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309,N(S(=O)(=O)N(C)C)CC(=O)NCC(C1CC1)NC(C(C)N(c1cnccn1)C)=O 310,c1(CC(=O)NC(C2CCCCN2C(c2ncoc2C(C)C)=O)C)ccc(O)nc1 311,N1(CC(C)NC(=O)Cn2cc(C(C)O)nn2)CCN(C(=O)C(Cl)=CCl)CC1 312,S(=O)(=O)(c1ccc(OC)cc1)NC(C(=O)NCC1CN(CCC)C(=O)C1)C 313,C=CCCCC(C1CC1)NC(=O)NCCc1nccn1-c1ccccc1 314,c1(C(N2CCN(C(=O)CC3CC34CC4)C(C3CCC3)C2)=O)cncc2c[nH]nc12 315,C1(C)(OC)CCCN(C(=O)Cn2cc(C3(O)COC3)nn2)C1 316,CC1(CNC(=O)CC2CCOCC2)CC(F)(F)CN1C(c1cnsn1)=O 317,c1(C(=O)NCC(CC=C)NC(=O)C(F)C2CCC2)cccc2nccnc12 318,C(=O)(C(=O)C(C)CC)N1CC(C(=O)NC2(CC#C)CC2)C(C)C1 319,N1(C(CCC2OCC(C)(C)C2)=O)CCc2[nH]nc(CNC(=O)C=CCO)c2C1 320,c1(OC)ccc(F)c(C(N2CCN(C(c3cc(OC)cc(F)c3)=O)C3CC23)=O)n1 321,O=C(C#CC1CCCCC1)NC(CC(=O)NC(CCO)C(F)F)C1CC1 322,c1(C(N2CCCC(C(N(C(C#C)C)C)=O)C2)=O)cc2ccccn2n1 323,N1(C(C2C(C)CCCC2)=O)CC2CC(NC(C3(c4ccccc4)CCC3)=O)CC1C2 324,Cc1nccc(C(=O)NC(CCF)C(=O)N(CC(F)(F)CO)C)n1 325,C1(CNC)CC(C(=O)Nc2csnc2C)CCO1 326,C1(C(C)NC(C2(O)CCOCC2)=O)CN(C(C2CC(F)(F)C2)=O)CCO1 327,N1(C(C2(C)N(C(c3c(C)nc(CC)o3)=O)CCC2)=O)CCCC(C)C1CO 328,N1(C(c2cc(OC)n[nH]2)=O)CC2CC1(C(=O)NOC(C)(C)CO)C2 329,c1(C(=O)NCC(C(C)C)NC(C(C(C)C)SC)=O)c(C)nn(C(C)(C)C)c1C 330,c1(Cn2c(C(C)(CCN(C)C)NCC(COC)(C)C)nnn2)nn(C)c(Cl)c1Br 331,Fc1ccc(C2=CCN(c3nc(Cl)nc4sccc34)CC2)cc1 332,c1(C(=O)NCC=CCNC(CCn2ccc(C)n2)=O)cc2c(s1)CCCNC2=O 333,N1(C(C=CCCC=C(C)C)=O)CC2CCC1CN2C(=O)Cc1ccccc1C 334,c1(C(N2CCC(NC(C3(F)CCCCC3)=O)C(O)C2)=O)ccc(=O)n(CCF)n1 335,CC(C(=O)OC(C)(C)C)C(=O)NC1CN(C(c2ccc[n+]([O-])c2)=O)CC1C 336,c1(C(N(CC(CNC(C2(C)CC=C(C)CC2)=O)O)C)=O)[nH]nc2c1COC2(C)C 337,C=C(C)CCC(=O)N1CCC(C(C)(C)NC(=O)C(C)OCC(F)(F)F)C1 338,CC1(C)CC(C(=O)NCC=CCNC(c2cc[nH]c(=N)c2)=O)CC(C)(C)O1 339,c1(CNC(=O)COC(F)F)cnn2c1CN(C(C1Cc3ccccc3O1)=O)CC2 340,c1(CCC(N2CCCC(NC(C3(C#C)CC3)=O)C2)=O)ccc([N+](=O)[O-])cc1Cl 341,c1(C(N2CCC(N(C(=O)C(O)CC(F)F)CCO)C2)=O)cc2c(s1)CCC2 342,c1(C(=O)NCC(CNC(C(CC=C)c2ccccc2)=O)(C)C)csc([N+](=O)[O-])c1 343,c1(C(c2n(CC=C)nnn2)NCC=CCl)cn(C)nc1-c1ccccc1 344,N1(C(c2cc(CC)on2)=O)CCN(C(=O)COCC(=O)OC)C(CF)C1 345,N1(C(C2(C)COC2)=O)CCCC(C2CC2NC(C2CCCO2)=O)C1 346,C1(CNC(COC2CCC(C)CC2)=O)CCCN(C(=O)CCN(C)C(N)=O)CC1 347,c1(C(N2C3CC(NC(C(C=C)O)=O)CC2CC3)=O)csc2ccc(Br)cc12 348,Cc1ccc(C(=O)NC(CNC(c2ccc(C#N)s2)=O)CO)c(=O)n1C 349,C#Cc1ccccc1CNC(=O)C(C)(C)NC(c1coc(CO)c1)=O 350,N1(C(C(C)N(C(C)=O)C)=O)CCC2(C1)CN(C(=O)Cc1ccccc1C)CCO2 351,C12(NC(c3c(CC)ocn3)=O)CCC(C1)N(C(=O)CN1CC(CC)C1)C2 352,C1(CN(C(CSCC(C)C)=O)C)CCCN1C(=O)Cc1cc(C(F)(F)F)n[nH]1 353,N1(C(CC#N)=O)CCc2nc(CNC(c3ccc4ccccc4n3)=O)sc2C1 354,C1(C(N2CC(C)(CCC(=O)NCCCC3CCOCC3)C2)=O)CCS(=O)(=O)C1 355,CCCC(C(=O)OCC(=O)Nc1ccc(-n2cncn2)cc1)S(N)(=O)=O 356,CCCC(C(=O)OC)C(=O)NC12CC(CNC(=O)Cc3coc(C)n3)(C1)C2 357,CC1(C(N2CC(C#N)C2)=O)CN(C(=O)CNC(=O)C(C)(C)C)C1 358,CC1(C(F)(F)F)CN(C(=O)Cc2cc(C(F)(F)F)nn2C2CCCC2)CCO1 359,c1(OC)ccc(F)cc1C(=O)C(=O)NC(CNC(=O)C1=CCCCO1)C1CC1 360,c1(OC)cncc(C(=O)N(C)CC2CCCN2C(c2ccnn2C(F)F)=O)c1C 361,C(=O)(C1=C(Cl)CCOC1)NCc1cn(CC(=O)NC(c2ccccc2)C)nn1 362,C(=O)(CC(C)CC(=O)OC)N1CC2C(CNC(CC3(OC)CCC3)=O)C2C1 363,C(CN=c1[nH]c(=NCC2CCC(=O)N2)[nH]c2c1CSC2)SCC 364,c1(CC(N2CCC(NC(CCC3C(C)C3)=O)C2C)=O)c[nH]c2cnccc12 365,C(=O)(C(O)CNC(c1sccc1CO)=O)N(CCOCCOC)C 366,C1(C(=O)NCC=C(C)C)C2CC(O)C(C2)N1C(C1CS(=O)(=O)C1)=O 367,CCCCCCCCCC(C)CC(C(=O)N(C)CCN(CC(C)C)CCOC)OC 368,C(=O)(C(CN(C)C)C(C)C)N1C(CNC(CC2(OC)CCC2)=O)CC1 369,N1(CC)CCCC(c2cn(CC(N3CCCN(CC(N)=O)CC3)=O)nn2)C1=O 370,N1(C(C(C2CCCC2)NC(C)=O)=O)CCC(C)C(CNC(=O)C=CC(N)=O)C1 371,O=C1NCC2CCCN(C(c3cncnc3)C(=O)NC3CCOC3)C12 372,N1(C(C(CC(C)C)N(C)C(c2cccc(O)c2F)=O)=O)CCN2C(=O)OCC2C1 373,c1(NCC)cccc(C(=O)NCC2CC2NC(C2CCNC2=O)=O)c1 374,C(=O)(C1=NOC(C)C1)N(c1scc(CC(N2CCCC2)=O)n1)CC.NC=O 375,Cc1onc(Br)c1Cc1noc(Cc2csc(C3CC3)n2)n1 376,c1(OC)cccc2c(C(N3CCN(C(=O)C(Cl)=CCl)CC3C(C)C)=O)cccc12 377,C(=O)(CCCCCF)NC(c1cnn(C)c1)C(=O)N(C(C)C(C)(C)O)C 378,C1(C(=O)NC(c2nncs2)C)CCN(C(C2(C(N)=O)CCC2)=O)CCO1 379,N1(c2nnc(C(N)=O)s2)CCOCC(CNC(=O)C(C2CCC2)C2CCC2)C1 380,C(=O)(C1Cc2cccc(Br)c21)NC1CCC(C(=O)OC)NC1 381,c1(C(N2CCN(C(C3CCCS3)=O)C3C2CCC3)=O)cc(=O)c2ccccc2o1 382,N1(C(c2c(C)nc(C3CC3)s2)=O)CCN(C(=O)CC2(O)CCC2)CC1C(C)C 383,C1(NC(C2C(C(=O)OC)C2)=O)CCC(O)CN(C(c2ccc(S(C)(=O)=O)s2)=O)C1 384,N1(C(CN(CC)CC)=O)CC(NC(c2cc(C#N)cs2)=O)C2(CC2)C1 385,c1(C(=O)NC2CC(F)(F)CC2NC(C2COC2)=O)cccc2c1OCC2 386,c1(OCC(=O)NC2CCC(N(C(Cn3ccc(C)n3)=O)C)C2)ccc(F)cc1Cl 387,n1(CC)cnc2c(NCC3(CO)CC3)nc(N3CCC(C(F)(F)F)C(C)C3)nc12 388,C1(NC(Cn2c(C(C)C)ncc2)=O)CN(C(=O)CCC2(C)CC2)C2(CCCC2)C1 389,CC(C(=O)N1CCC(O)(C(N)=O)C1)C(F)F.n12cc(nn1)CC(=O)NC1CC2C1 390,N1(C(C)=O)CCC2(CCC(CNC(=O)CN3OC(C)(C)CC3=O)CC2)CC1 391,C1(C)(CC(=O)NC(C)(C)C2CC2)CC(NC(CCC2C(C)C2)=O)C1 392,CCC(CC(=O)NC1CC(C)(NC(=O)COCC(=O)Nc2ccccc2)C1)SC 393,n1(CC)c(=N)[nH]c2cc(C(=O)NC3CC3NC(=O)CC(C)CCOC)ccc12 394,CC(CNC(C1(F)CCC1)=O)CC(=O)N1CC2C(NC(=O)OC(C)(C)C)C2C1 395,C1(F)(CNC(c2noc(CC)c2C)=O)CCCN(C(C2CC2c2nc[nH]n2)=O)CC1 396,Cn1ncc(CCC(=O)NCCC(O)CNC(C2CN(C(=O)CC3CC3)C2)=O)n1 397,c1(C(C(=O)NC2C(CNC(C3(C=C)CCC3)=O)CC2)O)cc(F)c(F)c(F)c1 398,C1(CC(=O)N(C2CCC(CC)CC2)C)CC(C)(C)CN1C(C1CCC(C)CC1)=O 399,CC(CCN(CCCN1CCNCC1)C)CC(C)(C)C 400,N1(C(C)C)CCCN(C(=O)CC23CCC2CN(C(C2CC2(F)Cl)=O)C3)CC1 401,c1(-c2nc(-c3c(C)nn(-c4cccc(Br)c4)c3Cl)on2)cn(CCO)c(=O)nc1O 402,C(=O)(C1CCCc2ncnn21)NCC1(NC(c2cncc(C#C)c2)=O)CCOC1 403,n1(-c2ccn(CC)n2)nc(CCCc2ccccn2)nc1CCc1ccccc1 404,N1(C(c2c(N)ccc(F)c2)=O)CCN(C(c2cc(O)ncn2)=O)C2CCCCC12 405,C(=O)(C(C)(F)C(=O)OC)N1CCC(CCC)C1.C(=O)(CCN1CCCC1)N 406,CCCCC(O)C(C)C(=O)NCC1(OC)CCN(C(C2(C)CCCC2)=O)CC1 407,CN1N=C(CC(=O)N2CCC(F)(F)C(CNC(C3(O)CCSCC3)=O)C2)CC1=O 408,c1(C(=O)NCCCN(C(CCC=C)=O)C2CC2)cccc2c1OC(C)(C)C2 409,C1(NC(C)=O)CC(n2cc(C3C4CC5C(C4)C35)nn2)C(CCC(=O)O)C1 410,CCCCC(C(=O)NCC1CCCCS1)NC(c1cccc(C#N)c1)=O 411,N1(C(C2(CC)C=CCN2C(=O)OC(C)(C)C)=O)CCC(F)(F)CC(C)C1 412,c1(CC(N2CC(NC(CCCOC)=O)(CO)C2)=O)c(C(F)(F)F)nn(C)c1Cl 413,CCCC(C(=O)NC)N(c1cccc(Cl)c1)Cc1cccc(O)c1 414,CC(C(=O)OC(C)(C)C)C(=O)N1CCC(CCNC(c2ccnn2C2CC2)=O)C1 415,Cn1cnc(CC(=O)NCC2C=CCN2C(=O)CCc2nnc(C(F)F)o2)c1 416,N(C1CCc2ccccc21)C(C(CNC(c1ncnc(C)c1C)=O)O)=O 417,C12(C(N3CCC(CNC(CC(C)N(C)C)=O)C3)=O)CCC(CC1)OC2 418,C(=O)(C1CCc2cccc(Cl)c21)N1C2CC(NC(C3(CC)COC3)=O)CC1CC2 419,C1(C(=O)NCCOC2CN(C(c3ccc(=N)[nH]c3)=O)C2)CC2(CCOCC2)CO1 420,C1(NC(C2CCC(C)CC2)=O)CCCC12CN(C(c1c(Cl)ccc(F)c1F)=O)C2 421,c1(OCC)cc(NC(C2(Cc3cnn[nH]3)CCCC2)=O)ccc1[N+](=O)[O-] 422,S(=O)(=O)(c1cccnc1)NCC(=O)N(C1CCN(C(=O)C(O)CC2CC2)C1)C 423,c1(-c2nc(C3CCN(c4c(C)con4)C3)on2)cc(F)cc(F)c1 424,N1(C(CS(CC)=O)=O)CC2CCCC2(NC(C23CC(COC)(CO2)C3)=O)C1 425,C1(CC)CN(C(=O)Cc2cc(Cl)cnc2C)CCN1C(=O)C1=CCSC1 426,O=C1NC(C(=O)NCC2CCN2C(=O)Cn2cnccc2=O)CCO1 427,C(Cn1cccn1)(C(=O)NOC1CC1)NC(C1CCCC(=O)N1)=O 428,c1(NC2(C)CC(NC(c3nn(C)c(NC(=O)CO)c3)=O)C2)ccc(Cl)c(Cl)c1 429,c1(C(N2CCCC(NC(c3c(C)[nH]cc3)=O)C2)=O)cn(C)c(=O)cn1 430,C1(C(N2C(CNC(C3N(C)CC(F)C3)=O)CCCC2)=O)CC(C)(C)OC1=O 431,C(N=C(NC1CCC1)N1CC(O)C2(CC2)C1)C1(O)C(C)(C)CCC1 432,N1(C(CCOCCC)=O)CCCC2CCN(C(c3cccn4cncc34)=O)CC12 433,N1(C(c2c(CCC)nco2)=O)CCC2(CC1)CC2C(=O)NC1(C)CCCC1(C)C 434,c1(C(=O)NCC(CNC(C(C)Cc2cnn(C)c2)=O)(C)O)cc2n(c1)CCOC2 435,C1(NC(n2ncnn2)=O)CN(C(=O)COCCOCCO)CC(F)(F)C1 436,C1(NC(=O)NCC2(OC)CC(C(F)(F)F)C2)CCCCC1Nc1ccn(C)c1C 437,N1(C(CCCC2(C)N=N2)=O)CC(NC(c2cc(C3CC3)n[nH]2)=O)C2CCCCC12 438,c1(NC2CCC2)ccc2nc(C(N3C(C)CN(C4CCOCC4)CC3)=O)oc2c1 439,c1(C(N2CCC(C=C)(C(N3CCC(CF)C3)=O)C2)=O)cccc2c[nH]nc12 440,c1(NC(c2nnnn2CCC)CCC)cc([N+](=O)[O-])ccc1C 441,CCCC(C(=O)N1CCCCC12CC(NC(=O)C(C)(CC)CC)C2)S(N)(=O)=O 442,C1(C(=O)NC2C(CNC(c3cccc(CO)c3)=O)C2)CCOC2(CCCCC2)C1 443,c1(SC)cccc2sc(NC(c3sc(-c4ccccn4)nc3C)=O)nc12 444,c1(C(C)(C)C(N2CC3CC(NC(=O)CC4CC4)C(C3)C2)=O)ccc2c(c1)OCO2 445,c1(C(=O)NC2C(CNC(c3cc(Cl)no3)=O)COC2)coc2ccc(Cl)cc12 446,CC(C)C(CO)C(=O)NC1CCCCC1CNC(c1cnc(-c2ccco2)s1)=O 447,C(=O)(C(CO)C(C)(C)C)N1C(CN(C(Cc2nc(C(C)OC)sc2)=O)C)CCC1 448,CCC(CO)C(=O)N1CC(C(C)NC(c2c(OC)noc2C)=O)C1 449,C12(C(N(CC(N3CCCC(CO)C3)=O)CC)=O)CCC(CC1=O)C2 450,CCCC(C)(O)CC(=O)N(C)CCOCCN(c1nnccc1C#N)C 451,c1(C(=O)OC)ccc2c(C(=O)NN3CC(OC(C)(C)C)CCCC3=O)cccc2n1 452,C1(NC(C(C2(O)CN(C(c3csc(C)c3C)=O)C2)F)=O)CCCCCC1O 453,C(N1CCOC2(C1)CN(C(=O)Cn1nc(C3CC3)n(C)c1=S)C2)C(C)C 454,N1(C(C(C2CCOCC2)C)=O)CC(NC)C(C)(C)C1.c1(C=O)c[nH]nc1Br 455,CC(C)C(C)C(=O)N1CC2C(CNC(=O)CCOCc3ccccc3)C2C1 456,Cc1ccc([N+](=O)[O-])c(NNC(=O)NC23CCCCC2OCC3)n1 457,C1(CNc2nc(COC)nc(N3CCC(CF)C3)c2)CC2(CCC2)CCO1 458,c1(C(C(=O)NC(C(F)F)c2ccco2)NC(CNC(=O)NC)=O)cccnc1 459,N1(C(CC(=O)OC)=O)CC(C2CN(C(c3cccc(-c4nnc(C)o4)c3)=O)C2)C1 460,c1(C(=O)NCCC(C)CCNC(=O)C(F)CC2CC2)cccc2ccnn12 461,C(N=c1[nH]c(=NC2CC(=C3CCC3)C2)c2[nH]ccc2[nH]1)c1ocnc1.FCF 462,Cc1c(C(N2CCOC(CCCN(C)C)C2)=O)cnn1CCC(C)C 463,N1(C(C(CC)=CCCC)=O)CC(C)CN(C(c2ccc(C(F)F)cc2)=O)CC1C 464,C1(C(=O)NCc2cnco2)CC(F)CN1C(c1ccccc1F)=O 465,N1(C(CCCn2ncc(C)c2)=O)CCC(n2cc(CNC=O)nn2)CC1 466,N1(C(C2N(C(C(CCC)CCC)=O)C3CCC2C3)=O)CCc2nc(C)sc2C1 467,C=C(Cl)CCC(=O)NCC(C)(CNC(c1csc(C(C)=O)n1)=O)OC 468,c1(-n2c(C3CCC(c4cccc(F)c4)C3)nc(CO)n2)cccc2ccccc12 469,C1(CC=C)(NC(CCN(C(=O)C(O)CN(C)C)CC#C)=O)CCCC1 470,c1(NCC(C)NC(C)CN2CCSCC2)c2c(nn1C)CCCC2 471,C=CC1CN(C(c2ccc(F)c(O)c2)=O)CC1NC(C1CCC(F)(F)CO1)=O 472,N1(C(C(C)CC(F)F)=O)CCC(CNC(c2ccc3n[nH]cc3n2)=O)C(F)(F)C1 473,c1(C(=O)NCC(C2CC2)NC(c2cnc(CC)s2)=O)c(F)cncc1Cl 474,c1(C(=O)NCC2(F)CC(NC(C(CC=C)(C)C)=O)C2)cc(F)c(C#N)c(F)c1 475,C1(NC(c2ccc(Cl)cc2F)=O)CN(C(=O)C2=CCCC2)CC1C1CC1 476,c1(OC)ccc(C2(CNc3cnc(I)cn3)CCC2)cn1 477,C1(C(=O)NC2(C)C(C)(C)C2)CCN(C(C2CC3(CC(=O)C3)C2)=O)C1(C)C 478,C1(CNC(c2c(SCC)cncc2)=O)COCCN(C(C2(C)CCCN2C)=O)C1 479,C1(CNC(C(C)N2CCC2)=O)CC2CCC1N(C(=O)CC(C)c1cccnc1)C2 480,c1(OC)ccc(Cl)cc1C(N1CCN(Cc2cn(C3CCC3)nc2C)CC1)=O 481,Cc1c(NCc2cnc(O)nc2O)ncnc1NC(c1ccc(F)cc1)C 482,C(C)(CCCC(C)C)NC(C(CC=CC)NC(c1c[nH]c(C)c1)=O)=O 483,Cn1ccc2cccc(C(N3CC(F)CC3C(=O)Nc3cc(O)ccn3)=O)c12 484,C(=O)(CCCCC(=O)NC1CC(OC)CN(C(c2coc(N(C)C)n2)=O)C1)NC 485,C(=O)(C(O)C(C)CC)NC(CC=C)CNC(c1ccc(C(N)=O)cc1)=O 486,c1(N2CCCC(CCOC)C2)nc2ncc(Cl)cc2s1.c12ccnc(c1)NC2=O 487,C1(C(=O)NC(C)C(C)(C)NC(C2CCC(C(=O)OC)CC2)=O)CCS(=O)(=O)C1 488,C(=O)(C1CCSc2ccccc21)N1C(CNC(c2cc3c[nH]nc3s2)=O)CCC1 489,C1(NC(c2sccc2F)=O)CC2CCC1CN2C(=O)Cn1cc(CO)nn1 490,C#Cc1cc(NC(=O)CN(C(=O)C(C(C)CC)N(C)C)CC(C)(C)C)cc(F)c1 491,N1(C(C(CCC)O)=O)CCOC2(CCN(C(=O)CC3(C(=O)OC)CCCC3)C2)C1 492,N#CC1CCCCN1C(C1CN(C(c2cccc(C(F)(F)F)c2)=O)C1)=O 493,C(c1cnn(C)c1C)=CC(N1CC(NC(c2nccc(CC)c2)=O)C(C)C1)=O 494,C1(CNC(C(CC)N(C)C)=O)CCN(c2ccc(CC(=O)OC)cn2)CC1 495,c1(OC)cn(CC(N2CC3C(N(C)C(c4scnc4C)=O)C3C2)=O)c(C)cc1=O 496,C1(NC(C(CC)C)=O)CCC(CNC(C2CCCC(C)O2)=O)CC1 497,c1(C(=O)NC2C(NC(C(F)=CC)=O)CCCC2)cn2c(Br)cnc2s1 498,C(=O)(CCCC(N)=O)NCCC1C(C)CN(C(c2c[nH]nc2Br)=O)C1 499,CC(O)(CC(=O)N1CC=CC(NC(=O)CCCCN2CCCC2)C1)C(F)(F)F 500,N1(C(C(N2CCOCC2)C)=O)CCC2(CCC(NC(c3cnc(O)o3)=O)C2)C1 501,CC(CNC(=O)C(N1CCNC1=O)C)CC(=O)N(C1CCCCC1)CCO 502,n1(CC)cc(Br)c(C2CCCN2C(=O)CNc2cnn(C)c2)n1 503,C1(c2ccc(Cl)cc2)(C(N(CC(CNC(CSCCC)=O)O)C)=O)CCN(C)C1 504,N1(C(=O)CCc2ccccc2Cl)CCCCC(C2CN(C(C3CC(O)C3)=O)C2)C1 505,c1(C(=O)NCC(F)CNC(C2CCC3CC23)=O)ccc(CN2CCCC2)c(F)c1 506,Cn1ncc2c1CCC(C(N1C3CCCC1CN(C(=O)CC(F)(F)F)C3)=O)C2 507,c1(C(N2C(CNC(C3(F)C(C)C3)=O)CC2)=O)cc2cc(Cl)ccc2o1 508,C1(C(CNC(C(C(C)C)c2ccc(F)cc2)=O)O)CCC(F)(F)CC1 509,CC1=CCC=CC1C(N1CCN(CCCNC(C2(F)CCCC2)=O)CC1)=O 510,CC(C)(C(=O)NCC1CCN1C(=O)CCN1CCCC1=O)c1ccccn1 511,CCN=c1[nH]cc(C(=O)NC(C)(CNC(C2CCCN2CC)=O)CO)s1 512,C(=O)(C(CC)C(=O)NC(c1cccnc1)C(=O)NCCO)OCC.C1CCCC1 513,c1(C(=O)NCCCN(CCCNC(C(CC)N(C)C)=O)C)cnc2[nH]cnc2c1 514,c1(OC)ccc(CCC(=O)NCCNC(=O)CC2COCCOC2)cc1N 515,N1(C(C(C)C(=O)OC(C)(C)C)=O)CCCN(C(c2c[nH]nc2Cl)=O)CC1C 516,CC1CCC(CCC(=O)NCC(C)(C)CNC(C23CC(CC(F)F)(C2)C3)=O)O1 517,c1(C(=O)NCC2(CCNC(c3n(C)ncc3)=O)CC2)cc(N2CCCC2)ccn1 518,N12CC3CC1C3NC2=O.c1(C2CCN(C(C3CC=CC3)=O)C2)nn(CO)cc1F 519,C1(NC(C2CCCN(CC)C2)=O)CCN(C(C2CCCC2O)=O)C12CCC2 520,N1(C(c2c(=N)cc[nH]c2)=O)CCC2(CCCN(C(C34CCC(CC3)C4)=O)C2)CC1 521,c1(C(=O)NCCC2CCC(NC(C=CC(=O)OCC)=O)C2)n[nH]c2c1COCC2 522,C1(NC(C2C(C)CC=CC2)=O)CC2CCC1CN(C(=O)CSc1n[nH]c(O)n1)C2 523,n1(CC)ncc2c(NC(=O)CC3(O)CN(C(=O)NCC4CCCC4)C3)ncnc12 524,CC1CC2(CCC(CNC(=O)Nc3ccnn3C)O2)CO1 525,CC(C)C(C(C)NC(C1(N(C)C)CC1)=O)NC(c1ccsc1Cl)=O 526,CCC(C(C)(C)O)NC(=O)CC1CCCC(NC(=O)CC(C)=C(C)C)C1 527,C1(OC)CC(C)CN(C(C2C(O)CCN2C(=O)C(C)=NOCC#N)=O)C1 528,c1(C(N2CCc3nnc(O)cc3C2)=O)c2c(nc3ccc(Cl)cc13)CCC2 529,C=CC1(C(=O)NCCC2CCCN(C(C3(C)CCCNC3=O)=O)C2)CCCCC1 530,c1(C(=O)NC(Cc2c(OC)cccc2)(C)C)[nH]nc2c(OC)cccc12 531,c1(C(=O)NC)ccc(C=CC(=O)N(C)CCN(C(=O)CCS(C)=O)C)cc1 532,C#CCCCCCCCNC(=O)C(CC1CCOCC1)NC(c1cnns1)=O 533,CC1c2c[nH]nc2CCC1C(=O)NC1C=CCN(C(c2csc(Cl)n2)=O)C1 534,c1(C(=O)NC(CN(C(C(C=CC)O)=O)CC)CC)ccc2nc3n(c2c1)CCC3 535,C1(CNC(C2(C(=O)NC)CC2)=O)CC2(CO1)CN(C(=O)C(C)CC1CC1)C2 536,C1(OCCC(=O)N(CCN(C(C(C)NC(=O)OC)=O)C)C)CCC(F)(F)CC1 537,C1(NC(=O)NCC(C)Oc2cccnc2)CCCCCC1C(N)=O 538,C1(CNC(C2C(C(C)NC(C(CSC)OC)=O)C2)=O)OCCCC1(C)C 539,Cc1cc(C#N)ccc1C(=O)NC(C)(C(=O)NCCOCCN=[N+]=[N-])C1CCC1 540,C(=O)(C(CNC(c1cccc(O)c1C)=O)CC=C)N(CC#C)CC1CCCO1 541,c1(CNC(=O)CCC2CCCN(C(=O)COC3CCOC3)C2)cc(F)ccc1O 542,C(=O)(C1=CCN(C)C1)N(CC(CNC(CCOCC)=O)(C)C)C 543,c1(NC(CSC(C2CCCOC2)C)=O)ccc(OC2CCCC2)nc1 544,CCC(C)C(O)CC(=O)N1CCC(C(=O)NCC(=O)N(C)O)C1 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563,Cc1nn(C)c(Cl)c1CC(=O)NCCCCCCNC(C1CCC(C)(C)CO1)=O 564,C#CCC(O)C(=O)NCC1CC1NC(c1cccnc1OCCCC)=O 565,c1(C(N2CCN(CC(COCC(C)C)O)CC2)C)ccc2c(c1)NC(=O)CO2 566,C(=O)(C1=CCCSC1)NCCN(C(C)C)C(c1ccccc1SCC(F)(F)F)=O 567,Cc1ccc(C)c(C(N2CCC(C)N(C(c3cc(Cl)no3)=O)CC2)=O)c1N 568,C1(C(N(CC(C)NC(=O)CSc2ccccn2)C)=O)CC(C2CCC2)C1 569,CC1CC(C(=O)NCc2ocnc2C(N2CCC(CO)C2)=O)CC(C)C1 570,C1(C(=O)NC2C(CNC(c3ccc(CC)cc3)=O)C2)CC2CC(=O)C1O2 571,C1(CNC(C2CN(C)C2)=O)CC2(CO1)CN(C(=O)CC1CCCCN1C)C2 572,N1(C(CCC=C)=O)CCC(CNC(C2CCC(F)CC2)=O)(COC)CC1 573,N1(C(c2ccc(C#C)cc2C)=O)CCC(NC(=O)C(O)C=C)C2(CCC2)C1 574,c1(OC)ccncc1CC(N1CC2CC1C2NC(=O)C(CO)NC(=O)C(C)C)=O 575,C1(C(N(C(C)CCNC(=O)Cc2ccc(O)nc2)C)=O)CCC(C)(O)CC1 576,c1(N2CCC(CCNC(C3C(C)CCCC3)=O)C2)ncnn2cccc12 577,N1(C(CC2CCC(C)C2)=O)CC2(CCN2C(=O)CC(C)(F)F)C1 578,CCCCCS(=O)(=O)CC(=O)N1C2CCCC1CN(C(=O)CCc1cccs1)C2 579,c1(C(=O)NC(C)CN(C)C(c2ccc(OCF)cc2)=O)ccc(O)nc1Cl 580,C1(C(=O)NCC2CCN(C)C2)(CNC(=O)CC2COCCO2)CCCCC1 581,Cn1c(O)nc2cccc(C(N3CCCCC(NC(=O)CCS(C)(=O)=O)C3)=O)c12 582,c1(OCC(N2CC(CCNC(C3CS(=O)(=O)C3)=O)(OC)C2)=O)ccc(F)nc1 583,CC(C)(Cc1cnn[nH]1)C(=O)N1CCC(N2CC=CC2)C1 584,C1(CNC(c2n(C)cc(F)c2)=O)COCCN(C(C2(C)CCOCC2)=O)C1 585,N1(C(c2nc(CC)sc2N)=O)CC2(C)CN(C(C3CCS(=O)(=O)N3)=O)CC2(C)C1 586,CC(C)C(F)(F)CC(=O)N(CCNC(C1CC(F)(F)C1)=O)CCc1ccccc1 587,Cc1cc(C(=O)NCC2CC(CNC(c3ccncc3Br)=O)CO2)[nH]c1C 588,N1(Cc2c(C)ccnc2)CCC(NC(c2cccc(F)n2)=O)C(F)C1 589,CC(=O)C(C)CC(C)C(=O)NCc1ccc(C(N2CCCC(CCF)C2)=O)nc1 590,C1(CCC)CN(C(c2ccc(OC)cc2OC)=O)CCN1C(=O)Cc1cnsc1 591,C(=O)(C(C)CC1CC1)NCC(C1CCCC1)NC(CSCC=C)=O 592,Cc1ccn(C)c(=O)c1NC(C1C(C)CN1C(c1cc(C(C)C)[nH]n1)=O)=O 593,Cc1cncc(C(N2CCC(CNC(c3cc(N)cc(O)n3)=O)CC2)=O)c1C 594,c1(C(N2CC(C)(C(NOCCCOC)=O)C2)=O)c(Br)nnn1C 595,c1(NC(c2ccc(-n3ccc(O)n3)cc2)=O)ccc(O)c(Br)c1 596,N1(CC)CCC(NC(C2OCCC2CNC(c2c[nH]c(C)cc2=O)=O)=O)C(C)C1 597,N1(C(C(CN(C)C)O)=O)CC(NC(=O)CSCc2cccs2)C(C)(C)C1 598,C12(CNC(C(CC(C)C)SC)=O)CC(C(N)=O)(C1)C1(CN(C(=O)C=C(Cl)Cl)C1)O2 599,c1(CC(=O)NCC(=O)NCC2(COCC(=C)C)COC2)cc(F)ccc1F 600,N1(C(c2cscc2F)=O)CCN(C(c2cccc(F)c2Cl)=O)C2COCC12 601,CC1(CN2C(=O)CCN(Cc3nocc3Br)C2=O)Cc2ccccc2C1 602,C1(CNC(=O)C(=O)Nc2ccc(C(C3(CC(N)=O)CC3)=O)cc2)CCCC(CF)C1 603,c1(CNC(=O)NC(C2CCN(C(=O)C(C)(C)C)C2)C(=O)OC)nc2ccccc2[nH]1 604,c1(C(N(CC(C)NC(=O)C(F)CC2CC2)CC)=O)ccc2c(C)nn(C)c2n1 605,C=C(C)CC(C)C(=O)NCC(=O)NOCCC(F)(F)F 606,C1(NC(CCC(=O)NCCC)=O)CC2(NC(C3CC4CCC3CC4)=O)COC1C2 607,C#CC1CCCN(C(=O)COC(C)(C)CNC(=O)CC(C)C(F)F)CC1 608,Cc1cc(CNCC(C)(O)C2CC2)ccc1Br 609,C(c1ccc([N+](=O)[O-])cc1)=CC(=O)NC1CN(C(c2cc(Cl)cnn2)=O)C1 610,C(=O)(C(C(C)(C)O)NC(=O)CC1CC2(CC2)CO1)NCCC(CC)(F)F 611,C1(F)(C(N(CCC(C)NC(C2CCCC23CC3)=O)C)=O)CCC(F)(F)CC1 612,C1(NC(C2CC3CC2C3)=O)CCCC2CN(C(c3coc4ccccc34)=O)CC12 613,C1(CNC(CCOCCCNC(C(C)=C2CCC2)=O)=O)CC(O)C12CCC2 614,C(=O)(C1=CCS(=O)(=O)C1)N1CC(N(C(=O)Cc2ccc(F)cc2Cl)C)C2(C1)CC2 615,C1(C2CC2)(NC(=O)C(F)n2ccnc2)CCN(C(c2ccc(Cl)o2)=O)C1 616,C1(C)(CC(=O)NC2CN(C(CCCOCCOC)=O)C(C)C2)CCS(=O)(=O)N1 617,C=C(C(=O)NC1CN(C(=O)Cn2nc(Cl)ccc2=O)CC1F)C(F)(F)F 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726,c1(C(=O)NC2C3(CC(NC(C(C)CN4CCCCC4)=O)C3)C2)cccc(N)c1F 727,C1(CC(=O)NC2C(C)COCC2)C2CCCC2N1C(C1C2CCCOC12)=O 728,C1(C(=O)NCC(C)NC(=O)CN2CC(C)(C)C2)COc2ccc(O)cc2O1 729,C(=O)(CS(=O)(=O)c1ccccc1F)N(C1CCN(C(CCCC)=O)CC1C)C 730,C1(C(=O)OC)CCCC(C(=O)NC23CC(CNC(=O)CC4CC4C)(C2)C3)C1 731,N1(C(C(=O)NCc2ccc(N(CC=C)C)cc2)=O)CCn2cc(C)nc2C1 732,C1(c2n(CC)nnn2)(Nc2ccc(C(C)C)c(O)c2)CC2CC(OC)C2C1 733,CC(C)CC(C(=O)N1CCOCC(NC(=O)C2=CCC2)C1)NC(=O)OC(C)C 734,C1(C(=O)NCC2(O)CCOC2)CC=CCN1C(c1csc(C2CC2)n1)=O 735,N1(C(c2cn(C(C)C)nc2)=O)CCN(C(=O)COc2ccc(F)cc2)C(C)C1C 736,C1(C(=O)NCc2nc(COC)sc2)CN(C)CCN1C(=O)C(CO)N(C)C 737,C(=O)(C#CC1CCCO1)N1CC(C)CC(NC(c2c(O)ccc(C)c2)=O)C1 738,S(=O)(=O)(c1cc(CC)ccc1C)N(CC(=O)OC(C1CCCCC1)=O)C1CC1 739,CCC(C(=O)NCCCC(C)NC(c1ccc(C)nc1N)=O)C(C)C 740,C1(CC(N2CC(OCC)(CNC(c3ccoc3)=O)C2)=O)CC(OC)C1(C)C 741,N1(C(CCC#C)=O)CCC(=O)NC2CN(C(=O)CCCC(F)(F)F)CCC12 742,C1(CNC(=O)NCC(C)OC)CN(c2cc(C3CC3)ncn2)CCO1 743,Cc1ccc(=N)[nH]c1C(N1CCN(C(=O)C(C)C2CCCC2)CC1C)=O 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762,N1(C(C=C(C)C)=O)CCCC2(CCN(C(c3c(Cl)ccc(Cl)c3O)=O)CC2)C1 763,C1(NC(C(C)(C)N2CCCCC2)=O)CC2(C1)CC(NC(C1CCC1C#N)=O)C2 764,Cc1cc(C(=O)NC2CCC2CNC(c2cn(CC(F)(F)F)nn2)=O)n[nH]1 765,c1(CC(=O)N(CCN(C(C(C2CCCC2)OC)=O)C)C)cccc2occc12 766,C(=O)(C1=CCCCCC1)NC1CC(N(C)C(C2CC23CCOC3)=O)C1 767,C1(C)(C(=O)NCC2CCCC(NC(COCC#C)=O)C2)CCOC(C)C1 768,C1(C2CCCN(C(C3CC3COC)=O)C2)(NC(c2c(C)nn(CC)c2C)=O)CC1 769,c1(NC)c(C(=O)NC(C)(C)CNC(=O)CC2CC3CC3C2)cccc1[N+](=O)[O-] 770,Cc1cnn(CCC(=O)NCC2(NC(C3CC3(c3ccccc3)F)=O)CCC2)c1 771,C(=O)(CCS(=O)(=O)c1ccc(Cl)cc1)NC(C(C)NC(CC(C)OC)=O)C 772,N1(C(c2c(CC)nccn2)=O)CCC2(CC1)CCN2C(=O)CCC1CCOC1 773,C1(C(N(C(=O)C=CC(C)(C)C)C)C2CC2)CCN(C(C2CC(N(C)C)C2)=O)C1 774,c1(C(N2CCCC(CCNC(C3(NC(C)=O)CCC3)=O)C2)=O)cnc(O)c(C)c1 775,C1(C)(C(=O)Nc2cccc(NC(c3c(C)nn(C)c3)=O)c2)CC2(C1)CC(F)(F)C2 776,N1(C(C2C(=C)C2)=O)CC2(CCN(C(c3sc(Cl)c(Cl)c3OC)=O)CC2)CC1C 777,C1(C(=O)NC2(CO)CN(C(CC3(C)CCC3)=O)C2)CCC(CCO)CC1 778,CCC(F)(F)C(C)(C)C(=O)NC1CCCCCC1NC(=O)CC1CCN(C)CC1 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887,N1(C(C(=O)NC(C)C)=O)CC(NC(=O)CSCC2CCCCO2)C(C(F)F)C1 888,C1(CNC(C2CCCC2C(F)F)=O)CC2(CCC2)CN1C(=O)CCOCC(F)F 889,c1(NC(=O)NCC2CC(CC)C2)ccc(C(N2CCCC2C(=O)O)=O)cc1C 890,c1(OC)cc(-c2cn(CCN(C(=O)CCn3ccnn3)C)nn2)ccc1F 891,C1(C(N(CC(F)F)C)=O)C(CNC(C2CCCS2)=O)C1(C)C 892,c1(C(N2CCC(OCCNC(C3(CC)CC3(F)F)=O)C2)=O)c([N+](=O)[O-])cnn1C 893,N1(C(CN(S(C)(=O)=O)C)=O)CCN(C(=O)CC2OCCCC2(C)C)C2COCC12 894,S(=O)(=O)(C1CCC2(CC1)CC2)NC1C(C)CCC1 895,c1(C(=O)Sc2ccc(C(=O)NC3C(C)CCC3)cn2)ccc2c(c1)N(C)CC2 896,N1(C(c2c(C)c(C3CC3)on2)=O)CC2CCCC1C2CNC(=O)Cn1cncn1 897,Cc1cc(C(=O)NC2CC3CC2N(C(=O)CSCc2cccs2)C3)nc(C)c1 898,c1(C(N2CC(OC)C(NC(C3CC=CCC3)=O)C2)=O)cc(F)c(N)cc1F 899,CC1=C(C(=O)NCC2CN(C(c3c(C)noc3C)=O)CCN2C)CCO1 900,N1(C(C(C(CC)C)O)=O)CC2CCN(C(C3(C)CN(C4CCC4)C3=O)=O)CC2C1 901,c1(C(N2CCC3CN(C(CCCSC)=O)CC32)=O)cc2cc(C)ccc2[nH]1 902,CCC(C)(F)C(=O)NC(C)CNC(C1(Sc2ccccc2)CC1)=O 903,O=C(CC1=CCCC1)NCc1ncccc1C(=O)NC1CCCCC12CC2 904,c1(N(CCCCN(C(=O)CC2COC(=O)C2)C)C)nnc(C2CC2)o1 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1140,Cc1ccc(CCCCC(=O)NC(CNC(c2cc(C)ncn2)=O)CO)cc1 1141,C1(CNC(C(COC)C)=O)COC(C)(C)CN1C(=O)CC1(N(C)C)CC1 1142,c1(OC)ccc(C)c(C(=O)NCC2CC(NC(c3ccc([N+](=O)[O-])s3)=O)C2)n1 1143,CC1(CNC(C2C(F)(F)C23CCC3)=O)CCN(C(C2C3CCCC23)=O)CC1 1144,C12(NC(=O)COC3CCC3)CCCCC1N(C(c1cc(Cl)ns1)=O)CC2 1145,c1(CSC)cc(C(=O)NC(CCNC(=O)Cc2cncn2C)C(C)C)ccc1F 1146,C1(C(=O)NC2CCN(C(c3cc(C(C)(C)C)ncc3)=O)CC2)CCOCC1(C)C 1147,C12(CNC(COCC(=O)NC)=O)CC1CN(C(=O)CNC(=O)CC(C)(C)C)C2 1148,Cc1cc(=NC(C)c2cnn(C)c2C)[nH]c(=NCC2CCCc3nccn32)[nH]1 1149,Cc1cnc(F)c(CNC(=O)CC(C(F)F)NC(C2(c3ccno3)CC2)=O)c1 1150,Cc1cc(OCC(=O)NCC(F)CNC(c2ccc(C3CC3)cn2)=O)cc(C)c1 1151,c1(N(C(=O)CC2CCN(C(=O)C(O)CN3CCCC3)C2)CC)ccc(F)cc1F 1152,CC1CCC(NC(C2CC3CCC3C2)=O)CN1C(C1CCCO1)=O 1153,c1(C(=O)NC(CCNC(Cc2c(C)cccc2)=O)C(C)C)ccc(C)n(C)c1=O 1154,C(=O)(C(CCCO)c1ccccc1)NC1CC(C)(C)C1O.C=O 1155,CCCC(C(=O)N(CC(CC)NC(c1[nH]nnc1C)=O)CC)NC(C)=O 1156,Cc1nn(C)c(C)c1C(=O)OCC1(NCc2ccc(-c3nn[nH]n3)cc2)CC1 1157,C1(C(=O)NCc2cccc(NC(C(C)(C)F)=O)c2)CCn2cncc2C1 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1230,C1(C2CC2)(CC)CN(C(=O)CC2(NC(c3csc(=N)[nH]3)=O)CCCCC2)C1 1231,c1(C(CC)NC2COCC2O)ccc(C#N)c(C)c1 1232,N1(C(C2CC(NC(c3ccnc(O)c3)=O)C(O)C2)=O)CC2(C1)CC2(F)F 1233,N1(C(C(F)=C(C)C)=O)CCC2(CCCN2C(=O)CCCc2ccc(Cl)c(Cl)c2)C1 1234,c1(C(N(CC(C)N(C(=O)CC2CCOC2)C)C)=O)cc(F)n[nH]1 1235,c1(C(=O)NCCC2N(C(C(CCC)C#N)=O)CCC2)[nH]c2ccccc2c1OC 1236,C(=O)(CCC(F)(F)C(=O)NCCN(C)C(C12CCCCC1C2(F)F)=O)OC 1237,C(=O)(CC(CC)C(C)C)NCc1ccc(CNC(c2cncc(C#C)c2)=O)cc1 1238,c1(C(=O)NC2C(CNC(C(C)C(F)(F)F)=O)CC2)cccc2nnn(C)c12 1239,c1(OC)ccc2c(N(C3CC(N)C3)Cc3ccc(O)cc3C)ncnc2c1 1240,C1(CC=C)(C(N2CCC(O)(CO)C2)=O)CCN(C(=O)C(C(C)OC)N(C)C)C1 1241,N1(c2cccc(NC(c3[nH]c(=N)sc3C3CCCC3)=O)c2)CCC(=O)NC1=O 1242,c1(CC)ccnc(C(=O)NCC(CC(=O)N2CCC(O)C2)C2CCC2)c1 1243,c1(CNC(CC2(C)N(C(c3c(CC)cc[nH]3)=O)CC2)=O)cnc(O)nc1O 1244,C12(C(N(CC(C)SC)C)=O)CCC(CC1)N(C(c1ccnc(CO)c1)=O)C2 1245,CC(C(=O)NNC(=O)CC1(OCCO)CC1)n1cc(CN2CCS(=O)(=O)CC2)nn1 1246,CN(C(=NCCCCl)NC1CCOC(c2ccc(F)cc2)C1)CCC(F)F 1247,c1(CCC(c2nnnn2C)NCC2(OC)CC2)ccccc1F 1248,c1(C2CCN(C(=O)NCCSCCC(F)(F)F)C2)ncc(Br)cn1 1249,C1(C(c2n(C)nnn2)Nc2ccc(Cl)cc2)CCC2(CC1)OCCCO2 1250,C1(CNC(C(C(=C)C)(C)C)=O)CC2(CO1)CN(C(c1ncc(C)cc1F)=O)C2 1251,Cc1cc(Br)cc(C)c1C(=O)OCC(N1CCCC(C(C)(C)O)C1)=O 1252,CCC(CC(=O)N1CCN(C(C2CCCN2C)=O)C(CO)C1)C(=O)OC(C)(C)C 1253,N1(C(COc2cn(C)nc2)=O)CC2CCC1C(CN=c1[nH]nc(O)s1)C2 1254,c1(NC(C(C)=C2CCC2)=O)ccc(NC(=O)C(c2cccc(N)c2)O)c(C)c1 1255,c1(N(CCN(C)C)C)nc(N2CCOC(C)(C)C2)nc2c1COCC2 1256,Cc1cc(C(=O)NC2(C)CNCC2(F)F)c(C)nn1 1257,C1(COCC)CCCN(C(C2(C(C)NC(c3[nH]cnc3C)=O)CC2)=O)C1 1258,C(=O)(C1=C(C)N2CCN=C2S1)N1CCC2(C(C(=O)NCCCOCC=C)C2)CC1 1259,c1(C(=O)NC(C2CCN(C(C3CC=CC3)=O)C2)C)cc(F)c(F)cc1N 1260,c1(N(C2CN(C(C(C=C)c3ccccc3)=O)C2)C)nc(C)ncc1F 1261,c1(-c2n(C)ncn2)ccc(C(N2CC(O)CC2CNC(C2(CO)CC2)=O)=O)cc1 1262,N1(C(C=CCC)=O)CCC(C)C(CNC(c2cc(C(=O)OC)oc2C)=O)C1 1263,S(=O)(=O)(c1ccc(C(=O)NC2CC3(C2)CC3NC(=O)CCCC(F)(F)F)o1)NC 1264,c1(CCC)cc(C(=O)N(C2CCCC(NC(c3cnc(O)n3C)=O)C2)C)sc1C 1265,c1(NC(CN(CCC)C)=O)sc2c(c1C#N)CCCCCC2.C1(C)CC(=O)N1 1266,Cn1nccc1C=CC(N1CC(NC(=O)C(F)C2CCC2)C1)=O 1267,c1(C(N2C(CNC(C(c3c(C)ccnc3)(C)C)=O)CC2)=O)cnc(Cl)c(F)c1N 1268,Cc1cc(NC(=O)CC2CC(C)N(C(C3COCCC3C)=O)C2)cc(C)c1F 1269,N1(C(C(C2(O)CCCCC2)NC(c2cc(C)c(C)s2)=O)=O)CCN(C)C(C2CC2)C1 1270,C=C(C)CC(C(=O)NCc1nc(C(N)=O)co1)NC(C1CCCN1C=O)=O 1271,N1(C(c2cc(C(=O)OC)oc2C)=O)CC2CN(C(=O)CN3CCOCC3)CC2C1 1272,N1(C(c2c(SCC)cccn2)=O)CC2CC(NC(=O)Cn3cnnn3)CC2C1 1273,C1(NC(c2c(C)sc(O)n2)=O)CCN(C(=O)C(C)Cc2ccccc2Cl)CC1C 1274,Cc1ccc(C)n1CC(=O)NCCCC(=O)NCC1CCC2CC12 1275,C1(F)(C(=O)NC(c2c(C)ncs2)C)CCN(C(c2ccc(C#N)[nH]2)=O)C1 1276,c1(CNC(NCc2nc(CC)on2)=NCC2CC2)cn2c(C)cc(C)cc2n1 1277,c1(C(c2n(CCC)nnn2)NCc2cncs2)cccc(C(F)(F)F)c1F 1278,C1(CNC(C2N(CC#C)CCC2)=O)CC(F)(F)CN1C(C1CN(C)CCO1)=O 1279,N1(CC2CC2)CCCNC(=O)C12CC2.c12cncc(c1)N(CC1CC1)NC2=O 1280,N1(CCC)CC(C(N2CCCC2CN(C)C(C2CCC(=O)N2)=O)=O)CC1=O 1281,CC#CCC(C(=O)NCCC(O)C1CCC1)NC(c1ccccc1OC)=O 1282,c1(C(=O)Nc2nccc(C#N)c2)cc2ncc(-c3cncs3)cc2[nH]1 1283,C1(CC)(NC(c2sc(-n3cccc3)nc2C)=O)CCCN(C(=O)C(C)COC)C1 1284,N1(C(c2n(CC(C)C)ncc2)=O)CCN(C)C(CNC(=O)CC2CC2C)C1 1285,c1(C(=O)Nc2cccc(CO)c2F)ncn2cc(-c3cnoc3)sc12 1286,c1(OC)ncc(C)cc1C(=O)NC1CC1CNC(=O)CC1COC(=O)C1 1287,Cc1c(F)ccc(C(=O)NC2CC3CC(NC(=O)C#CC(C)C)CC23)c1C#N 1288,C(=O)(C(CC(C)C)NC(=O)CCCCCSC)OCC#C 1289,N1(C(C=C(CC)C)=O)CCN(C(=O)Cc2cc(C)[nH]n2)CC1C1CCCC1 1290,c1(OC)cc(C(N2CC(NC(=O)C(F)(F)CN(C)C)C(O)C2)=O)cc(Cl)c1O 1291,c1(C(=O)OCC)cnc(N2CC(NC(=O)CN=S(C)(C)=O)CC2C)nc1C 1292,C(=O)(CCC(F)(F)C(F)F)N1CCN(CCCNC(c2cnsc2)=O)CC1 1293,C1(C)(C(N(CCCNC(=O)CC(=O)Nc2nccs2)C)=O)CS(=O)(=O)C1 1294,Cc1ccc(C)c(C(N2CCNC(=O)C2C(C)C)C(=O)Nc2ccccc2)c1 1295,C1(NC(C(C)(C)OC(C)C)=O)CN(C(=O)CC2CCCC2)C2(CCOC2)C1 1296,N1(Cc2n(C)c(-c3ccc(F)cc3)cn2)C2CCC1CN(C(=O)C(C)(F)F)C2 1297,Cc1c(C(=O)NC2CN(C(C3CCC3(C)C)=O)CC2C)ccn1C(C)C 1298,C(CCSC)(C(=O)NCC(C12CCC(CC1)C2)NC(C1(C)CC1(Cl)Cl)=O)OC 1299,c1(C(=O)NC2(CCNC(=O)CSC3CCC3)CC2)cnn(CC2CC2)c1Cl 1300,c1(C(N(C2CCN(C(=O)CCCNC(=O)OCC)C2)CCC)=O)cnc(O)n1C 1301,C1(C(N2C(C#C)CC2)=O)CN(C(c2occc2COC)=O)CC12CC2 1302,c1(C(N2C3CCC(CNC(c4nc(C)oc4C)=O)(C3)C2)=O)cccc2ccsc12 1303,N1(C(CCc2scc(C)n2)=O)CCN(C(C2CCCC3CC23)=O)C2(CCC2)C1 1304,C1(CC)CN(C(=O)Cn2cc(C)cn2)CCC1NC(=O)C(C(F)(F)F)OC(C)=O 1305,N1(C(C(C)NC(=O)NC)=O)CC2(C)CN(C(C3(F)CCOC3C)=O)CC2(C)C1 1306,N1(CCC(N2C(CNC(c3[nH]cc(C(=O)OC)c3)=O)CC2)=O)CCOCC1C 1307,CC(C)C(C)C(=O)N1CCN(C2CCCC2NC(=O)CCC2CCOCC2)CC1 1308,C(=O)(CC(F)(F)C(F)(F)F)N1CCC(C)(CNC(C(C(C)C)n2cccc2)=O)C1 1309,N1(C(c2cc(C(C)C)on2)=O)CC(NC(C2CC2(Cl)Cl)=O)C2(CCOCC2)C1 1310,N1(C(C2(CC#C)CCCC2)=O)CC2CC(NC(C3CCS(=O)CC3)=O)C(C2)C1 1311,CCC(CC)C(C(=O)N1CCN(CCNC(C23CC(C)(CCO2)C3)=O)CC1)OC 1312,c1(-c2ccc(CNC(c3cnn(C4(CO)CCNC4)c3)=O)s2)ccnc(F)c1 1313,C1(NC(C(CN(C)C)(C)C)=O)CC12CCN(C(c1sccc1I)=O)CC2 1314,N1(C(CC(=O)OCC)=O)CC(CNC(C23CC(C)(CO2)C3)=O)CC1C 1315,C1(CNC(c2ccncn2)=O)CN(C(C2CC3(C2)CC(F)(F)C3)=O)CCC1(F)F 1316,N1(C(COCCN(C)C)=O)CCC(C)(NC(C2CCCN(CC(F)F)C2)=O)C1 1317,C=CCCC(C(=O)OC)NC(C1CN(C(c2cscn2)=O)C1)=O 1318,C1(CNC(CC2C(CNC(C(CC)OC)=O)C2)=O)CCC2(CC1)CC2 1319,c1(C(N2C3(CC#N)CC(C2)C3)=O)ccc(OC(F)(F)F)cc1F 1320,C(CCCCCN(C)C(C1CCOC1)=O)NC(C(C)c1cncs1)=O 1321,N1(C(CC2(C#N)CC2)=O)CCC2(CCC2NC(=O)CSCc2ccccc2)CC1 1322,C1(NC(c2cccc(C#C)c2C)=O)CC2CCC(C1F)N2C(C1(CF)CC1)=O 1323,Cc1ccc2c(c1)CC(NC(=O)N(C)C(c1cccs1)C)CO2 1324,C1=C(c2cc(N3CC4CCC3C4)cc(CN3CCCCC3)c2)CCNC1 1325,C(=O)(C1=CCCC1(C)C)N(C1CCCN(C(c2csc(C)c2C2CC2)=O)C1)C 1326,C1(c2nnnn2C)(NCC(C2CCOCC2)OCCOC)CCCC1CCCF 1327,N1(C(C=CSC)=O)CCCC(CNC(=O)C(F)(F)C2CCOCC2)CC1 1328,C1(CC(=O)NCCC(=O)NCC(=O)OC(C(=O)N(C)C)(C)C)CC2(CC2)CO1 1329,N1(C(c2n[nH]c(C)c2Cl)=O)CCC2C(C(=O)NC3(C)CCCC3(C)C)C2C1 1330,C1(C(=O)NC2C3CN(C(C(C=C)(C)C)=O)C2C3)Cc2cc(C)ccc2O1 1331,Cc1nc2c(o1)CCN(C(=O)C(CCOCCO)NC(c1ccoc1Cl)=O)C2 1332,c1(C(=O)NCC2C(NC(c3c(C#C)ccc(F)c3)=O)C2)csc2c(F)cccc12 1333,N1(C(CCC2CC(OC)C2)=O)CCN(C(c2ccc(O)cc2Cl)=O)C(C(C)C)C1 1334,c1(CCC)ncoc1C(N1CC(Cn2cc(-c3cnc(C4CC4)o3)nn2)C1)=O 1335,C1(NC(c2c(C)ncs2)=O)COC2(CCN(C(C3(C#N)CCCOC3)=O)CC2)C1 1336,c1(NC(C2C3CC2N(C(=O)CCCn2ccnc2)C3)=O)cnc(Br)nc1 1337,C1(CC)CN(C(c2ccc(Cl)cc2Cl)=O)CCC1NC(c1cnccc1C)=O 1338,C(CC)(C(=O)N1CC(C(C(=O)NC2(C3CC3)CCCO2)OCC)C1)=CCCC 1339,C1(C(N2C3(C(=O)Nc4c(OC)ncnc4)CC3CC2)=O)CCCCC(=O)N1 1340,C(=O)(C#CC1CCOCC1)NC(C1CCN(C(c2cc(Cl)cc(C)c2O)=O)C1)C 1341,C1(C(=O)NCC(C)N(C)C)CCN(C(C2(N3CCCC3)CC2)=O)C1 1342,c1(C(N2CC(CCNC(C(C)(C)SC)=O)OC(C)C2)=O)cc2cc(C)ccc2[nH]1 1343,c1(C(=O)NCC2(NC(c3cn(C)c(=O)cn3)=O)CC2)coc2ccc(F)cc12 1344,c1(C(=O)NC(CC)(C)CNC(=O)COCc2nc(CC)no2)cc(Cl)ccc1N 1345,C(=O)(C(CC1CCC1)C1CCC1)NCCCCN(C(=O)C(c1cccnc1)O)C 1346,c1(NC(C2(CC)CCN(C(c3cc(O)cc(=O)o3)=O)C2)=O)ccc(O)c(Cl)c1 1347,C1(C(=O)NCC(C)CN(C)C(C2CC3CC3C2)=O)CCc2ccnn2C1 1348,C1(OC)CC(NC(c2ccsc2)=O)CN(C(c2cncc(OC(C)C)c2)=O)C1 1349,C1(C(N)=O)CN(C(C2(F)CN(C(C3(c4cccs4)CC3)=O)C2)=O)CCC1O 1350,O=C(N=c1cc2ccccn2[nH]1)N1CCOC(C2CCCCC2)C1 1351,CCCC(C(=O)NC1CN(C(c2ccc(OC)c(OC(C)=O)c2)=O)C1)S(N)(=O)=O 1352,CC#CCCCC(=O)N(C(C)CNC(=O)C(c1ccc(N(C)C)cc1)C)CC 1353,C1(NC(C(CC)CC)=O)CC(F)(F)CC1NC(c1cc(Cl)c(Cl)s1)=O 1354,c1(CS(=O)(=O)NC(C)C(=O)NC(CNC(c2ncc[nH]2)=O)CO)ccccc1 1355,C1(O)(C(N)=O)CCCN(C(C2CSCCN2C(c2cc(Cl)cs2)=O)=O)C1 1356,c1(CC(N2C(CNC(CC=CCC)=O)CC2)=O)cc2ccccc2nc1O 1357,N1(C(c2c(COC)cc[nH]2)=O)CC(NC(=O)C=C(C)C(F)F)C(C)C1 1358,C1(NC(C2C(CNC(CNS(N)(=O)=O)=O)OCC2)=O)C2C=CC(C2)C1CO 1359,C1(NC(C(C=C=C)C)=O)CN(C(=O)C(F)(F)C=Cc2ccccc2)CC12CC2 1360,C1(NC(C(C)OCCCC)=O)CCC(O)CN(C(C2(c3ccn(C)n3)CC2)=O)C1 1361,c1(CNC(C(=O)Nc2c(C(=O)OC)scc2)=O)cccc(NC(C)=O)c1 1362,C1(C(N(C2(CO)CC2)C)=O)CN(C(=O)CC2CCSC2)CCC1(C)C 1363,N1(C(C(CC)C#N)=O)CC2C3CCC(C2C1)N(C(C1CC1(C)C(F)F)=O)C3 1364,CCC(C(=O)NC(C)(C)CN(C(=O)CCc1ncccc1C)C)C(C)O 1365,C1(C(C)C)CCC(C(=O)N(C)CC2CCCN(C(C3(CO)CCCO3)=O)C2)CC1 1366,N1(CC(N2CC(CN(C)C(C3COCCO3)=O)C2)=O)CCCCC1=O 1367,c1(C(N2C(CNC(CCC#C)=O)CC(O)C2)=O)cc(OC)cc(F)c1 1368,CO[Si](C)(CCCOC(=O)CCc1ccc(F)cc1C)OC 1369,C12(NC(CC(=O)OC)=O)CCC(CCC3C(C)CN3C(C)=O)(C1)OC2 1370,CCCCC(C(=O)N1CCC(C)C1CNC(=O)C(C(C)C)SC)C(C)C 1371,N1(C(CCCOC)=O)CCCC2(NC(=O)C=CCOc3ccccc3)CC12 1372,N1(C(CCCC=C)=O)CCN(C(C23CC=CC(C2)OC3)=O)C(CC)C1 1373,c1(C(N2CC(NC(CSC(C)C)=O)C(C)(C)C2)=O)c(F)cccc1[N+](=O)[O-] 1374,c1(C(=O)NC2CC3(C2)CC(NC(C2CC2(F)Cl)=O)C3)cc2cccnn2n1 1375,CCC#CCN=c1nc(N2CCC(c3ccccn3)CC2)c2c([nH]1)CCC2 1376,c1(C(=O)NCC(CO)NC(CCNC(N)=O)=O)coc2c1C(=O)NCC2 1377,c1(NCC2CC(NC(c3nc(NC(C(C)C)=O)sc3)=O)C2)ccccc1[N+](=O)[O-] 1378,CCC(CC(=O)NC(CC(F)F)C(=O)N1CCCC(C(C)C)CC1)CC(C)C 1379,CN1CC=C(CC(=O)NC2CCN(C(C3CC3C(=O)NCCO)=O)C23CCC3)CC1 1380,Cc1cc(Cl)cc(C(N2CC(NC(C3(F)CCC3)=O)CC(C)C2)=O)c1N 1381,C1(C(=O)NC(C)(CNC(c2cnn(C(F)F)c2)=O)CO)COC2(CCC2)CO1 1382,c1(C(N(CC(CO)(CO)NC(C(C)NC(C)=O)=O)C)=O)c[nH]c2c(F)cccc12 1383,C(C(O)CCNC(C1CCC12CC2)=O)NC(CSCCC(C)C)=O 1384,C(=O)(C(CNC(c1ccc(C)nc1)=O)C(C)(C)C)NCCC(COC)O 1385,c1(CC(=O)N(CCCNC)C)cnoc1.C1(C(=O)NOC(C)(C)C)(CF)CCC1 1386,C12(NC(C3C(C)(C(C)C)C3)=O)CCCN(C(c3cccc4[nH]ncc34)=O)CC1C2 1387,N1(C(C23CC(C(C=CC(=O)NC4CC4)=O)C2C3)=O)CCC2(CCC(OC)CC2)C1 1388,N1(C(c2ccc(C(C)(C)C)o2)C(=O)NCCCC)CCCC(COCCOC)C1 1389,C(=O)(N=c1ccn(CC#N)[nH]1)OS(N(C)CC)(=O)=O.c1(CCC)cc(Br)ccc1 1390,C1(NC(C(C)CC#N)=O)CC(F)CN(C(c2nnc(O)cc2O)=O)C1 1391,C(C1=NOC2CCCCC12)n1cc(CCN(C)C)nn1 1392,Cc1ccc(N)cc1C(N1CC2(C1)CN(C(=O)C(c1ccccc1Cl)O)C2)=O 1393,C1(C(N2C(CCNC(C(C)C3CCCC3)=O)CCCC2)=O)CCC([N+](=O)[O-])CC1 1394,C1(NC(CCSC)=O)CCN(C(c2cnnn2C2CC2)=O)C1c1cn[nH]c1 1395,c1(-c2cn(C(CNC(c3cc(OC)n[nH]3)=O)C)nn2)cccc(F)c1N 1396,N1(C(C2CCC(C)CC2)=O)CCOC2(CCN(C(=O)C=C3CCC3)C2)C1 1397,N1(C(c2n[nH]cc2Br)=O)CCC(C2CC2)C1CNC(C1(CCF)CCC1)=O 1398,c1(C(N(C2CCN(C(CCC(=C)C)=O)CC2)C)=O)c(Cl)cccc1[N+](=O)[O-] 1399,N1(C(CSc2nc(C)[nH]n2)=O)CCCC2(C1)CN(C(c1nc(C)n(C)c1C)=O)C2 1400,C12(C(N3CC(NC(c4c[nH]nc4CC4CCOCC4)=O)C3)=O)C3C4C5C3C1C5C24 1401,C1(C(=O)NC2(COC)CC2)CCCN1C(C)C.C1=CC(=O)NC1(C)C 1402,C(CC(C)(C)C)(C(=O)NCCCC1(O)CCC1)NC(C(CCC)C)=O 1403,c1(SC)ccc(C(N2CC3CC3(CNC(=O)CC(C)C)C2)=O)cc1Br 1404,c1(C(=O)NC2(CC(=O)NC3CC(CC)(CC)C3)CC2)cccc(F)c1O.O 1405,N1(C(CC2ON=C(C)C2)=O)CCCC(CN(C(=O)C(c2ccc(Cl)cc2)O)C)C1 1406,c1(C(=O)NC2C=CC(CNC(c3n(CC)ncc3)=O)C2)c(F)cccc1F 1407,C(c1cc(F)c(F)c(F)c1)=CC(N1CCC(N(C(C(C)OC)=O)C)C1)=O 1408,N1(C(c2c(C)c[nH]n2)=O)CC(C(=O)N(C2CCCC2C#N)C)CC(C)C1 1409,C1(NC(CCn2c(C)csc2=O)=O)CC2(C1)CC(NC(C1(C3CC3)CC1)=O)C2 1410,N1(C(C2CN(C)C2)=O)CCC(NC(=O)CC(O)C2CC2)C2(CCC2)C1 1411,c1(CNC(CN2CCN(C(CC(C)N(C)C)=O)CC2)=O)ccc(C#N)cc1F 1412,C(=O)(C1CCCc2nncn21)N1CCC2(C(CNC(c3cn[nH]c3)=O)C2)CC1 1413,c1(C(=O)NCC(CNC(c2c(CC)nns2)=O)(C)O)ccc2ncncc2c1 1414,CON=C(C(=O)NCC1(C)CCN(C(=O)C2CC2)CC1)c1ccco1 1415,n1(C(C)(C)C)nc2c(c1C(=O)NCCCNC(c1cc(Cl)ccn1)=O)CCCC2 1416,Cn1c(=O)[nH]c(NCC2CCN(c3ccccc3Cl)C2)c(C#N)c1=O 1417,C1(CC#C)(C(=O)O)CCN(C(C2CCC(N)CC2)=O)CC1 1418,c1(C(N2CC3C(C(N4CC(C)NC(=O)C4)=O)(CC3)C2)=O)ccn2cncc2c1 1419,Cc1nc(C(=O)NCC2CC2CNC(c2ccc(Br)s2)=O)cn1C 1420,c1(NC(C2COCCN2C(=O)CCCc2ccccc2)=O)ccc(Br)cc1CO 1421,C1(C(=O)NCCN(C(COCC=C)=O)CCC)CC(C)CO1 1422,CC(C)(C)CC(=O)NC1CC2C(NC(=O)COC3CCCOC3)C2C1 1423,Cc1ccc(CC(=O)NCCC2(OC)CN(C(C3CCC(C(N)=O)O3)=O)C2)cc1 1424,c1(C(N(CC(N2CC(OC)C2)=O)C2CC2)=O)coc(CO)c1 1425,c1(C(=O)NCC(c2ccccc2F)NC(C(C)OC)=O)nsc2c(Cl)cccc12 1426,n1(CCCC)nnnc1C(CCC1CC=CCC1)NCC=C(C)C 1427,CC1CCN(C(c2cnn(-c3ccc(F)cc3)n2)=O)CC1NC(c1cnns1)=O 1428,C1(=O)CC(O)CN1CC.C1CCCS1.C(=O)(COCC(=O)NCC)NC.N(C)C 1429,C1(C(=O)Nc2cn(CC#C)nc2)CC2C=CC1N(C(=O)Cc1cnn(CC)c1)C2 1430,c1(SC)cccc(C(=O)NCC2(O)CCN(C(=O)C(c3cnn(C)c3)O)C2)c1 1431,C(N=c1cc(C)nc(Cl)[nH]1)C1CN(C(C2(COC)CCCCO2)=O)C(C)C1 1432,C=CC(C)(O)C(=O)NCC(C)(C(C)C)NC(c1cc(Cl)sc1Cl)=O 1433,C1(C(N2CCC(NC(C(C(C)C)n3cnnn3)=O)C2C)=O)CCCCC(C)(C)C1 1434,CC1CCC(CC(N2CC(CC(F)C(=O)N3CCC(CCCO)C3)C2)=O)C1 1435,N1(C(c2c(C)nsc2)=O)CC(N(C)C(c2cncs2)=O)C(F)C1 1436,CCC(CC(=O)N1CCCC1CCc1ccncc1)NC(=O)CSC 1437,C=CCC(CC(C)C)C(=O)N1CCCC(C)(C)C1CNC(C1(C(C)C)COC1)=O 1438,c1(C(C2(n3cc(Cl)cn3)CC2)NC2CN(C(C)=O)C(C)C2)ccccc1F 1439,CC1CCCC1(C)NC(=O)CCN(CCCO)C(C1CCC(N(C)C)C1)=O 1440,CC1CCCC(O)(C(c2c(F)ccc(NC3COCC4CCCC34)c2)=O)CC1 1441,Cc1nc(CC(C)C)sc1C(=O)NC1CCC(CNC(c2n[nH]c(=N)s2)=O)C1 1442,c1(NCc2ncc(CC)[nH]2)ncc(Br)c2cccnc12 1443,N1(C(C23CCC(C)(CC2)OC3)=O)CCCC2CN(C(C3CC3C3CC3)=O)CCC12 1444,C(=O)NNc1c(Cl)cccc1Br.O=C1CCC2CC12 1445,c1(Nc2cc(C(=O)OCC)sc2C)c(Cl)ccnc1Br 1446,c1(C(N2C(C(N3C(COC)C(O)CC3)=O)CC2)=O)ccc(C)c(C#N)c1 1447,C1(C#CC(=O)N2CCC(O)C2CNC(=O)CC2CC3(CC3)CO2)(CC)COC1 1448,N1(C(CCC(C)(C)F)=O)CCC2(CCCN(C(=O)CC(C)(C)C3CC3)C2)C1 1449,n1(CC)cc(NC(C2CC(C)CN2Cc2cnc(N(C)C)nc2)=O)c(C)n1 1450,N1(C(=O)NC(C)(CO)C(F)F)CCC2(C1)CN(C(c1ccccc1)=O)CCO2 1451,C#CCC(C)(C(=O)NC(c1ncccn1)CC)NC(=O)CC1CCC(=O)N1 1452,c1(C(=O)NCC2CC(OC)CN2C(c2cnnn2C)=O)cc(Br)cnc1N 1453,c1(C(N2CC(CN(C(c3cc(C)n(C)n3)=O)C)OCC2)=O)ccn2cnnc2c1 1454,c1(OC)ccc(C(=O)NCC2CC(F)(CNC(C3(F)CC3C)=O)C2)c(F)c1 1455,c1(C(=O)NCC2(F)CCC(NC(c3c(C)noc3)=O)C2)cnc2ccccn12 1456,n1(CC(N2CCCC(N(C(C(CCC)C)=O)C)C2)=O)ncc(C#N)c1Br 1457,C1(C(N(CCC(=O)NCC2(C3CC3)CCC2)CC#C)=O)CCCC(C#N)C1 1458,c1(C(N(CC(C)NC(=O)CCc2cn[nH]c2)CC)=O)ccc(SC(F)(F)F)o1 1459,C1(C(=O)Nc2cccc(CNC(C(CC)O)=O)c2)Cc2cc(C)c(C)cc2O1 1460,CCCCCC(O)CC(=O)NC(CNC(=O)CCOc1cccnc1)CCC 1461,C(=O)(CC1=NNC(=O)C1)NCCC(CCNC(C=CCCC)=O)C 1462,N1(C(c2c(C(C)C)c[nH]n2)=O)CCC2CN(C(c3csc(C(N)=O)n3)=O)CC2C1 1463,C(=O)(C1=C(C#N)CCC1)N1CCC(OC)(CNC(C2CN(C)C2)=O)CC1 1464,C(C(=O)N(C)CC1C2CN(C(=O)C=CC(F)(F)F)CC12)(C(C)C)n1ncc(C)c1 1465,N1(C(c2c[nH]c(=NC)s2)=O)CCN2CCN(C(=O)C(C)OCC3CCCO3)CC2C1 1466,C12(C(=O)NCC3CCN(C(C)=O)C3)CC(NC(C3CCCSC3)=O)(CCO1)C2 1467,C1(CC#C)(C(=O)NC(C)CC(C)NC(c2ccc(F)o2)=O)CCCCO1 1468,C1(C(=O)NC(CN(C)Cc2cn(CCCC)nn2)C)CCC(N(C)C)CC1 1469,C(=O)(C1=CS(=O)CCC1)N1CCC(CNC(C(C)SC(F)(F)F)=O)CC1 1470,Cc1cc(=NC2CCC(N(C)C)C2)[nH]c(NCc2[nH]cnc2C)n1 1471,O=C(C=CCC(=O)NCCN1CCCCC1)NOCCF 1472,n1(CC)c(C)cc2c1CCCC2NC(=O)C(=O)NCC1OC(=O)CC12CNC2 1473,c1(OCC)cc2[nH]ncc2cc1NC(C1CN(Cc2ccc(C)o2)CCO1)=O 1474,N1(C(c2ncn(CCNC(C(C)n3cccc3)=O)c2)=O)CCCCCC1C 1475,N1(C(C2C(COC)CC2)=O)CCc2ccccc2C1CO 1476,c1(C(=O)NC2C(CNC(COC(C)C)=O)C2)coc(Cl)n1 1477,C1(CNC(=O)C(O)CC2CCCCC2)COCCN(C(C2CCCS2)=O)C1 1478,C1(C(=O)Oc2c(OC)cc(Br)cc2)CC2(C1)CC(N=[N+]=[N-])C2 1479,C1(NC(Cc2ccc(C)cc2)=O)CCN(C(c2ccc(C)n2C)=O)CC1C(N)=O 1480,c1(C(=O)NC(CN(C(c2cc(CC)on2)=O)C)(C)C)sc2nccnc2c1N 1481,O(NC(=O)C(c1cn(C)nn1)NC(c1cc(C)[nH]n1)=O)C(C=C)C 1482,CC1CCN(C(=O)C(O)CC2CCCC2)CC1CNC(c1ccc(C2CC2)nc1)=O 1483,c1(OC)cc(CN2CCC(NC(c3cccc(F)c3I)=O)C(F)C2)ccc1C 1484,CN1C(=O)CSC1=CC(=O)NCC1CN(C(C2COC(C)(C)O2)=O)CCCO1 1485,C1(C2CCN(C(=O)C(F)=CCCF)CC2)(NC(C=C(C)C(C)(C)C)=O)CC1 1486,N1(C(C2C(C)(C(C)C)C2)=O)CC2CC1(CNC(=O)CN1CCOCC1)C2 1487,Cc1nccc(Cl)c1C(N1CC(N(C(=O)C(Cl)=CCl)C)C(C)(C)C1)=O 1488,N1(CC(=O)NCC2CC(F)(F)CN2C(=O)CCc2ccco2)CCCNS1(=O)=O 1489,c1(NC(C2(C)CCN(C(=O)Cn3cc([N+](=O)[O-])cn3)C2)=O)ccc2oncc2c1 1490,Cc1csc(C(=O)NC2(C(=O)N(C)CC3(O)CCOC3)CC(O)C2)c1 1491,N1(C(C2CCN(C(=O)OCC)CC2)=O)CCCC(NC(C2CC(C)(O)C2)=O)C1C 1492,C1(CNC(C2CCC(=C)CC2)=O)CC2CN(C(=O)Cc3coc(C)n3)CC12 1493,c1(OCCC)cccc(C(N2CC(O)CC2CNC(c2cnnn2C)=O)=O)c1 1494,C(C(C)C(F)C(=O)NCC1CCC(=O)NC1C)NC(CC=CC=C)=O 1495,C12CCN(C13CCC3)C2=O.O=C(CCCOc1ccccc1)NC1CC1 1496,Cc1cc(C)n(CC(=O)NC2(Cn3cc(-c4cscn4)nn3)CC(F)(F)C2)n1 1497,C1(CNC(CNC(=O)NC)=O)(NC(=O)C(CO)NC(N)=O)CCOC1.C(C)C 1498,C1(CC)CCCC1(C)C(=O)NCC1CCCC1NC(C1CCC(=O)N1)=O 1499,C#CCCN=C(NCC1CCCC(C)(C)C1)NC1CC(CS(N)(=O)=O)C1 1500,N1(C(C)C)CCC(CNC(=O)C(O)CNC(=O)C(F)=CC2CC2)C1 1501,C1(NC(C(c2cn(C)nc2)O)=O)CC2(C1)CN(C(C1CNC(=O)C1)=O)C2 1502,CC(C(=O)NC1CCCN(C(=O)C(=O)NCC(F)F)CC1)C(F)(F)C(F)F 1503,Cc1ccccc1C(N1CC2C(NC(C3(C(C)(C)C)CCCCC3)=O)C2C1)=O 1504,c1(C(c2n(C(C(=O)OC)C)nnn2)NC2C(C)C2(C)C)ccc(OC)nc1 1505,C1(NC(C(C2CCCCC2)OC)=O)C2CCCN(C(=O)COC(F)F)C2C1(C)C 1506,c1(C(N(C2CCCN(C(C3CCCCN3C)=O)C2)CC)=O)[nH]c(O)nc1C 1507,c1(NC(N(CC(C)OC)Cc2ccccc2)=O)ccc(O)c(Br)c1 1508,N1(C(C(CC)C(C)O)=O)CCC2CC(NC(c3cc(F)ccc3Cl)=O)CCC2C1 1509,N1(C(CC(=O)NCC#C)=O)CC2CC(NC(=O)CC3COCC3(C)C)C(C2)C1 1510,c1(C(N2CCN(C(C3(CF)CC3(F)F)=O)CC2)=O)cc(F)cc(Cl)c1O 1511,C(=O)(C(C)CC(=C)C)NCCCCN(CCCNC(CC=C=C)=O)C 1512,C1(OCC)CN(C(=O)C=Cc2csnc2C)CC1CNC(=O)CSC1CCCO1 1513,c1(C(=O)NC(CC)CNC(=O)C(=O)NC(C)C)sc(C(C)C)nc1C 1514,CCCC(C)CCN=c1[nH]ccc(=NCCOc2ccc(Cl)cc2Cl)[nH]1 1515,CC(C(=O)OCc1ccccc1)C(C)CN(C)C(c1cccnc1N)=O 1516,c1(C(c2n(CCSC)nnn2)NCc2cc(C)ncn2)ccc2nsnc2c1 1517,Cc1[nH]c(C)c(C(=O)NC2CC(NC(c3ccoc3C3CCN(C)CC3)=O)C2)c1C 1518,S(=O)(=O)(c1cccc(=NC2CCC(F)(F)C2)[nH]1)NCc1c(C)nc(C)c(C)n1 1519,C1(OC)CC(N=c2[nH]c(N3CCc4nc(N(C)C)sc4C3)nc(=N)[nH]2)C1 1520,C(=O)(C(C)(O)CCC)NCC(CC)NC(c1nn(-c2ccccc2F)cc1Br)=O 1521,N1(C(C2ON=C(C)C2)=O)CCN(C(c2cnccn2)=O)CC1c1cccc(F)c1 1522,CN1C(=O)NCC1C(=O)NCCN(C1CCCC1)C(c1ccc(F)cc1)=O 1523,C1(C)(CNC(C(C)C2CCOC2)=O)CCCN1C(=O)CS(=O)(=O)NC1CC1 1524,N1(C(c2cc(C)c(Cl)cc2Cl)=O)CCC2(CC(NC(=O)C=CC3CC3)CO2)C1 1525,C(=O)(C#CC1CCOCC1)N1CC(NC(c2csc(C)c2C)=O)CC(F)(F)C1 1526,N1(C(=O)C(F)(F)CC2CC2)CCc2ccccc2C1C(F)(F)F 1527,C1(CN(C)C(C2CC23CC(NC(C24CCC(C2)C4)=O)C3)=O)CCCCC1(C)C 1528,C#CCC(C)(CC)C(=O)N1CCC1CNC(C1(O)CCSCC1)=O 1529,Cc1ccc2c(N(CC(F)F)C)nc(N(C)CC3CCCS3(=O)=O)nc2c1 1530,C(C)(C(CC(=O)NCCN1CCCCC1)NC(=O)Cc1ccc(F)nc1)OC 1531,C1(NC(c2n(CC)nc(C)c2)=O)CCN(C(=O)CC2CCC3CC3C2)CCC1CO 1532,CC(C(C(=O)NCCCOCC1CC1)N1CCCC2(CC1)CC2)C(C)(C)C 1533,C1(CNC(c2cn(CC(C)C)nc2C(F)F)=O)CCCCN(C(=O)C=C(C)Cl)C1 1534,c1(CCC(=O)NC(CCNC(C2C(C(=O)OC)CCC2)=O)C)ccccc1OC 1535,CCCCCC(=O)NC(CO)C(C)NC(c1cccnc1S)=O 1536,Cc1cc(F)ccc1CC(=O)NCC1CC(NC(=O)C(C)(C)c2ccccn2)C1 1537,N1(C(c2ncn(CC)c2)=O)CCC(NC(=O)C(N)=O)C(C)C1 1538,N1(C(CN(C)C(N)=O)=O)CCCC(O)(CCNC(=O)C(O)Cc2ccccc2)C1 1539,C1(O)(CNC(=O)CN2CCCC2)CCCN(C(C2CCCS2)=O)CC1 1540,C(=O)(C(CO)c1ccccc1)NC(C1CCN(C(=O)CCc2cc[nH]n2)C1)(C)C 1541,n1(CC)ccc(CN(C(=O)COCCN(C(=O)C(C)C2CCOC2)C2CC2)C)n1 1542,c1(C(=O)NCCCN(C(CC2CC(CC)C2)=O)CC)ccc(F)cc1CC 1543,N1(C(CC(C=C)CC)=O)CCC(C(=O)N(C)CCc2ccccc2)C(C)(C)C1 1544,C1(NC(C2C=CCN(C(c3ccccc3)=O)C2)=O)CC2(CCC2)C1O 1545,C1(C(N2CCN(C(CC(n3ccc(C)n3)C)=O)CC2C)=O)CC2CCCCN2C1 1546,C1(CC(=O)NCC2N(C(C(C(C)C)OC)=O)CCC2)CCC(=O)NC1=O 1547,Cc1nc2ccc(CN(C3CCC(=O)NC3)C)cc2s1 1548,C1(N(C)C(C23CCC(C2)C3)=O)CCCC(NC(C2(C)CC2)=O)C1 1549,C1(CC(=O)NCC2CCC(C)C2)CCN(C(=O)C2=NNC(=O)C2)C1(C)C 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1568,C1(C(=O)NCC2CC(CC)C2)(OC)CCN(C(=O)CN(C)CCOC)C1 1569,CCCC(CCCNC(c1cc(CO)n(C)n1)=O)NC(C1(O)CCC1)=O 1570,c1(C(N(C(C)CCNC(=O)CC2CC2C2CC2)C)=O)ncc(C(F)(F)F)cc1Cl 1571,CC1(C)CC(NC(C2CC2F)=O)CCN(C(=O)CCc2cc(Cl)cs2)C1 1572,C1(C(=O)OCC)(C(=O)NC2CCN(C(c3cn(CC)nc3C)=O)C2)CCOCC1 1573,N1(C(C(C)(F)F)=O)CCCC(C2CCN(C(C3(C#N)CC4CCC3CC4)=O)C2)C1 1574,CN=c1[nH]c(C(N2CCN(CCNC(C3CC34CCOC4)=O)CC2)=O)cs1 1575,C1(CNC(c2n(C(C)(C)C)ncc2)=O)CN(C(C2CC2(F)F)=O)CCC1(C)C 1576,c1(NCC2(COC)CC(F)(F)C2)nccc(=NC2CCC3(CCCCC3)CC2)[nH]1 1577,N1(C(c2c(CC)oc(C)c2)=O)CC(CNC(C2(CC)CC2(F)F)=O)CC12CCC2 1578,c1(C(=O)NC(C)C(F)(F)F)cccc(S(=O)(=O)NCCC(O)C2CCCC2)c1 1579,Cn1ccn2ncc(CNC(=O)NC3CC3c3ccccc3)c12 1580,c1(N2CCC(NC(c3ccc(C)cc3)=O)C(C)C2)cc2nncn2c(C)n1 1581,C1(CC)CN(C(=O)C(C)(O)COC)CCC1NC(=O)CCCOC 1582,C(=O)(C(C)CCCC(C)=O)N1CCC(CCOC)(C(N2CC(C)C(O)C2)=O)CC1 1583,c1(N(CCOCC=C)C)nc(N2CCc3scc(Br)c3C2)c2c(n1)c(C)nn2C 1584,N1(C(CCS(CC)=O)=O)CC2CCN(C(c3nc4ccccc4[nH]3)=O)C2C1 1585,CCC(CC(=O)N1CC(CC(F)C(=O)N2CC(N3CCC3)C2)C1)C(C)C 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1691,c1(C(c2cn(C3CN(OC)CC3C)nn2)C2CC2)cc(N)c(=O)n2c1CCCC2 1692,c1(N(CC=C)C)ccc(S(=O)(=O)N2CCCC(O)C2)cc1C#N 1693,c1(C(=O)NCC2(C(C)NC(C3(CO)CCC3)=O)CC2)ccc(F)cc1C1CC1 1694,C1(C(=O)NCC2N(C(C(C(C)C)N(CC)CC)=O)CCOC2)CCCCCCC1 1695,S(=O)(=O)(c1cn(C)cn1)NC1CN(C(c2c(C)cc(C)s2)=O)C1.C1(=O)CN1C1CC1 1696,CC1(C(=O)NC2C=CC(CC(=O)NCCc3noc(=O)n3C)C2)CC=CCC1 1697,N1(C(c2c(C)nn(CC(F)F)c2)C(=O)N(C)C)CCNC(=O)CC1(C)C.C1CCN1 1698,N1(c2nc(C(C)C)nc(Cl)c2)CCS(=O)(=O)C(CCNC(=O)CC=C(C)C)C1 1699,N1(C(CC)=O)CCC(C)C(NC(=O)N(C(C2CCCCCCC2)C)CC)C1 1700,N1(C(c2cc(C)ns2)=O)CCC(NC(=O)Cc2ccsn2)C1C 1701,Cc1nc(O)ccc1C(N1CC=C(CNC(=O)C(C)CN(C)C)CC1)=O 1702,c1(C(N2CCOCC2)=O)ccc(Br)cc1.c12ccccc1CNC(=O)NC2 1703,c1(CN=c2ccnc(-c3ccc(OC)c(F)c3)[nH]2)ccc2[nH]cc(C#N)c2c1 1704,C1(NC(C2OCCN(C)C2)=O)CCN(C(=O)C=Cc2ccccc2F)CC1(C)C 1705,CN1CC=C(CC(=O)NCC2COCCN2C(=O)Cc2c(O)ncnc2O)CC1 1706,C1(C)(C(=O)NC(C)CNC(=O)C(Cc2ccccc2)n2cnnn2)COCCO1 1707,c1(C(=O)NC2(CN(C(=O)COC3CCOC3)C)CC2)ccn2nncc2c1 1708,C1(NC(C=NOC)=O)(CO)CCCN(C(=O)C(c2ccnn2C)C)C1 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1727,n1(CC(=O)N(CC(CO)(CO)NC(C2CC(C)(C)CO2)=O)C)cnc([N+](=O)[O-])c1 1728,C(C)(CO)(C(=O)NC1CC1NC(=O)CCc1ccccc1Br)OC 1729,c1(C(N(C2CN(C(c3c(F)ccc(F)c3N)=O)C2)C)=O)cccn2c(O)nnc12 1730,c1(OC)nc(N2CCC(C(=O)N(CC(c3ccccc3)O)C)C2)ncc1C#N 1731,CCCC(CNC(=O)CCNC(=O)CO)C(=O)NCC1COC(=O)N1 1732,N1(CC=CC(=O)NCC(C)CN(C)C(c2cn[nH]c2)=O)CCOCC1 1733,c1(CC(=O)NC2C3(CC(NC(C4N(CCC)CCC4)=O)C3)C2)cccc(F)c1F 1734,N1(c2cn(C)nc2[N+](=O)[O-])C(=O)NC2(CCN(C(=O)Nc3cccs3)C2)C1=O 1735,C1(NC(c2cc(Cl)c(Cl)[nH]2)=O)CN(C(c2cnn(CCF)c2)=O)CC2(CCC2)C1 1736,C1(COC)CC(N=c2[nH]c(=NCc3ccoc3C)[nH]c3c2CC(C)CC3)C1 1737,C(=O)(C1Cc2ccc(Br)cc21)OCc1cnc(C2(C)OCCO2)s1 1738,C1(CNC(C(CC#C)O)=O)CCN(C(c2scnc2CC)=O)CC1(F)F 1739,c1(C(N2CCC(CNC(C(C=C=C)C)=O)C2)=O)cc(C)nc2ccnn12 1740,CC(C)CC(CNC(C1CCCN1C=O)=O)NC(=O)C(C)(C)COCC(F)F 1741,c1(C(C(=O)NC(C)(C)C)N(CCC#C)C)cc(CC)cc(C)c1 1742,CN1CC(C(=O)NCCC2(NC(c3c[nH]c(C#N)c3)=O)CCC2)CCC1=O 1743,c1(C(N(CC(C)N(C(C(C)OCCC=C)=O)C)C)=O)ccc(Cl)cc1O 1744,C1(C(=O)NC(C)CCNC(c2cccnc2)=O)CCN(CCF)CC1 1745,c1(CN2C(CCNC(C3(C=C)CCCCC3)=O)CCCC2)ccc2c(c1)COC2 1746,C1(C(=O)NCC2(NC(c3cc(N)nc(Cl)c3)=O)CCC2)Cc2ccccc2O1 1747,n1(Cc2cn(CCC(=O)NCC(c3ccc(C)o3)O)nn2)ccc2ccccc12 1748,c1(C(=O)NCC2N(C)CCN(C(=O)CCn3ccnc3)C2)cccn2cncc12 1749,c1(OCCCC(=O)OCC2C3CCC23)ccc2ccccc2c1 1750,C1(C)(NC(c2c(C)csn2)=O)CCN(C(c2cc(Cl)n[nH]2)=O)C1 1751,CCC(C)(C)C(=O)C(=O)N1CCC(C2CCCN2C(c2ccc(Cl)o2)=O)C1 1752,c1(C(N(C2CN(C(CN(C)C)=O)C2)C)=O)cc(=O)cc[nH]1 1753,C(=O)(C1=CC2(CCOC2)C1)N1CCC(C(N(CC(CC)CC)CC)=O)CC1 1754,c1(C(=O)NC2C(CNC(c3scc(OC)c3OC)=O)C2)ccc2occ(C)c2c1 1755,C1(C2CCCN(C(C3C(C)(C)C3(F)F)=O)C2)(NC(C=C(CCC)C)=O)CC1 1756,c1(OC)ccc([N+](=O)[O-])cc1C(N1CCN(C(=O)Nc2nnc(C)s2)CC1)=O 1757,c1(C(=O)NC(C(=O)NC(CC#C)CCOC)CCC)cccc(C#N)c1C 1758,c1(CN2C(CC(=O)NC(C3CCCC3)C)CCC2)c(F)cccc1F 1759,c1(CNC2C(C(=O)NC(c3cncs3)C)CCC2)c2c(nn1C)CCC2 1760,c1(N(C(C2N(C(C(CC)Br)=O)CCC2)=O)C)cc(C)cnc1C(N)=O 1761,C1(O)(CC)CCCN(C(=O)C=CCNC(=O)CCn2nc(C)nc2C)C1 1762,Cc1nc2cc(C(=O)NCC(O)CNC(=O)CC3=CCN(C)CC3)cc(O)c2o1 1763,CC(C)CCC(F)C(=O)N1CCCC(C)(C)C1C(=O)N(C1COC(C)(C)C1)C 1764,C1(C)(NC(C2C(C)OCC2)=O)CCN(C(C2CCN(c3ccccc3)C2=O)=O)C1 1765,C(=O)(C(C)CCCOC)NCCCC(C)(C)NC(c1cc(CCCCC)[nH]n1)=O 1766,C#CCCCC(C)C(=O)NCC(CO)NC(c1cc(C(N)=O)[nH]n1)=O 1767,C(C(CC(=O)N1CCC(C)(N(C)C)C1)NC(C1CCC(CO)CC1)=O)OC 1768,C(=O)(C1CCOc2ccc(F)cc21)N1CC(CNC(C(Br)=C(C)C)=O)C1 1769,N1(C(C23C(C)(C)C(CC2)C3)=O)CCCCC(NC(C2CCCC3(CC3)C2)=O)CC1 1770,Cc1[nH]c(C#N)cc1C(=O)NC1(CO)CCN(C(C2CC(C)(C)CN2C)=O)C1 1771,CP(C)(=O)CCC(=O)NC1CCN(C(=O)CCCc2csc(=N)[nH]2)C1 1772,Cn1ccc2c(C(=O)NCCC3CN(C(=O)Cn4ccnn4)CCO3)ccnc12 1773,c1(SCC(=O)NCC2(COC)CN(C(C3CCC3(C)C)=O)C2)ccccc1Br 1774,c1(CC(=O)NC(CNC(c2n(CCC)ccc2)=O)C2CCC2)cnc(Cl)cc1C 1775,S(=O)(=O)(c1cccc(NC(=O)CNC(=O)NC(c2nc(=O)o[nH]2)C)c1)NC 1776,Cc1cnn(C)c1C(=O)NCC(c1ccccc1)N(C(=O)CCS(C)=O)C 1777,C(CCC(=O)NC(C)CNC(=O)CCc1nc(C)no1)=C(C)C 1778,C12(NC(CC3CCC(C)CO3)=O)CC(CNC(c3cncc(N)c3)=O)(C1)OC2C 1779,C1(C(=O)NC(c2nc(=O)o[nH]2)C)CC12CCN(C(c1ccc(C3CC3)cc1)=O)C2 1780,CS(=O)CCC(=O)N1CCCC(N(c2nccc(C(F)(F)F)n2)CCO)C1 1781,C1(C(=O)NC2(C(O)CO)CC2)CCCC2CN(C(=O)C3Cc4ccccc43)CC12 1782,N1(C(C2CCC3C(C)(C)C2C3)C(=O)NC2CC2)CC2CS(=O)(=O)CC2C1 1783,N1(C(C(C)OCCCCCC)=O)CCCC(N(C(=O)C(c2ccc(Cl)s2)=O)C)C1 1784,c1(NC(CC)(CNC(=O)C(C2CCCOC2)OC)CC)c(Cl)cncc1[N+](=O)[O-] 1785,Cc1noc(C)c1C=CC(=O)NC1CC2(C1)CC(NC(c1nonc1N)=O)C2 1786,c1(CC(=O)NC2CCN(C(C=CC(CC)C)=O)CC2CO)cn2ccccc2n1 1787,c1(OC)ccc(Cl)cc1C(=O)NC(C)CNC(c1cccc(F)c1O)=O 1788,CC(CC(F)(F)F)C(=O)NC(CC1CC1)C(=O)N1CC(N2CC(F)C2)C1 1789,c1(OC)c(NC(C2CSCCN2Cc2ncc(C)s2)=O)ccc(Cl)c1Cl 1790,C1(C(=O)NCCCOCCN(C)C)(COC)CCCN1C(=O)C(C)(F)F 1791,c1(CCC)cccc(C(=O)N(C)CC2COCCN2C(=O)CN(C)C(=O)OC)c1 1792,C1(CC(=O)NCCC(CNC(=O)CC(=O)Nc2nccs2)O)CC2C=CC1CC2 1793,c1(CNC(=O)OC2CN(C(=O)C3CC3)C2)ccc(I)nc1 1794,N1(C(C(C(CC)C)O)=O)CC2N(C(=O)Cc3nnc(C)o3)CCC2(C)C1 1795,CCCCC(C(=O)N1CCN(C(C2CC3C(C2)C3(F)F)=O)CC1)NC(N)=O 1796,c1(NC(C23CC(NC(c4ccncc4Cl)=O)(C2)C3)=O)ccc2c(Cl)n[nH]c2c1 1797,C(=O)(C(=O)N=S(C)(C)=O)N(CC(C)NC(C1CC(O)CN1C)=O)C 1798,C(=O)(C1SCCc2sccc21)NC1C2CN(C(c3cc(C)c(=O)n(C)c3)=O)C1C2 1799,c1(C(N(CCCNC(C(C(C)C)OCC)=O)CC2CC2)=O)cc(OC)nc(C)c1 1800,N1(C(C(C2(O)CCOCC2)(C)C)=O)CCCCC1CCNc1nccc(CO)n1 1801,N1(C(COCC(C)C)=O)CC(CNC(c2csc(Cl)n2)=O)OC(C(F)(F)F)C1 1802,C(C1CN(C(c2cc(C(N)=O)co2)=O)CC1C(N1CCC(C(N)=O)C1)=O)=CC 1803,c1(CC(=O)NC2CN(C(=O)C(O)CC(F)F)CC2O)cnc2ccccc2c1 1804,CC(O)C(C)(C)C(=O)N1CC(C(N)=O)(CNC(=O)C2=C(Cl)CCC2)C1 1805,C=CCCC(c1nnnn1C1(C)CC1)(C1CC1)NC(C)CCC=C 1806,c1(CN2CC3C(C(=O)NCCc4cscn4)C3C2)cccc2cccnc12 1807,c1(C(=O)NCC(CN(C(=O)CC2(O)CC2)C)O)n[nH]cc1-c1ccccc1 1808,c1(C(N2CCC(O)C(C(=O)OC)C2)C(=O)NCCOC)n[nH]c2cc(Br)ccc12 1809,N1(C(COCCCCC)=O)CCC(CNC(=O)C=CI)C(C)C1 1810,C1(NC(c2cnn[nH]2)=O)CC2CC(NC(c3cc(Cl)cs3)=O)CC2C1 1811,C1(C(=O)NC2C=CC(CC(=O)NC(C)C(C)(C)C#N)C2)CC2CC(=O)C1O2 1812,c1(NCC2C(C)CN(C(=O)CC(C)(F)F)CC2)ncnc2c1nnn2C1CC1 1813,C1(NC(COCCCC#C)=O)CC2(C1)CC2NC(=O)CCCOC1CCCCC1 1814,c1(CC)ccc(C=CC(N2CCCC2CN(C(=O)Cc2ncc(C)o2)C)=O)cc1 1815,N1(C(c2cc(OC)n[nH]2)=O)CCC(C)(CNC(C2CCC(=O)CC2C)=O)CC1 1816,N#CCCCCC(=O)N1CCN(C(=O)C=CCN2CCCC2)C(CCO)C1 1817,C1(OC)CC(NC(c2occc2CNC(=O)CNc2ncccn2)=O)CC1OC 1818,Cc1cc(N2CCC(NC(C3C(F)(F)C34CCC4)=O)C2C)n2nc(C)nc2n1 1819,C(=O)(CS(=O)(=O)C(C)(C)C)NC(C)CN(C(=O)C(c1cc2ccccc2o1)C)C 1820,C(=O)(C1=CC2CCC(C1)C2)NC1CCC(C(N2CCC(C(C)C#N)CC2)=O)C1 1821,C1(CNC(c2cnc(OC)nc2)=O)COCCN(C(=O)C(C)SC(F)(F)F)C1 1822,c1(C(=O)NCC(C)(C)NC(Cc2c(C)noc2)=O)cnc2c(c1)nnn2C 1823,C1(CNC(C(CC)C)=O)COC(C)(C)CN1C(c1cnc(SC)nc1O)=O 1824,C12(NC(Cc3cc(C)no3)=O)CCCCCC1N(C(C1CC(=O)C1)=O)CC2 1825,c1(CC(=O)NC2(NC(C=CC(=O)OCCCC)=O)CC2)c(CC)cccc1CC 1826,CC1CCCCN1C(=O)CCNC(=O)Nc1cccnc1COC1CCOCC1 1827,c1(C(=O)NCC2CC2CNC(C2CC(O)(c3ccccc3)C2)=O)ccc(O)cn1 1828,C1(NC(CCc2nc(C)c(C)o2)=O)CC2CC(NC(C3OCCC3(C)C)=O)CC12 1829,C=CC(CCC)CC(=O)NC(CNC(=O)C(C)N(C)C(C)=O)CC(F)(F)F 1830,C(CC(O)CNC(=O)C(Cn1ccnn1)NC(=O)CC1(O)CCOC1)OC 1831,Cc1ccc(C(=O)NC2CCCC(N(C)C(c3nocc3Cl)=O)C2)c(F)c1 1832,CC(CC(=O)N(C1CCCN(C(=O)CCN2CCC2)C1)C)C(F)F 1833,c1(C(N2C(CC)CN(C(=O)C(C3CCOCC3)F)CC2)=O)cc2c[nH]cnc-2n1 1834,c1(C(C)=O)cn(CC(N2CC(C)(OCC(=O)NC3CCCCS3)C2)=O)nn1 1835,c1(OCC(=O)NCCC2(NC(C3(CO)CCCCO3)=O)CCC2)ccc(F)cn1 1836,c1(C(N2CCC(CCNC(=O)C=CC3CCCC3)C2)=O)cccc([N+](=O)[O-])c1O 1837,N1(C(CCc2n(C)cnn2)=O)CC2CC2(NC(=O)CCC2CCCOC2)C1 1838,c1(CC(N2C(CN(C(C(C)C3CCCC3)=O)C)CCC2)=O)cc(O)ccc1Br 1839,C1(OC)CN(C(C2(CSC)CC2)=O)CCC1NC(=O)C(O)CCSC 1840,c1(C2C(C(N(CC(C)(C)C)Cc3csnn3)=O)C2)ccccc1 1841,Cc1nc(C(N2CC3(NC(c4cnoc4C)=O)CC2C3)=O)ccc1C#N 1842,CC1CCCCCN1C(=O)Nc1ccccc1-c1ccc(Cl)c(F)c1 1843,C1(C(N2C3(CN(C(C(CCC)CC)=O)C3)CC2)=O)Cc2ccccc2C(C)(C)C1 1844,Cc1cc(C(N2CCC(C(=O)NCC3CCCC3O)(CF)C2)=O)ncc1N 1845,C1(NC(N(CCN(C(C(C2CCCC2)NC(C)=O)=O)C)C)=O)CCC2CC1CO2 1846,Cc1cc(C)c(CN2CC(F)CC2C(=O)Nc2cccc(F)c2CO)cc1C 1847,c1(C(=O)OCC)cc(Cn2cc(-c3ccn(C)n3)nn2)cs1 1848,Cc1cc(S(=O)(=O)N2CCCCC(C)C2)c(C)cc1-c1cc(F)c2cc[nH]c2c1 1849,CC1(CNC(c2ccoc2)=O)CCN(C(=O)Cc2nnc(-c3ccccc3)o2)C1 1850,C(=O)(CC1C(=O)Nc2ccccc21)NC(C)C(CO)NC(=O)Cc1csc(Cl)n1 1851,C(=O)(CC(F)(F)C(F)F)N(CC(=O)NC1CC(CC)OCC1)CCOC 1852,N1(C(C(C=C)O)=O)CCC(C2OCCCC2NC(=O)C(c2ccccc2)O)CC1 1853,C12(C(=O)NCCCNC(C3(c4ccc(Cl)cc4)CCC3)=O)C=CC(CC1)C2 1854,C(C)(CC(=O)NCC(C1CC1)NC(=O)CC#N)(C(F)(F)F)N(C)C 1855,n1(CCCC)nc(-c2ccoc2)nc1-c1cc(-c2ccc(F)cc2)no1 1856,c1(CC)cc(C(N2CCC(NC(=O)Cc3ccsc3)C(O)C2)=O)cc(O)n1 1857,c1(C(=O)NC2C(C)CN(C(c3cn4ccsc4n3)=O)CC2)ccnc2cc[nH]c12 1858,Cn1cc(CNC(C2CC=CCN2C(=O)C(O)CC2CCCC2)=O)ccc1=O 1859,Cc1cnsc1C(=O)N(CC(C)C(=O)NC1CC(CF)C1)C 1860,CCC(CCCC(=O)NC(c1noc(CO)n1)C)NC(C1CC(F)(F)C1)=O 1861,c1(CC)nnc(CN(C(=O)CC=CCNC(=O)Cc2cccnc2)C)o1 1862,CCCC(C)CC(=O)NC1CCCC(CNC(c2c(C)nc(C)n2O)=O)C1 1863,CC1CC(c2nnnn2C)(NCC(c2ccccc2F)(C)C)CN1C 1864,c1(C(N2CC(NC(C(C)(C(C)C)OC)=O)C2)=O)c(C)nc(C(C)(C)C)nc1O 1865,c1(C(N2CCC(C)(NC(COC)=O)CC2)=O)nccc2cnn(C)c12 1866,c1(C(N2CCC(N(CCC)C(c3ncncc3Cl)=O)C2)=O)sc2cncn2c1C 1867,C1(NC(c2ccc(CN(CCC)C)o2)=O)CCCN(C(=O)CCN(C)C(C)=O)C1 1868,c1(CC)ccc(C(=O)NC(COC)C(=O)NCC(=O)NCC(F)F)o1 1869,c1(-n2c(CCCCC=C)nc(CCO)n2)ccc2ncsc2c1 1870,Cc1ccc(=O)n(CC(=O)NCC2CC2NC(=O)COC2(C)CCCC2)n1 1871,C1(NC(c2c(OC)cccn2)=O)CCCC12CN(C(=O)CC(C)(C)F)C2 1872,O=C(C1=CCCN(C(C2CCC2(F)F)=O)C1)NC(C(F)(F)F)C1CC1 1873,C12(C(=O)NCCCC3(C)CC3)CC1CN(C(=O)C(C)(C)n1cncn1)C2 1874,C1(C(N2CCCC(C)(NC(c3cccc(F)c3F)=O)C2)=O)Cc2cccnc2C1 1875,c1(OC)ccc(O)cc1C(N1CC=C(CNC(C2(OC)CC2)=O)CC1)=O 1876,CC1CCN(C(c2cc(C(C)(C)C)no2)=O)CCN1C(C1CC1C(F)F)=O 1877,CN1CC(C(=O)NC(C)(C)CC=CC(=O)NCCOC2CCCC2)NC1=O 1878,c1(C(=O)NC(C(=O)OCC=C)Cc2ccccc2)noc2c1CCCCC2 1879,N1(CC(=O)Nc2ccccc2)CC2(CCC(CNC(C34CCCCC3C4)=O)O2)C1 1880,C1(NC(c2c(C)n(C(C)C)cc2)=O)CCN(C(=O)CCC2CCOC2)CC1O 1881,N1(C(c2c(CC)nc[nH]2)=O)CCCC(O)(CCNC(c2cnc(C3CC3)[nH]2)=O)C1 1882,c1(C(C(C)C)NC(=O)NCC2CS(=O)(=O)C2)ccc(Cl)cc1 1883,N1(C(C2CCN(CCC#C)CC2)=O)CCC(CO)C(NC(=O)CP(C)(C)=O)C1 1884,C(=O)(C(C)(C)C(C)C)NCC(C)N(C(C1N(C(CCC)=O)CCCC1)=O)C 1885,C1(C(=O)NC2CCC2)CCOC(=O)CC1.CC1C(=O)CN1.C12CC1NCC(=O)N2 1886,CC1CCN(C(c2ccc(C(N)=O)cc2)=O)CCN1C(=O)Cn1ncn(C)c1=O 1887,CCCC(CNC(c1ccsc1C)=O)C(=O)NCC(F)(F)C(C)(C)O 1888,c1(C(=O)NCC2COC(CNC(c3cc(Cl)no3)=O)C2)cccc(CO)n1 1889,CC(C)(C)C(=O)NCC(=O)NCC1CCCN1C(=O)Cc1ncc(Cl)s1 1890,Cc1sc(NC(=O)Cc2nnc(S)n2C(C)C)nc1C1CCCOC1 1891,C1(C(N2CCC(Cn3cc(CCN(C)C)nn3)CC2)=O)CC1C1CCCC1 1892,CC1CCC(NC(=O)OC(C)(C)C)CN1C(c1ccoc1I)=O 1893,c1(C(N2CCN(C(c3ccc(C)cc3)=O)C3C2C3)=O)ccnc2ccnn12 1894,c1(C(C)NC(C2CC=CC2)=O)ccc(CNC(C2(c3cccs3)CC2)=O)cc1 1895,c1(OC)ccc(C(N2CC(OC)C(NC(=O)CSCC#N)C2)=O)c(N)c1Br 1896,C1(NC(c2cccc(OC)c2)=O)CCN(C(c2cn(C)nc2SC)=O)C1(C)C 1897,CCCC(O)CC(=O)N1CCC(C(F)F)(CNC(=O)CCS(C)(=O)=O)C1 1898,CCC(C)(COC)CNC(C1CCN(C(=O)CCCCN(C)C)C1C)=O 1899,N1(C(C=Cc2ccc(C)o2)=O)CCCC(NC(C2(N(C)C)CCCOC2)=O)C1C 1900,N1(C(C(CC#C)O)=O)CCC(C(=O)NCC2(OC)CCC2)CC1(C)C 1901,N1(C(c2cc(Cl)cc(Cl)c2O)=O)CCC2CCN(C(C34CCC(C3)C4)=O)CC12 1902,C1(C)(C(N(CC(CNC(c2c(C)n(C3CC3)nc2)=O)(C)C)C)=O)COC(C)CO1 1903,CC1(C)CC(NC(=O)NCC(C)(F)C(C)(C)F)c2ccccc2O1 1904,C(C)(C(=O)NCC(C)(C)CNC(=O)CC(C)C1CC1)(C(C)C)NC(C)=O 1905,C(=O)(CC(C)(O)COC)NC1CCN(C(c2c(N(CC)CC)nccc2)=O)C1C 1906,n1(CC)cnc2c(NC(C)CCCO)[nH]c(=NCCCCCN3CCCC3)nc12 1907,Cc1ccc(CCC(=O)NC(C2CCN(C(C3(C)CC3C)=O)C2)C)s1 1908,N1(C(COC)C)CCC(C)C(NC(C2CCCN(CC(=O)O)C2=O)=O)C1 1909,Cc1ccc(C)c(C(=O)NCC(CC(C)C)NC(c2cccnc2)=O)c1O 1910,C1(NC(CCOC(C)C)=O)CCC2(CCN(C(c3ccsc3C#N)=O)CC2)C1 1911,c1(C(N2CCC(O)(CC(N3CCC(C#N)CC3)=O)CC2)=O)c(Cl)cc(Br)cc1Cl 1912,C(CN=c1nc(Cl)[nH]c(C)c1C#N)C1(OC)CCC1.N12CCCCCC(C1)C2=O 1913,C1(n2cnnn2)(C(=O)NC(CCCNC(C(C)CC2CCC2)=O)C)CCCCC1 1914,N1(C(CC2CCN(C)CC2)=O)CC(NC(C2CC2c2ccncc2)=O)CC(O)C1 1915,c1(C(=O)NCCCN(C)C(C2CCCS2)=O)cc(S(=O)(=O)N2CCOCC2)c[nH]1 1916,C1(NC(c2c(C(N)=O)csc2)=O)CS(=O)(=O)C2CN(C(c3cnns3)=O)CC12 1917,c1(C(=O)NC2CC(CCNC(CC3(OC)CCC3)=O)C2)cncnc1C 1918,c1(CC)cnoc1C(=O)NC1CC(C)(NC(=O)C(C)C2CCCO2)C1 1919,CC1CC(CNC(=O)CN(CC(C)(C)C)C)CN1C(C1C2COCC12)=O 1920,CC(C)(CNc1ccc(Br)nc1)CC(F)F 1921,N1(C(CCOCC#C)=O)CC(CO)C2(C1)CN(C(C1(C(F)F)CCCCC1)=O)C2 1922,C(CCC(C)(C)NC(=O)COCCc1cccs1)NC(CNC)=O.CC(=O)NC 1923,CC1OCCCC1C(=O)NC(C1CN(C(C2CCCN2C=O)=O)CCO1)C 1924,CCC(CC)(CO)C(=O)NCC1(CN(C)C(C2CCC3CCC23)=O)CC1 1925,Cc1cnc2c(C(N3CCN(C(=O)CN4CCCS4(=O)=O)CC3)=O)cccn12 1926,C1(C)(CNC(c2n(CCOCC)nnn2)c2cscc2Cl)CC2(C1)CC2(F)F 1927,N1(C(C2CCN(C(c3cn(C(C)C)nn3)=O)CC2)=O)CCC(O)C(C(=O)O)C1 1928,C1(C)(CC)CC(NC(=O)CCN(CCCO)C(C2CC(C)(C)C2)=O)CCO1 1929,c1(C(N(CC(C)NC(=O)CCC2CCCC2)C)=O)ccc(N)c(Cl)c1 1930,c1(NC(=O)Nc2ccc(CNC(C)CN3CCCCC3)cc2)cc(Cl)nnc1O 1931,c1(OC)ccccc1C(=O)NC(C1CCN(C(c2c(Cl)cnn2C)=O)C1)C 1932,c1(C(=O)NCCOC2CN(C(c3c(C)oc(Cl)n3)=O)C2)ccc2c(c1)CC(=O)N2 1933,c1(CN(C(CC)C)C(C2CCCC23CC3)=O)ccc(F)cc1 1934,c1(OC)ccc(O)c(C(=O)NC2CCC(NC(=O)C(CCSC)NC=O)C2)c1 1935,c1(OC)nc(C)cc2ccc(C(=O)NC(C)CN(C)C(C3C=CCCC3)=O)cc12 1936,c1(C(=O)NC2CC(NC(C=CC3(C)COC3)=O)CC2O)cc2cnccc2o1 1937,C1(CN(C)C(c2ccnc(C(C)(C)C)n2)=O)CCN(C(=O)C(F)(F)CO)CC1 1938,C1(CNC(c2cc(C)oc2)=O)CN(C(c2c[nH]ccc2=O)=O)CCC12CCC2 1939,Cc1scc(C(=O)NCC(c2ccc(F)cc2)NC(c2nnsc2C)=O)c1C 1940,CC1CCC=C1C(=O)N1C(CNC(c2cc(-c3cnn(C)c3)[nH]n2)=O)CC2CC12 1941,Cc1cc(F)c(C(=O)NC2CCCCC2CNC(c2ncccn2)=O)c(Br)c1 1942,c1(C(=O)NC2C(C(F)(F)F)CCN(C(CC(=C)C)=O)C2)c(F)ccc2occc12 1943,Cc1cc(C(=O)N(CC(C)NC(C23CCCC2C3)=O)C)cc(C)n1 1944,C1(C(=O)NC(c2cccc(Cl)c2)C(F)F)C2Cc3cc(Br)ccc3C12 1945,c1(OC)ccnc(O)c1C(=O)N(CC(C)N(C)C(c1cc(C(F)F)[nH]n1)=O)C 1946,CC(C)(CCCCNC(c1cc(Cl)n[nH]1)=O)NC(=O)Cc1ncc(Cl)s1 1947,C1(NC(=O)C(F)Cc2ccccc2)COC2(CCN(C(c3cc[nH]c3)=O)C2)C1 1948,c1(NCC(C(C)C)OC)ccc(S(=O)(=O)Nc2ccnc(CN(C)C)c2)c(Cl)c1 1949,C1(C(=O)NCc2c(C)n[nH]c2)N(C(C2CN3CCC2C3)=O)CCCC1(C)C 1950,c1(C(N2C(C)(CNC(=O)C(F)CC3CC3)CCC2)=O)cccc2c1NCCC2 1951,N#Cc1sc(=NC2(C3CN(C(=O)CNCS(=O)(=O)C(F)(F)F)CC3)CCC2)[nH]c1Cl 1952,c1(C(N(CCCNC(C=C(C)C)=O)C(C)C)=O)nncn1C1CC1 1953,C1(NC(C(C)Cn2cccn2)=O)CCN(C(C23CCN(CC2)C3)=O)C12CCC2 1954,C1(C(=O)NC(C2(O)CCN(C(c3c[nH]c(C#N)c3)=O)C2)C)CCCCN1C 1955,c1(C(N(C)Cc2cc(OC)no2)=O)cc2ccncc2c(O)n1 1956,N1(c2ccnc(SC)n2)CCCC(N(C)C(C2CC2(F)F)=O)CC1 1957,C12CCN(CC1(C)C)C(=O)C(CC1CC1)NC2=O.n1(CC=C(C)C)cncn1 1958,c1(C(=O)NCC2CN(C(C3COCC3C(F)F)=O)C2)ccc(-n2cccn2)cc1 1959,N1(C(c2cn(CC)nc2)=O)CCN(C(c2cn(C)nn2)=O)C(CF)C1 1960,C1(C(N2CCC(Cc3cn(CC(CC)O)nn3)CC2)=O)CCc2ccccc2C1 1961,C1(NC(=NCC)NN2CC3CN(CCOC)CC3C2)CCc2nn(C)cc2C1 1962,C(=O)(C(C)(CC)CO)NCC(N1CCN(C(C2C(CN(CC)CC)C2)=O)CC1)C(F)F 1963,C(CCN=c1nc2c(c[nH]1)CCCC2)OCCNC(C1N(CC(C)C)CCC1)=O 1964,N1(C(CC2(N(C)C)CCCC2)=O)CC2CCCC1C2CNC(C1CC=CC1)=O 1965,CC1(C)CN(C(c2cccnc2)=O)CC(CNC(=O)Cc2ccc(F)cc2Cl)O1 1966,Cc1cnc(NCCC2CCS(=O)(=O)C2)c(S(=O)(=O)NCCCCCF)c1 1967,C1(NC(C(COC)(C)C)=O)CCN(C(=O)C(C)OCC(C)C)C12CC2 1968,N1(C(C2(C(F)(F)F)CC=CCO2)=O)CCN(c2ccccc2OC(F)F)CC1 1969,c1(C(=O)NC(C2CCN(C(C3CN(CC)C(=O)C3)=O)CC2)C)cc(C#N)[nH]c1C 1970,C(CC(=O)N1CC2(CCCC2)C1)(C(F)(F)F)NC(C1CC2(CCC2)C1)=O 1971,c1(-c2nc(-c3c(C)ccc(N4CC(C)OC(C)C4)c3)on2)cn2cccnc2n1 1972,C=C(C)CCCC(=O)NC(C)Cn1cc(CN(CC)CC)nn1 1973,N1(C(C=C2CCN(C)CC2)=O)CC2CN(C(=O)CC3CCCO3)CC2C1 1974,C1(NC(CC(C=C)C)=O)CC2CC1N(C(c1cnc(C(C)(C)C)o1)=O)C2 1975,C12(C(=O)NC3CCCN(C(c4[nH]cc(C)c4)=O)CC3)CCCC(CCC1)C2 1976,CCCCC(O)CC(=O)NC1CCCN(C(=O)C(C)(C)C(C)C)CC1 1977,C12(C(=O)NC(C(C)C(=O)NC(C)(C)C(O)CO)C)CCC(CC1F)C2 1978,N1(C(C2(C(=O)OC)C(C=C)C2)=O)CC2CCC1CN2C(=O)COc1ccccc1 1979,N1(C(Cc2n(C)nnc2)=O)CCC(CNC(C2CNC(=O)C2)=O)C12CC2 1980,C1(C(=O)NC2C(CNC(c3sc(CCC)c(COC)c3)=O)C2)C(C2CC2)C1(F)F 1981,N1(C(CCC)=O)CC(C(=O)NCc2nnc(C)s2)C(F)(F)C1 1982,C=CCCCCCCC(=O)NC1CCCC1NC(C1C=C(C)CS1)=O 1983,N1(C(C2(C)CC2)C)CCCCC(Nc2cc(C(F)(F)F)ncn2)C1 1984,C1(C(N2CC(CN(C)C(C3SC4C=CC3CC4)=O)C2)=O)C2(CCC2)C12CCC2 1985,n1(C(C)C)cc(CC(=O)NC2CCCC2NC(=O)CCOC2CCCCC2)nn1 1986,c1(C(=O)NC(C2CCOC2)CNC(=O)Cn2ccnn2)ccc(O)c(Br)c1 1987,C1(NC(C(CCCC#C)C)=O)CC2CCC1CN(C(=O)CC1CCCC1C)C2 1988,c1(C(=O)NCCC2(O)CCN(C(C34OC(C)C(C3)C4)=O)C2)cccc2occc12 1989,C1(c2nnnn2CCCF)(NCc2ccc(C(C)C)s2)CSC(C(C)(C)C)C1 1990,n1(CCC)ncc(C(N2CC(NC(=O)CCc3cnco3)C3CC23)=O)c1C 1991,c1(C(=O)NCC(C2CCC2)NC(c2csc(Cl)n2)=O)ccc([N+](=O)[O-])cn1 1992,C12(NC(C3CC3[N+](=O)[O-])=O)CCC(C1)N(C(=O)CNc1ccc(C(F)(F)F)cn1)C2 1993,C12(CNC(CC(=O)NC)=O)CN(C(=O)CCOCC3CC3)CC1CCO2 1994,N1(C(CC2(N(C(CC(C)C(F)F)=O)C)CC2)=O)CCC2(CCC(O)C2)C1 1995,C1(CNC(C2CCC(CC)O2)=O)(OC)CCN(C(=O)C(F)(F)C2CCCC2)C1 1996,Cc1ncnc(C)c1CC(=O)NCCCNC(C1CC2(F)CC1C2)=O 1997,c1(C(N2C(C(=O)NC(CC=C)CO)CCC2)=O)ccc(Cl)nc1F 1998,Nc1cc(C(N2CCCC2C2(NC(=O)C3=COCCC3)CC2)=O)cc(Br)n1 1999,C1(CCCCN2CCC(C)C2)CCN(C=O)C1.C(C(=O)OC)SCC 2000,C1(CC(=O)N(CCn2cc(-c3ccncc3)nn2)CC2(O)CC2)CC2COCC12 2001,N1(C(C2C3(CCN(C(C4(CCCC)CCC4)=O)C3)C2)=O)CCC(C2(C)CC2)CC1 2002,c1(C(N2CCOCC(NC(c3c(C)onc3)=O)C2)=O)cc2c(Cl)cccc2s1 2003,N1(C(C2C(CC)CCN2C(c2cc(C3CC3)[nH]n2)=O)=O)CCc2oc(C)nc2C1 2004,C1(NC(C(CC=C)N(C)C)=O)CCCCC12CCN(C(=O)C(O)C(C)CC)C2 2005,c1(OCC(C)C)ccccc1C(=O)NCCC(C)(C)NC(=O)Cc1ccsc1Cl 2006,CCC(CC)(C(=O)NC1(CO)CC2CCC1C2)c1ccccc1 2007,C1(NC(C(c2ccnn2C)C)=O)CCOCC1C(=O)N(C)Cc1cccnc1O 2008,C(=O)(CCC(C)(C)c1ccccc1)N(C)CCC(c1ccc(F)cc1)(C)C(=O)O 2009,C(=O)(C(O)C1=CCCCC1)N(CC(=O)NC(CCC(C)C)C)C 2010,N1(C(CC2COCC(C)O2)=O)CC(C(=O)N(C2CN(C)C2)C)C(C)(C)C1 2011,c1(CC)cccc2c1CN(C(=O)C(=O)Nc1ccc(Cl)cc1)CC2 2012,N1(C(C2(C)CC2C(F)F)=O)CCC2(CC(NC(=O)CC(F)(F)c3cccs3)C2)C1 2013,CCCC(O)CC(=O)NC(CNC(c1cc(N2CCCC2)ncn1)=O)CCOC 2014,Cc1cccnc1CNC1CCCC1C(=O)Nc1cnccc1C(F)(F)F 2015,C(=O)(C(C)C(CC)CC)N1CC(CC(NCP(OCC)(C)=O)=O)C2(C1)CC2 2016,c1(C(N(CC(C)NC(=O)CC2COCCO2)C)=O)ccc(-c2ccccc2)o1 2017,c1(C(=O)NC2(CO)CCN(C(c3ccc(Cl)cc3)=O)C2)cccc(F)c1O 2018,N1(C(CCCC(C)NC(C2C(=C)C2)=O)=O)CCCC2(CC1)CC2 2019,CC(N=c1ccnc(Cl)[nH]1)C1CCN(C(=O)C(C)Cc2ccccc2)C1 2020,C1(C(N2CCC(N(C)C(C3CC4CC4C3)=O)CC2)=O)CCc2ccc(F)cc2C1 2021,c1(C(N2CCC(N(C(c3cc(C)cc(O)n3)=O)C)C2)=O)ccc2c(c1)N(C)CC2 2022,Cn1cc(-c2ccccc2)c(=NC(=O)C2CC2CNS(=O)(=O)c2ccccc2Br)[nH]1 2023,C1(OC)(CNC(=O)Cn2cc(Br)cn2)CCN(C(C23COCC2C3)=O)CC1 2024,C1(C(=O)NC(c2nccc(O)n2)C)C=CCN(C(=O)Cn2ccnc2)C1 2025,C=CCCC(F)(F)C(=O)NC1CN(C(c2cc3ccccc3s2)=O)C1 2026,Cc1nc2cc(C(=O)NC(C)CCNC(C3CC(C)CC(=O)N3)=O)[nH]c2s1 2027,C(C(C)C(=O)NCCCC1(NC(C2CCC(=O)C2)=O)CC1)OC 2028,C1(C(=O)NC(C)CNC(=O)Cn2cnnc2)CCCCC12CCC2 2029,N1(C(c2c(C)noc2N)=O)CCCC(C)(C(=O)NC2CC(CC(C)(C)C)C2)C1 2030,C1(CNC(c2n(C)c(S)nn2)=O)CCN(C(=O)Cn2cc([N+](=O)[O-])cn2)C12CC2 2031,c1(C(C(=O)NCCOC)N(CC(C)S(C)(=O)=O)C)cnn(C)c1Cl 2032,C1(NC(C(C(COC)C)C)=O)CCCC12CCN(C(=O)Cn1nnc(=N)[nH]1)CC2 2033,C1(C(N(C)CC2COCCN2C(c2n[nH]cc2Br)=O)=O)CCC2(CCC2)O1 2034,c1(CC)ccc(C(=O)NCC2CC2CNC(=O)CC2CCCCCC2)cc1Br 2035,C1(NC(COCC)=O)CCN(C(C2C=CCCC2)=O)CC1OC 2036,C1(NC(C=CC(C)(C)NC(C2(COC)CCCCO2)=O)=O)CN2CCCC1C2 2037,c1(NC2C(C)S(=O)(=O)CC2)ccc(S(=O)(=O)NC2CCC(O)CC2)cn1 2038,C1(C(N(CCC(=O)NCC2CCCS2)CCO)=O)C=CCCC1 2039,c1(CNC(C(=Cc2cnc[nH]2)C)=O)cnn2c1CN(C(=O)C(=O)C(F)(F)F)CC2 2040,c1(OCC)c(Cl)cc(NC(c2ccc([N+](=O)[O-])o2)=O)cc1Cl 2041,O=[N+]([O-])c1cccc(F)c1Cc1noc(Cc2ccccc2)n1 2042,N1(C(C2N(C)CC(C)(C)C2)=O)CCC(c2ccccc2)C(F)(F)CC1 2043,N1(C(C(C)(C)c2cscn2)=O)CCC2(CCC2NC(=O)C=Cc2cccs2)CC1 2044,c1(C(=O)NC2CC3CN(C(CCCC(C)O)=O)CC32)ccc(Cl)c2occc12 2045,N1(C(CC(C)(C)O)=O)CCN(C(=O)C=Cc2ccccn2)CC1CS(C)(=O)=O 2046,C1(CNC(=O)COc2ccccc2)CCC(NC(C2CC2C2CC2)=O)CC1 2047,CCCC(C)CC(=O)N(C1CCCN(C(c2sc(N(C)C)nc2C)=O)C1)CCF 2048,C1(CNC(C2CCCC(=O)N2)=O)CCCCN(C(c2cc3c(s2)CCC3)=O)C1 2049,c1(CC(=O)NCCNC(c2c(Cl)csc2Cl)=O)ccc2cccnc2c1 2050,c1(C(=O)NCCSCCC(F)(F)F)cnc2c(Br)cc(Br)cc2c1 2051,C1(C(NOCCCC#C)=O)CCCN(C(=O)Cc2cccc(C)c2)C1.N1CCC1 2052,C(CC1CCN(C(=O)Nc2ccc(SC)c(C#N)c2)c2ccccc21)OC 2053,N1(C(CCCOCCC)=O)CCCC2CN(C(C3(F)CC34CCCCC4)=O)CC12 2054,c1(C(=O)NCCCCCNC(c2c[nH]c(=O)cn2)=O)cccc2cnccc12 2055,C=CCC(CNC(c1ccn(Cc2ccccc2)c1)c1nnnn1C)CC(C)C 2056,C(=O)(CS(=O)(=O)C1CC1)NCCC1CC(NC(c2c(NCC)c(F)ccc2)=O)C1 2057,C1(CC)CCCN(C(c2ccc(OC)s2)=O)C1C(=O)NC(C12CCC(CO1)C2)C 2058,c1(CC)c(C(=O)NCC2CN(C(c3csc(COC)n3)=O)CCO2)cccc1F 2059,c1(CC)nnsc1C(=O)NC1CN(C(=O)CCc2ncccn2)C1 2060,c1(C(=O)NC2C3CC(NC(C4C(=O)NCC4)=O)CC32)ccc2[nH]ccc2c1 2061,C12(NC(c3cnns3)=O)CCN(C(=O)CCc3cncc(Br)c3)CC1C2 2062,N1(C(CCOCC)=O)CCN(C(=O)Cn2c(C)c(C)sc2=O)CC1CC1CC1 2063,c12c(Cl)ccc-1c2F.N1(C(c2cc(Br)c[nH]2)=O)CCN(c2ccnc(O)c2)CC1 2064,c1(C(N2CCOC3CC23)=O)cnc(OC)cc1.c1(OCCC)ccc(NCC)cc1 2065,N1(C(C(CC)SC)=O)CCN(C(=O)CCCn2cncn2)CC1COC 2066,C=CCC(CC)C(=O)NCC1CN(C(c2nnn(C(C)C)c2C)=O)CCN1C 2067,c1(C(N2CCC(CNC(C3CN4CCC3C4)=O)C2)=O)cn2ccccc2n1 2068,C1(C(=O)NCC2(C)CCN(C(=O)CNS(=O)(=O)C3CC3)C2)CC2CC1CC2O 2069,CS(=O)(=O)c1ccccc1C(=O)NC1CCN(C(=O)CC2(C(F)(F)F)CCC2)C1 2070,C(C(=O)NCCC1(C)CC1)(c1ccns1)N(C(C)C)CCN(C)C 2071,C1(NC(c2cc(CC)sc2)=O)C=CCN(C(=O)CN(c2ccccc2)C)C1 2072,c1(CC)ccc(N)c(C(=O)NC2CN(C(=O)C(O)CC)CCC2C(F)(F)F)c1 2073,Cn1ncnc1C(=O)NCCNC(=O)CC1OCCO1 2074,O(C=CC(=O)N(C1CN(C(=O)CCc2ccc(Br)s2)C1)C)CC 2075,c1(C(=O)NCC(CO)NC(c2c(C)nn(C(C)(C)C)c2)=O)ccc(N=[N+]=[N-])cc1 2076,C=Cc1cnn(C)c1C(N1CCC(N(C(c2cc(OC)ccc2F)=O)CC)C1)=O 2077,C1(CNC(=O)NCCS(N)(=O)=O)(Cc2nccc(C(F)(F)F)n2)CC2(CCC2)C1 2078,N1(C(C2(OC)CCOC2)=O)CC2=C(C1)CN(C(=O)C(c1cncnc1)C)C2 2079,N1(C(c2cc(C)[nH]n2)C(N2COCC2C=Cc2ccco2)=O)CCC(O)C(C)C1 2080,C1(NC(C2C(C)C2)=O)CCCCC1NC(=O)CCOc1cccnc1 2081,N(C1CCCOc2ccc(Br)cc21)CC1(c2nccn2C)CC(OCC)(OC)C1 2082,C12(CC(=O)NCC3(F)CN(C(C4C(C)C4)=O)C3)CCCN1CCC2 2083,C(C(C)(C)C)N(CC(=O)N(CC=CC(=O)N(CCCC1CCC1)C)C)C 2084,c1(C(CC(N2CCC(N(C(C3CN(C4CC4)C3)=O)CC)C2)=O)C)c(C)noc1C 2085,n1(CC(=O)NC2CCn3nnnc3C2)nc2ccccn2c1=O 2086,c1(C(=O)NCC(CN(C(=O)COc2ccsc2)CC)O)cc(C)n(C2CC2)c1C 2087,c1(CSC2N(C(=O)OC(C)(C)C)CCC2)nccc(NCCP(C)(C)=O)n1 2088,c1(COC)cccc(S(=O)(=O)NC(CCc2ccccc2)C(F)F)c1 2089,c1(C(N2C(CNC(CCC=C)=O)C(C)CC2)=O)cnc2sc(C)nc2c1 2090,CCCC(CC(=O)N1CCC(C(N)=O)(OC)C1)NC(C1(n2cnnn2)CC1)=O 2091,Cc1cc(C(N2CC3CC(C(N4CC=CC4CF)=O)(C3)C2)=O)cc(O)c1 2092,Cc1nccnc1C(=O)NCC1(C(C)NC(C2CN(C(C)C)CCO2)=O)CC1 2093,c1(C(N2CCC(C#N)(NC(C3CCNC(=O)C3)=O)C2)=O)cc(O)c(O)c(O)c1 2094,CC1CC(C(=O)N(CCCO)CCCO)N(Cc2ccc(-c3cccs3)cc2)C1 2095,C1(NC(C(C=C)O)=O)CN(C(=O)CCc2cn(C)nc2C)C2(CCOCC2)C1 2096,C1(NC(C2N(C(=O)OCC)C(CO)CC2)=O)CCN(C)C(=O)C1 2097,CCCCC(O)C(C)C(=O)N(C(C)C(=O)NCCOC1(C)CCC1)C1CC1 2098,c1(-c2ccnc(N3CCC(O)C(C)C3)n2)c(C(C)C)nc2ccccn12 2099,c1(CC(=O)N(CCC(C)NC(C23CCN(CC2)CC3)=O)C)ccc2sccc2c1 2100,CCCCC(C)C(=O)NCc1csc(C(=O)NC(c2ccc(O)cc2)C)c1 2101,c1(C(N2C(C3(NC(CC(C)F)=O)CC3)CCC2)=O)ccc(OCCF)cn1 2102,Cc1c(C(=O)NC2CC(NC(c3cc(Cl)cc(Cl)c3)=O)C2)c[nH]c2nccc1-2 2103,Cc1c(F)ccc(C(=O)NC2(CNC(=O)CCOCCN(C)C)CCC2)c1N 2104,c1(C(N(CC(CNC(c2[nH]cc(C)c2)=O)C)C)=O)cn(C2CC2)nc1C 2105,c1(CC)ccc(C(=O)NC2(C)CCCN(C(c3cc(N)cc(O)c3)=O)C2)c(F)c1 2106,C(=O)(CC(C)CC(F)(F)F)NCC1CN(C(CC2(CSC)CC2)=O)C1 2107,c1(CC)ccc(Br)cc1C(=O)NC1CCCC1CO.N12CCC(CC1)CC2=O 2108,C(=O)(C(F)C1=CCCCC1)NC1C2CN(c3nnc(C(N)=O)s3)CC21 2109,C12(COC)CCC(C(N3CCC(CNC(=O)CC(C)(F)F)C3)=O)(CO1)C2 2110,N1(C(CSc2n(C)c(S)nn2)=O)CCCC(S(=O)(=O)N(C)C)C1 2111,C1(NC(c2ccc[nH]2)=O)CCC2CCN(C(c3cc(Cl)ns3)=O)C12 2112,c1(C(=O)NC(C)(C)CNC(C2(C)CCC(=O)NC2)=O)ccc([N+](=O)[O-])cc1F 2113,C#Cc1ccc(NC(=O)C(C)(C)C2CCN(C(=O)CCOCC)C2)cn1 2114,N1(C(c2cncc(OC)c2)=O)CCN(C(c2cc(N)c(Cl)cn2)=O)CC(C)(F)C1 2115,N1(C(c2c(COC)ncs2)=O)CC(NC(c2cnn(C)c2C)=O)CC1C 2116,C12(CNC(c3cnc4sccn34)=O)CCCC1CN(C(C1C(F)(F)C13CC3)=O)C2 2117,c1(C(=O)NC(CC2CN(C(C3(CCOC)CC3)=O)C2)C)ccc(O)nc1 2118,Cc1cc(NC(C2CC2NC(c2cc(Cl)ccc2O)=O)=O)ncc1F 2119,C(=O)(C1=CCS(=O)(=O)C1)N1CC(CNC(C2(C(=O)OC)CC2)=O)C(O)C1 2120,Cc1ccccc1OCCC(=O)NCC1CC(F)CN1C(=O)CC(F)(F)Cl 2121,N1(C(C2CN(C(CCC)C)C(=O)C2)=O)CCN(C(=O)C=C(C)C)C2COCC12 2122,C(CC(F)F)(C(=O)NCC1(O)CCN(C)C1)N(C(c1n(CCC)ccc1)=O)C 2123,C1(CNC(C2(OC)CCOC2)=O)CN(C(C2(F)CC2)=O)CCC1(C)C 2124,C(CCCCC(=O)NC1CCCC(C(CC)CC)CC1)=CC 2125,C1(C(N2C3(c4cn(C(CC=C)CC)nn4)COC(C2)C3)=O)CCC=CCCC1 2126,c1(CC(=O)NCCCC(C)NC(=O)COC2CCC2)c[nH]c2ncccc12 2127,c1(C(=O)NCC2(C)CCCN(C(C3(C)CS(=O)(=O)C3)=O)C2)cccn2nnnc12 2128,c1(C(=O)NC(C)CC2CN(C(c3cccc(CO)c3)=O)C2)ccn(C)c(=O)c1 2129,N1(C(CNS(NC)(=O)=O)=O)CCC2CCN(C(c3n[nH]c4c3CCC4)=O)CC12 2130,C12(CCC)CC(C(=O)NCCOC3CN(C(=O)CCC4CCCO4)C3)(C1)C2 2131,c1(C(=O)NC2CC3(C(C(N(C4CC(=C)C4)C)=O)C3)C2)ccc(C#N)cn1 2132,c1(C(N(CCN(C(C2C(C(C)C)(CC)C2)=O)C)C)=O)cncc2sccc12 2133,CCC(C)(COC)C(=O)NC(C(=O)N(C)CC1(COC)CCC1)C(C)C 2134,C(=O)(C1=CSCS1)NCC(CNC(=O)C=Cc1ncc[nH]1)F 2135,C1(NC(C2CCO2)=O)(CO)CCN(C(c2ccc(SC(F)(F)F)cc2)=O)C1 2136,c1(C(N2CCN(C(C#CC3(CC)CC3)=O)CC2)=O)cccc2cc(F)ccc12 2137,N1(C(c2cn(CC(N)=O)nn2)=O)CCCC(N(CCO)C(c2cnccn2)=O)C1 2138,Cc1nn(CC(N2CCN(C(=O)C3=CCCC3)CC2CF)=O)c2ncccc12 2139,CC(F)CC(=O)N1CCC(OCCCc2ccccc2)C1 2140,c1(OC(C)C(N2CCCCC2CNC(c2ccc(Cl)cn2)=O)=O)ccccc1F 2141,n1(CCC)nnnc1C(c1cn(C2COC2)nn1)NCc1nccn1C1CC1 2142,c1(C(=O)NC2CCN(C(C3CCC(CC)CC3)=O)C2)nn(C)c2ccc(Br)cc12 2143,N1(C(C2CCC(CC)CC2)=O)CCC2(COCC(CNC(=O)C(F)(F)CC)O2)C1 2144,c1(OC)ncc(C(=O)NCCC2CCN(C(C3CC(F)C3)=O)C2)cn1 2145,c1(C(=O)NCC(c2ccccc2)NC(C2(CC=C)COC2)=O)ccc(N)c(N)n1 2146,c1(C(=O)OCC)c(-c2nc(C(F)F)nn2C)ncn1C 2147,Cc1cc(C(=O)NC2CS(=O)(=O)CC2NC(c2cnc(C3CC3)o2)=O)cc(F)c1 2148,CC(O)CCC(=O)NCC(C)N(C(=O)CCc1ccco1)C 2149,Cc1ncc(Cl)cc1C(N1CCC(O)(C(F)(F)C(N)=O)C1)=O 2150,CS(=O)(=O)c1cnn(CCNCC2OCCC2C(=O)OC)c1.C(=O)O 2151,C1(=O)CN2C(=O)C(CCc3ccccc32)N1.C1(CNC(C#C)C)CCCN1C 2152,N1(C(c2c(C)cccc2Cl)=O)CCOCC12COCCN(C(C1CCOC1)=O)C2 2153,c1(C(N(CC(C)N(C(=O)CCc2ccon2)C)C)=O)ccc(S(N)(=O)=O)o1 2154,C1(N(CC#C)C(C2(OCC)CCCC2)=O)CCN(C(=O)C(C)OC)CC1 2155,c1(C(N2CC3C(NC(C4CCC(OC)C4)=O)C(C3)C2)=O)cccc(C)c1[N+](=O)[O-] 2156,C1(=O)CC(C(F)(F)F)CN1.Cc1ccc(CC(C)C(=O)NC(C)(C)C2CC2)cc1 2157,N1(C(C2CC(C)C2)=O)CCC(C(F)CNC(=O)CN2CCN(C)CC2)CC1 2158,C1(OC)(OC)CCC1C(=O)N(CC(=O)NCc1ccoc1)C(C)C1CC1 2159,N1(C(c2cc(CCC)on2)=O)CCC(NC(C2CC(CCC)C2)=O)CC(C)(C)C1 2160,c1(N2CCCC(N(C(COCc3cc(C)on3)=O)C)C2)ncc(Br)cc1C#N 2161,C1(COC)(NC(=O)C(C)n2cncn2)CCN(C(c2nccs2)=O)CC1 2162,c1(C(N(C(CC)C(=O)N(C2(C)CC2)C)C)=O)ccc2n[nH]cc2c1 2163,N1(Cc2cc(C)no2)CC2C(C(=O)NCCCn3cccc3)C2C1 2164,c1(NC2CN(C(C)=O)C2)ncccc1S(=O)(=O)N1CCC(=C(F)F)CC1 2165,C1(C(=O)NCC(CCOC)NC(c2nocc2Br)=O)CC1C1CCC1 2166,C1(C(=O)NC(CNC(CCCC)=O)C)Cc2c(F)cccc2C(=O)O1 2167,N1(C(C2(CCl)CCOCC2)=O)CCS(=O)(=O)CC1C1CCC1 2168,N1(C(Cn2c(CCC)ncc2)=O)CCOCC1CN(C)C(C1C=CCS1)=O 2169,c1(C(=O)NCC(CCC)NC(=O)CCc2nc(CC)no2)ccc(CCF)cc1 2170,c1(C(=O)OC)c(C)[nH]c(C(=O)N(C)CCNC(c2c[nH]nc2S(N)(=O)=O)=O)c1C 2171,N1(C(=O)Nc2ccc(C(=O)OC)c(Cl)c2)Cc2cccc(Cl)c2C1 2172,c1(C(N2CC(CO)CC(C)C2)C(=O)NCCCSC)cc(Br)ccc1C(F)(F)F 2173,C1(NC(C2(NC(c3cccc(=O)n3C)=O)CCN(C)C2)=O)CN2CCC1(F)CC2 2174,C1(O)(CC(N2C(Cn3cc(C(C)(C)OC)nn3)CCC2)=O)CCN(C)CC1 2175,c1(SCC#C)cccc(C(=O)N(C)CCOCCN(C(=O)C(C)=C2CCC2)C)c1 2176,C1(CC(=O)N(C2CCCC(CNC(=O)CO)C2)C)CC(=O)NC(=O)C1 2177,C1(NC(C(C(C)C)NC(=O)C(O)CN(C)C)=O)C=CC(C)(C)CC1 2178,c1(-n2c(CCCCCSC)nc(CCOC)n2)cc(C)ccc1C 2179,C1(CNC(CCC(C)C)=O)(NC(C2CC(OC(F)F)C2)=O)CCCCCC1 2180,C(=O)(C(C)(C)C(C)NC(=O)C=CC1(C)COC1)NCC1CCN(CCC)C1 2181,C1(C(N(CC(O)CNC(C2(Br)CC2)=O)C)=O)CC12CCOCC2 2182,N1(C(C2N(C(CCCCCC#N)=O)CCC(O)C2)=O)CC2(CCC(=O)NC2)C1 2183,CCC(Cc1ccccc1)C(=O)N1CCC1CNC(=O)CC1(CO)CCCC1 2184,C12(NC(C(CSC)OC)=O)CCCC1(F)CN(C(=O)CCCC(F)(F)F)C2 2185,N1(C(c2c(F)ccc(OC)c2)=O)CC(C)CN(C(=O)C=Cc2cocn2)C(C)C1 2186,N1(C(c2ccc(OC)cc2)=O)CCC(F)CC1C(=O)Nc1cc(C)cc(O)c1 2187,c1(OCC)nccc(C)c1NC(c1ccc(-c2c[nH]c(=N)c(C)c2)c(C)n1)=O 2188,C(=O)(CC(C)C(C)(C)C)N1CC(C=CC)C(C(N2CCN(C(C)CC)CC2)=O)C1 2189,c1(C(N2C(C3CCN(C(CCC4(C)CC4)=O)C3)CCC2)=O)cncc(Cl)c1 2190,c1(OC)ccc(C)c(C(N2CCC(C(C)NC(=O)CCN(C)C(C)=O)C2)=O)c1N 2191,C1(C(=O)NC2CC(CF)C2)C2CC(O)C(C2)N1C(c1ccn2ccnc2c1)=O 2192,Cc1cc(C(N2CCOCC(NC(c3ccc(C(N)=O)o3)=O)C2)=O)nc(C)c1 2193,CCCCCC(C)CC(=O)NC1CN(C(C2CC(F)(F)C2)=O)CC1SC 2194,C1(C(=O)NOCC=CCl)(CC)CCN(C(c2c[nH]c(=O)cn2)=O)C1 2195,CCC(C(=O)NC1(CC(=O)NCCc2cn(CC)nn2)CCC1)SC 2196,c1(C2(NC(c3n(C4(C)CC4)nnn3)CCOCC3CC3)CC2)ccccc1Cl 2197,c1(C(=O)NCC2(NC(C3CCCCC3F)=O)CC2)c(F)ccc(F)c1Cl 2198,C1(NC(C2CCCC2C(F)F)=O)CC2CC1N(C(c1ccncc1)=O)C2 2199,c1(CC)onc(C)c1CNC(=O)CCC1CCN(C(=O)CC2CCCC2)CC1 2200,Cc1c(C(=O)OCCCn2cc(Br)ccc2=O)cccc1Cl 2201,Cc1nc(C(N2CC(NC(c3cc(F)ncc3Br)=O)C(C)C2)=O)ccc1F 2202,C1(NC(C2C(C(C)=O)C2(C)C)=O)CC(NC(c2nn(C)cc2Cl)=O)C12CCC2 2203,N1(C(COC)=O)CC(S(=O)(=O)N2CCN(C(=O)C=C(C)C(C)(C)C)CC2)C1 2204,c1(C(=O)NC2C(CNC(C(CC#C)O)=O)C2)ccc(COC)c(F)c1 2205,C1(C(=O)O)(N)CCOc2ccccc21.C#CCC(C=O)C1CC1 2206,c1(CC)cnc(O)c(C(=O)NC2CN(C(=O)Cn3cc(CO)nn3)CC2C)c1 2207,c1(OC(C)=O)cccc(C(=O)NCC2(O)CN(C(=O)CC3(O)CCOC3)C2)c1C 2208,C(=O)(CC(C)CC)NC1(C(=O)NC(C(=O)N(CC)CC)C)CC1 2209,c1(CCNC(C2(NC(C3CCCC3)=O)CC2)=O)cccc(F)c1F 2210,c1(N(CCCS(C)(=O)=O)C)ccc(S(=O)(=O)N2CCSC3CCC23)cn1 2211,CC1CN(C(c2ccn(CC(F)F)n2)=O)CC1NC(C1CCC1(C)C)=O 2212,N1(c2cc(C)nc(C(F)(F)F)n2)CC2CCN(Cc3ccccc3)CC(C2)C1 2213,N1(C(C=CCN(C)CC)=O)CC2(CC2)CC1CC(=O)NCCC(C(C)C)C1CCC1 2214,C1(CNC(c2c(OCC)scc2)=O)CCC(C)(C)CN1C(=O)C(C)CF 2215,c1(C(=O)NCC(C2CC2)NC(c2c[nH]cc2Br)=O)ccc(C(F)F)c(F)c1 2216,N1(C(c2ncn(C(C)C)c2)=O)CC(C(N2CC(OCC(F)F)C2)=O)C(C2CC2)C1 2217,C(C)(CCC(=O)NCC1CC(C(=O)NCc2cccc(F)n2)C1)SC 2218,N1(C(c2cncc(OC)c2)=O)CCOCC12COCCN(C(=O)C(C)C(C)C)C2 2219,N1(C(C(CCCC)F)=O)CC2CCN(C(=O)CS(=O)(=O)C(C)(C)C)CC2C1 2220,c1(NC(c2ccc(C)nc2)=O)ccc2nc(C3CC3)oc2c1.C12CC1CNC2=O 2221,N1(C(COC)=O)CCN(C(=O)CC2C(=O)N(C)N=C2C)CC1CCOC 2222,c1(C(=O)NCC(CC(=O)NCCN(CCOC)C)OC)ccc2[nH]ccc2n1 2223,C=CCCC(F)(F)C(=O)N1CC(NC(=O)C(C)=C2CCC2)C(c2ccccc2)C1 2224,N1(C(C(C(C)C)O)=O)CCC(C)(C)C1CC(=O)NCC1CCCSC1 2225,C1(C(=O)OC)OCCC1C(=O)NCc1cc(C(N)=O)on1.C12(CCCO1)CS2 2226,c1(C(=O)NCCCCCN(C(=O)CCCN=[N+]=[N-])C)cc2n(n1)CCCC2O 2227,c1(C(=O)NC2CCN(C(c3cn(CC)nn3)=O)C2C)cc2ccc(Cl)cc2[nH]1 2228,C(=O)(CC1=CCOCC1)N(CCOCCN(C(C(CC#C)(C)C)=O)C)C 2229,C(CCN=C(NC(C)C)NC1CC1(C)C)N(CC)CC 2230,C=Cc1ccc(C(N2CC3CCC2C3NC(=O)Cc2ccn(C)n2)=O)cc1 2231,C(=O)(C(O)CC(F)F)N1C(CCN(C(CCC(C)C)=O)C)CCCC1 2232,C1(CNC(Cc2c(CC)con2)=O)CN(c2cc(C)nc(SC)n2)CC(C)(C)O1 2233,c1(-c2nc(SC)nn2-c2nc3ccccc3n2C)cc(C)nc2c1nc(C)n2C 2234,CC(C)(CC#N)C(=O)N1CCC(NC(=O)C(c2ccccc2F)(F)F)C(O)C1 2235,Cc1cc(CN2CC(c3ccccn3)(C(F)(F)F)C2)cc(C(F)(F)F)c1 2236,c1(NC(CN(C(=O)C(F)n2ccnc2)C(C)C)=O)cnn(CCN(C)C)c1 2237,c1(CC(=O)NCC2(C)CCC(NC(=O)C(N)=O)C2)ccc2c(c1)OC(F)(F)O2 2238,c1(C(=O)NCC(CNC(C(c2c(C)noc2C)CC)=O)C)ccc(C)c(F)c1N 2239,C(=O)(C(C)(C)C(=O)N1CC(NC(=O)Cc2ccc(CC)cc2)C(C)C1)OCC 2240,c1(C(=O)NC(C(C(C)C)NC(c2ccccc2O)=O)C)cncn(C)c1=O 2241,N1(C(C2CCCN(C)C2)=O)CCC(F)(CNC(c2sc(Cl)cc2Cl)=O)CC1 2242,CC1CCN(C(c2cccc(C3CC3)c2)=O)CCN1C(=O)Cc1ncc(Cl)s1 2243,C(=O)(CCCCCCS(N)(=O)=O)NCCC(C)NC(Cn1ncc(CC)c1)=O 2244,c1(CC(N2CCOCC(NC(c3ccn(C)c3)=O)C2)=O)cnc2ncccn12 2245,c1(C(=O)NCC(C2CC2)NC(CCCC#C)=O)[nH]c2c(c1C)CCCC2 2246,C1(CC)CCCCCCN1C(=O)CC(C)C(C)(C)NC(c1cccc(O)c1F)=O 2247,C(=O)(CC1=CCN(C(C2(N(C)C)CC2)=O)CC1)N1CC(CC)OCC1C 2248,CC(C)(CCC#N)C(=O)N1CCC2(CC(NC(C3(n4cnnn4)CC3)=O)C2)C1 2249,C=C=C(C)CC(=O)NCC(CNC(c1ccc(OC(C)C)nn1)=O)CO 2250,N1(Cc2nnc(C(C)C)o2)CCC(NC(c2c[nH]c(C(F)(F)F)c2)=O)C(C)C1 2251,Cc1cc(C(=O)NC2CC3C2CCN3C(c2[nH]cnc2C)=O)cc(C(F)F)c1 2252,c1(NC(C2N(C(c3cc(C)no3)=O)CC(F)C2)=O)cc2nccn2cn1 2253,Cc1nn(CC(C)C)c(C)c1CC(=O)NCC12CCC(CN1C(=O)COC(C)C)C2 2254,CCC(C)C(C(=O)NC1(C)CC2CC2C1)N(C)C(C1CC2CC1CC2=O)=O 2255,CCC(CC)CCC(=O)NCC1(NC(=O)CCC2CC2(Cl)Cl)CCOC1 2256,c1(NC(c2ccc(CNC(CCC(C)OC)=O)cn2)=O)ccc2c(c1)OCC2 2257,N1(C(CS(CC)=O)=O)CCN(C(c2cn(C3CC3)nc2C)=O)C2(CC2)C1 2258,N1(C(c2n(C=C)nnc2)=O)CCOC2(CCN(C(=O)CC(C)(O)COC)C2)C1 2259,c1(C(N(C)CC2C3CN(C(CCC(=C)Cl)=O)CC32)=O)cc(C)c(=O)n(C)c1 2260,C(CCC(N)=O)(C(=O)N(C1CC1)Cc1ccsc1)n1cc(C(C)CC2CCC2)nn1 2261,C(=O)(C(C)(C)CC#N)NCCCC(C)(C)c1cn(CCC(CC)O)nn1 2262,c1(N(C)C)ccnc(C(=O)NC2CCC2CNC(=O)CNc2cccnc2)c1 2263,N1(C(C(C(C)O)NC(C)=O)=O)CCc2ccccc2C(NC(=O)C(C)C(C)C)C1 2264,N1(C(c2c(C)nc(C)s2)=O)CCN(C(c2cccc(Cl)c2O)=O)C(C2CC2)C1 2265,Cc1ccc(C(N2CCN(C(=O)C(N3CCCC3)C3CC3)CC2C)=O)c(C)n1 2266,C12(NC(C3CN(C(c4ccc(NC)cn4)=O)CC3(C)C)=O)CC1COC21CCC1 2267,O=C1CCC(CCC(N2CCN(C3CCN(C(=O)C(O)C(F)F)C3)CC2)=O)CN1 2268,Cc1cc[nH]c(=N)c1C(=O)NCC(C)NC(c1cnn(-c2cccc(F)c2)c1)=O 2269,C(CC(C(=O)N1CSCC1C(N1CCC(CCCO)CC1)=O)OC)OC 2270,c1(C(=O)NCC(CC)NC(c2cn(C)c(C(F)F)n2)=O)cc(C)cc2c1CCC2 2271,N1(C(CCc2ccn(C)n2)=O)CC(CNC(C2(C#N)CC3CC3C2)=O)C(C)(C)C1 2272,C(=O)(C(CC(C)C)C(C)C)N(CC(C)NC(c1c(C)cc(C)nc1S)=O)C 2273,c1(CN(C(=O)NCC(C2CCOCC2)CC)C)cccnn1 2274,N1(C(c2cc(C)no2)=O)CCN(c2nccc(Br)n2)C(C#N)C1 2275,C(=O)(CC(CC)C(C)C)N1CCC(CN(C(=O)C(n2cc(C)cn2)C)CC)CC1 2276,C1(C(N2C(CCCNC(c3cn(CC)nn3)=O)CCC2)=O)CN(C)CC(C)O1 2277,c1(C(=O)NC2C(CNC(CCCc3onc(C)n3)=O)CCC2)cc(F)ccc1N 2278,c1(C(=O)NCC2N(C(C3CCN(CC)C3)=O)CCOC2)[nH]cc2c1CCCC2 2279,N1(C(c2ncn(CCNC(C(COC)OC)=O)c2)=O)CCC2CCC(C1)S2 2280,C(C(C)C(C)C(=O)NCC1(CNC(C23CCC(CC2)C3)=O)CCCC1)OC 2281,c1(C(=O)NCCn2ncc(C(=O)NC(CCC)(C)C)c2)cccc(O)c1C 2282,C=C=CC(C)C(=O)NC1CC(C)(NC(=O)CSc2ccc(C(C)(C)C)cc2)C1 2283,N1(C(=O)Cn2cnnc2)CCC2(CCN(C(c3c(F)ccc(F)c3F)=O)C2)C1 2284,c1(C(=O)NC2C(NC(C3N(C(C)=O)CCC3)=O)C2)cccc(F)c1Br 2285,C(=O)(CCC(=O)N1CCCC1(CC(C)C)C(=O)O)OCC 2286,n1(CCC)ncc(C(=O)NCC2CCCC(NC(=O)Cc3cnnn3C)C2)c1C 2287,FC1(F)C2(NCc3nccn3-c3ccc(F)cc3)CCCCC12 2288,C1(NC(c2cc(OCC)ncc2)=O)C2CC1CN(C(c1cscn1)=O)C2 2289,CC(CC(=O)N1C2CCC1(CNC(=O)CC1CC1(C)C)CC2)C(F)(F)F 2290,C1(NC(C(C)(F)F)=O)CCC(NC(=O)C(C)(O)c2ccccc2)CC1 2291,c1(CNC(C(C)OCCOC)=O)cccc(CN(C)C(c2sc(C)nc2C)=O)c1 2292,N1(C(C(CCC)OC)=O)CC2(CCCCN(C(=O)C(c3cncc(F)c3)C)C2)C1 2293,c1(CN(C)CC2CCCN(C(C3C(CC)CCCC3)=O)C2)ccc(O)c(O)c1 2294,C1(C(=O)NC(CCC)C)CN(C(=O)CCCF)CCC1(C)C 2295,c1(C(=O)NCCN(C(=O)C(n2ccc(Br)n2)C)CC)c(C)ncn1O 2296,c1(OC)cc(C)ccc1C(N1CCC(=CCNC(c2nc(CO)cs2)=O)CC1)=O 2297,c1(C(=O)NCCCC2N(C(C(C)SC(C)C)=O)CCC2)cc(Br)n(C)c1 2298,c1(C(N(C)CC2N(C(c3cc(C)nnc3)=O)CCOC2)=O)c(C)nn(C)c1C 2299,C1(NC(=O)Cn2cnnn2)CN(C(c2cc(F)c[nH]2)=O)CC2(CCC2)C1 2300,c1(CCC)[nH]ccc1C(=O)NCCCCNC(c1ccsc1CC(=O)OC)=O 2301,c1(C(N2C(CC(C)O)CCC2)C(=O)NC2CCC2)ccc(S(C)(=O)=O)s1 2302,C(=O)(C(C)(C)CC(=O)N(C)CC1(O)CCN(C(=O)C2=NNC(=O)CC2)CC1)OC 2303,C(Cc1ccccc1)(CCNC(=O)CN(C1CCC1)C)NC(C(C)O)=O 2304,N1(C(c2csc(Cl)c2)=O)CCCN(C(=O)C(O)C2CCCC2)C(CO)C1 2305,O=C(C1NCCc2ccccc21)NCC(C1CCCCC1)=O 2306,c1(C(=O)NC(C2OCCN(C(C(C)=CC3CC3)=O)C2)C)cncc([N+](=O)[O-])c1 2307,CCC(F)(CNC(=O)NC(C1CS(=O)(=O)C1)C)CC 2308,c1(C2CN(C(C(C)(C)C)=O)C2)nc(C2CC3CC2C3)[nH]n1.c1cccc(F)c1 2309,c1(C(=O)NCC2CCCC(NC(C(C#C)(C)C)=O)C2)nccc(F)c1Cl 2310,c1(C(=O)NCC(CNC(C2(OC)CCOC2)=O)OC)cc(C2CC2)n(C)n1 2311,C1(CN(C)C(C2(NC(=O)CC3CS(=O)(=O)C3)CC2(C)C)=O)COC(=O)N1 2312,C1(NC(c2c(C)nn[nH]2)=O)CCN(C(=O)Cc2cc(F)cc(Cl)c2)C(C2CC2)C1 2313,c1(C(=O)NC2CCC(CNC(CCCC=C)=O)CC2)c(C)cnc2ccccc12 2314,c1(CC)cc(F)ccc1C(N1CC(O)CC1CNC(C1(C#N)CC(C)C1)=O)=O 2315,n1(CCNC(=O)CC(CC=C)Sc2cn(CC=C)nn2)ccc2cccnc12 2316,C1(c2onc(CC(C(C)C)Sc3ccccc3)n2)CCCC(=O)N1 2317,CC1CN(C)CC1C(N(CCCCO)NC(=O)CSCC(F)(F)F)=O.c1(C)cccnc1 2318,C1(C(N(C(C2CCCCC2)C)C)=O)COC2(CNC2)C1 2319,c1(C(=O)NC2CCCC(N(C(CC3CC(OC)C3)=O)C)C2)ccc2cc[nH]c2n1 2320,Cc1cc(C(=O)NCC2CC(NC(=O)C(C#N)C(C)C)C2)c2c(C)nn(C)c2n1 2321,C(C(O)CC(=O)NC(C)(C)C)N(C)C.c12ccc(nc1)C(=O)N(C)CCNC2=O 2322,c1(NC23C(CN(C(=O)C4=CCCC4)C2)CCC3)ncc([N+](=O)[O-])cc1CO 2323,CC1=CCC(C(=O)NCC23CC(NC(c4cnn(C(C)(C)C)c4N)=O)(C2)C3)CC1 2324,C1(CC(=O)NC2(F)CN(C(=O)COc3ccc(CO)cc3)C2)CCCC1(F)F 2325,N1(C(Cc2c(C)nc[nH]2)=O)CCC(NC(=O)CCc2cncn2C)C12CCC2 2326,CCC(CCC(=O)NCCOCC1CCCC1)NC(=O)CS(=O)CC 2327,c1(NC(=O)NNC(=O)c2ccccc2F)ccc2cc[nH]c2n1 2328,c1(NC(C2C(NC(CCCOC)=O)CC2)=O)ccc(SC)nc1 2329,C1(C(=O)NC(C)(CO)C(=O)NCCC2(C)N=N2)CCC=CCCC1 2330,C1(C(=O)NC(CC#C)C(=O)NC(CO)C(C)(C)C)CC2C(C1)C2(F)F 2331,CC1(C)C(C(=O)NCC(CO)NC(=O)C2=NOCC2)CC1(F)F 2332,N1(C(CSCCC)=O)CCC2(CC2)CC1C(N1CC2CC2(C(=O)OC)C1)=O 2333,Cc1noc(Cl)c1CC(N1CCCC(c2cn(CCN(C)C)nn2)C1)=O 2334,N1(C(C(C)Sc2ccccc2Cl)=O)CC2(C1)CN(C(=O)C(C)N(C)C)CC2CO 2335,c1(CC(CC)C)nc(-c2nn(C)cc2Br)n(-c2cnnn2C)n1 2336,Cc1ccc(C(N2CCC2C(N2CC(CC(N)=O)C2)=O)=O)[nH]1 2337,Cc1ccn(CC(=O)N(CCNC(=O)Cc2nc[nH]n2)C(C)C)n1 2338,C=CCC(C)C(=O)NC1CC(NC(=O)CCSc2nccn2C)C1 2339,c1(OC)cc(C(N2CC(CC(C)NC(c3csc(Cl)n3)=O)C2)=O)cc(F)c1 2340,c1(C(=O)NCC(CC)NC(C2CCCC23CC3)=O)cnn(C(C)(C)C)c1Cl 2341,Cc1nn(CC(=O)NC2(CN(C)C(C3CCCNC3=O)=O)CC2)c(C)c1C 2342,CC(C)(C(=O)NC1CCCN(C(=O)CN2CC3C=CC2C3)CC1)C(N)=O 2343,C1(CNC(Cc2c(C)n(C)cn2)=O)CCCCCN1C(=O)C(c1cccn1C)=O 2344,C(=O)(CCC1=CCCCC1)NCC(COC)NC(=O)CC(C)O 2345,N1(CC)CC(NC(=NCc2ccoc2)NCc2nncn2C)CCC1=O 2346,S(=O)(=O)(c1cccc2scnc12)NC1CCN(C(c2ccn(CC)n2)=O)CC1F 2347,CON(CCC(=O)NC(CCO)C(F)F)C(=O)CC(C)c1ccco1 2348,c1(C(=O)Nc2cccc(C(=O)NCCC(O)CCO)c2)cc2ncccn2n1 2349,N1(C(c2cc(C)cc(C)c2)=O)CCN(C(c2nnsc2C)=O)C2CCCCC12 2350,CC1CC(NC(=O)Cc2cc(F)ccc2O)CN(C(c2cc(Cl)c(Cl)[nH]2)=O)C1 2351,C12(C(N3CCC(O)(CNC(C(CC)(F)F)=O)C3)=O)CC(C(=O)OC)(C1)C2(F)F 2352,C1(CC(=O)NC(C)CNC(c2cccnc2)=O)CC(F)(F)C1(F)F 2353,C1(C(C)(C)NC(=O)Cn2ncnn2)CCCCN1C(=O)CC1(O)CCC1 2354,C=CC(C)(C)CC(=O)N(C1CCCCC1N(C(=O)CN1CC2CC2C1)C)C 2355,C1(CCOC)CN(C(=O)CC(C)COC)CCN1C(=O)C(C)Cc1cnco1 2356,c1(C(=O)NC2(CNC(c3ccnnc3S)=O)CCOC2)ccc(Cl)cc1Cl 2357,Cc1cc(P(C)(C)=O)oc1C(N1CCC1CNC(=O)Cn1cc([N+](=O)[O-])cn1)=O 2358,N1(C(C2CCC(CNC(C3(C4(C)CC4)CC3)=O)CC2)=O)Cc2cncnc2C1 2359,C(=O)(C(C)(CO)NC(c1cnnn1C)=O)N(C(CC(C)C)C)C 2360,c1(CNC(CCN(C)C(C2CCCN2C)=O)=O)ncc(Cl)cn1 2361,c1(C(=O)NC2CC(C)(CNC(c3coc(Cl)c3)=O)C2)nnn2c1C(=O)NCC2 2362,c1(NC(C(C=C)F)=O)ccccc1NC(=O)CCc1ccc(C)cc1 2363,C(C)(CO)(C(=O)N(C)CC1(CNC(=O)CCn2ccnc2C)CC1)NC(C)=O 2364,N1(C(C=CC(C)C)=O)CC2CN(C(=O)CN3OC(C)(C)CC3=O)CC2(C)C1 2365,CC1CCN(C(c2cccc3c2CCC3)=O)CCN1C(=O)CCc1ccncn1 2366,CC1=C(C(=O)N2CCCC2CCNC(c2cnc(O)c(Br)c2)=O)CCO1 2367,C1(C(=O)NCCCCN(C(Cc2nc(NC=O)sc2)=O)CCO)CCC=CCC1 2368,Cc1ccccc1C(C)NC(=O)C(C1(O)CCC1)NC(=O)COC(C)C 2369,C=C(C)C1CN(C(c2cc(C)c(=O)n(C)c2)=O)CCO1.C12CCN1C2 2370,c1(C(N2C3(CNC(c4cc(C)[nH]n4)=O)CCC3CC2)=O)cc(S(C)(=O)=O)cs1 2371,N1(C(C(C)=CC)=O)CCC(NC(c2nccc(OC)c2OC)=O)C(CC)C1 2372,Cc1cccc(N)c1C(N1CC(CCNC(c2ccnn2C(C)C)=O)C(C)C1)=O 2373,CC1(S(C)(=O)=O)CC1C(=O)NCC1CCN(C(=O)CNc2ccccn2)C12CC2 2374,CCC(C)C(C)C(=O)NCCCCn1cc(-c2cn(C)nc2C(=O)OC)nn1 2375,c1(CNC)ccc(NC(c2sc(C(C)C)nc2C)=O)cc1 2376,CC1CN(C(=O)Cc2ccn(C)n2)CC1(C)CNC(=O)Cn1ccccc1=O 2377,c1(C(=O)OC)cn(C)nc1C(=O)NC(C)CN(C(=O)CC12CCCC1C2)C 2378,Cc1cc(C)c(C(=O)NC2CCCCC2N(C(=O)CCn2cnnn2)C)c(O)n1 2379,N1(CC(c2ccc(C)cc2)n2cc(-c3cscn3)nn2)CC(C)OC(C)C1 2380,c1(N2CCC(CC)C2)nc(N2CCC(C)(COC)C2)c2ncsc2n1 2381,C=CCCCC(C(=O)NCCNC(c1csc(C)n1)=O)NC(c1ccoc1)=O 2382,CS(=O)(=O)c1cc(C(=O)NCc2c[nH]nc2C(F)F)c(Cl)cn1 2383,CS(=O)(=O)C1(C(N2CC(O)(CNC(C3CCCCS3)=O)C2)=O)CCOCC1 2384,N1(C(C(Br)=C(C)C)=O)CCC(C2CC2)(CNC(c2ncnc3c2CCC3)=O)C1 2385,C1(C(N2CCSCC(C)C2)=O)COC2(C1)CN(C(c1c[nH]c(C#N)c1)=O)C2 2386,N1(C(c2cc(C)[nH]c2C)=O)CCN(C(=O)CC#N)C2CC12 2387,N1(C(C(COC)(F)F)=O)CCC2OCCN(C(=O)Cc3nc(CSC)no3)C2C1 2388,c1(C(N2CC(CNC(CCCOC)=O)OCC2)=O)cc(Cl)c(F)cc1OC 2389,c1(NC(C2CCCC2NC(C2CC23CCOC3)=O)=O)c[nH]ccc1=O 2390,C1(OCC)CC2CN(C(=O)C(CN(C)C)NC(c3c(C)noc3N)=O)CC12 2391,c1(N2CC(C=C)OCC2)cc(S(=O)(=O)NC2CC3(CC3)C2)ccc1C#N 2392,c1(C(N2C3CN(C(C(C)O)=O)C(C3)C2)=O)ccc2c(O)nnc(O)c2c1 2393,c1(C(=O)NCC2(C(=O)NC(c3ccc(F)cc3)C)CC2)ccc([N+](=O)[O-])cn1 2394,C1(CC(=O)NCC(CC)N(C)C(c2n[nH]c(C)c2C)=O)OCCCC1(C)C 2395,Cc1cc(Cl)cc(C)c1C(=O)OCCC(=O)NC1COC1.C1C=CC1 2396,C12(CNC(c3n(CC#C)ccc3)=O)CN(C(=O)CN3CCCC3)C(COC)(C1)C2 2397,C1(NC(CCCN(C)C)=O)CN(C(C2CC2c2ccc(F)cc2F)=O)CC12CC2 2398,C1(C(N(CCCN(CC)CC)C)=O)CN(C(=O)Cn2cccnc2=O)C(C)(C)C1 2399,N1(C(CNC(CN(S(C)(=O)=O)C)=O)C(F)F)CCN(C(C2(C)CC(C)C2)=O)CC1 2400,C(C(C)C(F)C(=O)N(CC(C)O)CC)NC(CC1(OCC)CC1)=O 2401,C1(C(=O)NC2CC(CNC(COCC=C)=O)C2)CC2(C1)CC1(CCC1)C2 2402,C1(CN(C)C(C2CC(C)(NC(=O)C(C3CC3)C3CC3)C2)=O)CCCCO1 2403,C1(CC)C(NC(c2cnc(CC(C)(C)C)o2)=O)CCCN1C(c1cnco1)=O 2404,c1(C(N2C(CNC(C3N(N=O)CCCC3)=O)C=CC2)=O)ncnc2ccsc12 2405,N1(C(C2N(CCC)CCC2)=O)C(C)CN(C(C2(C)CC=CC2)=O)CC1C 2406,CC(C)(C)CC(O)C(=O)N1CCN(C(=O)C=CCN2CCC2)CC(O)C1 2407,Cn1ncc2ncnc(N3CCN(C(C4CCC(C)CC4)=O)CC3)c12 2408,N1(C(CCNS(CC)(=O)=O)=O)CCCC1C1(NC(=O)C(F)OC(F)(F)F)CC1 2409,Cn1c(O)nc2c(C(=O)NC3CCN(C(c4cnc(O)s4)=O)CC3F)cccc12 2410,c1(SC)cc(C(=O)NCC(C2CCN(C(=O)C(O)c3ccco3)CC2)C)oc1C 2411,c1(C(N(CC(C)CNC(=O)Cc2cccnc2Cl)C)=O)ccnc2c1CC(=O)N2 2412,n1(C(C)C)nncc1C(=O)NCC(CNC(C1CC=CCC1)=O)CO 2413,N1(C(C(C(=C)C)(C)C)=O)CC(NC(=O)C(C)(C2CC2)OC)CC2(CCC2)C1 2414,c1(C(=O)NCCCCC(C)NC(Cc2c(C)nccc2)=O)ccc(S(C)(=O)=O)o1 2415,C(=O)(C#CC1(C)CCCO1)NC(CC(C)NC(c1nnc(C(C)C)s1)=O)C 2416,C1(N(C(=O)CC2CC2)C2CC2)CCCCC1.C1(C)CCOCC1 2417,C1(C(N2CC(C(C)NC(C3CCC(=O)O3)=O)C2)=O)CCC2CC2CC1 2418,O=S(=O)(c1ccc(NCC(O)CCC2CC2)c(F)c1)N1CC2CC3CC2C1C3 2419,C1(C(=O)NCc2ccc(C(=O)NC(CNC(=O)OC)C)s2)CCCC(C)C1 2420,N1(C(CS(N)(=O)=O)=O)CCC2CCN(C(=O)COCc3nc(C4CC4)no3)CC12 2421,C1(CN(C)C(c2csnc2Br)=O)CCCN1C(c1ccnnc1)=O 2422,CCC(C(=O)N1CCC(CCNC(c2c[nH]c(C)c2)=O)C1)OC 2423,C(=O)(C(F)C1=CCCCC1)NC(CCNC(c1ncc(CC)s1)=O)C 2424,Cn1cnc(CCC(=O)NCCSCC(N2CC(OCC(N)=O)C2)=O)c1 2425,Cn1ncc(NC(C2(CCCF)CC2)=O)c1-n1cc(C2(N(C)C)CCOC2)nn1 2426,C1(C)(C(=O)OC)CCN(C(C2CCN(C(C3CC4CC4C3)=O)CC2)=O)C1 2427,C(=O)(CC1=NNC(=O)C1)N1CCC(NC(C(C)N(CC)CC)=O)C(C)C1 2428,C1(NC(CN(C(C)C)C(C2CCC3CC2CO3)=O)=O)CN2CCC1CC2 2429,n1(CC(=O)NC2CCN(C(=O)C=CC3CCCCC3)C2)nc(Cl)ccc1=O 2430,CCC(CCC(=O)N1CC(CC(=O)N(C)Cc2cn[nH]c2)CC1(C)C)OC 2431,C(=O)(C1CNC(=O)c2ccccc21)N1CC2C(NC(CCOC)=O)C(C2)C1 2432,C1(C(C(N2CC(CC=CC)C2)=O)C)CCCN(C(=O)C(C)=C(C)CC)C1 2433,CC(CCCCO)NC(=O)C=CCN(C)C(c1cscc1Cl)=O 2434,C1(CCCNC(C=C(C)C)=O)CCCCN1C(C12CC(C(C)C)(CO1)C2)=O 2435,C1(CC(N2CC(C(C)(C)O)C2)=O)COC2CC1C2.C12CC(C1)C(C)NC(=O)C2 2436,c1(C(C)=O)ccccc1C(=O)NC1CCN(C(C)=O)C1C(=O)O 2437,c1(C(N2C(C(N(C3(CC)CC3)C)=O)CC2C)=O)ccc(C)c(F)c1 2438,C1(C(=O)NC2(C)CN(C(CC3C(C)CCC3)=O)C2)(CO)CCCCO1 2439,c1(NC(N2C(C(=O)Nc3ncn(CC(C)C)n3)CC2)=O)cc(OC)c(F)cc1F 2440,c1(C(=O)NNC2CC(CCO)C2)cccc2occc12.C1CCCNC1=O 2441,C1(C2CCN(C(=O)CC3(C#N)CCC3)C2)(NC(COC(C)(C)C(F)(F)F)=O)CC1 2442,N1(C(C2C(C)(C)C2(C)C)=O)CC2CCN(C(=O)C3Cc4ccccc43)C(C2)C1 2443,Cc1oc(C(C)C)cc1C(=O)NCCC(O)CNC(C1CC1c1ccccc1)=O 2444,C(CCC(=O)NCC=CCNC(c1c[nH]cc1C(C)C)=O)=C(C)C 2445,C12(C(=O)NC3(CCNC(C4C(c5n(C)ncc5)C4)=O)CC3)CC1COC21CCC1 2446,C(=O)(CC(O)CC(C)(C)C)N1CC(NC(CCCOC)=O)C2(C1)CC2 2447,c1(NC)c(C(N2CCCC(NC(C3(C)CCC(F)(F)C3)=O)C2C)=O)cccc1N 2448,C12(C(N3CCC(NC(C4C(CC)CCO4)=O)(CO)CC3)=O)CCC(F)(CC1)CC2 2449,Cc1nscc1C(=O)NCCCC1CCCN1C(=O)COCC1CCCCO1 2450,N1(C(CP(C)(C)=O)=O)CCOC(C(=O)NCC2CCCO2)CC1 2451,C1(CN(C2CCCCC2)CC(=O)NCCC)CCN(C)C1 2452,N1(C(C2N(CC)CCCC2)=O)CCCC(C2CCN(C(=O)C(C)CCO)C2)C1 2453,c1(C(N2CCC(NC(CC=C(C)C)=O)C2C)=O)ccc2c(c1)CCC(C)(C)O2 2454,C1(C(N2CCC(O)(CN(C)C(C3C=CCC3)=O)CC2)=O)C2CCC1(C)C2(C)C 2455,N1(C(CCCN(C)C)=O)CCC(CC(C)NC(=O)COC(C)(C)C)CC1 2456,c1(CC(=O)OC)ccccc1C(=O)NCC(CO)NC(=O)CC1OCCC1(C)C 2457,S(=O)(=O)(c1ccc(F)cc1)NCC(N1CCC(n2nncc2C)CC1)CC 2458,c1(C(=O)NCC(CNC(c2coc(Cl)c2)=O)OC)ccc2ccn(C)c2c1 2459,C(CCC(=O)NCCC(=C)CNC(=O)C(C)NC(=O)CC1C=CCC1)=CC 2460,C=C(Cl)CC(C(=O)N(C1CCCC1C)C)NC(C1CNC(=O)O1)=O 2461,c1(N(C(C)C)C)ncc(CN2CCSCC(C)C2)cc1F 2462,C1(N(C(C(CC)C)=O)C)CN(C(=O)Cn2nc(Cl)ccc2=O)CC1(C)C 2463,C(CN=C(NCc1ncnn1C)NCCN1CCOCC1)C1CC(C)OCC1 2464,C12(C(=O)NCC=CCNC(c3cccc(O)c3F)=O)CCC(CC1)CC2 2465,C1(C(N2C(C(C)NC(c3cc(C)sn3)=O)CCCC2)=O)CN2CCN1CC2C 2466,CCC(CC(F)(F)F)C(=O)NC(C)(CNC(=O)Cc1cc(C(F)(F)F)n[nH]1)CC 2467,C1(CNC(CCCCNC(C=CC(=O)OCC)=O)=O)CCCCC(O)C1 2468,C1(NC(NCC2(O)CCCC2)=NCCF)CC2(CCC2)C12CCC2 2469,c1(C(N(C(CNC(=O)COC2CC2)C2CC2)C)=O)ccc(S(N)(=O)=O)c([N+](=O)[O-])c1 2470,N1(C(CNC(C2(C#N)CC2)=O)=O)CCN(C(=O)CC2CC3(CC3)CO2)CC1 2471,c1(C(=O)NCCCCC(C)NC(=O)CN(CC(C)(C)C)C)cccc(C#N)c1Br 2472,C1(NC(c2c(C3C(C)C3)noc2)=O)CC(F)CN(C(=O)Cc2cn(C)nn2)C1 2473,c1(C(=O)NCCCCN(C(=O)Cn2cnnn2)C)sccc1Cl 2474,CC1CN(C(=O)CC2CCN(C(c3ccn4c3CCC4)=O)C2)CC(=O)N1C 2475,N1(C(CN(C)CC)=O)CC(CNC(=O)COCCCOC(C)=O)C2(CC2)C1 2476,c1(CCC)c(C(N2CC(CNC(c3occc3C)=O)CC2C)=O)nnn1CC 2477,N1(C(CC(C)=C(C)C)=O)CCC(C)(CCNC(c2ccc(C3CC3)o2)=O)C1 2478,c1(C(N2CCOC(CCCNC(=O)C3CC3)C2)C(=O)NC)ccc(C2CC2)cc1 2479,c1(CNC(c2ccc(NC(C3CCC(F)C3)=O)nc2)=O)cc(Cl)ccc1[N+](=O)[O-] 2480,c1(CC)c(C(=O)NCCC(C)(C)NC(=O)CCc2ncc(F)cn2)csc1C 2481,N1(C(c2nc(CC)oc2C)=O)CCN(C(c2ns[nH]c2=O)=O)CC2CCCCC12 2482,C(=O)(C1=CCC2CCC1N2C(=O)C(C(=O)OC)OC)N1C(CC)CC1 2483,C1(O)(CCNC(c2cc(C)oc2)=O)CCN(C(C2CC(N(C)C)C2)=O)C1 2484,N1(C(C(c2ccc(Cl)s2)C)=O)CC=C(CNC(=O)CC2(C(F)(F)F)CC2)CC1 2485,N(C(=NCCN1CCCCC1C)N1CCC2(CCCOC2)C1)Cc1cc(C)on1 2486,C(=O)(C1=NNC(=O)CC1)N1CCC(O)(CC(=O)Nc2cc(OC)cc(Cl)n2)CC1 2487,c1(CC(=O)NCCN(CCOC)C(c2cnc(O)o2)=O)ccccc1Br 2488,C1(NC(C2CCCC23CC3)=O)COCCN(C(c2ccc(F)cc2F)=O)C1 2489,c1(C(=O)NCC2(CNC(COC)=O)CCCC2)cnn(C)c1Cc1ccccc1 2490,Cc1cnc(NC(C2CC23CN(C(c2cnc(Cl)cn2)=O)C3)=O)cc1F 2491,c1(NCC(=O)NC(C2CS(=O)(=O)C2)C)cccc(Cl)c1Cl 2492,C1(NC(C(=Cc2cccs2)C)=O)CC(CNC(c2coc(C)n2)=O)C(O)C1 2493,c1(CC)nn(C)c(Cc2nc(-c3ccn(C)n3)nn2CC2CC2C)c1Cl 2494,Cc1cccc2c1N(C(C1CCCC1NC(=O)CCC1CCCCO1)=O)CC2 2495,c1(C(=O)NCC2(CN=c3nc(C4CCCC4)[nH]s3)CCC2)cnc2[nH]cncc1-2 2496,c1(C(=O)NC(CC)(C)CNC(=O)CC2CCN(C)C2=O)nccc2c1CNC2=O 2497,C1(C(=O)NC2C(=O)OCC2CO)(NC(C(C(C)C)F)=O)CCc2cc(Br)ccc2C1 2498,O=C1COc2ccc(C(=O)NC3CN(C(=O)C=CCF)CCC3F)cc2N1 2499,C(=O)(C(F)(F)CC1CN(C(=O)NCC2(n3cccn3)CC2)C1)OC 2500,CCCCC(CCCC)NC(=O)CC(C)(C)N(C(=O)Cc1cccc(C#N)c1)C 2501,N1(C(C(CC)C(C)C)=O)Cc2ccccc2OC2(C1)CN(C(C1CC13CC3)=O)C2 2502,C(=O)(C1=NNC(=O)CC1)NCC=CCNC(c1cnc(OCC)nc1)=O 2503,c1(C(=O)NC(CC)CNC(=O)C(C)=C(C)CC)ccc2nnnn2c1 2504,c1(OC)ncc(C(=O)NCC2(C)CN(C(=O)C(C)N(C)C)CCO2)nc1C 2505,N1(C(CCC=C(C)C)=O)CC2CC1(C(=O)NC1(C)CS(=O)(=O)C1)C2 2506,c1(C(=O)NC2(CN(C(CC(C)(C)SC)=O)C)CC2)cnc2c(C)cccn2c1=O 2507,C1(C(=O)NCCCCCCNC(CCCC)=O)C2CCC(C2)S1(=O)=O 2508,C(CC(=O)NCC1(NC(C2CC2CF)=O)CC1)OCC#C 2509,Cc1coc(C2CC2)c1C(N1CCC(OCCNC(C2CC(O)C(F)C2)=O)CC1)=O 2510,c1(CNCC23C(CN(C(c4cc(CC)nn4C)=O)C2)C3)c(Cl)ccnc1Br 2511,CCC(CC(=O)N(C)CC1CN(C(c2n[nH]c(C3CC3)c2C)=O)CCO1)C(C)C 2512,N1(C2CN(C(C(=O)NC)COC)C2)CC(NC(c2c[nH]nc2C(F)F)=O)CC1=O 2513,C#CC1CN(C(=O)CCC2CCCN(C(=O)C(C)=C(C)CC)C2)CC1OC 2514,C#Cc1ccc(C(=O)NCCN(C(=O)Cc2conc2C)CC2CC2)cc1Cl 2515,N1(C(c2ccc(CC(C)C)s2)C(=O)NCc2ccccc2)CC2CSCC2(C)C1 2516,CC(CC(=O)NCC1CC(NC(c2csc3c2CCCC3)=O)C1)C(F)(F)F 2517,CCC(CCOC)C(=O)N1CC(NC(C2Cc3nccn3C2)=O)C1 2518,c1(C(N(CCC(=O)NCC(O)CCC)CC=C)=O)ccc(C#N)n1C 2519,C(c1cc(C)no1)=CC(=O)NC(CNC(CNS(CC)(=O)=O)=O)(C)C1CC1 2520,N1(C(CC(C)CNC(C2(C)SCCCS2)=O)=O)CC2(CCOC2)C1 2521,C1(C(=O)NCC(C)CNC(C2(C)CC(C#N)C2)=O)CC(c2cccc(F)c2)=NO1 2522,c1(C(N2CC(N(C(C(C=C)O)=O)C)C(O)C2)=O)nn(C)cc1S(N)(=O)=O 2523,C(=O)(C(C(=O)NC1(CNC(C2CC2(Cl)Cl)=O)CCCCC1)C1CC1)OC(C)(C)C 2524,C1(NC(C2C=CCC2)=O)(CF)CCN(C(c2cncc(C(F)(F)F)c2)=O)C1 2525,C1(CNC(c2ncc(OCCOC)nc2)=O)CN(C(c2ccns2)=O)CC1(F)F 2526,CCCC(C)C(=O)N1CCC(C2OCCCC2NC(=O)CCc2cnco2)CC1 2527,C12(NC(C=COCC)=O)CCCC1N(C(c1cncs1)=O)CC2 2528,c1(CC)cnc(O)c(C(N2CC(NC(C3(CN(C)C)CC3)=O)C(C)C2)=O)c1 2529,N1(C(C(C)C2CC2)=O)CCN(C(C2CCC(OC(F)F)CC2)=O)CC1C 2530,N1(C(C)C)CCCC1CC(=O)N(C(C)CCNC(=O)CCCN(C)C)C 2531,C(N=c1cc[nH]c(=NCCc2cc3ccccc3[nH]2)[nH]1)c1c(C)occ1 2532,C(CCN(C)C(C1(Cl)CC1(C)C)=O)(C(C)C)NC(c1cc(CCCCC)[nH]n1)=O 2533,N1(C(c2ccc(CC)s2)=O)CCC(C)C(NC(=O)CCC(F)F)C1C 2534,CC1(C2CCCN(C(=O)CC3CCCN(C(c4cn[nH]c4)=O)C3)C2)CC1 2535,N1(C(CNC(C2C=CS(=O)(=O)C2)C)=O)CCCC2(C1)NC(=O)N(C)C2=O 2536,C1(CNC(CCN(C)CC)=O)COCC2(CCN(C(=O)C(F)=C3CCCC3)C2)O1 2537,c1(C(N(C(=O)C(N2CCCC2CC2CCC(OC)C2)=O)CC)C)cccc(C)c1 2538,C1(NC(C(CC#CC)NC(c2cc(C(C)=O)[nH]n2)=O)=O)CCN(C)CC1C#N 2539,N1(C(C2C(CC)OCC2)=O)CC(C2CCCN(C(=O)C(C)(C)C3CCC3)C2)C1 2540,C1(CC)CCC(C)CN1C(C1CN(C(c2cnn(C(C)C)c2)=O)CC1(C)C)=O 2541,C1(C(=O)NCc2c(C(=O)OC)nn[nH]2)CCCCN1S(C)(=O)=O 2542,c1(CC(=O)N(CCCNC(c2cccn2C)=O)C(C)C)cccc2ccccc12 2543,C(=O)(CC(C(F)F)NC(c1c(C)csc1C)=O)NC(COC)C(=O)OC 2544,C(=O)(N=c1[nH][nH]c2c1CNC2(C)C)C1CC1.c1(NS(CC)(=O)=O)ccc2ncsc2c1 2545,c1(C(=O)NC(C(C(=O)N(CC(=C)C)C)C)C)ccc(=NC)[nH]c1 2546,C(=O)(CC(F)(F)C(C)C)N1CC(CCNC(C2N(CC)CCCC2)=O)OCCC1 2547,c1(C(N2CCC(CN(C(C(CC)(C)OC)=O)C)CC2)=O)ncncc1C#N 2548,O=C(C(O)C(F)(F)F)NC1CCCS(=O)(=O)C1 2549,C=Cc1cncc(C(=O)NCC2CC3CC3N2C(c2cc(CO)[nH]n2)=O)c1 2550,CN1CCC(C(=O)NCC2CCCN2C(=O)CNC(C2CC2CF)=O)CC1=O 2551,c1(CN2CCCC(NC(c3ccc(CN(C)C)cc3)=O)C2)ccc(F)c(C#N)c1 2552,C1(CSCC(=O)NCCCNC(Cc2nc(C)oc2)=O)CCc2ccccc2O1 2553,C(=O)(CC1OCc2ncccc21)NCCCN(C(C(CCSC)O)=O)C(C)C 2554,c1(C(=O)NC2CCN(C(c3ccc(CNC(C)=O)s3)=O)C2)csc(C#N)c1 2555,N1(C(CC(C)(C)NC(Cc2scc(C)c2)=O)=O)CCN2CC(O)CC2C1 2556,C(C(C)C(=O)NCCC(Cc1ccccc1)NC(c1nscc1N)=O)SC 2557,CC(C)C(C)C(CNC(C1CCCCC1)=O)NC(c1cn(C)nc1C(C)(F)F)=O 2558,N1(C(C(c2scc(C)c2)C)=O)CCCCC2(CCN(CCN3CCCCC3)C2)C1 2559,CCC(C)CCCC(=O)N1CC2(CC2)CC1C(N1CCC2(CC1)N=N2)=O 2560,C(CCCC(C)NC(c1cnc(Cl)s1)=O)NC(C1(CC)CC1(F)F)=O 2561,C1(C(=O)NC(CSC)C)CC2CC1CN(C(c1ccc(O)cc1F)=O)C2 2562,C=C(C)C1OCCCC1C(N1CCC1CNC(c1cc(C)n(C)n1)=O)=O 2563,C(=O)(CC(O)C(Cl)(Cl)Cl)NCC1CCC(NC(c2c(C)ccc(F)c2)=O)CC1 2564,C1(CC#C)(C(N2CC(CC=C)(NC(=O)C(O)Cc3cnc[nH]3)C2)=O)CCCCO1 2565,N1(C(C2(CC)CC2)=O)CCOC(C)(C)CC1 2566,C1(C(N2CCC(C)(F)C2)=O)N(C(=O)Cc2csnn2)CC12CCCC2 2567,c1(CC)n[nH]c(CC)c1CC(=O)NC12CC(CNC(=O)C(C)C#N)(C1)C2 2568,C(=O)(C(C)(C)CC#N)NC(C(C)C)CCN(C(=O)C(c1ccccc1)C1CC1)C 2569,C#Cc1cn(C)nc1C(=O)NC(C)CC(C)NC(=O)C(C)(C)C#C 2570,c1(NC(CCC2N(C(c3c(C)ccc(F)c3)=O)CCC2)=O)ncnc2occc12 2571,C1(CNC(C2(C(CC)(F)F)CC2)=O)(NC(=O)Cc2ncccc2C)CCOCC1 2572,N1(C(C(CC)OC)=O)CCC(O)(C2(NC(=O)C(CC)NC(C)=O)CC2)CC1 2573,C1(CNC(CN(C2CCS(=O)(=O)C2)C)=O)CN(C(C23CC4CC2C3C4)=O)CCO1 2574,c1(OCC)c(C)n[nH]c1C.C(CCC(=O)N1CCC(C2CCCN2CC)C1)OCCO 2575,C(=O)(CC(C)C(C)C)NCC(CC(C)C)NC(c1scnc1C1CCCC1)=O 2576,C1(C(c2nnnn2CCC2CC2)NCCCOCCCCC)CC2CCC1CC2 2577,CN1CCN(C(=O)C=Cc2ccc[nH]2)C(C(=O)N(C2(C)CC2)C)C1 2578,CC1(C)OC2(CNC(=O)CCCC#N)CC1(NC(C1CC13CCCOC3)=O)C2 2579,C1(CNC(CCc2cccc(OC)n2)=O)CCCCN(C(=O)CCS(C)(=O)=O)C1 2580,C(CC=C)(CC(=O)N(CC(C1CCCC1)O)C)NC(C(C=C=C)C)=O 2581,C(C(=O)O)(C(C)(C)C)NC(C1N(C(=O)OC(C)(C)C)C2C(C1)C2)=O 2582,Cc1c(C(=O)NC2CCC23CN(C(C2COC(=O)C2)=O)C3)oc2ccc(F)cc12 2583,Cc1c(NC(=O)CN2CCN(C(c3ccccc3O)=O)CC2)cnn1C 2584,C1(NC(C2(C)CC3(CC3)C2)=O)CCCC(n2cc(-c3cnccn3)nn2)CC1 2585,C1(NC(CCCC)=O)CN(C(c2c(C)cc(OC(C)=O)cc2F)=O)CCC1(C)C 2586,c1(N(C(C)CCNC(c2ncn3ccccc23)=O)C)ncnc(Cl)c1C#N 2587,C=C(C)CCCC(=O)N1CC(NC(c2c[nH]cc(Cl)c2=O)=O)C(C)C1 2588,CCC1=C(C(=O)NC2COCC2NC(=O)C(C2CCC2)OC)SCCO1 2589,c1(C(=O)NCC2(C(=O)NCC3=CCCC3)CCCO2)ccnc(O)c1 2590,c1(C(=O)OC(Cc2ccc(OC)cc2)C)ccc2cc(OC)ccc2c1 2591,S(=O)(=O)(C1CN(C(=O)CCC(C)O)C1)N1CCN(C(CCSCCCC)=O)CC1 2592,N1(C(Cn2c(C)ccn2)=O)CCC2CCN(C(=O)CCC3CCCCO3)CC12 2593,c1(OC)ccc(F)cc1CC(=O)NC1(CNC(c2ncsc2C2CC2)=O)CCC1 2594,c1(N(CCCC)C)ccnc(C(N2CCC(NC(c3ccc(Cl)s3)=O)CC2)=O)n1 2595,C1(C)(NC(C(CNC(c2cn(C(C)C)nc2)=O)C)=O)CN2CCC1CC2 2596,c1(C(=O)NCCCCCCNC(C(CCC)CCC)=O)c(C)[nH]c2ncccc12 2597,C=CCC(C(=O)N1CC(C(=O)NC2(CO)CCC(C)C2)OC(C)C1)C(C)C 2598,N1(C(CC(COC)C)=O)CCC(F)(CNC(C2(C)CCC(C)C2)=O)CC1 2599,C1(=CCC)CN(C(=O)C(C)NC(=O)C(C)SC)C1 2600,C1(NC(CC2(OC)CCCC2)=O)CCN(C(c2nocc2C(C)(C)C)=O)CC1C 2601,C1(CC)CN(C(C2CCCN2C)=O)CCC1NC(=O)CCc1nccs1 2602,Cn1ccc2c(C(=O)NC3CCN(C(c4coc(O)n4)=O)CC3)[nH]cc2c1=O 2603,C1(CNC(CCCC=C)=O)(OC)CCN(C(c2ccnn2CCF)=O)CC1 2604,C1(Cn2cc(C(C)O)nn2)CN(C(c2csc(-c3ccoc3)n2)=O)CCO1 2605,N1(C(c2cc(CNC(C(CC)(C)CC)=O)on2)=O)CC(C)CC(C)(C)C1 2606,C12(CC1)C(=O)N2.C(CCN(C(=O)CN(C)CC)C(C)C)OCC 2607,N1(C(C2C(c3cn(C)nc3)C2)=O)CCCN(C(=O)CCc2cnc(O)[nH]2)CC1 2608,c1(C(N2CC(O)(CNC(C(CC)C)=O)C2)=O)scc(Br)c1Cl 2609,C1(C)(CC)C=C(C(=O)N2CC(CNC(C3(CS(C)(=O)=O)COC3)=O)C(O)C2)C1 2610,N1(C(C2CC3(CC(C)C3)C2)=O)CCC(C(=O)NC(C)CN(C)C(C)C)=C(F)C1 2611,C1(OCC)CCN(C(=O)C(C)(C)NC(C2CCC(F)C2)=O)CC1 2612,CC(=O)CCCCC(=O)NC1CC=C(C(=O)NCCN(C(C)C)C(C)C)C1 2613,N1(C(c2ncn(C)n2)=O)CC(O)CC1CNC(c1cc(C2CC2)n(C)n1)=O 2614,C1(CNC(C2CC(C)=C(C)CC2)=O)COC(C)(C)CN1C(=O)COCC1CC1 2615,C1(C(=O)OC)CC(C(=O)OC(C)C(=O)Nc2ccccc2F)CC(C(F)(F)F)C1 2616,c1(CC(=O)NCC23CC(C(=O)NC4C(CC)CCCC4)(C2)C3)ncc(F)cc1F 2617,C1(OC(c2ccc(-n3cnnn3)cc2Cl)=O)CCOC2(CCCC2)C1 2618,C12(NC(Cc3nc(C(C)(C)C)sc3)=O)CC1CN(C(C1CCC(C)(C)C1)=O)C2 2619,c1(C(N2CC(C(C(=O)NCc3c(CC)con3)OC)C2)=O)ncncc1C 2620,C(C)(CO)(C(=O)N1CC(C(N)=O)(CNC(c2cnn(C)c2Cl)=O)C1)OC 2621,c1(C(=O)NCCC(=C)CNC(=O)C(C)C(C)CC)cc(C(=O)OC)ccc1C 2622,c1(-c2c(C(=O)NCC(CNC(COCCOC)=O)OC)c[nH]c2)cnn(C)c1C 2623,c1(C(=O)NC(CC)CNC(=O)C(C)(C2CC2)OC)cccc2ccc(O)nc12 2624,C(=O)(CCN=c1cc[nH]cc1S(=O)(=O)N(C)CCN1CCCC1=O)N.CNCC 2625,c1(OC)ccc2c(n1)NC(C(N1CCC(NC(=O)CC(C)C)C(CO)C1)=O)C2 2626,c1(C(=O)NC2(CNC(C3(C)CCC3)=O)CCCCC2)ncc(F)c2ccccc12 2627,N1(C(C(C=CC)O)=O)CC(F)(F)CC1CCNC(=O)Cn1cncc1Cl 2628,Cc1cc(C)c(C(=O)NC2COCCC2NC(c2conc2C)=O)c(O)n1 2629,C(C(=O)NC1CCN(C(C2(C)CCOC2)=O)CC1)(C(F)(F)F)OC(C)=O 2630,CC(C)(C)CCC(C)(C(=O)O)NC(=O)NCc1ccc(N2CCC(O)C2)cc1 2631,CC1(C(=O)NCC2(NC(c3cn(C4CC4)cn3)=O)CCOC2)CCn2ccnc21 2632,C(=O)(C1CCCCc2ccccc21)NCCN(C(=O)C(C)C#N)CC 2633,C1(C(=O)NC2(CN(C(=O)CC3(C)CC3)C)CC2)CN(CC(F)(F)F)CCO1 2634,C(=O)(CC(C)C(=O)O)N1CCCC(n2cc(CC(OCC)OCC)nn2)C1 2635,C(=O)(CC1=CCCC1)NC1CC(C)(NC(=O)CNC(=O)CN(C)C)C1 2636,c1(C(N2C(C)CC(NC(c3cc(F)ccc3O)=O)C2)=O)n[nH]c2c1CN(C)CC2 2637,C1(C(N2CCC(NC(Cc3cc(C)no3)=O)C2C)=O)CC2(CCOCC2)C1 2638,N1(C(C=Cc2c(C)ncs2)=O)CC2CC(NC(c3snc(Cl)c3Cl)=O)CC2C1 2639,C1(CNC(CCNC(=O)OC(C)(C)C)=O)CCN(C(=O)Cc2ccoc2)C1 2640,C(CCC)(C(=O)NCCCN(C(C1CC1c1ccn(C)n1)=O)CC)=CCC 2641,C=C(C)C(C)(O)C(=O)N1CCCC(C)(NC(c2cccc(CC(F)(F)F)c2)=O)C1 2642,N1(CCC=C)CCC2(CN(C(c3nsc4ccccc34)=O)CC(C)O2)C1 2643,C(C(=O)NC1(CO)CC2CC2C1)(C1=CCSC1)N(CCN(C)C)CC 2644,C12(CNC(CSCC(C)C)=O)CCC(CC1NC(c1ccc(O)cc1F)=O)C2 2645,c1(C(=O)NCC2COCC2NC(C2CC2C2CCC2)=O)nccc2[nH]ccc12 2646,C12(CNC(C(CC)NC(C)=O)=O)CC(NC(=O)CC3(O)CCCCC3)(CO1)C2 2647,C(=O)(C1CCCc2nncn21)NC1C(C=C)CN(C(C2(n3cnnn3)CC2)=O)C1 2648,C=C1CCC(NC(=O)NC(Cc2ccccc2)C(=O)N2CCCCC2)CC1 2649,Cc1cc(F)cc(C)c1C(N1CC2CCC1CN2CC1CCS(=O)(=O)CC1)=O 2650,c1(CC(N2C(CC)C(NC(=O)C(C)CSC)CC2)=O)ccc(C)cc1C 2651,N1(C(CNS(CC)(=O)=O)=O)CC(C)(NC(=O)CC(C2CCC2)C2CCC2)C1 2652,CC1(C)OCc2c1n[nH]c2C(=O)NCC1(C)CCN(C(=O)C=C2CCCCC2)C1 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2816,N1(CC)C(=S)NC(c2cccnc2)C(CC(F)(F)F)(C2CC2)CCCCC1=O 2817,C(=O)(C(C)(C)CS(N)(=O)=O)NC1CCN(C(C2(Oc3cn(C)nc3)CC2)=O)C1 2818,CC1NC(=O)CCC1CNC(=O)CC1CCN(C(C2CC(=C3CC3)C2)=O)C1 2819,N1(C(c2c(OC)cc(Cl)cc2)=O)CCn2nnc(C(=O)NC3CCOC3)c2C1 2820,CC#CCCCC(=O)N1CCC(O)C(NC(C2CCCC(C)(C)C2)=O)C1 2821,CC(C)C(CO)C(=O)N(C(CNC(c1cnn(C2CC2)c1)=O)C1CC1)C 2822,C1(C(=O)NCC2(SC)CCC2)CN(C(=O)CCc2ccoc2)CCO1 2823,c1(CN2CC(CC(=O)Nc3nc(C(C)(C)C)[nH]n3)OCC2)cccc([N+](=O)[O-])c1 2824,C1(O)(CCNC(c2ccccc2Cn2cnnn2)=O)CCCN(C(=O)C2CC2)C1 2825,c1(C(=O)NC2CCC(NC(c3c(Cl)ncc(C)c3)=O)C2)ccc2nc(O)[nH]c2c1 2826,C1(CN(C)C(C2CC3(CC3)C2)=O)CCCN(C(c2snnc2C2CCC2)=O)C1 2827,N1(C(CCc2c(C(=O)O)c(F)ccc2)=O)CCC2(CC1)CC2CO 2828,Cc1cccc(CC(c2ncc[nH]2)NC(=O)N(C)Cc2ccccc2C)c1 2829,C1(C(=O)NC(COC)C(=O)OC)CN(C(=O)NC(C)(C)C)CC12CC2 2830,Cc1nn(CC(N2CC(NC(C34CCCC3(C(N)=O)C4)=O)CC2CO)=O)c(=O)o1 2831,c1(C(=O)NCCN(C(=O)C(c2cncnc2)C)CC)ccc(C)c(C#N)c1 2832,CC(C(=O)N1OC2C=CC1CC2)C1CCN(C(C2CC(C)(C)CO2)=O)C1 2833,c1(-c2cc(Cl)cc(Cl)c2)nc(-c2nc[nH]n2)nn1C1CCCc2ccccc21 2834,c1(CC)c(C(N2CCC(CF)(NC(c3oncc3C)=O)C2)=O)cccc1C 2835,c1(SCC(N2CCOC(Cc3ccc(Cl)cc3)C2)=O)ccccc1F 2836,C1(CNC(c2ccc(C#C)cc2)=O)CN(C(c2cnn(C)c2F)=O)CC(C)(C)O1 2837,CCCCC(C(=O)N1CCN(C(=O)CCOC)C(C2CC2)C1)COC 2838,N1(C(C(CC)COC)=O)CCOC2CN(C(=O)C(C)Cn3ccnc3)CC12 2839,N1(C(C)C)Cc2cccc(NC(C3CCCCC3C(N)=O)=O)c2C1 2840,c1(C(=O)NC(C(CO)NC(c2csc(C)c2C)=O)C)ncc(F)c2ccccc12 2841,N1(C(CNC(C)=O)=O)CCCC2C1CCN2C(c1snc(O)c1Cl)=O 2842,C1(C(=O)NC(CCNC(C(N2CC(C)C2)C)=O)(C)C)CCC(F)(F)C1 2843,CCCC(CCC)=CC(N1CCN(CC(=O)N(C2CCOC(C)C2)C)CC1)=O 2844,FC1(F)CCC2C(CNc3cccc(OC4CC4)c3)C12 2845,N1(C(C(COCC)(C)C)=O)CCCC(C)(c2cn(-c3ccc(Cl)cc3F)nn2)C1 2846,CCC(CC(=O)N(C(C)C(C)C(=O)NCCOCCC(C)C)C)CC(C)C 2847,c1(NC2(CNC(C3CCCC(F)(F)C3)=O)CCC2)ncc(Br)c(O)n1 2848,N1(C(C2CN(CC)C(=O)C2)C(=O)NCCC2CCOCC2)CC(CO)C2(CC2)C1 2849,N1(C(C(c2cnccn2)C)=O)CCC(O)(CCNC(C2(C)CC2)=O)C1 2850,C(c1cccnc1)=CC(=O)NC(CNC(C1CCN1C1CCCC1)=O)CO 2851,Cc1ccc(CCC(=O)N(CC(C)NC(c2c(C)ccn2C)=O)C)c(Br)c1 2852,C1(CNC(c2n(CCOC)ccc2)=O)CCCCN1C(=O)Cc1cnccc1C 2853,N1(C(CCS(N)(=O)=O)=O)CCOCC2(COCCN2C(c2cccnc2Cl)=O)C1 2854,c1(CNCC2(NC(CC3C(C)=NNC3=O)=O)CCCCCC2)cc(C)c(F)cc1N 2855,N1(C(C(=O)NCC=C)CCC)CCC(N2CCOC2=O)CC1.c1(C(C)S)ccccc1 2856,c12ccc(Cl)c(c1)C(=O)N2.N(C(=N)N)C(C)C 2857,c1(SC)nc(C(F)F)cc(=NC(CNC(c2ncccc2Cl)=O)C2CC2)[nH]1 2858,c1(C(N2CCC(N(C(c3cc(=O)cc[nH]3)=O)CC)C2)=O)c(C)ccc(F)c1O 2859,c1(C(=O)OC)cnc2c(c1)N(C(=O)CC(C)(C(=O)O)OC)CCO2 2860,C1(COC)(CNC(=O)CCCCCN(C)C)CCN(C(=O)CCCCSC)CC1 2861,C1(NC(COC(C)=O)=O)CN(C(=O)CC2CCC(=O)N2)C2(CCC2)C1 2862,C1(C(N(C2CCCN(C(C3CCC(=O)N3C)=O)C2)CC)=O)CCC(=C(F)F)CC1 2863,CCCC(CCCNC(c1scc(C)c1Cl)=O)NC(c1ccn(C2CCC2)n1)=O 2864,c1(C(=O)NC(COCCCNC(C(CC#C)O)=O)(C)C)cc(C)n(C)c1C 2865,N(C1CCCn2nccc21)C(C(C)(C)CCCNC(=O)CCN1CCCC1=O)=O 2866,c1(C(=O)NCC(CNC(Cc2ncc(C)o2)=O)(C)F)ccc(F)c(C)c1C 2867,C1(CNC(C=Cc2n(CC)ncc2)=O)C2CCCC1N(C(c1cnn[nH]1)=O)C2 2868,N1(C(Cc2cc(C)nn2C)=O)CCC2CCCC12CNC(c1cnc(C)nn1)=O 2869,C1(C(=O)NCC#CCC)CC2(CCC2)CN1C(c1cc(F)ccc1C)=O 2870,c1(C(=O)NCC(C)CNC(=O)CCCN(C)C)ccc(OC(F)F)cn1 2871,C(C(CNC(c1cnn(Cc2ccc(Cl)cc2)c1)=O)C(F)(F)F)NC(C)=O 2872,C12(NC3CCN(C4CN(C(=O)OC(C)(C)C)C4)C3=O)CCCC1C2(F)F 2873,C1(C(=O)NC2CCCC(F)(F)C2)Cc2cc(O)ccc2CN1S(=O)(=O)CCCl 2874,c1(C(=O)NC(C)CCN(C)C(C2CC2C2CCC2)=O)ccc2c(c1)C=CS2(=O)=O 2875,Cc1cc(=NCCCO)[nH]c(=NCC2CN(C(=O)NN3CC(C)CC(C)C3)C2)[nH]1 2876,C(N=c1cc(C(C)=O)c([N+](=O)[O-])c[nH]1)C1C(C)CCN(C(C(CC)(F)F)=O)C1 2877,C1(C)(C(N(C)CC2CCN(C(CCC(=C)Br)=O)CC2)=O)CC(OC)CN1C 2878,C(=O)(C1=CCCCC1P(C)(C)=O)NCC1N(C(CCCCCC)=O)CC(F)(F)C1 2879,CCCCC(CC)C(=O)NCCCN(CC(=O)N(C)CC1(C)CC1)C 2880,C1(CNC(c2cnc(C3CC3)s2)=O)CC2CCCC2N1C(=O)CN1CC2CC2C1 2881,C1(C#N)(C(=O)NCCCN(C(=O)CC2CCC2(C)C)C(C)C)CC1(C)C 2882,C#CC1CN(C(=O)CCCN(C)C)CC1OCC 2883,c1(C(=O)NC2C3CN(C(C=C(C)C(F)F)=O)C2C3)ccc(F)cc1C(F)(F)F 2884,c1(CNC(C2(c3c(C)c[nH]n3)CC2)=O)cc(O)nc(CNC(=O)CCC2CC2)n1 2885,C(=O)(CC1=NNC(=O)C1)NCC1OCCCN(C(CC2CC(C)OC2C)=O)C1 2886,C1(C)(C(N(CCN(C(C)C)C(C2CCC(F)(F)C2)=O)C)=O)CCCN1C 2887,CC(C)CC(C)CC(=O)NCC12CCCCC(N)(C1)C2 2888,CC(CCCCCO)NC(=O)C=CC(C)(C)NC(C1CC(=O)OC1(C)C)=O 2889,N1(C(=O)NCc2cc(CC)on2)CCC2COC(=O)C12 2890,C12(CNC(CS(CC)=O)=O)CCC(NC(c3nccc4ccsc34)=O)(CC1)CO2 2891,c1(CC(N2CC(C)C(NC(C3CC3C#N)=O)CC2)=O)ccc2c(c1)CCN2C 2892,C1(CC)CN(C(=O)OC(C)(C)C)CCN1C.C12CC(CCN1CC)OC2=O 2893,C(=O)(CC(CC)CC)NC(C(=O)NC(CCCCC)C)COC 2894,Cn1c(=O)c2ccc(NC(=O)NCC3(CCCO)CC3)cc2n(C)c1=O 2895,N1(C(C=CCC)=O)CCC(NC(C2(C)CCCC2(F)F)=O)C(O)C1 2896,N1(C(c2cc(C)sc2C)C(=O)NCCN2CCOCC2)CC2COCC2(C)C1 2897,C12COCCN(C1)C(=O)C1CC1C(=O)N2.c1(C(=O)OCC)c[nH]n(C(C)C)c1=N 2898,CC1CC(CNC(C2CN(C3COC3)C2)=O)CN1C(=O)CCCCN(C)C 2899,C1(CC#C)(C(=O)NCCC#CCO)CCN(C(=O)C(CC)n2cncn2)C1 2900,C(=O)(C1=NOC(CNC(=O)C(CC)CCC)C1)NCCC=CC=C 2901,CC1=C(C(=O)NC2CN(C(C3(C(F)F)CCCC3)=O)CC3CC23)CCO1 2902,c1(C(=O)NCC=CCNC(c2ccc(CC)s2)=O)cnn(CC2CCOC2)c1C 2903,c1(C(=O)OCC)[nH]c(C)c(C(=O)NCc2conc2C(C)C)c1CC 2904,C1(C(N2C(C(C(=O)NCCC(C=C)C)(C)C)CCC2)=O)CC12CCOCC2 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2923,c1(C(=O)NC2C(CNC(CCCNS(C)(=O)=O)=O)C2)c[nH]c2cc(F)ccc12 2924,c1(NC(c2cc(OC)c(-c3cccnc3O)cn2)=O)nccc2occc12 2925,C1(C(=O)NC(c2cccc(Cl)c2)Cc2cn(CCOC)nn2)CC(F)C(=O)N1 2926,C1(CC=C)(NC(=O)CCOCCOC)CCN(C(=O)CCc2cscn2)CC1 2927,c1(CC)nc(C)c(C(=O)NCC2(C(N)=O)CN(C(=O)C(Cl)=CCl)C2)s1 2928,C1(C(=O)NCCNC(c2cc3sccc3[nH]2)=O)Cc2ccccc2C(=O)O1 2929,c1(OC)nc(Cl)ccc1C(=O)NCC1CCC1NC(=O)COc1ccc(F)cc1 2930,c1(CC)cc(C(=O)NCC2CCCN2C(=O)Cn2cc(C)cn2)cc(N)c1 2931,C1(NC(=O)CN2CCC2=O)CC12CCN(Cc1cn[nH]c1)CC2 2932,n1(CC(=O)NC2CCCC(NC(c3oc(CC)c(C)c3)=O)C2)nc(O)ccc1=O 2933,C1(NC(CCC=C(C)C)=O)CCOC(C(=O)NCCc2c[nH]nc2O)C1 2934,CCC(CCC(=O)N(CC(N1CCN(C(=O)Cc2cccnc2)CC1)=O)C)OC 2935,N1(C(CCC#CC)=O)CCC(C(=O)NCc2ncccc2Cl)C(C)C1 2936,N1(C(C2(NC(Cc3scc(C)c3)=O)CCN(C)C2)=O)CCC2C(=O)NCC2C1 2937,c1(CC(N2C(CCCNC(C3(C)CC(=C)C3)=O)CCC2)=O)cccc2sccc12 2938,C(C(C)(O)CC(=O)NC1CCCCN(C(=O)CC2CCSCC2)C1)OC 2939,c1(C(N2CCC(N(C(c3c(CC)c[nH]c3)=O)C)C(C)C2)=O)cc2ccccn2c1 2940,C(=O)(C#CC(=O)N(C)C)NCC(C)CN(C(=O)C(C)(C)NC(=O)C(F)(F)F)C 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2959,c1(CC(=O)NCC2CCN(CC(=O)Nc3cccc(Cl)c3)C2)ccc([N+](=O)[O-])cc1 2960,C12CN(CCN1C(=O)OC(C)(C)C)C2=O.c1(CCC(=O)NC)cnc(C2CC2)o1 2961,c1(C(=O)NC(C(N2CCCC(CN(C)C)C2)=O)C2CCCC2)cc(O)nc(O)n1 2962,CC1(NC(=O)CN2CCCC2)CCN(C(c2sccc2C2CC2)=O)CC1 2963,c12ccc(cc1)NCC2N(C)C.c1(C(=O)OCC=C)ncnn1CC 2964,C(=O)(C(C)(C)CC(=O)NC(c1ccc(F)cc1)CNC(=O)COCCF)OC 2965,C(c1ccc([N+](=O)[O-])s1)=CC(N1CCN(C(CCC(C)C)=O)CC1CCO)=O 2966,C1(=O)CCC(=O)N2CC3C(C3C2)N1.N1(CCC)CCOC(C)C1 2967,c1(C(=O)OC)c(C)[nH]c(C(N2CC(C)(NC(=O)CNS(N)(=O)=O)C2)=O)c1C 2968,C(=O)(C(C)(C)Cn1cc(C2(C)CN(C(=O)CC=C(Cl)Cl)C2)nn1)OCC 2969,C(CCCCC(=O)N1CC(OC(F)F)C1)n1cc(COCCN)nn1 2970,C(CCC(=O)NC(C)CC(C)NC(c1ocnc1-c1ccccc1)=O)OCCC 2971,C12(C(N3CCC(N(CC#C)C(C4CCC5CC5C4)=O)CC3)=O)CCOC(C)(C1)C2 2972,N1(C(C(=C(C)C2CC2)F)=O)CC(NC(=O)Cn2nc(C)c(Br)c2C)CC(F)C1 2973,C1(COC)(NC(c2sccc2CN(C)C)=O)CN(C(=O)CCCC2CCC2)C1 2974,c1(NC(N2CCC(C(N)=O)CC2)=O)cc(C(F)(F)F)cnc1O 2975,N1(C(=O)C=CCF)CC2CCCC(C1)N(C(=O)Cc1ccsn1)C2 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2994,c1(C(=O)NCC2N(C(CC3C(C)(C)CCO3)=O)CCOC2)cccc2nsnc12 2995,Cc1cc(C(=O)NCC23CC(CN2C(C2CC=CCC2)=O)C3)nn1C(C)C1CC1 2996,Cc1nn(C)c(NNC(=O)Nc2nccc(C(F)(F)F)n2)c1C#N 2997,c1(C(N2CC(C(=O)OC)CC(O)C2)C(=O)NCCC)ccc(F)c2ccccc12 2998,Cc1ccc(C(=O)NCCCN(CCCNC(=O)C(C)n2ccnn2)C)cc1 2999,c1(C(c2n(CC)nnn2)NCc2ccn(C(C)(C)C)c2)ccc(C(F)F)cn1 3000,C(CCC[Si](C)(C)C)N(C(Cc1ccccc1)C(=O)NC1CC1)C 3001,n1(C(C)C)ccc(C(=O)N(C(C)CNC(C2CC2(C)C(F)F)=O)C)n1 3002,C#CCCCCC(=O)NCC12CCC(C1)N(C(c1ccc(C3CCC3)nc1)=O)C2 3003,c1(-c2ccnc(NC(C3CCN3c3cnncc3Br)=O)n2)cccc([N+](=O)[O-])c1 3004,c1(C(N(CCCNC(C=CC)=O)C)=O)cc2cccc(O)c2[nH]1 3005,c1(CC)cc(F)ccc1C(=O)NCC1CN(C(C2CC3C(C2)C3(F)F)=O)CCO1 3006,N1(C(=O)NCc2cnsn2)CCC2(CCOCC2C(N2CCOCC2)=O)CC1 3007,C1(NC(C#CC(C)(C)O)=O)CC2CC1CN(C(=O)CCC(C)(C)N1CCCC1)C2 3008,Cc1ncnc(N2CCC(C)(CNC(=O)Cn3nnnc3C3CC3)CC2)c1Br 3009,C(C1CCCN1C(c1csc(Cl)c1)=O)=CC(=O)N(CCSC)C 3010,C1(NC(c2c(CC)ccs2)=O)CC2CN(C(c3c(C)noc3CC)=O)CC2C1 3011,C1(C(=O)NC(C(C)O)(C)C)CCCCCC1NC(=O)CC1OCCO1 3012,c1(C(N2C(CCNC(COc3cc(C)on3)=O)CCCC2)=O)ccc(N)cc1C 3013,n1(CC(=O)N(c2ccccc2)CC)cc(-c2ccncc2)nn1.C1C(=O)N1.C1CO1 3014,Cn1cc(C2OCCC2C(=O)NC2CCC2NC(c2cc(C3CC3)on2)=O)cn1 3015,N1(C(=O)NCC(c2ccc(CC)cc2)O)CC=C(c2cccc(Cl)c2)CC1 3016,C(=O)(CCCC(=O)N1CC2CC2(NC(C2CCC3CCC2O3)=O)C1)OC(C)(C)C 3017,CN=c1ncc(-c2cnc(C(N3CCN(Cc4ccc(OC)s4)CC3)=O)nc2)c[nH]1 3018,C1(C(C)NC(C2(C(=O)NC)CCC2)=O)CCCN(C(c2sc(C)cc2Cl)=O)C1 3019,Cc1c[nH]cc1C(=O)NCCC(O)CNC(c1cnn(Cc2ccccc2)c1)=O 3020,c1(CC)[nH]nc(C(N2CC(OCCNC(=O)C(C3CCCO3)OC)C2)=O)c1Cl 3021,Cc1nc2c(cc1C(=O)NCCC1COCCN1C(=O)C=C1CC1)c(C)nn2C 3022,C1(C(N(CCN(C(Cc2cc(CC)no2)=O)C)C)=O)CC12CCC(=O)CC2 3023,Cc1ccc(C(N2CCC(C)N(C(=O)CS(N)(=O)=O)CC2)=O)c(N)c1Br 3024,C(C(=O)NC1(C2CCCN2C(c2nccnc2N)=O)CC1)(C(C)C)SCC 3025,C(=O)(C(O)CC(C)(C)C)N(CC(CNC(CC(C)(C)OC)=O)C)C 3026,CCCCC(O)C(C)C(=O)NC(C)C=CC(=O)NCCC(C)C(F)F 3027,c1(OC)c(F)cc(C(=O)NCC2CN(C(C3CN(C)CCO3)=O)CC2C)cc1Cl 3028,N1(C(c2cc(Br)cc(C)n2)C(=O)NC(C(=O)OC)C)CC(C)(C)C12CCOCC2 3029,C#CCCC(O)C(=O)NC(C)CCNC(c1snnc1CC)=O 3030,C1(C(N2CCCC(NC(CCc3ncc(C)[nH]3)=O)C2C)=O)CS(=O)(=O)CC(=O)N1 3031,C(=O)(CCCCC#N)NCC1N(C(COCC(=C)C)=O)CC(O)C1 3032,N1(C(CC)C(C)C)CC2COCC2(C(=O)NC2CCC(C(=O)OC)C2)C1 3033,CCCC(CCCS(C)(=O)=O)C(=O)NCC1(C)COCCN(C(C2COC2)=O)C1 3034,N1(C(C(C(CC)C)N(C(=O)CCN2CCCCC2)C)=O)CCN2CC(O)CC2C1 3035,N1(C(c2c(C)coc2)=O)CC2CN(C(=O)C=CC(C)C)CCC2(CO)C1 3036,C1(C(N2CC(CC(C)NC(=O)C(c3ccn(C)n3)C)C2)=O)OC2CCC1CC2 3037,CC1C(C)C(C)CN1C(=O)C(=O)Nc1ccc(OCC(=O)N(C)C)cc1 3038,CCC(CCC(=O)NCc1cn(C)nc1C)NC(=O)Cc1ccon1 3039,Cc1cc(=NC(=O)C(C)C(C)NC(c2cc(C3CC3)no2)=O)[nH]n1C 3040,c1(N2CC(C(=O)OC)(CNC(C3CN(C(C)=O)CCO3)=O)C2)ncc(C)cn1 3041,CC(C)CC(F)C(=O)NC1CCCN(C(=O)CCN(C)C(=O)OC(C)(C)C)C1 3042,C(CC(C)C)(C(=O)NC1C(C)C1C)ON(C(COC(CC)CC)=O)C 3043,c1(C(=O)NCC2CC(F)(CNC(CCOCCOCC)=O)C2)cc(O)nc(O)n1 3044,c1(C(=O)NCCN(C(CCCn2c(C)ncc2)=O)CC(C)O)c[nH]c(=S)cn1 3045,CCCC(C)CC(=O)N(CCCC(=O)NCCOC1CCOC1)C 3046,c1(C(C=CC(=O)N(C2CCC(C)C2)C)=O)ccc(C(F)F)cc1 3047,C(=O)(CC1OCc2ccccc21)N(CCNC(C(=O)NCC)=O)CCSC 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3066,C(C(O)CN=c1[nH]c(C2CCCC2)nc(=N)[nH]1)NC(C=C(CCC)CCC)=O 3067,C(N=c1[nH]nc(-c2cccnc2)s1)C1CCC(NC(c2cc(C)ncc2)=O)C1 3068,c1(N2CC(CNC(Cc3cccc(C)c3C)=O)OCCC2)nc2cccc(C)c2o1 3069,Cc1nn(CC(=O)NCC2CCC2NC(=O)CC=CC(C)(C)C)c(C)c1C=NO 3070,N1(C(Cn2c(C(=O)OC)cc(C)n2)=O)CCC(F)C(NC(c2sccc2Cl)=O)C1 3071,CC1CCN(C(c2cncnc2)=O)CC1N(C)C(C1CCCCCC1)=O 3072,N1(C(CCCCCOCC)=O)CCC2CCN(C(=O)C(C(C)C)C(C)C)CC12 3073,C(=O)(C(C)(C)CN(C)C(C1COCC(C)O1)=O)N(CC(CC)OC)C 3074,c1(N2C(CO)CN(Cc3ccncc3Br)CC2)ncnc2ccc(F)cc12 3075,c1(C(=O)NCC(CNC(=O)C=CCO)O)cc(Cl)cc2c1CCC2 3076,Cc1cccc(C(N2CCC(CNC(=O)CCCF)C2(C)C)=O)c1C 3077,c1(N2CCC(N(C)Cc3cccc(C)c3)C2)ncnc2oc(C)nc12 3078,C1(CNC(c2cc(O)ncn2)=O)CN(C(C2C(F)(F)C23CC3)=O)CCCO1 3079,c1(C(=O)NC(CNC(CCCCC)=O)CC(C)C)cc(C2CC2)ccc1F 3080,C(C(CC(C)C)C(=O)NC1CC(=O)N(C(C)C)C1)NC(C1=CC(C)(CC)C1)=O 3081,C1(CC(C)NC(=O)CSC(F)F)CCN(C(=O)COc2ccc(C(N)=O)cc2)CC1 3082,c1(C(=O)NC2CC(N(C(C=CSC)=O)C)C2)ccc(NC(=O)N(C)C)cc1 3083,N1(C(C2C(CC(C)C)C2)=O)CCCC1CN(C)C(C1(CCCO)CCCC1)=O 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3102,C1(NC(C(C2CCCC2)OC)=O)CCNC1(C)C 3103,c1(N2C(CNC(C3N(C(C)C)CCC3)=O)C(C)CC2)nc(Cl)ncc1C(F)(F)F 3104,N1(C(CC(=C)C)=O)CC2CC(C1)C2NC(c1sc(Cl)cc1Cl)=O 3105,C1(CNC(CCCC)=O)C(C)CCCN1C(c1ccc(CC(C)C)nc1)=O 3106,c1(C(=O)NC2CCCC(CNC(c3cnsn3)=O)C2)ccc2c(c1)CCCS2 3107,N1(C(c2c(SCC)cccc2)=O)CCCC2C1CCCN2C(=O)Cc1ccco1 3108,C1(CC2CCC2)CCC(C)(C)OC1.c12ccccc1-n1cc(nn1)C1CN(C1)C2=O.CO 3109,c1(C(=O)NC2CCN(C(CCCC(=C)C)=O)C2(C)C)ccc2cnnn2c1 3110,n1(CCO)c(CN2CCCSCC2C2CCCC2)nc2ccccc12 3111,C1(NC(c2scc(C)c2)=O)CCN(C(=O)Cc2cnn(C)c2C)CCC1CO 3112,N#Cc1cc(C(N2CC(NC(=O)C3CC3)C(C=C(F)F)C2)=O)cc(F)c1F 3113,N1(C(C=C(C)CNC(=O)Cc2scnc2C)=O)CCCC1CC(C)C 3114,CN1CC(NC(C2CN(C(=O)CN3CCNC3=O)CC23CC3)=O)CCC1=O 3115,C1(NC(C(c2ccc(Cl)cc2)C)=O)CN(C(=O)C(c2cccnc2)=O)CC12CC2 3116,CCC(C)(C)C(C)CC(=O)NCCC1CC(NC(c2ncc3[nH]ncc3n2)=O)C1 3117,CCCC(C)C(=O)N1CCCC1Cn1cc(CNC(=O)CSC(F)(F)F)nn1 3118,c1(OCC)cc(Cn2cc(-c3ccccc3C#N)nn2)ccc1Cl 3119,C1(NC(C2CC(C(C)C)C2)=O)CC2CCC(C1)N2C(=O)CSCCN(C)C 3120,c1(C(=O)NC(C)CC(C)NC(=O)C=CC=C(Cl)Cl)ccc(-c2cnnn2C)cc1 3121,N1(C(C=C2CCN(C(=O)Cc3ccccn3)CC2)=O)CC2COCC2(CO)C1 3122,C1(NC(C(C)C2(O)CCC2)=O)COCCC1C(=O)NOCC1CCOCC1 3123,C1(C(N(CC(CCC)O)C)=O)CC(OC)CN1C(=O)CC1CC2(CCC2)C1 3124,C1(C(=O)NC2(C)CC(=C)C2)CCN(C(C2CCCCCN2C)=O)C(C)(C)C1 3125,C(=O)(C(=O)CC(C)CC)NCCCC(N1CCCC(CC=CC)C1)=O 3126,C(=O)(C(C)CC(C)CC(C)C)NCC1(F)CC(NC(c2nnn(CC)c2C)=O)C1 3127,c1(C(N2CC3C(CNC(C4CCC(CC)O4)=O)(C3)C2)=O)ccc2c(c1)nnn2C 3128,C1(C(N2CCC(CNC(C3(C(=O)NC)CC3)=O)C2)=O)CCCC(NC(=O)NC)C1 3129,C1(CC)CN(C(C2CC2c2ccccc2)=O)CC1Cc1ccccc1.C(C(C)C)OC 3130,C1(C(N2CC(C)C2C(=O)NCCc2cn(C)nn2)=O)CC12CCCCC2 3131,N1(CC(=O)NC2CC2)CCC(N(C(C2CC23CCOC3)=O)Cc2nncs2)CC1 3132,Cc1ncc(NC(=O)C(CC2CC2)NC(=O)C(C2(O)CCCC2)F)c(C)c1C 3133,C1(OC)CC2C1CCN2C(C12CCC(CC1NC(=O)CCC1CC1(F)F)C2)=O 3134,c1(CC)cc(C(=O)NC(C)C(C)NC(=O)C(F)C2CCCC2)ccc1O 3135,C(=O)(C(F)C(C)CNC(C1CCS(=O)CC1)=O)NCc1c(OC)nn(C)c1 3136,C12(C(=O)NCc3cnc(C)o3)CC1CN(C(C1CCO1)=O)C2 3137,c1(CC(=O)NC2C(CNC(CNC(C)=O)=O)C2)cncs1 3138,Cc1nc2cc(NC(=O)C(C(C)(C)C)NC(N)=O)cnc2[nH]1 3139,C(CNC(=O)C(F)(F)C(F)F)(CC(F)(F)F)NC(C1CN(S(CC)(=O)=O)C1)=O 3140,C1(NC2(c3cc(OC)c(C)cc3)CCCCC2)CCN2CCCC2C1 3141,N1(C(=O)OC(C)(C)C)CCc2ccccc2C1CC(=O)OCC(F)F 3142,C1(C(=O)NC(C(N2CC(C)=C(C)C2)=O)CCN(C)C)CC2(CC(=O)C2)C1 3143,C1(C(C)CO)CCCN(C(=O)NC(=O)CCn2cc(CC3(C#N)CC3)nn2)C1 3144,C1(c2n(CCC)nc(-c3cc(OC)ccn3)n2)CCn2c(C)cnc2C1 3145,C(=O)(CCCCCc1cn(C(C)CN2CCCC2)nn1)Nc1cc(C)nn1C 3146,Cc1ccc(CCC(N2CCC(C)N(C(=O)C=CC(N)=O)CC2)=O)cc1[N+](=O)[O-] 3147,N1(C(CSCCC)=O)CC(NC(C2C=CC=CC=C2)=O)C(c2cncn2C)C1 3148,C1(C#N)(NC(C(C)C)=O)CCN(C(=O)CN2C(=O)CSC2=S)C1 3149,CCCC(C(=O)N1CC(C)(NC(c2nccn3ccnc23)=O)C1)C(C)C 3150,CC1(NC(c2cnc(Br)s2)=O)CCN(C(C2(O)CCC2)=O)C1 3151,CC(C)(C#N)CCCC(=O)NC1C2CN(C(c3n[nH]cc3C(F)(F)F)=O)CC12 3152,c1(CC)cc(C(N2CC(F)CC2CN(C(=O)C2=CCCS2)C)=O)sc1C 3153,c1(OC)ccc(Br)cc1C(c1nnnn1Cc1ccco1)NCCc1ccns1 3154,c1(CCC(C)NC(=O)C=CCN2CCC2)ccccc1[N+](=O)[O-] 3155,C1(CC(N2C(C(=O)NCC=C3CCSCC3)CC2)=O)CC2(CCC2)C1 3156,c1(C(=O)NCC#CCNC(C(C)C2CCC2)=O)cc(C(F)(F)F)cc(O)n1 3157,c1(C(N2CCCCC2c2n[nH]c(C(C)C)n2)C(=O)NCC(C)C)nc(Br)nn1C 3158,C1(CCC)CN(C(=O)Cn2nc(C)nc2C)CCN1C(=O)C1=C(Cl)CCC1 3159,N1(C(C2N(C(C3CC3c3ccc(Br)cc3)=O)CCC2)=O)CCN2CC(O)CC2C1 3160,C1(NC(C2CN(CC(C)C)C2)=O)CCC(CNC(=O)C=Cc2ncc[nH]2)C1 3161,C(=O)(C(C)(C)C(C)C)N(C)CC1CCN(C(CCOCCCOC)=O)C1 3162,C1(NC(CC(C)N(C)C)=O)CC(C(=O)NCC2=CCCC2)C1(C)C 3163,C1(C(=O)NC2CC(COC)C2)C(C)OCCN1C(c1cc(O)nn1C)=O 3164,C(=O)(C1=NN(C)C(=O)CC1)NC1(c2c(F)ccc(-c3ccc(OC)cn3)c2)CC1 3165,C(=O)(CCCCCF)NCCN(CCOC)C(C1CC1C1CCCC1)=O 3166,CCCC(C)(O)CC(=O)NC1(C)CCCCC1C(N1CC=CC1CF)=O 3167,CC(CNC(c1cscc1Cl)=O)C(F)C(=O)NC1(CO)CC1 3168,N1(C(c2cnc(OC)s2)=O)CC2(CCC2NC(=O)C(O)Cc2cn(C)cn2)C1 3169,CCC(CC)(CCNC(C1CC1[N+](=O)[O-])=O)NC(=O)C(C)Cc1cnco1 3170,c1(OC)cccc(-c2cn(C3CN(C(C4(C)CC=CCC4)=O)CC3O)nn2)c1Cl 3171,C1(CNC(C)=O)CCCN1C(=O)CCOC1CN(C(=O)CC(C)F)C1 3172,N1(C(C(C)OC)=O)CCN(C(=O)C(C)CN(C)C)C(C2CCCC2)C1 3173,N1(C(C(C)OC2CCOC2)=O)CC(CNC(=O)CCC2CCCOC2)C(F)(F)C1 3174,N1(C(C(F)=C(C)C)=O)CCC2(CCCC2NC(c2cc(C)sc2C)=O)C1 3175,C1(C(C)NC(c2c(C(C)C)c[nH]n2)=O)CN(C(=O)CCCC2CC2)CCO1 3176,C1(C(=O)NC2C(CNC(c3c(C)[nH]cc3)=O)COC2)CCn2cncc2C1 3177,N1(C(CCNC(=O)NC)=O)CCCN(C(=O)C(C#N)C(C)(C)C)C(C)C1 3178,CC(C)C(O)C(F)(F)C(=O)NCCc1ocnc1CNC(C1Cc2nncn2C1)=O 3179,c1(CCC)ncc(NC(=O)C(CCC2CC2)NC(=O)Cn2cccn2)cn1 3180,c1(-c2n(C(C)C)ncc2)cccc2c1nnn2C 3181,c1(CC)ncsc1C(=O)NCC1(CNC(=O)CC2CCCC2C)CC1 3182,Cc1cccc2[nH]c(C(N3CCC=C(CNC(C4COC(=O)N4)=O)C3)=O)cc12 3183,C(c1cn(C)nn1)=CC(=O)NC(C(=O)N(CCCC(=O)NC)C)Cc1cc[nH]n1 3184,C(=O)(N=S(C)(=O)c1cccc2cccnc12)c1c(N(CCN(C)C)C)nccc1 3185,C1(C(C)C)CN(C(=O)Cn2cnc(C(N)=O)n2)CCN1C(C1CCCCC1O)=O 3186,N1(C(C2C3CCCC(=O)C32)=O)CC2CCCN(C(C34CC(C3)C4)=O)C2C1 3187,c1(NC(COc2cn(C)nc2)=O)ccc(NC(C2(C)CC2C(F)(F)F)=O)cc1 3188,c1(NC(C(C)OC(c2cncnc2)=O)=O)nccc2ccn(C)c12 3189,N1(C(CCC(CC)C)=O)CCC2(CC1)CC(NC(C1CCNC(=O)C1)=O)C2 3190,Cc1cc(C(N2CCC(C)(C#N)C2)C(=O)NC(C)(C)C)cc(Br)c1 3191,N1(C(C(C)SCC)=O)CCCCC(NC(=O)C=C2CCC(C)CC2)C1 3192,C1(C)(CNC(CN2C(C)CC2)=O)CCN(C(=O)C(C(C)(C)C)C2CCC2)CC1 3193,C#Cc1cncc(C(N2CC(C(C)NC(C3CCS(=O)(=O)C3)=O)C2)=O)c1 3194,n1(CC)nncc1C(=O)NCC1CC(NC(=O)C(F)(F)c2ncccn2)C1 3195,c1(CNC(C2(C3N(C(CC)=O)CCC3)CC2)=O)ccnc(N2CCCC2)n1 3196,c1(C(NNC(C(C)n2cc(CO)nn2)=O)=O)cc(S(=O)(=O)NC2CC2)ccc1Cl 3197,C1(C(N(CC(F)F)CCOC)=O)CSCN1C(c1cc(OC)no1)=O 3198,CCC(CC(=O)NC12CC(NC(c3ccnn(C)c3=O)=O)(C1)C2)C(C)C 3199,c1(C(=O)NC2CC(CNC(C3CC(C#C)(O)C3)=O)C2)ccc2ncc(=O)[nH]c2c1 3200,c1(OC)cccc2c1CC(C(N1CCOC(CNCc3ccccc3)C1)=O)CO2 3201,C1(C(N2CCC(NC(=O)C3=CCCCO3)C(CO)C2)=O)CC2CCC(C1)S2(=O)=O 3202,N1(C(c2ccc(-n3c(C)ccn3)cc2)=O)CC2CCC(C1)N2C(C1CC1(Cl)Cl)=O 3203,CCCCCCCCC(=O)N(CC(C)N(C(=O)CC(C)(C)C1CC1)C)C 3204,C1(NC(C(CSC)O)=O)CC2CCC1CN(C(c1cc(Br)cs1)=O)C2 3205,N1(C(c2cscn2)=O)CCC2(CCCCN(C(C34CC(C3)C4)=O)C2)C1 3206,N1(C(C(C=C)(F)F)=O)CCCC(CCNC(C2CC3(CSC3)C2)=O)CC1 3207,C1(OC)CN(C(=O)C=C(C)Cl)C(C)(CNC(c2ccc(C(F)F)nc2)=O)C1 3208,Cc1cc(CC(N2CCC(NC(=O)Cc3ccc(Br)s3)C2)=O)c(C)s1 3209,Cc1nc2ccccc2n1CCC(N1CC2CC1C2NC(C1CCC(C)C1)=O)=O 3210,C1(C(=O)NCCCCCN(C(COCC(C)C)=O)C)CC(S(C)(=O)=O)C1 3211,c1(C(=O)NC(C2CCCN2C(C2CCC2C(F)F)=O)C)cncc(F)c1 3212,C1(C(N2CCC(NC(c3cccc(Cl)c3F)=O)CC2)=O)CCCCCCC1 3213,Cc1cc(C(=O)NCC2CCN(C(c3ncc(Cl)cc3Cl)=O)CC2)ccc1F 3214,c1(C(=O)NCC2CC(F)(F)CN2C(C2CC23CC(O)C3)=O)cn2cnnc2cn1 3215,C(=O)(C(C)CNC(C)=O)N(CCNC(=O)OCC)CCNC(=O)CCC1CC1 3216,C1(C)(C(=O)NCCC(C#C)OC)CCN(C(c2cccc(CO)n2)=O)C1 3217,C1(NC(CSSC)=O)CCC2CN(C(c3cnc4nccn4c3)=O)CC2C1 3218,C1(C(=O)NCC2(C3(O)CN(C(C4CC(=C)C4)=O)C3)CC2)CC2(C1)NC(=O)NC2=O 3219,c1(NC(C(CNC(C(CCC)=CCC)=O)C)=O)c(C)[nH]c(C)cc1=O 3220,c1(OC)ncc(C=CC(N2CCC(NC(=O)C(F)CC3CC3)C(CO)C2)=O)cn1 3221,C(=O)(NNC(=O)CCc1cccc(O)c1)c1ccc(C)cc1 3222,c1(CC)cc(C(N2CCC(c3cn(CCOC)nn3)C2)=O)nn1-c1ccccc1 3223,C1(CNC(Cc2c(CC)n[nH]c2CC)=O)C2CCC(C2)N1C(=O)Cn1ncnn1 3224,c1(C(=O)NC(CC)CNC(=O)C=CC(=O)N(C)C)ccnc(C(F)(F)F)c1F 3225,CCCCCCNCCC1CCN1C1CCCC1.C(=O)CCc1cccs1 3226,N1(C(CC=C)=O)CCCC(C)(CNC(=O)CN(C)CCC)C1 3227,N1(C(COC(C)C)=O)CCOC2CCN(C(=O)C=CCCc3ccccc3)CC12 3228,N#Cc1ccc(C(N2CCC(NC(c3ccc(-c4cc[nH]n4)cc3)=O)C2)=O)o1 3229,c1(C(N(CC(CNC(CCC(=C)Br)=O)O)C)=O)c(C)cccc1Cl 3230,N1(C(c2ccc(Br)cc2Br)=O)CC2CCN(Cc3cccc(F)c3O)C2C1 3231,C=CCC(C)C(=O)N(C1CN(C(c2cn(-c3cccc(CO)c3)nn2)=O)C1)C 3232,Cc1oc(S(N)(=O)=O)cc1C(=O)NCC1(F)CCN(C(c2cc(Cl)cs2)=O)C1 3233,CCC(CNC(=O)OC(C)(C)C)(CC)C(=O)NCc1ncc(C2CCOC2)s1 3234,CCCC(C(=O)NCC(C)(CNC(c1ccc(=O)n(C2CC2)c1)=O)OC)C(C)C 3235,C(C)(CCCNC(=O)C(N1CCC(C)C1)=O)NC(COCCCC#C)=O 3236,c1(C(N2CCC(C)(C(N)=O)C2)C(=O)NCCC2(C)CC2)ccc(F)c(Cl)c1Cl 3237,c1(C(=O)NC(C(C)NC(C(C)OC)=O)C)ccccc1Oc1ccncc1 3238,C1(CNC(Cc2n(C)cnc2)=O)CCCN(C(=O)CCNC(C2CCC2)=O)CC1 3239,CCCCCC(F)C(=O)NCC1CC1NC(c1onc2c1CCCC2)=O 3240,C1(CNC(C(C)=C2CCCC2)=O)CN(C)CCN1C(=O)CNC(=O)C(F)(F)F 3241,C1(CC=C)(NC(=O)CN2CC(C)(C)C2)CCCN(C(=O)C(C)OC2COC2)C1 3242,C1(C(N(CC(C)O)CC)=O)CCCN1C(=O)C(n1ccc(C)n1)C 3243,CCC(C)(C)C(=O)C(=O)NC1COCC1CO.C1CCC(=O)N2CC1C2 3244,N1(C(C(C(=O)OCC)F)=O)CCC(CNC(=O)Cn2nnc(=O)[nH]2)C(F)(F)C1 3245,C1(C(=O)NC(C)CNC(c2csc(COC)n2)=O)(COC)CCCC1 3246,N1(C(CCCC#C)=O)CCC2CCN(C(c3cn(C)c(C)n3)=O)CC12 3247,N1(C(CCC(=C)Cl)=O)CCC(C2CCN(C(c3cc4sccc4[nH]3)=O)C2)CC1 3248,c12cc(OC)cc(c1)NC(=O)Nc1ccc-2cn1.c1(OC)ncccc1OC 3249,c1(COCC(=O)NC(C)CN(C(=O)Cc2cncn2C)C2CC2)cccnc1 3250,N1(C(C(C)COCCc2ccccc2)=O)CC2CN(C(=O)CSC3CC3)CC2C1 3251,c1(CC(=O)NC2C(CNC(CN(CC(C)(C)C)C)=O)CC2)ccccc1Cl 3252,CC(C(=O)N(C(C)C(=O)NCCC1OCCC1(C)C)C)C(C)(C)C 3253,N1(C(C2C3COCC23)=O)CC2CCN(S(=O)(=O)c3ccccn3)C2C1 3254,CN1C(=O)CCCC1C(N1CC23CC1(C2)C(=O)NC3)=O.c1(CO)nnnn1C 3255,CC(C)(C)C(O)CC(=O)N1CCCC(O)(CCNC(c2cc(F)cc(Cl)c2)=O)C1 3256,c1(C(N2CCN(C(C3CCCN(C)C3)=O)CC2CC#N)=O)ccc(C#N)c(Cl)c1 3257,O=C(CC1CC(=O)c2ccccc21)Nc1ccc(Cl)c(S(=O)(=O)N2CCCC2)c1 3258,C(CO)(CCCCNC(c1nnc(C)s1)=O)NC(C(CC)CC1CCCC1)=O 3259,c1(C(N2CC(NC(C)=O)C(c3ccccc3F)C2)=O)cccc(CC2CC2)n1 3260,N1(C(CCOC(CC(C)C)C)=O)CC2CCC(C1)N2C(=O)CC(F)(F)F 3261,c1(SC)cccc(F)c1C(=O)NCCCNC(=O)C(O)c1cnc[nH]1 3262,C=C=CCCC(=O)N(CC)CC1CCCCN1C(=O)CC1(OCC)CCC1 3263,N#CC1(C(N2CC3CC2CN3C(=O)C=CBr)=O)CCOCC1 3264,c1(OC)cc(C(N2CCC2CNC(c2cccc(N)n2)=O)=O)ncn1 3265,C(=O)(C(CCOC)NC(C1(C)CC(C#N)C1)=O)NCCCOCCOC 3266,C(=O)(C(CCCC)N(C)C)N1CCC(O)(c2cn(C3C(OC)CCC3)nn2)C1 3267,c1(NCC2CC(NC(C3(C)CC3)=O)C2)ncc(C(F)F)cn1 3268,N1(C(C2(CCC=C)CC2)=O)CCN(C(=O)CCn2nc(C)cc2C)CC(C)C1 3269,C1(C)(C(=O)NCC2(NC(C(N3CCC(O)CC3)C)=O)CCCC2)COCCO1 3270,c1(C(N(c2ncnc(OC)c2C)C2CNCC2F)=O)ccc(F)c(Br)c1F 3271,CC1(C)CCc2cc(C(N3CCN(C(c4cnsc4)=O)CC(O)C3)=O)ccc2O1 3272,c1(OC)ccc(CN2CCCCC2C(=O)NC2CC(CO)C(O)C2O)cc1O 3273,c1(CCC(N2CCN(CCNC(C3(C)CC3)=O)CC2)=O)c(F)cccc1Cl 3274,C1(C(N(CCC(=O)NC2C=CCCC2)CC#C)=O)CCCC(=O)CC1 3275,C(=O)C1=NOC2(CCN(C)C2)C1.c1(C(N2CC(C)(C)C2)=O)csc2c1CCCO2 3276,c1(C(N2CC(N(C(c3c(C)onc3)=O)C)C2)=O)cn2c(n1)CCC2 3277,CC1Cc2cc(C(N3CCN(C(=O)CC(C)(C)C(F)(F)F)C(C)C3)=O)ccc2O1 3278,N1(C(C(CC)C(=O)OC)=O)CCC2CN(C(C3CC(F)(F)C3(C)C)=O)C(C)C12 3279,CC1COC(C(N2CCN(C(C3(Cl)CC34CCC4)=O)CC2)=O)CO1 3280,c1(C(N)=O)c[nH]c(C(=O)NCCOCCNC(c2nncs2)=O)c1 3281,C1(OC)COCCC1CC(=O)NC(C)(C)CNC(C1(NC(N)=O)CCCCC1)=O 3282,c1(C(=O)Nc2nc(C(C)NC(=O)OC(C)(C)C)cs2)c(C#N)ccc(Cl)c1F 3283,C1(CSc2n(-c3ccc(OC)cc3)c(C)nn2)Cc2ccccc2C1C 3284,Cc1[nH]c2ccc(C(=O)NCC(C(C)C)NC(=O)CC3CC=CCC3)cc2c1C 3285,N1(C(C2=CC(C)(C)C2)=O)CCC2CN(C(c3ccc4c(c3)CCOC4)=O)CC2C1 3286,C1(NC(C(c2c(C)cccc2)(C)C)=O)CC2CCC1C(NC(=O)C(O)CF)C2 3287,N1(C(C2(C)CC3CC3C2)=O)CC2(CC(NC(c3c[nH]c(C(N)=O)c3)=O)CO2)C1 3288,C1(C(=O)NCC[Si](C)(C)C)(CC)CN(C(=O)C(C)c2cccs2)C1 3289,Cc1cc(C(=O)NC(c2nccs2)C)c(C)n1N 3290,C1(CC(=O)NCC2C(C(=O)NCCc3onc(C)n3)C2)C(C)(C)C1(C)C 3291,c1(C(=O)NCC2CC(NC(C(c3n(C)ncc3)O)=O)C2)cc2cc(F)ccc2o1 3292,CN=c1[nH]cc(C(N2CCCC2C2(O)CN(C(c3cscc3C)=O)C2)=O)o1 3293,c1(OC(C)C)ccc(Cn2nc(-c3ccsc3)nc2CN2CCOCC2=O)cc1 3294,c1(C(=O)OCC(=O)Nc2c(C)ccc(Br)c2)cncc2c(Cl)cccc12 3295,C(=O)(CC(C)C(=O)OC)N(C(C(=O)NC1(COC)CCC1)C)C1CC1 3296,Cc1cncc(CC(=O)NCC(C)(C)CN(C)C(C2NC(=O)OC2C)=O)c1 3297,C=CC(C)(CC)C(=O)NCC(C)CNC(c1cn2ccnc2s1)=O 3298,C(=O)(CC(C)CCC=C(C)C)NCC(=C)CCNC(C1CCCCN1CCC)=O 3299,CN1CCOCC(NC(C2(NC(=O)C(O)CC(N)=O)CSC2)=O)C1 3300,c1(SCC)nc(N(c2ccco2)CCNC(=O)CNC=O)cc(Cl)n1.CCO 3301,CC#CCC(C(=O)N1CCC(C(C)C#N)CC1)NC(=O)C(n1cc(C)cn1)C 3302,N1(C(c2cc(OCCC)ncn2)=O)CCC(C)(CNc2ncc(COC)s2)CC1 3303,N1(C(C2CCC(C#C)CC2)=O)CCCN(C(c2cncc3sccc23)=O)C(C)C1 3304,c1(C(N(CC(CC)NC(=O)C(c2cccc(C)c2)C)C)=O)cncc(F)c1C 3305,C(=O)(CCCC(F)(F)F)NCC(CNC(C1CC(C)(C)OC1)=O)O 3306,C12(C(=O)NCC(CNC(c3ccccc3-n3cccc3)=O)F)CC1CCC2(F)F 3307,C#Cc1ccnc(C(=O)NCC(C2CC2)NC(=O)C(N2CCNC2=O)C)c1 3308,c1(CC)cc(C(=O)NC2CCC(N(C)C(c3ccnnc3)=O)C2)cc(F)c1 3309,C1(CC)CC(CC(=O)NC2CC(CNC(=O)CC(C)(F)F)C2)CCO1 3310,c1(SCC)cccc(CC(=O)N(C)CC2(NC(=O)CC(C)n3cccc3)CC2)c1 3311,c1(NCC(CCCC)NC(C2(CO)CCCO2)=O)cc(=O)n2cc(Cl)ccc2n1 3312,C1(c2nnnn2C)(CNCCC(C(F)(F)F)OC(C)(C)C)CC2CCC1CC2 3313,Cc1ccc(NC(=O)C(c2ccoc2)NC(=O)Cn2ccnn2)cc1CO 3314,N1(C(C(CC)(F)F)=O)CC(CCNC(c2ccc(NC)cc2Cl)=O)OC(C)C1 3315,c1(OC)csc(C(=O)NCCN(C(=O)C(n2ccnc2C)C)CC2CC2)c1 3316,n1(C(CC)C)ncc(C(=O)NC2(C(C)O)CC2)c1C 3317,N1(C(c2c(OC)c(Cl)ccc2)=O)CCC2(CCN(C(=O)CN(S(C)(=O)=O)C)C2)C1 3318,C(=O)(C(C)P(C)(C)=O)NCc1c(CCNC(CCNC(CC(C)C)=O)=O)ocn1 3319,N1(C(c2c(C)nsc2)=O)CC(NC(=O)Cc2cc(C3CC3)no2)C(C(F)F)C1 3320,N1(C(c2c(C)c[nH]n2)=O)CC2CCOCC2(NC(c2ccc3c(c2)OCC3)=O)C1 3321,N1(c2cc(NC(CCC)CCO)ncn2)CCC2(CC1)CC(CO)C2 3322,C1(C(=O)OC)C(C(N2CCC(NC(=O)Cc3cscn3)C2)=O)C1(F)F 3323,C(CCN=C(NCC1CN2CCN1CC2)NC(c1ccc(F)c(F)c1)C)OC 3324,C12(NC(=O)CCCn3ccnn3)CCN(C(c3ccc[n+]([O-])c3)=O)CCC1C2 3325,C(=O)(C(C)(C)C(C)(C)C)N1CC(NC(c2c(C(C)C)con2)=O)C(F)C1 3326,C(=O)(C(C)S(=O)Cc1cccs1)OC(c1ccccc1)Cc1ccc(OC)cc1 3327,C12(C(=O)NC3C(C)CN(C(c4coc(Br)n4)=O)C3)CC(C)(C1)OC21CCC1 3328,c1(OCC(N2CC(CNC(CC(=C)Br)=O)C(C)C2)=O)cccc(C)c1F 3329,c1(C(=O)NCC2C=CC(NC(=O)C=C3CCCC3)C2)cc(F)c(F)cc1Cl 3330,CC1CCN(C(C2CCOC2C2CC2)=O)C1C(=O)NC1C(C)C1C 3331,C1(O)(C(C)NC(=O)CCC2CCC(O)CC2)CCN(C(c2ccon2)=O)CC1 3332,C1(C)(NC(C(CC)N(C)C)=O)CCN(C(c2cnc(O)cc2OC)=O)CC1 3333,n1(CC)ccc(C(=O)N(CCN(C)C(c2ccn(COC)n2)=O)C(C)C)n1 3334,c1(C(=O)NC(CNC(Cc2nc(CC)sc2)=O)C)c(-c2ccccc2)noc1C 3335,c1(-c2c(C(=O)NCC3(C#N)CCC3)cncc2)cc(F)c(CO)cc1F 3336,N1(C(C2CCN(C)C2=O)=O)CCC2(CC1)CC2NC(C1(O)CC(C)(C)C1)=O 3337,C12CCCN(C1)C2=O.C1(O)(CN(C(c2ccn(C3CC3)n2)=O)CC)CCCC1 3338,c1(C(C(=O)N(C)CCF)NC(CC(=O)OC)=O)c(C)cccc1Br 3339,Nc1cccnc1C(N1CCC(NC(C2(c3ccccc3)CC2)=O)C1C1CC1)=O 3340,C1(c2ccccc2)(CCNC(=O)CC2(O)CN(C(C34CCC3C4)=O)C2)CCCO1 3341,c1(C(=O)NCCCN(CCO)C(C2CCCC2)=O)cc(F)cc(F)c1Br 3342,Cc1cccc(C(N2CCC=CC2C(=O)NCCC2=CCCC2)=O)c1 3343,C1(NC(c2c(C)cns2)=O)CN(C(=O)Cc2cn(C(C)C)nn2)C2(CCC2)C1 3344,C1(NCc2nnn(C)n2)CCN(C(c2cccc(Cl)c2)=O)CC1(C)C 3345,C1(CC)CCC(NC(=O)CCCn2cncn2)CC1 3346,c1(C(N2CCN(C(C=C(C)C)=O)CC2c2ccncc2)=O)ccc2c(c1)CCC2 3347,c1(C(=O)NCC2(F)CCC(NC(C3(C(F)F)CC(=C)C3)=O)C2)ccc(N)c(Cl)n1 3348,C1(CCCC)CN(C(c2ccsc2SC)=O)CCN1C(C1(Br)CC1)=O 3349,c1(OC)cc(C(=O)NCCOCCN(C(=O)C(C)C)C)on1 3350,Cc1oc2ccccc2c1C(=O)NCCC1CC(NC(c2cc(O)nn2C)=O)C1 3351,N1(C(c2c(N)ccc(C(=O)OC)c2)=O)C2CCC1CN(C(=O)CN1CCC1C)C2 3352,c1(C(N2CCC(C)(CNC(C3C(C)C3(F)F)=O)C2)=O)n[nH]c2cccnc12 3353,N1(C(c2c(C)snn2)=O)CCC(C2(NC(C3CCC(=O)O3)=O)CCC2)CC1 3354,C(=O)(C(CNC(=O)Cc1nccn1C)C(C)(C)C)NC(C)Cc1ccccn1 3355,CC(N=c1[nH]c(N(C)Cc2ccn(C3CC3)n2)nc2c1CCC2)c1csc(Br)c1 3356,c1(-n2cc(C3CCN(C(C4CN(CC)C(=O)C4)=O)C3)nn2)ccc(F)c(Br)c1 3357,c1(OC)cc(O)ncc1C(=O)NCCC1(O)CN(C(c2ccc(N)c(N)n2)=O)C1 3358,c1(NC(c2oc(CC)c(C)c2)=O)cc(C2CC2)cc(F)c1 3359,N1(C(=O)OC(C)(C)C)CC2(CNC(c3ccccc3)C3CC3(Br)Br)CC1(C)C2 3360,c1(C(N)=O)cccc(OCC(N2CCN(C(C3CC=CCC3)=O)CC2)=O)c1 3361,C1(C(=O)NCC(CNC(C2C(C(=O)OC)CCO2)=O)CO)CCC(F)(F)CC1 3362,c1(C(=O)NC2C(NC(C3(CSC)CCOCC3)=O)CCC2)cc2scc(C)c2[nH]1 3363,N1(C(c2c(C)coc2)=O)CCCC(C)(C)C1C(N1CCCC(O)C1)=O 3364,c1(CS(C)(=O)=O)ccnc(C(=O)NC2CC2NC(=O)CC23COC(CF)(C2)C3)c1 3365,C=C1CC2(C1)CC(C(=O)NCC1CCCCN(C(C3(COC)CCC3)=O)C1)C2 3366,C1(CNC(c2cc(C)c(C)nc2)=O)CC2COCC2N1c1ncc(F)cn1 3367,CC1CCCc2ncc(C(=O)NC34CC(NC(C5CC56CCSCC6)=O)(C3)C4)n21 3368,C1(O)(CC(=O)NCC(C)(C2CCC2)NC(=O)CCc2nccs2)CCOC1 3369,CC1CC(CCNC(=O)Cc2cncs2)CCN1C(c1csc(C(N)=O)n1)=O 3370,N1(C(c2n(C)ccc2)=O)CCC(C)(C)C(CNC(=O)CC2CCC3(CC2)CC3)C1 3371,C1(C(=O)NC2CC(N(C(c3noc(CC)c3C)=O)C)C2)CCc2n[nH]cc2C1 3372,N#Cc1c[nH]c(C(N2CC3CC3(NC(c3cc(-c4ccccc4)cs3)=O)C2)=O)c1 3373,CC(C(=O)NCC1(CC(=O)NCCCc2nc[nH]n2)CC1)C1CCCO1 3374,C12(CNC(CSCC#C)=O)CCC(NC(=O)CCC3CCCCC3)(CC1)CO2 3375,c1(CN(CC(=O)NCC2C(NC(CC=C)=O)COC2)C)cccc(C#N)c1 3376,N1(C(C(CC(C)C)=O)=O)CC2C=CC1C(C(=O)N(C1(C)CC1)C)C2 3377,C=CC(C)(CCOC)C(=O)N(C1CCCC1)CCNC(=O)CC(F)(F)C(F)F 3378,C12(CNC(c3ncn(C(C)C)n3)=O)CCC(CC1)N2C(C1(Br)CC1)=O 3379,N1(C(C(c2nc(C)sc2)=O)=O)CC(NC(c2ccc(C(F)F)nc2)=O)C(C)(C)C1 3380,N1(C(=O)CON2CCC2OCc2cn(CC3CCOC3)nn2)CCC(CO)CC1 3381,CN1CC=C(C(=O)NC2COCCN(C(C3(C#N)CC3C(F)(F)F)=O)C2)C1 3382,c1(CN2CC(C(CF)(F)F)(C(=O)O)C2)cnn2c1OCC2 3383,C(c1cccc(Cl)c1)=C(C(N1CC(NC(C(C)(C)SC)=O)C1)=O)C 3384,c1(C(CC(=O)OC)NC(=O)C(C)NC(C2CSCN2C(C)=O)=O)ccc(Br)cc1 3385,C1(NC(=O)CCc2cnccn2)CCN(C(c2ncccc2Br)=O)CC1CO 3386,N1(C(C(N2CCNC2=O)C)=O)CCC(C(=O)NCCCn2cnnc2)CC1 3387,N1(C(CCc2ccnc(C)n2)=O)CCN(C)C(CNC(c2csnn2)=O)C1 3388,c1(N2CC(C)C(NC(c3occ4c3CCC4)=O)CC2)ccc([N+](=O)[O-])cn1 3389,c1(C(N2C(CNCc3c(C)n[nH]c3)CCCC2)=O)cnc2c(c1)CCCC2 3390,CC1CC2(C(N3CC(F)(CNC(C4(CCOc5ccccc5)CC4)=O)C3)=O)CC12 3391,CC1CCCN(C(C2CCS2(=O)=O)=O)C1CNC(=O)CCN1CCOC1=O 3392,c1(C(=O)NCC2(C)C(C)CN(C(C(CCSC)O)=O)C2)cc(Cl)c(Cl)cc1N 3393,C1(CNC(CCSCCC)=O)C(C)CCCN1C(c1cc(C2(C)CC2)on1)=O 3394,C(=O)(C1=CC2CCCCCC12)NCC(CC)N(C(=O)C=C(CC)CC)C 3395,c1(C(C(=O)N(C2CCN(C(C3CCCC(C)C3)=O)CC2)C)O)cc(F)cc(F)c1 3396,N1(C(C2(C)CC(=C)C2)=O)CCC(CNC(c2cnn(C3CC3)c2)=O)C(O)C1 3397,C1(C(=O)NC)CS(=O)(=O)CN1CCN(C(CNC(CC)=O)=O)C.C1CCO1 3398,N1(C(C(C)N(C(=O)CCN2CCCCC2)CC)=O)CCc2ccncc2C1 3399,CC1CCCc2ccc(NC(=O)NCC(C3(O)CCCC3)N(C)C)nc21 3400,C=C(C)C(CC(=O)N1CCCC1CN(C(=O)C=Cc1ccccn1)C1CC1)OCC 3401,C1(NC(C2(CC=C)CC=CC2)=O)COCCC1NC(=O)CCN1CCOCC1 3402,c1(NC(C(=O)Nc2c(Cc3ncc(C)[nH]3)cccc2)=O)c(C)cc(C)cc1C 3403,c1(C(N2CCCC2c2cn(C3CCC3)nn2)=O)cnc(CC2CCOC2)s1 3404,C(=O)(C1=CC2CCCC12)N(C1CCN(C(c2ccc3nncn3c2)=O)CC1)CC 3405,C(=O)(CCCCC(=O)OC)N1CCN(C(COCCC=C)=O)CC1C(C)(C)C 3406,CCC(CC)(CC)CN=c1[nH]c(=NCC2CC23CCOC3)[nH]c2c1CSC2 3407,CC1(CCC(=O)Nc2cnsc2)CCCN1C(=O)Cc1ccc(Cl)s1 3408,C1(N(C(=O)Cc2csc(Cl)n2)C)CN(C(=O)C#CC2CC2)CC12CC2 3409,C1(C(=O)NCCCC(=C)Cl)CN(C(=O)C(C)NC(C)=O)CC12CC2 3410,c12cc(F)ccc1[nH]c(=O)[nH]2.N1(CC)CCC(N2CCN(C)CC2)C(C)C1 3411,N1(C(C(C)C(F)F)=O)CC(CC(=O)NC2CCN(C(N)=O)CC2)C2(CC2)C1 3412,N1(c2snc(C)n2)Cc2ccccc2C(CNC(C23CCC(C2)OC3)=O)C1 3413,C1(C(N2C(C(=O)NC3(CCC)CC3)CCCC2)=O)C2CCCC(=O)C12 3414,Cc1ncc(CNC(C2(C)CCCN2C(c2cc(C(C)C)[nH]n2)=O)=O)n1C 3415,CCCC(CNC(c1cccn1C)=O)C(=O)N(CC)CC1CCCO1 3416,c1(N(c2cnn(C)c2)C)nnc(-c2cnsn2)n1C 3417,C1(CC(=O)NCCn2ncc(CC)c2)CCN(C(c2cnc(NC)cn2)=O)CC1 3418,N1(C(C=CC)=O)CC(C)(C)OC2(C1)CN(C(c1ccc(S(N)(=O)=O)c(N)c1)=O)C2 3419,Cc1cc(=O)ccn1CC(=O)NCCCN(C)C(c1coc(C(F)(F)F)n1)=O 3420,C12(C(N3CC4C(N(C)C)C4C3)=O)CC(CN(C(=O)CN3CCSCC3)C1)C2 3421,c1(C(N2CCCN(C(C3CC(NC)C3)=O)CC2)=O)nc(C)ccc1C(=O)OC 3422,Cc1cc(S(=O)(=O)CCN2CC(C)OC(C)C2)c(C)cc1-c1ccc[nH]1.C1CN1 3423,C=CCC(CC)C(=O)N1CCOC(C)(CNC(c2cnn(CC3CCC3)c2)=O)C1 3424,C1(NC(Cc2cc(OC)no2)=O)C2CN(C(C3CC(C)OC3C)=O)CC12 3425,N1(C(C2CCCC(=O)N2)=O)CC(NC(=O)CCc2ccccc2Cl)CC(F)(F)C1 3426,c1(C(=O)NC(CC)CNC(=O)COC2CCCOC2)c(Cl)n[nH]c1C1CC1 3427,OC1CCC2(CC1)CCN(CC1CC3(CCC3)CCO1)C2 3428,c1(OC)ccc(O)cc1C(N1CC2CC1CC2NC(c1ncc[nH]1)=O)=O 3429,N1(C(c2c(C)nc(CC)o2)=O)CCN(C(=O)COCC2CCOC2)C(C(F)F)C1 3430,C(=O)(C1=CCN(C)C1)NCC(CC(C)C)NC(=O)Cc1ccno1 3431,Cc1ncc(NC(C2CCCN(C(=O)C(C)C3CCC3)C2)=O)cc1Cl 3432,Cc1cc(F)ccc1C(N1CCC(N(CCO)C(C2OCC2(C)C)=O)C1)=O 3433,N1(C(c2cc(C)sc2)=O)CC2(C=C(C(=O)N(C3CCCCC3(C)C)C)CO2)C1 3434,C(CCC1CC1)(C(=O)N1CCC(CCF)CC1)NC(c1cc(Cl)c[nH]1)=O 3435,Cc1c(F)cc(CNC2CCC(NC(c3cnn(C)c3)=O)C2)cc1F.C(N)=O 3436,c1(C(=O)NCC2N(C(c3cc(N)c(F)cn3)=O)CC(F)C2)ccc2c(c1)OCC2 3437,C(CO)(CCCCNC(C1CC(O)C1)=O)NC(c1cscc1Cl)=O 3438,CCCCCCCC(=O)N1CCCC(NC(=O)Nc2cccc(Cl)c2F)C1 3439,C1(C(=O)NCCCN(C(=O)CCn2cnccc2=O)C)CN2CCN1CC2 3440,C1(C(=O)NCC=CC(=O)N(CC(COCC)O)C)CCC(C)O1 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3458,N1(C(C(C(=O)OCC)(C)C)=O)CCC2(CCN(C(=O)CCC3(C)N=N3)C2)C1 3459,C1(NC(C(C)CCN(C)C)=O)CN(C(C2CC2(F)F)=O)CC(C)(C)C1 3460,c1(NCC2CCCN(C(CCC(C)OC)=O)C2)c(C(C)=O)cc([N+](=O)[O-])cc1Cl 3461,Cc1nc(C)c(C(=O)NCC2(CNC(=O)CCC(=O)N(C)C)CCOCC2)[nH]1 3462,N1(CC=C(C)C)CCN(C(=O)C(CC2CC2)NC(C2CNC(=O)C2)=O)CC1 3463,CN1CCCCCC1C(=O)NC1CC(O)CN(C(=O)C2=C(Cl)CCC2)C1 3464,C1(C(=O)NCC2(C)N(C(c3ccnc(C)n3)=O)CCC2)COC2(CCC2)CO1 3465,n1(CCC#C)c(N2CCC(NC(C)=O)C2)nnc1-c1cnn(CCC=C)c1O 3466,c1(OC)cccc(COCC(=O)NC2CC(CNC(=O)COC(F)F)CC2O)c1 3467,c1(CN2CCC(CC(=O)Nc3cccnc3F)C2)cnc(O)nc1O 3468,N1(C(CC(CC(=O)OC)C)=O)Cc2ccc(C(C)NC(C3CN(C)C3)=O)cc2C1 3469,CC1CN(C(=O)OC(C)(C)C)CC1CC(N1CCC(c2nnc(O)n2C)CC1)=O 3470,CC1CN(C(=O)CCc2ccc(O)nn2)CCCN1C(c1ccc(F)cc1Cl)=O 3471,N1(C(c2c(CC)noc2)C(=O)NC2CCOC2)CCOC(CF)C1 3472,c1(C(=O)NC(CCOC)CNC(=O)C(C)CSC(F)(F)F)cnc(C#N)s1 3473,N1(C(C2(c3c(C)cccc3)CCCC2)=O)CC2(CCN(C(=O)CC(C)F)CC2)C1 3474,C1(C(N2CCCC2CNC(c2ns[nH]c2=O)=O)=O)(OC)CCSC1 3475,S(=O)(=O)(c1ccsc1C(=O)NCCCCC(C)NC(=O)C(F)(F)CO)NC 3476,Cc1nn(C)c(C(=O)NCc2cc(O)nc(CNC(=O)C(C)O)n2)c1Cl 3477,C(=O)(C(C)(C)CC(C)C)C(C)=O.C1(N)CC1C1CCCC1.C123CC(C1)(C2)CC(=O)N3 3478,C1(CCC=C)(C(=O)NCc2cc(COC)on2)CN(C(=O)CCc2cnc[nH]2)C1 3479,C1(NC(C2(C)C=CCC2)=O)CCC2(CC1)CC2NC(c1cncc(O)c1)=O 3480,c1(N2CC(CCCCNCc3n(CC)ncn3)C2)cnc2c[nH]nc2c1 3481,C1(C#CC(=O)NC2CCC(CNC(c3csc(C(C)=O)n3)=O)C2)(CC)CC1 3482,c1(NCCOCCCCC)noc(CC(C(N)=O)NC(=O)CC)n1 3483,CN1CC=C(C(=O)NC2CCC(NC(=O)C(CCO)N(C)C)CC2)C1 3484,N1(C(CCC(=O)OC(C)(C)C)=O)CCN(C(C2CCC(F)C2)=O)CC12CCC2 3485,C(C(CCC)C(=O)NCc1ccn(C2CC2)n1)NC(COC1(C#C)COC1)=O 3486,N1(C(C2C(NC(C3CCCC3F)=O)CCOC2)=O)C2C=CCC1CCC2 3487,C(=O)(CS(C)(=O)=O)N1C(C(=O)NC(C=C)(C)CC)CC1 3488,Cc1cc(C(N2CCCC2CNC(=O)CCc2cc[nH]n2)=O)cc(C)c1F 3489,c1(CC(=O)NC2CC(NC(c3ccc(F)cc3O)=O)C2)cc(F)cc(Cl)c1 3490,C1(C(N2CC(O)CC(NC(c3c(C)cccc3N)=O)C2)=O)CC2C=CC1C21CC1 3491,c1(OC(CC)C)cc(NCC2(O)CCN(C(C3CCCC3C)=O)CC2)nc(C)n1 3492,c1(C(N2CC(NC(CSCC)=O)C(CO)CC2)=O)cc2c(C)sc(C)c2s1 3493,Cc1cnc(CCNC(=O)C(C2CCN(C(=O)Cn3cc(CO)nn3)C2)F)nc1 3494,CC1OC(=O)NC1C(=O)NCC#CC(=O)NCC#CCCO 3495,Cc1ccc(-c2nc(CC(C)Oc3ccccn3)n(-c3ccc(F)cc3)n2)cc1 3496,c1(CNC(C2CC(OC)C(OC)C2)=O)ccc(CN)cc1F 3497,N1(C(c2cc(C)c(O)cc2)=O)CC(C)(CNC(C2CCC(=O)NC2)=O)CC1(C)C 3498,CC(C)CC(Cn1cc(C2(C)CC2)nn1)NC(=O)CSc1ccccc1 3499,N(C1CCc2ccccc21)(CC(=O)OC)C(=O)CO 3500,C1(CC)C(NC(c2cc(Cl)ccn2)=O)CCN1C(C1CC1c1ccccc1)=O 3501,CC1CN(C(=O)CSCCC#N)CCC1CNC(=O)Cn1ccccc1=O 3502,N1(C(C2CC(OC)C2)=O)CCC2(CC(NC(=O)Cc3ccnc(Cl)c3F)CO2)C1 3503,N1(C(c2ccc(C)c(Cl)c2)C(=O)NC(C)(C)C)CCOCC2(COCCN2C)C1 3504,c1(C(N2CC(O)CC(NC(C=CSC)=O)C2)=O)cc2cc(Br)ccc2o1 3505,c1(C(=O)NC2(C(=O)NCC(C)(C)C#N)CC2(C)C)ccc(C#N)cc1 3506,N1(C(CC(CC)(F)F)=O)CC2(CC(C(=O)NC34CC3COC4(C)C)CO2)C1 3507,c1(CC)ccc(C(N2CC(CNc3ncc(Br)c(C)n3)CC2C)=O)cc1F 3508,C(CC1=CCN(Cc2ncc(C(F)F)o2)CC1)NC(=O)CCC1CCCCO1 3509,c1(OC)ncnc(OC)c1CNC1CN(c2nccc(C(F)F)n2)CC12CC2 3510,c1(C(N2CC(C)C(CNC(C34CCN(CC3)C4)=O)CC2)=O)ccn2ccnc2c1 3511,N1(C(CNc2ccc(OCC)cc2)=O)CC(C(=O)O)c2ccccc21 3512,N1(C(C(CCC)=CCC)=O)CCCCC(NC(=O)C(C)N2CC(C)C2)C1 3513,C(CCCCCCC(=O)OC(C)(C)C)NC(CCC)CCc1ccccc1 3514,N1(C(C(C(C)C)NC(N)=O)=O)CC(NC(c2coc(C3CC3)n2)=O)C2CC2C1 3515,c1(NC(C(=O)NC(CC(C)NC(=O)C(C)OCC2CC2)C)C)cc(Cl)ccc1Cl 3516,C#Cc1cccc(C(=O)NCC2CCCCC2NC(C2CCSCC2)=O)c1C 3517,c1(C(=O)NC2CC(C)CN(C(C3(O)CCOC3)=O)C2)ccc(S(N)(=O)=O)c(F)c1 3518,Cc1cc(C(N2CC3CC(NC(=O)CCCc4ccccn4)C3C2)=O)cc(O)n1 3519,c1(C(N2CCC(CN(C(c3cnc(C)[nH]3)=O)C)CC2)=O)nc(Cl)ccc1F 3520,C1(C(N(C(CCC)C)C)=O)(COC)C=CCN1C(C1CN(C(N)=O)C1)=O 3521,N1(C(C(C)(C)CF)=O)CCC(CNC(=O)C(c2ccc(F)cn2)(F)F)C(F)(F)C1 3522,C1(C(=O)NCCC2(O)CN(C(c3nccc(C)c3)=O)C2)CCCS(=O)(=O)C1 3523,Cc1nc2n(n1)CC(C(=O)N(CC(c1ccccc1)C1CCC1)C)CC2 3524,N1(C(CCN(C(C(C)OCC(=O)OC)=O)C)=O)CCN(C)C(C(C)C)C1 3525,C(=O)(C(CCCC=C)NC(=O)C(C1C=NN(C)C1=O)C1CC1)N1C(C#C)CC1 3526,c1(C(=O)NCC(C2CCN(c3snc(SC)n3)CC2)(C)C)cc(C#N)ccc1Cl 3527,c1(C(N2CCCC(N(C(C(CCC)C)=O)CC)C2)=O)c(C)nc(C)n1O 3528,CCC(CC(=O)N1CCC(CN(CC)CC)CC1)C(C)C.c12ncoc1N2 3529,c1(C(N(C)CC2N(C(C(C3CCOC3)OC)=O)CCCC2)=O)cc(C#N)n(C)n1 3530,C1(NC(C(c2ccc(OC)cc2C)C)=O)CN(C(=O)C(N)=O)C2(CCCC2)C1 3531,N(C(=NCCc1nnc(C)s1)NCC(c1ccccc1)C)CC(C=C)C 3532,c1(N(CC=C(Cl)Cl)C(C)C)ccc(C(C)(C)C)cc1 3533,C1(CNC2(c3cccc(C(=O)NC(C)C)c3)CCC2)CCCS1(=O)=O 3534,C(=O)(C1=CCCOCC1)NCC(C(N1CCCC[Si](C)(C)C1)=O)CC1CC1 3535,Cc1cc(C(=O)NC2CC(CNC(c3[nH]cnc3C)=O)CC2O)nnc1O 3536,C1(NC(C=CC=CC)=O)CN(C(=O)C(CC)C(C)=O)CC1C(F)F 3537,C1(N(C(C)C)C(=O)NCC(C2CCCO2)O)CCN(C)CC1 3538,C#CCC(C(=O)N1CCC(CC(=O)Nc2ccccc2OCC)C1)C1CC1 3539,Cc1cc(C(=O)NC2CCN(C(c3cn(C)nn3)=O)CC2C)ccc1Cl 3540,C(CC(C)C)(C(=O)N1CC(CNC(c2c3c(nn2C)CCC3)=O)C(C)(C)C1)OC 3541,S(=O)(=O)(c1cccc(Oc2ccccc2)n1)N(C(CCC)C(=O)O)C 3542,c1(C(=O)OC)cc(NC(=O)NC(c2cccc(OC(F)F)c2)C)ccc1F 3543,N1(C(C2CN(C(=O)NC)C2)=O)CC(C2(NC(c3nc(C4CC4)oc3C)=O)CC2)C1 3544,C(C(N)=O)(C(C)CC)NC(C(C1CCN(C(CC2ON=C(CC)C2)=O)C1)C)=O 3545,N1(C(C(C=C)O)=O)CCC2(CCC(NC(c3cc(C)c4[nH]nnc4c3)=O)CC2)C1 3546,n1(CC#C)cccc1C(=O)NC1(C(=O)NCC2CN(C(C)C)C2)CCSC1 3547,N1(C(c2ccc(Cl)c(C(F)F)c2)=O)CCc2ccc(Br)cc2CC1 3548,c1(CN2C(CC(C)C)(CC)CCC2)cn2ccccc2n1 3549,c1(C(N2C(CCC(=O)NC(CC=C)C3CC3)CCC2)=O)ccc([N+](=O)[O-])[nH]1 3550,C(=O)(C1=NN(C)C(=O)CC1)N1CC(NC(CCN(C(CCC)C)C)=O)C(O)C1 3551,C1(CNC(=O)CNC(=O)Cn2cccc2)C2CN(C(=O)CCC3CCOC3)CC12 3552,c1(OC)ccc2c(C)c(C(=O)NC3CCC4(CC3)CC4)[nH]c2c1 3553,c1(C(N(CC(CN(C(=O)Cc2cnoc2)C)O)C)=O)ccn(CCF)n1 3554,C1(F)(CNC(c2nc(CC)oc2C)=O)CCCN(C(c2ccon2)=O)C1 3555,N1(C(=O)Cn2ccc(C(F)(F)F)n2)CCCC2CCN(C(=O)C3=COCC3)CC12 3556,C=Cn1nncc1C(=O)NC1(CN2CCN(C(=O)C(C)O)CC2)CC1 3557,c1(CCCSC)cn(CCN(C)C(C2CC2(C)C)=O)nn1 3558,S(=O)(=O)(c1c[nH]ccc1=NC(CF)CF)NC(c1cc(C)no1)C 3559,Cc1ccsc1CCCC(=O)NCCOCCNC(=O)C(C)C1(O)CCC1 3560,c1(C(N(C2CN(C(c3onc(CC)c3C)=O)C2)C)=O)cc(F)cc(Br)c1O 3561,C1(CNC(CCCCC=C)=O)CN(C(=O)C(F)(F)C(O)CC)CCC1(C)C 3562,C(=O)(C(C)(CC)CCC)N1CC(C(C(N2CCCC(OCCC)C2)=O)O)C1 3563,CCS(=O)(=O)CC(=O)NC(C)C(C)NC(c1ccoc1CC(N)=O)=O 3564,C(=O)(C(COC)NC(=O)COC)N1CC(OCCOCC)C1 3565,C1(C2CCN(C(=O)COc3ccccc3F)C2)(NC(c2cccs2)=O)CC1 3566,C1(C(=O)NC(C(=O)N2CC(OCCCCC)C2)CO)COCCN1CC 3567,c1(CC)ccnc(C(=O)NCCn2cc(C(N3CCCC3(C)C3CC3)=O)nn2)c1 3568,N1(C(CC(C)(F)F)=O)CC2(CCC(NC(=O)CC3NC(=O)NC3=O)CC2)C1 3569,C1(C)(C(=O)NC2C(NC(CSC(C)(C)C)=O)C2)CC2(C1)CC(F)(F)C2 3570,C1(C(=O)NCCCNC(C(C(C)(C)C)O)=O)CC(O)c2ccccc2O1 3571,C(=O)(C1CCc2nccn21)NCC(=O)NCc1c(C)nsc1 3572,CC1=C(C(=O)NC2CCCCCC2NC(=O)Cn2nc(C)nc2C)CCS1(=O)=O 3573,N1(C2CN(C(C(=C3CCCCC3)C)=O)C2)CCN(C(c2ncn(C)n2)=O)CC1 3574,c1(C(N2CCN(C(Cc3scc(C)c3)=O)CC2C)=O)nn(C)c2c1CCC2 3575,c1(CC)nc(O)c(C(N2CC(CNC(c3occ(C)c3C)=O)C2)=O)cc1C 3576,C(CC(C)N=c1[nH]c(=NCC2CC2c2ccc(Cl)cc2Cl)c2ccccc2[nH]1)OC 3577,C12CCN(C1)C2=O.C1(CCOC)(NC(=O)Nc2cn(C)nn2)CCCC1 3578,CCC(CN(C)C)CC(=O)N(C1CN(C(=O)C(C)NC(C2CCCC2)=O)C1)C 3579,C1(=O)CC(C)(C)N1C.C1(C(F)(F)F)(C(=O)O)CSC1 3580,C1(O)(CN(C(COCC)=O)C)CCN(C(c2c(C)cncc2C)=O)CC1 3581,Cc1cnc(NC(CNC(C2CC23CCOC3)=O)C2CCC2)nc1O 3582,C#CCCCCC(=O)NCC(C)(O)CNC(c1ccc(C(=O)C2CC2)cc1)=O 3583,C1(NC(c2ccc(CNC(CC(C)O)=O)cn2)=O)CCCN(C)C1C 3584,c1(C(=O)NC2C(NC(c3c(N)nc(Cl)cc3)=O)COC2)cnn2c(=O)cc[nH]c12 3585,C(=O)(CC(C)CC(C)(C)C)N1CC(O)(CN(C(C#CC(C)C)=O)C)C1 3586,C(CCC)(C(O)C(=O)N1CC=CC1CF)NC(C(C)OCC#C)=O 3587,N1(C(c2c(OC)csc2)=O)CCCN(C(c2ccnn2C(C)C)=O)C(CO)C1 3588,c1(C(=O)NCCC(CNC(=O)C=Cc2ccccc2)O)cccc2ccnn12 3589,C(CC(=O)NC)C(C(N1CCCC1)N(C(=O)CCOCCOCC)CC#C)=O 3590,c1(CNC(c2sc(C(=O)NC3(C)CN(CC)C3)c(C)c2)=O)ccc(C)c(C)c1 3591,C(=O)(CCS(=O)(=O)Cc1ccncc1)N1CCC(NC(C(CC)(C)C)=O)C1 3592,N1(C(CCN(C(C)C)C(C2CCOC2=O)=O)=O)CCC2(CC1)CC2C#N 3593,C1(CNC(C2C(C(=O)OC)CC2)=O)CC2CN(C(c3cc(C)nc(C)c3)=O)CC12 3594,C(=O)(C1=C2CCN=C2NC=C1)N1CCC(N(C(=O)CS(C)(=O)=O)C)CC1 3595,C(N=c1nc(N2CCC3(CCCN(C)C3)C2)c2sccc2[nH]1)C1C(C)C1C 3596,c1(OCC)ccc(Cl)nc1C(=O)NC1CCN(C(=O)CCCOCCOCC)C1 3597,CC1CC(c2nn[nH]n2)CC(C)N1CC(C)(C)CO 3598,Cc1ccc(C(=O)NC2CCC(C)N(C(C3CC4CCC3CC4)=O)C2)cc1CO 3599,c1(CC)cccc(C(=O)NC2CC2NC(=O)COc2ccc(C)cc2)c1C 3600,N1(C(C(C(=C)Cl)(C)C)=O)CCC2(CCN(C(=O)C(C)(C)COCC(F)F)C2)C1 3601,C1(CC(=O)N(CCC(N)=O)C)CN(C(c2cc(O)cc(=O)o2)=O)C(C)(C)C1 3602,N1(C(COCCC)=O)CCC(C(=O)NCc2cn(C3CC3)nn2)C1C 3603,c1(C(N2CC(C(C)NC(=O)C(C)(C)c3cc[nH]n3)OCC2)=O)cnc(O)c(Cl)c1 3604,c1(C(=O)NC(C)C(C)(C)NC(C2CCC(F)(F)C2)=O)cccc[n+]1[O-] 3605,c1(N(C)C)ccc(C(=O)NC2(CNC(c3ccc(C#N)[nH]3)=O)CCCCC2)cn1 3606,CN1CCC(C(=O)NCC23CC(CNC(=O)CC(F)(F)F)(CO2)C3)CC1=O 3607,c1(SC)ccc(C)c(C(N2CCOCC2CNC(c2ccc(C)c(C)c2)=O)=O)c1 3608,C1(C(N(CCC2CN(C)C2)C)=O)CN(C(=O)Cn2nccn2)CCN1C 3609,c1(CC(=O)OC)ccc(C2CNC2)cc1.C1C(C)C(=O)NC(=O)C(=O)N1 3610,C1(C)(C(N(C(CNC(=O)CCC2CCCOC2)C2CC2)C)=O)CCCO1 3611,C(=O)(C(C)(C)C(C)(C)O)N1C(CNC(c2cccc(COC)c2)=O)CCC1 3612,c1(N2CC3CC4C(O)C2C3C4)nc(C2CC2)nc2ccccc12 3613,c1(C(N(C2CCCCC2)CCNC(c2c[nH]cc2Br)=O)=O)nsnc1O 3614,Cc1nc(C(N2CCC(F)(C(N3CC=CC3CO)=O)C2)=O)ccc1Br 3615,C(CC(CC)C(=O)NC1C=CCC(C(=O)N(CCN2CCOCC2)CC)C1)=CC 3616,C1(CNC(c2c(CC)scc2)=O)CCC2CN(C(C3CN(C)C(=O)N3)=O)CC12 3617,C(=O)(C(CNC(c1cc(C2CC2)no1)=O)C(C)(C)C)NC(c1nncn1C)C 3618,N1(C(CCCC(C)n2cc(-c3cnc(C(=O)OC)s3)nn2)=O)CC2(CCCCC2)CC1C 3619,C(=O)(C1CNC(=O)c2ccccc21)NCC1C2CN(C(C(N)=O)=O)C1CCC2 3620,C=CC(O)(C(=O)NC1CC(NC(c2cnn(C)c2C)=O)C(O)C1)C(F)(F)F 3621,c1(OC)cc(C)c(C(=O)NCCOc2ccc(NS(C)(=O)=O)cc2)o1 3622,C1(NC(c2n[nH]c(CC)c2Cl)=O)CC(OC)CN(C(=O)C(C2CCCC2)OC)C1 3623,C1(CCCNC(C(F)=CCC)=O)CN(C(c2ccnc(OC)n2)=O)CCO1 3624,n1(CC(=O)N(CCCCCNC(C2CC2Cl)=O)C)ccc([N+](=O)[O-])n1 3625,CCC(CNC(C1CN(C(=O)CCC(C)(C)C)CCN1C)=O)CC(C)C 3626,C(CC(=O)N1CC(NC(C2(c3ccc(F)cc3)CCOCC2)=O)C1)(C(F)(F)F)OC 3627,N1(C(=O)CC(F)(F)CCc2ccccc2)CCC2(CC1)CC(F)CO2 3628,C1(NC(C2CN(C)C2)=O)CCN(C(=O)CCNC(N)=O)CCC1c1ccccc1 3629,C=CCC(CC(C)C)C(=O)N(C(C)CCNC(=O)Cc1nsc2ccccc12)C 3630,N1(C(C(C)SC(F)(F)F)=O)CC2CCN(C(c3nnn4c3CSCC4)=O)CC2C1 3631,c1(C(=O)NC2C(CNC(Cc3nc(C)sc3C)=O)CCCC2)cccc(Cl)c1N 3632,C1(NC(c2cc(CCC)[nH]n2)=O)CC(O)CN(C(=O)Cn2cc(F)ccc2=O)C1 3633,C(CC(O)C(F)(F)F)NC(C(CC=CC)NC(=O)CC1CCOC1=O)=O 3634,C(=O)(C1=COCCC1)NCC(CC(C)C)NC(c1cncc(CO)c1)=O 3635,N1(C(C2CCCC(OC)C2)=O)CCC2(CC1)CCN(C(C1CC1C)=O)CC2 3636,CCC(C)C(C(=O)OC)N(C(=O)C(C)NC=O)C.C1CCCC(=O)N1C 3637,N1(c2ncc(CC)cn2)CC2CC(NC(=O)CCCc3cccnc3)CC1C2 3638,c1(C(=O)NC(CNC(C(C(C)C)n2cccc2)=O)CO)cn2cnnc2cn1 3639,c1(CC(C)C(=O)NC(C)(C)C)ccc(F)cc1.c12ccc(o1)COCCNC2=O 3640,N1(C(C2(CC#C)CCCOC2)=O)CCC2(CC1)CC2CNC(=O)CCOC 3641,C(=O)(CCN(OC)C(=O)c1ccc(C#N)[nH]1)N1C(C)CC1 3642,N1(C(Cc2ccc(C)cc2)=O)CCCC(C)C1CNC(=O)C=CC1CCOCC1 3643,c1(C(=O)NCC2CC2NC(=O)C(O)Cc2ccc(Cl)cc2)nccc2[nH]ccc12 3644,C1(C(N(c2cn(CC)nc2)C)=O)CCC(C)(C)N(C(c2cc(OC)n[nH]2)=O)C1 3645,CC1CC2(CCO1)CC2C(N1CC(OCCNC(c2conc2C2CC2)=O)C1)=O 3646,c1(C(=O)NCCOC2CCN(C(c3c(OC)nccc3)=O)C2)c(C)cnnc1O 3647,N1(C(CCCC(N)=O)=O)CCC2CN(C(=O)C=CCN3CCOCC3)CC12 3648,N1(c2c(OC)cncn2)CC(NC(c2ccc(C)[nH]2)=O)C(C)(C)C1 3649,N1(CC)CC2CN(C(=O)C(CC)NC(c3ccc(F)cn3)=O)CC2C1 3650,Cc1c[nH]c(C(N2CCOCC2CCNC(C2(C(F)(F)F)CCC2)=O)=O)cc1=O 3651,C(c1cscn1)=CC(=O)N(C1CCN(C(c2sccc2C2CC2)=O)C1)CCC 3652,c1(C(=O)NC2(C(=O)NCCNC(C=C(COC)C)=O)CC2)ccnc(C)n1 3653,c1(NCC(C2CC2)NC(C2(OC)CCCC2)=O)ncnc2ccccc12 3654,c1(C(=O)NCC(CNC(=O)C2=CCCS2)O)coc2c(Cl)cccc12 3655,Cc1nc2cccc(C(=O)NC3CC(NC(c4cc5sc(C)c(C)c5[nH]4)=O)C3)n2n1 3656,CCC(C)C(O)C(C)C(=O)NCC(C)(C)C(N1CCCC(F)(F)C1)=O 3657,N1(C(c2cc(CC)c(C)o2)=O)CCCC(CO)(NC(C2(SCC)CC2)=O)C1 3658,c1(C(N(CC(C)(C)CNC(=O)Cc2nncn2C)C)=O)cnc2c(c1)ncn2C 3659,N1(C(C2CC(CC)C2)=O)CCN(C(c2ccc(Cl)nc2N)=O)C2CC12 3660,C1(c2n(CCOCC)nnn2)(NCc2nc(C)c(C)o2)CCC(F)CC1 3661,Cc1cc(C)c(C(=O)N(CCNC(c2cncc(O)c2)=O)C(C)C)cc1C 3662,C1(NC(c2n(CC)ccc2)=O)CN(C(=O)C=CC2CCCO2)CC2(CCC2)C1 3663,N1(CC)CCCC1C(=O)NC(C)CCCNC(=O)CCc1cc[nH]n1 3664,c1(C(C(=O)NCCCC)N(CC(c2cccc(Br)c2)C)C)ccc(Br)c(Cl)c1F 3665,N1(C(C(CC)C(C)C)=O)CC2CCCC(NC(C3CCCS(=O)(=O)C3)=O)C2C1 3666,c1(C(=O)NCC(COC)NC(c2c[nH]nc2C)=O)ccc2n[nH]cc2c1Cl 3667,n1(CC)nccc1C=CC(=O)NC1CN(C(=O)CCc2cccc(O)c2)CC1F 3668,c1(C(=O)NCC2CC(OC)CN2C(=O)C(C)C2CCCC2)c(Cl)c(C)nn1C 3669,N1(C(=O)NC(C)CCC#N)CCC(CCc2ccc(O)cc2)CC1 3670,C(=O)(C(O)CCS(C)=O)NC1CC(CCNC(CCCCOC)=O)C1 3671,N1(C(CN(C)C(c2ccco2)=O)=O)CCN(C(C2CCCS2)=O)CC1 3672,c1(C(N(C2CCCC(NC(c3cc(C)oc3C)=O)C2)C)=O)cnc2n1CCCC2 3673,N1(C(CCSCC)=O)CCC2CCCC12C(=O)N(CC(N1CCCC1)=O)C 3674,Cc1nn(C2CCC2)cc1C(=O)N(C)CCNC(=O)CCc1cccs1 3675,C(=O)(C(CNC(c1nc(Cl)cs1)=O)C(C)(C)C)NC1C(C=C)COC1 3676,N1(C(C2(CC)CC=CC2)C(=O)NC2CCOC2)CCC(C)(CN(C)C)C1 3677,Cc1ncccc1N(C(N1CCC(Cc2ccc(Br)cc2)C1)=O)CC1COC1 3678,C(=O)(C#CC1(C)CCCO1)NC(C1CC1C(=O)NC1(C)CCCC1(F)F)C 3679,CC1(C)OC(=O)CC1C(N1CCCC(C(=O)Nc2ccc(F)cc2)C1)=O 3680,N1(C(CC)=O)CCC(C)(C(=O)Nc2cnc(C(F)(F)F)nc2)C1 3681,C1(NC(C(CC)(C)O)=O)CN(C(=O)CCn2ccnc2C)CC(C)(C)C1 3682,N1(C(C(CC)OC)=O)CC2(CNC(c3ccc(C(N)=O)[nH]3)=O)CC1CO2 3683,c1(C(=O)OCC)ccccc1-c1ccc(C(C(=O)NC2CC2)N2CCCC2)o1 3684,C(=O)(C(C(=O)N1CC(=C(F)CNC(c2cc(C(C)(C)C)on2)=O)C1)OC)OCC 3685,N1(C(c2cc(C)n(C)c2C)=O)CC2CC(NC(=O)C(c3ccccc3)O)CC1C2 3686,C(=O)(CC1CCc2ccccc21)N1C(CNC(=O)C#CC2CCOCC2)CC1 3687,c1(C(N2C(CNC(c3cn(CC)nc3)=O)C=CC2)=O)cc2cc(Cl)cnc2o1 3688,CC1CCCN(C(=O)CCC2(NC(=O)C=C3CCC3)CCC2)C1CO 3689,N(C1CN(Cc2ccccc2)Cc2ccccc21)C(Cn1c(=O)ccc(C)n1)=O 3690,Cc1cc(F)cnc1C(c1nnnn1C1CCCCCC1)NC1CC(F)(F)C1 3691,C1(NC(CCC=C)=O)CC2C(NC(=O)C(C)(C)n3cnnn3)C2C1 3692,c1(N2CCC(NC(c3c(C)ccs3)=O)C(C)C2)nc2ccc(Br)cc2o1 3693,c1(C2(C(=O)N(CC=CCNC(C3NC(=O)C4CC34)=O)CCO)CCCC2)ncccc1F 3694,C1(C(F)(F)F)(C(=O)NCC(C)CNC(C2(C)CSC2)=O)CC(C)(C)C1 3695,Cn1ncc(C(=O)NCC(C)(C)OCC(=O)NCC2C(C)(C)C2(F)F)c1Cl 3696,n1(NC(=O)NCC2(O)C(SCC)CC2)ccc(Br)cc1=O 3697,CC(C)(C(=O)NC1(C)CN(C(=O)CCOCC(F)F)C1)c1cccnc1 3698,N1(C(C2(C#C)CC(=O)C2)=O)CCCC(CC(=O)NCC(C)C(=O)OC)CC1 3699,c1(OC)cc(OC)cc(OCC(=O)NCC(O)CN(c2cc(F)ccc2Cl)C)c1 3700,N1(C(C2(C)N(C(c3c(C)oc(C#N)c3)=O)CC=C2)=O)CCC(O)C(F)(F)C1 3701,C1(C(C(=O)OC)NCC=CC(=O)OCC)CS(=O)(=O)C1 3702,C(=O)(CCS(=O)(=O)N1CC(F)CC1C(=O)NCCN1CCNC1=O)OC 3703,O(NC(=O)C(C(C)NC(c1cn2ccccc2n1)=O)C(C)C)C(C(=O)OC)C 3704,CC(C)(C)C(C(=O)NC1CCN(C(C2CCCCNC2=O)=O)CC1)NC(N)=O 3705,N1(C(C=CC(C)NC(C=Cc2cc(C)no2)=O)=O)CC(CC2CC2)CC(C)(C)C1 3706,C(CCC(C)C)(C(=O)N1CCC(O)(CO)CC1)NC(C1(OC)CCOCC1)=O 3707,N1(C(C(CC)n2nccc2C)=O)CC2(CCC(CNC(=O)C3=COCCC3)O2)C1 3708,c1(CN2CCC(C(=O)Nc3cc(SC)n[nH]3)C2)ccc(O)nn1 3709,c1(C(CC(F)(F)F)=O)cc(O)c2c(C(N3CCCC(C4CCC4)C3)=O)cnn2c1 3710,c1(C(C)C(=O)NCC2CCN2C(C2CC(OC(C)(C)C)C2)=O)cc(F)cc(F)c1 3711,N#Cc1cc(CN2CC3C(C2)N3C(c2ccncc2O)=O)ccc1Cl 3712,N1(C(C23CCC(OC)C2C3)=O)CC2CCCC(C1)N2C(=O)CCc1cncs1 3713,c1(OCC)ccc(C)cc1NC(C1(F)CCCN(C(=O)CCC=C(C)C)C1)=O 3714,C=CCC(CNC(C1CC(C)(C)CN1C(=O)CCCCOC)=O)CC(C)C 3715,CC(CC(=O)N1CCCCC1C(N)=O)C(C)(C)NC(=O)Cn1cnnc1O 3716,C(=O)(CC(C)(CN(C)C)C(F)(F)F)N1CCC2CN(C(CCC(=O)NC)=O)C2C1 3717,N12CCN(CC1)C(=O)C2.c1(C(=O)NC(C)CCO)cnn(C)c1 3718,c1(CCC(=O)NC2(CNC(c3cc(C)nc(C)n3)=O)CC2)cc2ccccc2[nH]1 3719,c1(C(=O)NCC(C2CCOC2)NC(C=CC=CC)=O)ccc(OC)nc1C 3720,c1(C(=O)NC(C(=O)N(CCC(=O)OCC)C)c2ccco2)cc(CC)c[nH]1 3721,C=CCCN=C(NCc1cc(Cl)cn1C)NC1CCOC(c2nccn2C)C1 3722,C1(C(CC2N(CC#C[Si](C)(C)C)CCOC2)=O)CCOC2(CCC2)C1 3723,C=CC1CCN(C(C2(NC(C3CC4CC4C3)=O)CC(O)C2)=O)C1 3724,c1(OC)ccc(CNC(=O)NCC2CCCC(F)C2)nc1 3725,C(=O)(CC(C(F)(F)F)c1ccon1)NCCN(C)C(C1CCC(=O)NC1)=O 3726,Cc1nsc(N2CC3C(CNC(=O)CNC(=O)C(C)(C)C)C3C2)c1C#N 3727,N1(C(=O)COCCF)CCC(F)(C(N2CCC(F)(CO)C2)=O)CC1 3728,C1(CCNC(C(C)NC(C=CCOC)=O)=O)CCN(C)C1 3729,CC1CN(C)CC(C(=O)NC(C)C(N2CC(O)(CC(N)=O)C2)=O)O1 3730,CCC(CC)C(C(=O)N1CC(OC)CC1CNC(C1(C)CC1)=O)OC 3731,C12(NC(c3ncoc3C)CC)COC(CN(c3ccc(C(=O)OC)cn3)C)(C1)C2 3732,c1(CC)ccc(C)c(C(N2CC3(C2)CN(C(=O)C(c2ccc(Cl)s2)C)C3)=O)c1 3733,N1(C(c2c(OC)n(C)nc2C)=O)C2CCC1CN(C(C1CN(CC(C)C)C1)=O)C2 3734,c1(C(N2C(C)(CNC(c3cnc(Br)s3)=O)CCC2)=O)ccc2ocnc2n1 3735,C12(NC(C(CCSC)OC)=O)CC1CN(C(=O)C(c1ccccc1Cl)C)C2 3736,c1(C(N2C(CNC(C3(CC=C)COC3)=O)CC2)=O)cc(Br)cnc1O 3737,c1(CC)cnccc1C(N1CCC(CC)C1C(=O)NCc1ncn(C)n1)=O 3738,c1(C(=O)NCCCC2(NC(C3C(C)CCS3)=O)CC2)ccc(OC(F)(F)F)cc1 3739,c1(CC(=O)NCCC(C)CO)cccc(NC(=O)CC(C)n2ccnc2)c1 3740,c1(OC)ccc2nc(N3CCC4(CCC(CNC(=O)OC(C)(C)C)C4)C3)sc2c1 3741,CN1C2CCC1CC(=CC(=O)NCC1CCN(C(C3(CF)CC3)=O)CC1)C2 3742,c1(C(=O)NCC2CCC(C(N(CC=C)Cc3ccco3)=O)O2)c(C)noc1C 3743,c1(-n2cc(CN(CC)CC)nn2)ccc(C(F)(F)F)cc1.C(=O)C(C)O 3744,c1(C(N2CC(NC(=O)C3=COCC3)C3C2C3)=O)cc2n(n1)CCNS2(=O)=O 3745,CCC(C)(C)CC(=O)NC1(CO)CCN(C(c2csc3cncn23)=O)C1 3746,C1(CC(=O)N(C)CCC2CCCO2)COCCN1C(c1nocc1Cl)=O 3747,c1(C(N(C2CCN(C(=O)CCC3CCCC3)C2)CC)=O)ccc2nc(O)[nH]c2c1 3748,C1(C(N2CCN(CCOC)CC2)=O)C2C(CN1c1ncc(Br)c(SC)n1)C2(C)C 3749,c1(C(=O)NCC2(CNC(CCC(=O)OCC)=O)CC2)ccc(C)cc1OC 3750,C(=O)(C1CCc2c[nH]nc21)NCCC1(C)CCN(C(C(CCCC)O)=O)CC1 3751,C1(NC(=O)CN2CSCC2=O)CN(C(=O)C(F)=C2CCCC2)CCC1C(F)(F)F 3752,c1(C(N2CC(C)CCC2C)C(=O)NC(CC)C)ccc(F)c(C)c1F 3753,N1(C(C2CC(C)N(C)C2)=O)C2CCC(C(=O)NCC3CCC3(F)F)C1CC2 3754,C1(F)(C(=O)NCC2CCCC(CNC(C(C)NC(C)=O)=O)C2)CCC2(CC1)CC2 3755,c1(SC)ccc(OCC(=O)NC(C)CN(C)C(c2ccc(F)s2)=O)cc1 3756,c1(C(N(CCNC(=O)C(C)S(N)(=O)=O)CC)=O)c(OC)ccc(F)c1N 3757,C(C(CC(C)C)C(=O)NC1CN(C(=O)Cc2coc3ccccc23)CC1O)OC 3758,c1(OCC)cc(OC)cc(S(=O)(=O)NCC(c2ccncc2)OC)c1 3759,C#CCC1CC(=O)N1.C(=O)(CC(=O)OCCC(=C)C)OC(C)(C)C 3760,Cc1nn(C)c2nc(NC3CC4CC(C3)N(C(=O)CCC(N)=O)C4)c(C#N)cc12 3761,C1(C(=O)NCCC(CC)(F)F)CC2(CCN(C(=O)C(O)CC(C)(C)C)C2)C1 3762,CCCC(CC1CCCCC1)C(=O)NC1CCCC1NC(c1coc(C)c1)=O 3763,C1(NC(c2cn(CCNC(C(C(C)(F)F)F)=O)nc2)=O)CCn2nnnc2C1 3764,c1(C(N(CC(C)NC(=O)CC(C)C(=O)OC)CC)=O)ccc2ccnc(Cl)c2n1 3765,Cc1cc(C(=O)NC2CCC2NC(=O)C(C)N(C)C)ccc1O 3766,CC1(C)COC(CC(=O)NCC2(NC(=O)CC34CCCC3C4)CCCC2)CO1 3767,C1(NC(CC(c2cccs2)NC(C)=O)=O)(CN(C)C)CCN(C(=O)CO)C1 3768,c1(CC)cc(C(=O)NCC(CO)NC(c2cc(N)ccc2Cl)=O)c2c(c1)CCO2 3769,c1(OCC)cc(NC2CC3CCCC(C2)N3C(=O)CSC)ccc1[N+](=O)[O-] 3770,C1(C(N(CCOC)C2CC2)=O)CN(C(=O)C(C)C(F)F)CCO1 3771,Cc1ccc(C(C)NCCC(O)CC2(O)CCOCC2)cc1C#N 3772,C(c1cccc(F)c1)=C(C(=O)NC(C)CNC(=O)CC1(CN(C)C)CCCC1)F 3773,c1(C(=O)NCCC)ccc(C(=O)NCC(C)(C2CC2)NC(=O)CCC(C)C)cc1 3774,n1(CC(N2C3C(NC(=O)CC45CCCC4C5)C(C3)C2)=O)cnc2sccc2c1=O 3775,CC1CC2(CCN(c3ccnc(N(C)Cc4nn(C)cc4Br)n3)C2)CO1 3776,C1(C(=O)NC(C)Cc2ccccn2)C2CC1N(C(=O)Cc1ccns1)C2 3777,C(CCCCC1CC1)(c1n(CC=C)nnn1)Nc1cnn(CCC)c1 3778,N1(C(=O)Cc2ccco2)CC2CCCC(C1)N(Cc1ccc3nonc3c1)C2 3779,c1(C(=O)NCCN(C)C(C2(CO)CCOCC2)=O)sc2cccnc2c1Cl 3780,N1(C(C=CSC)=O)C2CCC1CC(C(N1CC3(COCCO3)C1)=O)C2 3781,c1(OC)cc(C(=O)NCCN(C(=O)CSCCC(C)C)CC2CC2)cnc1O 3782,c1(-c2cn(C(C(=O)N(CCOCC=C)CC)CSC)nn2)ccc(OC)cc1Br 3783,N1(C(c2ccn(C(C)(C)C)c2)C(=O)NC2(C)CC2)CCC2C(C(N)=O)C2C1 3784,C1(NC(CCCOC(C)=O)=O)C2CC3C1C3C2C(=O)NC1(C)CCCC1C 3785,C1(N(C)C)CCN(C)C(COC(c2cc(Br)ccc2OC(F)(F)F)=O)C1 3786,C1(CC(=O)NC(c2c(C)nccc2)C)CN(C(C2(N(C)C)CC2)=O)CC12CC2 3787,C=CCC(C(=O)NCC1CCC(C(=O)N(c2cccc(OC)c2)C)O1)OC 3788,CC(C)C(O)C(F)(F)C(=O)NC(C1CC(NC(c2ccncc2)=O)C1)C 3789,n1(C(C)C)ccc(C(=O)N(CC(O)CN(C(=O)CN(S(C)(=O)=O)C)C)C)n1 3790,C(N=c1[nH]c(N(C)Cc2ccc(Br)nc2)nc2c1CSC2)C1(OC)CCOCC1 3791,N1(C(C2N(C(C)=O)CCC2)=O)CCCCC1CCCNC(=O)CC1(CO)CC1 3792,CC1CN(C(C2C3CCOCC23)C(=O)NCC2CCOC2)CCS(=O)C1 3793,C1(CCC(C)(C)NC(C2CCCC2(C)C)=O)CCCCN1C(=O)CSC(F)(F)F 3794,C(=O)(C(C)CC(=O)N1CC2CC1C2NC(=O)Cc1ccc(Cl)c(Cl)c1)OC 3795,c1(C(=O)NCCCN2CCN(C(C3C(OC)CC3)=O)CC2)cccc(=S)n1O 3796,C1(C(C)NC(c2cnc(C3CCC3)s2)=O)CCCN(C(C2CNC(=O)N2)=O)C1 3797,N1(C(C(C(C)C)NC(CC(C)C)=O)=O)CCC2(CCN(C(=O)C(=O)N(C)C)C2)C1 3798,c1(C(=O)NC2C(OC)CN(C(=O)CCc3csc(=N)[nH]3)C2)cc(C)nc(C)n1 3799,CC(C)(C)C(CC(F)(F)F)NS(=O)(=O)Cc1ccc(F)cc1Br 3800,Cc1ccc(CCCNC(CC2CCC2)C2CC2)c(C)c1 3801,C(C)(C1=CCN(C)CC1)NC(C(c1ccccc1)NC(c1[nH]cc(C)c1)=O)=O 3802,c1(C(=O)NCC(C)CNC(c2n[nH]c3c2CCC3)=O)cc(O)nc(Br)c1 3803,C1(C(=O)NCCCN(C(=O)CSC(F)F)C)CC(=O)N(c2ccccc2F)C1 3804,CCC1CN(C2CCN(C(=O)C(C)n3cncn3)CCC2C)Cc2ccccc21 3805,c1(C(=O)NC2CCC(CCC(=O)NC(C#C)(C)CC)C2)cnc(C)n1C 3806,c1(C(=O)NCC2CCC(NC(C3CC(C)N(C)C3)=O)C2)cc(Cl)ccc1[N+](=O)[O-] 3807,c1(C(=O)NC(CNC(C2N(C)CCC2)=O)(C)C)ccc2c(=N)[nH]cnc2c1 3808,CC(=O)CCCC(=O)NCC12CC1CN(C(=O)COc1ccc(F)nc1)C2 3809,n1(CC)cc(C(N2CCOC(CCCNC(=O)C=C(C)C(C)(C)C)C2)=O)c(C)n1 3810,c1(NC(=O)Nc2c(SCC)cc(Br)cc2)ccc([N+](=O)[O-])cc1Cl 3811,c1(SC(C)C(=O)N(C)CC2CCN(C(=O)C=CCn3cncn3)C2)ccccn1 3812,c1(C(C)C(c2c(-n3cc(C4(N)CC4)nn3)ccs2)=O)cc(C2CCC2)nn1C 3813,CCC(C)(C)CCCC(=O)NC(CNC(c1cc[nH]c(=NC)c1)=O)(CC)CC 3814,c1(CC(=O)N(CC(=O)N(CCCO)CCO)CC#C)cncnc1 3815,c1(NC(=O)NC2C(OC)C2)ccc(SC2(C)CCC2)c([N+](=O)[O-])c1 3816,C1(C(N(C(CC(=O)NC(COC)C)(C)C)C)=O)CC2CC1CC2=O 3817,C(=O)(C1=CCCN(C(C2CC2C(=O)OCC)=O)C1)NC(CCC)(C)CC 3818,CC1CN(C(=O)CSCC(N)=O)CCC1CNC(c1ccnn1CC(F)F)=O 3819,c1(OC)cccc(C(=O)NCCC2CC(NC(=O)C(C)CS(C)=O)C2)c1C 3820,C#Cc1ccc(F)c(C(N2CCCC(CCNC(C3CCC(=O)C3)=O)C2)=O)c1 3821,N1(C(CCC(=O)N(C)C)=O)CC2CCC1CN2C(C1CC2CC2CO1)=O 3822,CN1CC=CCC1CCC(N1CCC(CC(=O)NCCc2ccon2)C1)=O 3823,N1(C(c2cncc(F)c2)=O)CCCC(C2CCCN(C(c3c[nH]nc3F)=O)C2)C1 3824,N1(CC(=O)Nc2c(OC)cccc2)CC(C)(C)C(O)C(C)(C)C1 3825,CC1CN(C(=O)CC2C=CCC2)C1C(=O)NCC(C)(C)CC1CC1 3826,C#Cc1ccc(C(=O)NC2CCN(C(C3NC(=O)CC3C)=O)CC2)cn1 3827,c1(C(=O)NC2CC(CCNC(C(N3CCSCC3)C)=O)C2)ccc2ccoc2c1 3828,c1(C(N2C3CCC(NC(=O)C=CBr)C(C3)C2)=O)cnc2n1CCCCC2 3829,N1(C(C(=O)OCC)c2cccs2)CCOC(C2CC2)CC1.C(CN)S 3830,c1(C(C)(C)C)cc(C(N2CCC(C)(NC(=O)Cc3ccoc3)C2)=O)ccc1O 3831,c1(OC)c(C(=O)N(CCCNC(=O)COC)C)ncnc1C 3832,C(=O)(C(C)COC)NC(C(=O)N(CCC)CC)c1cccs1 3833,c1(OC)ccc(F)cc1CC1CCCCC1C(N1CCCC(Cn2cccn2)C1)=O 3834,C1(C(=O)OC)CCC(C2CC2)N1C(c1cccc(N(C)C)c1)=O 3835,C12(CNC(C34CC(C)C3C4)=O)CC1CN(C(C1(CO)CC(C)(C)C1)=O)C2 3836,c1(C(N2CCC(F)(CNC(CCOCC#C)=O)C2)=O)cc2ccncc2s1 3837,N1(C(=O)NC(C2(N3CCOCC3)CC2)=O)CCCC(NC(C23CCCC2C3)=O)C1 3838,N1(C(C(=O)NCC)=O)CCC2(CCCN2C(=O)C(O)CC(C)(C)C)C1 3839,n1(CCC(N2CC(CCNC(C3C(C)(C(C)C)C3)=O)C2)=O)ccc2cccnc12 3840,CC(C)CC(F)C(=O)NC1(C2CN(C(=O)Cc3cc(-c4ccco4)on3)C2)CC1 3841,C1(NC(=O)CCc2cccnc2)CC2CC(NC(c3ccc(Cl)s3)=O)C2C1 3842,C=CCCC(C)NC(C1CCCC1CNC(C1CN(C)C1)=O)=O 3843,C1(CNC(C(COC)O)=O)C2CCCC1N(C(c1ccc(O)c(Cl)n1)=O)C2 3844,CC1(C)OCC2CC12C(N1CCN(CC(C)(C)NC(=O)CC2=CCCC2)CC1)=O 3845,Cc1nc(CNC(C2CCOC2C(C)C)=O)sc1CNC(=O)COCC1CC1 3846,c1(CN(C)CC2CN(C(c3c(C)cco3)=O)C2)ccc(Br)c(C)c1 3847,C(=O)(CS(=O)C(F)(F)F)NC(CNC(c1c(CC)ocn1)=O)C1CCC1 3848,CC#CCC(C(=O)Nc1ccc(CC)nc1)NC(=O)CCn1cncn1 3849,CCCCCC(O)C(=O)N1CCC2CC12C(=O)NCc1nnnn1CC 3850,N1(C(C(C=CC)O)=O)CC(NC(C2CC(OCc3ccccc3)C2)=O)CC1(C)C 3851,C(=O)(C(C(=O)NC(C)(C)C(C)NC(c1occc1CN(C)C)=O)OC)OCC 3852,c1(C(=O)NCC2(C)CCC(NC(COCCOC)=O)C2)cc([N+](=O)[O-])ccc1N 3853,C1(CC(=O)NCC(C2CCCOC2)OC)CCCNC12CC2 3854,C1(CC=C)(NC(C2CCS(=O)(=O)C2)=O)CCN(C(C2CCCNS2(=O)=O)=O)CC1 3855,Cc1cc(C)c(C(=O)NCc2ccccc2C)c(Cl)n1.N12CCC(C1)NC2=O 3856,CC1(C)OC(=O)NC1CC1CCC(C(N2CCC(C(c3ccccc3)=O)CC2)=O)CC1 3857,c1(SC)cccc(Br)c1CC(=O)NC(C)CCn1cncn1 3858,Cc1ocnc1CC(=O)N(CC(=O)N(CC(F)F)C)C1CCC1 3859,N1(c2nc(C(=O)OC)c(C)s2)CCC(C)C(NC(c2cn(C3CCC3)nn2)=O)C1 3860,CC(C)C(C)CC(=O)NCC1(C)CCCN1C(=O)CCc1ccc(C2CC2C)o1 3861,C1(C(C)C(=O)NCC(=O)N(CCCO)C2CC2)CCC(=O)N1 3862,N1(C(CC2CN(C(c3c(CC)ccs3)=O)C2)=O)CCCCC1C1(COC)CC1 3863,CC(C)C(CCS(C)(=O)=O)NCC(=C1CCNCC1)F 3864,c1(OCC(=O)NCCCN(C(CC(=C=C)C)=O)C)ccc(C)cc1CC 3865,C1(C(=O)NCC(CC)(C)NC(=O)Cc2cc(C)cs2)CCc2ccccc2C1 3866,C12(C(=O)NCCCC(C)(C)OC)CC(CN(C(c3nnccc3C)=O)C1)C2 3867,C1(CNC(COCCC)=O)CC2(CC2)CN1C(c1cn(C2CCOC2)cn1)=O 3868,Cc1ccccc1OCc1nc(-c2ccc(C(F)F)cc2)nn1Cc1cccs1 3869,c1(C(=O)NCC(C)N(C(c2scc(C)c2Cl)=O)C)cc(O)nc(Cl)c1 3870,C=CC(C)(CC)C(=O)N(CCCNC(c1ccc(C(=O)OC)nc1)=O)CCO 3871,c1(NC(C2CC(F)CN2C(c2ccc(I)cc2)=O)=O)ccnc(-n2cccc2)c1 3872,C12(CNC(c3cc(C)no3)=O)CCC1CCN2C(c1ccc(O)c(F)c1)=O 3873,C(=O)(CCCCN=[N+]=[N-])N1C(C(=O)NC(CC=C)C(=O)OC)CC1C 3874,C1(CCC)(C(=O)NCC(c2cccc(Cl)c2)NC(c2ccco2)=O)CCNC1=O 3875,Nc1cccnc1C(=O)NCC1CCCCC1C(=O)NCc1ncc(CO)[nH]1 3876,C(=O)(CC(C)C(F)F)NC1C(C(NOC(CC)CC)=O)CC1 3877,C=CCC(CNC(C1(CC=C)CCCC1)=O)NC(C1(c2cc[nH]n2)CCC1)=O 3878,C1(NC(Cc2nn(C)nc2Br)=O)CN(C(C2CCCN2C=O)=O)CCC1CO 3879,C(CC(C(=O)N(CCC(=O)NCCc1ccccc1O)CC1CC1)OC)OC 3880,c1(C(=O)NCC2(C#N)CCC2)c(NC(C2CC(O)CN2)=O)sc2c1CCCC2 3881,C=CCC(C)(CO)CN=c1ccnc(N2CCC(COc3ccccc3)C2)[nH]1 3882,c1(CC)cccc(C(=O)N(CCNC(=O)CCc2ccn(C)n2)C2CC2)c1 3883,C#CC1CCCN(C(C2COC3CN(C(=O)CC(=O)N(C)C)CC23)=O)CC1 3884,N1(C(C(COCC)C)=O)CCSCC1CCNC(=O)Cc1ccnn1C1CC1 3885,C1(NC(C2(OC)CC2)=O)CC(O)CN(C(c2cnc(C3CCC3)s2)=O)C1 3886,C1(COCC(=O)NCC2CC(NC(c3cc(Cl)no3)=O)C2)CCCCO1 3887,Cc1nsc(NC(C2CCN(C(=O)CCC3CC3(C)C)CC2)C)c1C#N 3888,N1(C(C2CN(C)CC2C(F)(F)F)=O)CCCC(NC(C2(CF)CCC2)=O)CC1 3889,N1(CC(C)NC(=O)CS(=O)(=O)N(C)C)CCN(C(C2C=CCS2)=O)CC1 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3927,C1(=O)C(OC)CCN1.C(C(CCO)c1ccncc1)OC 3928,N1(C(C(c2ccncc2)C)=O)CCC(O)(CCNC(=O)Cc2n[nH]c(=N)s2)CC1 3929,CC(N=c1[nH]c2c(c(=NCCn3ccnn3)[nH]1)CCCCC2)c1ccns1 3930,O=C(CN=c1cc(F)nc(-c2ccccc2)[nH]1)C1CC2(C1)CC(F)(F)C2 3931,C1(NC(C(C)(C)N(C)C)=O)CCCCCN(C(c2c[nH]nc2C(F)(F)F)=O)C1 3932,C=Cc1cc(C(=O)N(CC(N2CCC(C(=O)NC)C2)=O)CC)cc(F)c1 3933,c1(C(N2CC(CCC)N(C(c3ns[nH]c3=O)=O)CC2)=O)c(F)ccc(F)c1F 3934,c1(OC)ccc(F)c(CC(=O)NC2CC(OC)CN(C(=O)CSC(F)(F)F)C2)c1 3935,N1(C(C(C)C(F)F)=O)CCCN(C(=O)CC23CCC(CC2)OC3)C(CO)C1 3936,C1(C(c2ccccc2)C)CCN(C(=O)CSc2ccc(F)cc2)CC1O 3937,C=CCCC(O)CNC(=O)CC(O)CNC(c1nonc1C)=O 3938,C1(NC(C(Cn2cncn2)NC(COCCCCC)=O)=O)CCCC2(CCC2)C1 3939,c1(-n2ccc(C(=O)NC3CC3C(=O)NCC3(O)CCCC3)n2)ccc(F)cc1 3940,C1(C(=O)NCC(C2CCCCC2)C)CCN2CCCC2C1 3941,N1(C(C(C)C2CCCO2)=O)CCC(CCCNC(c2ncc[nH]c2=O)=O)CC1 3942,C1(C(=O)NCc2c(C)nn[nH]2)CC2(CCN(C(C3CC(=O)OC3(C)C)=O)C2)C1 3943,N1(C(c2ccc(C(C)=O)nn2)=O)CC=C(CNC(c2cnn(C3CC3)c2)=O)CC1 3944,CC1(C)CC(NC(c2csc3nccn23)=O)CN1C(c1ccncc1Cl)=O 3945,c1(NC(CC(C2CC2)NC(CC(C=C)C)=O)=O)cc(O)c(C)cc1C 3946,CC1C(O)CCCN1C(c1ccc(CNC(=O)CCN2CCCCC2)s1)=O 3947,Cc1[nH]nc(C(=O)N(C2CC(NC(=O)Cn3ccccc3=O)C2)C)c1C 3948,C(=O)(CC(C)(C)CNC(C1CC1(C)C)=O)NC1(C(=O)OC)CC1 3949,c1(OC)cc(C(N2CCC(O)(CNC(=O)Cc3cccc(Cl)c3)C2)=O)ccn1 3950,N1(C(c2ncc(Cl)s2)C(=O)NC(C(=O)OC)CC(C)C)CCC2C(O)CCCC2C1 3951,CC(CN(C)C)CCC(=O)NC1(C(=O)NC2(CO)CC3CCC2C3)CCOCC1 3952,CCC(CCC(=O)Nc1cnsc1)NC(=O)C(C)(O)CCN(C)C 3953,N1(CC2C(C)(C)CCO2)C(=O)CN(CCOc2cc(Cl)cc(Cl)c2)C1=O 3954,C12(C(N3CC4C(NC(C5C(OC)C5)=O)(C4)C3)=O)C3C4C1C1C2C3C41CO 3955,c1(N2CC3CN(C(CN(C)C(N)=O)=O)CC3C2)nc2cc(F)cc(F)c2o1 3956,N1(C(C2(N(C)C)CC2)=O)CCCC(C2CCN(C(=O)C(O)c3ccsc3)C2)C1 3957,C(=O)(C(CC)(CC)C(=O)OC(C)(C)C)NC(CN(C(CCC(=C)Br)=O)CC)C 3958,c1(C(N(C(CNC(C2(C(=O)NC)CC2)=O)C2CC2)C)=O)ccc(O)nc1C 3959,c1(C(C)C)noc2ncc(C(=O)NC3CCC3CNC(c3ccccc3)=O)cc12 3960,C(N=c1[nH]cnc2cc(F)c(F)cc12)C1N(C(C2(C)CCOCC2)=O)CCCC1 3961,Cc1nccn1CCC(=O)NCC1CCC1N(C(C1(C2CCCCO2)CC1)=O)C1CC1 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3981,C1(CNC(CC(C(CC)C)O)=O)CC2(CCN(C(=O)Cc3cnc[nH]3)CC2)C1 3982,C(=O)(C(CCSC)NC(=O)C(Cl)Cl)NC1(CC=C)CC1 3983,N1(C(CN(C(=O)OC(C)(C)C)CC)=O)CCC(CC(C)NC(=O)C(F)CC)CC1 3984,CCCC(C(=O)N1CC(CC(C)NC(C2CCN(CC)C2)=O)C1)OCC 3985,C1(C)(C(N2CC=CC(NC(c3c(OC)nn(C)c3)=O)C2)=O)CC(O)CN1C 3986,CCC(CC1CCCC1)C(=O)NC1CN(C(c2sc(CO)nc2C)=O)C1 3987,c1(C(=O)NC2C(NC(C(c3cn(C)nc3)=O)=O)CCCC2)cnc2[nH]cnc2c1 3988,C1(NC(=O)Cc2cnccn2)CCCCN(C(C2CCC(F)(F)CO2)=O)C1 3989,C1(N(C)Cc2ccccc2)CN(CC2CNCC3(CCC3)O2)C2(CCC2)C1 3990,CCCC(C(=O)N(C)CC1(NC(c2ccc3nn[nH]c3n2)=O)CC1)S(N)(=O)=O 3991,CC(F)(F)C(C)(C)C(=O)NCC1CC2(CC2)CN1C(c1ccc(F)cc1C#N)=O 3992,c1(C(=O)NC2C(C)CN(C(c3ncccc3O)=O)CC2)nnn2c1CCCC2 3993,C1(C(N(CC(CC)O)C)=O)CC12CCN(C(c1n[nH]c3c1COC3)=O)CC2 3994,O=C1CCC(C(=O)NCCC2CCCCN2C(c2ccsc2C(F)F)=O)CN1 3995,c1(C(N2CCC(CC(=O)NCC(CSC)OC)C2)=O)[nH]c2ccc(F)cc2c1C 3996,CCCC(C(=O)N(C)CCN(C)C(c1cc(F)c(C(F)F)c(F)c1)=O)C(C)C 3997,c1(C(N2C(CNC(c3ccns3)=O)CC(OC)C2)=O)cc(Cl)c(F)cc1O 3998,Cc1ccc(OCCC(N2CC(NC(=O)CCC(C)C#N)C3(CC3)C2)=O)cc1C 3999,CCCC(C(=O)N1CC(NC(N)=O)C1)c1ccc(Cl)cc1 4000,c1(CNCC(CC)CC)cncc(Br)c1 4001,CC(C)(C)CC(O)CC(=O)NC1CCCC1C(=O)NC(CCO)C(F)(F)F 4002,CCCC(C(=O)N(CCC(=O)NC12CCC(CC1)C2)CC)N(C)C 4003,c1(C(C)OC)nc(C(=O)NC(CNC(c2cn(CCF)nn2)=O)CO)co1 4004,c1(C(N(C2CCCN(C(C(CC)O)=O)C2)C)=O)cc(O)cc(N)c1Cl 4005,N1(C(CC2C(OC)CC2)=O)CCN(C(=O)COCCN=[N+]=[N-])CC1C 4006,c1(C(=O)NC2C(CNC(c3n[nH]c(C)c3C)=O)C2)c(C)[nH]c2ncccc12 4007,CCCCC(CC)CC(=O)N1CC=CCC1C(N1CC(C2=NOCC2)C1)=O 4008,C1(NC(C23CC(C)C2C3)=O)CC(O)CN(C(=O)CCCCCN2CCSCC2)C1 4009,Cc1nnc(O)c(C(=O)NCCC2CSCCN2c2ncc(Br)cn2)c1C 4010,c1(CNC(C2(c3cnn(C)c3)CCCO2)C)nc2ccc(F)cc2s1 4011,c1(CC(N2CC(F)(CNC(C3CC4(CCCO4)C3)=O)C2)=O)n[nH]c2c1CCCC2 4012,c1(CNC(C2CCCN(C(=O)COC3CCCCC3)C2)=O)cc(Br)ncc1F 4013,c1(C2C(CNC3C4CN(C(=O)OC(C)(C)C)CC43)CCO2)ccc(Cl)c(F)c1 4014,N1(C(c2ccc(F)c(Cl)c2)=O)CC2CCC1CN2C(C1SC2C=CC1CC2)=O 4015,N1(C(C(C)=CCC)=O)CSCC1C(N1CC(CCN(C(=O)C2CC2)C2CC2)C1)=O 4016,C1(NC(CCC(C)OC)=O)CC2CN(C(C3(COC(C)C)CC3)=O)CC12 4017,Cc1ccc2ccccc2c1COC(c1sc(CC2CC2)nc1C)=O 4018,c1(N2CCC(N(CC#C)C(c3cscc3C)=O)CC2)ncnc2cc(Br)sc12 4019,C12COCCC1CC(=O)N1CCCC1CN2.C(=O)(C1=COCC1)N(C1CC1)CC 4020,c1(C(=O)NCCOCCNC(C2(SC(F)F)CC(O)C2)=O)cccc(C(F)(F)F)n1 4021,C1(N(C(c2ccoc2C2CC2)=O)C2CC2)C=CCN(C(=O)COCC(F)(F)F)C1 4022,C(=O)(C(O)CC(N)=O)NC(C)CCC(=O)N(C)Cc1cccc(O)c1 4023,CC1CCC2(CC1)CCC(CNCc1cccc(S(=O)(=O)N3CCCC3)c1)O2 4024,c1(C(=O)NCC2CCC(NC(C(CC)(C)CO)=O)C2)n[nH]c2cccc(OC)c12 4025,C1(C(=O)NC(CNC(C(CC)=CC)=O)(C)C2CC2)CCc2cn(C)nc2C1 4026,C1(NC(Cn2ccc(C)n2)=O)CCN(C(C2CC(n3cnnc3)C2)=O)CC1F 4027,C(=O)(CCC(=O)N(C)C)N(C(C)C)CCN(C)C(C1COC(C(F)F)C1)=O 4028,C1(O)(CCNC(CCCC)=O)CCCN(C(C2CC2c2cccc(OC)c2)=O)C1 4029,c1(C(=O)NCCNC(c2cn(CCNS(C)(=O)=O)nn2)=O)snc2ccccc12 4030,C(CCC(C(=O)Nc1ccccc1)N(C1CCN(C)CC1)C)=C(C)C 4031,C12(NC(c3csnn3)=O)CCCC1CN(C(=O)C=Cc1ccc[nH]1)C2 4032,C(=O)(CC(F)(F)C(F)F)N1CCCN(C(C(c2ccc(OC)cc2)C)=O)CC1 4033,N1(C(CC(CN(C)C)O)=O)CCC(CNC(=O)CC(C)(C)C)(COC)CC1 4034,c1(OC)noc(C)c1C(N1CCC(C(C)NC(=O)CC2(C)CCCCC2)C1)=O 4035,N1(C(CC=CC)C(=O)NC2CC(C(=O)OC)C2)CC2(C1)CC2(F)F 4036,C(=O)(C(CC(C)C)NC(c1cnc(Cl)n1C)=O)NCC1CC(CC)C1 4037,N1(C(C(CC=C)CC)=O)CCC(C2(NC(=O)COC3CC(F)(F)C3)CC2)CC1 4038,c1(C(N(C(C)CCNC(C2CCOC(C)C2)=O)C)=O)cc2c(cc1F)NCCC2 4039,c1(C(=O)NCC2C=CCN2C(C2CCCC2(F)F)=O)ccc2c(n1)OCCO2 4040,C1(O)(CN(C(CSC(C)C)=O)C)CCCN(C(=O)CCn2cccnc2=O)C1 4041,C1(NC(C(C)OCc2ccccc2)=O)CN(C(=O)C(=O)Nc2ncc[nH]2)CC1O 4042,c1(C(N(CCCCN(C(c2nccc(CC)c2)=O)C)C)=O)nc[nH]c2ncnc1-2 4043,c1(OC)ccc(Cl)c(C(=O)NCC23CC2CN(C(=O)CC(C)(C)OC)C3)c1 4044,N1(CCC(=O)N(CCC(=O)NC(CO)C2CC2)CC=C)CCOC1=O 4045,c1(C(N2CCCC(N(CCF)C(C3CC3C(F)F)=O)C2)=O)cnccc1Cl 4046,C1(CNC(c2n(CC)ccn2)=O)CCN(C(C2CSCN2C)=O)C12CCC2 4047,N1(C(C2(OC)CCCOC2)=O)CCN(C(=O)COCCC(C)C)C(C(N)=O)C1 4048,C(C(CC(F)(F)F)NC(=O)Cc1cc(F)cc(F)c1)NC(C(CC)NC(C)=O)=O 4049,C1(NC(CC2(C=C)CC2)=O)CCCC(NC(=O)C=CC)CC1 4050,C(CCC(C)C)(C(=O)NCCc1nccnc1C)NC(c1c(CC)c[nH]n1)=O 4051,C(=O)(C(C)(O)C(F)(F)F)Nc1ccc(C)c(Cl)c1.C=C1CNCC1 4052,c1(-c2nc(NC(N3CCC(CS(N)(=O)=O)C3)=O)sc2)nc2ccc(F)cc2s1 4053,Cc1ccc(C)n1CC(=O)NCC1CC1C(=O)NCC1(OCCO)CCCCC1 4054,C1(C(N(C(C)CN(C(=O)C(C2CC2)C2CC2)C)C)=O)CCCC2C1C2(F)F 4055,N1(Cc2onc(C(C)OC)n2)CCCC(CO)(NC(c2cn(C)nn2)=O)C1 4056,C(=O)(C(C1=CCC(C(C)C)CC1)N1CCOC(C(C)(C)O)C1)NCC=C 4057,C(N=c1ncc(C(C)(C)O)c[nH]1)C1CC(NC(C2CC(C(C)(C)C)C2)=O)C1 4058,N1(C(c2c(N)cc(F)cn2)=O)CC=C(CC(=O)NC2CC2O)CC1 4059,C1(NC(C2N(C(C3CC(CC)(CC)C3)=O)CC(OC)C2)=O)CC2(CC(OC)C2)C1 4060,C(CCC(C)(C)CO)NC(C(CNC(C1C(C)CCCC1)=O)(C)C)=O 4061,C1(NC(C(F)=CC)=O)CS(=O)(=O)CC1NC(=O)Cc1cnc(C(C)C)[nH]1 4062,C(C(C)(CO)CC=C)NC(c1cccc(CNC(C(CC#C)O)=O)n1)=O 4063,C1(C(N(C)CC2(N(C)C)CC2)=O)CN(C(=O)CCn2cnc(=N)[nH]2)CC1(F)F 4064,c1(NC2CC(C(=O)Nc3nc(C)c(C#N)nc3)C2)ncnc2sc(Br)cc12 4065,c1(C(COC(COC(CC(C)(C)C)=O)=O)OCC)cc(F)cc(Cl)c1.N1CCCC1 4066,N1(C(C(CCCOC)C)=O)CC2CCC(NC(=O)CC(O)C3CC3)CC2C1 4067,c1(-n2c(Cc3ccc(OC)cc3C(F)(F)F)nc(CO)n2)cccc2nsnc12 4068,N1(C(C2CC(C)C2)=O)CCOCC(F)(CNC(=O)Cc2cnn3c2CCCC3)C1 4069,c1(C(C(=O)N(CC(CC)NC(=O)CCc2ccc(C)s2)CC)C)ccccc1C 4070,C1(F)(C(=O)NCCCCNC(=O)CCC2NC(=O)NC2=O)CCS(=O)(=O)C1 4071,C1(C(=O)NCCCN(C(=O)C(C)(C)C)CC)CCCSC1 4072,N1(C(C=CC)=O)CC2CC(NC(=O)C(C3CCC3)OC)CC1C2 4073,N1(C(CCOCC(C)C)=O)CC(F)CC1CNC(=O)CCC1CCCCC1 4074,c1(C(=O)O)ccc(C(CO)N(CCN2CCCC2)C(C2(F)CC2)=O)cc1 4075,ClC1=CCCCC1(c1nnnn1-c1ccccc1)Nc1cccc(Br)c1 4076,N1(C(c2c(C#N)csc2)=O)CC2(CCC(CNC(C3CCCCNC3=O)=O)O2)C1 4077,C1(C(=O)NCCNC(C=C(C)C(C)C)=O)CCCOC1c1cn[nH]c1 4078,C12(NC(=O)Cc3ccoc3)CCCC1N(c1cc(Cl)nc(C(F)(F)F)n1)CC2 4079,O(N1CCC(N=c2cccc(S(=O)(=O)N3CC(C)OC(C)C3)[nH]2)CC1)CC 4080,c1(CC(C)C(N2CCCCC(NC(=O)CC3(O)CCC3)C2)=O)ccc(Cl)cc1Cl 4081,C1(C(N(C(C)CCNC(=O)CC(C)n2cccn2)C)=O)CCC(C)(C)CC1 4082,C12(COC)CC(NC(N3CCCC(C(C)(C)C(=O)O)C3)=O)(CO1)C2 4083,C1(CC(=O)N(CCCOCCN(C(CC2CC(C)C2)=O)C)C)OCCC1(C)C 4084,c1(C(N2CC3(CNC(CCC#C)=O)CC(F)(C2)C3)=O)cnc2c(C)nccn12 4085,c1(C(=O)NC(CNC(CCCCCSC)=O)CO)ccnc2c1CCCN2 4086,C1(CCNC(C2N(C(CC)=O)CSC2)=O)COCCN1C(=O)COC1CC1 4087,N1(C(C2C(NC(C3CCN(CC)C3)=O)C2(C)C)=O)C2CSCC1C2 4088,Cc1cc2c(Br)ccc(C(=O)NCCCNC(c3ccnc(O)c3)=O)c2o1 4089,c1(OC)ncc(NC(=O)CC(CNC(=O)C(N2CCNC2=O)C)OC)cn1 4090,Cc1cc(Br)cnc1C(=O)NC(CNC(=O)COC(F)(F)F)CO 4091,c1(C(=O)NC2CC(CNC(c3cc(CCOC)on3)=O)C2)nc(Cl)c(Cl)s1 4092,CC1=C(C)CC(C)(C(=O)N(CCNC(=O)CCC#N)C(C)C)CC1 4093,c1(C(=O)NCCN(C(=O)CC(=O)Nc2nccs2)CCOC)ncsc1C 4094,c1(N2CCC(CC=C)C2)ccc(S(=O)(=O)NC2COc3cc(F)ccc32)cc1Br 4095,Cc1nc(N2CCC3(NC(=O)C4=NNC(=O)CC4)CCCC23)c2ccsc2n1 4096,C1(C)(C(N2CCN(C(COCCCC#C)=O)CCC2)=O)CC(C(C)(C)C)=NO1 4097,C1(CNC(CCN(S(C)(=O)=O)C)=O)C2CN(C(c3cc(C4CC4)cs3)=O)CC12 4098,N1(C(c2nc(C(C)NC(CSCC#C)=O)oc2)=O)CCC2(CCCN2C)C1 4099,c1(CNC(CSCC)=O)ccccc1CNC(c1ccsc1CC)=O 4100,Cn1cnc(CNC(=O)CC2(NC(C3CCCCS3)=O)CCC2)n1 4101,c1(C(=O)NCC2CCCC(NC(C(CC)(C)CO)=O)C2)ccc2cnoc2c1 4102,Cc1ncc(N)cc1C(=O)N(CC(C)NC(=O)C(C)NC(=O)Nc1ccco1)C 4103,Cc1cnc(CNC(=O)CCCC2CN(C(=O)OC(C)(C)C)C2)o1 4104,Cc1nc(N2CCC(N(c3ncc(N(C)C)cn3)C)C2)c2ccccc2n1 4105,n1(CC)ncc(C)c1C(=O)NC1CN(C(c2csc(C)n2)=O)CC1OC 4106,c1(OC2CCN(C(C3CC3C(F)(F)F)=O)C2)cccc(F)c1 4107,c1(C(=O)NC2(C(=O)NC3CN(C(C)=O)C3)CC(O)C2)cn(C)cc1C 4108,C1(C(=O)OC)CCOC1C(=O)NCCCNC(=O)CC1(C)CCC1 4109,[N-]=[N+]=NC1CN(C(C2(F)CCN(C(c3n[nH]cc3Cl)=O)CC2)=O)CC1O 4110,Cc1ccc(C(N2C3CCC2C(NC(C2CC4CCC2C4)=O)C3)=O)cc1C 4111,C1(CN(C)C(c2ccc(O)nc2)=O)CCCN(C(C2(C(F)F)CCCCC2)=O)C1 4112,C(=O)(C1CC=Cc2ccccc21)N1C2CN(C(C#CC3(C)COC3)=O)C(C2)CC1 4113,Cc1nc(CNC(=O)CCc2cccn2C)oc1C(=O)NC(C)Cn1cnnc1 4114,N1(C(C2CC(C(C)C)OCC2)=O)CCC(F)(CNC(C2CN(C)C2)=O)CC1 4115,c1(OC)cc(OC)cc(C(N2CC(NC(c3cc(C#N)oc3C)=O)C(C)C2)=O)c1 4116,C1(NC(C2CCCO2)=O)CCN(C(C2CCC=CO2)=O)CC1 4117,Cc1ccc2c(C(=O)NCC3CC(NC(=O)C(=O)N(C)C)C3(C)C)csc2c1 4118,C(=O)(C#CC1(C(F)(F)F)CC1)N1CCC(OCCNC(C=C(CC)CC)=O)C1 4119,C=CCCC(C(=O)N1CCCC(O)(CC)C1)NC(=O)CN(C)CCOC 4120,C1(F)(C(=O)NCCN(C(=O)CC2CCOC2(C)C)CCC)C2CCCC12 4121,C1(C(=O)NC(C)C(C)NC(=O)C(C)(C)C2CC2)CCN(CC(F)F)CC1 4122,Cc1cocc1C(=O)NC1CCCC1CC(=O)NCC1(C)CC1(F)F 4123,N1(C(c2cc(OCC)n[nH]2)=O)CCC(C(=O)NCC2CC3(CCO2)CC3)C(O)C1 4124,Cc1nc(C(N2CC(OCC(N3CC(C)CC3C)=O)C2)=O)c(C)o1 4125,CC1CC(C(N2CC(NC(c3c(Cl)noc3C)=O)C2)=O)CC(C)C1 4126,N1(C(c2c(C)cc[nH]2)=O)CCC2(CC1)CC2NC(c1cc(I)ccc1C)=O 4127,N1(C(c2ccc(F)nc2)=O)CC2(CCN(Cc3ccc(-n4cncn4)cc3)C2)C1 4128,C1(CC(=O)N(C)Cc2c(C)nco2)CN(C(=O)Cc2ccc(F)cc2)CCC1C 4129,C(=O)(C(CO)C(F)(F)F)N1CC(C)CC(NC(CCc2cc(C)[nH]n2)=O)C1 4130,N1(C(C2ON=C(CC)C2)=O)CC2CC1CC2NC(=O)Cn1cc(CC)cn1 4131,c1(C(=O)NCC2(NC(C3N(CCC)CCC3)=O)CC2)nc2ccccc2s1 4132,C12(C(=O)NC3C(C(C)C)C3)CCCC1CCN2C(=O)CCCN(C)C 4133,c1(C(=O)OC)ccc2c(C(NC(=S)NC3COCC3O)=O)n[nH]c2c1 4134,C1(CNC(c2c(C)scc2)=O)CC2CCC1N2C(=O)C(F)(F)c1nccs1 4135,c1(N2CCC3(C(CNC(C4N(C(C)C)CCC4)=O)C3)CC2)ccnc2c1CCO2 4136,C1(CN(C(=O)CN2CC(C)(C)C2)CC)CCN(C(=O)C(C)CC#N)CC1 4137,C=C=CCCC(=O)NCC1CN(C(=O)C=C(CCC)CCC)C1 4138,Cc1ncc(Br)c(C(N2CCC(NC(=O)C3=CCCCO3)C(O)C2)=O)n1 4139,C1(S(C)(=O)=O)(C(=O)OC)CC(NCC2CC2C)C1 4140,C1(C(=O)NC2CC3CC4C(C3)C24)(CC)CCCN(C(=O)COC2CCC2)C1 4141,C1(NC(CCC#CC)=O)CCC2(CC1)CC2NC(C1CC(=O)N(C)C(=O)N1)=O 4142,c1(C(=O)NCC(C2CCC(F)(F)CC2)OCC)ccc2n[nH]cc2c1 4143,CC1CCC(NC(c2cc(O)cc(Br)c2)=O)CN1C(C1CCOCC1)=O 4144,S(=O)(=O)(c1cccc(=NCCc2cnccn2)[nH]1)N(C(C)CC#N)C 4145,C(CCCCCN=[N+]=[N-])NC(C1C(c2c(OC)cccc2)C1)=O 4146,CC1(C)CN(C(=O)CN2CCOC2=O)CCC1C(N1CCCN(CCO)CC1)=O 4147,N1(C(C(C)CN(C)C(C2CCCCC2O)=O)=O)CCOC2(CCC2)CC1 4148,C1(NC(c2c(C)sc(-c3ccco3)n2)=O)CN(C(c2ccoc2)=O)CC12CCC2 4149,c1(C(=O)NCCCNC(c2nnn(C)c2C(F)(F)F)=O)ccc(C2CC2)nc1O 4150,Cc1cc(C(=O)NC2(CO)CCN(C(C3OCCN(C)C3=O)=O)C2)nnc1C 4151,C1(NC(C2=C(C)CCC2)=O)COC2C(NC(c3cccc(O)n3)=O)COC12 4152,C1(NC(C2(C)CC(C)C2)=O)CN(C(=O)CCc2ccc(F)cc2F)CCC1CO 4153,N1(C(CC2CCN(C)C2)=O)CC2CCC(CNC(=O)Cc3cnc[nH]3)(C2)C1 4154,O=C(C1CCc2nccn21)N1CC(C2=NOCC2)C1 4155,Cc1c(CN2CCCC(C(=O)Nc3ncc(Br)nn3)C2)cccc1Cl 4156,c1(C(C)=O)[nH]ccc1C(=O)NCC1(NC(=O)CN2CCC(C)C2)CCC1 4157,C(=O)(C1=CC2(CCOCC2)C1)N1C(CCNC(=O)CC2CCC2)CCC1 4158,c1(CC)ccc(O)c(C(=O)NCC2CCN(C(=O)C(C3CCCOC3)OC)C2)c1 4159,C1(C(N2CCN(C(CC3CNC(=O)O3)=O)C(CCO)C2)=O)CC2C=CCC(C1)C2 4160,N1(C(c2ccc(C(C)F)cc2)=O)CCCCC(NC(C2(n3cnnn3)CC2)=O)C1 4161,C1(CC(=O)N(C2(COC)CCOC2)C2CC2)C(=O)NN=C1C.C12(CCC1)C(=O)N2 4162,c1(CCC)nc(C(=O)N(C2CCN(C(C3(C)CCCO3)=O)C2)CC)cs1 4163,c1(OC)cccc(OCCC(=O)NCCC2COCCN2C(=O)C(F)C(C)C)c1 4164,C1(O)(CCNC(c2cn(C3CCOCC3)nn2)=O)CN(C(C2CCC2(F)F)=O)C1 4165,C(=O)(C1=CS(=O)CCC1)N(CCN(C(=O)CN(C)S(=O)(=O)N(C)C)CC)CC 4166,c1(NC(C2(F)CCN(C(c3ccc(F)c(F)c3)=O)C2)=O)nc2ccc(Cl)cc2[nH]1 4167,n1(CC=C)cc(CNC(c2cn(CCNC(=O)C(F)C3CCOC3)nn2)=O)nn1 4168,c1(CNC(Cc2onc(CC)c2CC)=O)cc2ccccc2nc1NC 4169,c1(SC)ncc(Br)c(C(=O)NCC2CC(F)CN2C(=O)CCc2scnc2C)n1 4170,c1(CNC(C2C(C(=O)OC)C2)=O)ocnc1C(=O)NCC1CCOC1 4171,C1(CCCNC(c2c(C)c[nH]n2)=O)CCN(C(c2cccnc2C2CC2)=O)CC1 4172,C12(CCOCC1)n1cc(nn1)CNC2=O.c1(C(=O)OCC)cc(C(=O)OC)on1 4173,C(C(=O)N=S1(=O)CCC(OC)(OC)CC1)n1nc(C)c(NS(CC)(=O)=O)c1C(F)(F)F 4174,N1(C(C(C(CC)C)O)=O)CCC2CCCC12C(=O)NCC(F)(F)C(F)F 4175,Cn1nccc1C(CNC(=O)Cc1ncco1)NC(=O)C(F)C1CCCC1 4176,c1(SCC2(CC)CCOCC2)ccc2ccccc2c1.C1(CCC(F)F)C(=O)N1 4177,c1(OC)ccncc1NC(=O)C=C(C)CNC(=O)Cc1ccncc1Cl 4178,C1(CNC(C=CC=CC)=O)CCCN1C(=O)C(F)n1ccnc1 4179,N1(C(c2nncc(C)c2)=O)CCC(F)(F)C(CNC(C2CC=CCC2)=O)C1 4180,O=C(N=c1[nH]nc(Cl)cc1Br)C1CCCN1C(c1cn2c(Br)cccc2n1)=O 4181,C(=O)(CCC(C)OC)N1C(CNC(CCCOCC)=O)CCC1 4182,CCC(CC)CCCC(=O)C(C(CNC(C(COC(C)C)N)=O)O)=O 4183,c1(C(C(=O)NCCCN(C(C(C)(C)OC(C)=O)=O)C)C)ccc(C)cc1 4184,c1(C(c2cc(C(C3CCCN3CCNC(C)(C)C)(C)C)on2)SC)ccccc1Br 4185,C1(C(=O)NCCCOCC)CCCN(C(c2nc(C)sc2C)=O)CC1 4186,C1(CC)CCN(C(c2cc(F)c[nH]2)=O)C1CNC(=O)CCc1nncs1 4187,Cc1ccc(OCC(=O)N(C)CC2(CO)CC2)c(C)c1.C(=O)CCC=CC(C)C 4188,C=CC(CC)CC(=O)NC1C2CCN(C(=O)C(N3CCCC(C)C3)=O)CC12 4189,C(=O)(C(O)CCCNC(=O)C(C1CCOCC1)C)N1CCC(OC)C1C(C)C 4190,c1(C(N2CC3C(C(=O)NC(C(C)C)C)C3C2)=O)c[nH]c2ccccc12 4191,CCCC(C)(CC)C(=O)NCC1(NC(C2C=CCC2)=O)CCCCC1C 4192,C1(NC(c2c(CC)nc[nH]2)=O)COCCC1NC(C1(C2CCC2)CC1)=O 4193,c1(C2(C(=O)NC3CCC(CCNC(c4n(C)nnc4)=O)C3)CC2)ccc(Cl)cc1 4194,c1(C(=O)NC(C)C(C)NC(c2csc(O)n2)=O)ccc(-c2cnnn2C)cc1 4195,C(C(=O)NCc1cc(C2CC2)no1)(C(C)(C)C)NC(c1ccn(CCC)n1)=O 4196,C=CC1OCCC1NC(=O)COCC1CCCC1.N12CCCCC1C2=O.CC 4197,C1(NC(c2n[nH]cc2[N+](=O)[O-])=O)CCCCN(C(c2ccc(C3CC3)cc2)=O)C1 4198,N1(C(C(=O)NC(C)C)=O)CCC2CCC(NC(=O)CCCC(F)(F)F)C12 4199,C1(C(=O)NC(CC)(CNC(=O)C(C)CC2CCCO2)CC)CC2(COC(=O)N2)C1 4200,c1(-c2ccc(C(=O)NCCCCOC)nc2)cccc2nn(C)c(C)c12 4201,C1(NC(COCCCC)=O)CCCC1(C)C(C)NC(=O)CC1CC1C(F)(F)F 4202,C1(NC(=O)CCn2ccnc2)C2CCN(C(=O)C(F)(F)c3nccs3)CC12 4203,C1(CNC(CC(c2cccc(C(F)(F)F)c2)C)=O)CC(F)(F)CO1 4204,c1(NC2(c3n(CC=C)nnn3)CCN(C(C)C)C2)nc2ccc(OC)cc2n1C 4205,Cc1cc(C(=O)NC2(c3cn(-c4ccc(Br)cc4F)nn3)CCC2)cc(O)c1 4206,CC1CCn2c(C(=O)NCC3(NC(C4(CCF)CC4)=O)CCC3)cnc2C1 4207,c1(NC(=O)N(C2CCOC2C(F)(F)F)Cc2cccc(F)c2)cccc(Br)c1 4208,Cc1ccc(CC(N2CCC(C(C)C3CC3)C2)=O)cc1Cl.C(=O)(CC(=O)N)N 4209,N1(C(C(C)OC)=O)CCC(F)(C(=O)NCCc2cnn(C)c2C)C1 4210,S(=O)(=O)(c1cncc(C(=O)O)c1)NCC1(C(N)=O)CC(OC)(OC)C1 4211,c1(C(=O)NC2C(NC(C3C(C)OCC3)=O)COC2)cnccc1C(F)F 4212,c1(NC(c2cccc(O)n2)=O)cccc(NC(C2(N3CCOCC3)CC2)=O)c1 4213,c1(C(=O)NCC(C)(C)OCCNC(C(C(CC)O)C)=O)c([N+](=O)[O-])cnn1CC 4214,C1(CC(N2CCN(C(=O)NCc3n(C(C)C)ccn3)CC2)=O)CCC(F)(F)CC1 4215,CC1(C)CCN(C(=O)C(c2ccc(F)cc2)(C)F)C(C(=O)O)C1 4216,c1(C(=O)NCCCOCCNC(=O)Cn2cncn2)coc2c1C(O)CCC2 4217,c1(CCC)cc(C(=O)N(C2CCC(NC(C3CC4CC3C4)=O)C2)C)cc(O)n1 4218,N1(C(Cc2c(C)nccc2)=O)C(C(=O)NCC2(C)CSC(C)=N2)C2CC(O)C1C2 4219,N1(C(C(CC2CC2)OC)=O)CCC(C2CCN(C(=O)C(C)(C)CF)C2)CC1 4220,CCC(C(=O)NC(CNC(=O)CCC(=O)NC)CC(F)(F)F)C(C)(C)CC 4221,c1(C(=O)NC2C(OC)CN(C(=O)CC=C(C)C)C2)cc2occc2[nH]1 4222,c1(-c2ccc(CN(C(C)(C)C)CC)cc2)ccc(F)c(C)c1 4223,S(=O)(=O)(c1ccc(Br)cc1NCC(C(F)F)n1cccn1)NC(C)(C)COCCO 4224,Cc1ccc(C=C(C#N)C(=O)N2CC(=CCNC(=O)C(C)OCCOC)C2)cc1 4225,C(CC(C(=O)N1OC2CCC1CC2)NC(c1cncnc1CC)=O)=CC 4226,Cc1nc2cc(C(N3CC4CC3C4NC(C3COCCN3C)=O)=O)cnc2[nH]1 4227,c1(CC)ccc(C(=O)Nc2ccccc2COC)cc1.N12CCCC1(C)C2=O 4228,N1(C(C(C)Cc2ccccn2)=O)CCN(C(c2cc(Cl)ccc2O)=O)C(C)C1 4229,C1(C(=O)NCc2cccc(F)c2)CC12CCN(CC1N(C)CCN(C)C1)CC2 4230,CC(CC(F)F)C(=O)N1C(C(=O)NCC(=O)NCC2CC2)CCC1C 4231,N1(C(C(CC)(C)O)=O)CCN(C(=O)CCCCCNC(C)=O)CC(C)(C)C1 4232,c1(C(=O)NCC2CCN(C(C3CSCC(=O)N3)=O)C23CC3)cn2ccccc2n1 4233,N1(C(C)C=O)CCC2(CC(C(=O)OCF)=NO2)C1.c12ccc(cc1)n2F 4234,c1(C(=O)NCC(CNC(CN(C(=O)OC)C)=O)C(F)(F)F)cc(C)c(F)c(C)c1 4235,C1(C(=O)NC2C(C(N3CC(OCCOC)C3)=O)CCCC2)C2CCC(C2)C1C 4236,c1(CCNC(C(=O)Nc2c(C(C)(C)C)cccc2)=O)nc2ccccc2s1 4237,C(C(CC(=O)N1CCC(NC(C2(C)CCCCCCC2)=O)C1C)C(F)F)N(C)C 4238,c1(CC(=O)OCCCCC(C)=O)c[nH]c2ccc(F)cc12 4239,S(=O)(=O)(c1cc(F)ccc1C#N)NC1CCC(C)(C)CC1CN=c1[nH]ncs1 4240,C1(NC(CC2COCC(C)O2)=O)CC=C(C(=O)NCCC(C)N(C)C)C1 4241,c1(-c2cn(C(C)C(N3CCC(OCCO)C3)=O)nn2)c(Cl)cncc1Cl 4242,c1(C(N2C(CNC(CC(C)SC)=O)CC(O)C2)=O)cc2c(s1)CCOC2 4243,C(C)(C)(CC(F)C(=O)NC1CC(CO)C2CC12)NC(C(n1c(C)ccn1)C)=O 4244,c1(C(=O)NCC2(C)CC(NC(c3c(C)nc(O)cc3)=O)C2)ncnc2ccsc12 4245,S(=O)(=O)(c1ccc(N2CC=CC2)c2cnccc12)N1CC(C)(CC)OCC1 4246,C1(OC)CN(C(=O)CC2CC3CC3C2)CC1CC(C)=O.C1(=O)CCN1.C(=O)(C(=O)N)N 4247,N1(C(C(C)OCCOC)=O)CCCC(NC(c2ccnn2CCN(C)C)=O)C1 4248,Cc1ccc(C#N)c(NC(=O)CC2CN(Cc3ccc4c[nH]nc4c3)CCO2)c1 4249,CCC(CC(F)(F)F)C(=O)NC1(C)CC(NC(c2cc(Br)cn2C)=O)C1 4250,N(C(=NCCCCl)NC1CC2(CC2)C1)C(c1c(C)nns1)C 4251,C(C)(C(=O)NC1CCC(n2cc(-c3ccc(C)nc3)nn2)CC1)(C(C)C)OC 4252,c1(C(N(C(CN(C(CSCCC(C)C)=O)C)C)C)=O)csc(N=S(C)(C)=O)n1 4253,C1(C(=O)NC(c2occ(C(N(C3CCOC3)CC)=O)n2)C)CC(C)N(C)C1 4254,C1(CNC(CNC(c2ccc(SC)s2)=O)=O)CCCN(C)C1=O 4255,c1(SCCSCC(=O)NC2C(NC(=O)CC3(O)CCCOC3)C2)ccccc1Cl 4256,c1(OC)cccc(NC(c2cc(C)cs2)c2nnnn2-c2ccccc2C)c1 4257,C(=O)(CC(O)CC(C)C)NCC1CC(OC)CN1C(=O)C(C(C)C)NS(N)(=O)=O 4258,C(=O)(CC1=NNC(=O)C1)NC1CN(C(c2n(C)cnc2)=O)CC(O)C1 4259,Cc1cccc(F)c1C(N1CCN(Cc2ccc(Cl)cc2O)CC1C)=O 4260,N1(C(C(COC)C)=O)CCCC12CCN(C(C1CCC(=O)C1)=O)CC2 4261,c1(CC(C(=O)NC2(CC)CCOC2)C)ccc(OC)c(OC)c1 4262,c1(C(=O)NCC2(O)CCN(C(C3(C)CNC(=O)C3)=O)CC2)cnn2c1CCCC2 4263,[N-]=[N+]=NC1CCC2(C(=O)NC3CC(F)C3)CC12 4264,N1(C(C2C(C=C)C2)=O)CCC(C2(NC(=O)Cc3cc(C(F)(F)F)n[nH]3)CC2)CC1 4265,c1(OCC)nc(Br)cnc1C(N1C(CC(=O)NS(=O)(=O)CC(C)C)COCC1)=O 4266,C1(NC(c2ccc(CC)o2)=O)CCN(C(=O)C(O)Cn2cncn2)C1(C)C 4267,c1(C(=O)NCC(C23CCC(CC2)C3)NC(CC(=C)C)=O)ccc2ncncc2c1 4268,N1(C(CC)=O)CC2CC2(CNC(=O)C(N2CCNC2=O)C)C1 4269,N1(c2cc(C)nc(Cl)n2)CC2CC1CCC2NC(=O)CC(C)C1CCCCC1 4270,CC1CC(C(=O)N(C(C)CNC(C2CCC(C(C)(C)C)O2)=O)C)CC(C)C1 4271,C1(C(=O)NC2CC(CNC(CC=C(C)C)=O)C2)CCc2ccccc2O1 4272,C12(C(N(CCC(C(C)C)NC(c3ccc(F)cc3)=O)C)=O)COCC(C1)OC2 4273,N1(C(c2cn(C(C)C)nn2)=O)CCCC(C2(NC(c3cccc(O)n3)=O)CC2)C1 4274,C1(CNC(C(C)CC2CCC2)=O)COCCN(C(=O)C(C)(C)C2(O)CCOC2)C1 4275,N1(C(C(C)Cc2ccccc2)=O)CCSC(C(N2CCC(C3CC3)CC2)=O)C1.C 4276,n1(COC)nnc(C(=O)NCc2ccc(Cc3ccccc3F)cc2)c1C(=O)O 4277,N1(C(C=CC(=O)N(C)C)=O)CCC(C)(C)C1CC(=O)N(C)CC=CCO 4278,c1(C(=O)NC2(COC)CCN(C(=O)C(F)C3CCC3)C2)cc2c(cn1)OCCC2 4279,c1(C(=O)NCC(C)(C2CC2)NC(C(C)OCC#C)=O)cncc(F)c1C(F)(F)F 4280,CC1CN(C(=O)NC2CCC(CCCN3CCCC3)O2)CC1CN(C)C 4281,C(=O)(C(CC(C)(C)C)NC(=O)C1=C(C)OCCC1)N1CC(CCC)C(OC)C1 4282,c1(C(C(=O)NC(C(C)(C)NC(c2c(C)con2)=O)C)C)cc(F)cc(F)c1 4283,S(=O)(=O)(c1ccc(Cl)cc1)N1CCCC(C(C)C)(C(=O)NC(C)CO)C1 4284,c1(C(N2C(CNC(CSCCCC)=O)C(CC)CC2)=O)cc(F)cnc1O 4285,C1(C(C)NC(=O)CCCC2CCCO2)CCCCN1C(=O)CSCc1csc(C)n1 4286,CC1(C)C(NC(c2cc(Cl)ccc2Cl)=O)CC1N=c1ccnc(Cl)[nH]1 4287,C1(CNC(C(C)NC(c2ccco2)=O)=O)CC12CCN(C(=O)C=C1CCC1)CC2 4288,CCCC(O)C(=O)N(CC)CC1CCCN(C(=O)C(C)CC2CCCCC2)C1 4289,CC(C)CCN=C(NCC1(C)CCCO1)NC1CCCN(c2ccccc2Cl)C1 4290,N1(C(C2(C)C(C(=O)OC)C2)=O)CCC2(C1)CN(C(=O)C(C)(C)CC(C)=O)CCO2 4291,C1(NC(C(C)(C2CCC2)NC(C=CCC)=O)=O)CCCCNC1=O 4292,C(=O)(CCP(C)(C)=O)N(C(C)C)CCNC(C1(c2cccc(Cl)n2)CC1)=O 4293,N1(C(c2c(C)[nH]nc2Br)=O)CCN(C(=O)CC2CCCOC2)C(C(F)F)C1 4294,c1(C(=O)NCC(C)(C)O)cc(F)ncc1NC(C1(CCCCO)CC1)=O 4295,CC1(CCNC(=O)CC2(O)CCCC2)CCN(C(C2C3CCCC23)=O)C1 4296,N1(C(CNC(=O)NC(CC)COCC2CC2)C)CCCCC1 4297,c1(C(=O)NC2C(CC)CN(C(=O)C(CC3CC3)OC)C2)c(C)nn(C2CC2)c1Cl 4298,N1(C(C2(CC)CC2)=O)CC2CCC1C1CN(c3c([N+](=O)[O-])c(C)nn3CC)CC21 4299,c1(OC)cc(C)ccc1C(N1CC2CC1C2NC(c1ccnnc1)=O)=O 4300,c1(C(=O)NCCN(C(c2ccc(O)c(O)c2)=O)CC)cc2cc(C)ccc2s1 4301,CC1COCC(CC(N2CCCC2(C)C(=O)NC(c2nncs2)C)=O)O1 4302,C1(C(=O)NC(CNC(CC)=O)C)CCC2(CC1)CC(OC)C2 4303,c1(OC)cc(C(N2CCCCC2CN(C(=O)C(O)COC)C)=O)ccc1F 4304,c1(C(=O)NCC2CC(OC)CN2C(C2CC(OC)C2)=O)ccc2c(c1)N(C)CC2 4305,N1(C(C(CCC)OC)=O)CCN(C(=O)CCCS(N)(=O)=O)CC(CO)C1 4306,c1(C(N2CCN(C(C(C)CC3CC3)=O)CC2)=O)cccc2c1OC(C)C2 4307,n1(CCC(=O)NCC2CN(C(c3cnccc3Cl)=O)CCO2)cnc([N+](=O)[O-])c1 4308,c1(CN(C)C(C2CCN2C(C2CCCC2O)=O)=O)nccn1C 4309,c1(C(N(C)CC2CN(C(c3cn(CC)nn3)=O)C2)=O)ccncc1OC 4310,Cc1ccc(C(=O)NCCC2(NC(c3cccnc3N)=O)CCC2)c(Cl)c1 4311,N1(C(C23N(C(c4c(NC)cncc4)=O)CCC2C3)=O)CCC12CCCSC2 4312,Cc1n[nH]cc1CNC(c1c[nH]nc1-c1ccsc1)c1nnnn1C1CCCC1 4313,Cc1nc(NCCCC(C)C)cc(=NCc2ccc(C3CCCC3)cn2)[nH]1 4314,C(CCCCCCn1cc(-c2csc(C3CC3)n2)nn1)NC(C1C(C(=O)O)C1)=O 4315,N1(C(C=CC=CC)=O)CC2CCCCC2(CNC(c2cc(F)ccc2F)=O)C1 4316,N1(C(c2nc(CC)oc2C)=O)CC2CC1CN(C(C1(C(N)=O)CCC1)=O)C2 4317,C(=O)(CC(c1ccccc1)C1CC1)NCCC(C)N(C(CCNC(C)=O)=O)C 4318,N1(C(CN2CCC(C)CC2)=O)CCC(NC(C2CSC2)=O)C(c2ccccc2)C1 4319,N1(C(C2CCC(N(C)C)CC2)=O)CCCC2(NC(=O)C3=CCOCC3)CC2C1 4320,c1(CNC2CC(CC(N3CCC(F)C3)=O)C2)cnn(-c2ccccc2)c1 4321,N1(C(c2cc(C)c(F)cc2)=O)CC2CCN(Cc3ccc(C(F)F)cn3)CC2C1 4322,CCC(C)CCC(O)CC(=O)NC1(CNC(C2CCCN2CC(C)C)=O)CCC1 4323,C#Cc1cc(C(C(=O)NCC2CCOC2)N(CCC#N)CC2CC2)cc(Br)c1 4324,N1(C(c2c(NC)cccc2)=O)CCC(NC(c2ccc(C)nc2N)=O)C(C)(C)C1 4325,C(C(CC1CC1)C(=O)N1CCCC1CCCO)NC(CC1CC(=C)C1)=O 4326,c1(CCN(C)C)ccc(C(=O)NCC(CO)NC(c2occc2C2CC2)=O)cc1 4327,C1(OC)CCCC(C(=O)NC(CNC(C2CCOCC2)=O)C(C)C)C1 4328,c1(C(N2CC(C(N)=O)(CNC(C3C(C(=O)OC)C3)=O)C2)=O)c[nH]cc(F)c1=O 4329,CCCCCC=CC=CC(=O)NCCOCCNC(c1cc(C)no1)=O 4330,N1(C(C(C)(CO)OC)=O)CCC2(CC1)COC(CNC(c1coc(C)c1)=O)C2 4331,Cc1ccc(C(N2CCC(C(C)C(=O)NC3CCCCC3)C2)=O)cc1C#N 4332,C1(NC(=O)C=Cc2ccc(C(F)F)o2)CN(C(=O)C(Cl)=CCl)CC2(CCC2)C1 4333,C(CC(C)(C)C(=O)NC(C)CC(C)NC(C1(C)SCCCS1)=O)OC 4334,Cc1ccc(F)c(NC(C2CC(O)CN2Cc2ccc(OC(F)(F)F)cc2)=O)c1 4335,CC1CCC(C(=O)NCc2cscn2)N(C(C2CC2C(=O)OC)=O)C1 4336,CCCC(CNC(=O)C(C)(C)CC1CC1)C(=O)NCCC1CCCCC1O 4337,Cc1nn(C)cc1CC(=O)NCC1COCCN1C(C1CC(CC(F)(F)F)C1)=O 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4463,Cc1cc(NC2CCC(NC(C3CCCSS3)=O)CC2)n2nc(C)nc2n1 4464,N(C)(S(=O)(=O)NOC(C1(OCC)CC=CCC1)=O)CC#C 4465,CCC(CNC(=O)C=Cc1ccccc1C)(CC)C(=O)N1CCC(N(C)C)C1 4466,N1(C(C2CCCC2)=O)CCCC(N(CCO)CC2CCC(c3ccccc3)CC2)C1 4467,C(CCCC(C)(C)C(=O)NNC(=O)C1SCCC1C)NC(c1[nH]cc(CC)n1)=O 4468,c1(NCc2c(C)nn(C)c2Cl)[nH]c(=NC(C)CC2CCOC2)nc2c1ncn2C 4469,C(=O)(C(C(C)C)C1CCC1)NCC1(OC)CN(C(c2cnc(O)o2)=O)C1 4470,Cn1ncc(CNCc2ccccc2I)c1C1CCC1 4471,c1(C(=O)NC(C)C(N2CCN(C(c3cncnc3)=O)CC2)=O)ccc(F)cc1F 4472,C1(OC)(CNC(C2(F)CCN(C(=O)Cn3cnnc3)C2)=O)CCCCC1 4473,C1(O)(CNC(C(N2CCNC2=O)C)=O)CCCN(C(=O)CCc2cnn[nH]2)CC1 4474,C1(C(=O)NC2CC(F)(CNC(C(C)OCC)=O)C2)CC(C)(C)CC(C)(C)C1 4475,c1(C(=O)NCC(C)NC(CCC(C)c2ccccc2)=O)cc2ccccc2n1C 4476,C(=O)(C(C(C)(C)O)NC(=O)C(C)=C1CCCC1)NCCC(CC)C 4477,c12cnn(c1C)CC1CC(F)(C1)CNC2=O.CCCC(C1CCC1)NC(=O)C1CC1 4478,C1(C2CCN(C(=O)CNC(=O)C3CC3)C2)(NC(=O)CCOc2ccccc2Cl)CC1 4479,C1(NC(c2n(C)nnn2)CCC2(C)CC2)CCc2cc(C#N)ccc2C1 4480,CC(C)C(CCN(C)C(c1cnc(S)[nH]1)=O)NC(=O)C(C)C1CC1 4481,c1(OC)cncc(C(=O)NC23CC2CN(C(=O)CSCc2cccs2)C3)n1 4482,C(N=c1ccnc(N2CCCC3(CC2)CC3)[nH]1)c1c(C)n[nH]c1 4483,N1(C(C2OCCN(C)C2)=O)CCC2(CC1)CN(C(c1ncccc1N)=O)CCO2 4484,c1(NC(C)C)ccc(C(=O)NCC2CC2CNC(c2cc(Cl)no2)=O)cn1 4485,O=C(C1CCCc2ccnn21)NCC1CCN1C(c1cnc(O)n(C2CC2)c1=O)=O 4486,N1(C(CN(C(CC2CC(=C)C2)=O)CC2CC2)=O)CCOC(CC(N)=O)C1 4487,c1(CC(=O)NC2CN(C(CC(C)(C)C#N)=O)CC2(C)C)csc2c(F)cccc12 4488,CC1CCN(C(=O)CN2CC3CCC2C3)CC1CNC(c1cc(Cl)on1)=O 4489,C1(C)(C(=O)NC(C(C)C)C2CC2)C=CCN1C(c1ccsc1C#N)=O 4490,C1(C(=O)OC)CN(C(C2CN(Cc3nc(Br)cs3)CCS2)=O)CCC1O 4491,N1(C(c2cc(F)cs2)=O)CCCC(Cl)(O)CC1 4492,N#Cc1ccc(C(=O)NC2(C(N3CCC3CO)=O)CCSC2)s1 4493,CN1C2(CCN(c3ncnc(Cl)c3Br)CC2)C(NC(=O)C(O)C2CC2)CS1(=O)=O 4494,C1(CNC(Cc2cc(C)sc2)=O)COCCN1C(c1cnc(C2CCC2)s1)=O 4495,C(=O)(C(CCC(C)C)NC(c1cc[n+]([O-])cc1)=O)N1C(CC)CCC(C)C1 4496,N1(C(C(Cc2cc[nH]n2)NC(c2cnc(Cl)s2)=O)=O)CCC12CCCC2 4497,n1(CC(N2CCC(C(=O)NCCOC(c3onc(C)n3)C)C2)=O)nc(C)cc1C 4498,CCC(CN=C(NCCn1cnnn1)NC1CCC1)c1cccs1 4499,c1(CN(C(C(=O)OC)C2CC2)C)ncc(C(C)(C)C)o1 4500,N1(C(=O)OC(C)(C)C)CCC=CC1C(=O)NCC12CC3CC1C2C3 4501,Cn1nc(C(N2CC3CCC(C2)N(S(=O)(=O)CC#N)C3)=O)c2cc(Br)ccc12 4502,c1(CC(=O)NCC23C(CN(C(C(CC#C)O)=O)C2)CC3)ccc(F)cc1[N+](=O)[O-] 4503,C1(C2CCN(C(=O)NCC(=O)OC)C2)(NC(=O)COC(CC(C)(C)C)=O)CC1 4504,C1(CCC(=O)NCC(CO)NC(=O)CSc2nncn2C2CC2)CCC(O)CC1 4505,C1(CNC(C2C(=C)C2)=O)(COC)CCN(C(c2cc(C)ccc2N)=O)CC1 4506,N1(C(C(C(C)C)O)=O)CCC2(CCN(Cc3cc(-c4ccc(F)cc4)n[nH]3)C2)C1 4507,Cc1cnc(C(=O)N(C2CN(C(c3cnnc(O)c3)=O)CC2F)C)c(Br)c1 4508,N1(C(c2oc(C)c(CO)c2)=O)CCC2(C1)CN(C(C1CC13CCOCC3)=O)C2 4509,N1(C(c2c(SC)cn(C)n2)=O)CC(NC(C2(C(=O)OC)CC2)=O)CC(C)C1 4510,C(=O)(CCCC(=O)C(C)(C)C)N(CC(C)NC(C1(CF)CC1)=O)C 4511,c1(C(N(CCNC(C(C)P(C)(C)=O)=O)CC2CC2)=O)cnc2ncnc(O)c2c1 4512,N1(C(C2C(=C)C2)=O)CCCN(CCNC(C2CCCC(C(F)(F)F)O2)=O)CC1 4513,CCCC(CCCNC(C1CC1CF)=O)NC(c1ncccc1CC)=O 4514,C1(C2CCN(C(=O)C(F)CC3CCCCC3)CC2)(NC(C(CC)C)=O)CC1 4515,C1(C(N2CCC(C(F)F)(CNC(C3CN(C(C)C)C3)=O)C2)=O)CC2C(C1)C2(F)F 4516,C1(N=[N+]=[N-])(C(N(C(C#C)(C)C)C2CC2)=O)CCN(C(=O)CN2CCSCC2)C1 4517,c1(OC)cc(NC(C2CCN2C(=O)C(C)(C)n2ccnn2)=O)ccc1Cl 4518,c1(-c2cc(C(=O)NC3CN(C(c4cnn(CC(F)F)n4)=O)C3)n[nH]2)ccccc1O 4519,C(=O)(CCCC(C)NC(=O)CN1CCCCC1)NCC(C)C#N 4520,N1(C(C(C)(C)CCC#N)=O)CCN(C(=O)CCC2CCC(=O)NC2)CC(C)(F)C1 4521,Cc1cc(CC(=O)NCc2nc(C(=O)N(CC(C)O)C)co2)no1 4522,C(=O)(C1=CCCC1P(C)(C)=O)N(C)CC1CCN(C(c2c(C(C)C)con2)=O)C1 4523,C1(CC(=O)NCc2c(COC)cccc2)CCCN(C(=O)C(C)(C)O)CC1 4524,CC(N=c1cc(NCc2c(Br)cnn2C)nc(C(F)(F)F)[nH]1)c1nncn1C 4525,CC(C)C(C(=O)N(C)CCc1ccncc1)C(C)NC(=O)CC1CC(=O)C1 4526,C(=O)(CCN(OC)C(=O)C(C)N(C(=O)C(C)C#N)C1CC1)OC 4527,N1(C(CC#N)=O)CCC2(NC(c3ccc(-c4ccon4)cc3)=O)CCCC12 4528,CC1(C)OC(=O)CC1C(N1CCN(C(=O)Cc2ccc(Cl)s2)C(CF)C1)=O 4529,Cc1ccsc1CC(=O)N(C(c1ccccc1)CNC(C1(CC2CC2)CC1)=O)C 4530,c1(-c2c(C)ccnc2F)ccc2ccnc(NC(=O)C3=CCCCO3)c2c1 4531,c1(C(=O)NCC2C(CNC(c3c(C#N)nc[nH]3)=O)C2)cc2ccccc2o1 4532,n1(CC(=O)N(CC(C)NC(C2C3COCC23)=O)C)nc2n(c(=O)c1=O)CCC2 4533,C(=O)(CCCCCN(C)C(c1cn(C2CC2)nn1)=O)NCC(CCCC)O 4534,C1(NC(C(c2cncc(F)c2)C)=O)C2CC1CN(C(c1ccc([N+](=O)[O-])[nH]1)=O)C2 4535,N1(C(CC(C)C)=O)CCC(CNC(=O)C(O)CN2CCOCC2)C1(C)C 4536,c1(OC)nc(C(=O)NC2CCCCC2n2cc(C3(C)CCOC3)nn2)ncc1F 4537,N1(C(C(C)(O)CCc2ccccc2)=O)Cc2ccc(O)cc2C1 4538,C=CCC(C)C(=O)NC1CCCC(CNC(C2CCN(C(=O)C(C)C)CC2)=O)C1 4539,C(N=C(NC(C)C)N(C)Cc1ccc(Br)cc1)C1(COC)CCCO1 4540,c1(Cn2cc(CC3(C)CSC3)nn2)cc(Cl)ncc1Cl.N12CCCC(C1)C2 4541,C1(C)(NC(c2nc(C)sc2)=O)CCCCC1C(=O)NCCc1cscn1 4542,CCC(C#N)(CC)C(=O)N(C)CCC1CCCCN1C(=O)C1=C(C)CCOC1 4543,C(CC(C)(C)CC(=O)NCCCN(C(=O)CCCCc1cnn[nH]1)C(C)C)OC 4544,N1(C(c2cn(CCCC)nn2)=O)CCOCC(CNC(=O)C(O)C(C)CC)C1 4545,C12(C(=O)NCCC3CC(C(=O)NC(C(=O)OC)(C)C)C3)CCCC1C2(F)F 4546,C1(C(N2CCCC(n3cc(CCCCCO)nn3)C2)=O)CC12CCCC2 4547,N1(C(C=Cc2cnc(C)s2)=O)CC2CC(NC(c3cc(C#N)c[nH]3)=O)C1C2 4548,Cn1ncc2cccc(C(=O)N(C3CCC(NC(=O)C4=NOCC4)CC3)C)c12 4549,c1(NC(C2CC(F)(F)CO2)=O)cc(F)cc(I)c1 4550,n1(C(C)C)nncc1C(=O)NCC(C)NC(=O)C(C)(C)c1ccsc1 4551,C1(NC(=O)CCc2ncc(F)cn2)CCCC12CCN(C(c1ccc(Cl)cc1)=O)C2 4552,C(=O)(C1=C(C)OCCS1)N1CCCC(CCC(=O)NC(CC=C)CC(F)F)C1 4553,N1(C(C(CC)OC)=O)CCC2(C1)CN(C(=O)CC1CN3CCN1CC3)C2 4554,N1(C(CC(CC)OC)=O)CCN(C(=O)CCc2ccc(F)cc2F)C(C(C)C)C1 4555,N1(C(Cc2cn(C)nc2Cl)=O)CCCC(NC(=O)C(C)(C)n2cnnn2)CC1 4556,c1(NC(C2(C)CN(C(C3CC34CCC4)=O)C2)=O)ccc(O)c(N(C)C)c1 4557,Cc1sc(Cl)c(C(=O)NCC2(O)CC(CNC(=O)CCCC#N)C2)c1C 4558,N1(C(c2cc[nH]n2)=O)CC23CCCCC2(C1)CN(C(c1ccc(Br)o1)=O)C3 4559,Cc1ccc(C2(C(=O)NCC(C)(CO)NC(c3cc(Br)n[nH]3)=O)CC2)cc1 4560,C(=O)(C1=NOC2(CCC2)C1)N1CCN(C(C(C)=C(CC)C)=O)CC(O)C1 4561,C1(NC(c2nocc2Cl)=O)CCCC1CNC(C1(C(F)F)CCC1)=O 4562,C(=O)(C(C)(C)C1=CCN(C(=O)C(C2CCCCC2)F)C1)C(CCC=C)=O.N 4563,C(=O)(C1CCc2ccccc21)N(C(CCNC(CC(CC)C)=O)C)C 4564,c1(C2CC(NCC3(C)CCCS3)C2)cccc(Br)c1 4565,C1(NC(c2c(C)noc2)=O)C=CCCC1C(=O)NCC(F)(F)Cl 4566,C1(COC(Cc2c(C(=O)OC)csc2)=O)CCC(OC2CCCCC2)CC1 4567,CC1(C)CCN(C(=O)C(=O)NC2CC2)CC1CNC(C1CCC=CCCC1)=O 4568,c1(C(=O)NC(CNC(C(C(CC)O)C)=O)COC)cc2cnccc2[nH]1 4569,N1(C(C2CCN(C3CC4CCC3C4)CC2)=O)CCN2CCC1C2 4570,c1(NC(C2(C)CCN2C(C2CC2F)=O)=O)cncc(F)c1I 4571,C1(NC(C2CSCN2N2CC(C)(C#N)C2)=O)CN(C(c2cnsn2)=O)CCC1F 4572,c1(OC)ccc(Cl)c(C)c1C(=O)NC1CC(C)N(C(c2ccc(F)s2)=O)C1 4573,c1(OC(C)C)cc(C(=O)N(CC(C2CCCCC2)C)C(C)C)cc(F)c1F 4574,N1(C(N=c2[nH]nc(SCC)s2)=O)Cc2cccc(Br)c2C1 4575,N1(C(C#CC(C)C)=O)CC2(C1)CN(C(c1cnn3cc[nH]c13)=O)CC2CO 4576,C1(NC(c2cc(Cl)ncn2)=O)C2CN(C(=O)CCOc3ccccc3Cl)CC12 4577,C(=O)(CCN(CCCO)C)N(CC(F)(F)F)C(COC)C1CC1.C1C(=O)N1 4578,Cc1cccc(Br)c1C(=O)NC(C)C(=O)N(C)Cc1ccc(Cl)nc1 4579,c1(OCC)ccc(Cl)cc1C(=O)NCC12CCC(CC1)N2C(C12CC(O)C1C2)=O 4580,c1(C(N2CC(F)(CNC(C3CCCC(CC(F)(F)F)C3)=O)C2)=O)cccc(F)c1 4581,C(=O)(C(C)(CC)CCC(C)C)N(CCNC(C(CC)N(CC)CC)=O)C 4582,c1(C(N(CC(CN(C(=O)Cc2ccc(O)nc2)C)O)C)=O)ccc2oncc2c1 4583,Cc1sncc1C(N1CCCC1C1CCN(C(c2csc(C(N)=O)n2)=O)C1)=O 4584,N1(C(C2CC3CN(C(CCOCCOC)=O)CC2C3)=O)CCc2ccccc2C1 4585,N1(C(CC2(C(=C)F)CCC2)=O)CCCCCC1CNC(=O)C(O)C(C)CC 4586,c1(C(=O)NC2CN(C(C3C(C(C)C)CCO3)=O)CC2(C)C)cnc2ccoc2c1 4587,N1(C(C(C)C#N)=O)CCC(C(F)(F)F)CC1CNC(c1ccnc(S)c1)=O 4588,C1(C(=O)NC2CN(C(c3n(C(C)C)cnc3)=O)C(C)C2)CC(O)C12CCC2 4589,CCC(C)CCCCC(=O)NC(C1(O)CN(C(c2cc(F)cc(Cl)c2N)=O)C1)C 4590,c1(C(c2n(CC)nnn2)Nc2ccc(CCO)cc2)cccc(C(=O)OC)n1 4591,CCC(F)(F)C(C)(C)C(=O)NCC1CCN(C(c2nn(C)cc2[N+](=O)[O-])=O)CC1 4592,C1(C(N2C(C)CC(CCNC(C3CCC3)=O)CC2)=O)CCc2nn[nH]c2C1 4593,N1(C(C=C(CCC)C)=O)CCC2(CCC(NC(=O)C(O)C(C)OC)CC2)CC1 4594,c1(C(=O)NC2CN(C(CC=C=C)=O)CC(O)C2)nc2ccc(Br)cn2c1Cl 4595,N#Cc1cccc(NC(=O)CC2CCCC2NC(c2ccc(Cl)s2)=O)c1F 4596,C(CCCC(C(=O)NC1CCN(C(=O)OC(C)(C)C)C1)Nc1csnc1OC)OC 4597,C1(c2n(C)ncc2)CN(C(=O)CNS(=O)(=O)C2CC2)CCN1C(=O)CO 4598,c1(CC(N2CCC(CNC(c3c(C)scn3)=O)CC2)=O)ccc2n[nH]cc2c1 4599,C1(CC(=O)N(C)Cc2c(C)nsc2)CCC(NC(=O)CC2CCN(C)C2=O)CC1 4600,c1(C(=O)NC(C2CN(C(c3ccc(CCC)cc3)=O)C2)C)ccc2cnnn2c1 4601,c1(C(=O)NCC2CCN(CC)C2)sc(F)cc1C.C1(C)CCC(=O)N1 4602,Cc1nc([N+](=O)[O-])cn1CCC(=O)NCC1CN(C(=O)CC(C)O)CC12COC2 4603,C(=O)(C(O)C(C)(C)C)N1CC(C)C(n2cc(C3CCCCC3O)nn2)C1 4604,C1(NC(c2c(C)nccc2Cl)=O)CN(C(C2CCCC2(F)F)=O)C2(CCCC2)C1 4605,C1(NC(c2n(C)c(C#N)cc2)=O)CCCC12CN(C(=O)Cc1cnccn1)C2 4606,C(CC(C)C)(C(=O)NCCCNC(N)=O)NC(C1N(CC)CC1)=O 4607,C1(NC(=O)CN2CCC(c3ccccc3Cl)C2)CCC(N)C(F)(F)CC1 4608,C(CC(C(=O)NCCC(C)(O)CC)NC(=O)C(C)=CCC)=CC 4609,C(=O)(C(C)(C)C(F)F)N1CCC(C2N(C(C3C(C)C3)=O)CCCC2)C1 4610,C(C(=O)N1CCCO1)NC(C1(N(C(=O)C=Cc2nccs2)C2CC2)CCC1)=O 4611,C1(C(=O)NCCN(C(=O)C(O)Cn2cncn2)C)(CC)CCCCO1 4612,CCCC(C(=O)OC)N(C)N1CC(C)CCC1C(=O)OC 4613,N1(C(CC2(CN(C)C)CCC2)=O)CCC(CNC(c2cncc(N)n2)=O)C(C)C1 4614,c1(C(N(CCN(C(=O)CC2CCOC2)CC)CCN(C)C)=O)nonc1N 4615,c1(C(=O)OC)ccc2c(c1)nc(CNC(=O)NC1CC(CC(=O)O)C1)n2C 4616,C(CCNC(=O)C(CO)OC)(C(=O)NOCCCCCC1CC1)OC 4617,c1(C(C(=O)NC2CC(C)(NC(C3CC=CCO3)=O)C2)O)ccc(F)c(F)c1 4618,c1(SCCc2c(C)n[nH]c2)ccc(-c2nc(NC(=O)OC(C)(C)C)cs2)cc1 4619,C=C1CNC(=O)CCCN(CC2CC2)C(c2ccccc2)C(=O)NCC1.N(C)OC 4620,c1(C(N2CCC(CC)C2C(=O)N(C(C)CCC(C)C)C)=O)n[nH]c2ccccc12 4621,N1(C(C(C(C)(C)C)O)=O)CC(C2CCCCN(C(C3(n4cccn4)CC3)=O)C2)C1 4622,c1(SCC)cc(C(N2CCCC(NC(=O)Cc3[nH]cnc3C)C2)=O)ccn1 4623,C12CN(CC1CC(F)(F)F)C2=O.c1(COCC(=O)OC2CCOC2)ccccc1 4624,N1(C(c2csc([N+](=O)[O-])c2)=O)CC2CC1CC2NC(C12CC3CC1C2C3)=O 4625,c1(C(=O)NC2CCN(CCNC(C(CC)(C)O)=O)CC2)cc(C)cc(O)c1 4626,C(=O)(C1=CCCC1)NC(C1CN(C(C23CCCCC2C3)=O)C1)C 4627,c1(C(=O)NCC(CCC)C(=O)N2CCC2CN=[N+]=[N-])cc2cccnn2c1 4628,C1(=CC(=O)NCC(CN(C(C(C)(C)OC(C)C)=O)C)O)C2CC3CC(C2)CC1C3 4629,N1(Cc2cccc(CC(=O)OC)c2)CCCN(C(C2CCCSC2)=O)CC1 4630,C1(CC)(CC)CN(C(c2ccc(OC)nn2)C(=O)NCCOC)CCS1=O 4631,C12(NC(c3cc4sccc4[nH]3)=O)CCN(C(=O)C3=CCCSC3)CC1C2 4632,C1(C(=O)NC(C2CC(NC(=O)C(N3C(=O)CCC3=O)C)C2)C)CC(=O)C1(C)C 4633,c1(NC(C2CC(CNC(c3c(NCC)scn3)=O)OC2)=O)ccc(Cl)cc1 4634,CCS(=O)(=O)CCCNC(=O)NCC(N1CCCCC1)(C)C 4635,C1(OC)CC(NCc2nc(-c3ccccc3Cl)no2)C12CCC2 4636,c1(C(N2CC3N(C(C(C(C)C)SCC)=O)CC(C3)C2)=O)cn2cc(Cl)cnc2n1 4637,CC1CCCCC1CC(=O)NCC(C)(C)OCCNC(=O)Cc1cnccn1 4638,C1(NC(CN2CCN(C)CC2)=O)CN(C(c2ccc(CF)cc2)=O)CC1C1CC1 4639,c1(OC)ccc2c(Cl)nc(COC3CCN(C(C)C(=O)OC)C3)nc2c1 4640,c1(CC)c(N2CCC(CNC(C3(OC)CCCC3)=O)C2)nc(C)nc1Cl 4641,N1(c2ncc(CCC)cn2)CCCC2C1CCN2C(c1csc(Br)c1)=O 4642,N1(C(CCC#CC)=O)CCCC(N(C(=O)COc2ccccc2)C)CC1 4643,c1(C(N2CCC(N(C(=O)CCN3CCC(O)CC3)C)C2)=O)ccnc2c1CCO2 4644,CCCCCC(F)C(=O)C12CC(C)(C1)CNC(=O)C(C)(CO)NCC2 4645,C1(NC(C=CC=CCC)=O)CN(C(c2cn(C)nc2Cl)=O)C2(CCOC2)C1 4646,Cc1cc(C(=O)NCC(C2CC2)N(C(=O)CC(O)C(C)C)C)cnc1C(F)(F)F 4647,c1(C(N2C(C)CC(NC(COCCC=C)=O)C2)=O)nccc2ncncc12 4648,C1(CNC(c2c(N)cc(Br)cn2)=O)CCC2(CCC2)C1NC(c1cnco1)=O 4649,C#CC1CC2(CC(C(N3CC(NC(c4cc(C)ccc4OC)=O)C3)=O)C2)C1 4650,C1(C(=O)OCC(c2cc(CSc3nnc(O)o3)on2)=O)CCC(=O)NC1 4651,Cc1cccc(C(O)C(=O)NCc2cn(CC(C)(C)[N+](=O)[O-])nn2)c1 4652,CC(C)CC(O)C(=O)NC1CN(C(=O)C=Cc2ccc(SC(F)F)cc2)CC1C 4653,C(=O)(C1=CCN(C(C2COCCO2)=O)C1)NC(C(C)C)C1CCC1 4654,C(=O)(C(F)(CNC(C1CC(CF)C1)=O)C(C)C)N1CCC(C=C)CC1 4655,N(C1CCOc2ccc(Cl)cc21)CCC(C)Sc1nnco1 4656,N1(Cc2c(C)cc(Br)cc2)CCN(C(=O)Cc2ccc(Cl)s2)C(C#N)C1 4657,c1(C(N2CC(CC)N(C(=O)C(C)OCCOC)CC2)=O)cc(C)c(OC)c(Cl)c1 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4728,C1(NC(C2CC(S(C)(=O)=O)C2)=O)COC2CN(C(C3CC4C(C3)C4(F)F)=O)CC12 4729,c1(OC)nc(C)cc(=NCC(C)(C)C2CCCCN2C(C2CC(C)(C)C2)=O)[nH]1 4730,c1(CNC(C2N(C(c3cncc(CC)c3)=O)CCC2CC)=O)cccc(C)c1O 4731,Cc1cc(C)nc(N(C2(C#N)CCNC2)C(C2CCC(=O)NC2)=O)n1 4732,N(C1CCOc2c(F)cc(F)cc21)C(C(C)Oc1ccccc1CC(=O)O)=O 4733,c1(C(N(C2CCCCN(C(C(C)S(N)(=O)=O)=O)C2)C)=O)csc(=NC2CC2)[nH]1 4734,N1(CC#CCOC)CCCCC(NC(c2cnnn2-c2ccccc2)=O)C1 4735,C1(C(N(CC(=O)NC)C)=O)(OC)CCN(C(C2C(C)C2C)=O)C1 4736,S(=O)(=O)(c1cccc(Cl)n1)SCCC(N1CC(c2ccccc2)(O)C1)=O 4737,C1(C(=O)NC2C(CNC(c3cncc(N)n3)=O)CCC2)CC2CCC1C21CC1 4738,n1(CCOC)ncc(NC2(c3nnnn3CCCF)CCOC2)c1C 4739,CC(CCCC(=O)NC1CN(C(=O)Cc2ccccc2)C1)c1ccccc1 4740,Cc1cc(C(N2CCOC(C(=O)N(CCCc3ccccc3)C)C2)=O)nn1C 4741,C(=O)(C1=C(C2CCOCC2)N(C)C(=S)NC1c1cccc([N+](=O)[O-])c1C)OCC 4742,C1(C)(COC)CC(NC(c2ccoc2)=O)CN1C(=O)Cc1ccc(Cl)c(OC)c1 4743,n1(CC=C)c(N(CC(C)CC)C)nnc1C1COc2ccccc21 4744,CC1CC(C(=O)N2CC(C)(NC(C3CC(Cc4ccccc4)=NO3)=O)C2)=NO1 4745,C1(NC(c2c(COC)ncs2)=O)C2CC1N(C(=O)CCc1cccc(Cl)c1)C2C 4746,C(CN=c1cc(F)nc[nH]1)(c1ccccc1F)NC(C(C(C)C)C)=O 4747,N1(C(c2ccsc2Br)C(=O)NC2CC2)CCC2(C1)OCCO2 4748,C1(CCC)CN(C(=O)C(=O)NCC2CC(CC)C2)C1 4749,c1(C(N2C3CN(C(C(CC)C(C)O)=O)C(C3)C2)=O)onc2ccccc12 4750,C12(NC(C=C(C)C(C)(C)C)=O)CCC(F)(F)CC1CN(C(=O)C(C)(C)CF)C2 4751,C1(CC)CCC(C(=O)N(C2CCC(NC(c3cccc(N(C)C)n3)=O)C2)C)CC1 4752,c1(C(NC(NC(C#C)CC2CC2)=NC)C)ccc(CC)cc1 4753,C(=O)(C1CCc2cc(F)ccc21)NC1(C)CN(c2cc(C(C)C)nc(Cl)n2)C1 4754,c1(CC(N2CC(NC(c3n[nH]cc3Br)=O)C3C2C3)=O)cccc(F)c1O 4755,c1(C(N2C(CN(C(=O)C(C)(C)CF)C)CC(F)C2)=O)ccc2c(c1O)CCCC2 4756,C1(CC(=O)NC(C#C)C(C)C)N(C(=O)CC2CCC(C)CO2)CCC1(C)C 4757,N1(C(C2(C)CCOC2)=O)CC(O)CC1CNC(C1CC2(CCC2)C1)=O 4758,CC(C)(C)CCCC(=O)NC1CCC(NC(=O)CCc2c[nH]c3ccccc23)C1 4759,C1(CNC(C2CC23CCOC3)=O)CC2(CC2)CN1C(=O)C(F)n1cccn1 4760,CC1(C(=O)NCCC2(O)CN(C(C3CC4(CCCC4)C3)=O)C2)CCCC1(F)F 4761,N1(C(c2n[nH]c(C)c2C)=O)CC(NC(=O)C(CC2CC2)CC2CC2)CCC1C 4762,Cc1cc(C(N2CCC(N(CCO)C(C3(C)CCC(=O)NC3)=O)C2)=O)ccc1F 4763,N1(C(C(SC)SC)=O)CCCCC(N(C)C(c2ccc(F)c(F)c2)=O)C1 4764,c1(OC)cc(C(=O)NCCNC(c2c(C3CC3)cnn2C)=O)cc2cn(C)nc12 4765,C(CC(C)CCNC(=O)C=CCOC(C)(C)C)NC(c1cn(CC=C)nn1)=O 4766,N1(C(CC2C(C)(C)C(NC(=O)COC3CCOCC3)C2)=O)CCC2(CC1)CSC2 4767,C1(C(=O)NC(C)CN(C)C(C2CCCS2)=O)CCCN(c2ccccn2)C1 4768,c1(CC)ccc(C(=O)NCCCC(C)NC(=O)C(O)Cc2ccsc2)cc1C#N 4769,N1(C(CC(C)O)=O)CCCCC1CNC(=O)CSc1nncn1C1CC1 4770,C1(C(=O)NCC(=O)N(C(C)CO)CC2CCC2)C2CN(C)CC12 4771,c1(OC)cccc2[nH]cc(CC(=O)N(C)CC3(O)CCC(F)(F)CC3)c12 4772,C(=O)(C(F)(F)C(F)(F)F)N1CCC(N(C)C(c2cc(C(F)(F)F)ccc2Cl)=O)C1 4773,C=CCC(C)(C)CNC(C1CCN(C(=O)CP(C)(C)=O)C1)=O 4774,CC1C(NC(=O)Cc2cnsc2)CC2CCC1N2C(=O)C(F)(F)c1cnccn1 4775,N1(C(c2c(C)n[nH]c2)=O)CCN(C(=O)C=CCCC=C(C)C)CC1c1ccnn1C 4776,N1(C(C(C)Cc2cnc[nH]2)=O)CC2CCCCC2(NC(c2cc(Cl)ccn2)=O)C1 4777,c1(C(N2CCOCC2C2CCOC2)C(=O)NCCOC)cc(OC)cc(SC)c1 4778,c1(CCC)c[nH]ccc1=NC(=O)Cc1ccc2nonc2c1 4779,C(c1cc(Cl)ccc1Cl)=CC(N1CCN(C(C(C)(C)OC)=O)CC1)=O 4780,C1(C(N2CCC(C(C)Nc3nc(C)nc(O)c3C)C2)=O)CCC2(CC1)CC2(F)F 4781,c1(CNC(C(CO)NC(C2C(C)CC2)=O)=O)ccc2c(c1)CC2 4782,c1(C(=O)NC(C)CNC(=O)C=CCOCC(F)(F)F)snc(Cl)c1Cl 4783,C(CN=c1cc(NCc2ccc(C(N)=O)o2)nc[nH]1)(C1CC1)OC 4784,CCC(C)CC(=O)C(=O)NC(C1CC1C(=O)NCc1ccc(C2CC2)o1)C 4785,C1(CNC(C(C(C)(C)C)SC)=O)CC12CCN(C(c1cscc1C(N)=O)=O)CC2 4786,c1(N(C(C)=O)C)ccccc1C(=O)N(CC(C)CNC(C1CC(N=[N+]=[N-])C1)=O)C 4787,CCCCC(C)CCC(=O)NC1COCC1NC(c1cc(Br)cs1)=O 4788,CC1CN(C(=O)OC(C)(C)C)CCC1N(C)CC1(O)CCOCC1 4789,C(c1ccc(Cl)c([N+](=O)[O-])c1)=CC(=O)NC1CC2(CNC2)C1 4790,C(CCCCCNC(C1(OC(C)C)CCC1)=O)N(C(c1c(C)snn1)=O)C.CCO 4791,c1(C(=O)NCC2N(C(C(C)SCc3ccccc3)=O)CCC2)c(O)cccc1F 4792,C(c1cncn1C)=CC(=O)N(CCC(=O)N(CC(O)C1CCC1)C)CC 4793,N1(C(C(COC)NC(C)=O)=O)CCC2CC1CN2C(c1cccc(C)n1)=O 4794,c1(SC)ccc(C=CC(=O)NCC2CC(NC(=O)COc3ccsn3)C2)s1 4795,C1(N(C(C2(C)COC2)=O)Cc2nccs2)CCC2(CCNC2)CC1 4796,CC(C)C(CC(=O)NCC(F)CNC(c1cocn1)=O)c1ccccc1 4797,CCC(CC)CC(F)C(=O)NC1CC2CC1N(C(c1cscc1C(N)=O)=O)C2 4798,Cc1cccc(CCNC(=O)NCC(c2ccc(C(C)C)cc2)(C)C)c1F 4799,C1(CNC(COCC)=O)CN(C(C2(CC(C)=O)CC2)=O)CCC1(C)C 4800,C1(C(N(CC(C)(C)OC)C)=O)CN(C(C2CC(C)=NO2)=O)CC12CC2 4801,c1(CNC(CC2(CC)CCC2)=O)cc(C(=O)N(C2CC2(C)C)C)on1 4802,CCCCC(C(=O)NCc1ocnc1CC)NC(c1cc(C)c(C)[nH]1)=O 4803,c1(CCNC(C=CC(C)(C)NC(c2cc(O)cs2)=O)=O)ccncc1F 4804,C1(CNC(C(CCC)C)=O)CCC(C)N(c2nccc(C)c2C(=O)OC)C1 4805,CCC(C)CC(CO)N(C(=O)CC(CC)N(C)C(C1CC(=O)N(C)C1)=O)C 4806,Cc1nc2ccc(-n3cc(C4CCN4C(c4cccc(O)c4)=O)nn3)cc2o1 4807,C(=O)(C(F)CCC(C)C)N1C(C)CCC(NC(C2C=C(C)CS2)=O)C1 4808,Cc1n[nH]c(=NC2CCCC(NC(c3cnn(C4CCCC4)c3C)=O)C2)s1 4809,c1(C(=O)NCCC2N(C(C=C(CCN(C)C)Cl)=O)CCC2)c[nH]cc(C)c1=O 4810,N1(CC)CCCCC1C(N1CC=CC(NC(C2(C(F)(F)F)CCCC2)=O)C1)=O 4811,C1(NC(CCCC(C)C)=O)CCN(C(c2cc(O)cc(=O)o2)=O)C12CCCC2 4812,C1(CNC(=O)CSCc2cscn2)CC12CCN(C(C13CCC(CO1)C3)=O)CC2 4813,c1(C(N2CCOC(C3CCOCC3)C2)=O)[nH]cc2c1CCC2 4814,c1(C(=O)NCC2C3CN(C(CCCCCC)=O)CC32)cc2n(n1)C(C)CCC2 4815,c1(OC)c(C(=O)NC(CNC(C2CC2(Cl)Cl)=O)C(C)(C)C)cnn1C 4816,c1(C(=O)NC(C)CC)cc(N(CC=C)CC)c(OC)cc1-c1ccc(CC)cc1 4817,N1(C(CC(C)SC)=O)CCC(F)(F)C(CNC(C2(C)CC(C)(C)C2)=O)C1 4818,C1(NC(C2CC3CCC2C3)=O)CC2CCC1N(C(=O)CN1CCCS1(=O)=O)C2 4819,C1(CNC(C(CC)N(C)C)=O)CC2COCC2N1C(c1cc2cccnc2s1)=O 4820,C12(C(N3CC(O)(C(=O)OCC)C3)=O)CC1CN(C(=O)CC1CCCO1)C2 4821,N1(C(C(CCCC)O)=O)CC(NC(c2ccncc2)=O)C2CCCC2C1 4822,c1(C(=O)NCC2C(C)(C)N(c3ncc(Br)cn3)CC2)ccnc2c1CCC2 4823,c1(C(N2CCOCC(NC(CC3(CSC)CC3)=O)C2)=O)cc(O)cc(C#N)c1 4824,C=CCC(C(=O)NC(C1CC(NC(C2(CC)CCCCO2)=O)C1)C)C(C)C 4825,C(CC(C)C(=O)NCC1CCN1C(=O)CN1CCCCC1)OC 4826,C1(NC)CCCC(C(=O)NCCNc2ccc(F)cn2)C1 4827,CC1CN(C(c2c(F)cccc2Cl)=O)CCN1C(c1ccc(C2CC2)cc1)=O 4828,N1(C(c2ncn(C)n2)=O)CCOCC12COCCN(C(C1C3CCCOC13)=O)C2 4829,N1(C(c2scc(C)c2C)=O)CC2(CCN(C(=O)C(F)C3CC3)C2)C1 4830,C(CCCCC(=O)NC1CCC(CCC(=O)N(CC(C)C(=O)OC)C)C1)SC 4831,c1(C(=O)NCC(C)=CC(=O)NCCN(CC(C)(C)C)C)cnc(C)c(C)c1 4832,CC(C(F)(F)C(F)(F)F)NC(=O)Nc1ccc(Br)c(Cl)c1F 4833,S(=O)(=O)(c1ccc(CNC(N)=O)cc1)N(C(C)C)Cc1ccc(CC(=O)O)cc1 4834,c1(NC)ncc(C(=O)N(C2CCCCC2)CCNC(C2(CO)COC2)=O)cc1Cl 4835,CC(C)CCCCCC(=O)NCCOC1CN(C(=O)Cc2ccsc2)C1 4836,n1(CC(=O)NC(C(=O)NC(c2cnn(C)c2)CC)c2ccco2)[nH]cnc1=N 4837,C(=O)(CCCC(N)=O)N(C(C)CCNC(=O)CC1CN(C)C1)C 4838,CCCCCC(O)C(=O)N(CC(N1CC(c2ncc[nH]2)C1)=O)CC1CC1 4839,c1(OCC)cc(NCc2ccc(CNC(c3cscc3Cl)=O)cc2)ncn1 4840,c1(N(C)CC)nc(NCC2CCC3(CCCC3)C2)c2ncn(CC)c2n1 4841,C(=O)(C(O)C(F)(F)F)NCC(C)(C)NC(c1cn(C)c(O)n1)=O 4842,c1(N2CCOCC(=C)C2)nc2c(c(=NCC3CCC(O)C3)[nH]1)CCC2 4843,c1(C(c2c(C)nc(C)[nH]2)Sc2ccccc2)c(C#N)c(C2CC2)nn1C 4844,C1(n2c(C(CCC=C)NCc3cc(Br)no3)nnn2)CCC(F)(F)CC1 4845,c1(C(N2CCCC(NS(CC)(=O)=O)CC2)C)cccc2ccccc12 4846,N1(C(c2ccc(C)s2)=O)CC2CCN(C(C3CCCCNC3=O)=O)C2C1 4847,C1(C(=O)OC)CC2CC(NC(=O)Cc3cnc(C)nc3O)C2C1 4848,C(CC(=O)NCC1C=CC(NC(=O)C(C)CC2CCC2)C1)(OCC)OCC 4849,N1(C(C2C(C)(C)CO2)=O)CC2CC(NC(=O)CCCC3CCCCC3)CC2C1 4850,c1(C(=O)NCCN(C(c2[nH]nnc2C(F)F)=O)CC)cnc(O)n1CC 4851,N1(C(CCOCCCOC)=O)CCC(C(F)F)(CNC(c2sccc2Cl)=O)C1 4852,Cc1noc(N)c1C(N1CCC(NC(c2csc(C(F)(F)F)c2)=O)C1)=O 4853,c1(C(=O)NCCN(C(=O)Cc2ccc(Oc3ccccc3)cn2)C)nnc(S)n1C 4854,N1(C(CC(CC)C2CC2)=O)CC(NC(C2CCN(OC)CC2)=O)C2(CC2)C1 4855,CC1CC(c2cn(-c3ccncc3)nn2)CCN1CC(N1CCC(O)CC1)=O 4856,C1(C(=O)NC2CN(C(Cc3cccc(C#N)c3)=O)CC2O)CCc2ncnn2C1 4857,S(=O)(=O)(c1cccc(N(C)CC2CC2)n1)NC(C)Cc1ccc2ccccc2c1 4858,C12(OC)CN(C(=O)Cc3ccnc(C(=O)OC(C)(C)C)c3)CC(C(=O)O)(C1)C2 4859,N1(C(C(CC)(C)OC)=O)CCCC(CC)(NC(=O)CCc2ccccc2F)C1 4860,CC(C)S(=O)c1ccc(C(N2CCCN(C(=O)C(C)(C)C(N)=O)CCC2)=O)cc1 4861,C1(C(=O)NC(CC)CN(C(=O)Cc2nonc2C)C)CCC(=O)NC1 4862,n1(CCC(=O)NCCC2COCCN2C(=O)Cn2ncnn2)cc([N+](=O)[O-])cn1 4863,c1(C(=O)OC)ccc(S(=O)(=O)NC2CCCN(C(c3cncs3)=O)C2)cc1 4864,C1(CC=C)(NC(=O)CC(O)CCSC)CCCN(C(c2ccc(C=CC)o2)=O)C1 4865,N1(C(C(CC=CC)CC)=O)CC2OCC(NC(=O)CCCCCCC)C2C1 4866,c1(C(N2CCC(C(N(CCOC)C(C)C)=O)CC2)=O)nccc2ccccc12 4867,N1(C(C=CC(CC)=CC)=O)CC2CC(CNC(c3ccc(Cl)o3)=O)C2C1 4868,c1(NC(C2(CC)CN(C(=O)CC3CCCCO3)C2)=O)cccc2cccnc12 4869,c1(SCC(C2CCCOC2)OCC)ccnc(OC)c1I 4870,c1(C(N2CCCCC(NC(C(CC)(F)F)=O)C2)=O)cc2c(cn1)NC(=O)CO2 4871,C(CC)(CCCC(=O)NCC(C)(C)CCOC)NC(c1cnc(CC)o1)=O 4872,c1(C(N2CCCN(C(c3cnccc3Cl)=O)CCC2)=O)noc2c1CCCC2 4873,C(C1=CCCN(C(=O)C=C2CCCCC2)C1)NC(C(CC=C)OC)=O 4874,Cn1cc(C(=O)NC2CCCN(C(=O)CCC3CCCCC3)C2)c(O)nc1=O 4875,c1(OC)cc(C)ccc1C(N1CC2CC1CN2C(C1C2CCC(F)(F)C12)=O)=O 4876,CC1CCC(C)(C(N2CC(NC(=O)C(C)(Cl)Cl)CC(O)C2)=O)CC1 4877,c1(NC(C(C)C)=O)ccc(C(=O)NC2CCN(C(=O)C(C)(O)C3CC3)C2)cc1 4878,c1(C(N2CC(OC)C(NC(=O)C=CS(C)=O)C2)=O)ccc(C)c(C(F)(F)F)c1 4879,C1(C(=O)NCC=C2CCN(C(C(CC)(C)O)=O)CC2)CC(C(C)C)=NO1 4880,c1(-c2n(C(CC)CC)nc(C3CCOC3)n2)ccc(C)c(Br)c1 4881,Cc1c(Cl)cc(C(N2CCC(N3CC(CSc4ccccc4)C3)CC2)=O)cc1Br 4882,CCS(=O)(=O)c1ccc(C(N2CCC(C(F)F)C2)=O)cc1 4883,C12(C(N(C)Cc3ccn(C)n3)=O)CC1CCN2C(C1CC(C)(O)C1)=O 4884,N1(C(c2ccc(CC(C)(C)C)cc2)=O)CCC12CN(C(C1SCCCS1)=O)C2 4885,c1(NCC23OCC(NC(=O)CN4C(=O)CCC4=O)(C2)C3)ncc2ccccc2n1 4886,c1(CN(C(CCC)(C)c2nnnn2C)C)ccc(SC2CCOCC2)cc1 4887,CCCCC(CC(=O)N(C(C)CC(C)CC)C)NC(=O)CC1(C)CC1 4888,N1(C(CCSCCC)=O)CC2(CCC(CNC(=O)CC3(OC)CCOCC3)O2)C1 4889,c1(OC)cc(C(=O)Nc2c(Cl)c(C)nn2C)cnc1-c1ccccc1 4890,C1(NC(c2c(CC)ccs2)=O)CCCCN(C(C2CCCC(C)CC2)=O)C1 4891,c1(OCC)ccc(C)nc1C(=O)NCC(F)CNC(C1CC1C(F)(F)F)=O 4892,c1(C(N2CCCC(CN(C)C)C2)C(=O)NCCCF)cc(Br)ccc1F 4893,c1(OCC(N2C(C3(NC(c4c(C)con4)=O)CC3)CCC2)=O)c(C)cccc1Cl 4894,C1(C(=O)NCC2CC(CNC(C3CC4C=CC3C4)=O)C2)CCCCCC1(F)F 4895,C1(F)(CNC(c2cccc(C)c2)=O)CCCN(C(c2occc2C(C)C)=O)CC1 4896,N1(C(=O)OC)CCC(C(N2CCCC(CNC(=O)CSC(C)C)C2)=O)CC1 4897,CN1CCN(C)C(C(=O)NC2CCC2CNC(=O)CC#N)C1 4898,c1(C(=O)NC(C(C)NC(C2CCS(=O)(=O)C2)=O)CO)ccnn(C)c1=O 4899,CC1(C(N2CCCC(NC(c3coc(CC4CC4)n3)=O)C2)=O)CC2(CCC2)C1 4900,N1(C(c2cc(OC)n(C)n2)=O)CCN(C(=O)C2CC2)C(c2ccncc2)C1 4901,N1(C(C(C=C=C)C)=O)CC2CCN(C(c3cc(CC)oc3C)=O)CC2C1.[SH](C)(=O)=O 4902,c1(C(=O)NC2C3CN(C(C4(n5cncn5)CC4)=O)CC23)c[nH]c2cccnc12 4903,N1(C(c2cnc(C)o2)=O)CC2CCC(NC(c3cccc(F)c3Cl)=O)CC2C1 4904,Cn1c(C(N2CC(F)(F)CC2CCNC(C2CC3(CCC3)C2)=O)=O)cccc1=O 4905,c1(NC(C2CC(F)CN(CC3CCC(F)(F)CC3)C2)=O)ccc(C(F)(F)F)cc1O 4906,C(=O)(C(O)CC[S+](C)C)N1CCC(NC(c2c(C)oc(C(F)(F)F)n2)=O)C(O)C1 4907,C#CCC(C(=O)N1CCC(N(C(=O)CN2CCC(C)(O)C2)CC#C)CC1)C1CC1 4908,C1(CNC(C(Cc2ccoc2)NC(C2SCC(=O)C2)=O)=O)CC(O)C12CCC2 4909,C1(C(=O)NCC=CCNC(C(N2CCC(O)CC2)C)=O)CCCC(CF)C1 4910,Cc1cc(CC(=O)NC2(c3ccccc3)CN(C(=O)Cc3occc3C)C2)n[nH]1 4911,C1(C(=O)NCC2(C(=O)NC(c3ccncc3)C)CC(C)(C)C2)CCC(C#N)CC1 4912,C1(C(N2C(CN(C(=O)CC3CCC34CCC4)C)CCC2)=O)CCC2(CC1)CC2 4913,N1(C(CS(=O)(=O)NC)=O)CCCC(C(=O)NC(c2cnc(C)s2)C)CC1 4914,C(=O)(CCCCCN=[N+]=[N-])NCCC1(OC)CN(C(=O)COCC2CCC2)C1 4915,Cc1nn(C)c(C)c1CC(C)C(=O)NCC(CO)NC(=O)CN1CCCCCC1 4916,c1(C(C)C)conc1C(=O)NC1(CNC(=O)CC2(C#N)CC2)CC1 4917,n1(CC)cc(C(=O)NC(C)C(C)NC(c2cc(C(F)(F)F)ns2)=O)nn1 4918,c1(C(N(CCN(C(c2c(CC)onc2)=O)CC)CC)=O)cc2n(c1)CCC2 4919,c1(C(=O)NCC2(NC(c3cc(SC)oc3)=O)CC2)c(F)cc(Cl)cc1Cl 4920,N1(C(C2CN(C(c3cc(C)c(F)cc3)=O)CC(F)C2)=O)CCCC(S(C)(=O)=O)C1 4921,CCCCC(O)C(=O)NCCN(C(c1ccc(OC)cc1F)=O)C(C)C 4922,N1(C(CCc2n(C)ncc2)=O)CCOC(CCNC(C2CC2(C)C(F)F)=O)C1 4923,c1(C(C)(C)C)ccc(NCc2cccnc2)cc1Cl 4924,Cc1cc(C)c(C(=O)NC(C)C(C)NC(c2coc(N(C)C)n2)=O)cc1N 4925,CC(O)CC(=O)N1CC(N(C)C(C2CSC2)=O)C1 4926,C12(NC(CC3(C)CC3)=O)CC3CC(C1)CC(NC(C1CCCC(O)C1)=O)(C3)C2 4927,Cc1cc(O)cc(C)c1C(=O)NC12CC(C(=O)Nc3cccc(C4CC4)c3)(C1)C2 4928,c1(C(=O)NCC=C)cccc(S(=O)(=O)NC(C)CNc2cccnc2)c1 4929,CC1CCCCC1(CNC(=O)CCn1cnccc1=O)NC(C1CC(=O)N1)=O 4930,c1(NCC(=O)N(CCCN(C(=O)CNC(C2CCCSC2)=O)C)C)cccnc1 4931,N1(CC(=O)N(C)CC2CC2)CC(=O)NCC1SCCCN=[N+]=[N-] 4932,N1(C(c2cc(CC)oc2C)=O)CCCCC(CNC(=O)CCc2nncs2)C1 4933,C1(NC(C2N(C)CCC2)=O)CN(C(=O)CCc2ccc(=N)[nH]c2)CC12CCC2 4934,N1(C(c2ccc(C#C)c(C)c2)=O)CCC2CCN(C(c3scnc3Cl)=O)C2C1 4935,c1(C(=O)NCC(CC)(C)NC(=O)C(C)NC(=O)COC)cc2cncn2c(O)n1 4936,CCCCS(=O)(=O)NCC(N1CC(N(C)C(c2nn(C)cc2SC)=O)C(O)C1)=O 4937,N1(C(CNC(CCCCC)=O)=O)CCN(C(=O)C(C)CO)CC1C(F)F 4938,C(=O)(CC(C)(C)C(F)F)N1C(CC(N2CCC(OC)C2C)=O)C2CCCC21 4939,c1(C(N(C(CNC(C2(Cl)CC2(F)F)=O)C2CC2)C)=O)cnc2c(Cl)cccn12 4940,C1(C(=O)NCc2nc(C)sc2)C=CCN(C(=O)C(F)CC2CCOC2)C1 4941,N1(Cc2cc(C(N3CCCC3C#N)C(=O)NC(C)(C)C)no2)CCCOCC1 4942,N1(C(C2(CCC=C)CN(C(=O)CC=CC)C2)=O)CC2CCC1C(O)C2O 4943,c1(C(=O)NC(C2CCOC2)CNC(c2c(C)ccs2)=O)nc2c(s1)COCC2 4944,C(=O)(C1CCC(NC(=O)Nc2cc(Cl)cc(Cl)c2C(C)=O)c2ccccc21)OC 4945,Cc1ccc(O)cc1C(N1CC2CC(C1)N2C(c1nc(Cl)ccc1F)=O)=O 4946,N1(C(CCCC#C)=O)CCC2C(C1)CN2C(C1CC2(CCOCC2)C1)=O 4947,N1(C(c2ccnn2CC(F)F)C(=O)NC)CCCC2(CCCO2)CC1 4948,CCCCC(C)C(=O)NC12CC(C(=O)NCC3COC(C)(C)C3)(C1)C2 4949,C1(CC)(NC(=O)C=CSCc2ccco2)CN(C(=O)CNC(c2ccoc2)=O)C1 4950,c1(CN(C(C)CNC(=O)Cc2cccc(O)c2)C)ccc(Br)c2nsnc12 4951,c1(C(N2C3(C(=O)NC4C(OC)COC4)CC3CC2)=O)cccc(F)c1F 4952,c1(CNC(C2(C(=O)OCC)CC2C)=O)cc(O)nc(CNC(=O)CC2CCCC2)n1 4953,c1(OC(C)C)ccc(C(=O)NCCCN(CCO)C(c2cn(C)nc2Cl)=O)cc1 4954,N1(C(CC(C)OC)=O)CCCC(O)(CNC(=O)C(F)(F)CN2CCCC2)C1 4955,c1(C(=O)NC(C)Cc2nccn2C)n[nH]c2c1CN(C(=O)CCOC1COC1)C2 4956,CC1CC2(CCN(C(c3cc(N)ccc3Cl)=O)CC2)CN1C(=O)C(O)CN(C)C 4957,c1(C(=O)NC2C(NC(c3c(Cl)nc(OC)s3)=O)COC2)ccc(=O)n2c1CCC2 4958,C(=O)(C1=C(C)N(C2CCC2)C(=S)NC1c1cc(I)c(Br)c(F)c1F)NC(C)=O 4959,C1(C(=O)NCCC(CCC)C2CC2)CC2(CCC2)CN1C(=O)C1=NOCC1 4960,C(C)(CCN=c1c(Cl)c[nH]cc1[N+](=O)[O-])NC(CCCc1cc(C)no1)=O 4961,c1(NC)ncccc1C(=O)NCC(C)(C1CCC1)NC(c1ncc(OC)cn1)=O 4962,c1(C(=O)NC2(CF)CCN(C(C(C=C)(C)O)=O)C2)cc(C)nc2c1nc(C)n2C 4963,C(=O)(C1CCCn2ccnc21)N1CCC(C)C1CNC(=O)CCCC1CCCC1 4964,N1(C(c2nc(C(C)OC)sc2)=O)CCOCC1CCNC(C1CC=CC1)=O 4965,C(C)(CCC(C)C)N(C(C1C(C)=CCS1)=O)C 4966,N1(C(C(C)CC2CCC2)C(=O)NCCN2CCOCC2)CC2CN(C)CC2C1 4967,c1(CNC(C2OCCN(C(CCCN(C)C)=O)C2)=O)ccc(F)c(O)c1 4968,c1(NC(C)CCC(F)(F)F)[nH]c(=NC2CSc3ccc(F)cc32)nc2sccc12 4969,CC(CNC(=O)CN(C)C(=O)Nc1ccccc1OC1CCCC1)CC(F)F 4970,C1(C2CCN(C(=O)C=Cc3ccc([N+](=O)[O-])s3)C2)(NC(CCSC)=O)CC1 4971,CC(=O)CCCC(=O)NCC1(CCNC(C2CCCN2C(=O)C(C)C)=O)CC1 4972,C1(NC(=O)NC2CCC3(C(=O)OC)C2C3)CCC2OCCC2C1 4973,C12(NC(c3cncc(Cl)c3)=O)CCCCC1N(C(C1CC(O)C1)=O)CC2 4974,CN1CCOC2CN(C(C3(CNC(=O)COC4CCC4)CC=CC3)=O)CC12 4975,c1(OC)cccc(C(C(=O)NC(C)CCNC(=O)C(F)C2CC2)C(C)C)c1 4976,c1(C(=O)NCC2CN(C(CCC(C)C)=O)CC2O)cn2c(n1)C(C)CCC2 4977,C1(C)(NC(c2cc(OC)no2)=O)CCCC1C.C12(C)CC(C1)C(=O)NOC2 4978,C1(C2CCC2)(NC(C2C=CCCN2C(=O)CCCc2cnn[nH]2)=O)CC1 4979,Cc1cc(C(=O)NC2CN(C(c3ccc(Br)cc3)=O)C2)nnc1C 4980,C1(CC=C)(NC(=O)C(F)=CC)CCCN(C(=O)Cc2cc(Br)cs2)C1 4981,Cc1cncc(C(N2CCCCC2CN(C(=O)CSc2ccncc2)C)=O)c1C 4982,c1(C(N2C(CNC(CC(C=C)CC)=O)C(C)CCC2)=O)ccnc2c1CCC2 4983,C1(C(N(C(CC)C)C)=O)C=CC(NC(=O)C(CO)N(C)C)C1 4984,C1(CCNC(CCCOCC)=O)CN(C(=O)Cc2scnc2C)CCO1 4985,C1(O)(CNC(C2(C)CC2)=O)CCN(C(c2cc(C(F)(F)F)no2)=O)C1 4986,C1(CNC(C(CC)n2cncn2)=O)CCN(C(c2c(C)noc2C)=O)C12CCC2 4987,Cc1cnoc1Cn1cc(CCCNC(c2[nH]nnc2-c2ccccc2)=O)nn1 4988,C1(F)(C(=O)NC(C)Cc2ncn(C)n2)CCN(C(=O)C=C2CCC2)C1 4989,C12(NC(C(N3CCNC3=O)C)=O)COC(CNC(c3cc(N(C)C)ccn3)=O)(C1)C2 4990,N(S(=O)C12CC3CC(CC(C3)C1)C2)CC(c1cccc(C#N)c1)=O 4991,C1(CNC(C2(N(C(c3ccc(COC)o3)=O)C)CC2)=O)CC(O)C(O)C1 4992,C(=O)(CC(C(F)(F)F)c1ccccc1)NC1CCN(C(CSCCOC)=O)C1 4993,c1(C(N(C(C(=O)NCC(CSC)OC)C)C2CC2)=O)cccc(F)c1N 4994,C(=O)(CC(O)c1cnc(Cl)s1)N(CCNC(C1(CCC=C)CC1)=O)C 4995,C(C(C(=O)NOCCCCCC1CC1)NC(=O)C(O)CCN(C)C)OCC 4996,CC1(CNC(=O)NCCC2CCCCO2)Cc2ccccc2C1 4997,C1(NC(CN(C)C(C2CCCC2)=O)=O)CCC2(CCCNC2)C1 4998,c1(OCCC(N2C(C)(CNC(CCC=CC)=O)CCC2)=O)cccc([N+](=O)[O-])c1 4999,c1(CNC(N(C2CCS(=O)(=O)C2)CC)=O)cccc(C(C)(C)C)c1 5000,C1(CNC(c2cccc(C3(C)CC3)c2)=O)CC2(C1)CN(C(=O)C#CC1CCC1)C2 5001,N1(C(c2scc(CC)n2)C(=O)NC2CC2)CCn2c(Cc3ccccc3)nnc2C1 5002,C1(NC(CCCc2onc(CC)n2)=O)CCC(C)(CNC(=O)Cc2ccco2)C1 5003,c1(C(=O)NC2CC(N(C(=O)Cn3cccn3)C)C2)cc(Cl)cc2ccccc12 5004,N1(C(C=C=C(C)C)=O)CCC(CNC(C2CCCO2)=O)C(C2CC2)C1 5005,C(=O)(C(C)C(F)F)NCC(N(C(Cc1cc(C)no1)=O)C)C1CC1 5006,C(=O)(C(F)C(C)CC(C)(C)C)N1C(C2(NC(COC(CC)C)=O)CC2)CCC1 5007,c1(C(N2CC(CNC(CC(=O)OC)=O)C3(C2)CC3)=O)ccccc1N=S(C)(C)=O 5008,c1(C(C)C)ccccc1C(=O)NC(C)(C)CN(C(=O)CC1CCN(C)C1)C 5009,c1(C(=O)NC(C)C(C)NC(=O)COc2ccsc2Cl)ncoc1-c1ccon1 5010,c1(C(=O)NC(CC=CC)C(=O)N2CCC(C)(CC)C2)ccc(C)cc1C 5011,C1(NC(C2CC(OCC)C2)=O)CC2C(NC(c3ccc(C)cc3)=O)C2C1 5012,c1(C(C(=O)NC2CCN(C(C(C)N3CCC3)=O)C2)=O)ccc(O)cc1 5013,N1(C(c2ccc(CC)[nH]2)=O)CCC(C2(NC(C3CC3C(C)C)=O)CC2)C1 5014,C(=O)(C1CCc2c[nH]nc21)N1C(CNC(c2cccc3nccn23)=O)C=CC1 5015,C1(N(C(=O)C(=O)Nc2ncsc2Br)CCOC)CCCCCC1(C)C 5016,c1(C(N2CC(CC(C)NC(C(CC)C(C)C)=O)C2)=O)cc([N+](=O)[O-])cnc1N 5017,C12(OC)CCC(C(=O)NC3CCC(C)N(C(c4ccon4)=O)C3)(CC1)CC2 5018,C1(NC(C(C)OCCCC)=O)CN(C(=O)C(c2ccccc2)C)CC(C)(C)C1 5019,CC(C)CC(C)(O)CNC(=O)CNC(=O)Cc1ccc(C#N)cc1 5020,N1(c2nnc(SC)s2)CCCC(C)(C)C1CNC(=O)CSc1ccncc1 5021,CCCCCCC(=O)NC1CC2(C1)CN(C(=O)C(C)C(C)c1ccc(F)cc1)C2 5022,c1(N(CC)CC)ccc(C(=O)NC2CC(NC(c3ccoc3Br)=O)C2)cc1 5023,C(=O)(C1c2ccccc2CN1C(c1snc(Cl)c1Cl)=O)N1CC(c2n(C)cnn2)C1 5024,C1(CNC(c2c(OC)csc2)=O)CCCCN(c2cc(C)nc(CO)n2)C1 5025,c1(OCC)cccc(Cl)c1NC(=O)OC(C)(C)C.C12(C)CC(CN1C)OC2=O 5026,C(N=c1[nH]c(C)cc(=NCC(C)N2CCC(C)CC2)[nH]1)C1CC(OC)C1 5027,c1(CC)cc(N)c(C(=O)NCC(C)CNC(c2ncc(C)cc2F)=O)c(F)c1 5028,C(=O)(CC(C)COC)N(C(C(N1C(C(CC)C)CCC1)=O)C1CC1)C 5029,CCC(C(=O)NC(C)C(C)NC(=O)Cn1ccc(Br)n1)OC 5030,c1(CNC(C2CC(F)CN(c3ncc(C(F)(F)F)cn3)C2)=O)cccc(F)c1O 5031,Cc1cc(O)nc(N2CC(NCc3cc(C(c4cccs4)=O)no3)C2)n1 5032,C1(C(=O)NC2C=CC(CNC(c3ccc(CO)s3)=O)C2)CCC12CCC2 5033,Cc1cc(CN2CCCC(NC3CCN(C)C3)C2)cc(C)c1 5034,C1(NC(c2nc(C(C)C)sc2)=O)CN(C(C23CSC(C2)C3)=O)CC1(C)C 5035,N1(C(c2cnc(CC)[nH]2)=O)CCN(C(=O)CC2(C(F)F)CC2)C2CC12 5036,n1(CC(=O)NCC2C(C(=O)NC3(CC#C)CC3)CCC2)nc(C)cc1C 5037,C(CC(=C)Cl)(C(=O)NCCC1CCOCC1)NC(C(CC=C)NC(C)=O)=O 5038,C(=O)(C1=NN(CCO)C(=O)CC1)NCC1CC(NC(C(CCCCC)O)=O)C1 5039,C1(C(=O)NCC(C)N(C(=O)CCNC(C)=O)CC)CCC2(CCOCC2)CO1 5040,C(=O)(CC(C)(F)F)NC(C1CCN(CC(=O)N(CC)Cc2ccc(F)cc2)C1)C 5041,CCCC(C)(CC)C(=O)NCC1(F)CCCN(C(=O)CSC(C)(C)C)C1 5042,CCCCC(C)CCC(=O)NC(C)C(C)(C)NC(c1nc(CC)c[nH]1)=O 5043,c1(C(=O)NC(CCSC)C(=O)NO)ccc2c(c1)OCO2 5044,CCCC(CNC(=O)C(C)(C)c1ccno1)C(=O)N(C)CC1CC1(C)C 5045,c1(C(=O)NC2CN(C(c3cncc(SC)c3)=O)C2)cc2c(C)cccc2o1 5046,C1(NC(C=NOC)=O)(CO)CCN(C(c2c[nH]nc2-c2cnn(C)c2)=O)CC1 5047,C(CCC)(C(=O)N(C1CCCC(NC(=O)CCC2CC(OC)C2)C1)C)=CCC 5048,C1(NC(=O)COC2CC=CC2)CCCCC1NC(=O)C=CC1CCOCC1 5049,C(=O)(C1Cc2ccc(Cl)cc21)N(CCNC(c1cc(C(C)C)nc(O)c1)=O)CC 5050,N1(C(COCc2cccc(C)c2)=O)CCCC12CCN(C(c1ncoc1C)=O)C2 5051,C1(NC(=O)C(c2ccccc2)F)CCN(C(=O)CC(O)c2cnc(Cl)s2)CC1 5052,O=C1NC2(C(N3CCC(CO)(Cc4cn(C5CC5)nn4)C3)=O)CC3CC1C2C3 5053,C(=O)(CC(C)C(F)(F)C(F)(F)F)N1CC(NC(COCC)=O)C(F)CC1 5054,CCC(C)C(C(=O)NC(CC(C)C)C(=O)N1CC(C)C(C)C1C)N(C)C 5055,Cc1n[nH]c(C)c1C(=O)NCC1CN(C(=O)C(C)Oc2ccccc2F)CCO1 5056,C1(C#CC(=O)N2CCN(C(=O)CC(C)O)CC2CCc2ccccn2)(CC)CC1 5057,C1(N(C)C)CCC(C(=O)NCC2(O)CCN(C(c3cccnc3)=O)C2)CC1 5058,c1(C(=O)NC2C(CCC)CN(C(=O)C(CC)OC)C2)cc([N+](=O)[O-])ccc1CC 5059,c1(SCC(=O)NCCNC(=O)COCC2CCCCO2)cc(F)cc(F)c1 5060,c1(CCOC)nc(=NC(C)C2CN(C(C3(C)CC=CCC3)=O)CCO2)s[nH]1 5061,c1(CC)ccc(C(=O)NC2CN(C(=O)C(CC)SC)CC2(C)C)cc1C#N 5062,Cc1nc2c(N3CCC(O)C(C(N4Cc5ccc(Cl)nc5C4)=O)C3)ncnc2[nH]1 5063,C1(NC(Cc2c(C)n[nH]c2)=O)CC2(CCN(C(=O)C(C)C3(O)CCC3)CC2)C1 5064,C1(CNC(c2cc[nH]n2)=O)CCCCN(C(=O)CN2CCCCCCC2=O)CC1 5065,CCCCC(O)C(=O)NC(CNC(=O)Cc1ccc(F)cc1CC)CC 5066,C1(CNC(C(C2CC(NC(c3cc(C)c(C)s3)=O)C2)F)=O)CC2(CC2)C(=O)O1 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5084,C1(CCC)(NC(C2CCN(C(c3nccnc3N)=O)C2C2CC2)=O)CCNC1=O 5085,Cc1nn2cc[nH]c(=O)c2c1C(=O)NC1CCCN(C(=O)C(C)(C)C)CC1 5086,N1(C(C(CC)CN(C)C)=O)CC(C(N2CCCCC2CN(C)C)=O)C2(CCC2)C1 5087,Cc1nc(NC2CCCC(NC(=O)Cc3ccc(C)nc3)C2)c2scc(C)c2n1 5088,C1(N(C(c2n(CC)nnc2)=O)C)CCC(NC(c2oc(C)cc2C)=O)CC1 5089,c1(C(N2CCCCC(NC(C3(COC)COC3)=O)C2)=O)cc([N+](=O)[O-])ccn1 5090,c1(NCCCCC=C)nc[nH]c(=NCc2cc(C)ncn2)c1C 5091,C=CCC(CC(F)F)NC(=O)C(F)C(C)CNC(=O)Cc1ccoc1 5092,c1(C(N2CC(C)N(C(C3COC(=O)O3)=O)CC2)=O)nn(C)c2ccccc2c1=O 5093,C1(C)(CC)CCCN(C(C2(CC)C=CCN2C(C2CCC3(CC3)C2)=O)=O)C1 5094,N1(C(C(CNC(C)=O)(C)C)=O)CCN(C(c2cc(C)cc(C)c2)=O)C2CCCC12 5095,C1(C)(C)CCCCC(=O)N1.C1(COC)CCC(NC(=O)C=CCF)CC1 5096,c1(C(N(CCNC(C2CC(CS(C)(=O)=O)C2)=O)CC)=O)cccc2ccnn12 5097,C1(C(N(CCCOCCNC(CC=CC)=O)C)=O)CCC(NC)CC1.C(C)(=O)O 5098,CCCCC(CC)CC(=O)N1CC(F)(F)CC1CCNC(=O)CCOC1CCC1 5099,CCC(C)(C)CC(=O)NC(C)CC(=O)N1CC(CC(F)(F)F)C1 5100,C(CC(=O)NC1CCC1N(C)C)NC(CC1(C(=O)OC)CC1)=O 5101,c1(C(N2CC(C)C(NC(c3cc(Cl)cs3)=O)C2)=O)cc(N)c(F)c(F)c1Cl 5102,C1(Cl)(C(=O)NCC(C)NC(c2cnnn2C)=O)CC12CCC2 5103,c1(OC)ccccc1CNCc1cc(C(=O)Nc2cc(O)ccn2)ccn1 5104,Cc1ccc(NC(C2(C)CCCN2C(c2cc(Cl)c(F)cc2F)=O)=O)cc1C#N 5105,c1(C(c2nnnn2CC2CCOCC2)NCC2(CCO)CC2)cc(Cl)no1 5106,C12(C(=O)NCC3C(NC(c4cc(CC)n(C)n4)=O)CCCC3)CC(C)(C1)OC2C 5107,C1(C)(CNC(CN2CCN(C)CC2)=O)CN(C(C2CC(C)(O)C2)=O)C(C)(C)C1 5108,C1(NC(CC2(COC)CCCC2)=O)CCCCC1CNC(=O)C(C)=C1CCC1.C 5109,C1(NC(=O)NCc2cccc(OCC#C)c2)Cc2ccccc2N(C)C1 5110,CC(C)(C(=O)NCCN(C1CCCC1)C(=O)CC1CCC(=O)N1)C1CCCCC1 5111,O(NC(=O)C(O)CNC(=O)C(F)(F)CC=C)CCC#C 5112,C(=O)(C1CC(N)c2ccccc21)N1CCC(C)(c2ccc(Cl)cc2)C1 5113,C12(NC(=O)CC3CCCO3)CCC(CNC(=O)Cn3cnnc3O)(C1)OC2 5114,N1(C(c2ccc(OCCF)cc2F)C(=O)NCCSC)CCN2C(=O)NCC2C1 5115,C1(CC(=O)NC(COC)C(=O)NCCCC2CCCC2)COCC(C)O1 5116,N1(CC(=C)Cl)CC2CCC(NC(c3ncn(CC)n3)=O)CC2C1 5117,c1(CN2CC(C(=O)NC(c3ccc(C(N)=O)cc3)=O)OCC2)cc2n(n1)CCC2 5118,C=CCC(C(=O)NC(CO)C(C)NC(=O)CCC(N)=O)c1ccccc1 5119,c1(CCCC=C)ccc(C(=O)NCC(C2CC2)NC(C2(N3CCCC3)CC2)=O)cc1 5120,C(CC(C(=O)NCCC1CCN(C)C1)NC(=O)Cn1ccc(C)c1)OC 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5139,c1(C(N2CCC(CNC(c3cnc(Cl)[nH]3)=O)C2)=O)ccncc1N1CCCC1 5140,c1(NC(CC(C)(C)C)c2nnnn2Cc2ccccc2)ccc(CO)c(I)c1 5141,C1(CNC(C2CCCO2)=O)(CO)CC12CCN(C(=O)CC(F)(F)C(F)(F)F)CC2 5142,N1(C(C(C)SC)=O)CCN(C(=O)CCCCCc2cccs2)CC1c1ncc[nH]1 5143,N1(CCC)CCCC1C(=O)NC1CC(C)(NC(=O)C(c2ccc(C)s2)C)C1 5144,C1(C(=O)NCCN(CCOC)C(c2cnn(C3CC3(F)F)c2)=O)CCNC(=O)C1 5145,C1(NC(CC2C(C)CCO2)=O)CC2(CCN(C(c3ccoc3C3CC3)=O)CC2)C1 5146,C1(CNC(C(C2CCCC2)OC)=O)CCCN1C(C1CCS1(=O)=O)=O 5147,Cc1nn(C)c(Cl)c1C(N1CCN(C(c2coc(Cl)n2)=O)C(c2cn[nH]c2)C1)=O 5148,CC1OC(C)CC1C(=O)NCC1(NC(c2sc(N(C)C)nc2Cl)=O)CC1 5149,Cc1ccc(Cl)c(F)c1C(=O)NCC1CCC(NC(=O)Cc2cccc(F)c2)C1 5150,c1(C(=O)NCC2N(C(Cc3ccc(C)s3)=O)CCC2C)ccc(=O)n(C)n1 5151,C1(Cl)(C(=O)NC2CC(NC(C(C)OCC)=O)C2)CC1(C)C 5152,c1(CNC(C(=O)Nc2ccc(NC(=O)OCC)c(C)c2)=O)c(C)ccc(C)c1O 5153,c1(C(=O)Nc2ccc(C)nc2Cl)ccc2c(C(N3CCC(C#N)C3)=O)n[nH]c2c1 5154,c1(OC)ccc(Br)c(CNc2csc(-c3c(O)cccc3F)n2)c1 5155,C1(C(=O)NC(CC=C)CO)CCN(C(=O)C(C)COC)C12CC2 5156,C(C)(CCCCNC(c1cnc(OC)s1)=O)NC(c1cnc(CCCC)s1)=O 5157,Cc1ccc(C(=O)NCCN(CC(C)O)C(=O)CC2CC=CCC2)cc1O 5158,N1(CC(=O)NCCC(C)NC(C2(CO)CC2)=O)CCCC(C(=O)N(C)C)C1 5159,S(=O)(=O)(c1cccc(N2CCCC2)n1)NC1C(NC(c2nncs2)C)COC1 5160,C(=O)(C1CCc2cc(F)ccc21)N1CCC(C2CC2)(NC(CC=C(C)C)=O)C1 5161,N1(C(C(C)N=[N+]=[N-])=O)CC(C)(C)CC1CC(=O)NCCC(=O)NC(C)(C)C 5162,C(=O)(C1Cc2ccc(F)cc21)N1CC(OCCNC(=O)Cc2sc(O)nc2O)C1 5163,C1(NC(CC2CC(=C)C2)=O)CC12CCC(NC(c1cc(C(=O)OCC)on1)=O)CC2 5164,CC(C)(CCCNC(C1CC12CC2)=O)C(=O)N1CCCC(CC2CC2)C1 5165,C(=O)(C(=O)CC(C)C)N1CC(CC=C)(NC(=O)Cc2cn[nH]c2)C1 5166,CC(C)C(C)(CNC(=O)C(CNC(=O)C=Cc1cncn1C)N(C)C)C(C)C 5167,C1(C(=O)NCCC(C(=O)NCCCCN=[N+]=[N-])OC)CC2(CCCO2)C1 5168,C1(C2CCN(C(=O)CC3(C)CCS(=O)(=O)N3)C2)(NC(c2cc(C)no2)=O)CC1 5169,c1(C(=O)NC2CC(NC(c3nc(OC)c(F)cn3)=O)C2)ccc(C#N)cc1F 5170,C1(NC(C2C(C)CCC2)=O)CCOC12CCN(C(=O)C(C)(C)CCCO)CC2 5171,c1(CC(=O)NCC2(OC)CN(C(C3CC3(C)C)=O)C2)ccc(F)cc1C 5172,c1(C(=O)NC2C(CNC(C(COC)(F)F)=O)C2)c(Br)nc2n1CCCC2 5173,C1(OC)CCC(CC(=O)NCCNC(c2cnn(-c3ccc(Cl)cc3)c2C)=O)CC1 5174,Cc1ccc(C(=O)NC(CO)C(C)NC(=O)CC2(CO)CC2)c(N)c1Br 5175,c1(OC)cc(C(N2CCC(C3(NC(=O)CCC(C)(F)F)CC3)C2)=O)cc(N)c1O 5176,Cc1cnn(C)c1C(=O)NC(CCC(=O)NCc1cn(C2CC2)cn1)C 5177,c1(C(N2CC(NCc3c(C)cccc3O)C(F)CC2)=O)ccc2cnccc2c1 5178,C(=O)(C1CCCn2c(C)nnc21)NC(C(C)(C)NC(Cn1c(C)cc(C)n1)=O)C 5179,C1(C(=O)NCC(C(C)(C)C)NC(C=Cc2c(C)ccs2)=O)CCc2nc[nH]c2C1 5180,C(CC(C)(C)CC(=O)NCC1CCCCN(C(=O)CC2CC(=O)C2)C1)OC 5181,CC1CCC(C)N1CC(=O)NCC1(F)CC(NC(=O)COCC2CC2)C1 5182,N1(C(c2cccnc2S)=O)CC2CN(C(c3c(Cl)cncc3Cl)=O)C2C1 5183,N1(C(CCSCC)=O)CCC(C2CC2)C1CNC(=O)C(F)=CC1CC1 5184,Cc1c(C(=O)N(CC(O)CN(C(=O)CC2COCCN2C)C)C)nc2sccn12 5185,c1(CC)ccc2c(c1)C(NC(C1(C)CN(C(=O)OC(C)(C)C)C1(C)C)=O)CCO2 5186,N1(C(C2C(C)C2)=O)CCc2cc(C(=O)Nc3cc(F)c(Cl)cc3I)cnc2C1 5187,c1(OC)ccc(C=CC(=O)NC(CO)C(c2ccc([N+](=O)[O-])cc2)O)cc1F 5188,C12(C(=O)NCC3(OC)CCOC3)COCC1CN(C(C1CCC1C#N)=O)C2 5189,c1(NC(CN2CCN(C(c3c(C)nc[nH]3)=O)CC2)=O)cc(Cl)cc(Cl)c1Br 5190,c1(CCC(=O)NCC2(C)CCN(C(CCS(C)=O)=O)C2)ccc([N+](=O)[O-])cc1 5191,CON1CC(C(N2CCC(NC(C3CC=CCO3)=O)CC2)=O)CC1=O 5192,C=CCCCC(C(=O)NCCS(C)(=O)=O)NC(C1C2CCCCCC12)=O 5193,N#Cc1cccc(C2CC2C(=O)NC2(C3CN(C(C4CCSCC4)=O)C3)CC2)c1 5194,N1(C(c2n(C=C)ncc2)=O)CCC(C)CC1CNC(=O)CC 5195,Cc1cccn2cc(C(N3CC(C(=O)NCCNS(C)(=O)=O)C(F)C3)=O)cc12 5196,Cc1sncc1C(=O)NCC1CC1CC(=O)N(CCS(C)(=O)=O)C 5197,c1(C(c2nnnn2C(C)C)NCCC(C)CO)cccc(Br)c1OCC(F)F 5198,C(=O)(CCCCC(C)(C)C)N1CCC(F)(CNC(c2c(C)con2)=O)CC1 5199,CC1(NC(=O)CC2CC=CCC2)CCN(C(C2CCC3CCC2O3)=O)CC1 5200,C(CC1CC1)(C(=O)NC1CC(CF)C1)NC(=O)Cc1cc[nH]n1 5201,N1(C(c2ccc(CCC)cc2)=O)CC(C)CCC1CNC(C1CN(C(C)C)C1)=O 5202,c1(C(N2CCC(NC(c3cncc(NCC)c3)=O)C2)=O)cc(C)ccc1O 5203,c1(CC(=O)N(CCCCCNC(C(CCC)F)=O)C)ccc(F)cc1C 5204,Cc1cnccc1C(N1CCCC1CN(C)C(c1cnn(CC(F)F)c1C)=O)=O 5205,C1(C(=O)OC)C(F)(F)C12CC(C(N1CCN(C(c3cnns3)=O)C(C)C1)=O)C2 5206,C(CC(C)C)(C(=O)NCCCCCN(C)C(C1CC12CC(C)(C)C2)=O)NC(C)=O 5207,C(=O)(C1=CC2CCCCC12)N1CC(CNC(c2c(CC)cncc2)=O)N(C)CC1 5208,C1(C(N(CC(C)(C)CNC(C2CCCCC2F)=O)C)=O)CCC(=C(F)F)CC1 5209,c1(C(N2CC(OC)(CNC(=O)C(C)C(C)(C)C)C2)=O)ccc2ncccn12 5210,CC1OC2(C(=O)NCCCN(C(=O)CC#N)Cc3ccccc3)CC1C2 5211,CC(C)(C)CC(=O)OCC(C)(C)C.C1CC(O)CNC(=O)C=CCS1 5212,CCCC(CC)C(c1nnnn1Cc1ccco1)NCc1nnnn1C1CC1 5213,CC1c2ccccc2CC1C(=O)NCC1(CNC(c2cnc(C(F)F)s2)=O)CC1 5214,N(C(=NCc1cccc(F)c1)NCC12CC(C1)C(C)O2)C(C)C1CC1 5215,CC(C)C#CC(=O)NCC1CCCN(C(=O)CCCc2ccccn2)C1 5216,N1(C(C(C)OC2CCOC2)=O)CCC2CN(C(c3cnn(C)c(=O)c3)=O)CCC12 5217,c1(C(CS)C)cn(CCCCC2CCC2)nn1.C(C(=O)NCCOCCO)N(C(C)C)C 5218,CN1CCC(C(=O)NC2CCN(C(c3oc(C(F)(F)F)nc3C(F)F)=O)C2)CC1 5219,C1(C(=O)NCC(C(C)O)O)CCC2(CC2)N1C(c1cccc(CO)n1)=O 5220,c1(C(=O)NCC2CCN(C(=O)CC3CCSC3)CC2)ccnc2ccnn12 5221,C1(CNC(C2C(C)(C)C2)=O)(CNC(C2CC(n3cnnc3)C2)=O)CC12CCC2 5222,C1(CNC(CC(C)(C)SC)=O)CCC(C)N(C(c2ccc(F)o2)=O)C1 5223,C(=O)(CC(C)CC(C)(C)C)NCC(CC)(CC)NC(c1cc(C)c(O)c(C)c1)=O 5224,CCC(C)(C)C(O)C(=O)NC1CN(C(c2cc(Cl)cc(C)c2O)=O)CC1OC 5225,C1(C(N(C(C(N)=O)C2CC2)C)=O)CC=CCN1C(c1cccc(CC#N)c1)=O 5226,c1(C(N2CCC(C)(CNC(Cc3c(C)nsc3)=O)C2)=O)ncc(C2CC2)cc1F 5227,N1(C(C(COCC)CC)=O)CC2(CCN(C(=O)C(C)P(C)(C)=O)CC2)C1 5228,CC1SCCCC1C(=O)NCC1(C(=O)N(C)CC2(C#N)CCC2)CC2(CC2)C1 5229,c1(OCCOC(c2cn(C)nc2C2CC2)=O)ccccc1[N+](=O)[O-] 5230,N1(C(C(C(=C)Cl)(C)C)=O)CCC2CN(C(c3ccn4nncc4c3)=O)CCC2C1 5231,N1(C(C(CC)C)=O)CC2CCOC2(CNC(c2cncc(C)c2C)=O)C1 5232,N1(C(C(C(=C)C)(C)O)=O)CCC2(CC1)CC(CNC(=O)CCC(C)C)C2 5233,c1(C(=O)Nc2scc(C(=O)NCCNC(C)=O)n2)c(O)ccc(F)c1F 5234,C(=O)(C(CC(C)C)NC(=O)Cc1c(C)cnn1C)NC(CC)COCC1CC1 5235,Nc1ccccc1OCSC1(O)CCNC1.C1C(=O)O1 5236,S(=O)(=O)(c1cc([N+](=O)[O-])c(N)cc1Br)NC(C1CN(C)S(=O)(=O)CC1)=O 5237,C1(NC(CSCC)=O)CN(C(=O)C(c2ccn(C)c2)C)C(C)(C)C1 5238,C1(NC(COCCC)=O)COCCN(C(=O)C(c2cccc(C#N)c2)(C)C)C1 5239,Cc1c(C(=O)NC2CCCC2CNC(C2(CN(C)C)CC2)=O)c[nH]c1C#N 5240,N1(C(C2CCCCCCN2C(C2CCC3CC2CO3)=O)=O)CC2(CCOCC2)C1 5241,CC1CC(C(=O)NCCC2CCCCC2O)N(C(c2ncncc2Cl)=O)C1 5242,C(C(CC)(CC)NC(=O)Cc1ncc(C)s1)NC(C(CC)F)=O 5243,C1(CC=C)(NC(=O)C(C)=C(C)C)CC2CCC(C1)N2C(c1snc(C)c1N)=O 5244,C(=O)(CC(C)CC(=O)NCC(O)C(=O)NC1CC(C(C)O)C1)OC 5245,C1(NC(CCC(=O)OCC)=O)CC(O)CN(C(c2cocc2C)=O)C1 5246,C1(CC=C)(NC(c2cnc(O)cc2O)=O)CC2CCC(C1)N2C(=O)C(C)(C)CF 5247,C(=O)(CS(=O)(=O)CC(C)C)NC1CCC(CNC(C(CC(C)=O)(C)C)=O)C1 5248,CC1CCN(C(C2CCOC2(C)C)=O)C(CNC(c2cc[nH]c2)=O)C1 5249,c1(OC)nc(Cl)ccc1C(N1CC2C(NC(=O)C=Cc3cnccc3C)C2C1)=O 5250,N1(C(c2ccc(CSC)cc2)=O)CCC2(CNC(C3CC3(C)C)=O)CCCC12 5251,C1(CNC(Cc2ccc(OC)cn2)=O)CC12CCN(C(=O)C(C)(O)C(C)C)CC2 5252,C(CCCC(=O)N(C)CC1CCC(=O)N1)N(C(=O)Cn1cnc(C#N)n1)C 5253,CCC(C)(C)C(C)(O)c1nc(C(c2ccccc2)C)no1 5254,c1(C2N3CCN(CC3)CCNC2=O)ccc(C(F)(F)F)c(F)c1.C1CC1.CCO 5255,C(=O)(C(C)CC(N)=O)N1CC(O)(CNC(C(C)Oc2cccc(N)c2)=O)C1 5256,C1(NC(COCCCCC)=O)C(C)(C)CN(C(=O)C(C)CC(C)CC)CC1(C)C 5257,N(C1c2ccccc2CC12CCOCC2)Cc1cccc(CO)c1 5258,N1(C(CC(C=C)C)=O)CCC(C(=O)NC(c2nc(=O)o[nH]2)C)C1(C)C 5259,N1(C(=O)Cc2ccccc2F)CC2CC(C1)N2C(c1cc(F)ccc1I)=O 5260,c1(C(=O)NCC2CC(F)(CNC(C3CCC(C)O3)=O)C2)cnc(O)c2ccsc12 5261,c1(C(N(C2CCCN(C(C3CCS3(=O)=O)=O)C2)CC)=O)ccnc2c1nnn2C 5262,c1(C(=O)NCC2(CNC(=O)Cn3cnnn3)CCC2)ccc2c(n1)OCCO2 5263,C1(C2CC2)(CNC(CCC(C)(F)F)=O)CCN(C(c2cncc3ccsc23)=O)C1 5264,c1(C2(C(=O)NC3CCN(CCCNC(COC)=O)C3)CC2)cnn(C(C)(C)C)c1 5265,C(=O)(C(C(C)CC)N(C(=O)CCC(C)SC)C)N(CCC)C 5266,Cc1nn(C)c(Cl)c1CN1CCCC1CNC(c1cc(C(C)C)nn1C)=O 5267,CCC1=C(C(=O)NCC2CC(CNC(c3cc4cscc4s3)=O)CO2)CCCO1 5268,N1(C(CCC=C(C)C)=O)CC(CN(C(=O)C(O)C(C)(C)C)C)C2(CC2)C1 5269,CCC(CCOC)C(=O)N1CC(OC)CC1CNC(C1(CO)CCOCC1)=O 5270,c1(CC)ccc(C)nc1NC(C1(F)CCCN(C(C2CCCCO2)=O)C1)=O 5271,CC1CC(N(C(=O)CC2(CNC(=O)COCCCF)CC2)C)CC(C)C1 5272,CC1CC(C)CN(C(=O)CNc2cnn(-c3cc(F)ccc3F)c2)C1 5273,N1(C(COCCC(C)C)=O)CC2CC(O)C1C2NC(c1ncoc1C1CC1)=O 5274,c1(C(=O)NC2CC(C)(NC(Cc3scc(C)c3)=O)C2)cc2n(c1)CCOC2 5275,c1(OC)ccnc(C(=O)NC2CC(CNC(=O)CC3CC(C)=NO3)C2)c1 5276,C1(C(N)=O)CCN(CC2CCC(C(=O)O)N2C(=O)CC2CSCCO2)CC1 5277,c1(C(c2n(CCCSC)nnn2)NCc2cccc(Cl)c2)c(F)ccc(Br)c1Cl 5278,C1(C(C)(C)C)CCCN1C(=O)C(O)CNC(=O)CC(C1CC1)C1CC1 5279,C1(CNC(C2C(C=C(C)C)C2C)=O)(NC(c2nncn2C)=O)CCCCC1 5280,c1(CC)ncncc1C(=O)NC(CC1CCCC1)C(=O)NCCN1CCCC1C 5281,c1(SCC)cccc(C(N2CCCC2C2CCCN(C(C3CCCC3)=O)C2)=O)c1 5282,c1(COCC(C)NC(C2(Cc3ccccc3)CCO2)=O)ccccc1 5283,c1(C(=O)NCCCCNC(C2(CC#C)CCOC2)=O)cc(-n2ccnc2)ccn1 5284,O=C(C1=CCCC1)NCC1CN(C(=O)CCC(=O)c2ccc[nH]2)C2CC12 5285,CC1CN(C)CC(C(=O)NCC(C)(C)CNC(=O)COc2cccc(O)c2)O1 5286,c1(CC(=O)NCCN(C(C2CC(O)C2)=O)C2CC2)cccc2[nH]ncc12 5287,c1(C(c2nnnn2CC2CCCO2)NCCCCCC)cccc(Cl)c1Br 5288,Cc1cccc(C2(CNC(C3CCCCC3N3CCOCC3)=O)CC2)c1I 5289,N(C(=NCc1cc(CN2CCCC2)on1)N1CCC(COC)C1)C(C=C)C 5290,C1(C)(C(=O)NC(CCCC)CNC(C2(C)CCCC2(F)F)=O)CCC(C)(C)CC1 5291,N1(C(C(C)CN(C)C)=O)CC(CC(=O)N(C)CCC2CCOCC2)C(C)C1 5292,C1(N(C2C(C=C)C2)C(C)=O)COCC1NC(=O)C(=O)NC1CCCC1 5293,N1(C(c2ccc(OCC)nc2)=O)CC2(C1)CN(C(=O)CC1CCCC(=O)N1)C2 5294,c1(CS(=O)(=O)N(C2CC3CNC2C3)Cc2c(C)nc[nH]2)ccc(Cl)cc1 5295,c1(CC)cccc(C)c1C(N1CCN(C)C(CNC(C2CC(OC)C2)=O)C1)=O 5296,c1(C(N2CCCN(C(=O)C(C3CC3)C3CC3)CC2)=O)cc2c(nc1O)CCOC2 5297,Cc1cnc(C#N)nc1N(C1CCCN(C(C2COC3COCC23)=O)C1)CCO 5298,CC(C)(C)C(CNC(C1CCC(F)(F)C1)=O)NC(c1ncccc1Br)=O 5299,c1(C(=O)NCC=CCNC(c2cnc(C(C)C)s2)=O)ccc(Br)nc1O 5300,C(=O)(CC(F)(F)Br)N(C1CCN(C(C2CCN(C)C2C)=O)C1)CC 5301,C(=O)(C1=CCC(C)(C)CC1)NCC1N(C(c2snc(C)c2N)=O)CCC1 5302,C1(NC(C2(C)CC2)=O)CCC(C)(C)CC1CNC(c1nccc(N)c1Cl)=O 5303,Cc1cnc(C(=O)NCCCCC2CCCC2)c(S(=O)(=O)N2CCC(CF)C2)c1 5304,CC1(C)CN(C(c2cnc[nH]2)=O)CCC1NC(C1CC2(CC2)CO1)=O 5305,C(C#Cc1cccnc1)NC(C(CCOCC)NC(C1CN(C)CCN1C)=O)=O 5306,N1(C(C2CC(C)(F)C2)=O)CCCC12CCCN(C(c1cccc3c1CCN3)=O)C2 5307,N1(C(CN(C2CC2)CC)=O)CCN(C(=O)CC2C=CCC2)C(c2ccnn2C)C1 5308,C1(C(=O)NCC2(OC)CN(C(CC=CC)=O)C2)Cc2cccc(F)c2O1 5309,c1(C(N2CCC(C)(CNC(=O)Cc3ccoc3)CC2)=O)ccc2nc[nH]c2n1 5310,c1(C(N(C2CCN(C(=O)CC3(OC)CC3)C2)CCC)=O)ccnc(C(C)(F)F)c1 5311,c1(C(N(CCN(C(=O)CN2C(=O)CCC2=O)CC)CC)=O)cccc(C2CC2)c1 5312,C1(C(N(C2CN(c3ccnc(C(=O)OC)c3)C2)CCC)=O)CC12CCCOC2 5313,CCC(CC(C)C)C(=O)NCCC1(NC(=O)CCc2cncs2)CCCC1 5314,Cc1nc2n(c1CC(N1CC(NC(=O)CC3CCC(C(N)=O)C3)C1)=O)CCCC2 5315,n1(C(C)C)cc(C(=O)NCC(C)NC(C2CCN(c3nccn3C)C2)=O)cn1 5316,C1(NC(=O)C(N2CCC(C(F)(F)F)C2)=O)CCC2CN(CC3CCOC3)CC2C1 5317,c1(CN2CC3N(S(C4(CC=C)CC4)(=O)=O)C(C3)C2)cc(OC)c(O)c(I)c1 5318,N1(C(CN(C2CCCC2)C)=O)CCC1CNC(C1CC(n2ccnc2)C1)=O 5319,c1(CN2CCCC(Cc3nc(C)on3)C2)noc2c1CC(C)CC2 5320,CCC(C)C(C(=O)NC(c1nnc(O)o1)C)NC(C1CC(=O)NC(=O)C1)=O 5321,C(=O)(C(C)C(O)CC(C)C)N1CC(F)(C(=O)NC(CCC=C)(C)C)C1 5322,CCCCCCC(F)C(=O)NC(CNC(c1cnccc1Cl)=O)C(C)C 5323,c1(OC)ccc(Cl)cc1C(N1CCCC(C(=O)NCCC(O)c2cccs2)C1)=O 5324,C=CCC(CNC(C1CC(CC)(CC)C1)=O)C(=O)NCC1CC12CCC2 5325,c1(C(C)=O)csc(C(=O)NCC(C)(C)CN(C(=O)C(F)(F)c2ccncc2)C)c1 5326,N1(C(CCCC#C)=O)CC(C)N(C(C2CC2(C(=O)OCC)C(C)C)=O)CC1C 5327,N1(C(C)=O)CCC(c2nc(CC(C)C(C)(C)C)n(C3CCS(=O)(=O)C3)n2)CC1 5328,C#CCC(CC(=O)OC)NC(C1(CCN(C)C)CC1)=O.C12CCCCC1NC2=O 5329,C1(C(N2CC(n3ccnc3)C2)=O)(CC)CCN(C(c2n[nH]c(C)c2Cl)=O)C1 5330,Cc1cnc(C(N2CCC(NC(c3sc(C)c(C)c3C)=O)C(O)C2)=O)cc1C#N 5331,C1(NC(COCCCC#C)=O)CN(C(c2ccc(F)c(C)c2)=O)C(C)(C)C1 5332,Cc1cc(C(C)NC2CCN(C(=O)OC)C2)cc(C)c1F 5333,c1(C(N2CC3CC(CNC(c4n(C)c(S)nn4)=O)C3C2)=O)cc2cccnc2[nH]1 5334,c1(CC(=O)N(CCN(C(c2c(CC)cco2)=O)C)C)csc2nccn12 5335,c1(NC(C2(C(=O)NCC3C(C(N)=O)C3)CC2)=O)cnc2ccccn12 5336,Cc1nn(CCO)cc1C(=O)NCC(O)CN(C)C(C1(C(C)C)CNC(=O)C1)=O 5337,c1(N2CC(CNC(C(C)C3CC3)=O)OCCC2)c(Br)cncc1[N+](=O)[O-] 5338,c1(CNCC2(CC(=O)OC(C)(C)C)CCOC2)ncccc1Br 5339,c1(C(=O)NC2(CNC(c3ncncc3Cl)=O)CCOC2)cn2ccccc2n1 5340,CC(CNC(=O)C(C)(C)C1CC1)C(F)C(=O)N(CCCO)CCO 5341,c1(OC)cc(C)ccc1C(N1CCNC(=O)C1c1cccc(Br)c1)=O 5342,C1(C(N2C(C(N3CCC(OC(C)C)CC3)=O)CC(F)C2)=O)CC2(CCO1)CC2 5343,C(=O)(C(O)CC(=O)OC(C)(C)C)N(C1CCCN(C(c2cc(Cl)no2)=O)C1)CC 5344,C1(F)(CNC(C(C)(C)F)=O)CCN(C(C2(c3cccnc3)CCC2)=O)C1 5345,c1(N2CC(C)C(NC(=O)Cc3cc(C4CC4)on3)CC2)ncnn2cccc12 5346,c1(C(N(CC(CNC(c2c(C)ccc(C)n2)=O)O)C)=O)cc2cc(F)ccc2o1 5347,C1(C(CO)NC(C2(CO)CCCN2)=O)CCCOC1 5348,C(=O)(C1c2ccccc2C2(CC2)CN1CC)NCc1ccnn1CCF 5349,N1(C(c2c(C(C)=O)cco2)=O)CCC2(CCN(C(c3c(Cl)nn(C)c3C)=O)C2)C1 5350,CCCCCC(CC)C(=O)NCCC1CCCN(C(c2cc(N)cc(F)c2)=O)C1 5351,c1(C(N(C2CCCN(C(=O)CC34CC(C3)C4)C2)CC)=O)noc2c1CCCCC2 5352,CC1CC(C(N2CCC(O)C2c2ccccc2)=O)N(C(=O)C=CC2CC2)C1 5353,C1(C(N2CCCC(CNC(c3ccc(C)cn3)=O)CC2)=O)Cc2cccnc2C1 5354,C1(C(=O)NC(CC(=O)NC)C)(COC)CCN(C(=O)C=Cc2cocn2)C1 5355,C(C1=CCCCC1)(c1nnnn1CC)NC(c1ccc(F)cc1)C(=O)NCC 5356,C1(F)(CNC(c2cnco2)=O)CC2CCC(C1)N2C(c1noc2ncccc12)=O 5357,C(=O)(C(F)C(C)C)NC(C(=O)NC(CN(CC)CC)C)C1CCCC1 5358,CC(C(C(=O)O)NC(=O)OC(C)(C)C)c1ccccc1.c12nc(no1)C2 5359,C1(N(C2CCOCC2)C(c2ccc(OC)cc2)=O)CCNCC12CC2 5360,c1(OC)cc(C(=O)NC2CC(CC(=O)NOCC(C)C)C2)ccn1 5361,C1(NC(C2CCCC3CCCN23)=O)CN(c2nncs2)CC2(CC2)C1 5362,C1(CNC(c2c(C(C)C)ncnc2)=O)CCCCN(C(C2COC(=O)N2C)=O)C1 5363,N1(C(C2C(OCC)C2)=O)CCN(C(=O)C(C)(C)CNC(C)=O)CC(C)(F)C1 5364,c1(COCC)ccccc1NC(=O)C(C)NC(c1cc[nH]c1SC(C)C(=O)O)=O 5365,N1(C(C(C)(C)C2CCN(C(C3CC34CCC4)=O)C2)=O)CC2CC2(CO)C1 5366,CC1CC(NCc2cccc(F)c2)CN(C(c2ccc([N+](=O)[O-])o2)=O)C1 5367,c1(C(=O)NC(C)CNC(c2cc(C#N)cn2C)=O)cccc2nc(O)[nH]c12 5368,n1(CC(=O)NCC2CC(CNC(C3(C(=O)OC)CC3C)=O)C2)cc(C(N)=O)cn1 5369,CC(F)(F)CC(=O)NC1CCC1NC(=O)COc1ncccc1C(F)(F)F 5370,N1(C(C(C)N(C)C)=O)CC(O)CC1CNC(C1CCC(CC(=O)N(C)C)CC1)=O 5371,Cc1cncc(C(=O)NC2CN(C(c3cn(C)nn3)=O)CCC2C(F)(F)F)c1C 5372,c1(C2(NC(CNCc3n(C)cc(Br)c3)=O)CC2)ccc(C(F)(F)F)cc1Cl 5373,c1(CC)cc(C(=O)NCC2CCN2C(c2c(NC(C)=O)c[nH]c2C)=O)cc(O)n1 5374,CCCCC(C(=O)N(CCNC(c1cnn(C)c(=O)c1)=O)C(C)C)N(C)C 5375,c1(CN(C(=O)CC2(CNC(C3CC3Cl)=O)CC2)C)cncnc1 5376,N1(C(C(CCC)NC(C)=O)=O)CCN(C(C2CN3CCN2CC3)=O)C(C(C)C)C1 5377,C1(C(=O)Nc2ccc(OCCOC)cc2)CCCN(C(=O)CSC(C)=O)CC1 5378,N1(CC(=O)NC2CCC(CCC(=O)N3CC(SC(F)F)C3)C2)CCNC(=O)C1 5379,Cc1cccc(CC(=O)NCC(C2CCC2)NC(c2cc(O)ncn2)=O)c1 5380,CC1(C)CCC2(CCCN2C(c2ccc(S(C)(=O)=O)cc2)=O)CC1 5381,C1(NC(c2nc(CNC(C=C(C)C(C)(C)C)=O)oc2)=O)CN(C)CC12CC2 5382,c1(NC(C2C3C(NC(C(CC)=CCCC)=O)C4C(C3)C42)=O)c[nH]c2ncccc12 5383,n1(CC)ncn(NC(=O)CN(C(=O)C(CC(C)C)NC(N)=O)C2CC2)c1=O 5384,N1(C(c2cncc(SC)c2)=O)CC(NC(=O)C(C)C(C)(F)F)CC1(C)C 5385,CCC(C)C(C)C(=O)NCC1(C)CCN(C(c2cn(C)nc2C2CC2)=O)C1 5386,N1(C(C2N(C(c3csnn3)=O)CCC(=C)C2)=O)CCN2CCCCC2C1 5387,CCCCC(C(=O)N1CC2(CCN(C(C3CN4CCN3C(C)C4)=O)C2)C1)C(C)C 5388,CN=c1cc(C(=O)NCC23CC(NC(C4CCOC4C)=O)(CO2)C3)cc[nH]1 5389,c1(OCC=C)cccnc1C(=O)N(CCNC(=O)COCC(F)F)C1CC1 5390,c1(C(=O)NCC2OCCN(C(c3c(C)ccs3)=O)C2)ccc(N)c(F)n1 5391,Nc1c(C(N2CC=CC2CNC(=O)C(c2ccc(F)cc2)O)=O)nc(O)nc1O 5392,C1(O)(C(N2CCCC(CCNC(CCC=C)=O)C2)=O)CCCC(C)(C)C1 5393,C(=O)(C1CCc2c[nH]nc21)N(CCNC(C1CC2(CCO1)CC2)=O)CC 5394,C1(NC(Cn2cc(-c3cc(N)cc(F)c3)nn2)=O)CCc2nncn2C1 5395,Cc1nc2ccc(C(N3CCCC3C(C)(C)CNC(=O)CCC3CC3)=O)cc2o1 5396,C1(NC(C2C(C=C)C2)=O)COC2(C1)CN(C(=O)Cc1cncc(O)c1)C2 5397,c1(C(N2CC(NC(C3(COC)CC3)=O)C(OC)C2)=O)ccc(O)c(CO)c1 5398,c1(C(=O)NC2C(CNC(c3n(CC)cc(Cl)c3)=O)CC2)n[nH]c2c1CC1CC21 5399,CCCCC(C)CCC(=O)NC1CC(NC(=O)C(C)n2cccc2)C1 5400,c1(N(CC(N2CCCCC2C)=O)Cc2c(C)n[nH]c2C)ccc(N)cc1F 5401,CCC(C)CC(C)C(=O)N1CCCC(NC(=O)CN2Cc3ccccc3C2)C1C 5402,C1(N(C(=O)CCc2ncc[nH]2)C)CCCCN(C(c2c[nH]c(Br)c2)=O)C1 5403,c1(C(C)=O)cc(C(=O)NCC2CCC(NC(=O)COC3CCOC3)C2)cs1 5404,C=CCN=C(NCCC1CC1(F)F)N1CCC(COC(F)(F)F)CC1 5405,N1(C(Cn2ncc(C#C)c2)=O)CCC(C(=O)NC(c2ncc(C)o2)CC)CC1C 5406,N1(C(C2CN(CC)C2)=O)CC(Nc2cnccc2C2CC2)C(F)(F)C1 5407,N1(CC(C(=O)C(F)CC2CCOCC2)=O)CCCN(c2nnc(COCCO)s2)CC1.OC 5408,C1(CN(C(=O)C2=CC(C)(C)C2)C)CN(C(c2cc(Cl)c(Cl)n2C)=O)CC12CC2 5409,S(=O)(=O)(c1ccc2c(c1)OCCO2)NC1CCN(C(=O)OCc2ccccc2)C1 5410,c1(C(=O)NC(C(C)C)CNC(=O)Cc2cnoc2)cccc2nncn12 5411,N(C1CCc2ccc(Br)cc21)C(C(N1CCCC(CCC(C)O)C1)=O)=O 5412,N1(C(CC(COC)C)=O)CC2CCCC(CNC(C3(O)CCCC3)=O)(C2)C1 5413,C(=O)(CC(C)(O)C(F)(F)F)NCC1(CNC(C=C(C)c2cccs2)=O)CC1 5414,c1(C(N2CC(Cn3cc(-c4cncc(C)n4)nn3)C2)=O)ccc(Br)c(Cl)c1F 5415,c1(NC2(c3n(C4(C)CC4)nnn3)CSC2)cnc(NC2CCOC2)c(Cl)c1 5416,c1(OC)ccc(NC(C2(C)CCCN(Cc3cccc(F)c3)C2)=O)c(F)c1 5417,C1(C(N2CC(c3ccco3)C2)=O)CC2CCC1N2C(=O)C(O)CC1CCCC1 5418,CCCCC(C(=O)NC1CCC(NC(c2ccc(F)cn2)=O)C1)C(C)C 5419,C1(CNC(CCN(CCC)C)=O)CC(F)(F)CN1C(=O)C(CC)NC(N)=O 5420,CCC(C)CC(C(=O)NCc1cncc(F)c1)NC(c1c[nH]cc1C)=O 5421,C(=O)(CC(C)(C)COC(C1COC(C)(C)OC1)=O)OC 5422,N1(C(c2ccc(OC)o2)=O)CC(NC(c2ncoc2-c2cc(C)no2)=O)C(C)C1 5423,C1(F)(CNC(C(C)OCC)=O)CCCN(C(C2(CO)CC(C)(C)C2)=O)CC1 5424,C1(NC(=O)CCOCC2CC2)CC(O)CN(C(C2CCC3(CC3)C2)=O)C1 5425,C1(C(=O)NCC(CCNC(=O)C=CCF)OC)CCc2nn[nH]c2C1 5426,CC12CC(C(=O)NC3CN(C(C4(O)CCSCC4)=O)CC34CCC4)(C1)C(C)(C)O2 5427,N1(C(C(CC=C)(C)C)=O)CC2(CCN(C(C3C=CCS3)=O)C2)C1 5428,C1(NC(=O)COCc2nc[nH]n2)CC2(C1)CC2NC(C1CC(n2ccnn2)C1)=O 5429,N1(C(C2ON=C(C)C2)C(=O)NCC2CC2)CCC(=Cc2ccccc2)CC1 5430,CC1CCN(C(=O)C(C)Sc2ccc(Cl)cc2Cl)CCN1C(C1CC1C)=O 5431,CC(C)C(C)C(=O)NC1CC(CCNC(=O)C(N2CCSCC2)C)C1 5432,C(=O)(CN=c1ccc(Cl)n[nH]1)NC1CCN(C(c2ccnc(OC)n2)=O)C(C)C1 5433,CCC(CC)C(C)C(=O)N1CCN(C(=O)C(=O)NCC2CC2)CC1CC 5434,CC12CCC(C(=O)NC3CC(NC(c4ccnc(O)c4)=O)C34CCC4)(CC1)CO2 5435,C(=O)(CC1=C(C(=O)OC)C(c2[nH]cnc2C)NC(=O)N1C1CC1)OC 5436,N1(C(C2CCN(C(C)=O)C2)=O)CC2CCN(C(=O)COc3ncccc3O)C2C1 5437,c1(C(N2C(CNC(CC(C)OC)=O)COCC2)=O)cccc(Cl)c1C(F)F 5438,C1(NC(CC2N(C)CCCC2)=O)CCC2CN(C(C3CC3(C)C(F)F)=O)CC2C1 5439,c1(CN(C)CC2N(c3nnc(C)s3)CCCC2)ccc2c(c1)C(=O)NC2=O 5440,CC1(C)C(NC(c2ccncn2)=O)C2CCCN(Cc3csc(Br)c3)C12 5441,c1(COC)nc2ccccn2c1C(=O)NCC(C)NC(C1(C#N)CCOC1)=O 5442,c1(C(=O)NC2(CC=C)CN(C(=O)CC(C=C)CCC)C2)cc2c(cnn2C)nc1C 5443,C1(NC(C2C(CC)OCC2)=O)CCSC12CN(C(C1CC(=O)N(C(C)C)C1)=O)C2 5444,C1(C(CNC(C=CSC)=O)(C)O)CCCN(C(c2ncsc2C)=O)C1 5445,CCCS(=O)(=O)c1ccccc1S(=O)(=O)CCNC(=O)NC1(C(=O)OC)CC1C 5446,c1(C(=O)NC(CNC(=O)OCC)C)cn(C)nc1C(N1CCCC1)=O 5447,C#Cc1ccc(CNC(=O)Nc2c(C)nn(C)c2CC)nc1 5448,C1(C(N2CCC(O)(CNC(CCS(C)(=O)=O)=O)C2)=O)CS(=O)(=O)CC12CC2 5449,CCN=C(NCCC12CC(CO1)C2)NC1CCCC(F)C1 5450,c1(CNC(=O)NC(C2CCCO2)CC)ccc(S(C)(=O)=O)c(OC)c1 5451,N1(C(CO)=O)CC(=O)NC1=O.C1(CNC(COCCCN(C)C)=O)CCN1C(=O)C 5452,N1(C(CCCCC=C)=O)CC2(CCN(C(c3nc4ccccc4[nH]3)=O)CC2)C1 5453,C1(CC)C(C(N2CCC3CCC23)=O)CCN1C(C1CCN(C)C1)=O 5454,C1(CN)CCCCC1C(N(C(C)C(C(=O)C(C)CC1CCCC1)=O)CC)=O.OC 5455,Cc1c(C(N2CCCC(NC(C3(C)CNC(=O)C3)=O)CC2)=O)cccc1C1CC1 5456,CC(CCCC(=O)N1CCOC(CCF)C1)NC(=O)COCCN(C)C 5457,c1(C(=O)NCCCOCCN(C(c2c(C)cco2)=O)C)cc2cc(O)ccc2[nH]1 5458,C1(C(N(CCCNC(C(C)OC)=O)CCO)=O)CC(=O)NC(=O)N1 5459,C1(NC(c2ncn(CC)c2)=O)C(C)CN(C(C2(OC)CCOCC2)=O)CC1C 5460,C1(C)(C(=O)NCc2ccc(CC)cn2)CC(O)CN1C(c1cnccc1C)=O 5461,N1(C(c2ccc(CC)nc2C)=O)CCN(C(c2ocnc2C)=O)CC12CCC2 5462,c1(CCC(=O)NCC2(F)CCN(C(C(C)C(F)F)=O)C2)ccc2cccnc2c1 5463,C(C1CN(C(c2csnn2)=O)Cc2ccccc21)NC(CCC1(C)CC1(F)F)=O 5464,N1(C(c2c(C)ncc(C)c2)=O)CC2CCN(C(c3ccc(C)c(Cl)c3N)=O)CC12 5465,c1(N(CC(=C)C)C)nc2cc(OC)ccc2c(=NCC2(CC)CCC2)[nH]1 5466,c1(C(=O)NCCOC2CN(C(C3CC(O)C(F)C3)=O)C2)cc2c(cn1)OCCC2 5467,CCC(C)(CNC(=O)CC(C)N(C)C)C(=O)NCC1(CO)CC12CCC2 5468,C(=O)(C(F)(F)C1CCCC1)NCCN(C(=O)CCc1n[nH]c(=N)s1)C(C)C 5469,C1(C(N2C(CNC(c3cc(CC)[nH]n3)=O)CC(O)C2)=O)CCC(F)(F)CO1 5470,C1(CNC(c2ccc(CO)s2)=O)CCCCCN1C(=O)C(F)CC1CCC1 5471,S(=O)(=O)(c1ccc(C#N)c(NCCC2CC2(Cl)Cl)c1)NC(C=C)(C)CC 5472,c1(SCC(=O)NCC=CCNC(C2=C(C#N)CCC2)=O)ccc2c(c1)OCCO2 5473,N1(C(CN2CC(CC)C2)=O)CCCC(O)(CNC(C2CC3C=CC2O3)=O)C1 5474,CC1CCCc2c(C(=O)O)cnn21.C12NC(=O)CCC1NC(=O)Cn1cc2nn1 5475,N1(C(C2(CC)CC2)=O)C2CCC1C(C)C(NC(c1c(C)coc1C)=O)C2 5476,C(=O)(CCCS(N)(=O)=O)N(CC)CC1CCCCN1C(C1CC2CCC1O2)=O 5477,C(=O)(C(O)C(C)(C)c1ccc(Cl)cc1)N(C1CCN(C(=O)CO)CC1)CC 5478,Cc1ccccc1CC(=O)N(CC(C)CNC(c1ccc(SC(F)(F)F)s1)=O)C 5479,C1(N(C(CCCOC)=O)C)CC2CCC(C1)N2C(=O)Cc1cccc(Cl)c1F 5480,c1(C(N2CCC(C)C(NC(c3scnc3Cl)=O)C2C)=O)cc([N+](=O)[O-])cnc1N 5481,c1(C(=O)NCc2nc(C)c(C(N3CC=CCC3)=O)o2)cc2cccnc2[nH]1 5482,Cc1ccnc(O)c1C(=O)NCC(C)CNC(=O)C(c1ccc(C#N)cc1)O 5483,c1(C(=O)NCC(CNC(c2c(C)con2)=O)CO)cc2c(C3CC3)cccc2[nH]1 5484,C(N=C(NCC1CSCCO1)N1CCC(O)CC(C)(C)C1)c1n(C)ncc1 5485,Cc1nccc(C(=O)NC2(CCNC(=O)COc3ccsc3Cl)CC2)n1 5486,N1(C(C2C(OCC)C2)=O)CC(C)C(Nc2ncnc(C(C)(C)C)n2)C(C)C1 5487,C(=O)(CC(C)(C)C(=O)OC)NC1C(C(=O)Nc2cnc(CCC)nc2)CCC1 5488,c1(C(C)=O)cc(=NCCCCNC(c2ccc3c(c2)NC(=O)CO3)=O)[nH]cn1 5489,C(=O)(CCCCCNC(=O)C(c1cc(C)sc1C)N(CC(=O)NC1CC1)C)OC 5490,CN1C(=O)CCC1(C)CNC(=O)CCCNC(C1CC=CCC1)=O 5491,Cc1cc(F)cnc1C(=O)NC1COCCN(C(=O)CCC2(C)CC2(F)F)C1 5492,N1(C(C2C(C)(C)C2C#N)=O)CC23CCCC2(C1)CN(C(=O)CCOC1CC1)C3 5493,N1(C(C(=O)NCCOC)=O)CCCN(C(c2ccnc(OC)c2)=O)CC1C(C)C 5494,C12(CNC(C(C)N(C)C(C3CC(CC4CC4)C3)=O)=O)CCCCC1C2 5495,C(C(C(=O)N(CCNC(c1cccn1C)=O)C(C)C)NC=O)SC.C(C)(=O)O 5496,N1(C(C(CCCNC(CC(CC)O)=O)O)=O)CCC(C2CCC2)CC1 5497,N1(CC(c2c(C)c(I)nn2C)=O)CCC(OCCO)C(F)(F)C1 5498,C(=O)(C(F)(F)c1ccncc1)N(C1CCN(C(C2CCCC2C(=O)O)=O)C1)C 5499,c1(-c2n(CCC=C)c(N3CCn4cccc4C3)nn2)ccc(S(=O)(=O)NC)cc1 5500,C(=O)(C(Cl)=CCl)NCCN(CC(C)O)C(c1cn(C2CCCCC2)nn1)=O 5501,C1(CNC(CC(=C)C)=O)(CO)CC12CCN(C(=O)COCP(C)(C)=O)CC2 5502,c1(C2C(C(N3CC(NC(CNC(CC(C)(C)C)=O)=O)C3)=O)C2)ccc(F)cc1Br 5503,c1(NC(C2CCCN(C(=O)CC3CCCOC3)C2)C)ncccc1C#N 5504,N1(C(CN2CCC(N(C(C(C)CC3CC3)=O)C)CC2)=O)CCc2ccccc21 5505,N(C(=NCC1OCCC1)N1CCC2(C1)CC(F)(F)C2)CC1CCCS(=O)(=O)C1.C1(C)CC1 5506,c1(CN(C(CC(C)(C)n2cc(CCC(C)O)nn2)=O)C)c(C(=O)NO)cnn1C 5507,c1(NC(C2C(C(N(c3ccn4ccnc4c3)C)=O)C2)=O)cc2ccccc2n1C 5508,c1(C(N(C2CCN(C(=O)CC3COCC3O)C2)CCC)=O)ccoc1Br 5509,C1(NC(c2ccc(C(C)=O)[nH]2)=O)CCCCC1CC(=O)NC(C)C 5510,c1(C(=O)NC2CC(CCNC(=O)CSc3ccccc3)C2)cncc2nc[nH]c12 5511,N1(C(C)Cn2cc(CCC(=O)CC(F)(F)Br)nn2)CC(CC(=O)O)OC(C)C1 5512,N1(C(c2cc(F)cc(F)c2)=O)CC2CCC1CN2C(C12CC3CC1C2C3O)=O 5513,C(=O)(C1=NOC(C)(C)C1)NCC(CNC(c1cc(CC)[nH]n1)=O)OC 5514,CCC(C)C(O)CC(=O)N(CCC(=O)NCCC1CC(=O)N(C)C1=O)C1CC1 5515,N1(C(C=C(C)C(F)F)=O)CC2CCC1C(NC(=O)CC1CC3CCC(C1)N3C)C2 5516,C=CC(C)(C)CCCNC(c1cccc(Br)c1Cl)C 5517,CC1CCN(C(=O)COCC(c2ccccc2)C)CCN1C(c1cc[nH]n1)=O 5518,C1(C(C)C)CCC(C)CC1C(=O)NCC1C(C(C)C)CCN1C(=O)CN=S(C)(C)=O 5519,C1(CNC(=O)C=Cc2ncc[nH]2)CN(C(C2(C3CCC3)CC2)=O)CCC12CCC2 5520,c1(OCCNC(=O)Nc2ccc(NS(C)(=O)=O)cc2)cc(Cl)c(Cl)cc1Cl 5521,N(C1CCS(=O)(=O)c2ccc(Cl)cc21)C(=O)NC(CCCCC)C 5522,CC1CCCC(NC(C2(CN(C3CN(C(=O)OC(C)(C)C)C3)C)CC2)=O)C1C 5523,C1(NC(C(C)=CC)=O)CN(C(c2cnn(CC(F)F)c2)=O)CCC1C 5524,C(CN=C(NCc1cccs1)N(C)CC1CCOC1)c1c(C)n(C)nc1 5525,N1(C(CC2CCCC(NC(CN(CC)CC)=O)C2)=O)Cc2cccc(O)c2C1 5526,c1(C(=O)NCCCN(C(=O)Cc2cc(C)ccc2F)CC)ccc(N)cc1F 5527,C1(C(N2CCC23CCCSC3)=O)CCN(C(=O)Cc2ccsc2)O1 5528,N1(C(CCC)C(=O)NCc2ccc(Br)cc2)CC2CC3CC2C1C3O 5529,N1(C(C2C=CCN2C(=O)CN2CSCC2=O)=O)CCC2(CCOC2=O)C1 5530,Cc1cc(C2CC2)ncc1C(=O)NC1CC(CCNC(C2(C)CCCN2C)=O)C1 5531,N1(C(c2nc(C)oc2)=O)CC2CCC1C(CNC(=O)CCCCF)C2 5532,c1(C(N2CC(CC(CNC(CC3ON=C(C)C3)=O)(C)C)C2)=O)cc(C)nc(O)n1 5533,c1(C(=O)NC(CNC(C(C)OCCCC)=O)C)cccn1C1CC1 5534,C(=O)(C(C)(C)C(F)(F)CC)NCC12CC(NC(CN(CC)CC)=O)(C1)C(C)(C)O2 5535,C1(NC(=O)Cc2ccc(O)cn2)CC2CCC(C1)N2C(=O)C1=NNC(=O)C1 5536,C1(N(C(C2C(C(=O)NCC#C)C2)=O)C)CN(C(c2cc[nH]n2)=O)CC12CC2 5537,CC1CN(C(c2csc(Cl)n2)=O)CCC1NC(C1(c2ccccc2)CCC1)=O 5538,N1(CC)CCN(CCC(N2CC3CC3(NC(=O)CC3CC4CC4C3)C2)=O)CC1 5539,C1(C(N2CCN(C(c3nc(N(C)C)nc(=N)[nH]3)=O)CC2)=O)Cc2ccncc2C1 5540,c1(C(N(CCOCCNC(C2C(=C)CC2)=O)C)=O)ccoc1CC(=O)OCC 5541,C=C1CC(CC(N2CC(C)(OCC(=O)N(C(COC)CO)C)C2)=O)(CO)C1 5542,C1(NC(c2cc(OCC)n[nH]2)=O)C2CC1N(C(C1(C(F)(F)F)CC(F)C1)=O)C2 5543,C1(NC(c2c(OC)cc(O)nc2)=O)C(C)(C)C(NC(=O)C=CC(=O)N(C)C)C1(C)C 5544,c1(C(=O)NCC(CCNC(CCSCC)=O)O)ccc2cnc(C)n2c1 5545,CCC(C)(O)C(=O)N1CC(NC(=O)C(O)Cc2cnn(C)c2)C(O)C1 5546,c1(OCC)ccc(Cl)nc1C(=O)NCC1CCCC1NC(=O)C(C)c1ccco1 5547,c1(CC(N2CC(O)(CNC(C3CCSCC3)=O)C2)=O)cncc(O)c1 5548,C(=O)(C1CCc2c(F)cccc21)NC(c1ccc(OC)cc1Br)C 5549,c1(C(=O)NC(CC(C)NC(c2ncoc2C2CC2)=O)C)ccnc(NC(N)=O)c1 5550,c1(C(N2CC3C(NC(C4C(C)(C)C4(F)F)=O)(C3)C2)=O)oc2ccccc2c1Cl 5551,C1(CNC(CC(CCC)O)=O)CCN(C(C2(SCCCC)CC2)=O)CC1(F)F 5552,c1(C(N2CC(OC)C(NC(=O)Cn3cccnc3=O)C2)=O)cnc2[nH]ncc2c1 5553,N1(C(CC2N(CC)CCC2)=O)CC2CCCC(CNC(=O)COC(F)F)(C2)C1 5554,C(CC(CC)C(=O)NC1CC(C(F)C(N2CCC3(CC2)N=N3)=O)C1)=CC 5555,C1(NC(=O)CCC2CCCC(O)C2)CC2CC1N(C(C1CC3C=CC1CC3)=O)C2 5556,N1(C(Cn2ncc(C#C)c2)=O)CCC2CN(C(=O)CCC3CC(F)(F)C3)CCC12 5557,c1(C(=O)NCC2N(C(CC=C=C)=O)CCC(C)C2)cc(OC)c2c(c1)CC(C)O2 5558,c1(COC)ccoc1C(N1CCC1CNC(c1ccn(C2CC2)n1)=O)=O 5559,Cc1ccc(C(=O)NCC2C3CN(C(C4CC(n5cccn5)C4)=O)CC23)cc1 5560,C1(C(=O)OC)CCCN(Cc2ccc(F)cc2-c2nn[nH]n2)C1C 5561,N1(Cc2cc(OCC)c(O)cc2)Cc2[nH][nH]c(=NC(=O)c3cnn(C)c3)c2C1 5562,C1(NC(C2C(OC)CCC2)=O)(CO)CCN(C(c2ccc(C)[nH]2)=O)CC1 5563,CC1CCC(C)CN1C(=O)CSCCNC(c1csc(O)n1)=O 5564,C(=O)(CC(CN(C)C)C(F)(F)F)N1CC(O)(C(C)NC(C=C(C)C2CC2)=O)C1 5565,C(C(CC(C)C)C(=O)NC(CC(F)F)C(=O)N1CCC(n2cnnn2)C1)OC 5566,N1(C(c2cccnc2O)=O)CC2CC(C1)N2C(=O)CC(O)c1ccccc1 5567,c1(C(=O)NCC2C(C)CN(C(C3CC34CCCC4)=O)CC2)cccc2cnsc12 5568,C(CC(F)F)(C(=O)NC(C)C(O)C(F)F)NC(c1c(C)non1)=O 5569,c1(C(=O)NCC(Cc2ccc(C)cc2)F)cc2c(Br)cncc2[nH]1 5570,Cc1cccc(C(N2CC=CC2CNC(=O)CC2CC(c3ccccc3)C2)=O)n1 5571,n1(CCOC)ncc(C(=O)NCC2CN(C(c3sc(C)nc3C)=O)C3CC23)c1C 5572,c1(CC(=O)NC2CCC(C(N3CC(C)C(O)CC3)=O)CC2)c[nH]c2ccccc12 5573,N1(C(C2N(C(c3coc(CO)c3)=O)CCN(C)C2)=O)CCC12CC(C)(CO)C2 5574,N1(C(CCCC#C)=O)CCCC2CN(C(=O)CCS(=O)(=O)NC)CCC12 5575,CC(C(=O)N1CC(C2CCCO2)C1)C(=O)c1ccccc1 5576,N1(C(CC(CC)O)=O)CCCCC(C2CN(C(c3cc(C)ccc3F)=O)C2)C1 5577,N1(C(CC(C)n2cccn2)=O)CCC2(COC(CNC(c3cnns3)=O)C2)C1 5578,c1(OC)nc(NC2CCCCC2NC(=O)CCc2ccc(F)nc2)nc(C)c1F 5579,N1(C(c2cc(COC)[nH]n2)=O)CC(C)CN(C(=O)Cc2c(C)noc2C)C(C)C1 5580,Cc1cc(NC(C2C=CCCC2)=O)ccc1NC(c1cn(CCN(C)C)nn1)=O 5581,C1(CNC(CCCC(=C)C)=O)CN(C(=O)C=C(C)C(F)F)CCC12CCOC2 5582,N1(C(c2c(OC)cncn2)=O)CC(O)CCC1C(=O)N(C)CC1(CO)CC1 5583,C1(OC)CC2(C1)CC2NC(C1(COC)CCN(C(c2cc(C(C)C)no2)=O)C1)=O 5584,C12(C(=O)NC3(C=C)CCC3)CCC(CN(C(C3C4COCC34)=O)C1)C2.OCC 5585,c1(NCC(=O)OC)ccc(C(=O)NCCC2OCCCO2)c(OC)c1 5586,c1(C(N2CC3(CCC3(F)F)C2)=O)nn2c(c1Br)OCCC2 5587,C1(OC)(OC)CCC(C2(NC(c3ccccc3)CC3CS(=O)(=O)C3)CC2)CC1 5588,C(N=c1[nH]c(N2CCCCC(F)(F)C2)nc2c1CCC2)C1(Br)C(F)(F)C1 5589,C(=O)(C1CCCc2nccn21)NC(CCCC)CNC(c1cc(C)oc1C)=O 5590,c1(C(=O)NC(CNC(COCC(=C)C)=O)C)c(C)c(Br)n(C)c1C 5591,C(=O)(C(C)CNC(=O)C1CC1)N(C(CSC)C)C 5592,CC1CC2(CCO1)CC2C(=O)NCC1CCCCN(C(c2c[nH]ccc2=O)=O)C1 5593,O=C1CCCC(c2ccccc2)(CNCCCF)N1 5594,N1(C(=O)CCC=CBr)CC2(CCN(C(C3CCC4CCC(=O)N34)=O)CC2)C1 5595,C(C(O)C(=O)NC(c1cc(C)[nH]n1)C)SCC 5596,C12(CNC(=O)CC3CCC34CCC4)CCCC1N(C(=O)C=C1CCCCC1)CC2 5597,c1(C(N2CCCN(C(C3CCN(C(C)=O)C3)=O)CC2)=O)ccc(Cl)c(N)c1Cl 5598,C1(C(=O)NCC2(F)CN(C(CC=CC(C)(C)C)=O)C2)CC2C=CC1C2 5599,C1(NC(C(CC)NC(=O)C(C2CCOCC2)F)=O)CC2OC(=O)CC12 5600,C1(CCC)CN(C(C2(C#N)CCCC2)=O)CC1C(=O)N(CCCO)CCC 5601,c1(C(=O)NC(CC=C)CNC(=O)Cc2cncnc2)cncc(Cl)c1C 5602,C1(N(C(C=CCCC)=O)C)CCCC(NC(=O)CCn2ccnc2)C1 5603,c1(C(N2C(C(C)(C)NC(CC(C)OC)=O)CCC2)=O)ccnc(C(F)(F)F)c1 5604,c1(C(N(c2cc(OC)ncn2)C2CC2)=O)ccc2c(C3=CCNCC3)n[nH]c2c1 5605,Cc1nc2nc(=S)n(CC(=O)NNC(=O)c3ccc(C#N)cc3)n2c(C)c1C 5606,C12(C(=O)NCCCOC=C)CCC(NCc3cc(O)cc(Cl)c3)(CC1)CC2 5607,N1(C(Cc2cc(C)no2)=O)CCC(NC(C2C=CCS2)=O)C(O)C1 5608,c12ccc(nc1)C(=O)NC2.C1(CC)CCCC1C(=O)NOCC=CCl 5609,c1(C(=O)Nc2cccc(C(=O)NC(CC)C)c2)cnc(F)c(C)c1 5610,C(=O)(C1=C(Cl)CCC1)NC1CC(F)(CNC(c2c(NC)nccc2)=O)C1 5611,N1(C(CNC(=O)OC)=O)CCOC(C)(CNC(=O)Cc2cnc[nH]2)C1 5612,CC(CC(N)=O)C(=O)N1CCCC(N2CCN(C(c3c[nH]ccc3=N)=O)CC2)C1 5613,N1(C(c2ccc(OCC)cc2)=O)CC2(CCC2NC(c2ccc(CO)s2)=O)C1 5614,C1(NC(CC=CCC)=O)CC(C)CN(C(c2ccc(=O)n(CC(F)(F)F)c2)=O)C1 5615,N1(C(C(C)C2CCC2)=O)CCOCC(NC(c2occc2-c2cnn(C)c2)=O)C1 5616,C1(C(N)=O)CN(C(c2cccc(O)c2)=O)CCC1NC(=O)CC1CC=CCN1C 5617,C1(F)(CNC(COCc2n(C)ncc2)=O)CCC(CNC(C2CCCO2)=O)CC1 5618,C(C(=O)N(C)CC1CCCC1NC(=O)COC1(C)CCCC1)(C(C)(C)C)OC 5619,C1(NC(c2c(C)onc2C2CC2)=O)CCN(C(c2ccc(N)c(Cl)n2)=O)CC1F 5620,Cc1c(C(=O)NC(C(N2CC[Si](C)(C)C2)=O)C2CCCC2)ccn1C 5621,C1(NC(C=CCC2(NC(C(C(CC)O)C)=O)CCC2)=O)CC(C2CCCC2)C1 5622,C(=O)(C1=CC2(CCN(C(=O)CCc3nccn3C)C2)C1)NCC(=O)N(C)C 5623,N1(C(C2C(C)(C)CC2)=O)CC(NC(c2cc(N)ccc2O)=O)CC(O)C1 5624,CC1(C)CC(O)(CC(=O)NCC(F)(C2CCOC2)NC(C23CC(C)(CO2)C3)=O)CO1 5625,CNS(=O)(=O)N1CCC(C(=O)N(CCCN(C(=O)CCNC(=O)CO)C)C)CC1 5626,C1(C)(CC)CC(NC(=O)Cc2ccc(C)s2)CN1C(=O)CCCCOC 5627,c1(N(CCOCCN(C(C2C(CCC)CCC2)=O)C)C)ncnn2c(Br)ccc12 5628,c1(OC)ccc(OC)c(C(=O)NCC(C)(O)CNC(C2(C)CC(C)=NO2)=O)c1N 5629,c1(C(=O)NCC(c2cccc(OC(C)C)c2)O)ccc(S(C)(=O)=O)nc1 5630,c1(C(N2CC(C(=O)NCC3OCCN(C)C3)OCC2)=O)cccc2ccoc12 5631,n1(CC(=O)NC(C(C)NC(c2cnc(C)s2)=O)C(C)C)ccc(=O)cc1C 5632,CC(C)CC(C)CC(=O)NC1CCN(C(=O)C2=CS(=O)CCC2)CC1O 5633,c1(CCC(=O)NC23CC(NC(C4NC(=O)OCC4)=O)(C2)C3)cc2ccccc2[nH]1 5634,C(=O)(C#CC(C)(C)CNC(=O)C=C(C1CC1)C1CC1)NCC1C(C)C1 5635,c1(SCC=C)ccccc1C(N1CC(NC(=O)C(c2cccnc2)O)C(C)C1)=O 5636,C1(C(N2C(CNC(c3c(C)cnnc3O)=O)CC2)=O)Cn2c(C)nnc2CN1C 5637,C1(CNC(C(C)(C)C2CCCCO2)=O)CCN(C(=O)Cc2nc[nH]n2)CCC1(F)F 5638,c1(CC)cnc(C(c2nnnn2CCOC)NCc2ccc(OCC3CC3)s2)[nH]1 5639,Cc1ccc(NC(C2CCCC(NC(=O)Cc3ccc(Br)cc3I)C2)=O)c(I)n1 5640,c1(C(=O)NCCCCCC(=O)N2CCC(OC)C2C)nccc2[nH]ccc12 5641,N1(C(c2ncc(C)s2)=O)CCc2c(Br)ccc(NC(c3ccnnc3)=O)c2C1 5642,C12(c3onc(-c4c(OC)ccc(F)c4F)n3)CCCN(C1)S(=O)(=O)C2 5643,CC#CCCCC(=O)NC1CC(CNC(C2CCCCO2)=O)C1 5644,C1(C(=O)NC2CN(C(=O)Cc3ccc(-n4cccn4)cc3)C2)CC(C2CC2)=NO1 5645,C(c1ccc(F)c(F)c1)=C(C)C(=O)NC1(C)CCN(C(C2CCOCC2)=O)C1 5646,C1(NC(c2nc(C)[nH]c3nccc2-3)=O)CC2CCC1(N=c1[nH]ccnc1F)C2 5647,c1(OC)cc(C(N2CCC(NC(c3ccc(C)c(N)c3)=O)C(C)C2)=O)ccc1Cl 5648,c1(C(=O)NCC(CC)NC(C2CCC2c2nc[nH]n2)=O)nc2cccnc2s1 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5685,c1(C(N2C(C(=O)NCC(C3CCC3)OC)CC(O)C2)=O)cc2cccnn2c1 5686,Cc1nccc(=NCC2CCN(C(C3(C)CC=CCC3)=O)C2)[nH]1 5687,C1(CNC(C)=O)(CSC2(c3ccc(F)cc3)CC3(CC3)C2)CCCCC1 5688,Cc1cc(C(=O)NCCC2(C)CCN(C(=O)Cc3nc(=N)[nH][nH]3)C2)c(C)s1 5689,N1(C(c2c(COC)noc2)=O)CC2CC(C1)CN(C(=O)C(C)(C)C1CCC1)C2 5690,c1(C(=O)NCCC2(C)CC2(F)F)cc(S(=O)(=O)Cc2ccccc2)ccc1F 5691,c1(OC)ccc(CN2CCN(Cc3ncccc3O)C3CC23)c(C)c1C 5692,CC(C)(C)CC(C(=O)NC1(C)CC2(CCC2)C1)NC(=O)Cc1cncnc1 5693,c1(OCC(=O)NC2CCCC2CNC(c2ccnc(O)c2)=O)ccc(Cl)cc1F 5694,Cn1cc(S(=O)(=O)N2CCCC2c2cn[nH]c2)c(C(C)(C)C)n1 5695,C#Cc1ccc(C(=O)NC(CCC=C)C(=O)NC(C)CCC=C(C)C)nc1 5696,c1(C(=O)NC2CCN(C(c3nn(C)c(Cl)c3)=O)CC2F)c(Br)cc(F)c(Cl)c1F 5697,C(=O)(CCCCC(C)CC)NCCC(=C)CNC(c1csc(Cl)c1)=O 5698,CCCC(C)(CC)C(=O)NC1CCCC(NC(c2ccc(O)c(C)c2)=O)C1 5699,N1(C(C2C(C(=O)OC)C2)=O)CCN(C(=O)COc2cccc(Cl)c2)CC1CC#N 5700,N1(C(c2cc(C)c(Cl)c(N)c2)=O)CCC2(CC1)CN(C(=O)CC1CC3CC3C1)C2 5701,C1(NC(=O)CCc2ccncc2)CCCCC1NC(=O)Cn1cc(Br)cn1 5702,C(=O)(C1CCc2ccccc21)N1C(CN(C)C(C2CC(N=[N+]=[N-])C2)=O)CCCC1 5703,CC(C)CCCCC(=O)N(C(C)CN(C)C(c1cccc(Cl)c1)=O)C 5704,CC(C(=O)NC1CC(NC(=O)COCc2nnc(S)n2C)CC1O)C(F)F 5705,CCC(CCO)NC(=O)CCC1(NC(=O)C=Cc2cc[nH]c2)CCC1 5706,C12(Cn3c(=O)c3=O)CCC(CC1)CN2.c1(C(N2CCCC2)C)ccnn1C 5707,CCCCC(CN=c1nc(CC(C)C)cc(C)[nH]1)NC(c1n[nH]c2c1CCC2)=O 5708,N1(C(c2c(CC)cco2)=O)CC(NC(=O)Cc2cc(C)cc(F)c2)C2(CCC2)C1 5709,c1(C(=O)NC2CCC(NC(c3cnc(CCC)s3)=O)C2)ccnc2c1nnn2C 5710,C1(C(=O)NCC2(NC(CSCCCC)=O)CC2)CNC(=O)N1C 5711,c1(OC)cccc(Br)c1C(N1CCC(N(C(=O)CCSC)C)C(C)C1)=O 5712,Cc1cc2ncc(C(=O)NCC3CC(C)CCN3C(C3CC3(Cl)Cl)=O)c(C)n2n1 5713,N1(C(C2CC(OC)C2)=O)CCN(C(=O)C=C2CCN(C)C2)C2CCCC2(C)C1 5714,Cn1cc(C(=O)NC2CC(C)(NC(=O)C=CS(C)=O)C2)c(=O)c2cc(Cl)ccc12 5715,Cc1nc(C2CC2)ccc1C(=O)N(C)CCN(C(=O)Cc1cnc[nH]1)C 5716,C(c1cc(F)c(F)c(F)c1)=CC(N1CCCN(C(C2(COC)CC2)=O)CC1C)=O 5717,CCC(C(=O)NC1(CNC(=O)CC2(C#N)CC2)CCCC1)n1ccnc1 5718,c1(NC2CCN(C(C(=O)NC(C)C)=O)C23CCC3)ccc([N+](=O)[O-])c(C#N)c1 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5754,C(C(=O)N(C)CC1CC(F)CN1C(c1ccc(C)s1)=O)(C(C)C)OC 5755,C1(CC)CCCCCCN1Cc1cc(C(F)(F)F)ncc1Br 5756,c1(OC)ccc(Cl)cc1NC(N1CC(c2ocnc2CNC(=O)C(C)(C)C)C1)=O 5757,C1(O)(C(C(=O)NC(C)CCN(C)C(c2ccns2)=O)(F)F)CCCCC1 5758,N1(C(c2nc(CCCC)sc2)=O)CCCN(C(c2cc(C)ncn2)=O)CCC1 5759,c1(C(=O)NC2CCC(Cn3cc(C4(C)CCCC4)nn3)C2)cnn2c1CCCC2 5760,N1(C(COC(C)=O)=O)CCN(C(=O)C(F)C2CCC2)C(C2CC2)C1 5761,CCC(C(=O)N1CCOCC1(C)c1cn(Cc2ccnc(Cl)c2)nn1)C(=O)O 5762,Cc1ccc(C(C)(C)C(=O)OC2CCC2=O)c(C)c1 5763,c1(CC)noc2ncc(C(=O)N(CCN(c3nnc(C)s3)C)C(C)C)cc12 5764,c1(CC(=O)NCCNC(=O)C2=CC3CCCC23)c[nH]c2cc(Br)ccc12 5765,N1(C(C2(NC(=O)C3=C(Cl)CCC3)CC(F)C2)=O)CCCN2CCCC2C1 5766,CC(CCCC(=O)N(CC(F)F)C)NC(c1ccc2c(c1)CC2)=O 5767,C(C(COC)CC(=O)N1CC(CCNC(C2(Br)CC2(C)C)=O)C1)OC 5768,C(=O)(CC(CCC)NC(=O)C=Cc1ccncn1)NCC(=C)Br 5769,N1(C(C=C(CC)C)=O)CC2CN(C(c3ccc(NCC(N)=O)cc3)=O)CCC12 5770,C#Cc1ccc(Br)c(C(=O)NC2CC(C)CN(C(c3[nH]cnc3C)=O)C2)c1 5771,C1(NC(C(F)=C(C)C)=O)CC2CC1CN(C(=O)C(c1c(C)noc1C)(C)C)C2 5772,c1(N2CCN(CC(=O)Nc3ccc(Cl)cc3F)CC2)ncnc2[nH]ccc12 5773,Cc1cc([N+](=O)[O-])cc(C(=O)NC2CN(C(c3c(C)cnn3C)=O)C(C)(C)C2)n1 5774,c1(OC(C(=O)NC2CC(c3ncc[nH]3)C2)C2CCC2)ccccc1 5775,N1(C(CCc2cc(OC)c(F)cc2)=O)CC2CCC(C1)N2C(=O)C(C)CC(N)=O 5776,C1(C2CCCCC2)(C(=O)NCC2CC(NC(C3(C#N)CCOC3)=O)C2)CC1 5777,C1(NC(C=CCOC)=O)CCN(C(C2CCC(=O)N2C(C)C)=O)CC1O 5778,N1(C(C)C)CCOC(C(=O)Nc2cnccc2C(=O)OC(C)(C)C)C1 5779,c1(N(C)CC)ccc(C(=O)NC(C)CCN(C)C(c2cc(C3CC3)on2)=O)cc1 5780,c1(C(=O)NC2C(C(N(C3CCCC3)CC(C)C)=O)CC2)ccc2occc2c1 5781,C(=O)(C(CC)CC(C)C)N1C(CC=C)(C(=O)NCc2nc(C)c(C)s2)CCC1 5782,c1(C(=O)NC2CC3CN(C(C(C=C=C)C)=O)C(C2)C3)n[nH]c2c(C)cccc12 5783,N1(C(CCCCC)=O)CC2OCC(NC(C3CC4(CSC4)C3)=O)C2C1 5784,c1(NC)cnc(C(=O)N(C)CC2CCCN2C(C2CCN(C)C2)=O)cn1 5785,N1(C(C(CC)(C)OC)=O)CCOCC(F)(CNC(c2cn(C)nc2C(C)C)=O)C1 5786,CCCCCCC(C)C(=O)NCC12CCC(C1)N(C(=O)CN1CC(=O)NC1=O)C2 5787,C1(C(N(C2CCN(C(=O)C(C)(C)C3CCC3)CC2)CCOC)=O)C2CC2C2CC12 5788,N1(C(C2CCC(C)(C)N(C(=O)CSC(C)(C)C)C2)=O)CCC12CCC(C)CC2 5789,C(CC(=O)NCC1(CC2CC2)CC1)(CC(C)C)NC(C=Cc1cccc(C)c1)=O 5790,C(=O)(C(C)(C)CC(C)C)N(C(CC(=O)NC(C(=O)OC)C)(C)C)C 5791,C1(NC(C2(C)CCNC2=O)=O)CC2(C1)CN(C(=O)C(C1CC1)C1CC1)C2 5792,N1(c2ncnc(N(CC(CC)C)C)c2C)CCc2c[nH]nc2C1 5793,c1(C(=O)NCC2C(NC(c3cc(OCCC)ncc3)=O)CC2)nn(C)c(C)c1Cl 5794,c1(OCC)nn(C)cc1NC(C1CC(C)N1C(C1C=CC=CC=C1)=O)=O 5795,CCCC(C)(C)C(=O)NC1CC(CCNC(=O)COCCOCCO)C1 5796,CCC(C)(F)C(=O)N(C)CCN(C)C(C1(N2CCSCC2)CCCCC1)=O 5797,C1(N(C(CS(CC)=O)=O)C)CCCC2CN(C(c3ccc(N)c(Cl)c3)=O)CC12 5798,c1(C(=O)NCC(c2ccc(Br)cc2)(C)C)ccc2c(c1)NC(=O)C2 5799,S(=O)(=O)(c1ccc(NC(c2cc(C)ccc2F)CO)nc1)N1CCC=C(C)C1 5800,C12(NC(c3c(C)ocn3)=O)CC1CN(C(=O)Cn1nc(C(F)F)cc1C(F)F)C2 5801,c1(C(=O)NCc2scc(CNC(CCC=C=C)=O)n2)cccc(F)c1C 5802,N1(C(c2ccn(CCNC(C3CN(C(C)=O)C3)=O)c2)=O)CC(S(C)(=O)=O)C1 5803,Cc1cc(C(=O)NC(CCNC(C2CCCS2)=O)C(C)C)cnc1C(F)F 5804,c1(C(N2CCC(O)(CNC(C(CC)(C)C#N)=O)C2)=O)cc(S(N)(=O)=O)cn1C 5805,N1(C(=O)OC(C)(C)C)CC2CN(C(c3ccc(Cl)cc3N3CCCC3)=O)C2C1 5806,c1(C(N(CC(CNC(C(COC)NC(C)=O)=O)O)C)=O)sc(C(C)(C)C)nc1C 5807,CC(C)CS(=O)(=O)CC(=O)NC1CC2CC(NC(c3coc(C(F)F)c3)=O)C2C1 5808,C(CS(=O)(=O)C1=NOC(C)(C)C1)NC(c1ccc(C(F)(F)F)cc1)C(=O)OC 5809,OCCC(N=c1[nH]c(=NCC2CCOC2)[nH]c2c1CCCC2)c1ccc(F)cc1 5810,c1(NC(C2(C)OCCN(C(C)=O)C2)=O)ccc(C(=O)NC2(O)CCC2)cc1Cl 5811,C1(C(N2CC(NC(C(C)NC(C3CCCCC3)=O)=O)C2)=O)CCCC2CC12 5812,C(=O)(CC1=NNC(=O)C1)NC1CCC(N(C(CN(CC)CC)=O)C)C1 5813,c1(C(N(CCN(C(C=CC)=O)C(C)C)C)=O)cccc(C2CCCOC2)c1 5814,N1(C(c2ccc(C)n2C)=O)CC2CCC1CN2C(c1ccc(F)cn1)=O 5815,C1(CCNC(CCSCC(C)C)=O)CN(C(c2cc(CO)[nH]n2)=O)CCO1 5816,C12(CCNC(C3(CC=C)CC=CC3)=O)CC(CO1)N(C(=O)CC1(C)CC1(F)Cl)C2 5817,Cc1cccc(NCC(N2CC(N(CCCS(N)(=O)=O)C)C2)=O)c1 5818,c1(C(N2C(CC)CCC2C)=O)n[nH]c2c1CCN(C(=O)Cc1cc(C)n(C)n1)C2 5819,S(=O)(=O)(c1cccc(=NCc2cc(OC)c(C)cc2C)[nH]1)NCC(CC)N(C)C 5820,Cc1cc(S(=O)(=O)NC(c2cnccc2-n2ccnc2)=O)sc1C 5821,C1(C(=O)NCCC2CN(C)C(=O)C2)CCC2(CC2)N1C(=O)CCc1ncccn1 5822,C1(NC(C(CCC)(C)O)=O)CCC2(CC1)CN(C(=O)C(CC)SC)CCO2 5823,C1(S(N)(=O)=O)(C(N(C2CCC(NC(C=C(C)Cl)=O)CC2)C)=O)CCC1 5824,c1(C(=O)NC2CCN(C(CCC(C)OCC)=O)CC2)ccc2nc(S)[nH]c2c1 5825,CC(C)(F)C(C)(F)CNC(c1cccnc1CNC(=O)CCC1CCCOC1)=O 5826,C1(n2cc(CCCC)nn2)CCC(NC(C2(O)CC2)=O)CC1 5827,c1(NC2CC(C)SCC2)[nH]c(=NC2CCS(=O)(=O)C2)nc2scnc12 5828,c1(CCC(=O)N(C2CCN(C(CC)C)C2)CC)ccc(C(=O)OC)nc1 5829,O=S1(=O)CCCC(NC(=NCc2cccc(C(N)=O)c2)NCc2cc(Cl)c[nH]2)C1 5830,C1(NC(CN(C2CC2)CC)=O)CCCC(NC(c2ccnc(C3CCC3)c2)=O)C1 5831,C(=O)(C(C#N)C(C)C)N1C2C(C(N(CC(C)(C)O)CCC)=O)C(C2)C1 5832,C1(CNC(COCCC#C)=O)CCCCN(C(c2csc(-c3ccsc3)n2)=O)C1 5833,C(=O)(C1=COc2ccccc2O1)NC(C(C(C)C)C)CNC(=O)CCSC(F)(F)F 5834,C1(NC(C2(CCC=C)CC2)=O)CS(=O)(=O)CC1NC(c1cc(C(F)(F)F)no1)=O 5835,C1(NC(c2cc(C3CC3)cs2)=O)CC12CCN(C(=O)CC1CC1(Cl)Cl)C2 5836,c1(C(N2CC(SC)C(NC(C3CC3C3CC3)=O)C2)=O)ccc2c(C)cc(O)nc2c1 5837,c1(C(N2C(C)CN(C(C3CN(S(=O)(=O)C(F)F)C3)=O)CC2)=O)ccn2cccc2c1 5838,N1(C(C2CC=C(C)CC2)=O)CCC2CN(C(C3CCC(=O)N3)=O)C2C1 5839,n1(CC(=O)N(C)CC2CCCN(C(c3cccn3C)=O)C2)cc(Cl)c(O)nc1=O 5840,C1(C(N(C2COC(C)(C)C2)C)=O)CN(C(=O)Cn2cncn2)CC12CC2 5841,c1(C(=O)NCC(C)(C)NC(c2ccc(N)cn2)=O)ncc2cc(Br)ccc2n1 5842,CCC(C)C(O)C(=O)NCC1CC(C)(C)CN1C(C1CC1(F)F)=O 5843,C(=O)(CC(CCCC)NC(=O)Cn1ccnc1C)N1C(C#C)COCC1 5844,c1(C(=O)NC(CN(C(=O)C=C(C)C(C)C)CC)C)ccc(O)c(C(C)(C)C)c1 5845,Cc1c(F)ccc(C(c2nnnn2C(C)C)NCC2(C)CC3(CC3)C2)c1Cl 5846,c1(CC(C(=O)O)NC(c2ccc(-c3ccncc3)cc2)=O)coc2ccccc12 5847,C12(NC(CCC=C)=O)CCOCC1CN(C(=O)Cc1ccc(C)c(C)c1)C2 5848,c1(SCCC(=O)NCCC2(CNC(=O)Cn3cnnn3)CC2)ccccc1Cl 5849,C1(NC(C2(C)CC=C(C)CC2)=O)COC2C(NC(c3ccccc3C)=O)COC12 5850,C1(C(N2CCC(COC)(CNC(=O)C(=O)NCC(F)F)C2)=O)OCCCC1(C)C 5851,c1(OC(C(=O)NCCC(C)NC(C(C)(C)OCC)=O)C)cccc(COC)c1 5852,CC1CN(C(C2CCCC(F)C2)=O)CC1NC(c1ccc(=N)[nH]n1)=O 5853,n1(CC(=O)NCC2CCCC2C(=O)Nc2cc(O)cc(F)c2)cc([N+](=O)[O-])cn1 5854,CC(C)CCCCC(=O)NCC1CCC1C(N1CCC(n2cncn2)C1)=O 5855,C12(NC(Cc3nc(CC)sc3)=O)CCC(C1)N(C(C1CC3CC3C1)=O)C2 5856,C=CC(C)CCN=c1[nH]c(=NCC2(CCO)CC2)c2cc(Cl)ccc2[nH]1 5857,N1(C(C(COC)C)=O)CCC(CC(C)NC(=O)CN2CCNC(=O)C2)CC1 5858,CCCCC(CNC(=O)CCC(=O)N(C)C)NC(=O)CC1CC(CC)=NO1 5859,C(C(C)C(C)C(=O)NCC(C)CN(C(=O)CC=Cc1ccc(F)cc1)C)OC 5860,C1(COC)N(C(C23CC2CN(C(c2cc(C4CC4)no2)=O)C3)=O)CC1(C)C 5861,N1(C(COCCC=C)=O)CC(O)CC1CNC(c1c[nH]nc1CCC)=O 5862,Clc1cccc(CCC(c2ccccc2)NCC23CC(C2)NC3)c1 5863,N1(C(C=Cc2n(C)cnc2)=O)CCN(C(c2cccc(Br)c2O)=O)C2CCC12 5864,C1(C(=O)Oc2cccc3c2OCCO3)COc2c(cc(Cl)cc2[N+](=O)[O-])C1 5865,C1(C(=O)NCC(CO)C2CC2)CC(O)CCN1C(=O)CC1CC=CC1 5866,CCCC(O)CC(=O)NC(C)(CNC(=O)Cn1cc(C2CCC2)nn1)CO 5867,N1(C(c2c(C)n(C(C)C)nc2)=O)CC2CC1CN(C(=O)CC1CC3(COC3)C1)C2 5868,c1(C(C(=O)NCC=CCNC(C2CCC(F)C2)=O)(F)F)c(F)cccc1F 5869,N1(CC(=O)NC(CN(C(C(C)CC2CCCC2)=O)C)C)CCCNC1=O 5870,c1(OC)nccc(C(=O)NC(C)C(C)NC(C2CC(=O)C2C)=O)n1 5871,C1(C(=O)NC(C)CNC(=O)C=Cc2cnc(C)s2)(CC)CCC(O)CC1 5872,C1=CCCC(Nc2cc(-c3ccccn3)ncn2)CCC1 5873,C(CC(C)(C)CC(=O)N1CCCN(C(=O)Cc2c[nH]c(=N)nc2O)CC1)OC 5874,N1(C(C2(C(=O)OCC)CC2)=O)CCN(COc2cc(F)cs2)CC1c1ncc[nH]1 5875,C1(CC)(NC(=O)COc2ccccn2)CCN(C(c2coc(CC3CC3)n2)=O)C1 5876,N1(C(c2cc(C)c(F)cn2)=O)CCC(C)(C)C(C(=O)NC(c2cccnc2)C)C1 5877,c1(C(C)NC(c2nc(C)c(C)[nH]2)c2nnnn2C2CC2)cc(Cl)ccc1F 5878,C1(C(C)N(C(=O)C(N2CCCC(N3CCN(C)C3=O)C2)=O)CC)CN(C)CCN1C 5879,CCCCCC(O)C(=O)N1CCN(C(c2cnc3occc3c2)=O)C(C(C)C)C1 5880,c1(N2CCC(O)(CSc3scc(CCCCCC)c3)C2)ncnn2cccc12 5881,c1(C(N2CCCC(NC(C3(C)CCCS3(=O)=O)=O)C2)=O)cc2c(Cl)nccc2o1 5882,c1(C(=O)NC2C3CN(C(C4(SCC)CC4)=O)C2C(O)C3)sc2cccnc2c1Cl 5883,C1(CNC(c2cnoc2)=O)CCN(C(c2cn3ccccc3n2)=O)CC1(F)F 5884,Cc1ccc(C(N2CC(C(F)Cn3cc(C4CCCC4O)nn3)C2)=O)o1 5885,CC1(C)C(NC(=O)CCSc2ccccc2)CCN1C(=O)C=C1CCCC1 5886,N1(S(CC)(=O)=O)C2CCC1CN(C(c1ccc(OC)c(I)c1)=O)C2 5887,N1(C(c2cnn(C(F)F)c2)=O)CCC2CN(C(=O)C(F)=CC3CC3)CCC2C1 5888,C1(N(C(COc2ccc(SC)cc2)=O)C)CCC(C)N(Cc2ccccc2)C1 5889,C=Cc1cc(C(=O)NCC2CCC(C)CN2C(c2nnc(CC)s2)=O)cc(F)c1 5890,N1(C(C2C(CNC(c3cnn4c3CCC4)=O)OCC2)=O)CCC12CCCOCC2 5891,CCCCC(C(=O)NCC1(CCNC(=O)C(CC)C(C)C)CC1)NC(N)=O 5892,c1(C(=O)NC(COC)C2(C)CC2)cccc(CN2CCNC(=O)C2)c1C 5893,N1(C(c2ccc(Cl)c(N)c2Cl)=O)CCN(C(=O)C2=NOCC2)C2CCCCC12 5894,c1(CCC)nc(=NC2CC(C)N(C(=O)CCC3CCCO3)C2)s[nH]1 5895,N(C(=NCCc1nn(C)cc1C)N1CCCC(CNC(N)=O)C1)C(COC)C 5896,c1(CN(C(c2c(CC)ccs2)=O)C)cnn2c1CN(C(c1c[nH]c(=N)s1)=O)CC2 5897,n1(CC(=O)NCC2N(C(C3C(C#N)C3)=O)CCCCC2)ncc(=O)c2ccccc12 5898,N1(C(C=CCCCCC)=O)CCCCC1CCC1CCCN1C(=O)COC1CC1 5899,c1(OC)nscc1C(=O)NC1COCC1NC(C1CC1(C)C)=O 5900,C(=O)(C(F)(F)C(F)(F)F)NCCCCN(C(=O)CC1(C)CCS(=O)(=O)N1)C 5901,c1(C(N(CC(C)NC(c2cnc(CC)o2)=O)CC)=O)ccc(C(F)F)cn1 5902,N1(C(c2[nH]cc(C)c2)=O)CCN(C(c2sc(C)cc2OC(F)F)=O)C(C(F)F)C1 5903,CC(=O)CCCC(=O)NC(C(=O)NCCCOC1CCCC1)C(C)C 5904,C(=O)(C(O)CC(C)C)N(CCN(C(COCc1onc(CC)n1)=O)C)C1CC1 5905,N1(C(c2snc(C)c2N)=O)CCC(N=[N+]=[N-])(C(=O)NCC(O)CF)C1 5906,CCC(CC)C(C(=O)NC(C)C(=O)NC(C)(C)CC(C)(C)C)OC 5907,O=[N+]([O-])c1ccc(NCc2cnn(-c3ccccc3)c2)cc1I 5908,N1(C(C(C)(C)OC)=O)CC2CC2(C(N2CCN(CC3CC3)CC2)=O)C1 5909,C1(C)CCCN(C(=O)C(=O)NCC2C(NC(C3(CC=C)CCCC3)=O)CC2)C1 5910,Cc1ccc(O)c(C(=O)NC2CCCC2NC(C2CCN(C)S2(=O)=O)=O)n1 5911,N1(C(=O)Cc2cn[nH]c2)CC(C2CN(C(=O)CCSc3ccc(F)c(F)c3)C2)C1 5912,C1(C(N(CCCn2cc(CN3CC4CC4C3)nn2)C)=O)CCC(=O)C(C)C1(C)C 5913,C1(CC(C)NC(C2(C)CCCS2)=O)CCN(C(=O)CC2CCC(=O)N2C)CC1 5914,N1(C(CC(=O)OC)=O)CCCC(O)(CNC(c2cc(Cl)ncc2OC(F)F)=O)C1 5915,C1(CC(=O)N(CCCN)C(C(=O)Cn2nccn2)=O)CCCCC1(F)F.C1CC1 5916,N1(C(C(C(C)C)C)=O)CCC(C)N(C(=O)CCCCOCC(F)F)CC1 5917,S1(=O)(=O)c2ccc(c(Cl)c2)N1.C1(CN2CCC(NC=O)CC2)CC2CCCCC12 5918,C12(CNC(=O)Cc3csnn3)CCCC1CCN2C(c1ncccn1)=O 5919,n1(CCC)ccc(C(N2CCC(CC(=O)NCCCN3CCOCC3)C2)=O)n1 5920,C(=O)(CC(C)C(=O)N1CCC(NC(=O)CC2(C)CC2(Cl)Cl)C1C(C)C)OC 5921,c1(C(N)=O)nc(C(N2CCC2CNC(c2cc(O)cs2)=O)=O)cs1 5922,CC(C#N)CN=C(NCC(C)(C)CN(C)C)NC(c1ccccc1)C 5923,Cc1c(C(=O)NCC2(NC(c3csc(C(F)(F)F)c3)=O)CCC2)cnn1C 5924,C(CC(C(=O)NC(C)C(C)OC)NC(=O)CC1CC1)OC 5925,CC12CCN(CC1)CC2C(=O)NCC1CC(NC(c2cc3ncccc3s2)=O)C1 5926,N(C1c2ccccc2CC1C)C(C1CN(c2c(OC)cccc2)C(=O)C1)=O 5927,c1(C(N2C(Cc3cccc(SCC)c3)COCC2)=O)cc2n(c1)CCCNC2=O 5928,N1(CCC)CCC(O)(NC(c2cnc(CC(=O)Nc3cccc(OC)c3)[nH]2)=O)C1 5929,S(=O)(=O)(c1cnccc1N(C)CC1(CF)CCC1)N(C)CC1N(C)CCC1 5930,c1(CNCC2CCN(C(C)=O)C2)cc2ncncc2s1 5931,c1(OC)cc(F)c(F)cc1C(=O)NCC1(CCNC(C23CC4CC2C3C4)=O)CC1 5932,C(=O)(C(Cc1cn[nH]c1)NC(c1cnc(O)o1)=O)N(CCOC)CC 5933,C1(C2CCN(C(=O)CCC(F)(F)F)CC2)(NC(C2CC(C)(C)OC2)=O)CC1 5934,C1(NC(C(C)(N(C(=O)C(=O)C(C)(C)C)C)C2CC2)=O)CCCOC12CCC2 5935,c1(CC)ccc(Br)cc1C(=O)NC(C)CCN(C)C(C1C(C)(C)C1(C)C)=O 5936,CN1CC(NC(=O)NCC23CC(C2)C(C(F)(F)F)O3)Cc2ccccc21 5937,c1(C(N2C(CN(C)C)CCCC2)=O)nc2ccccc2o1.C1(N)CCC12CCNCC2 5938,C1(C)(NC(CN(CC(C)C)C(c2ccn(CCC)n2)=O)=O)CCC(C)(C)C1 5939,c1(-n2c(CC3SC(=N)NC3=O)nc(COC(C)C)n2)ccc(Cl)c(F)c1 5940,C1(NC(c2c(C)scc2)=O)CN(C(c2cc3n(n2)CCC3)=O)CC12CCC2 5941,N#Cc1cncc(CN2CC(c3ccccc3)(C(N3CCCC3)=O)C2)c1 5942,c1(CC(C(=O)NC(C)CCCNC(C2CC2(C)C(F)F)=O)=O)ccc(F)cc1 5943,Cc1ncc(Cl)cc1C(N1CC(N(C(=O)CC2CCCCC2(C)C)C)C1)=O 5944,N1(C(CCc2n(C)ncc2)=O)CCC(C(N2CC(O)(C(F)F)C2)=O)C12CC2 5945,S(=O)(=O)(c1cccc(=NCCCN2CCCOCC2)[nH]1)N1CCC(OC)(CO)C1 5946,c1(CC)cnoc1C(=O)N(CCC(=O)NCCOC)CCO 5947,c1(NC(=O)NC)ccc(S(N)(=O)=O)c(OC)c1.C123CCC1CCCN2C(=O)OC3=O 5948,c1(C(N2CCC(CNC(C3(C#C)CC3)=O)C2)=O)cn(CCO)nc1C 5949,c1(OC)cc(C(N2CCC(C(=O)Nc3cccnc3C(F)(F)F)C2)=O)cc(Br)c1 5950,c1(C(=O)NCC2CCCN(C(C3C(C#C)C3)=O)C2)cc2sc(Cl)cc2s1 5951,N1(C(CCC)=O)CCC(N(C2CCC2)C(C2CCCN2C(=O)OC)=O)C1 5952,CC(C(C)C(=O)NCCN(C(=O)CCS(C)(=O)=O)c1ccccc1)C(C)(C)C 5953,c1(CC)cccc(C(=O)NCC2CCC(C(=O)N(C)CC3CCOC3C)CC2)n1 5954,c1(NC(CCCC)CC)ncnc(NC(c2cc(C)oc2C)C)c1C 5955,O(NC(=O)C(CNC(C1CCCSC1C)=O)N(C)C)CCCOCC 5956,C1(c2c(OC)nccc2)CCN(C(=NCC2CC(CF)C2)NCC(F)F)C1 5957,c1(Cn2c(-c3nc(Br)cs3)nc(C(CCC)C)n2)ccc(F)c(F)c1 5958,CC1CCN(C(=O)CC(c2ccon2)C2CC2)C1CNC(=O)CC1OCCC1C 5959,C1(C)(C(N2CCC(O)(CN(C(=O)C3=CCOC3)C)CC2)=O)CC(C(C)(C)C)=NO1 5960,C12(C(N(C)CC3(CC(C)C)CC3)=O)CC(CNC(c3nnc(S)n3C)=O)(CO1)C2 5961,c1(C(=O)NC2CC(NC(=O)CCc3nccs3)C2)ccc(CO)nc1 5962,c1(CC(C)C)ccc(CN2CC(O)(CNC(C3CCCOCC3)=O)C2)cc1 5963,c1(C(=O)NC2CC(NC(=O)Cn3ncccc3=O)C2)cccc2c1C(=O)NC2 5964,C1(CC)CN(C(=O)C(c2ccccc2)C)CCC1N=c1[nH]c2ccc(O)cc2s1 5965,S(=O)(=O)(c1cnn(C)c1)N(C)CC1CCC(=O)NC1.C12CCN(C1)C(=O)CN2C 5966,CC1CC(C(=O)NC2CCC2C(=O)NC2CCCCCC2C)=NO1 5967,c12nn(C)c3c1CN(CC3)C(C)C(=O)N2.C(=O)(C(C)CN(C(C)C)CC)OCC 5968,CC#CCCCC(=O)NCC1CN(C(c2c(Br)nnn2C)=O)CCCO1 5969,c1(C(n2cc(C3CCN(C(C4COCCO4)=O)C3)nn2)CC)ccccc1F 5970,C1(C(N(CCNC(C(C)CF)=O)CC2CC2)=O)CCc2ccccc2C1 5971,C(=O)(C(F)(F)CCn1ccnn1)NCC1(NC(C2C(C)(C(F)F)C2)=O)CCC1 5972,c1(-n2cc(CN(C(CC)=O)C)nn2)c(C)cccc1[N+](=O)[O-] 5973,C(=O)(C(CC(F)F)NC(c1ccoc1Cl)=O)N1CC(N(C)C)(C(N)=O)C1 5974,C1(CC(=O)NC2CN(C(C3(CF)CCOCC3)=O)C2)(OC(C)(C)C)CCOCC1 5975,c1(OCC)ccc(OCC)c(NC(=O)NC2CCNC2C)c1 5976,CC(C(=O)NCCOCCCNC(C1CC(=O)NC(=O)N1)=O)C(C)S(C)(=O)=O 5977,n1(CC)cccc1C(=O)NCC(CCNC(c1ccc(SC)o1)=O)OC 5978,C(=O)(C1=CS(=O)CCC1)N1C(CN(C(=O)C=CC2CCOCC2)C2CC2)CCC1 5979,c1(CC(N2CC(NC(CC(CC)CC)=O)C3C2C3)=O)ccc2c(c1)NC(=O)C2 5980,C(C(=O)N1Cc2ccccc2CO1)C1CCC(NC(CCC=CC(C)C)=O)C1 5981,Cc1ccc(NC(=O)CC2CCCN2C(C2CC3CC3C2)=O)c(C)c1 5982,c1(CN2CC(C#N)C(NC(c3ccc(S)cc3)=O)C2)cc(Br)cc(F)c1F 5983,N1(C(C(C2CCCCC2)OC)=O)CC(CNC(=O)CC(C)(C)CC)C(C)(C)C1 5984,N1(C(C2(CNC(C(C(C)C)OC)=O)CCC2)=O)CCC(C(=O)NC)CC1(C)C 5985,N1(C(CNC(=O)NC)=O)CCOCC1CC(N1CC(F)(F)C1C1CC1)=O 5986,c1(C(=O)NCCCC(=O)NC(COCC)CO)c[nH]ccc1=O 5987,C(=O)(C1=NN(CCO)C(=O)CC1)NCCC(C)(C)NC(C1N(CC)CC1)=O 5988,C(=O)(C1CCCn2nccc21)N1CC2N(C(c3cc(C)cc(Cl)c3)=O)C(CC2)C1 5989,C(N=c1[nH]c(NC2CCN(C)C2C)nc2cccnc12)c1c(C)n(C)nc1 5990,Cc1cc(CNC(C2CC(C)N2C(=O)CCC2(C)CC2)=O)ccc1F 5991,CC(C)CC(C(=O)N1CC2CC1C2)NC(C1CN2CCC1C2)=O 5992,c1(CNC(C2CC(CC)C2)=O)nc(CNC(=O)C(C)OCC(C)C)cc(O)n1 5993,c1(C(=O)NCc2scc(CC(=O)O)c2)cc2c(nc1O)CCC2 5994,c1(C(=O)NCC2CN(C(CCCCOCC)=O)C(C)C2)ccc(CC)cc1F 5995,N1(C(C(COC)OC)=O)C2CCC1CC(NC(c1ccccc1SC(C)C)=O)C2 5996,C1(C(=O)NCCC(C)O)COCCN(C(=O)CCc2cccnc2)C1 5997,CCC(O)C(C)(C)C(=O)NCCCN(C(=O)COc1ccc(CO)cc1)CCO 5998,c1(SCC(=O)N(CCCN(C(C(CC)F)=O)C)C)nc(C)c(C)c(C)c1C#N 5999,C1(CC(=O)NCc2cn[nH]c2)CCN(C(C2CCO2)=O)CC1 6000,N1(C(CCSCCC)=O)CC(NC(c2c(C)csc2Cl)=O)CC1(C)CC 6001,C1(NC(CCc2ccc(OC)cc2)=O)COC2(C1)CN(C(=O)C(F)=C(C)C)C2 6002,C1(C(=O)NCCCCNC(=O)C=Cc2cccnc2)CCC(=O)N2CCCC12 6003,N1(C(C2CC23CCC3)=O)CC2CCC(C1)N2C(=O)C(O)CC1CCCCC1 6004,CCC(C)(O)CNC(=O)CCCC1(NC(=O)COCCF)CCC1 6005,Cc1nc(C#N)c(NCCC(=O)NCC2CCCC2NC(=O)C(F)C(C)(C)O)o1 6006,C1(C)(C(=O)NC2CC(NC(CCCSC)=O)CC2O)CC=C(C)CC1 6007,c1(N(CCOC)C)cccc(S(=O)(=O)N2CCSC(C)C2C)n1 6008,CCCCC(CN=c1[nH]c(Cl)nc(CC)c1Cl)SCC(=O)Nc1ccccn1 6009,C(CCCCC(=O)NCC1(O)CCCN(C(=O)CC2CC(F)C2)C1)OCC 6010,C1(N(C(c2cncc(C)n2)=O)C)CCCN(C(c2cc(Br)nn2C)=O)CC1 6011,c1(C(=O)NC(C(=O)NC(C=C)CO)c2ccco2)cnccn1 6012,S(=O)(=O)(c1c(F)cc(F)cc1F)NCc1scc(C(=O)Nc2cccc(Br)n2)n1 6013,CCCCC(C(=O)NCc1cc(C2CC2)no1)NC(C1OCCC1(C)C)=O 6014,n1(CC(=O)Nc2cccc(C(N(CC)CC)=O)c2Cl)c(C)cc(C)nc1=O 6015,c1(C(=O)NC2CN(C(C3C(C)CCC3)=O)CC2F)cn2ccc(Br)cc2n1 6016,C1(O)(CN(C(C(C)SC(C)C)=O)C)CCN(C(c2n[nH]c(C3CC3)c2Cl)=O)C1 6017,C=CCC(CC)C(=O)N1CCN(C(=O)CN(CC)CC)CC1CC(F)(F)F 6018,C1(C(=O)NC(C)Cc2nc(-c3ccccc3)no2)CC(O)C(O)C1 6019,N1(CCC#C)CCC(C(N2CC3CC3(NC(=O)C(O)CF)C2)=O)CC1 6020,Cc1cc(C(=O)NC2CC(N(C)C(C3CNC(=O)N3)=O)C2)c2sc(=N)[nH]c2n1 6021,N1(C(C2C(C)(CCC)C2)=O)Cc2cccc(CNC(=O)C(CC)CC)c2C1 6022,Cc1nc(C(=O)NCCC2CCCN2C(=O)CO)ccc1Br 6023,c1(N2CCC(CC(C)N)CC2)ncc2ccccc2n1.C(=O)(C(=O)NC)NC1CC1 6024,c1(C(N2CCCC2CNC(C2CC(F)(CO)C2)=O)=O)coc2ccccc12 6025,C1(C(=O)NC2CN(C(c3cc(C)ncc3)=O)CC(F)C2)CCn2ncnc2C1 6026,N1(C(CC2(C=C)CC2)=O)CCCC2(NC(C3CCC(C(N)=O)CC3)=O)CC2C1 6027,c1(C(N2CC(NC(c3coc(Br)n3)=O)C3C2C3)=O)cc2scnc2[nH]1 6028,C1(C(=O)NC2CC(NC(=O)CCC3CCCCC3)C2)CCCN(C(=O)C2CC2)C1 6029,c1(CC)nn(C)cc1C(=O)NCC1(C)CCN(C(c2cnc(C)o2)=O)C1 6030,CCCCC(CNC(=O)CCCC1CCCC1)NC(=O)CC(C)C1CC1 6031,C(N=c1nc(N2CC3CCN(C)CC3C2)c2[nH]ccc2[nH]1)c1c(OC)cncc1 6032,c1(C(c2nnnn2CC)NCCCn2cc(C(CC)O)nn2)c(C)cccc1Br 6033,N1(C(C(C)=C2CC2)=O)CCCC2(CCCCC2NC(=O)CN2C(C)CCC2C)C1 6034,Nc1c(F)c(F)cc(C(N2CCN(C(C3CC(O)C3)=O)C3CCC23)=O)c1Cl 6035,CC(CCC(=O)Nc1cn(C)nc1Cl)NC(c1ccncc1Cl)=O 6036,c1(OCC)ccc(C)nc1C(=O)NCC1CC1NC(c1cc([N+](=O)[O-])c[nH]1)=O 6037,c1(C(=O)NCC(CNC(C=NOC)=O)F)cc2ccc(F)cc2s1 6038,Cc1cc(F)c(C(=O)NC2CC(CCNC(C3CCOC3C)=O)C2)cc1F 6039,C1(C2CC2)(C(=O)NCCCCCNC(=O)CCN2CCOCC2)CCC1 6040,C(=O)(C1SCCc2sccc21)N1CCC2(CC(NC(=O)CC=C(Cl)Cl)C2)C1 6041,c1(C(=O)NCC2(NC(=O)CC3CC4CCC3C4)CC2)ncc(Br)cc1O 6042,C1(C(=O)NC2CC(CNC(c3ccc4nncn4c3)=O)C2)CCc2nnnn2C1 6043,O=C(C(F)C1=CCCCC1)NCC1CC2CCC1N2C(=O)Cc1ccc(Cl)cc1 6044,c1(OC)ncc(Cl)c(C(N2CC3(NC(=O)C(C(C)C)SC)CC2C3)=O)c1Cl 6045,c1(OCC)nccc(C(=O)NCC(C)(CO)NC(=O)C=C(CC)CC)c1F 6046,Cc1nc(CO)ncc1C(N1CCC(NC(C2C(C)OC(C)C2C)=O)C1(C)C)=O 6047,c1(C(=O)NCCNC(=O)Cc2c[nH]ccc2=O)cnc2ccccn2c1=O 6048,C(=O)(C1=CC2(CCOCC2)C1)NC1CC(C)N(C(=O)C(=C2CCCCC2)F)CC1 6049,S(=O)(=O)(c1cccnc1N1CCCOC1)NC(=O)CC12CC1CCN2 6050,C1(C)(CNC(C(C2CC=CCC2)NC(c2cnc(C)o2)=O)=O)CCN(C)C1 6051,C1(C(=O)NCC2C(NC(c3nc(C(C)=O)sc3)=O)COC2)CCN(CC)C(=O)C1 6052,C=CCCCCCCCC(=O)N1CCC2(CC2NC(=O)C(C)CC(C)C)C1 6053,N1(C(C(C)CC2CCCO2)=O)C2CCC1CN(C(=O)CN1CC(C)(N(C)C)C1)C2 6054,c1(C(N(C(C(=O)N(CC=C)CC)C2CC2)C)=O)cnncc1C 6055,c1(CC2(C(=O)NC3CC(O)(CNC(C4CCCO4)=O)C3)CC2)cccc(F)c1 6056,N1(C(CCc2cn(C)nc2)=O)CCC(NC(=O)CSc2cn[nH]c2)C1C1CC1 6057,C(=O)(C(CC(F)F)NC(=O)Cc1cn[nH]c1)N1CCN(C(C)(C)C)CC1 6058,C1(CNC(COC)=O)CC2CC1CN2C(c1ccc(-c2ccsc2)cc1)=O 6059,Cc1nn(CC(N2CC(NC(c3ncc(F)cn3)=O)C(C)C2)=O)cc1Br 6060,C1(NC(C(n2ncc(C)c2)C)=O)CCCCC1NC(=O)C=Cc1ccoc1 6061,C(=O)(C(F)(CNC(C1CC(C(=O)OC)C1)=O)C(C)C)N(c1cccc(CC)c1)C 6062,N1(CC(=O)NC(C2CN(C(=O)CCNC(N)=O)CCO2)C)CCC(F)(F)C1 6063,C(=O)(C(C)(C)C(=O)Nc1ccc(F)c(F)c1)NC1CC(C)N(C(C2CSC2)=O)C1 6064,c1(C(CC)C)ccc(C(=O)NCC(C(C)C)NC(C2(O)CC2)=O)c(O)n1 6065,c1(NCC2(NC(=O)OC(C)(C)C)CC2)n[nH]c(=N)[nH]1 6066,C1(C2CC2)(NC(CN(CCC)C(C2CC2C(F)(F)F)=O)=O)CCCC1 6067,c1(NC(c2ccc(OC=C(Cl)Cl)cc2)=O)cccc(-c2nc(O)n[nH]2)c1 6068,c1(COC)cc(N(CC(C)CNC(C2CCCOCC2)=O)C)nc(SC)n1 6069,CCCCC(CN1CCCC(C(N2CCCC(CO)C2)=O)CC1)CC 6070,CP(C)(=O)C1CCCN(C(=O)N(C2CC2)Cc2ccncc2)C1 6071,N1(C(C(CC2CC2)NC(C2CCCN2C2CC2)=O)=O)CC2(CCC2)C1 6072,N1(C(C(C2CC2)OCC)=O)CCC2(CCCN2C(c2cc(N)c(Cl)cn2)=O)CC1 6073,C1(NC(CCC(C)OC)=O)CC2CCC(C1C)N2C(=O)C1=CCCCO1 6074,C1(CNC(c2[nH]nnc2C2CC2)=O)CN(C(=O)CCc2ccccc2O)CCO1 6075,CC1=CCSC1C(=O)NC(C1CCN(C(=O)CC2CCCC2O)C1)(C)C 6076,C1(CC=C)(OC)CCN(C(c2cnc(O)n2C)=O)C1.c12nc(Cl)c([nH]1)CNC2=O 6077,C1(N(C(=O)C(=O)NCc2cn(-c3nccs3)nn2)C)CS(=O)(=O)C12CCOCC2 6078,N1C2c3ccccc3CC2N(C=O)C(C)(C)C1=O.C(=O)(C(O)C1CC1)C(N)=O 6079,CCCC(CC)C(=O)NC1CN(C(=O)C2=NNC(=O)C2)CC1CC 6080,C1(NC(C(CC)CC2CCCC2)=O)CC2CN(C(c3ccccc3F)=O)CC2C1 6081,N1(C(C(C)N(CCC)C(C2CC(NC(C)=O)C2)=O)=O)CCOC2C(O)CC12 6082,C1(NC(C(CC=C)C)=O)CC(OC)CN(C(c2cc(C)n(CC)n2)=O)C1 6083,C=CCCC(C(=O)N1CC(OC)CC(F)C1)NC(=O)C(C(C)(C)C)SC 6084,C1(NC(c2c(OC)csc2)=O)CC2CN(C(c3ccc(CO)s3)=O)CC2C1 6085,N1(C(COCC=C)=O)CCC(NC(=O)COc2cccc(C)c2)C12CCC2 6086,CC1(C)C2CC1CN(C(=O)CC(=O)NCC(F)(F)F)C2 6087,C1(CNC(Cc2c(C)con2)=O)(CNC(c2cc(C)n(CO)n2)=O)CC12CCC2 6088,S(=O)(=O)(CC(=O)Nc1c(C(N)=O)ccnn1)C(N(CCNC1CC1)CC1CC1)=O 6089,C1(NC(C(CCOC)NC(=O)Cn2cnnc2)=O)C2CCCC1COC2 6090,C1(CNC(C(C)NS(C)(=O)=O)=O)CCC2(CN(C(=O)Cc3cnccn3)C2)O1 6091,N1(C(CC=CC)=O)CC=CC(NC(c2ccc(C3CCC3)nc2)=O)C1 6092,Cc1ccnc(C(N2CCC(N(C(=O)C(N3CCCCCC3)C)CCO)C2)=O)c1N 6093,Cc1cncc(C)c1C(N1CCCCC1CNC(c1ccc(C#N)n1C)=O)=O 6094,C(CCCCCN(C(=O)CCn1ncn(C)c1=O)C)NC(C1(CC)CC1(F)F)=O 6095,C(=O)(CCN1C(=O)C(C)Oc2ccccc21)NC(CC)C(=O)NC 6096,n1(CCC(=O)NCC(CC)(CC)NC(C2CCO2)=O)c(C)c(C)sc1=O 6097,N1(C(C2CC(OC)C2)=O)CCOC2CN(C(c3nccc(Cl)c3O)=O)CC12 6098,N1(C(C(C)n2cccc2)=O)CCC2(CC2)CC1C(=O)NCCN1CC=CC1 6099,O(NC(=O)C(O)C1CN(C(c2ccc(=N)[nH]n2)=O)C1)CC1CC(=C)C1 6100,C(=O)(N=c1[nH]n(-c2ncccn2)cc1I)c1ccc(-c2n(C)cnc2)cc1 6101,C#Cc1ccc(CNC(=O)C(C)C(C)NC(=O)CCN2CCOCC2)cc1 6102,n1(CC)c(=O)cnc2ccc(NC(=O)Cc3ccc4c(c3)NC(=O)CC4)cc12 6103,N1(C(C(CC)NC(=O)C(=O)NCC2CC2)=O)CCOC(C)(C)C1C 6104,Cc1sc(-c2nc[nH]n2)nc1C(N1CC(O)(CCNC(C2(F)CC2)=O)C1)=O 6105,C1(NC(Cc2c(C)cco2)=O)CCCN(C(=O)CC23CCC(CC2)C3)C1C 6106,c1(OC)ncc(Cl)cc1C(=O)NC1CN(C(C2CC(=C3CC3)C2)=O)CCC1C 6107,C=CC(C)(C)CC(=O)N1CCC(CO)C(NC(=O)CN(C)CCOC)C1 6108,c1(CNC(c2c(C)noc2C)c2nnnn2C2CC2)ccc2c(c1)OC(C)(C)O2 6109,C1(C)(C(N(C)CC2CCN(C(C3(C)CCCO3)=O)C2)=O)CCCNC1=O 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6128,C1(CNC(C(=O)NCC)=O)CN(C(C23CCC(F)(CC2)CC3)=O)C2CCN1C2 6129,CC12CC13CCN(CC3)C(=O)C1(CC1)OC2=O.c1(COC(C)(C)C)ccccc1 6130,C1(CC(=O)NCCC(F)(F)CO)CCCC(NC(c2csc(O)n2)=O)C1 6131,C1(NC(Cc2ncc(C)[nH]2)=O)CCCC(NC(=O)CCSc2ccccc2)C1 6132,C1(CNC(C(CC(C)C)F)=O)CN(C(c2cnc(C3CC3)s2)=O)CCC1(F)F 6133,N1(C(=O)CCOc2ccccc2Br)CCCC2(CCN2)C1 6134,N1(C(Cc2c(C)n(C)cn2)=O)CCN(C)CC1CNC(=O)C1=CCN(C)C1 6135,CN1CC=C(CC(=O)NC2CCC2NC(c2cc(Cl)c(Br)[nH]2)=O)CC1 6136,C1(OC)CN(C(=O)C=CCBr)CCC1NC(=O)C(C)(C)c1cc[nH]n1 6137,CC(C)(C(=O)NC(c1sc(Cl)nc1Cl)C(=O)O)C1=CCSCC1 6138,N1(C(C(CC(C)C)C)=O)CC2CCCC(NC(=O)CSCCC#N)C2C1 6139,CCC(O)C(C)(C)C(=O)NC1CCCC1NC(c1cccc(OC)c1O)=O 6140,C1(NC(CCCCOCC)=O)CCN(C(c2ccccc2C#N)=O)CC1(C)C 6141,CC(C(=O)N(CCCO)CCO)(C1CCC1)NC(c1cnn(C(F)F)c1)=O 6142,C#Cc1cn(C)nc1C(N1CCCOC(CNC(C2CCC2(OC)OC)=O)C1)=O 6143,CN1C(=O)CCCC1c1nc(-c2cccnc2O)nn1C1CCCC1 6144,Cc1cc(C(N2CC(NC(=O)CC3CC3)C3CC3C2)=O)c(C)n1-c1cnccn1 6145,C1(CNC(COCCC#C)=O)COCCN(C(=O)CC(CC)NC(=O)OC)C1 6146,C(C1COC(C)(C)O1)=CC(=O)NC1(CCNC(C(CCC)NC(N)=O)=O)CC1 6147,C1(NC(c2c(CCC)n[nH]c2)=O)CN(C(=O)CC#N)CCC12CCC2 6148,n1(CC(=O)NC2CC(C)(NC(CC=C=C)=O)C2)nc(C)c([N+](=O)[O-])c1C 6149,Cc1cnc(F)cc1CNCCC1CCC(C(F)(F)F)O1 6150,C(CCCCCC(=O)NCc1ccnc(F)c1)NC(C1(CC#C)CCC1)=O 6151,Cc1ccc(C(=O)NCC(O)CNC(=O)C2=C(Cl)CCOC2)c2cccnc12 6152,c1(CC(=O)NCCC(C)N(C(c2nc(OCC)oc2)=O)C)ccc(F)cn1 6153,C(=O)(CC(CC)C(C)(C)C)NC(CCC)C(=O)N(CCS(N)(=O)=O)C 6154,N1(C(COCCC(C)C)=O)CC2CCN(C(c3cn(C)c(O)n3)=O)C(C2)C1 6155,c1(C(N2CC3C(CNC(C(N)=O)=O)(CC3)C2)=O)c[nH]ccc1=NC(=O)C(F)(F)F 6156,C#Cc1cc(C(=O)NCC2C=CCN2C(c2cc(Cl)c([N+](=O)[O-])[nH]2)=O)cc(F)c1 6157,CCCCCCN(C)C(C1CC(CNC(=O)CC2CC2CC)C1)=O 6158,CCCCC(O)C(C)C(=O)NCC(CNC(=O)C(CC)SC)S(C)(=O)=O 6159,c1(CCNC(=O)C(N2CCC(N3CCCNC3=O)CC2)=O)ccc2c(c1)CCOC2 6160,C(=O)(CC(F)(F)C(F)(F)F)NCC(C(C)C)NS(CCCNC(COC)=O)(=O)=O 6161,c1(NC(=O)NCCCNC2CNC(CO)C2)ccccn1 6162,c1(CCC(=O)N(C)CC2CCN(C(CC(=O)OC)=O)C2)cc(C)cc(C)c1 6163,C(=O)(C(O)CCC(C)C)N1C2CCC(NC(C=Cc3ccc(SC)s3)=O)(C2)C1 6164,N1(C(COCc2cc(C)no2)=O)CCC(C)CC1CNC(c1ccc(C#N)s1)=O 6165,c1(OC)c(C)csc1C(N1CCC(CN(C)C(C2(C#N)CC2)=O)C1)=O 6166,C(C(C)(O)CC(=O)N1CC2(C1)CN(C(C1(c3ccccc3)CCOC1)=O)C2)OC 6167,C12(CNC(CC(CNC(c3ocnc3C(C)C)=O)OC)=O)CCC(CC1O)C2 6168,n1(C(C)C)ccc(C(N2CCCC2C(C)NC(=O)CCOCC2CCC2)=O)n1 6169,N1(C(c2ccc(CNC(C3CN(C4CCC4)C3)=O)nc2)=O)CCC2CCCCC2C1 6170,C1(C(=O)NCC(C)(C)CCO)CCOCCN1C(C1CC(C)(C)CO1)=O 6171,Cc1c(C(=O)NCC2CCC(C)CN2C(=O)CC2CC=CC2)sc2nccn12 6172,N1(C(C2C(=C)C2)=O)Cc2n[nH]cc2C1C(=O)NCCCOCCCC 6173,Cc1cc(C)n(C2CCCN(C(c3nnc(C(C)C)s3)C(=O)NCC(C)C)C2)n1 6174,CCCCCCC(=O)NC(c1nc(C(=O)NC(CC)CC(F)(F)F)co1)C 6175,Cn1ccnc1CC(=O)NCC1CC1C(=O)NCC(C)(C)n1ccnc1 6176,c1(NC(CN(C(Cc2ccc(C)nc2)=O)C)C)ncc([N+](=O)[O-])cc1C#N 6177,c1(C(N2CC(C(=O)NC(C#CC)(C)C)N(C)CC2)=O)coc2ccccc12 6178,C1(C(N2CC3(CCC3NC(C3CC=CCC3)=O)C2)=O)(CC)CCC(F)(F)CC1 6179,Cc1noc(C)c1C(N1CC2(NC(=O)Cc3csc(Cl)c3)CC1C2)=O 6180,N1(CC(N2CCC(CCNC(c3cc(C)on3)=O)C2)=O)CCC(F)(F)C1 6181,Cc1ccc(C(=O)N(CCN(C)C(c2coc(Cl)n2)=O)C(C)C)nc1 6182,Cc1cccc(F)c1CC(=O)NC1CC(N(C)C(c2c(C)ncn2C)=O)C1 6183,Cc1noc2ncnc(NC(C3(O)CCN(C(=O)CCn4cnnn4)C3)C)c12 6184,C1(C(=O)NCCOCCOCCO)CC2(CC(NC(=O)CCC(N)=O)C2)C1 6185,c1(C(=O)OC)cc(C(=O)NC(C)(C)CCCNC(=O)C=CCO)ccc1F 6186,C1(C)(CNC(c2c(C)ncs2)=O)CCCN(C(=O)Cc2csc(NC=O)n2)C1 6187,Cc1cncc2nc(CC(N3CCCOC(COc4ccccc4)C3)=O)cn12 6188,N1(C(c2snc(C)c2N)=O)CCCN(CCNC(C2CN(C)C2)=O)CC1 6189,O=C1CCC(C(=O)N2CCC(NC(c3cc(C(F)(F)F)cc(Cl)c3)=O)C2)=NN1 6190,C1(NC(c2nc(C)sc2)=O)COC2(CNC(=O)CCOC3CCCOC3)CC1C2 6191,N1(C(c2c(OC)cc(N)cc2)=O)CCC2CN(C(C3CC3(Cl)Cl)=O)CC2C1 6192,C1(NC(C2CC3CC2C2CC32)=O)CCCCN(C(c2cc3occc3[nH]2)=O)C1 6193,N1(C(c2c(N)cccn2)=O)CCC2(CCOC2)C(CNC(=O)Cc2csnn2)C1 6194,C12(CNC(C(COC)O)=O)CCCCC1N(C(c1cc(OC)nn1C)=O)CC2 6195,C1(C(N2CC(CC(C)NC(C(C)C)=O)C2)=O)(N(C)C)CCCCC1 6196,C(=O)(C(CC(C)(C)C)NC(=O)C(C1(O)CCCC1)F)N1CC(SCC)C1 6197,C(CCCCNC(=O)COCC(C)(C)C)N(C(CCC1CC(C)C1)=O)C 6198,c1(C(=O)NC2CCC(NC(Cc3ccn(CC)n3)=O)C2)ccc(C)c(C)c1N 6199,c1(C(CNC(c2c(C(C)C)noc2)=O)NC(c2ccoc2)=O)ccccc1F 6200,C1(CC)CC(O)CN1C(c1conc1CNC(=O)Cn1cnc(C#N)n1)=O 6201,N1(C(c2ccn(CCNC(c3c(C)cc[nH]3)=O)c2)=O)CCC(CO)(CO)C1 6202,C=CCCC(=O)NCC(C1CCC1)NC(C1CN(C2CCOC2)C1)=O 6203,CCCCCCC(C)C(=O)N(C1CN(C(c2cc(C#N)cn2C)=O)CC1(C)C)C 6204,C(=O)(C#CC1CCCO1)NC1CC(F)(CNC(c2c(C)nn(C(C)C)c2C)=O)C1 6205,c1(C(N2CC(OCCOC)C(O)C2)=O)cc(C)ccc1Br 6206,C1(C(N(C2CN(C)CC2O)C)=O)CCCC(NC(=O)C=CCN2CCCC2)CC1 6207,c1(C(=O)NC(C(C)C)C(=O)N(C2CCCCC2)C(C)C)cc2c(O)cccc2[nH]1 6208,C(=O)(C(CO)C(C)C)NC(CNC(CCn1c(C)cc(C)n1)=O)(C)C1CC1 6209,C(CC(C(C)C)NC(c1cscc1C(=O)OC)=O)N(C(C=C(CCC)C)=O)C 6210,N1(c2nnc(SCc3cccc(NC)c3)n2CCN(C)C)CCCC2(CCC2)C1 6211,c1(C(=O)NCC(CNC(CNC(=O)OCC=C)=O)(C)O)cc2n(n1)CCCC2O 6212,C1(CC(=O)OC)(C(=O)NCC(C)C(=O)NCC(C)(C)n2ccnc2)CCCC1 6213,N1(C(CNC(=O)NC)=O)CC(C)C(NC(c2ccc(C(C)(C)C)s2)=O)C(C)C1 6214,c1(CCC(=O)NC(C2(CNC(C3CC(N(C)C)C3)=O)CC2)C)cccnc1 6215,C1(NC(c2nc(CC)oc2)=O)CC12CCN(C(=O)Cc1ccoc1C)CC2 6216,N1(C(C(CCN(C)C)NC(CC2C(C)C(=O)CC2)=O)=O)CC2CSCC2C1 6217,c1(CNC(CN(C(=O)C=C2CCC2)C(C)C)=O)ccc(CO)o1 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6237,Cc1cc(OC=CC(=O)NC2CN(C(=O)COC(C)C)CC2C)ccc1F 6238,c1(C(C)=O)c(C)[nH]c(C(N2CCC(OCCNC(=O)CC3CCCC3)C2)=O)c1C 6239,C(=O)(CC(CC)CC(C)C)NCCC(=C)CNC(c1ccc(F)cc1)=O 6240,O=S(=O)(c1ccc(Cl)c(F)c1F)N1CCCCCC1Cc1ccc(O)cc1 6241,c1(NC(=O)NCC2C(OCC)CC2)ccc(N2C(=O)CCC2C)cc1 6242,CCC(CC)C(C)C(=O)N(C)CC1CCCN(C(c2nc(C)n(C)c2C)=O)C1 6243,C1(C(N2CCC(NC(C3CC(F)(F)C34CCC4)=O)C2)=O)Cc2ccccc2C1 6244,Cc1ccnc(C=CCNC(C2CCN(CC3CN(C)C3)C2)=O)c1 6245,N1(C(C2C(C)C2C)=O)CCCC(C2CCN(C(C3(O)CCCCC3)=O)C2)C1 6246,c1(NCC)ccc(Cl)cc1C(=O)NCC(F)CNC(C1CC2CC1CO2)=O 6247,N1(C(C2CC=CCC2)C(=O)N(c2c(C)cccc2)C2CC2)CCS(=O)C(C)(C)C1 6248,C(=O)(CC=C(Cl)Cl)NCCC(C)N(C)C(c1ccccc1OCC1CCCO1)=O 6249,CSC1=C(C(=O)NCC(C2CCOC2)NC(=O)CC2=NNC(=O)C2)CCCC1 6250,N1(C(CCC(c2cc(C)c(O)cc2)=O)=O)CCCC(C2CC2NC(=O)C(C)C)C1 6251,N1(C(C(C)CN(C)C)=O)CC2CCC1C(CNC(C1(C3CC3)CCCO1)=O)C2 6252,c1(C(N2CCC(n3cccn3)C2)C(=O)NC(CC)C)cc2ccc(OC)cc2o1 6253,C(=O)(C(C(F)(F)F)C(F)(F)F)N1CC2(OCC(NC(C(CC(N)=O)O)=O)C2)C1 6254,c12ccc(c(C)c1)S(=O)(=O)N2.C1(C(=O)OC)C(Cl)(Cl)C12CC2 6255,c1(C(=O)NC2(C)CN(C(C3CC4(CC4)CO3)=O)C2)cc(C(C)(C)C)ccn1 6256,N1(C(CCCC)=O)CC2CN(C(c3cccc(C(C)=O)c3)=O)CC2C1 6257,C1(NC(C(COC)NC(C2CCOCC2)=O)=O)CCCC(F)(F)C1 6258,C(C(C(=O)N(CCN(C(=O)C(C)(C)c1cnn(C)c1)C)C(C)C)N(C)C)OC 6259,c1(C(N2CCOCC2C(=O)Nc2cc(F)c(Cl)cn2)=O)cccc(Br)c1F 6260,c1(CC)cc(C(=O)NC(C2CCCC2)CNC(C2CC3CCC3C2)=O)cc(O)n1 6261,C12(C(=O)OC)CC(C(=O)NCC(CNC(=O)CN3CCCC3)CO)(C1)OC2(C)C 6262,C(=O)(CCC(C)(C)[N+](=O)[O-])NC1CCN(C(C2N(C)CC(O)C2)=O)CC1O 6263,c1(C(=O)NC(c2ccccc2)C(C)NC(=O)CC(F)(F)F)cc(Cl)ccc1O 6264,N1(C(=O)CC2CCOC2)CCN(CC(N2CCC(CC3CCCO3)C2)=O)CC1 6265,Fc1ccc(I)cc1C(NC1(CCC(F)(F)F)CC1)N 6266,C(=O)(C1=COCC1)NC(C1CC(C(C)(C)C)C1)=O.C1(=O)CSCCO1 6267,CCCC(C(=O)N1CCCC1C(C)NC(c1cncc(F)c1)=O)OCC 6268,c1(NC)cnc(C(=O)NC(C)(C)CNC(=O)C=C2CCC(C)C2)cn1 6269,Cc1ncccc1C(=O)N(C1CC(NC(c2cc(C(C)(F)F)n[nH]2)=O)C1)C 6270,c1(CC)ccc(S(=O)(=O)N2CCC(C)(C(=O)Nc3c(C)ccc(I)c3C)C2)cc1 6271,CC(CC1CCCC1)N=c1[nH]c(=NCC2(C)CCCC(=O)N2)c2ncccc2[nH]1 6272,C1(NC(c2cc(CC)no2)=O)CCN(C(C2CC3CC2C3)=O)C1(C)C 6273,C1(C(=O)NCc2cccc(NC(CN(C(=O)OC)C)=O)c2)CCCCN(C)C1=O 6274,C1(NC(CC=CC=C)=O)CC2CC(NC(=O)CCc3ccccc3F)CC12.C1(C)CC1 6275,c1(OCC(N2CC(CNC(C3CCCN(C(N)=O)C3)=O)C2)=O)ccc(Cl)cc1Cl 6276,c1(C(N2CCC(CC(=O)NCCc3ccco3)C2)=O)ccc(F)c(F)c1 6277,CCC(CC)(CC(=O)OC)C(=O)NC1CCCN(C(=O)CC(=O)NC2CC2)CC1 6278,c1(C(N2C(CNC(c3ccc(CO)cn3)=O)CCC2)=O)cn2cccc(Br)c2n1 6279,c1(CCC(=O)NCC(C)(C(C)C)NC(CCC(=C)C)=O)nnc(S)nc1O 6280,CC1(NC(=O)CCc2ccc(F)cc2)CCN(C(=O)C(F)C2CC2)CC1 6281,c1(C(N2CCN(C(C3(CO)CCCO3)=O)CC2)=O)ncc(F)cc1F 6282,Cc1cc(Cl)c(C(=O)NC2CCC(CNC(C3CNC(=O)N3C)=O)C2)cc1N 6283,C(=O)(C(C)C(=O)N1CCC(C)(NC(C2(CSC)CC(F)(F)C2)=O)C1)OC 6284,N1(C(CC(C)c2ccncc2)=O)CCC2(CC1)CC2CNC(=O)Cn1ccnn1 6285,C1(NC(C(F)=CCC)=O)(CO)CCCN(C(c2cc(C3CCCO3)n(C)n2)=O)C1 6286,N1(C(CC2(OC)CC2)=O)CC2CC1C2NC(c1ccnc(-n2ccnc2C)c1)=O 6287,CC(F)(F)CCC(=O)NC1CC(NC(C2CC3(C2)CC3(F)F)=O)C1 6288,C1(NC(CC(CC)SC)=O)C2CC3C1C3C2C(=O)NC(c1ccccc1)C 6289,C(=O)(CCS(C)(=O)=O)NCC1(CC(=O)NCCC=C=C)CC1 6290,N1(C(C(C)=C2CC2)=O)CCN(C(=O)COC2CCC2)CC1c1cnn(C)c1 6291,c1(C2C(C(=O)NC(CC)CNC(c3cnn(C(F)(F)F)c3)=O)C2)cccc(Br)c1 6292,Cc1cc(N)c(C(N2CC3C(NC(C4CC=CCC4)=O)C3C2)=O)cc1F 6293,Cc1cccc(OCC(=O)NC(CNC(=O)C(N2CCOCC2)C)CO)c1F 6294,C1(CC=C)(NC(c2csc(C(C)(C)C)n2)=O)CCN(C(=O)C(C2CC2)OC)CC1 6295,N1(C(C(C)C)=O)CCC2(CC1)CC2CNC(C1CCn2cncc2C1)=O 6296,C1(C(=O)O)CC2(CC(NC(C3CCCCN3Cc3cscn3)=O)CCS2(=O)=O)C1 6297,c1(C(N2C3C(NC(c4cc(C)ncc4)=O)C(C3)C2)=O)cnc2n1CCS2 6298,C1(OCC)(CNC)CCSCC1.C(c1cn(C)cn1)=CC(=O)O 6299,N1(C(C(C)(C)C2CCC2)=O)CC2CC(C1)N(C(c1cc(S(N)(=O)=O)cs1)=O)C2 6300,Cc1cncc(OCC(=O)NCC2(C)CCN(C(=O)CC3(O)CCC3)C2)n1 6301,C1(CNC(Cc2ccc(C)cc2)=O)CN(C(c2ncnc(O)c2F)=O)C(C)(C)C1 6302,C(=O)(C(F)(F)c1ncccn1)NCCCCNC(c1ccoc1C1CC1)=O 6303,C1(NC(CCCC)=O)CN(C(C2CNC(=O)O2)=O)CCC1C 6304,CC1CCN(C(=O)CC2CCC(=O)N2)C(CNC(C2CC(NS(C)(=O)=O)C2)=O)C1 6305,c1(C(N(CCCN(C)C)CCNC(C(C=C)O)=O)=O)cc(OC)cnn1 6306,C1(N(C(c2cc(CC)no2)=O)CCO)CCCN(C(c2n[nH]c(C)c2F)=O)C1 6307,C(CCN(C(=O)COC1(C)CCC1)C)(C(C)C)NC(CC1(OC)CCCC1)=O 6308,N1(C(c2cnc3cc[nH]c3c2)=O)CC23CCCC2(C1)CN(C(C1CCCS1)=O)C3 6309,Cc1ccc(C(N2CCC(CN(C)C(C3CC(=O)NC3(C)C)=O)C2)=O)cc1CO 6310,CCCCC(F)C(=O)NC1CCCCC1C(=O)NCc1cc(C)nn1C 6311,C1(OC)CC(F)CN(C(C2CCC(C)N2C(=O)CCn2cnccc2=O)=O)C1 6312,C1(COC)(NCc2cscc2Cl)CCCC1 6313,c12cc(nc(C3CC3)n1)S2.CC1CCC(C)N1CC(=O)NC1CC(C(F)(F)F)C1 6314,C(=O)(CC(C)(C)CC(F)F)NC1C2CC(NC(Cc3c(C)n[nH]c3)=O)CC21 6315,C(C(C)(C)CC(=O)N(CC(C)(C)CNC(c1ccn(C2CCC2)n1)=O)C)N(C)C 6316,C1(CC=C)(NC(C2CCC(N(C)C)CC2)=O)CCN(C(=O)C(O)CC)C1 6317,Cc1c(C(=O)NCC2C3CN(C(c4nccn4C)=O)CC23)ccn1C 6318,c1(C(=O)NC2C(NC(c3c(COC)cc[nH]3)=O)CC2)ccc2c(c1)NC(=O)CS2 6319,N1(C(C(C)NC(=O)NC)=O)CCC(C)(CC(=O)NCC(C)CO)C1 6320,N1(C(C=CCC)=O)CC(O)C(O)C1CNC(=O)CCc1cccs1 6321,CC1(C)COCC1C(=O)NCCC(O)C(=O)N1CC(CO)C1(C)C 6322,c1(NC)ncnc(N2CCN(C(C3CC=CCC3)=O)CCC2C)c1[N+](=O)[O-] 6323,C#Cc1cc(C(=O)NCCC2CCN(C(=O)CC3(C)CC3(F)F)CC2)ccc1C 6324,N1(C(C(F)=CC)=O)CC(NC(=O)Cn2cnc(Br)n2)CC(O)C1 6325,C(=O)(C(C)(C)CCC#N)NC(CNC(c1c(NC(C)=O)cncc1)=O)C1CCC1 6326,N1(C(C=CC(C)=O)=O)CCCC(C(N)=O)(NC(=O)C(C)Cc2ccc(F)cc2)C1 6327,CCCCCC(F)C(=O)NCC1CN(C(=O)COC2CCCCC2)CC12CCC2 6328,N1(C(CN(C)C2CC2)=O)CCN(C(C2CCN(C)S2(=O)=O)=O)CC1CC(F)F 6329,C1(O)(CNC(Cc2cc(C)[nH]n2)=O)CCN(C(C2CC2c2ccccc2)=O)CC1 6330,C1(NC(CC(C)(C)OC)=O)CC2CCC(C1)N2C(=O)Cc1ccc(C(C)C)cc1 6331,C1(C(C(N2CC(F)(CC)C2)=O)C)CCCN(C(c2cncnc2C)=O)C1 6332,c1(C(N(CCN(C(c2c(OC)n[nH]c2)=O)C)C(C)C)=O)cn2cc(C)ccc2n1 6333,c1(C(=O)NCC(C)NC(=O)CCc2ccccn2)cc(F)c(F)c(N)c1Cl 6334,N1(C(c2c(CC)noc2)=O)CC2(CCN(C(c3ccc(CSCC)[nH]3)=O)C2)C1 6335,N1(C(=O)Nc2ccc(OC(C)C)cn2)CC2(CC2)c2ccc(Br)cc21 6336,c1(NC23C(CN(C(c4scc(OC)c4)=O)C2)CCC3)nc2ccc(F)cc2o1 6337,C1(NC(=O)CN(C(=O)CCC2OCCO2)C2CCC2)CCC2CC12 6338,C1(NC(C(C2CCCCC2)OC)=O)CCNC(=O)CC1 6339,CN1CCc2cc(C(N3CCN(C(=O)C(C)(C)C(F)F)CC(CO)C3)=O)sc2C1 6340,c1(OC)cn(CC(=O)NC2COCCN(C(=O)C(C3CC3)OC)C2)c(C)cc1=O 6341,Cc1ncnc(C)c1CC(=O)NCC(CNC(C1COC(C)(C)C1)=O)C(F)(F)F 6342,c1(CNC(c2ccc(OCCCC)nc2)=O)ccc2cccc(Br)c2n1 6343,c1(C(N(CC(CN(C(CSCCCC)=O)C)O)C)=O)oc(C2CC2)nc1C 6344,CC1CCC=C1C(=O)NC1(C(=O)NC(CCO)C2CC2)CCSC1 6345,CC1CN(C(c2nccnc2C(N)=O)=O)CC1NC(C1C2CCCC12)=O 6346,c1(C(=O)OC)ccc(C(=O)NCCC(C)(C)NC(=O)CC(C)(C)O)c(F)c1 6347,Cc1cc(-c2cn(CC(F)(F)CNC(=O)C(C3CCOCC3)F)nn2)ccc1F 6348,Cc1cc(C(C)NC(c2ncsc2Br)c2nnnn2C2CC2)no1 6349,N1(C(=O)C(c2cccc(C(F)(F)F)n2)(F)F)C2CCCC1CC(O)C2.O=C 6350,C1(C(C)NC(C(F)=C(C)C)=O)CCN(C(c2coc(CO)c2)=O)CC1 6351,C1(NC(CC(C(C)C)O)=O)CCN(C(C23CCCCC2C3(F)F)=O)C12CCCC2 6352,N1(C(C(CC)NC(N)=O)=O)CC2N(C(C3CCC(O)CN3C)=O)CCC2(C)C1 6353,CCCCC(C)CCC(=O)N(CCCCN(C(=O)CC(C)(C)O)C)C 6354,C1(NC(COC(CC)CC)=O)(CNC(=O)C(COC(C)C)N(C)C)CCOC1 6355,c1(C(=O)NCCN(C(=O)C(C2CCCO2)OC)CCC)cc(C(F)(F)F)no1 6356,c1(C(N2CCC(C)(CNC(C3C(C)CCC3)=O)CC2)=O)ccccc1N=[N+]=[N-] 6357,N1(C(CC(OCC)OCC)=O)CCC(F)C(NC(c2ccc(Cl)c(OC)c2)=O)C1 6358,C=CC(O)(C(=O)NC1CC2CCC1N(C(=O)CCn1cncn1)C2)C(F)(F)F 6359,N1(C(C(CCOC)NC(c2cnc(C)cc2C)=O)=O)CCC2CCCC2CC1 6360,N1(C(C(CC)(F)F)=O)CCCC(C)(CNC(c2ccc(Br)c(OC)c2)=O)C1 6361,c1(Cc2onc(-c3cccc(-c4cccc(Cl)c4)c3)n2)ccc2cnccc2c1 6362,N1(C(C=CC(C)C)=O)CCC2(CC(NC(=O)Cc3csc(Br)n3)C2)C1 6363,C1(CC=C)(NC(c2cc(CC)on2)=O)CCN(C(C2COCCC2C)=O)CC1 6364,C(=O)(CCC(C)(C)[N+](=O)[O-])NC1CCN(C(C(C)(C)SC)=O)CC1F 6365,c1(OCC)cc(CNc2cccc(-c3cc(CC)n[nH]3)n2)cc(F)c1 6366,C(=O)(C(F)(F)C(C)O)NC(CNC(COC(CC)C)=O)CC(C)C 6367,N1(C(c2cc(O)ncn2)=O)CCC2(CC1)CC(C(N1CCC(CC3CC3)C1)=O)C2 6368,Cn1ncc(C(=O)NC2CCN(C(=O)C(C3CCC(=O)CC3)F)C2)c1Cl.C1CC1 6369,C(CCC(C)C)(C(=O)NCCc1nc(C)cs1)NC(C1C(=C)C1C(=O)OC)=O 6370,c1(C(=O)NC(C)CCNC(c2scnc2Cl)=O)ccnc(O)c1 6371,c1(NC)ccc(C(=O)N(CCCOCCNC(=O)Cc2c[nH]nc2O)C)nc1 6372,CS(=O)(=O)C1(C(=O)NCCN2CCC(NC(=O)CC3C=CCCC3)CC2)CCC1 6373,CCCCC(CNC(=O)Cc1cncn1C)NC(=O)CC(C)N(C)C 6374,Cc1nccnc1-c1cn(CC(=O)NC2CC(C(N)=O)C2)nn1 6375,C1(C(N(CC(=O)NCCC2(COC)CCC2)C)=O)C=C(C)CS1 6376,N1(C(CC(=O)N(C)C)=O)CCC(NC(=O)CN(C)S(=O)(=O)N(C)C)C(CO)C1 6377,N1(C(CC(CC)NC(C2CC2C)=O)=O)CCC(CC)(CC)CC1 6378,c1(C(N2CC(N(C(C(CC3CC3)OC)=O)C)C2)=O)c(Br)ccc(F)c1C 6379,CC1SCCCC1NC(c1ccc(CO)cc1)=O.C12(CCSC1)C(=O)N2 6380,C#CC1(F)CN(C(c2ncoc2CNC(=O)C(C(C)C)OC)=O)C1 6381,C1(CNC(=O)CCc2ncc[nH]2)CN(C(=O)C2=CSCCO2)CCCO1 6382,C(=O)(CCC(C)(C)C)N1C(C)CC(NC(C(Cc2ccc(C)cc2)N(C)C)=O)C1 6383,Cc1cnoc1C(=O)NCC(C)(O)CNC(c1[nH]cnc1C)=O 6384,C1(CCNC(c2ccc(F)cc2)c2n(CCC)nnn2)CCC(C)(C)O1 6385,c1(CN2CCC(C(N(c3ccc(Cl)cc3)CCC)=O)CC2)cccc(OC)c1Cl 6386,C1(F)(CNC(c2n(C)nnc2)=O)CCCN(C(=O)C(C)(C)CF)C1 6387,C1(NC(C=CC=CC)=O)CN(C(=O)Cc2ncc(C)[nH]2)C2CCCC12 6388,C1(NC(C(C)(C2CC2)OC)=O)CCCCC1C(=O)NCCC12CCCC1C2 6389,C(=O)(C(C)(C)CC(F)F)NCC(C(C)C)NC(c1c(Br)cn(CC)n1)=O 6390,c1(CCNC(c2c(Br)cc(C)c(C)n2)=O)ccc2c(n1)OCCO2 6391,C1(C(N2CC(N(C)CC)C2)=O)CCCC(NC(C2(C#N)CCC2)=O)CC1 6392,C1(CNC(C(Br)=C(C)C)=O)CN(C(C2CC2c2cncn2C)=O)CCCO1 6393,c1(CNC(CC2N(C(C(C)n3cccc3)=O)CCC2)=O)ccc2nc[nH]c2c1 6394,C(CCN=c1nc2c(ncn2CC)c(NC(C2CC2)C)[nH]1)N(S(C)(=O)=O)CC 6395,C(=O)(C(C)(C)Cc1ccc(O)cc1)NCC(CNC(c1n(CC)nnc1)=O)OC 6396,Cc1cc(C(=O)OC2CCC23CCC3)sc1-c1cccnc1 6397,O=C(N=c1[nH][nH]c2c1CN(Cc1c(O)cccc1Br)C2)c1cc(F)c(F)cc1F 6398,N#CC1=C(C(=O)N2CCCC(CCNC(C34CCC(CC3O)C4)=O)C2)CCC1 6399,C(C(O)CC(=O)NC1CCCC(C(=O)NCCc2nc[nH]n2)C1)N(C)C 6400,N1(C(c2nc(OC)oc2)=O)CC2CC3CC2C1C3NC(c1cc(C)cc(F)c1)=O 6401,Cc1[nH]c(C#N)cc1C(=O)NCCC1CN(C(C2CCCOC2C)=O)CCCO1 6402,C(=O)(C(C)C(C)NC(=O)CC1CNC(=O)O1)NCc1c(C(C)(C)C)n[nH]c1 6403,C1(C(N2CC3(C(NC(CCCOC)=O)CCC3)C2)=O)CCC2(CCCC2)CC1 6404,CC(CC(=O)NCc1ncoc1CCNC(=O)C#CC1CCOC1)C(C)(C)C 6405,S(=O)(=O)(c1cc2sc(=NCc3cc4n(n3)CCCO4)[nH]c2cc1Cl)NCCC 6406,N1(C(=O)C=CCO)CCCCCCC1C(N1CC2(CO)CC2(CO)C1)=O 6407,C=CC1OCCCC1C(=O)NCCN(C(C1CCCCC1)=O)CC1CC1 6408,C(=O)(CS(=O)(=O)CC(=O)N(C)CCNC(C1CCCC2(CCC2)C1)=O)OC 6409,N1(CC(N2CC3CC(O)CC2C3)=O)Oc2ccccc2S1(=O)=O 6410,C1(CNC(CCC(=C)Br)=O)C(C)CCCN1C(=O)CCc1ccc(F)nc1 6411,C1(NC(C2C3CCCOC23)=O)CCCN(C(=O)CC(F)(F)Cl)C1 6412,C1(C)(C(C)NC(C(c2ccc(O)cc2)OC)=O)COCCO1 6413,C(CCS(C)(=O)=O)(C(=O)N(C1CCCN(C(=O)COCCC(C)C)C1)CC)OC 6414,CC(CN=c1cc[nH]cc1S(=O)(=O)NCC1CCCC12CCC2)S(N)(=O)=O 6415,c1(C(=O)N(C2CCCCC2C(N)=O)c2n(C)nnn2)cc(C(F)F)ccc1F 6416,CC1=CCC(C(N2CC(COC)(NC(C3CCCC34CC4)=O)C2)=O)CC1 6417,N1(CC)CCC=C(c2cc(C(=O)N(CC(F)(F)F)C)cc3c[nH]nc23)C1 6418,C(CCCCC(=O)NC1CCC(C)(CNC(c2[nH]ccc2C)=O)CC1)=CC 6419,C1(CC)C(C(=O)NC2CC(NC(=O)C=CCNC(=O)OC(C)(C)C)C2)CCN1C 6420,N1(C(c2cc(S(N)(=O)=O)cs2)C(=O)NC(CC)C)CCC2(C1)C(=O)NC(=O)N2C 6421,N1(C(C(C(C)O)C)=O)CCN(C2CCCN(C(c3c[nH]ccc3=O)=O)C2)C(=O)C1 6422,C(=O)(CC(C)(C)N(C)C(C1CCC(=O)O1)=O)NC(c1ncn(C)n1)C 6423,c1(C(=O)NC(C(C)NC(c2cccc(C(C)C)n2)=O)CO)cc(Cl)c(F)cc1O 6424,c1(C(=O)NCCCNC(COCCOC)=O)csc(I)c1 6425,Cc1ccc(F)c(C(N2CC(O)(CNC(=O)C(C)C(C)C3CCCCC3)C2)=O)c1 6426,CC#CCCC(=O)NC(C)(CNC(=O)C(C)n1ccnn1)C(C)C 6427,C(C(C)C(C)C(=O)NCC1(F)CN(C(=O)CSc2ccc(C)cc2)C1)OC 6428,N1(C(c2c(O)cc(C)nn2)=O)CC(NC(=O)CCC2CC2(Cl)Cl)CC12CCCC2 6429,c1(C(=O)NC(CCNC(C)=O)C(C)C)cc(O)nc2c(Br)cccc12 6430,C(=O)(C(O)C(F)(F)F)NC(CCNC(C1CN(C2CCN(C)CC2)C1)=O)C1CC1 6431,N1(C(c2ccc(OC)cc2I)=O)CC2OCCN(C(=O)Cc3cc(C)on3)C2C1 6432,C(=O)(C(C)C(O)CC)NCCCOCCC(=O)NCCN(CCC)CC 6433,N1(C(Cc2c[nH]c(=N)s2)=O)CCC(Oc2cccc(F)c2)CC1 6434,C(=O)(CC1COCc2ccccc21)NCCN(C(Cc1ccc(C)s1)=O)C1CC1 6435,C#Cc1ccc(F)c(C(=O)N(CC)CC2CCCN2C(C2CC(F)C2)=O)c1 6436,C1(NC(Cc2ccc(C)s2)=O)CC2(NC(=O)CCC3(C)CC3)COC1C2 6437,C1(C2CCCN(C(=O)CC3(C)CC3(Cl)Cl)C2)(NC(c2c(C)con2)=O)CC1 6438,c1(C(=O)NCC=C)cnc2n1CCN(C(c1cc(-c3ccccc3)on1)=O)C2C 6439,c1(C(N)=O)cccc(CNC(C2CC(F)CN2C(C2CNC(=O)O2)=O)=O)c1 6440,N1(C(c2c(C)nccn2)=O)CCN(C(C2OCCCC2(C)C)=O)C2CC12 6441,C1(C(=O)NCC2(C)N(C(C(C)=C(C)C)=O)CCC2)CC2(C1)CC(C)(C)C2 6442,CN1CCOc2c(C(N3CC(CNC(C4(C)COC4)=O)CC3(C)C)=O)cccc21 6443,c1(NCCCN(S(=O)(=O)c2cnn(C)c2)C)cccc2c1OC(C)(C)C2 6444,c1(CNCCSC(C)(C)C)cc(N2CCOC(CCO)C2)ncn1 6445,c1(C(N2CC3C(C2)C3(F)F)=O)cn2cc(-c3c[nH]c4ccccc34)ccc2n1 6446,CC1CC(C(=O)NCc2cc(C(=O)NCC3CC4(CC4)CO3)ccn2)CN1C 6447,N1(C(C2(CC#C)CCOCC2)=O)CCC2CN(C(=O)C(C)OCC(F)(F)F)C2C1 6448,N1(C(CCC=CC)=O)CCC(C)C(NC(c2ccc(O)c(C(N)=O)c2)=O)C1 6449,C12(C(N3CC4CC4(CNC(c4snc(O)c4Cl)=O)C3)=O)CCCN1CCC2 6450,c1(C(=O)NC2CCCN(c3ccccc3F)C2=O)cc2cccc(F)c2s1 6451,C1(C(=O)NC(CNC(c2c(CC)nccn2)=O)CCOC)CC2(CCC2OC)C1 6452,c1(C(=O)NC2CC(NC(c3cccc(C4CC4)c3)=O)C2)cnn2cccc(Cl)c12 6453,Cc1cn2c(C(N3CC(N(C(=O)CC(O)CC4CC4)C)C3)=O)c(C)nc2s1 6454,c1(C(C)C)noc(CNC(c2nnnn2C2CC2)C2(C)COC2)n1 6455,C1(OC)CN(C(=NCCCSC)NCC2CCN(C(C)=O)C2)CC1OC 6456,C(=O)(CCCCCn1cnnn1)NCCC(C)(C)NC(C1(C)CC1)=O 6457,CCCC(C)(O)CC(=O)NCCCC(C)(C)NC(=O)Cc1ccc(Br)cc1 6458,C1(c2ccc(OCC)cc2)CCN(C(=O)C(F)C(C)C)CC1NC(=O)C(C)CC 6459,C1(C(N2CCCC2CC(c2cccs2)O)C(=O)NC2CCCC2)CC12CCC2 6460,C(CCC(C)(C)NC(=O)CC1(N(C)C)COC1)NC(C1(C(C)C)CC1)=O 6461,N#Cc1cc(S(=O)(=O)NC2CCCC23CCOCC3)ccc1Br 6462,C(=O)(C1=CC2CCC1C2)NC1CCN(C(c2ccc(C)c(O)c2)=O)C1 6463,C12(C(=O)NCC(CC)NC(=O)CCN3CCCS3(=O)=O)CCCC(CO1)C2 6464,Cc1cc(N)c(C(=O)N(C2CN(C(C3CCN3C)=O)CC23CC3)C)cc1C 6465,c1(C(=O)NC(C)(C)CNC(C2CCc3n[nH]cc3C2)=O)ccc(F)c2ccoc12 6466,c1(C(=O)Nc2ccc(CC)c(F)c2)nsc2ccc(C)cc12 6467,CN(Cc1c(Oc2ccccc2)cccc1F)N1CC(COc2ccccc2)C1 6468,CC1CCCC(C)N1CCC(=O)NCC1(C)CCN(C(c2sccc2F)=O)C1 6469,C1(CN(C)C)COCC(=O)NC2(C)CC1(NC(C(CSC)OC)=O)C2 6470,C(=O)(C(O)C(C)(C)C)NC1(CNC(c2nccc(CC)c2)=O)CCCC1 6471,c1(CC)nnc2cc(N3CCCCC3CNC(C3(C)C(C)(C)C3(C)C)=O)ncn12 6472,N1(C(CN2C(C)CCC2)=O)CCOC2(CCN(C(=O)CC3CNC(=O)C3)CC2)C1 6473,N1(C(CCC2N(C(CC=C)=O)CCCC2)=O)CCOC(C(=C)C)C1 6474,Clc1ccc2[nH]c(=NCc3ccccc3C(c3c(Cl)sc4nnsc34)=O)sc2c1 6475,CON(CN1CC(=O)N(c2cccc(F)c2)C1=O)CCC(C)C 6476,Cc1cc(C#N)sc1C(=O)NCC1CC(CNC(c2nc(Cl)cs2)=O)CO1 6477,C1(NC(C(C2CC2)OC)=O)CCC(N(C(=O)C(CC#N)c2ccccc2)C)CC1 6478,C1(NC(c2scc(OC)c2)=O)CCS(=O)(=O)C12CN(C(C1(C)CC=CCO1)=O)C2 6479,C(=O)(CCC(C)SC)NC1(CNC(c2cc(COC)on2)=O)CC1 6480,C1(NC(CCNC(CCOC)=O)=O)CC(N=c2[nH]c3cc(C)ccc3o2)C1(C)C 6481,c1(OCC(N2CCC(=C)CC2C(=O)OCC)=O)c(Cl)cc(Cl)cc1Cl 6482,C1(CSC)CCN(C(=O)C(C)(C2CCC2)NC(c2cc(Cl)cs2)=O)C1 6483,C1(F)(C(N2CC(C(=O)Nc3cc(C)cc(F)c3)C2)=O)CCCCC1(F)F 6484,C1(CNC(C2(CC=C)CC=CC2)=O)C(C)CCN1C(c1nn(C)nc1Br)=O 6485,Cc1oc(C#N)cc1C(N1CCC(C)(C)C1C(N1CCCC(CO)CC1)=O)=O 6486,N1(C(C(CCSC)O)=O)CC2CCC(NC(c3cnc4sccc4c3)=O)CC2C1 6487,c1(C(=O)NCC2C(CNC(c3c(CC)[nH]c(=N)s3)=O)C2)cscc1S(C)(=O)=O 6488,C(CNC(=O)CCN1CCCCC1C)(CC(C)C)NC(CSCNCCCC)=O 6489,c1(CNC(COC2CC(NC(C(CC#C)O)=O)C2)=O)cc(F)c(N)cc1F 6490,C1(NC(N2CC(n3c(C(=O)OCC)ncn3)C2)=O)CCc2ncccc2C1 6491,N1(C(c2c(=N)[nH]cnc2)=O)CC(F)(F)CC1CCNC(c1ncc(Cl)cc1Cl)=O 6492,c1(NCC)c(NC(c2cc(OC)cc(C)n2)=O)cc(Cl)cc1Br 6493,C=CCC(C)(C)C(=O)NCC(C)(C1CC1)NC(c1nccnc1N)=O 6494,N1(C(c2cc(C)sc2C)=O)CC2CCC1(CNC(c1n[nH]cc1C)=O)CC2 6495,N1(C(c2cc(C)nn2C)=O)CCOC2CN(C(c3conc3C(C)(C)C)=O)CC12 6496,c1(C(N2CC(CC(C)NC(=O)CNc3cccnc3)C2)=O)ccnc2ccnn12 6497,c1(C(=O)NCC(C)N(C(C(CC)n2cncn2)=O)C)cn(C)nc1COC 6498,c1(CSCC(=O)N(C)CC2CCC2NC(c2ccns2)=O)nc2ccccc2[nH]1 6499,CCC(C)C(CC(=O)NCC(C)(F)C(C)C)NC(c1cccc2ccnn12)=O 6500,c1(CNC(C2CCN(Cc3ncccc3F)C2)=O)ccccc1[N+](=O)[O-] 6501,N1(C(c2ccn(CC)n2)=O)CC2CCCN(C(c3cccc4c3CCC4)=O)C2C1 6502,Cc1noc(C)c1C(=O)NCC(F)CNC(C1(C)CC(C)(C)C1)=O 6503,c1(C(=O)NCC2N(C(C3CC(C)N(C)CC3)=O)CC2)ccc2cccnn12 6504,C(C)(C)(C(=O)N(C)CC1(CNC(c2coc(C(F)F)c2)=O)CC1)OC 6505,N1(CC)CCCCCC(N=c2cc(C)[nH]cc2C#N)C1.N1CC(O)CCC1=O 6506,c1(C(=O)NCC2(NC(C3CCC(N(C)C)CC3)=O)CC2)ccc(N)c(O)c1 6507,c1(OC)nnc(NCCCCc2cccnc2)cc1N 6508,c1(N)cccc2ccc(O)cc12.N1(NC(=O)C)CC2CC(C1)CS(=O)(=O)C2 6509,c1(CNC(=O)CC2CCCN(C(=O)CC3CCC3)CC2)ccc2cc[nH]c2c1 6510,c1(Sc2cc(C#C)n(C3CCCCO3)n2)sc2c(c1F)CCCC2 6511,C(C(C)C(=O)Nn1cccn1)N(C(C1C(C)=CCS1)=O)C 6512,C(=O)(C=C1SCC(=O)N1C)NCC1C(NC(C(C2CC2)OC)=O)COC1 6513,N1(C(Cn2ncc(C#C)c2)=O)CC(C)CN(C(=O)CCCCC=C)C(C)C1 6514,CCCC(CCC)=CC(=O)NC1CC(NC(=O)CCCn2cccn2)C(O)C1 6515,C1(C#N)(C(=O)NC2(CNC(CC3(NC(C)=O)CC3)=O)CCC2)C(C#N)C1(C)C 6516,c1(C(=O)NC(CC)CN(C(=O)CC(C)CC)C)cc2c(OC)cc(OC)nc2[nH]1 6517,N1(C(CC(=O)OC)=O)CCC2(CCCC2CNC(=O)Cc2csc(C)c2)CC1 6518,C1(C2CCN(C(C3CC(F)C3)=O)CC2)(NC(c2coc(Br)n2)=O)CCC1 6519,c1(C(N2CCC3CN(C(CC4CCN(C)C4)=O)CC32)=O)coc2ccc(O)cc12 6520,c1(OC(C)C)ccc(C(=O)NC2CC23CC(NC(c2c[nH]cc2CN)=O)C3)nc1 6521,C1(CNC(C(C)NC(c2ccoc2)=O)=O)C2CC1N(C(=O)CCC1OCCO1)C2 6522,C1(c2nc(-c3ccc(N)cc3)nn2Cc2cccnc2)CC12CCS(=O)(=O)CC2 6523,CC1CC(C(=O)NC2(C(=O)NC(c3cncs3)C)CSC2)CC(=O)N1 6524,c1(CC)cc(=NCC2CCCC(NC(C3CC(N(C)C)C3)=O)C2)[nH]cn1 6525,C12(CNC(C(CCCCC)F)=O)CCCC1N(C(=O)COC)CCC2 6526,C(C(=O)NC1CN(C(c2cc(O)nn2C)=O)CC1C(F)(F)F)(C(C)C)SCC 6527,N1(C(c2ccc(C(C)=O)cc2)=O)CCC(NC(c2n[nH]c(C3CC3)n2)=O)CC1C 6528,C12(NC(C3CCCCC34CCC4)=O)CC(C3CCCC3)(C1)C2 6529,N12CCOC3(CCCC3)C1C(=O)OCCCC(C)C2=O.C(CC#N)NC(=O)NC 6530,c1(CC=CC(=O)NCC(CNC(C2(N3CCCC3)CC2)=O)OC)ncccc1O 6531,Cc1c(Br)ccnc1C(=O)NC1CCC1CNC(c1snnc1C1CC1)=O 6532,c1(C(=O)Nc2cnccn2)ccc(=NCc2cc(F)ccc2Br)[nH]c1 6533,Cc1ccc(OCC(=O)NC2CC(F)CN(C(c3c[nH]nc3F)=O)C2)c(F)c1 6534,N1(C)CC2(CCC(CNC(=O)Cn3cc(C4CC4)cn3)O2)C1.C1(=O)CN1.C(C)CC 6535,Cc1cnc(C(=O)NC(C)CCN(C)C(C2CC2(C)C(F)F)=O)c(Br)c1 6536,Cc1ccc(C)c(C(=O)NC(CNC(c2cn[nH]c2)=O)C(C)C(C)C)c1 6537,C1(O)(CNC(CN2CC(C)(C)C2)=O)CCCN(C(c2cnc3n2CCC3)=O)C1 6538,N1(CCN(C(C2(OC)CCCC2)=O)C)CCN(C(=O)CCS(C)=O)CC1 6539,c1(C(=O)NC(C(C)NC(c2c(C)oc(C)c2C)=O)C)ccc2c(c1)COC2 6540,C1(CCC)CN(C(=O)Cc2nocc2C)CCN1C(c1cc(C)n(C(F)F)n1)=O 6541,c1(OCC(=O)N(CC(C)NC(c2cc(CC3CC3)on2)=O)C)ncc(Cl)cc1Cl 6542,c1(N(C2(C#N)CCNC2)Cc2c(C)noc2C)ncnc2cnn(C)c12 6543,C(=O)(C(CC)NC(=O)CCn1cnc(=N)[nH]1)NC1CC(CCOC)C1 6544,O=C(C1=NOC2(CCC2)C1)NCC1(C(N2CCCC(CO)C2)=O)CC12CCC2 6545,N1(C(c2ccc(C#C)cn2)=O)CCC2CCC(NC(c3ncoc3CC)=O)C1C2 6546,C1(O)(CNC(c2cc(I)c(Cl)cc2F)=O)COCCC1O 6547,C12(COC)CC(CNC(=O)C(C)CC(N)=O)(CN1C(c1n[nH]c(C)c1O)=O)C2 6548,c1(-c2cn(CC3CCC(NC(C(C)(C)CO)=O)CC3)nn2)cccc2c1OCC2 6549,N1(C(C2(CC=C)CCCC2)=O)CCCC(C(C)NC(=O)C(N)=O)C1 6550,Cc1csc(CCCC(=O)NCCC2CCN(C(=O)CC34CC(C3)C4)C2)n1 6551,N1(C(Cc2cc(C)on2)=O)CC(C(=O)NC(c2ncc(C)o2)C)OC(C)C1 6552,C1(CNC(c2c(C)nn(CC(F)F)c2)=O)CC2(CC2)CN1C(=O)C(C)CCO 6553,N1(C(C(=O)Cc2ccccc2)=O)CCC2(C1)CN(C(C1CC=CCC1)=O)C2 6554,C12(C(N3CCC(C)(CNC(c4nnc(C)s4)=O)CC3)=O)CCC(CC1)C(C)O2 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6750,C(=O)(C(C)CC(=O)NCCCN(CCCNC(=O)C(C)OC)CC(C)C)OC 6751,c1(N(c2ncnc(OC)c2C)C(c2ccccn2)=O)ccc2c(c1)CCNC2 6752,Cc1ccc(C(F)F)c(C(=O)NCC2CC(NC(C3(C)CC4CC4C3)=O)C2)c1 6753,CC(CCC(C)(C)C)C(=O)N1CC2CC1C2NC(=O)CNC(=O)CC(F)(F)F 6754,C12(C(N3CCCC(CN(C)C(c4ccn(C)n4)=O)C3)=O)CC(C3COC3)(C1)C2 6755,C1(CNC(=O)CC(O)C2CCCC2)(NC(C2CCC2)=O)CC(F)(F)C1 6756,C1(C(N2CCCC(CCNC(C(CC)(C)C)=O)C2)=O)CCOC(C)(C)C1 6757,c1(CCC(=O)NCC2(NC(C3CCN(C)C3)=O)CCCC2)ccc(N(C)C)cc1 6758,C1(C(N2CCC(C(N(C)CCc3cnc[nH]3)=O)C2)=O)Cc2ccccc2C1 6759,C1(CNC(C(C)=C2CC2)=O)CC(NC(c2cnn(CCC(F)(F)F)c2)=O)CC1O 6760,N1(C(C2CCC(F)(F)C2)=O)CCC2(CCCN2C(=O)CCCn2ccnn2)C1 6761,c1(N(C)C)ccc(F)c(C(=O)NCCC2CCC(NC(C3C4COCC34)=O)C2)c1 6762,c1(NCC(C)NC(C(=O)N(CC(C)N(C(C)=O)C)C)=O)ccccc1 6763,CCC(C)C(C(=O)N1CC(CO)=C(F)C1)N(C(=O)CC(Cl)Cl)C 6764,C(=O)(C1=CC2C=CC(C1)C2)NCCOCCNC(C(Cc1cn(C)nc1)O)=O 6765,C(CC(=O)N1CC=CC1C(=O)NCC1(OC(C)C)CCC1)(C(N)=O)NC(C)=O 6766,C=CCCCCC(O)CNC(c1ncsc1C(C)C)=O 6767,Cc1ccc(OCC(=O)NCC2CN(C(C3CCCN3N=O)=O)CC2O)cc1C 6768,c1(C(N2CCC(O)(C(C)NC(C(CSC)O)=O)CC2)=O)cc(F)c(C)cc1F 6769,c1(C(N2CCC(CC=C)(NC(=O)C(=O)N(C)C)CC2)=O)ccc(S(C)(=O)=O)o1 6770,C=CC(O)C(=O)N1CCC1CNC(c1cc(C2(C)CC2)n[nH]1)=O 6771,c1(C(=O)NC(CNC(c2nc(C)n(C)c2)=O)C(C)C)ccc([N+](=O)[O-])n1C 6772,N1(C(COC(CNC(CCC=C)=O)(C)C)=O)CC(COC)CC1(C)C 6773,C(CCN=c1[nH]ncs1)OC(C1(c2cccc(Cl)c2)CC(OC)C1)=O 6774,C(=O)(C(C)(C)CC(C)(C)C)N(CC(CC)NC(c1cnc(C)c(C#N)c1)=O)C 6775,C(c1c(F)ccc(Cl)c1F)=CC(N1CCC(O)(CNC(c2c(CC)nc[nH]2)=O)C1)=O 6776,N1(C(c2c(CC#N)cccc2)=O)CCC(C2CC2NC(c2csc(O)n2)=O)CC1 6777,Cc1oc2ccccc2c1CC(N1CCC(NC(C2(CCF)CC2)=O)C(F)C1)=O 6778,C(=O)(CS(=O)(=O)CCC(F)(F)F)N1CCCC(NC(C(N2CC(C)C2)C)=O)C1 6779,C(=O)(NNc1ncnc2[nH]cnc12)c1[nH]cc(OC)c(=O)c1 6780,n1(CC(=O)NCCC(C(C)C)NC(C2CCC(C)(C)C2)=O)cc([N+](=O)[O-])cn1 6781,CC(CNC(=O)CSc1ccccc1)(CO)NC(c1cscc1C(F)F)=O 6782,c1(OC)cc(C(=O)NC(C)CN(C)C(c2ccnnc2O)=O)ccc1Br 6783,N1(C(c2ccn(CC)n2)=O)CCC(O)C(N(C(=O)C(C)CSC)C)C1 6784,CC(C(=O)NC(C1CCN(C(C2CCCN(C(N)=O)C2)=O)C1)(C)C)S(N)(=O)=O 6785,CCCCCCC(=O)NC1CC(CCNC(c2cc(Br)n(C)c2)=O)C1 6786,C1(C(C)C)CCC(C)CC1C(=O)NC(CNC(C1(CCO)CC1)=O)CO 6787,CC1(O)CCCN(C(=O)C(C2(O)CCC2)NC(c2ccc(F)cc2)=O)CC1 6788,C(=O)(C1=NOC(C)C1C)NC1C2(CC(NC(c3c(OC)cncc3)=O)C2)C1 6789,CCC(C)C(C(=O)NC1(C(C)O)CC1)N(C)C(C1CCCCN1C)=O 6790,c1(C(N2CC(C)C(C(=O)Nc3cc(S(N)(=O)=O)co3)C2)=O)csc2ccccc12 6791,C=CCCC(C)NC(C1(CNC(c2occc2CSC)=O)CCC1)=O 6792,c1(OC)ccc(C(=O)NCC2(NC(=O)Cc3ccsc3Cl)CCOC2)cc1OC 6793,C(CCCCC(=O)NCCCN(C)C(C1(NC(N)=O)CCCCC1)=O)=CC 6794,C1(C(N2C(C#C)(C)CC2)=O)OCCC12CN(C(=O)OC(C)(C)C)C2.C1(C)CC1 6795,C1(C(N2C(C)CCCC2)=O)N(C(c2ccco2)=O)CCCC1(C)C 6796,c1(OC)ccccc1C1CC1C(N1CC(NC(C2COCCOC2)=O)C(C)C1)=O 6797,CC1(C)OC(=O)CC1C(N1CCC(CNC(c2cncnc2)=O)C1)=O 6798,C1(C(=O)NCC2C(C(NOCCCCC=C)=O)CCCC2)CCC2(CC1)CC2 6799,C1(NC(C(CC=CC)C)=O)CC2(C1)CC(C(=O)N(C)CC1(CC3CC3)CCC1)C2 6800,Cc1cc2ccc(C(=O)N(CC(C)N(C(=O)CCc3ccco3)C)C)cc2o1 6801,c1(CCC(=O)N(CCN(C(c2c(C)nn(C)c2)=O)C)C)ccc(Cl)cc1F 6802,c1(C(=O)NCC2CCCCN2C(c2cnc(Cl)cn2)=O)cc2cccc(Cl)c2o1 6803,c1(CC(C)(C)CO)nc(C2(C3CCCNC3)CCC2)n(C2CCSC2)n1 6804,CCC(CC(=O)N1CCC(N(C)C(C23CSCC2C3)=O)C1)C1CCC1 6805,c1(C(=O)NC2C3(CN(C(C4C(C)C4)=O)C3)CCC2)coc2c1C(=O)NCC2 6806,C1(NC(C(C)NC(CC)=O)=O)CCCCN(C(=O)CCC=CC(C)C)C1 6807,C1(C)(C(=O)NCCC(C)N(C(=O)CC2C=CCCC2)C)CC(F)(F)C1 6808,C(=O)(C1=C(C)OCCC1)N(C1CCC(CNC(c2c(OC)scc2)=O)CC1)C 6809,c1(CC(=O)N(CCCN(C(=O)CSCc2ccccc2Cl)C)C)ccc(O)nc1 6810,CC1CCN(C(=O)CCOC2CN(C(c3ccc(C(N)=O)[nH]3)=O)C2)CCS1 6811,c1(CNC2(C)C(NC(=O)OCC)CCC2)cc(C)nc(C)c1.C123CC(C1)(C2)C(=O)N3 6812,c1(C(N(C2CCN(C(C(CC)F)=O)C2)C)=O)ccc([N+](=O)[O-])cc1Br 6813,N1(C(c2cn(C)nc2)=O)CCC(NC(c2cn(-c3ccccc3)nn2)=O)C12CC2 6814,CCCCCCCCCC(O)C(=O)N(C(C)CNC(C1(C)CC(C)(C)C1)=O)C 6815,C1(CNC(C2C(NC(COCC(=C)C)=O)COC2)=O)CCCCN1C 6816,C1(NC(c2c(OC)noc2C)=O)CCCCN(C(=O)CC(C)c2cccnc2)C1 6817,C(C1C(C(=O)NCC2(F)CC(NC(=O)COCC(C)(C)C)C2)C1(C)C)=C(C)C 6818,C1(F)(C(=O)NC2CC=C(C)CC2)CCCN(C(=O)CCC2CCCO2)C1 6819,C1(C(=O)NCC(=C)CCNC(c2cc(N)ccc2Cl)=O)CCS(=O)(=O)C1(C)C 6820,C1(O)(CC(=O)NCC(CNC(c2c(C)nc(C3CC3)[nH]2)=O)(C)O)CCCCCC1 6821,C12(CCN(C(c3cnc[nH]c3=N)=O)C1)N(CC)C2=O.C(=O)(C1CC1)NC 6822,c1(OCC(=O)NCC2CCCN2C(=O)CC23CCCC2C3)ccc(C(F)F)nc1 6823,c1(C2(CC)CC2)ccc(C(=O)NC2CCC(NC(C3(C)CCCO3)=O)C2)cc1 6824,C(=O)(C1=CCCCC1P(C)(C)=O)N(C)CC1N(C(COCC=C)=O)CCOC1 6825,CCC(CC(=O)N1CCC(C)(C(=O)OC)C1)NC(=O)CCc1cccn1C 6826,N1(C(c2ccc(C)cn2)=O)CC2CC1CC2N1CCC(C)C1(C)C 6827,CC1COC(C(=O)NC2(C)CN(C(=O)CNC(c3ccc(Br)o3)=O)C2)C1 6828,c1(C(=O)NC2CCC(NC(CC=C(C)C)=O)C2)ccc2c(Br)n[nH]c2c1 6829,c1(C(=O)NCc2cccc(C(N(CC(C)C)CC)=O)n2)cccc2ccoc12 6830,n1(CC(C(N2C(CNC(CSCCC)=O)CCC2)=O)C)ncc2ccccc12 6831,c1(OCC(=O)OCC2(C)CCC2)ccc(Cl)cc1.c12coc(n1)CC1(CC1)NC2=O 6832,C(=O)(CCCCC(C)(C)C)N(CC(CC)NC(c1cncc(OC)n1)=O)C 6833,n1(CCC(=O)NC(CNC(c2c(C)ocn2)=O)C(C)C)c(C)cc(O)cc1=O 6834,CCCCCC(C)(C)CNC(=O)CNC(=O)C(F)CC1CCCCC1 6835,c1(N2CCC(CC(=O)NCCC=C)C2)cc(OC)nc(OC)n1 6836,C1(NC(c2nc(COCC)sc2)=O)C=CCN(c2nccc(CO)n2)C1 6837,N1(C(C2CC(NC(C(C)OCCCC)=O)C2)=O)CCC2(CCCN2C)C1 6838,C1(CNC(c2ccc(Cl)o2)=O)CCCN(C(c2cc(O)ncn2)=O)CC1 6839,C1(COC)(NC(c2cc(Cl)c[nH]2)=O)CCN(C(=O)Cc2ccc(F)cn2)CC1 6840,c1(C(=O)NCC(C)(C2CC2)NC(C(C)NC(=O)NC)=O)ccc2c(c1)CCCS2 6841,N1(C(CN(CCC)C)=O)CC(NC(C2(O)CCSC2)=O)CC2(CC2)C1 6842,N1(CC(=O)NC(CC=C)CNC(=O)C(C)OC)C(=O)c2cc(Cl)c(Cl)cc2C1=O 6843,C(=O)(CS(=O)(=O)C(C)(C)C)N1C2C(CNC(C3=NOC(C)C3C)=O)CC(CC2)C1 6844,c1(C(=O)OCC)ccc(S(=O)(=O)N2CCC(N)C(c3ccccc3)C2)c(F)c1 6845,C(CCSC)(C(=O)N1CC(OC)C(O)C1)NC(CC1(CC)CCC1)=O 6846,N1(C(CNC(=O)OC)=O)C2CCC1CC(CNC(=O)CC1CCCOC1)C2 6847,N1(C(c2nccn2C)C(=O)NC(CC)C)CCC(CC(N2CCCC2)=O)CC1 6848,c1(C(c2ccsc2)N(CC(C)N(C(=O)C(C)O)C)C)ccc2ccccc2c1 6849,C1(CC)CN(C(=O)C(CC)NC(C)=O)CC1NC(=O)Cn1cncn1 6850,c1(C(=O)NCC2OCC(CNC(CC(=C=C)C)=O)C2)ccc(Cl)c(CC)c1 6851,C1(CC(=O)N(C(C(=O)NCc2nc(CC)sc2)(C)C2CC2)C)C=NN(C)C1=O 6852,N1(C(CC2C(C)(C)C2)=O)CC(NC(c2ncc3[nH]ncc3n2)=O)C(N=[N+]=[N-])C1 6853,CCC(CCO)NC(C1CC1CNC(=O)C(c1cnn(C)c1)=O)=O 6854,C1(NC(c2c(CC)onc2)=O)CCCN(Cc2cc(F)ccc2F)CC1 6855,N1(C(C2(C#N)CC2)=O)CCOCC2(C1)CN(C(=O)C(C1CCCCC1)=O)CCO2 6856,C1(C(=O)NCC(=O)OCC=C)CC2CCC1N2C(C1CC(=O)C1)=O 6857,N1(C(CN2CCN(CC)CC2)=O)CCCN(C(=O)C2=CCC(C)CC2)CC1CO 6858,C(=O)(C1=CCN(C)C1)N(CC(CNC(C=Cc1c(C)n[nH]c1)=O)(C)C)C 6859,C(=O)(CC(C)CC(C)(C)C)NCC1C2(CCC(NC(CCS(=O)(=O)NC)=O)CC2)C1 6860,c1(CCC(=O)NCC2CCN2C(c2cnn(C(F)(F)F)c2)=O)nnc(C(F)F)o1 6861,C1(C)(C(=O)NC(c2nccn2C)CC)CN(C(=O)Cc2n[nH]c(=N)s2)CC1C 6862,C(C(CNC(c1ccc([N+](=O)[O-])[nH]1)=O)C(F)(F)F)NC(C1N(CC)CC1)=O 6863,Cc1ccc(C(C)(C)F)cc1NC(c1cc(F)ncc1F)CCl 6864,C(=O)(C(C)C(C)S(C)(=O)=O)NC1(CCNC(c2ccn(CCC)n2)=O)CCCC1 6865,CCCC(C(=O)NCCCC(C)(C)NC(=O)C(C)OC1CCCCC1)NC(C)=O 6866,Cc1ccc(C(=O)NC2CC(CNC(c3cc(=O)n(C)cn3)=O)C2)c(C2CC2)n1 6867,NS(=O)(=O)C1(C(=O)NC2CC(NC(=O)C=Cc3cocn3)C23CCC3)CCC1 6868,CN1C(=O)CCC1C(=O)NCC1CCCCC1NC(c1cccc(C2CC2)c1)=O 6869,CC(CCCCN=c1[nH]cc2ccnc-2[nH]1)NC(c1cnc2c(n1)CCCC2)=O 6870,N1(C(CCNC(=O)OCC)=O)CCCCC(C(=O)Nc2cnn(CCOC)c2)C1 6871,CC1CCCC1(CO)NC(=O)Cc1cn[nH]c1 6872,C1(C(=O)NCc2ccc(C)cc2)C2C3CC4C1C2C34C(=O)Nc1ncccn1 6873,C(=O)(CCC(C)(F)F)N1CC(CN(C(=O)CSC(C)(C)C)C)OCC1 6874,C12CCN(CC1)C2.N1(CC=CC(=O)NC(N)=O)CCOCC1 6875,c1(C(=O)NC(CNC(c2c(C#N)ccs2)=O)C2CC2)cccn2c(O)nnc12 6876,N1(C(c2c(ON=C(C)C)cccc2)=O)CCC2(CC(NC(=O)CC3(O)CC3)C2)C1 6877,C1(CNC(CC=C=C)=O)(CO)CCCN(C(=O)Cc2c(C)nn(C(C)C)c2C)C1 6878,c1(C(N(CCCNC(=O)C(C)C(F)F)CCC)=O)cccc2ncnn12 6879,C(C(=O)NC1CCN(CC(=O)Nc2cccc(C)c2)CC1C)(C(C)(C)C)OC 6880,CC1(C)C(C)(C(=O)NC2CCC(NC(=O)CC(=O)NC3CC3)C2)C1(C)C 6881,Cc1cc(=NCC2CC(NC(=O)C3COc4ccccc43)C2)[nH]c(S(C)(=O)=O)n1 6882,C(C(CC(=O)NCC(C)C(=O)SC1CC1)N(C)C)NC(CN(CC)CC)=O 6883,C1(N(C)C(c2cnsn2)=O)CN(C(=O)C=Cc2ccc(O)cc2)CC1(C)C 6884,C(CC(N)=O)(C(=O)N1CCNC(=O)C1)NC(C1OCCN(C)C1)=O 6885,C1(C(=O)O)(C(N2CC(O)(CC(C)C)C2)=O)CC2CCC1C2.c1(CC)nn[nH]n1 6886,CC1COCC(C(=O)N(C)CC=CC(=O)N(C2CCCC(O)C2)C)O1 6887,N(C1CCC2(CC2)c2cc(Br)ccc21)Cc1cc2ccc(O)cc2cc1 6888,c1(SCC)cc(Cl)ccc1C(=O)NC1CCC(NC(=O)C(C)n2cccc2)CC1 6889,N1(C(=O)NC2CC(F)C2Cc2cccc(-n3ccnc3)c2)CC(O)C(O)C1 6890,CC1(C)CC(NC(C2C3COCC23)=O)CCN(C(c2ccnc(C3CC3)c2)=O)C1 6891,N1(C(c2c(CC)nn(C)c2)=O)CC(F)(F)CC1(C)CNC(c1ccnn1CC)=O 6892,C1(NC(c2c(C)nccn2)=O)CCCC12CCN(C(=O)C1=CCS(=O)(=O)C1)C2 6893,Cc1nc(S(=O)(=O)N2CCCCCC2CNC(=O)C(F)CC(Cl)Cl)ccc1Br 6894,C(=O)(C1=CCCCCC1)NC1CC(F)(CNC(=O)CC2CCCNC2=O)C1 6895,CCCCCC(O)CC(=O)N(CCCN(C)C(c1ccnc(F)c1N)=O)C 6896,C1(NC(C2N(C)CC(C)(C)C2)=O)CCC2CC1CN2C(=O)C1=CCOCC1 6897,C(CC(C)(C)CNC(=O)C(C1CCN(C(=O)C(CO)NC(N)=O)C1)F)OC 6898,N1(CC)CCCC2(CCCO2)C1.c12ccccc1CN(C)C2=O 6899,c1(CC)ccc(Cl)c(COC(C2(n3cc(C#N)cn3)CC2)=O)c1 6900,CC(C)(CCC(=O)N1CCC(NC(C2CCC=CCCC2)=O)C12CCC2)[N+](=O)[O-] 6901,CC1(C)CCC(CNC(=O)C(CNC(=O)C(F)=CC2CC2)CC2CC2)O1 6902,N1(C(C=CCCC)=O)CCCC2(C1)CN(C(=O)Cc1nc(C)c(C)[nH]1)C2 6903,C1(NC(CN2CC(=O)N(C)C2=O)=O)CCCCCN(C(=O)C(F)C2CCC2)C1 6904,Cc1cc(N)c(C(=O)NC2CC(CNC(c3cn(C)c(O)n3)=O)C(O)C2)c(F)c1 6905,c1(C(N(CC(CC)NC(c2ncc(OC)cc2F)=O)C)=O)c(C)cc(C)nc1S 6906,N1(C(C2(C(C)NC(C(C)SCC)=O)CC2)=O)Cc2c[nH]nc2C1 6907,C12(NC(C3CCCCC3)=O)CCCC1N(Cc1cscn1)CC2 6908,c1(CC(=O)NCCCCC2CCCN(C(C(C)(C)O)=O)C2)cccc2nsnc12 6909,C1(CNC(C(C)(C)F)=O)CC2CN(C(c3cncc(C(F)(F)F)n3)=O)CC12 6910,N1(C(C(C2CCCC2)OC)=O)CCC(NC(=O)C(N)=O)C(C)(C)C1 6911,C1(NC(c2c(COC)ncs2)=O)CN(C(C2COCCN2C)=O)CCC1O 6912,C1(C2CC2)(NC(CCC(C)(C)F)=O)CCN(C(c2cc(Cl)cnc2O)=O)C1 6913,C1(CNC(c2n(C=C)ncc2)=O)CCN(C(c2ccc(F)cc2C)=O)CC1C 6914,N1(C(c2n(CC)ncc2)=O)CCOC(C)C1C(N1CC2(CO)CC2(CO)C1)=O 6915,C(CC(=O)NOC1CCOC1)(C(F)(F)F)NC(=O)CN1CC=CC1 6916,c1(NC(C2(C)N(C(CC)=O)CC2)=O)ccccc1S(=O)(=O)C(C)C 6917,N1(C(c2c(C)nn[nH]2)=O)CCN(C(c2ccc(Cl)s2)=O)C(C)C1C 6918,CC1CCN(C(=O)C(O)Cc2cn(C)cn2)C(CNC(c2cnccn2)=O)C1 6919,N1(Cc2ccc(C(C)C)cc2)CCN(C(C2CCC2)=O)CC1C1CC1 6920,CC1(C)CCC(NC(C2CC2CNC(=O)CC2CC3CCC2O3)=O)CC1 6921,C1(NC(C2OCCC(C)C2)=O)CN(C(C2CC3(CCO2)CC3)=O)C2(CCCC2)C1 6922,Cc1ccc(NC(=O)CCCCNC(c2ccccc2CC#N)=O)cc1O 6923,C(=O)(C(C)(C)COC)NCC(CC)NC(c1cccc(F)n1)=O 6924,C(=O)(CN=c1cc[nH]cc1)N(CCOCCC(=O)NC(C)CCn1cncn1)C 6925,Cc1cnc(O)c(NC(C2(O)CCN(Cc3ccc(Br)c(O)c3)C2)=O)c1 6926,N1(C(CCCC(C)c2cn(C(C)C(=O)O)nn2)=O)CCC2COC(=O)NC2C1 6927,C(=O)(CC1CCOc2ccccc21)N(C(CCNC(CCC(=O)NCC)=O)C)C 6928,c1(OC)cc(C(=O)NCC=CCC(=O)N(C)CCc2cnccn2)n(C)n1 6929,CC1CN(C(C2(CCNC(c3n[nH]c4c3COC4)=O)CC2)=O)CC(C)(C)O1 6930,N1(C(CCCCOCCC=C)=O)CCN(C(=O)CCC(C)SC)CC1CC(F)(F)F 6931,C1(CC(=O)NCCCN(C(C2(C)CC2Br)=O)CC)(CO)CCCC1 6932,C(=O)(C(O)C(C(C)C)OC)N1CC(CC)C(NC(c2cnn(C)c2C#N)=O)CC1 6933,C(C)(C(O)C(=O)N1CC2C(NC(C3(c4ccc(N(C)C)cc4)CC3)=O)C2C1)SC 6934,C1(F)(C(=O)NCCc2c(C(N(CC)CC3CCCO3)=O)c[nH]n2)CCOCC1 6935,Cn1cnc2c(C(N3CCN(C(C4CCC(=O)O4)=O)CC3CO)=O)[nH]nc2c1=O 6936,Cc1cccc(C(CN)NC(=O)NCC2(C3CCCO3)CCC2)c1 6937,CN(C1CCCc2ccc(F)cc21)CC1CCN(C(=O)CCc2nc[nH]n2)CC1 6938,S(=O)(=O)(c1cccc(F)c1)N1C(C(N2CCCN(C(=O)CO)CC2)=O)CC(O)C1 6939,CC1(C)CCN(C(c2c[nH]ccc2=O)=O)CC1CNC(C1CCC(F)CC1)=O 6940,C1(CN(C(=O)C(O)COC)CC)CCCN1C(c1cnn(C(F)F)c1)=O 6941,N1(C(CCOCCOCC)=O)CCC(N(C(=O)C=CC(F)(F)F)C)C1 6942,c1(-c2nc(C(C)C3CC3)nn2C2CCCOC2)ccnc(O)c1Br 6943,c1(OC)c(Cl)cc(NC(C2CC(O)CN2S(=O)(=O)c2cccnc2)=O)cc1Cl 6944,Cc1cnc2n1CCCC2C(=O)N1CCN(C(C2C=CC=CC=C2)=O)C(CO)C1 6945,CC(C)C(N=[N+]=[N-])C(=O)N1CCC(C)(NC(c2ncn3ccccc23)=O)C1 6946,C(C)(CNC(=O)C(C1CCCCCC1)C)(CC(C)C)NC(C=C=C(C)C)=O 6947,Cc1ccc(C(N2CC(F)(C(N3CCN4CCOCC4C3)=O)C2)=O)c([N+](=O)[O-])c1 6948,c1(C(C(=O)N(CCNC(c2csc(S)n2)=O)CC)C)c(C)n[nH]c1C 6949,N1(C(C(C2CCN(C(c3ccnc(O)c3)=O)CC2)C)=O)CCc2ncccc2C1 6950,C1(O)(CN(C(C(CC=C)C)=O)C)CCCN(C(c2cnc(C(C)(C)C)o2)=O)C1 6951,C(=O)(CCC(C)(F)F)NC(CC(=O)NC1(CO)C(C#C)C1)COCC 6952,CC(C)(C(=O)NCC=CC(=O)N(C1CC(C#N)C1)C1CC1)C1CCCC1 6953,c1(NC(C)CNC(=O)C(F)(F)c2cncs2)ncc(F)cn1 6954,Cc1[nH]nc(C(N2CCC(C)C2CNC(c2cc(CN(C)C)on2)=O)=O)c1N 6955,n1(CCCC(C)O)cc(C#CCNC(=O)CSC)nn1.C(C)(C)(C)OC(=O)NCC 6956,N1(C(c2ccc(C3C(C)C3)o2)=O)CCC(F)(CNC(=O)C(O)CC(N)=O)CC1 6957,C1(C(=O)NCc2ccc3nccn3c2)CN(Cc2ccc(O)nc2)CCC1(F)F 6958,CC1CC(F)(F)CN1C(C1(NC(=O)C(O)C2CCCC2)CCSC1)=O 6959,CC(C)C(F)(CNC(=O)C1=CCCC1C)C(=O)NC(CO)C(=O)N(C)C 6960,c1(OC)cc(N2CCC(NC(C3(C4CCOCC4)CC3)=O)C2)c(F)cc1[N+](=O)[O-] 6961,C1(C(=O)NCC2(OC)CCCCC2)CN(C)CCN1C(c1cc(C)n(C)c1C)=O 6962,C1(C(=O)NC2CN(C(COC)=O)C2)CC(C)(C(C)(C)C)C1.C1(CC)COC1.CO 6963,C1(NC(C(C(=O)OC)C)=O)CC(F)(F)CC1NC(c1conc1C)=O 6964,N1(C(c2ccc(C#C)cn2)=O)CC2(CCN(C(=O)C(C)(CC)CO)CC2)C1 6965,Cc1ccc(F)cc1CNC(=O)C(F)C1CC(NC(c2cc(=O)n(C)cn2)=O)C1 6966,O=C(CCC(=O)C1CCCC1)NC1CCOCC1NCC1CC1c1ccccc1 6967,N1(C(c2c(C)nns2)=O)CC(NC(c2ocnc2C2CCC2)=O)CC(O)C1 6968,Cc1cc(C(=O)NCC(=O)NC2COCCC2NC(=O)CC2CCCO2)n(C)n1 6969,c1(OC)c(C(=O)NC(C)CCCCNC(C2CCC(=O)O2)=O)cc(F)cc1F 6970,C1(C)(CNC(C(C)SCc2cccc(C)c2)=O)CN(C(=O)C(C)(F)F)CCO1 6971,Cc1c(F)ccc(F)c1CN1CCC(O)(CC(N2CCCOCC2)=O)CC1 6972,N1(Cc2onc(CC)n2)CCC(CO)(NC(C2CCCN2C(C)=O)=O)CC1 6973,Cc1c(Cl)ccnc1NNC(=O)CN1CCCCC1=O 6974,n1(CCC)nc(C)cc1C(=O)NC1CCC(CNC(=O)CCC=C(C)C)C1 6975,c1(CCC)c(C(N2CCC2CNC(c2nccnc2N)=O)=O)nnn1CC 6976,C1(CNC(C2C3(CCN(CC(=O)NCC#C)CC3)C2)=O)CCC2(CCCC2)CC1 6977,n1(CC(=O)N(CC(CN(C(=O)CC2C=CCCC2)C)O)C)ccc(Br)n1 6978,c1(C(N2CC(NC(CCN(C(C)=O)C)=O)C2)=O)cc(F)c(Br)cc1F 6979,C1(C(=O)NC(C2CCCC2)CC)CN(C(c2[nH]ccc2C2CC2)=O)CCN1C 6980,c1(CC(=O)NCC(C)N(C(=O)CC2CC(=O)NC2=O)C)c[nH]c2c(F)cccc12 6981,C1(N(C(c2cnc(C(C)C)s2)=O)C)CCN(C(C2CCC=CCC2)=O)CC1C 6982,C1(c2n(-c3c(SC)cccc3)nc(-c3cncnc3)n2)CC(=O)NC1(C)C 6983,c1(C2(NC(=O)NCC(F)C3CCC3)CCC2)ccccc1 6984,C1(CNC(C2C(C=C)C2)=O)CCN(C(=O)CNc2ccc(F)cc2Br)C1(C)C 6985,C(C(CC(=O)NCC(O)CNC(c1ccc2ccnn2c1)=O)C(F)F)N(C)C 6986,C1(C(N)=O)CCC(C(=O)NC2CC(F)(CNC(=O)CC3COCCO3)C2)CC1 6987,C1(NC(c2cc(C)cc(N)c2)=O)COC2C(NC(c3n[nH]c(CO)n3)=O)COC12 6988,c1(OC)cc(CN2CCN(C)CC2C(C)C)ccc1OC(F)F 6989,N1(C(=O)C2CC2)CC2(COC(CNC(C3(C(=O)OC(C)(C)C)CCOC3)=O)C2)C1 6990,C(=O)(C1=CCOCC1)N1CC(CC)C(C(=O)N(C2CCCCC2)CC)C1 6991,CC(CCP(C)(C)=O)(c1nnnn1CC1CCOC1)NCCC1CCC1 6992,N1(C(C(C=C)O)=O)CCCC(NC(=O)C(N2CCN(C)CC2)C)CCC1 6993,c1(CC(C(=O)O)NC(c2cc(C3CCCC3)no2)=O)ccc(Cl)nc1 6994,N(C(=NCC1(C)CCNC(=O)C1)N1CCN2C(CCS2(=O)=O)C1)C(COC)C 6995,C(C)(CN=c1[nH]ccc2cccc(C)c12)(CC(C)C)OCC 6996,C1(C(N)=O)CCCN1C(=O)CCC1CCN(C(C2CCCSC2)=O)C1 6997,C=C1CC2CCC(C1)N2C(=O)C(C(C)CC)NC(c1ncc(F)cc1F)=O 6998,c1(OC)cc(CN2CCOC(C(=O)NCc3ccn(C)n3)C2)ccc1C 6999,CC1CC(NC(c2ccccc2C(C)(C)C)=O)CN1C(=O)CC1(C)CC(F)(F)C1 7000,Nc1cnccc1C(=O)NC1CCNC(c2ccccc2)C1 7001,C1(CNC(CC(CC)OC)=O)CCC2(CCC2)CN1C(C1CC1C1CCC1)=O 7002,C1(C)(CC)CN(Cc2cn(CCC3CCCNC3)nn2)CCO1 7003,N1(C(C2N(CC)CCC2)=O)CCN(C(c2c(Cl)cnn2C)=O)CC1CC(=O)NC 7004,c1(C(N2CC(C)C2Nc2ncc(C(C)(C)O)cn2)=O)ccc2sccc2c1 7005,c1(CO)cc(NC)n(C)n1.N1(NC(CCc2ccc(C(=O)OC)s2)=O)C2CCC1CC2 7006,CC1(C)CN2CC1COC(=O)C1(c3cccc(c3)C2)CC1.S(C)(=O)(=O)NC 7007,C(=O)(C(C1=NOCC1)N1CCN(C2CCOCC2)CC1)NCCCOC 7008,N1(C(C(=O)NC2CC3(CC(OC)C3)C2)=O)CC2(CCC2)CC1CO 7009,Cc1cnoc1N.C1(CC(=O)N(CCC(C)C)CC(C)C)CCN(CC(C)C)C1 7010,N1(C(c2c(C)nns2)=O)CCC(CNC(c2cnc(O)c(F)c2)=O)C(O)C1 7011,C12(NC(C(C)CN(C)C)=O)CCOC(CNC(c3ncccc3C3CC3)=O)(C1)C2 7012,c1(C(N2CCC(CN(C(C(CC)N(C)C)=O)C)CC2)=O)cc(F)c(Cl)cc1F 7013,c1(NC(C2CC2NC(CNC(CN2CCN(C)CC2)=O)=O)=O)c(F)cccc1F 7014,c1(CNC(c2c(NC(CC(=O)OC)=O)ccs2)=O)ccc2c(c1)COC2 7015,c1(CNC(CCSC)=O)ccccc1N1CCN(C(C2NC(=O)CC2C)=O)CC1 7016,N1(C(CN2CCC(C)(O)C2)=O)CCN(C(=O)C(C)(C)O)CC12CCC2 7017,c1(C(N2C(C(=O)NC3(CO)CC(O)C3)CC(=O)C2)=O)cccc(F)c1O 7018,C(CNC(C1C2COCC12)=O)(CC(F)(F)F)NC(c1c(SCC)nccn1)=O 7019,C(=O)(C(C)CS(C)(=O)=O)N1CCC(NC(c2sc(CC)c(C)c2)=O)C1 7020,CC(C)(C(=O)NCCCCNC(C1(c2ccc(Cl)nc2)CC1)=O)C(F)(F)F 7021,N1(C(CSCCCC)=O)CCOCC(F)(CNC(=O)C=Cc2cnc[nH]2)C1 7022,CCC(C)(CNC(=O)CC1CN(C(=O)C(C)(C)C2CC2)CCO1)CC 7023,S(=O)(=O)(c1ccc(C(C)(C)C)cc1)NCC(=O)Nc1cc(C)c(F)cc1 7024,C1(C)(C(N(CCCCN(C(c2ccc(SC)o2)=O)C)C)=O)CC=CCO1 7025,C1(CNC(c2cnc(C3CC3)s2)=O)CCCN(c2cc(-c3ccccc3)ncn2)C1 7026,N1(C(CC(C)OC)=O)CCC2(CC1)CN(Cc1ccc(Cl)cc1C)CCO2 7027,c1(C2(CCNC(=O)CC)CC2)ccccc1Cl.C1(C)C(=O)N1.C1(CC)CN(CCO)C1 7028,C1(NC(C2CCCS2)=O)CCSC12CN(C(=O)CCc1nc3ncccn3n1)C2 7029,CC#CCCCC(=O)NCC1C=CCN1C(c1ccc(CC)c(N)c1)=O 7030,c1(N(C)Cc2cccc(OC)c2)nc(N2CCC(S(C)(=O)=O)C2)c2c(n1)COC2 7031,Cc1cc(=NCc2csc(C)c2)[nH]c(N2CCS(=O)C(C)(C)C2)n1 7032,n1(CC#C)cc(CNC(C2CC(NC(=O)CC3(N(C)C)CC3)CCO2)=O)cn1 7033,c1(CN(C(C)C)C(=O)Nc2cccnc2Oc2ccccc2)cc(Br)ccc1O 7034,Cc1onc(C(=O)NC2CC2CNC(=O)CSc2ccccc2)c1Br 7035,C1(CNC(C2CC(=C)C2)=O)COC(C)(C)CN1C(=O)Cn1cnnc1O 7036,c1(OC)cc(C(F)F)c(C(N2CC(C)(NC(=O)C=CC(C)(C)SC)C2)=O)cn1 7037,C(=O)(CC(CC)C(F)F)NCCC(C(N1CCC(C#C)CC1)=O)(C)C 7038,Cc1oc(C)c(C(=O)NC(C2CCN(C(=O)C(c3cccc(O)c3)C)C2)C)c1C 7039,C1(C(=O)NC2CC(N(C(CSCCCC)=O)C)C2)CCc2nc(O)[nH]c2C1 7040,c1(OCC(=O)NCC2(NC(c3csc(CO)n3)=O)CCOC2)cccnc1.C1CC1 7041,Cc1nn(C)c(C)c1OCC(=O)NC1CC(CO)N(C(=O)CC2(C(F)F)CC2)C1 7042,C1(NC(c2cc(C(N)=O)[nH]c2)=O)(CO)CCCN(C(C2CCCCO2)=O)C1 7043,C1(CNC(c2ncc(CC)cn2)=O)CN(C(c2c(C)nsc2C)=O)CCC1(F)F 7044,c1(CN2C(C(N3CCC(F)(F)C3)=O)CSCC2)cnc(Cl)cc1Cl 7045,C1(C(=O)NCC(n2cc(CCN3CCC(O)CC3)nn2)C)CCCC2NCCC12 7046,C1(CNC(C(c2n(C)ncc2)(F)F)=O)CN(C(c2ccsn2)=O)CCO1 7047,Cc1cnncc1C(=O)NCC(C)(C)CN(C(=O)COCC(=O)N(C)C)C 7048,N1(C(C(CC)=CC)=O)CCOC(C(C)NC(c2ccc(Cl)cn2)=O)C1 7049,c1(CNC(=O)NC(CC(=O)OC)C2CCCCC2)nccc(C(F)(F)F)n1 7050,N1(CC)CC(C(=O)N(C)CCC2CCCCN2C(=O)CCSC)CC1=O 7051,C(=O)(CC(C(=O)NC1(C)CN(C(c2scnc2C(C)C)=O)C1)N(C)C)OC 7052,C1(C(N2CCC(NC(C=NOC)=O)C2(C)C)=O)CCc2nccn2C1 7053,N1(C(CC(CC)C)=O)CCC2OCCN(C(c3cc([N+](=O)[O-])cnc3N)=O)C2C1 7054,C#Cc1ccc(C(N2CCC(c3n[nH]c(CNC(=O)C(O)C(C)C)n3)C2)=O)nc1 7055,C(=O)(C1CCc2c[nH]nc21)N1CC(C(C(=O)NCCc2cnccc2Cl)OC)C1 7056,C1(C(N(CCC(=O)N(c2ccsc2)CC)CC#C)=O)CCCSC1C 7057,CN1CCC(CC(=O)N(C2CC3CNC2C3)Cc2cnco2)CC1 7058,C1(C(=O)NC2C(NC(c3ncc(OCC)nc3)=O)CCCC2)CC2(C1)CC21CC1 7059,C1(NC(c2cnc(CC)s2)=O)CCN(C(=O)COCCCN(C)C)CC1F 7060,Cc1cc(C)c(C(N2CC3CC(NC(=O)CC4C=CS(=O)(=O)C4)C2C3)=O)cn1 7061,C1(=CC(=O)NCC(CNC(c2nccc(Cl)c2F)=O)OC)CCCCC1(C)C 7062,CCC(C)(CNC(=O)CSCC(N)=O)NC(=O)C(C)(C)c1cc[nH]n1 7063,c1(OC)cc(CC(N2CCN(CCNC(C3(O)CCCC3)=O)CC2)=O)ccc1C 7064,N1(C(CC(CC)(O)c2ccccc2)=O)CC2CN(C(=O)C(F)=CC3CC3)CC2C1 7065,c1(C(=O)NC2CN(C(c3cc(C)cc(O)n3)=O)CC2C)[nH]cc2c1CCCC2 7066,C1(C(N(CC(C(=O)NC2CCC(C#C)C2)(C)C)C)=O)CC2COCC2C1 7067,c1(CNC(C(CC)C)(C)c2nnnn2CCC2(C)CC2)cn2c(C)cccc2n1 7068,C(=O)(C(F)(F)C(F)(F)F)NC(CNC(CCc1ccnc(C)n1)=O)C 7069,c1(CC)[nH]c(=N)sc1C(=O)NC1CC(CNC(c2c[nH]cc2Br)=O)CC1O 7070,N1(C(C2C3CN(C(CC4(NC(C)=O)CC4)=O)C2C3)=O)CCCCCCC1C 7071,N1(C(C(C(C)OC)N(C)C)=O)CC(C)(C)CC1C(=O)NCC(C)(CO)CO 7072,c1(CN(C)CC2CN(C(c3cn(CC)nc3)=O)C2)c(F)ccc(OC)c1Br 7073,O(NC(=O)C(c1cccs1)NC(c1coc(CO)c1)=O)CCCC#C 7074,C(C)(C)(CC(=O)NCC(Cl)C(C)(F)F)N(C(CN1CCC(C)C1)=O)C 7075,N1(C(c2nc(OC)oc2)=O)CCC2(CCCN2C(C2(O)CCC(C)(C)CC2)=O)C1 7076,c1(NC(c2nccs2)C)nccc(N2CCC(N3CCOCC3=O)CC2)n1 7077,N1(C(C(C2CCN(C(c3cnc(C#N)s3)=O)C2)C)=O)CCOC(C2CCC2)C1 7078,c1(C(C(N2CCC(NC(C(C)OC(C)(C)C)=O)C2)=O)(C)C)cc(Cl)cc(Cl)c1 7079,C(C(CC(C)C)C(=O)NC(CNC(c1cscc1C)=O)C1CC1)OC 7080,c1(C(N(C)CCNC(C2CCC2C(C)(C)C)=O)=O)cc2sc(Cl)cc2s1 7081,N1(C(c2n(C)ncc2Cl)=O)CCC(NC(=O)Cc2c(O)ncnc2O)CC(O)C1 7082,CCC(O)C(C)(C)C(=O)NC1CCCC(CC(=O)NCC(O)(COC)CO)C1 7083,N1(C(CCSCC)=O)CCCOC(CCNC(=O)Cn2ccc(C)n2)C1 7084,Cc1c(C(C)NC(C2(c3ccccc3)CCOC2)C)cnn1-c1ccccc1 7085,CCCC(C)C(=O)NC(C1CN(C(C23CC(CO2)C3)=O)C1)C 7086,c1(OCC)cc(NCC2CC2NC(c2cn3cccnc3n2)=O)ccc1[N+](=O)[O-] 7087,CCC(C)(C)CCCC(=O)NC1CC1NC(c1c(C)ccc(F)c1O)=O 7088,c1(C(N2CC(C)(CC)OCC2)C(=O)Nc2ccccc2)noc2ccccc12 7089,N1(C(CCOCCC)=O)CCC2CCCC12C(=O)NC(CO)C(C)(C)CO 7090,C1(C(=O)NCC2N(C(C3(C)N(C(C)=O)CCC3)=O)CC2)CC(S(C)(=O)=O)C1 7091,S(=O)(=O)(c1ccn(CCF)n1)N(C)Cc1c(F)cc(F)cc1F 7092,O=C(N=c1ccn(CCC(=O)N2CCCC2)[nH]1)c1ccnc(F)c1 7093,C1(C(=O)NCCN(C(=O)CC(=O)NCC(F)(F)F)C)CC2CCC1O2 7094,n1(CC(=O)N(C(CNC(CC2(OC)CCC2)=O)C)C)cnc(C(N)=O)n1 7095,C1(CNC(C=CC=CCC)=O)CCCN1C(=O)C(F)(F)c1cnn(C)c1 7096,c1(C(N(C2CCN(C(C3CCC(=O)C3)=O)C2)CC)=O)cnn2cccc(Cl)c12 7097,c1(CC(N2CCC(F)(CNC(C(CCC#C)O)=O)C2)=O)ccc([N+](=O)[O-])cc1F 7098,c1(-c2cccc(C(C)O)c2)ncc(Cl)cc1C(=O)Nc1cccnc1C(F)(F)F 7099,C1(C)(C(=O)NC2CCN(CCCC)C2)CCN(C(=O)OCc2ccccc2)C1 7100,CC(C)CC(C)C(=O)N1CCC(N(C)C(C2CC3C=CC2CC3)=O)CC1 7101,C(=O)(CC(=O)NC(C)C(=O)NCCc1cscn1)OC 7102,Cc1nn2c(C(=O)NC3CN(C(c4cc[nH]c4)=O)CC(C)(C)C3)c(C)nc2s1 7103,c1(C(N2C(C)CCN(C(c3cnc(OC)s3)=O)CC2)=O)cc2c(nn1)CCCO2 7104,N1(c2n(CC(C)C)c(Cc3cscc3Br)nn2)CC2C(C1)C2(F)F 7105,N1(C(C2(C#C)CC2)=O)CCC2CCN(C(C3CC4(C3)CC4F)=O)CC2C1 7106,C(C1=NOC(C)C1)NC(C(Cc1ccoc1)NC(CC(C)SC)=O)=O 7107,CCCCCC(O)CC(=O)NC(C1CCN(C(=O)C(C#N)CC)C1)C 7108,c1(C(C(=O)NCCSC)NC(=O)CN(C)C)cncn1C 7109,c1(C(=O)NC(CN(C(=O)CCc2cncn2C)CC)C)cc(N)cc(F)c1 7110,C1(NC(C2CC3(COCCO3)C2)=O)CC2CC1C1CNCC21 7111,c1(CNC(C(C)Cn2cccn2)=O)cccc(NC(=O)OCC(F)(F)C(F)F)n1 7112,C1(Nc2cc(N3CCCC(CN(C)C)C3)ncn2)CC2CC1CC2(C)O 7113,C12CCN(C(=O)C(OC)CCOC1=O)O2.N1(CCC)CCOCC1 7114,c1(CC)ncc(C(=O)NCC2(CN(C)C(c3ccc(SC)s3)=O)CC2)s1 7115,C1(C(N2CCN(C(CSCC)=O)CC2CC(F)(F)F)=O)Cc2cc(C)ccc2S1 7116,C1(CNC(C(C)Cc2ccco2)=O)CN(C(c2ccc(F)s2)=O)CCO1 7117,C(c1ccco1)=CC(N1CCC1C(N1CCCC1C(O)CO)=O)=O 7118,c1(C(=O)NCC(CNC(c2c(C(C)C)nns2)=O)F)cccn(C2CC2)c1=O 7119,C(=O)(CC(CNC(C1C(C)(C)C1(F)F)=O)C1CCC1)N1CC(COC)C1 7120,c1(CNC(C(C2CC(NC(C3(C)CC3(F)F)=O)C2)F)=O)ccccc1O 7121,N1(C(c2c(C)onc2)=O)CC(F)CC1CNC(=O)C(c1ccc(Br)cc1)O 7122,Cc1nn(C)cc1NC(=O)CNC(=O)NC(c1ccccc1C(C)C)C 7123,Cc1c(C(=O)NC2CCC2CNC(=O)C=CC=CCO)cc(C(C)(C)C)n1C 7124,C(C(C)(C(=O)N(CCCCC(=O)NC1CC1c1ccsc1)C)OC)OC 7125,N1(CC(=O)N(CC(C)CNC(c2ccc(NCCO)cc2)=O)C)CCCS1(=O)=O 7126,C=CC(CC)CC(=O)NC1CCCN(C(=O)Cc2csc(C3CC3)n2)C1 7127,C1(CC=C)(C(=O)NC(c2cncnc2)C)CCCN1C(=O)Cn1cc(C#N)cn1 7128,c1(C(N2CCCN(C(C(C)(C)OC)=O)CC2)=O)ccc2c(c1)C(=O)NCC2 7129,c1(OCC)ccc(Cl)nc1C(N1CC2C(C1)N2C(=O)COC)=O 7130,N1(C(C(C)C2CCC2)=O)CC2CC1CN(C(=O)CC1CSC1)C2 7131,c1(C(=O)NC2(C)CCN(C(CC(C)C3CC3)=O)C2)ccc2c(c1)CCCCC2=O 7132,c1(C(N2CCC(F)(F)CC(C)C2)C(=O)NCCCOC)cccc2cnn(C)c12 7133,C1(C(=O)Nc2ccc(C)nc2)CCN(C(=O)C=CC2CC2)C12CC2 7134,c1(CC(=O)NCc2csc(C(N3CC4CC4C3)=O)n2)cccnc1F 7135,c12cccc(C(=O)O)c1N2.N1(C(=O)OC(C)(C)C)CCCC(C(F)(F)F)(CO)C1 7136,C(=O)(C1=COCCO1)N(CCNC(c1cncc(OCC)c1)=O)CC1CC1 7137,c1(C(N(c2nccc(OCC)n2)CC2CCCN2)=O)ccc(F)nc1C 7138,CCCC(O)C(=O)N1CC(NC(c2csc(Br)n2)=O)C(O)C1 7139,CCC(CC)(CO)C(=O)NCC(CC(F)(F)F)NC(C1CCCCC1C(N)=O)=O 7140,C1(NC(C2(OCC)CCOC2)=O)CCCCC1CNC(=O)CCC1CCOCC1 7141,c1(-c2cn(CC3N(C(C(CCC)N(C)C)=O)CCC3)nn2)ccc([N+](=O)[O-])o1 7142,CC(CN=c1[nH]cnc(Cl)c1Br)N(C)C(c1cnc2[nH]cncc1-2)=O 7143,N1(c2n(CCCOCC)c(-c3occc3C)nn2)CCCC2(CCCO2)C1 7144,N1(C(C2CCCC(NC(Cn3c(C)ccn3)=O)CC2)=O)CCC2CCN(C)CC12 7145,CCCCC(CN=c1ccc(C(F)(F)F)n[nH]1)NC(C1(CCOC)CC1)=O 7146,C12(C(=O)NCCCC(C)(C)C)CCC(CN(C(c3cc(=N)[nH][nH]3)=O)C1)C2 7147,N1(C(c2scc(Cc3c(C)ncs3)c2)=O)CCCC1(C)c1cn(CCON)nn1 7148,N1(C(c2nc(C)c(C)s2)=O)CCCCC12CC(NC(C1CC1C(F)F)=O)C2 7149,c1(C(N2C(C(=O)NCCCS(C)(=O)=O)CC(O)C2)=O)cc(F)c(Cl)c(C#N)c1Cl 7150,C1(CC)CN(C(=O)C=CC(=O)N(C)C)CCC1NC(=O)C(=O)NCC1CC1 7151,c1(-c2cccn(C)c2=O)nc2ccc(C(=O)NC(C3(C)CCOCC3)=O)cc2s1 7152,c1(C(N2CC(CNC(C(CSC)O)=O)C(F)(F)C2)=O)cc(C)c(Cl)c(C)c1 7153,c1(OCCC)cccnc1C(=O)N(CCCCN(C)C(c1cccs1)=O)C 7154,C#Cc1ccc(CC(=O)NC2(C(=O)N(C3CC4CC4C3)C)CC(CO)C2)cc1 7155,C#Cc1cnc(C(=O)NC(C2CCOC2)CNC(C2(CC)CC2)=O)c(C)c1 7156,N1(C(C2N(C(C)=O)CCOC2)=O)CCCC(O)(CNC(c2ccnc(O)c2)=O)C1 7157,C1(CNC(C(=Cc2ccco2)C)=O)CCN(C(=O)CCC2CC2(Cl)Cl)CC1 7158,c1(CCNC(C(=O)N(C(COC)C)C)=O)ccc(OC)cc1.c1ncccc1F 7159,CCCCC(CNC(c1c(C)noc1C)=O)NC(c1cc(C(C)(C)C)n[nH]1)=O 7160,c1(CCC(=O)NCC2C3CN(C(C(=C(C)C4CC4)F)=O)CC32)cccc(Cl)c1Cl 7161,N1(C(c2c[nH]nc2C)C(=O)NCc2c(OC)cccc2)CCc2cc(Br)ccc21 7162,N1(C(CN(C2CC2)CC)=O)C2CCC1CC(C(=O)Nc1c(F)cccc1F)C2 7163,Cc1nn(C(C)C)c(C)c1CC(=O)NC(C)CNC(c1cc(C(F)(F)F)no1)=O 7164,Nc1cccc(Cl)c1C(N1CCCC(N(C(=O)C#CC2CC2)CCF)C1)=O 7165,c1(C(=O)NC2(C)CCN(C(c3cncs3)=O)C2)cc([N+](=O)[O-])ccc1N 7166,N1(C(C(C(C)C)C2CCC2)=O)CCC(NC(=O)CCC2(C)CC2(F)F)C12CC2 7167,n1(CC(N2CC(C(N(CC(COC)O)C)=O)(SC)C2)=O)cccnc1=O 7168,C(=O)(C(C#N)C(C)(C)C)NC(CCC(=O)NC1CC(OCC)C1)C 7169,C(C(C)N=c1[nH]c2c(c(=NCC=CCl)[nH]1)COC2)Oc1cc(C)oc1C 7170,n1(C2CN(C(C(c3ccc(Cl)s3)C)=O)C2)cc(-c2ncccn2)nn1 7171,CCCCS(=O)(=O)N1CCCCC1C(=O)NCCCCc1cn(CC(=O)O)nn1 7172,CCC(C)(CO)C(=O)N1CCC(CN(C)C(c2cccc(C3CCCC3)c2)=O)C1 7173,C1(CC)(CN(C(C2CCCN(C)C2)=O)C)CCN(C(=O)C(F)C(C)C)C1 7174,c1(NC(C2C(NCC(CC)CC(=O)OC)C3CCC2C3)=O)ccn2ncnc2c1 7175,C1(C(N(C2C(C)C2)C)=O)CCCCN(C(C2CCC2)=O)C1 7176,C1(C)(NC(C2C(C)CN(C)C2)=O)CCC(NC(C2C3CC4C(C3=O)C24)=O)CC1 7177,CCCCC(C)(F)C(=O)NC1CCC(C(=O)NCC(C)N(C)C)C1 7178,C1(NC(=O)CCC2(NC(c3cc[nH]n3)=O)CCC2)CC12CCCC2 7179,n1(CCC2CC(NC(CN(C)CC)=O)C2)cc(C2CCCO2)nn1 7180,c1(C(=O)NCC(CCCC)NC(c2c(C)cnn2C)=O)nnc(Cl)cc1N 7181,C1(NC(C(c2cnccn2)C)=O)COCCC1NC(c1ccc(C(N)=O)[nH]1)=O 7182,c1(SC)ccc(C)c(C(=O)NCC2COCCN(C(=O)Cc3cc(C)ns3)C2)c1 7183,c1(C(N)=O)ccnc(C(N2CC(OCCNC(=O)C(O)C3CC3)C2)=O)c1 7184,N1(C(C(C=CC)O)=O)CCCC(C2(NC(c3cc(=O)n(C)cn3)=O)CC2)C1 7185,N1(C(C2CCN2C(C2(n3cccn3)CC2)=O)=O)CCC(CO)C(O)C1 7186,C(C(=O)N1CCC(OC2CCOC2)CC1)(C(C)C)c1cnc(C)s1 7187,C(C(C)(CC)OC)N(C(C(C)N(C(=O)CCc1nccs1)CCC)=O)C 7188,c1(OC)cc(NNC(=O)OC(c2c(C)n[nH]c2C)C)ncn1 7189,C1(CNC(N2CCC(c3ncn(C)n3)CC2)=O)CCc2nc(O)[nH]c2C1 7190,C(=O)(C1=CC(C)(C)C1)N1CCC(N(C(C(C)NC(=O)NC)=O)CCO)CC1 7191,c1(C(=O)NC2CCCOC2)cn(CC2(C(N(CCO)CC)=O)CC2)nn1 7192,c1(CN2CCN(c3ncc(-c4cccc(SC)c4)cn3)CC2)c(Cl)ccnc1Br 7193,N1(C(C2CN(C(C(C=C=C)C)=O)CC23CC3)=O)CCc2ccccc2C1 7194,C1(C(=O)NCCCCOC)CN(C)CCN1C(=O)C(C)CC(C)C 7195,CC1(C)COC(CC(N2CC=CC2CNC(=O)C(F)(F)CO)=O)CO1 7196,c1(CNC(C2CC(CNC(=O)CN3CC=CC3)C2)=O)ncc(F)cn1 7197,Cc1cc(CC(=O)NCc2cc(C(=O)NC(C)CC(C)O)cs2)on1 7198,c1(CNC(C(C)N(C(C2CCN(CC)CC2)=O)C2CC2)=O)cc(C)nc(O)c1 7199,C1(c2n(CCC)nnn2)(Nc2ccc(F)c(F)c2C)CCCN2CCSCC12 7200,C1(C(=O)NCCCN(C(C2C(=C)C2)=O)C2CC2)CCc2nc[nH]c2C1 7201,C1(CNC(CNC(CC(C)(C)C)=O)=O)CN(C(C2CCNC(=O)C2)=O)CCCO1 7202,N1(C(C2C(=C)CC2)=O)CCC(C(C)(C)CNC(=O)Cc2cccnc2OC)CC1 7203,c12cccc(c1)CN2.c1(S)nc(C(=O)NCC)cs1.C(N)(=O)N 7204,N1(CC(=O)NC(C)(C)CN2CCOCC2)CCOC(Cc2ccc(C)cn2)CC1 7205,C(=O)(CC(C)CCC=C(C)C)NC1C2CN(C(C3(COCC)CC3)=O)CC21 7206,C1(CNC(c2n(C)nc(C(F)(F)F)c2)=O)CC2CCC1N2C(=O)CN1CCC1C 7207,N1(C(CC2C(C)CCN(C(C3(F)CCC3)=O)C2)=O)CCn2ncc(O)c2C1 7208,C1(C(N(CCC)CCC)=O)CC12CCN(C(=O)C(C)n1ccnn1)CC2 7209,Cc1ccc(CNCC2CCN(C(C3CNC(=O)N3C)=O)C2)cn1 7210,c1(C(C(=O)NCC=C)N(CC)Cc2ccc(C)c(C)c2)csc2ccc(C)cc12 7211,C1(NC(C(C)n2ccnc2)=O)CN(C(=O)COC2(C)CCOCC2)CC1C1CC1 7212,N1(C(CCSCCCC)=O)CC(C2CCN(C(c3c(O)cccc3F)=O)CC2)C1 7213,c1(CNC(=O)Cc2cccc(F)c2)ccnc(OC2CCOC2)c1 7214,C1(NC(c2ccc(C)nn2)=O)CN(C(C2CCCCS2(=O)=O)=O)CC1(C)C 7215,N1(C(C(C)=CC)=O)CC(NC(c2c(C)noc2CC)=O)CC12CCCCC2 7216,C1(C)(C(N(CC(C)(C)NC(=O)CSC(C)(C)C)C)=O)CC(C#N)C1 7217,c1(C(=O)NC2C(CNC(=O)CCCCC(F)F)CCC2)cnc2cccnc2c1 7218,N1(C(C(CCSC)(C)C)=O)CCC2CCN(C(=O)Cc3ncc(C)o3)CC2C1 7219,CC1CCCCC1C(=O)NC(C1CN(C(c2cncnc2)=O)CCO1)C 7220,N1(C(c2n(C)nnc2)=O)CCC(=CCNC(=O)CC2CCCSC2)CC1 7221,N1(C(C(C)CNC(=O)CCCN(C)C)=O)CCCC(O)CC1 7222,c1(C(=O)NC2(CC=C)CCN(C(=O)CCNC(=O)CO)C2)cc2ccncc2s1 7223,Cc1ccc2ncccc2c1NC(C1CCN1C(c1cccc(CBr)c1O)=O)=O 7224,C1(NC(C2CN(CC(C)C)C(=O)C2)=O)CCN(c2nnco2)C(C)C1 7225,C1(CNC(c2c(C)coc2)=O)CCN(C(=O)CSCC(F)(F)F)CC1C 7226,N1(C(c2c(OC)cc(C)cc2C)=O)CC2OCCN(C(=O)C(C)NC=O)C2C1 7227,N1(C(CC(CC)C)=O)CCN(C(c2ccc(-c3ncccn3)cc2)=O)C(C#N)C1 7228,C1(C(=O)NCCN(C(c2c(N)ccc(CCC)c2)=O)C)CC2CC(O)CC(C1)C2 7229,CC#CCC(C)NC(=O)C(C)(C1CCC1)NC(=O)CNC(N)=O 7230,c1(OC)cccc2c(C(N3CC(NC(c4cnc(O)s4)=O)CC(C)C3)=O)csc12 7231,C1(NC(c2c(C)nc[nH]2)=O)CC(CNC(c2nc(Br)c[nH]2)=O)C1(C)C 7232,c1(SCC)cnc(O)c(C(=O)NCCC(C)N(C(=O)C(C)N(C)C)C)c1 7233,C=C(C)CC(C(=O)N1CCCC1C(N1CCC(n2cnnn2)C1)=O)OC 7234,C1(C(N2C(CCCNC(C=NOC)=O)CCCC2)=O)CCC=CCCC1 7235,C(=O)(C(C)(O)CC(F)(F)F)NC(c1ccc(Br)cn1)C 7236,C12(C(N3CCC(C(N4CCC(c5cn(C)nc5)CC4)=O)C3)=O)CC=CCN1CCC2 7237,O=C(NN1CCCCC1)N(CC(F)(F)F)CC1CC1.C12CCCCN1C2=O 7238,c1(OC)nc(N2CC(C(C)NC(c3snnc3C(C)C)=O)C2)cc(C)n1 7239,N1(C(c2c(C)c(C#N)[nH]c2)=O)CCOC2CN(C(=O)CC(C)C(C)(C)C)CC12 7240,C1(NC(C2(C)CC2)=O)CN(C(c2ccc(Cl)c3occc23)=O)Cc2ccnn2C1 7241,c1(CC)nc(C)c(CNC(=O)C(c2ccccc2)NC(=O)CC2CCCC3CC23)o1 7242,c1(C(=O)NC2C(NC(CNS(CC)(=O)=O)=O)COC2)oc2cc(Cl)ccc2c1C 7243,c1(OC)ccc2c(=NCCC#N)[nH]c(NC3CN4CCC3CC4)nc2c1 7244,CC1CC(NC(c2ccnc(C3CC3)n2)=O)CN1C(c1cnn(C)c1Br)=O 7245,CC1(C)CCCOC1CNC(=O)CC12CCC1CN(C(=O)CC(Cl)Cl)C2 7246,c1(C(N(C2CCN(C(=O)NCCNC(=O)C(C)(C)C)C2)CC)=O)cnc(C)s1.OC 7247,C1(C(=O)NC2CCCN(C(c3cn(C)nn3)=O)CC2)CCC2(CC1)COCCO2 7248,c1(C(=O)NCC#CCNC(CC(C)O)=O)cc(Br)ccc1Cl 7249,Cc1ccc(C)c(C(=O)NCC23CC(NC(c4ccnnc4)=O)(CO2)C3)c1 7250,c1(C(N2CC(C)N(C(=O)CCc3cc(Cl)no3)CC2)=O)cccc2oc(=N)[nH]c12 7251,N1(CC)CC2CN(C(=O)C=CCC3(NC(C4CC(=O)OC4(C)C)=O)CCC3)CC2C1 7252,c1(C(N2CC(NC(C(c3ccccc3F)(C)OC)=O)C2)=O)cnc(C(F)F)nc1 7253,C(CO)(C(C)(C)CO)NC(CCNC(C1(C)CC1(F)F)=O)=O 7254,C1(CN(CC(CC)OC)C)CCCN1C1CCC(c2ccccc2)C1 7255,c1cc(-c2noc(-c3cc(C4COCCO4)ccn3)n2)c2c(c1)CCCC2 7256,N1(C(C2CCC(CC)CC2)=O)CCCN(C(=O)CC23CCCC2C3)C(C)C1 7257,c1(N2Cc3c(C)cnn3CC2)nc(=NCC2CCO2)[nH]c2c1CCCCCC2 7258,C1(NC(C2C(C(=O)OC)C2)=O)CCC(NC(=O)Cc2ccccc2C)CC1 7259,C(C(=O)NC1CC2CCC1(NC(C1CCCCC1)=O)C2)(C(C)(C)C)NC(C)=O 7260,C(=O)(C(CCO)N(C)C)NCCC(=C)CNC(c1sc(C)nc1CC(C)C)=O 7261,C=CC1(NC(C2CC2NC(=O)COCC(=C)C)=O)CCCCC1 7262,c1(CNC(CCN(C(=O)C=Cc2ccccc2)CC)=O)cc2ccccc2[nH]1 7263,C(=O)(C1CCCc2scnc21)NC1CCN(C(C2(CN(C)C)CC2)=O)CC1F 7264,C(=O)(C1=C(C)OCCS1)NC(COCC)C(=O)Nc1ccc(C)c(CC)c1 7265,C1(NC(C(C(C)C)OC)=O)CN(C(=O)CCc2ccc(F)nc2)CCC1C 7266,C1(Nc2onc(OC)c2Br)CCN(C(=O)CCCNC(=O)C(C)(C)C)CC1O 7267,c1(OC)ccc2[nH]c(C(N3CC4CC4(CNC(=O)C(C)CF)C3)=O)cc2n1 7268,NS(=O)(=O)c1cc(C(=O)NCC2CCC(NC(=O)Cc3ccco3)C2)co1 7269,C1(C2(O)CCN(C(C3COCCN3C)=O)CC2)(NC(C(C)SC)=O)CC1 7270,C=CC1(CC(=O)NCCC(C)NC(=O)C(O)Cc2ccccc2)CCCCC1 7271,CC(C)(C)C(CC(=O)N1CC(NC(c2ccc3c(c2)nnn3C)=O)C1)C(F)F 7272,c1(C(=O)NC(C)CC2CN(C(c3cnccc3Cl)=O)C2)cc2cncn2c(O)n1 7273,Nc1cc(CC(N2CCCOC(CNC(=O)CCC(F)F)C2)=O)ccc1[N+](=O)[O-] 7274,N(C(=NCCN1CCOCC1)NCC1CN(C)CCN1C)CC(C)OC 7275,C1(C(NOCC#C)=O)(COC)C=CCN1C(=O)C(C)C1CC1 7276,C(C(C)(C)C(=O)NCC1(F)CCC(NC(C2CCCC(=O)N2)=O)C1)N(C)C 7277,C1(N(C(=O)CNC(N)=O)C)CN(C(c2cscc2C2CC2)=O)CC12CC2 7278,C1(NC(C2(C#N)CC2)=O)(CF)CCN(C(=O)Cc2ccccn2)C1 7279,C#CCC(C)(C)C(=O)NCCOC1CCN(C(=O)CC2CCOC(CC)C2)C1 7280,S(=O)(=O)(c1cc(C(=O)OC)c(C)c(Br)c1)NC(CCOC)Cc1cccnc1 7281,Cc1cccc2[nH]cc(C(N3CCC(C)(CNC(C45COCC4C5)=O)CC3)=O)c12 7282,N1(C(C2CC(C)N2C(c2ccn(C)n2)=O)=O)CCc2cnccc2C1 7283,C1(COCC(=O)N(C)C2CC2)CCCN(C(C2(c3cccnc3)CCCC2)=O)C1 7284,Cc1ccc(-c2c[nH]nc2C(=O)Nc2ncc(CCO)s2)cc1C 7285,C(=O)(C(=O)N=c1ccc(C#N)c[nH]1)OCC(C)OCCN 7286,c1(C(N(CCN(C)C(=O)OC(C)(C)C)C)=O)cnn(CC2CC2)c1 7287,C(=O)(CS(=O)CCC(F)(F)F)NCC1(NC(c2cc(C#N)oc2)=O)CCCC1 7288,c1(C(C(=O)NCCCSCC)N(CCCCC)C)cn(CC)nc1C.CC 7289,c1(CNC(CCN(CC#C)C(C2CC2(Cl)Cl)=O)=O)ccc(NC)nc1 7290,S(=O)(=O)(c1cnc(NC(c2nccnc2C)C)c(Cl)c1)NCC=CCCC 7291,N1(C(CN(C(c2cnn(C(C)C)n2)=O)CC)=O)CC(C)C(F)(F)C1 7292,C(=O)(C(C)C(F)(F)F)NCCCCCNC(C(c1cccc(C)c1)F)=O 7293,C1(NC(C(c2cccnc2)OC)=O)COC2(C1)CN(C(c1csnn1)=O)C2 7294,n1(CC#C)c(C(=O)NCCNC(c2cc([N+](=O)[O-])c[nH]2)=O)cc2ccccc12 7295,Cc1ccc(C)c(CN(C)C(C2CCCN2C(=O)C(O)CC(C)C)=O)c1 7296,Cc1cc(C)c(C(=O)NC(C2CCCC2)CNC(=O)CC2CCC(C)C2)c(C)c1 7297,Cc1cccc(Br)c1S(=O)(=O)N(CCC[Si](C)(C)C)C 7298,C1(C(=O)NC2(C)CN(C(CCN(C)CC)=O)C2)CCc2ncnn2C1 7299,N1(C(CSCC)=O)CCN(C(=O)CC2C(=O)NN=C2C)C(CS(C)(=O)=O)C1 7300,O=S(=O)(c1ccc(NC2C=CCCCC2)c(Cl)c1)NCC(CC1CC1)CO 7301,C1(CNC(CCN(C(C)=O)C)=O)CN(C(c2coc(Cl)n2)=O)C2CCN1C2 7302,Cc1cc(NC(=O)C(C2CCN(C(=O)CC3CCCC3O)C2)C)cc(O)c1 7303,C(=O)(C(O)CC(F)(F)F)N1C(CCNC(Cn2ncc(C)c2)=O)CCCC1 7304,N1(C(c2c(C)nc(Br)o2)=O)CCN(C(C2CCCCCC2)=O)C2(CC2)C1 7305,N1(C(C2N(C)CCCC2)=O)CCN(C(c2cccnc2F)=O)CC1C(F)(F)F 7306,C12(NC(c3nnnn3CCOCc3ccccc3)CC3(C)CC3)CC1CS(=O)(=O)C2 7307,C1(=CCNC(c2ncsc2C2CC2)=O)CCN(C(C2C(CC)(COC)C2)=O)CC1 7308,C=CC(C)(CC)C(=O)NC(c1ccccc1F)CNC(=O)C=Cc1cnc[nH]1 7309,c1(C(=O)NCC(C(C)(C)C)NC(CN(C)CCO)=O)ncc(Cl)cc1Cl 7310,c1(C(=O)NC2COCC2C(N2CC3CC2C3)=O)ccc2cc[nH]c2c1 7311,N1(C(C(C)(C)OC)=O)CC(CNC(c2cc(-c3ccccn3)c[nH]2)=O)C(C)(C)C1 7312,C(C)(C(F)(F)C(F)(F)F)NC(CCCCOC(C)(C)C)=O 7313,CC1CCC(C)N(C(=O)CC2CN(C(=O)COC3CCC3)CCO2)C1 7314,C12(NC(=O)OC(C)(C)C)CCCN(Cc3c[nH]c(-c4ccccc4)c3)CC1C2 7315,Cc1cc(N)c(C(N2CC3=C(C2)CN(C(C2(C)CC(=O)N(C)C2)=O)C3)=O)cc1C 7316,C1(=CCNC(C(C)(C)N2CCCCC2)=O)CCN(C(=O)CSC(F)F)CC1 7317,N1(C(C2(OC)CCOC2)=O)CCCC(C)(NC(=O)Cc2csc(C3CC3)n2)C1 7318,C1(C(=O)NC(C(=O)NCCNC(C(C)(C)C)=O)CC2CCCC2)CC12CCCC2 7319,N1(C(c2cc(OC)n(C)n2)=O)CC2(COC(CNC(c3ccc(SC)o3)=O)C2)C1 7320,Cc1nccn1CC(=O)NC1(CNC(c2cc(-c3ccn(C)n3)on2)=O)CCC1 7321,N1(C(C2CCCC(O)C2O)=O)CCC(C2CCCC2)C1 7322,C(=O)(C1=Cc2ccccc2C1)NCC1C(C)CN(C(=O)CCP(C)(C)=O)C1 7323,O=C1CCC(CC(N2CCCC(CCNC(c3cc(=O)cc[nH]3)=O)C2)=O)CN1 7324,c1(CC)ncccc1C(=O)NCCN(C(=O)CC12COCC(C1)C2)C1CC1 7325,C1(CNC(=O)CCc2ccoc2)CCN(C(=O)C(F)(F)CO)CCC1(F)F 7326,Cn1cnc2c(C(C(=O)NC3CC3)NCC3CCN(C4CC4)CC3)cccc12 7327,C1(C(N2CC(O)(C(C)NC(=O)Cc3cncc(O)c3)C2)=O)CC2(CCCO2)C1 7328,C(=O)(C1CCCn2cnnc21)NCC1(CN(C)C(c2cn(CCO)nn2)=O)CC1 7329,CC1(C)CCC(C(=O)NC2CCC(NC(=O)C=CC=C(Cl)Cl)CC2)CO1 7330,C(CC#CC)(C(=O)NC1CCCSC1)NC(CC1CC(=C)C1)=O 7331,c1(C(N(CC(C)NC(C2(NC(C)=O)CC2)=O)CC)=O)ccc2c(c1)CCS2(=O)=O 7332,c1(NC(Cc2scc(C)n2)=O)ncnc2c1c(Br)cn2C 7333,N1(C(C2CC(C)OC2=O)=O)C2CCCC1CN(C(=O)C=CC1CCC1)C2 7334,c1(COC)cc(C(=O)N(C(C)CN(C(=O)CCCC2CCCO2)C)C)ccc1F 7335,O=S1(=O)CCCC(n2nc(-c3ccccc3)nc2-c2ccc(OC(F)F)nc2)C1 7336,C(=O)(C1=C(Cl)CCOC1)NCC(CC)(C)NC(c1cccc2sncc12)=O 7337,c1(OC)ccc2c(c1)NCCN(Cc1ccccc1OC1CC1)C2 7338,N(C1CCCc2cc(F)ccc21)C(Cc1ccc(C(=O)O)nc1)=O 7339,CC1(C)C2CC(NCC3CCCN(S(=O)(=O)C(F)(F)F)C3)C3(CC3)C1C2 7340,N1(C(C2C(CNC(Cn3c(=N)nc[nH]3)=O)CC2)=O)CC2CCCC2C12CC2 7341,N1(C(C(CC)OC)=O)CCN(C(C2(C#N)CC2(C)C)=O)CC1C 7342,c1(C(=O)NC2C3OCC(C(N4C(C)(CCO)CC4)=O)(C3)C2)cccc2occc12 7343,C1(C(=O)NCC2C(NC(c3n(C=C)nnc3)=O)CCC2)SC2C=CC1CC2 7344,Cc1ccc2ncc(C#N)c(N3CCN(C4CC4)C(C)C3)c2c1 7345,CCS(=O)c1ccccc1C(=O)NC1CN(C(c2cnoc2C)=O)CC1C1CC1 7346,C1(C(C)C)CN(C(=O)CO)CCN1C(=O)CO[Si](C)(C)C 7347,CCCCC(C)CCC(=O)NOCC(=O)NC1CCN(C(=O)CC)C1 7348,c1(C(=O)NCCC(C)NC(C(CC)CC2CCCC2)=O)cc(OC)cc(C)c1 7349,N1(C(C2C(C)CCOC2)=O)CCC(CNC(=O)CCCC(N)=O)C(O)C1 7350,c1(CNC(C2(c3ccccc3)CC2C(F)(F)F)=O)cnc2ccccn12 7351,C=CC(C)(C)CC(=O)N1CCCC1C1CCCN(C(=O)CCN(CC)CC)C1 7352,c1(CC)c[nH]cc1C(N1CCCC1C(C)(C)CNC(=O)C=CC1CCOC1)=O 7353,c1(CC(N2C(CCCNC(C3CCCCCC3)=O)CCC2)=O)ccc(O)nc1 7354,N1(C(C(c2ccccc2)OC)=O)CC2CN(C(c3ccc(C#N)cn3)=O)CC2C1 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7391,c1(C(N2C(C(C)(C)NC(C(COCC)C)=O)CCC2)=O)nc2ncc(C)cn2n1 7392,Cc1c(-n2cc(C3CCN(C(=O)CC(C)C4CCCCC4)C3)nn2)cccc1F 7393,c1(OCC(N)=O)cccc(C(=O)NC2CCC(NC(=O)CSC3CC3)C2)c1 7394,C1(C(=O)OCC)CCCCC1Nc1ccccc1NC(=S)NC1CCN(C)C1=O 7395,Cc1ccc(N)cc1C(N1CCCC(F)(CNC(=O)CNC(=O)CC(C)C)C1)=O 7396,CCC(CC(C)C)C(=O)NC1(C)CC(C(=O)NC(C2CCCCC2)CO)C1 7397,CC1COc2ccccc2CN1C(=O)C(F)Oc1ccccc1 7398,C1(NC(CC(C)c2ccncc2)=O)(CO)CCN(C(C2(CF)CCC2)=O)C1 7399,C(=O)(C(F)C(=O)N1CCC(NC(=O)CC=C(C)C)C1C(C)(C)C)OCC 7400,c1(NC(C(C(C)C)SC)=O)ccc(C(=O)NC2CCCC2)cc1F 7401,c1(N(C(C2CC2c2ccc(Cl)cc2)=O)CC2CCC2)ccccc1Cl 7402,C(=O)(CCC(F)(F)F)NC1C(C)CN(C(=O)CCc2nnc(S)n2C)C1 7403,C(C(=O)N(C)Cc1cnc(C)s1)(C(C)CC)N(C(c1cccc(CC)n1)=O)C 7404,n1(CC)nc(C)c(CN2CCSCC2C(=O)NCc2cc(C)cnc2Cl)c1C 7405,C(=O)(C1CCCc2nc[nH]c21)N(CC(C)N(C(c1nc(OC)c(F)cn1)=O)C)C 7406,C1(C2CCCN(C(c3scnc3C(F)(F)F)=O)C2)(NC(C(CSC)OC)=O)CC1 7407,Cc1cc(C(=O)NCC(O)CNC(C2(S(N)(=O)=O)CCCC2)=O)ccc1[N+](=O)[O-] 7408,C1(CNC(c2cc(OC)n[nH]2)=O)CC(O)C(O)CC1C(=O)NC(CO)C(C)C 7409,N1(C(C2(OC)CCC2)=O)CC2(COC(CNC(=O)CC3CCCC34CC4)C2)C1 7410,C(CCC(C(=O)N(C)C)N1CCN(C(C(=O)OC)C(C)O)CC1)OCC=C 7411,c1(C(=O)NCC2(OC)CN(C(c3ccnn3CC3CCC3)=O)C2)cnnc(C)c1 7412,c1(C(=O)NC(C2CCOC2)CNC(CSCCC)=O)sc(C)cc1Cl 7413,C1(CCC)CN(C(c2oc(C)cc2C)=O)CC1NC(C1(CO)CCOCC1)=O 7414,N1(C(C=C)=O)CC2(COC(CNC(c3cc(CO)n(C)n3)=O)C2)C1 7415,c1(C(=O)NC2C(CNC(C=COCC)=O)COC2)ccc(F)cc1Cl 7416,C(CCC(C)C(=O)N1CC(O)CC(F)C1)OC 7417,CC1CN(C(C2CCCN(C)C2)=O)CC(C)C1N=c1nc[nH]n2c(Br)ccc12 7418,c1(C(=O)NCC(C)(CNC(=O)C(C)CC#N)OC)c(C)nc(O)nc1C 7419,C1(C)(CNC(c2c(CC)non2)=O)CCCN1C(=O)CCc1cccs1 7420,Cc1ccc(C(=O)NC2CCCC(C(=O)NC(=O)CN3CCOCC3)C2)c(F)c1 7421,C(=O)(CCP(C)(C)=O)N1CCC(NC(Cc2n[nH]c(=NC)s2)=O)(CO)C1 7422,C1(CNC(C2C(C)CCC2)=O)CCC2(CCN(C(=O)C#CC(C)(C)C)CC2)CO1 7423,C1(CNC(CC#N)=O)CC2(CC(NC(c3ccccc3C(F)(F)F)=O)C2)C1 7424,Cc1nnccc1C(=O)NC1COCC1CNC(=O)CCc1cnn(C)c1 7425,n1(CC)nnnc1C(c1cnn(CCCl)c1)NC(C1(OC(C)C)CC1)=O 7426,N1(C(c2ccc(OC)cc2)=O)CCOC2(C1)CN(S(=O)(=O)CC1CCC1)C2 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7462,CC1CCC(C(=O)N(C2CC3CC3C2)C)N(C(=O)Cc2ccon2)C1 7463,N1(C(C(C)(C)OCC)=O)CCC(C)(CNC(=O)CC(c2cccc(F)c2)C)CC1 7464,C1(F)(C(N(C)Cc2cnco2)=O)CN(C(=O)CC2CC(F)(F)C2)C1 7465,CC1(C)CN(C(c2coc(C(F)F)n2)=O)CCC1NC(=O)CNC(=O)C1CC1 7466,C1(C(=O)NCC(C)(CO)NC(c2c(C)n(C(C)C)cc2)=O)CCCCC(C)(C)C1 7467,c1(CC)cccnc1C(=O)NC(C)(CNC(=O)CCC1C(=O)NN=C1C)C1CC1 7468,N1(C(c2cc(CNC(C3CC(C)C3)=O)oc2)=O)CC2CCCC2C1 7469,CP(C)(=O)C1(C(N2CC(O)(C3CCCN3C(=O)CC3CCC3)C2)=O)CC1 7470,CC(C)(C)CC(F)C(=O)N1CCC(F)(c2cn(CC3CC4CC4C3)nn2)C1 7471,c1(OC(C)C(=O)NCC2CC(C)N(C(=O)CC(O)C3CC3)C2)ccc(F)nc1 7472,CC1(C)CCC(C(=O)NC2CC(C(F)C(=O)NCCN(C(C)C)C3CC3)C2)C1 7473,N1(c2nnc(COC)s2)CC2CC1CCC2NC(C1(O)CCSCC1)=O 7474,C1(CNC(C2C(OC)CCC2)=O)(CNC(c2ocnc2C)=O)CCCCC1 7475,C12(NC(C3C(CC)C3(F)F)=O)COC(C1)C(NC(c1cnn(C)n1)=O)C2 7476,c1(C(=O)NC2C(C)CN(C)C2)cnc2nc(C#N)ccn12 7477,CC1CN(C(=O)C(=O)NCc2cn(CC3CCCO3)nn2)CC1(C)CO 7478,N1(C(C2CC(=C)C2)=O)CCCC(C2CN(C(c3cc(O)n(C)n3)=O)C2)C1 7479,c1(C(N2CC(C(C)OC(C(=O)OC)OCC)C2)=O)ccc(C(=O)CC)cc1 7480,Cc1n[nH]c(C)c1C(=O)N(C)CC1(O)CN(C(=O)C(C)(C)C2CCOC2)C1 7481,CCC(C)(C)CNC(C1CC(CNC(c2cccnn2)=O)C1)=O 7482,C1(NCC(C)CC2CCC(F)(F)CC2)CCc2c(nnn2C)C1 7483,C(=O)(C1=CC2CCCC12)N(CC(CNC(c1cccc(SC)n1)=O)C)C 7484,Cc1nc(C(=O)NC2CC(NC(=O)C(C)(C)Br)CC2O)c2ccccn12 7485,CC1C2C(CCN2C(C2CCc3n[nH]cc3C2)=O)CN1C(=O)CC1CC(F)(F)C1 7486,Cc1cc(C(=O)N(C2CN(C(C34CCC(C)(C3)OC4)=O)C2)C)cc(N)c1O 7487,N1(C(COCc2ncc(C)o2)=O)CCCC(C(N(c2ncncc2Cl)CO)=O)C1 7488,CC(C)C(C)(F)CNC(=O)CNC(=O)CNC(c1nc(Cl)cs1)=O 7489,c1(CN2C(C)(C(=O)Nc3cc(OC)ncc3)CC2)c(C)cc(O)cc1O 7490,CCC(CC)C(C(=O)NCC1(CNC(c2cnnn2CC)=O)CCOCC1)OC 7491,c1(CC)[nH]nc(C(=O)N(CCC(N2CCC(CC3CC3)CC2)=O)CC)c1C 7492,C1(CCC(=O)NCC(C)NC(C=C(C)Cc2cccc(Cl)c2)=O)CCCN(C)C1 7493,c1(N(C)C)cc(F)ccc1NC(=O)C(C)(C)NC(C1C2CC(=O)CC12)=O 7494,C12(CNCc3cnc(C)[nH]3)CN(C(=O)OC(C)(C)C)CC(F)(C1)C2 7495,N1(C(=O)NC(c2cncn2C)C)CCCCC1C1OCCO1 7496,C1(NC(C2(OCC)CCC2)=O)CCN(C(c2ccc(O)c(Cl)c2)=O)C(C)C1 7497,c1(C(N(CCC(C)NC(=O)Cc2cnn(C)c2)C)=O)ccc2nccnc2c1 7498,c1(C(N2CC3C(NC(CN(C)CC)=O)C(CC3)C2)=O)cc2c(cn1)OCCC2 7499,CC1=C(C(=O)NC2CN(C(c3ccc(C)nc3)=O)CCC2C(F)(F)F)CCO1 7500,C(=O)(C1CCc2c[nH]nc21)N1CCC(CC(=O)NCCC(C(=O)OC)(C)C)CC1 7501,C#CC1(C(=O)Nc2cnc(C3CC3)nc2)CCN(C(=O)CC=C(C)C)C1 7502,C1(C(=O)NC(c2n(CC)ccn2)C)COCCN(C(=O)CCc2ccnn2C)C1 7503,N1(C(CCOCC(C)C)=O)CCOCC(C(=O)Nc2cc(C(N)=O)cc(F)c2)C1 7504,c1(CC)c(C(=O)NCC2CCC(NC(c3cc[nH]n3)=O)CC2)[nH]c(C)c1C(N)=O 7505,C(=O)(CCCC1CCC1)NCCCOCCC(=O)NCC(c1cncnc1)C 7506,N1(C(CNS(CC)(=O)=O)=O)CCC(C2CC2NC(C2CC=CCC2)=O)CC1 7507,C1(C(=O)NC2C(NC(=O)CCc3ccnc(Cl)c3)C2)CN2CCCCC2CO1 7508,C12(C(=O)NCC(CNC(c3ccc(N)c(O)c3)=O)O)CCCCC(=O)N1CCC2 7509,CCC(C)(CCNC(=O)CC1CC=CCN1C)NC(=O)CSC 7510,Cc1ccccc1C1(C(=O)NCC=CCNC(=O)C(F)n2ccnc2)CCC1 7511,N1(C(COCc2ccc(C)cc2)=O)CCC2CC(NC(=O)C=CCF)CCC2C1 7512,N1(C(CSCC)=O)CCC2(CC1)OCCC2NC(=O)CSCC(=O)OC 7513,C(CNC(C1CC12CCCC2)=O)(CC(=O)N1CCOC(C)C1)OC 7514,C1(NC(CCc2ccc(C#C)cc2)=O)CCC(O)CN(C(=O)COCCOC)C1 7515,N1(C(C(=O)NC(C)CN(C)Cc2ccc(C3CCCO3)nn2)C)C(C)CCC1C 7516,C1(CN(C(CCC=C(C)C)=O)C)C2CN(C(c3nocc3C3CC3)=O)CC12 7517,N1(C(C(CCC#C)O)=O)CCCC2(CCN(C(C3(S(C)(=O)=O)CC(O)C3)=O)C2)C1 7518,N1(C(=O)OC(C)(C)C)CCC(C2CC(CC(=O)N=c3cco[nH]3)C2)C1 7519,c1(CN2C(CNC(c3nc(C(C)C)oc3)=O)CC2)c(F)cccc1Cl 7520,N1(C(C2N(C(C(CC)(C)C)=O)C(C)C2)=O)CCC12CCCSC2 7521,Cc1cc(Cl)cc([N+](=O)[O-])c1C(=O)NC(C)CCNC(c1c[nH]nc1[N+](=O)[O-])=O 7522,CCCC(C)(CCC)C(=O)NC1CN(CC(=O)OC(C)(C)C)CC(C)(C)O1 7523,C1(CCCC)CCCCC1C(=O)NC1CN(C(=O)CCC(=O)OC(C)(C)C)C1 7524,C1(NC(c2c(SC)csc2)=O)CC2(C1)CC(NC(c1coc(C3CC3)n1)=O)C2 7525,O=C(CC1=CCCCC1)N1CC2CCCC1(CNC(C1(O)CCSCC1)=O)C2 7526,Cc1ccc(CO)cc1-c1cn(C2CCN(C(c3coc(C4CC4)c3)=O)C2)nn1 7527,C(CC1CC1)(C(=O)NC(C)C(=O)NCc1coc(C)n1)OC 7528,c1(OC)c(C(=O)NC2CC(O)CN(C(C3CCN(C)CC3)=O)C2)cc(F)cc1F 7529,c1(CC(=O)NCC(C2(O)CCN(C(c3c[nH]nc3F)=O)C2)C)c[nH]ccc1=O 7530,C(C1c2ccsc2CCN1C(=O)Cc1ccc(I)cc1Br)OC 7531,C(=O)(C(CC(F)F)NC(C1CCCC(=O)C1)=O)NCC1(CO)CC(C)C1 7532,N1(C(c2n(C(C)C)ncc2)=O)CC2CCCC2(NC(=O)C(=O)NCC(F)(F)F)C1 7533,N1(C(C2CCCN(C(C)=O)C2)=O)CCCN(C(C2CCN2C)=O)CC1C 7534,C1(N(C(Cc2nnc(C)s2)=O)Cc2ccccc2)CCCN(C(C2CC2F)=O)C1 7535,N1(C(C(CC)(C)O)=O)CC2CS(=O)(=O)CC2(CNC(c2cccnc2NC)=O)C1 7536,C1(C(=O)NCC(C(C)C)NC(=O)CC(C)(C)N(C)C)CCCC(F)C1 7537,c1(C(=O)NC2CN(C(C=CC(CC)C)=O)C3(C2)CCC3)ccc2c(c1O)CCC2 7538,N1(C(=O)CCc2nncs2)CCC(NC(C2(CC3CCC3)CC2)=O)C12CCC2 7539,C12(C(=O)NC3CCC(NC(=O)C4=CSCCO4)CC3)CCCC1CS(=O)(=O)C2 7540,C1(CNC(=O)NC2CCOC2)CCCN1C(c1cc(-c2ccccc2)[nH]n1)=O 7541,C1(CNC(c2n(CC)cnc2C#N)c2nnnn2C2CC2)CCCC(C)(C)CC1 7542,N1(C(CC(COC)C)=O)CC(C)OC2(CCN(C(C3(CO)CCCCC3)=O)C2)C1 7543,c1(C(=O)NC2C3(CN(C(C(C)(C)O)=O)C3)CC2)cnc(O)n(C2CC2)c1=O 7544,C(CC(C(C)(C)C)NC(=O)CC1CC=CCC1)N(C)C(c1sccc1C1CC1)=O 7545,Cc1ccc(Cl)cc1C(C(=O)NCc1nnn(C)n1)N(C(C)CS(C)(=O)=O)C 7546,C1(C(N(CC(C)N(C(C)=O)C)C)=O)CCN(C(=O)C(C)Cn2ccnc2)C1 7547,N1(C(CC2CCC(NC(c3c(C)occ3)=O)CC2)=O)CC2C(C1)C2(F)F 7548,C1(NC(c2cc(C(=O)OC)ncc2)=O)CN(C(C2CC(C)=NO2)=O)CC(C)(C)C1 7549,c1(CSc2n(CC)c(CCc3ccco3)nn2)ccc(Cl)cc1F 7550,N1(C(c2c(NCC)cccn2)=O)CC(NC(C2CC2C(F)F)=O)CC2(CCC2)C1 7551,c1(C(=O)NCC2CCCC(CNC(C(C)N3CCC3)=O)C2)noc2c1CCCC2 7552,N1(C(C(c2cccs2)SC)=O)CCCC(C)(C)C1CNC(C1CC(CF)C1)=O 7553,N1(C(C(n2cc(Cn3c(C)ccc3C)nn2)C)=O)CCOC(C2CC2)CC1 7554,C(=O)(C(C)(C)S(C)(=O)=O)NCCCC(C)NC(=O)CCCOc1ccccc1F 7555,C(C(=O)NC1CC1CN(C(=O)CNC=O)CC1CC1)(C(C)C)OCCOC.OC 7556,N1(C(C(C(C)C)OCC)=O)CCC2(CCC(NC(=O)C3=CCC3)CC2)CC1 7557,CCC(C(=O)NC1CC(C(=O)N2CCC(O)(CO)CC2)=CC1O)C(F)(F)F 7558,Cc1nn(C)c(NC2CC(C)CC(C)C2)c1C#N 7559,N1(C(c2ccc(COC)o2)=O)CC(CC(=O)NCCN(C)C(C)C)CC1(C)C 7560,N1(C(c2ccc(Cl)s2)=O)CCN(C(=O)C=CC2CCCO2)C(CF)C1 7561,CCC(C)(CN(C)N1CC(O)CC1Cc1ccccc1)OC 7562,c1(C(=O)NCC2CN(C(CS(CC)(=O)=O)=O)CC23CC3)cnc2c(C)cnn2c1 7563,C1(CC=O)(NC)CCOCC1.CC1CCN(C(=O)C(C2CCN(C(C)(C)C)C2)F)C1 7564,C12(NC(CN3CCC(C)CC3)=O)CCCC1CN(C(C1(C)CCCNC1=O)=O)C2 7565,C1(NC(CCSCCC)=O)C=CC(C(=O)NC(C)Cc2cnccn2)C1 7566,C1(NC(C2(C)ON=C(C)C2)=O)CN(C(=O)CC2(O)CCCC2)CC1(C)C 7567,Cc1ccc2c(c1)C(C(=O)NCC(F)CNC(c1ncccc1CO)=O)OCC2 7568,N1(C(CSCCC)=O)CCCC1C(C)NC(=O)C(C)OC1CCOC1 7569,CC1CCC(NC(=O)C(O)C2CCC2)CN1C(=O)CCCC1CC1 7570,N1(C(c2ccc(SC)o2)=O)CC(NC(=O)CCc2ccc(O)nn2)C(C)(C)C1 7571,C1(C#N)(C(=O)NCCC(C)N(C)C(c2cc(-c3cccs3)on2)=O)CCSCC1 7572,N1(C(Cn2ncn(C)c2=O)=O)CCC2CC1CN(C(=O)CCC1CC1(C)C)C2 7573,C1(NC(CN(C(=O)C(CSC)OC)CCC)=O)CCN(CCOC)C1 7574,c1(N(CCC)C)ccc(CN2CC(CC(=O)O)C(O)C2)cc1 7575,c1(N2CCN(C(c3c(C)noc3C)C(=O)NCC(C)C)CC2)ccc(C#N)nc1 7576,N1(C(C2(CC)CCCC2)=O)CCN(C(=O)COCCSC)C(C2CC2)C1 7577,c1(SCC(=O)NCCC(C)N(C)C(C2COC3(CCC3)C2)=O)ccsc1[N+](=O)[O-] 7578,S(=O)(=O)(c1cnn2ccc(=NCc3csnn3)[nH]c12)N1C(CCC)CCC1 7579,C12(CNC(CNS(N)(=O)=O)=O)CCCC1N(C(=O)CC1CCNC(=O)C1)CC2 7580,N1(C(CC=C)=O)CC(NC(c2cccc(-c3cscn3)c2)=O)C2(CCC2)C1 7581,c1(C(=O)NC2CCN(C(CCC#CC)=O)CCC2CO)cc2c(Cl)ccnc2s1 7582,C12(c3cn(CC)nn3)COC(C1)C(O)C2.N1(C(CC2CC(C)C2)=O)CCCC1C1CC1 7583,C1(O)(C(C(=O)NCC2C(C(C)C)C2)F)CN(C(C2CCOC2=O)=O)C1 7584,C1(C(=O)NCC2CN(C(c3ncc(C)nc3)=O)C2)CC(C)CC(C)(C)C1 7585,n1(CCC(N2C(CNC(=O)CC3CSC3)CCC2)=O)ncc2c1CCCC2 7586,C(=O)(C(C)S(C)(=O)=O)NCC=CCNC(C1CCN(c2cc(C)ncn2)CC1)=O 7587,C1(S(C)(=O)=O)(C(=O)NC2C(CNC(c3[nH]cc(CC)c3)=O)C2)CCCC1 7588,C12(CNC(CCCSC)=O)CC(NC(=O)CC3CSCCS3)(CO1)C2 7589,c1(C(=O)NCCN(C(=O)C(C2CCCCCC2)O)CC)cc(C)cc(Cl)n1 7590,N1(CC)N=C(C(=O)N2CCCC(C)C2CNC(=O)CSC2CC2)CCC1=O 7591,C1(CC(=O)NC2CCC(N(C(C(CC)N(C)C)=O)C)CC2)C(=O)N(C)N=C1C 7592,N(C(=NC1CCS(=O)(=O)C1)N1CCC2(CC1)CC(O)c1nn(C)cc1O2)C(C)C 7593,N1(C(c2cnc(C)nc2)=O)CC(NC(=O)C=Cc2cc[nH]c2)C2(CC2)C1 7594,N1(c2ncc(C)c(I)c2)CCCc2sccc2C1 7595,c1(C(N2CC(COC)(CNC(=O)C(C)C3CCC3)C2)=O)cccc(CO)c1 7596,c1(C(=O)NCC2CCC(NC(c3c(C)cc(Br)cn3)=O)C2)cc2ccncc2[nH]1 7597,CCC(C(=O)NC1CCN(C(=O)Cc2cc[nH]c2)C12CCC2)C(F)(F)F 7598,N1(C(CC=C=C)=O)CCC2CN(C(=O)CN3C(=O)CC(C)(C)C3=O)C2C1 7599,C(=O)(C(CNC(=O)CC(O)C1CCCC1)C(C)(C)C)NCCC=CCCC 7600,C(=O)(C1=CCCN(C(=O)CC(F)(F)F)C1)N(CC(N)=O)C 7601,Cc1ccc(C(c2nnnn2C2CCC2)NCCCn2cncn2)cc1C 7602,CCN=c1[nH]c(CNC(=O)N(C2CC(O)C2(C)C)CC)cs1 7603,Cc1cccc(C(=O)NC2CC(NC(C3(NC4(F)CC4)CC3)=O)C(O)C2)c1 7604,N1(C(c2ccnc(C)n2)=O)CC2CC(NC(c3ccc(C)c(F)n3)=O)C2C1 7605,C(=O)(C(CC)CC(F)F)NC1(CN(C(c2cc(CC)c(F)cc2)=O)C)CC1 7606,Cc1cc(C(=O)NC2CC(NC(C3(Br)CC3)=O)C2)[nH]c1C 7607,N1(Cc2ccn(C)n2)CCC(CO)(NC(c2nnc(O)nc2O)=O)CC1 7608,C1(C(N2C(CNC(=O)CC3(O)CC3)COCC2)=O)CCOC2(CCCC2)C1 7609,n1(CC(=O)NC(C2(CNC(C3OCCCO3)=O)CC2)C)cnc(Br)n1 7610,CC1(C)CCC(CCC(N)=O)OC1.C12CN(C(C)(C)C1)C(=O)C(=O)N1CCC21 7611,N1(C(C(n2cc(C)nc2)(C)C)=O)CCC2(CCC2)C(NC(C2CCS2(=O)=O)=O)C1 7612,N1(C(C2(CC=C)CC=CC2)=O)CC2CC(NC(c3c[nH]nc3CCC)=O)C2C1 7613,c1(C(=O)NCCn2cc(CNS(CC)(=O)=O)nn2)cc[nH]c(=N)n1 7614,CC1C(C)N(C(=O)CCCSC(C)(C)C)CCN1C(C1C2CCC1CC2)=O 7615,c1(C(N2CCCC(CNC(c3ncn(CC)n3)=O)C2)=O)cnc2cc[nH]c2c1 7616,C1(C(=O)NC2C(C)N(C(=O)CC3CCN(C)CC3)CC2)CCC=CCCC1 7617,C(=O)(C(C(C)(C)C)c1ccccc1)N1CC(NC(CCCSC)=O)C(C)C1 7618,Cc1nc(N2CC(NC(=O)CCC(C)(C)[N+](=O)[O-])C(C)C2)c(Cl)cc1C#N 7619,c1(C(=O)NCC(C)(CNC(C2C=CCCC2)=O)OC)cn(C)nc1C(C)C 7620,CC1C(NC(=O)CCc2cn[nH]c2)CCN1C(=O)CN1CCOCC1=O 7621,C(C1CCOCC1)=CC(=O)NCCC1CS(=O)(=O)C1 7622,CCCC(O)CCNC(=O)CSCCNC(=O)CCCOC(C)C 7623,Cn1ccc(=O)c(C(N2CCC(O)(CNC(=O)C(F)n3ccnc3)CC2)=O)c1 7624,C1(NC(C(=O)NC(CC)CC2CC2)=O)COC2(CCC2)C1 7625,N1(C(C2CCCN(C)C2)C(=O)NC2CC(F)(F)C2)CCc2cccc(F)c2C1 7626,C1(C(C)C(=O)NCCn2cnnn2)CCCN(C(C2SCCS2)=O)C1 7627,c1(C(=O)OC)cc2c(cc1NCCc1ccc(C)cc1Cl)CN(C(=O)OC)CC2 7628,c1(OC)cc(Br)cc(CN2CCCC2(C)C(=O)Nc2cnc3cc[nH]c3c2)c1O 7629,C=C(Cl)CC(C(=O)NCC(C)(C)C1CC1)NC(C1CC(=O)OC1(C)C)=O 7630,c1(CC)noc(C(N2CCSCC2CCNC(c2cnc(C)nc2)=O)=O)c1C 7631,N1(C(C2SCCN(C(c3c(C)ccc(OC)c3)=O)C2)=O)CCC2(CC1)CC2(F)F 7632,c1(C(N2CCNCC2c2ccccn2)=O)cnc2c(Br)n[nH]c2c1C 7633,c1(N2CCCC(CNC(CCOCC#C)=O)C2)cc(-c2ccco2)nc(C)n1 7634,Cn1cnc(I)c1CN1CCCC1(C)C1CCCCC1 7635,C(=O)(CC(F)(F)C(F)(F)F)NC1CCCN(C(C(CCC)c2ccccc2)=O)C1C 7636,C1(NC(C(CC)Cc2ccccc2)=O)C(C)CCN(c2cncc(Cl)n2)C1C 7637,c1(CC(N2CC(NC(c3ccc(Cl)nc3Cl)=O)C(F)C2)=O)cc(F)c(F)cc1Br 7638,N1(C(C)=O)CC(CC(=O)NC(C(=O)NCC(C)(C)SCC#N)C2CCOC2)C1 7639,C1(NC(Cc2cccc(OCC)c2)=O)CCSC12CN(C(=O)C(O)C(F)(F)F)C2 7640,c1(NC(CN(C2CC(C#N)C2)C(C2C(C(C)C)OCC2)=O)=O)ccc(F)c(CO)c1 7641,n1(CC(=O)OCC)nc(-c2cccc(F)c2)nc1-c1c[nH]c(=O)cn1 7642,c1(C(=O)NCC=CCNC(C2C(C=C(C)C)C2(C)C)=O)cc(N)c(Cl)c(O)c1 7643,c1(CC)cn2cccnc2n1.C12(CCC(=O)NC1=O)c1ccc(cc1)NC(=O)C2 7644,C(CC(=O)NCC1CC(NC(=O)C(C)n2ccnc2)C1)OCCCOC 7645,CC1(C)CCC(C(=O)NCCC2CCCN2C(c2cc(O)cs2)=O)C1 7646,c1(OC)ccc(C(=O)NCC(O)CNC(C2(C)CC3CC3C2)=O)cc1N 7647,Cc1ccc(C(N2CC3(C2)CN(C(=O)C(=O)N(C)C)CC3CO)=O)c(N=[N+]=[N-])c1 7648,c1(OC)cncc(C(=O)N(C(C)CNC(=O)CC2CCC(=O)O2)C)c1C 7649,Cc1c(C(N2CCCN(c3ccccc3)CCC2)=O)nn2ccccc12 7650,CCCCCC(F)C(=O)N1CCC(C)C1C(=O)NCCc1nc[nH]n1 7651,c1(N(CCC)C)ccc(C(N2CC(CC(C)NC(=O)CCC(C)C)C2)=O)cc1 7652,C1(NC(CC(=C)C)=O)CCC2(CC1)CN(C(=O)C1=COCCC1)CCO2 7653,c1(C(=O)NC2C3CN(C(C(CCC)OC)=O)C2CC3)sc(=NCC)[nH]c1C 7654,c1(C(=O)NCC23CC(CN2c2ncnc(Cl)c2Br)C3)cc2nccnc2cc1F 7655,CC(C)CS(=O)(=O)CCC(=O)NC1COC2CN(C(C3(C)CNC(=O)C3)=O)CC12 7656,N(C1CCCc2c(Br)cccc21)C(c1n(C(CC)(C)C)nnn1)(C)CCC 7657,N1(C(CC2(NC(c3cccc(C(C)C)c3)=O)CCC2)=O)CCC(O)C(C)(CO)C1 7658,C1(CC)CCN(C(c2ccc(=N)[nH]n2)=O)C(C(=O)NC(C)CCCO)C1 7659,CC(C)CC(O)C(C)C(=O)N(CCC(=O)NCCCC(C)CO)CC1CC1 7660,C1(NC(c2c(SC)cccc2)=O)CN(C(c2cnc(C3CC3)s2)=O)CCC1(C)C 7661,C(N=c1cc(C(F)(F)F)nc[nH]1)C1(NC(C(CC)SC)=O)CCOCC1 7662,C1(=O)C(C)(C)CC(C)(C)N(CC)C=CC2=NC2=NNC=CCO1 7663,N1(C(=O)Cc2ccc(Cl)s2)CCC(O)(C(N2CCC(CN3CCCC3)CC2)=O)C1 7664,C(=O)(C1CCCc2nn(C)cc21)NC(CC(C)C)CNC(=O)CSS(C)(=O)=O 7665,C1(C(N2CCC(NC(C=C(COC)C)=O)(CO)CC2)=O)C2CCC(C2)C1(C)C 7666,N1(C(c2ccc(C#C)cc2)=O)CCCC2CN(C(=O)C(n3ccnc3C)C)CC12 7667,N1(C(C(c2cc(OC)cc(CC)c2)N(C)CC)=O)C2CCC1CC(=O)NC2.C1(CC)CC1 7668,c1(N2CCC=C(C(=O)OC)C2)ncnc2c1ncn2C1CCC(CO)O1 7669,N1(C(c2c(CC)occ2C)=O)CC(NC(=O)CP(C)(C)=O)CC(O)C1 7670,C=CCCCC(=O)NCC12CC(CN1C(=O)CCc1cnn(C)c1C)C2 7671,Cc1cc2[nH]c(C(N3CCN(C(=O)CSCc4cccs4)C(C)C3)=O)cc2s1 7672,Cc1c(C(N2C3CCC2CN(C(C)C)C3)=O)sc2ccnc(O)c12 7673,CCC(CN(C)C)CC(=O)NC(C(=O)N(C1CCSCC1)C)C1CCC1 7674,c1(CC(=O)N(CCCN(C)C(C2CC2(F)F)=O)C)ncccc1Br 7675,C1(NC(C2CC23CCC3)=O)COCCC1NC(C1CCS(=O)CC1)=O 7676,N1(C(Cc2cccc(C(N)=O)c2)=O)CC(NC(c2cc(Br)co2)=O)C2(CCC2)C1 7677,C(C1CCOC1)=CC(=O)NC(C(=O)NCC1CC12CCC2)C1CCCC1 7678,Cc1cc(F)sc1C(=O)NCCC1CC(C(=O)NCC(O)CC(C)C)C1 7679,c1(C(=O)NC(CNC(C(C2CCC2)OC)=O)C)cc(O)c2cnn(C)c2c1 7680,N1(C(C(C)NC(COC)=O)=O)CCCCC1C(N1CC2CC2(CO)C1)=O 7681,CCC(CC(=O)NCC1CCCCCN1C(=O)COCc1nnc(C)s1)C(C)C 7682,c1(NC(c2scc(C)c2C)c2nnnn2C2CCOC2)ccc(Br)c(C#N)c1C 7683,C(=O)(C1=CC2(CN(C(=O)C(C)(C)n3cccn3)C2)OC1)NC(COC)C(C)C 7684,C1(CN(C(=O)CC2CCOCC2)CC)CCN(C(c2cnn(CC)c2)=O)CC1 7685,C1(CNC(c2cc[nH]n2)=O)(NC(c2ccc(-c3ccccc3)o2)=O)CCCCC1 7686,C1(NC(C(CC#C)C2CC2)=O)CN(C(c2ccc(F)c(CO)c2)=O)CC1N=[N+]=[N-] 7687,c1(C(=O)NC(CC)CN(C)C(C2(CC)CCOCC2)=O)ncc(C)cc1Br 7688,C(C(C(C)(C)C)CC(=O)O)COCCOC.C1(C(=O)O)CC(SC)C1 7689,C#Cc1cccc(OCC(N2CCCC2(C)NC(=O)C=CCCC)=O)c1 7690,Cc1cccc2[nH]c(=NC3CCCCC3CNC(=O)CCc3ccn(C)n3)sc12 7691,CC1(C(F)F)CC1NC(=O)NOCCn1cccn1 7692,c1(C(N2CCC(NC(C3CC(C)(CC)C3)=O)C(C)C2)=O)ccc2c(c1)CC(=O)N2 7693,C1(NC(=O)NC2CCN(c3ncco3)C2)CC2OCCC12 7694,C1(CNC(c2cc(CC)n(C)n2)=O)CCC(C)CN1C(=O)CSc1ccncc1 7695,C(=O)(C(C)C(C)C(C)(C)C)NCC(CC)NC(c1ccc2c(c1)nnn2CC)=O 7696,CC(C)S(=O)(=O)CC(=O)NCC(CNC(C1C2CCCCC12)=O)CO 7697,N1(C(c2c(CC)n[nH]c2)=O)CC2CN(C(=O)C(n3nccc3C)C)CCC12 7698,c1(OCC(=O)NCC2C(C)CN(C(c3ns[nH]c3=O)=O)C2)ccccc1C#N 7699,C(=O)(C1=CC(C)(CC)C1)N(CC1CCN(C(CC(=C)C)=O)CC1)CC 7700,c1(C(N2CCC(C)(NC(C(CC)C)=O)C2)=O)nn(C)c2ccc(Br)cc12 7701,c1(C(=O)NC2CN(C(C3(OCC)CCOC3)=O)C2)cc(F)cc(C)c1N 7702,c1(C(N(CCCCN(C(=O)C(F)CC2CC2)C)C)=O)ccccc1C#CC1CC1 7703,Cc1[nH]cc(C(=O)NC2CC(CO)N(C(=O)CCCN(C)C(C)C)C2)c(=O)c1Cl 7704,c1(OC)ccc2c(=NCC3(OC)CC3)[nH]c(=NC(C)Cc3cnccn3)[nH]c2c1 7705,N1(C(C(CC=C)C)=O)CCCCC(C2CN(C(c3ccc(O)c(N)c3)=O)C2)C1 7706,C1(C)(OC)CCCN(C(=O)C(CCF)NC(=O)CCCOC(C)=O)C1 7707,N1(C(C(C(C)O)NC(C(CC#C)O)=O)=O)CCCCC1C#C 7708,c1(NC(C2(Cc3scc(C)n3)CC2)=O)ccc(-c2ccns2)cc1 7709,C1(NC(c2scc(C(=O)OC)c2)=O)CC2CCC1N2C(=O)CC1CC2(CCC2)C1 7710,C1(C(=O)NCCCC(=O)OC)(CO)CCOCC1.C1(C=O)CC12CCCC2 7711,n1(CC(=O)NCC(C)(C)c2nc[nH]n2)cccc(N)c1=O 7712,c1(C(N2CCC(CNC(c3c(C)nc(C)s3)=O)C2)=O)oc(P(C)(C)=O)cc1C 7713,c1(NC(N2CCC(c3nc(=O)o[nH]3)CC2)=O)cncc(-c2ccc(Cl)cc2)c1 7714,N1(C(CCC#C)=O)CC(C)C(NC(c2cnc(S(C)(=O)=O)s2)=O)C(C)C1 7715,c1(CN(C)C)cccc(C(=O)NCC=C2CCN(c3ncc(Br)cn3)CC2)c1 7716,C1(CC(=O)N(CCCCCNC(=O)Cc2nn(C)cc2Cl)C)COCC(C)(C)O1 7717,C1(CC(C)C)(C(=O)NC2(C(=O)OC)CCC2c2ccccc2)CCNC1=O 7718,CCC(C(F)C(=O)OCC)NCc1cccc(C(F)(F)F)c1N 7719,c1(C(N(CC(C)NC(C2CC(=O)N2)=O)C)=O)ccc(F)c(O)c1 7720,C#CCC(CC(=O)NCc1c[nH]nc1C1CC1)NC(=O)CCN(C)C 7721,N1(C(C2CCCCCCN2C(=O)C(O)C2CC2)=O)Cc2cccnc2C1 7722,c1(C(=O)NCC(CNC(c2[nH]cc(CC)c2)=O)C)sc(CC(F)(F)F)nc1C 7723,c1(C(N2CC(CC=C)(NC(=O)Cc3ccc(O)nc3)C2)=O)ccc(Cl)c(C)c1O 7724,c1(N(CC(C)O)C(=O)NCc2cc(Cl)ccc2F)ccc2c(c1)OCCO2 7725,n1(C(C)C)cc(C(N2CC(C)(CCNC(=O)C(=O)NC3CC3)C2)=O)c(O)nc1=O 7726,c1(C(N(CCCCN(C(CCCC(C)=O)=O)C)C)=O)[nH]c2c(c1C)CCCC2 7727,C1(O)(CCNC(CCC2N(C)CCC2)=O)CCN(C(C2(C)CCCCO2)=O)C1 7728,Cc1cc(S(=O)(=O)NCCC(c2cccc3c2OCCO3)=O)cnc1C(F)(F)F 7729,c1(C(=O)OCC)ccnc(N(C)CCNC(C2(C(F)(F)F)CCC2)=O)c1[N+](=O)[O-] 7730,C=CCC(C)(CC)C(=O)NC(CNC(c1ccc(-c2cc[nH]n2)cc1)=O)CC 7731,c1(C(=O)NCCC2CCC(NC(C(C)C)=O)C2)ccc(F)cc1C1CC1 7732,Cc1conc1CC(=O)NCC1CCCN1C(C1CCCN1C1CCOCC1)=O 7733,Cc1ccccc1C=CC(=O)NCC1C2CN(c3nccc(C(C)(C)C)n3)CC12 7734,c1(-c2cnc(Cc3n(C(C(N)=O)C#N)nc(-c4ccco4)n3)o2)ccc(F)c(F)c1 7735,C=CCC(CC(F)F)NC(C1C(CC)CCN1C(c1cccc(F)c1)=O)=O 7736,N1(C(C2(CC)CCC2)=O)CC2CCCC2(NC(=O)CCN2CCCCCC2)C1 7737,C1(OC)CC(CCNC(=O)CCc2cnn(C)c2)N(C(c2cnc(C)n2C)=O)C1 7738,C12(c3nc(CC)nn3-c3ccc(OC)c(OC)c3)CC(C)(C1)OC2C 7739,N1(C(=O)NC(=O)C2=CCCCO2)CC(CCC2C(C=C(C)C)C2(C)C)C(C)(C)C1 7740,C(=O)(C(CNC(=O)C(C)NC(N)=O)OC)N(CCCF)CC 7741,C(=O)(C1=CCCOC1)N1C(CNC(c2ccc(C#N)n2C)=O)CC(OC)C1 7742,C1(C(N2C(CN(C(=O)CCc3ccoc3)C)CCC2)=O)CC(F)C(=O)N1 7743,N1(C(c2cc(OC)c(OC)nc2)=O)CCCC2(C1)CN(C(=O)C(C)=C1CC1)C2 7744,c1(C(=O)NCC=CCNC(=O)CC2CCCOCC2)ccc(F)c(Br)c1 7745,C1(NC(C2(CNC(=O)CC3CNC(=O)O3)CC=CC2)=O)CC2CCCCN2C1 7746,CC1(CC(=O)NC(CO)CCC2CC2)CCN(C(=O)CSc2nc[nH]n2)C1 7747,C1(C(=O)NC(COC)C)CN(C(c2cnc(C(C)=O)cn2)=O)CCN1 7748,CC1CC2CN(C(=O)CN3CCOCC3=O)CC2N1C(=O)CC1(CO)CC1 7749,C1(CNC(Cc2ccc(C)cc2)=O)CC(C(=O)N(C)Cc2scnc2C)=NO1 7750,C#CCCC(C(=O)NC1CC(O)C(O)C1)NC(c1snc(C)c1N)=O 7751,c1(CC(=O)NC2CC(O)CN(C(=O)CC3CC3)C2)c[nH]c2ncccc12 7752,C(=O)(C(C(C)(C)C)NC(c1cnc(OCC(F)(F)F)c(Cl)c1)=O)OCC 7753,Cc1c(C(=O)NC(CNC(C2CCCN2C(N)=O)=O)CO)oc2ccc(Cl)cc12 7754,N1(C(C=CC(C)C)=O)CC2CCN(C(c3ccncc3C(F)F)=O)CC12 7755,N1(C(C(C)(F)F)=O)CC2(CCCN(C(=O)C=Cc3ccc(C(F)(F)F)cc3)C2)C1 7756,c1(N(C(C(=O)NC(COCC)C(C)C)=O)C)cc(Br)cn1C 7757,CC(C)CC(CNC(c1cncc(C2CC2)c1)=O)NC(=O)C(C)c1ccco1 7758,c1(CC)cn2c(n1)CC(C(N1CCCCC1CN(C(=O)CCF)C)=O)C2 7759,Cc1nc(C(C)C)sc1C(=O)NCC1(O)CN(c2nc(CC3CC3)ns2)C1 7760,C#Cc1ccc(C(=O)NCCC(=O)N(CCCO)C2CC2)c(C)c1 7761,c1(C(N2CC(C(C)NC(c3nc(C)oc3)=O)C2)=O)cc(C(N)=O)ccc1F 7762,c1(C(=O)NCC2COCC2CN2CC(N3CCOC3=O)C2)cnn(CCO)c1 7763,C1(CNC(C2(C(C)C)CCCO2)=O)CCC2(CO1)CC(NC(C1(O)CC1)=O)C2 7764,c1(CC(N2CC(F)(CNC(C34CC(C)C3C4)=O)C2)=O)ccc(S(C)=O)cc1 7765,CC1CN(C(=O)CCN=[N+]=[N-])CC(C(N2CCC2CC2CCCC2)=O)O1 7766,C1(NC(=O)Cc2cccc(C(N)=O)c2)CC2CN(c3ncncc3Cl)CC12 7767,CCC(C)(CNC(=O)Cc1cc[nH]n1)NC(c1nocc1C)=O 7768,CN1CCN(CCOc2ccc(-c3ccccc3)cc2)CCC1C 7769,C(=O)(CC(C)CCCCCC)NC1C(C)CCN(C(C(C=C)(C)CCOC)=O)C1 7770,CC(C)C(O)C(C)C(=O)NCC(CO)NC(=O)CS(=O)(=O)Nc1ccccc1 7771,C1(CC)CCN(C(C2CC(F)C2)=O)C1CNC(=O)C(SC)SC 7772,C1(O)(CNC(C2CC(CCC)OCC2)=O)CCN(C(C2CCCC2C)=O)CC1 7773,c1(C(=O)NCC2(CN(C(c3nc(COC)oc3)=O)C)CC2)n[nH]c2ccccc12 7774,C1(CNC(=O)OC(C)(C)C)CC(NCCCC(C)(C)C)C1(C)C 7775,c1(OCCC)ccc(C(=O)NC(C)CCCNC(=O)Cn2ccc(C)n2)cc1N 7776,c1(C(=O)NC2(CO)CN(C(C=C(CC)CC)=O)C2)cc(C)ncc1C 7777,C1(F)(C(=O)NC2CC(OCC(=O)N(CCN(C)CCO)C3CC3)C2)CCCCC1 7778,N1(C(CCSCCC)=O)CCN(C(=O)C(C(C)(F)F)c2ccccc2)C(CC)C1 7779,NC(=O)CCCC(=O)NCCC1CCCCN1C(=O)CCNC(c1ccsc1)=O 7780,N1(C(C(=O)NCCCNC(C2CC23CCCC3)=O)=O)CCc2sccc2C1 7781,C1(NC(CC(CC)C)=O)COC2(CCN(C(c3ncc(Cl)cn3)=O)C2)C1 7782,c1(C(=O)OC)cc(C)c(F)c(S(=O)(=O)NCc2cc(C(=O)O)nc(C)c2)c1 7783,c1(C(=O)NCC2(O)CCN(C(C(C)C#N)=O)C2)c(C2CC2)nc2sccn12 7784,Cc1nccnc1C(=O)NCC(C(C)C)NC(=O)C=CCN1CCCC1 7785,C(C(C)(CNC(=O)C(COC)NC(C)=O)OC)NC(COC)=O 7786,N1(C(CNS(CC)(=O)=O)=O)CC(NC(c2ccc(CO)c(F)c2)=O)CC(F)C1 7787,N1(C(C2(COC)CCC2)=O)CC(CNC(=O)C(C)Cc2cnn(C)c2)C(C)C1 7788,Cc1cc(C)c(OCC(=O)NC(C)C(C)NC(c2cccc(=S)n2O)=O)c(C)c1 7789,C(=O)(CCCCCCS(N)(=O)=O)NC1C2(CN(C(CCC#C)=O)C2)CC1 7790,C1(C(=O)NCCC(C)N(CCC)C)(NC(=O)C(C)CC2CCCC2)CCN(C)C1 7791,c1(C(=O)NC2CCC(CNC(c3n(CC)nnc3C)=O)C2)cc(OC)ccc1Cl 7792,c1(C(=O)OC)sc(N(C(=O)C(=O)NCC23CC(C(N)=O)(OC2)C3)C)nc1C 7793,C1(CC=C)(C(=O)N(CC)Cc2nccs2)CCCN1C(=O)CC1CC2(CCC2)C1 7794,N1(C(C(C)OC(C)(C)C)=O)CCCN(C(C2CN3CCN2CC3)=O)CC1C 7795,N1(C(C2C(NC(C3(CC#C)CCOC3)=O)CCC2)=O)CCOC(CCC)C1 7796,N(C(=NCC(C)(C)CS(N)(=O)=O)N1CCC(Cc2ccccn2)CC1)C(C=C)C 7797,C(C(=O)NC1CN(C(C2CSCC(=O)N2)=O)C1)(C(C)C)c1cnc(C)s1 7798,c1(C(=O)OC)cc(S(=O)(=O)N2CC(CCO)C2)c(F)cc1C 7799,N1(C(C2C3CCN(C(CC(CC(C)C)O)=O)CC32)=O)CCC2CCN(C)CC12 7800,CCC(CC(C)C)C(=O)NCC1(NC(c2cnc(SC)s2)=O)CCOC1 7801,c1(NC)ncccc1C(=O)NCCN(C(=O)C(C1CCC(=O)N1)C)C(C)C 7802,c1(C(C)=O)cc(C(N2CCCC(C)(CNC(=O)C(O)C(C)C)C2)=O)ccc1C 7803,N1(C(CC2CC(=C)C2)=O)CCCN(C(C2CCCN(CC(F)F)C2)=O)CC1C 7804,c1(C(=O)NCC(C(=O)NCCCC(CC)C)(C)CC)cc2ccccn2c1 7805,C(C(CC(C)C)C(=O)N(CCC(=O)N(C)CCN1CCCCC1)C)OC 7806,C1(NC(c2ccc(CC)cn2)=O)CN(C(c2cnc(S)[nH]2)=O)CCC1O 7807,Cc1nc2c(s1)CCCC2C(=O)NCC(C)NC(C1COC(C)(C)CO1)=O 7808,c1(C(N2CCC(F)C2)=O)ncn2cc(N)ccc12.N1(C(=O)C)Cc2ccccc2C1 7809,N1(C(c2c(CC)nns2)=O)CC(Nc2ncc3c(n2)CCCC3)CC2(CCC2)C1 7810,C1(OC)CC2(C1)CC(CN=C(NCC1CC1(F)F)NC1CC1)C2 7811,N1(C(c2c(C)ocn2)=O)CCN(C(=S)NC(c2ccc(S(C)(=O)=O)cc2)=O)CC1 7812,c1(CCC(=O)N(CCNC(C2CC(CC)C2)=O)C)ccc(Br)cn1 7813,C1(C)(CNC(C2(SC)CCCCC2)=O)CCN(C(c2ccc(=N)[nH]n2)=O)CC1 7814,C1(NC(CN2CC(C)(C)C2)=O)CCN(C(C2CCC(C)(C)OC2)=O)CC1(C)C 7815,N1(C(c2c(C(F)(F)F)n[nH]c2C)=O)CC2CCN(C(=O)C3=CCCCO3)C(C2)C1.CS 7816,C1(C(C)C)CN(C(c2ccc(C(F)F)nc2)=O)CCN1C(=O)C#CC(=O)O 7817,C1(NC(CNC(=O)OCC=C)=O)CCCC1NC(=O)CC12CC(CO1)C2 7818,CC1(C)CC2(CC2C(=O)N=S(C)(=O)C2CCOC2)c2ccccc2O1 7819,c1(OC)cccc(C(=O)NCc2cc(C(=O)NCC3CC3)n[nH]2)n1 7820,CCC(C)(C)C(=O)C(=O)NCC1(CCNC(C2CC(O)CN2C(C)=O)=O)CC1 7821,c1(C(C)NC(=O)NC2CC(OC)(C(F)F)C2)cc(Cl)c(C)cc1O 7822,c1(NC(c2cnc(C)[nH]2)=O)cccc(NC(=O)CC(C)(F)F)c1 7823,CCC(N(C)N1CCN(C(c2ccc(F)cc2)=O)CC1)c1cc(Cl)cc(Cl)c1 7824,C(=O)(C1=CS(=O)CCC1)NCC1N(C(C(C(COC)C)C)=O)CCCC1 7825,C(N=c1cc(C)nc(C)[nH]1)C1C(NC(CCCC)=O)CCC1 7826,C#CCCC(C(=O)NC(c1ccn(C)n1)C)NC(C1CC2(CCC2)CO1)=O 7827,N1(C(c2cc(SC)oc2)=O)CC2CC1CCC2NC(=O)Cc1ccc(F)cc1F 7828,N1(C(C=CC=C)=O)CCC(F)(C(=O)NC2CCC2)CC1.CCOCCO 7829,C1(C(N(CC(CC)NC(C(CC)C2CCOCC2)=O)C)=O)CC(C)CC(=O)N1 7830,N1(C(c2cn(CCNC(C3(C)CCCCO3)=O)nc2)=O)CC(CSC)C2(CC2)C1 7831,c1(NC(C(C(=O)OC)C)=O)ccc(C)c(C(=O)NC2CCCC(O)C2)c1 7832,N1(C(Cc2c(C)ccs2)=O)CC(O)CC1CNC(C1CC1c1ccncc1)=O 7833,C1(CC)CCOC1C(=O)NCCCC(=O)NCC1CCCCO1 7834,C1(C)(CNC(CC(CCC)O)=O)COCCN(C(=O)CC2CN(C)C2)C1 7835,N1(C(c2n(CC)cnn2)=O)CCC(C2CC2)C1CNC(c1nc(F)ccc1Cl)=O 7836,N1(C(=O)CC2CSC2)CCC2CCCN(C(c3ccccc3C3CC3)=O)C2C1 7837,C(CNC(=O)C(F)(F)C(C)(C)O)(CC(=O)N1CC(O)CCCO1)OC 7838,N1(C(C2(NC(=O)C(O)C(C)(C)C)C(C)(C)C2)=O)CC2C3CCC(C3)C2C1 7839,C(=O)(C1COc2ccc(F)cc21)NC1C(NC(=O)Cc2ccc(Cl)cc2)C1 7840,C#CCC(CC(=O)NC1(CC)CCC1)NC(C1CCN(C(C)=O)C1)=O 7841,N1(C(C(C)CSC(F)(F)F)=O)C2CCC1CN(C(=O)CCCn1ccnc1)C2 7842,c1(C(N2C(CO)CC(NC(C3=NOC(C)C3)=O)C2)=O)cncc2ccccc12 7843,C1(N)(C(=O)O)CCS(=O)(=NC(=O)Cc2cc(NC(c3ccccc3Cl)=O)cs2)CC1 7844,N1(C(c2ccc(CCC)c(N)c2)=O)CCCC2(C1)CN(C(=O)C(C)(CC)CO)C2 7845,C1(NC(C2CCN2CC)=O)CCCC1NC(C1(F)CCC1)=O 7846,C1(CCC(C)(C)NC(C2(N3CCCCC3=O)CC2)=O)CCN(C(=O)C2CC2)CC1 7847,CC1CCCCC1Cc1nc(-c2cccc(Cl)c2)nn1-c1nccn1C 7848,C=CC(C)(CCOC)C(=O)NCC1(NC(=O)CNC(C)=O)CCCC1 7849,Cc1c[nH]nc1C(=O)NCCN(C(=O)C(F)n1cccn1)C1CC1 7850,N1(C(c2n(C)nnc2)=O)CCCC(CNC(c2cnn(CCO)c2)=O)C1 7851,C1(NC(c2nncs2)=O)CC2CC(NC(C34CCCC(CO3)C4)=O)C1C2 7852,Cc1cc(Cl)ncc1CC(=O)NC1CC2CCC1(NC(=O)C=Cc1cc[nH]n1)C2 7853,CCC1=NOC(CNC(=O)Nc2ccnc(OC(C)C)c2)C1 7854,Cc1nc(C)n(CC(=O)NC(CNC(=O)CCSC(F)(F)F)C(C)(C)C)n1 7855,c1(C(N2CCC(CC(C)NC(C3(C=C)CC3)=O)CC2)=O)ccc(F)c(Cl)c1N 7856,C1(NC(=O)C#CC2CC2)CN(C(=O)Cc2c(F)cccc2F)C2CCCCC12 7857,C(c1ncc[nH]1)=CC(=O)NCC(C)(C1CC1)NC(C1CC(CC2CC2)C1)=O 7858,C1(CC)(CC)C(CO)CC1NC(N1CCN(OCc2ccccc2)CC1)=O.C1CO1 7859,c1(C(N2CC(C)N(c3nnc(CO)s3)CC2)=O)cccn2nnnc12 7860,N1(C(C(n2c(C)ncc2)C)=O)CC(NC(=O)CC(F)(F)C(F)F)CC12CCC2 7861,C1(CN(C(CC(=C)Br)=O)C)CCN(C(C2CCCC(OC)C2)=O)CC1 7862,c1(NC(=O)NCC2(O)C(C)(C)COC2)cc(F)cc2ncoc12 7863,Cn1c(O)nc2cc(C(=O)NC(C)(C)CCNC(=O)CSC(C)(C)C)ccc12 7864,c1(C(=O)NC(CCCC2(C(=O)NCCCC)CC2)C)ccsc1C#N 7865,N1(C(CC2(OC)CCC2)=O)C2CCCC1CN(C(C1CC(O)C1)=O)C2 7866,n1(CC)ncc(Cl)c1C(=O)NC1CCC(CNC(=O)Cc2cccc(N)c2)CC1 7867,c1(C(=O)NCC2C3CN(C(C4CN(C)C(=O)C4)=O)C2C3)n[nH]c2c1CCC2 7868,C1(CC(=O)N(CC(C)N(C)C(c2cc3sccc3s2)=O)C)CCC(C)(C)CO1 7869,c1(COC)cccc(C(=O)NC2CN(C(=O)C=CC(C)(C)C)CC2O)n1 7870,c1(N2C(C=C)(C)COCC2)sc2cc(Cl)ccc2c1Cl 7871,C=CCC(C)C(=O)NCC(C(=O)N1CCC(COC)C1)N(C)C 7872,Cc1c(F)ccc(C(=O)NCCCC2CN(C(c3ccc[nH]3)=O)CCO2)c1Cl 7873,N1(C(COC)=O)CCN(C(=O)CP(C)(C)=O)C(CO)C1 7874,Cc1cc2[nH]c(C(=O)NC3CC4CC3N(C(c3ccsc3)=O)C4)cc2o1 7875,N1(C(=O)OC(C)(C)C)C2CCC1C(C(=O)NC(C1CC3CNC(C1)C3)C1CCC1)C2 7876,C(CCN=c1ccc(C(F)(F)F)c[nH]1)N(C)C(c1cccc(Br)c1Br)=O 7877,Cc1nc(N2CCC(F)C(NC(=O)OC(C)(C)C)C2)c(C)c(C)n1 7878,N1(C(c2cc(C)[nH]n2)=O)CC(C)OC2(CCN(C(=O)Cc3cccn3C)C2)C1 7879,c1(NCC(C)(CC(C)C)NC(CCCCCCC)=O)ncnc2c1nnn2C 7880,C1(C(C)(CSC)NCCCOCCO)CCOCC1 7881,CC(CN(C)C)CCC(=O)N1CC(CNC(c2cccs2)=O)CC1(C)C 7882,N1(C(C2C(C)CCN(C(C(F)=CCC)=O)C2)=O)CC(C)(CO)CC1(C)C 7883,C1(CNC(=O)Cc2cccc(F)c2)CN(C(C2CCCC(F)(F)C2)=O)CC12CC2 7884,N1(C(CN(CC)CC)=O)CC2CCC1C1CN(Cc3ccccc3)CC21 7885,C1(CNC(C(c2cccc(Cl)c2)C)=O)CCN(C(C23CC(C)(CO2)C3)=O)CC1C 7886,C(=O)(C(C)CC(F)F)NCC(CC=C)NC(c1ccnc(OCC)c1)=O 7887,Cn1c(C(=O)NCC=CCC(=O)NC2CC(=O)N(O)C2)ccc1C#N 7888,CC1CCCC1(O)CNC(=O)C(c1ccnn1C)NC(c1cnc(C2CC2)o1)=O 7889,c1(C(=O)NC2CCN(C(C3CN(CCC)C(=O)C3)=O)C2)ccc2c(c1)CCCN2 7890,C1(OC)CCC12CC(C(=O)NCCC1(C(=O)NCC34CCN(CC3)C4)CCC1)C2 7891,C(c1ccc(F)cc1)=C(C)C(=O)N1CCC1n1cc(COCC(=O)O)nn1 7892,C(=O)(C(C)S(N)(=O)=O)N1C(C(N2CC(CO)C2)=O)(COC)C=CC1 7893,N(C(=NCCC(=C)C)NC1CCN(c2ccc(-n3cncn3)cc2)CC1)C1C(=C)C1 7894,N1(C(CC(C(C)C)c2ccon2)=O)CC2CCC1C(CNC(C1(CO)CC1)=O)C2 7895,c1(C(=O)NCC2C(C)CN(C(C3(CO)CC3)=O)C2)ccc2c(O)ncnc2c1 7896,C(=O)(C1=CC2(CCOC2)C1)NCCN(C(=O)CCc1cnc[nH]1)C 7897,c1(CNC(C(CC)SC)=O)nc(CNC(C2CCC3CC2CO3)=O)cc(O)n1 7898,c1(CC)cnc(C(=O)NC2CCC(C(=O)N(C(C)CC(C)C)C)C2)nc1 7899,Cc1cc(=NC(=O)C(=O)N2CCC(C3NC(=O)OC3C)C2)[nH]o1.C1CCN1C 7900,c1(C(=O)NC2C(NC(C3(CC)CCOCC3)=O)CC2)cncc(C)c1C 7901,C1(NC(C2CC(C#C)(O)C2)=O)CC2CCCC(C1)N2C(=O)C#CC1CCOC1 7902,O=S(=O)(c1cnc(NC2CCOC2C2CC2)c(Cl)c1)NC1CCC=CCC1 7903,N1(C2CCN(C(C3CN(C)C3)=O)CC2)Cc2cccnc2N2CCCC2C1 7904,C1(c2onc(C(C)C)n2)CN(C(=O)NCc2csnn2)CCO1 7905,c1(N2CCN(CCCNC(C3CC(=O)NC3=O)=O)CC2)ccccc1[N+](=O)[O-] 7906,N1(C(c2cnc(CCC)s2)=O)CCCC(C)(NC(=O)CC(C)(C)OC)C1 7907,c1(C(=O)NCCN(C(CC(C)SC)=O)CC(C)O)cc(F)c(F)c(N)c1Cl 7908,c1(SCC(=O)NCC(C)(C)NC(C(CO)N(C)C)=O)nc2ccccc2o1 7909,N1(C(C)C)CC(NC(=O)C(C(C)(C)C)NC(=O)C=Cc2nnn(C)n2)CCC1=O 7910,C1(CN(C)C)CCC(C(=O)NC2CC23CC(NC(=O)CSc2cccs2)C3)CC1 7911,C(=O)(C(CCNC(c1cccn1C1CC1)=O)OC)NC1(CC#C)CC1 7912,N1(C(C2(CC)CCN(C(=O)CN(C)C)C2)=O)CC(=O)NC(C)C1 7913,N1(C(COCCC#C)=O)CCC2C(NC(=O)COC(F)(F)F)C2C1 7914,N1(C(CC2(CC)CCC2)=O)CC(CNC(C2(F)CCCC2)=O)C2(CC2)C1 7915,C(=O)(C(CC(C)C)NC(=O)C(C#N)CC1CC1)OCC 7916,c1(NC(CCC(=O)C2CCCCC2)=O)nc(F)c(I)cc1F 7917,C1(O)(C(=O)NC(C2CCCN(C(=O)C=Cc3cnc[nH]3)C2)C)CCCCCC1 7918,C1(NC(C2(C)C=CCC2)=O)CCCC2CN(C(=O)Cc3csc(Cl)c3)CC12 7919,CC1(CNC(=O)CC2NC(=O)NC2=O)CCN(C(=O)CCc2ncccn2)C1 7920,c1(CC)ccc(F)cc1C(=O)NCCCCCCNC(c1cc(F)ccc1O)=O 7921,N1(C(C(C)SCC)=O)CCN(C(=O)CCOC(C)=O)CC1CC(F)F 7922,C12(C(N3CC=CC(NC(CSCCOC)=O)C3)=O)CCC(C1)C(C)(C)O2 7923,c1(C(N2CC(CCNC(C(C)OC)=O)C2)=O)ccc2nc(O)[nH]c2n1 7924,N1(C(=O)CC23CCCC2C3)CC=CC(C(=O)N(C2CC2)CC2CCC2)C1 7925,C(CC(C(C)(C)C)NC(c1cn(C)cn1)=O)N(C)C(C1CCOC(C)(C)C1)=O 7926,N1(C(CCOCC(C)C)=O)CC2(CCCC2)C1C(=O)NC(C1(O)CCC1)C 7927,N1(C(CNC(C(C)(C)C)=O)=O)CCC(N=[N+]=[N-])(C(=O)NCC2(O)CCCOC2)C1 7928,C1(NC(C(C)c2ccco2)=O)COCC1CNC(c1csc(C(C)(C)C)n1)=O 7929,C1(N(C(C(C)SCCCC)=O)C)C2CN(C(c3cc[nH]c(=N)n3)=O)CC12 7930,c1(C(=O)NCC2CN(C(CCC3C(C)=NOC3=O)=O)C2)nc(O)nc(O)c1N 7931,Cc1cc(C(N2CCC(OC(C)C(N)=O)CC2)=O)c(Br)cc1F 7932,CCC(C)C(O)CC(=O)NC(CNC(=O)CCCCN(C)C)CC(F)(F)F 7933,C1(OC)CCC(NC(=O)CCN(C)C(c2ccc(C)o2)=O)C1 7934,c1(OC)ccc2cc(C(N3CCC(NC(=O)Cc4cnc(C)o4)C3C)=O)[nH]c2c1 7935,C=CC(O)C(=O)NC(Cn1cccn1)C(=O)N1CC(C)(C(N)=O)C1 7936,N1(CC)CC(C(=O)NCC2CCCC2NC(=O)CC2CCCOCC2)CCC1=O 7937,N1(C(C(C(C)C)F)=O)CCC12CN(C(C1(c3ccc(O)cc3)CC1)=O)C2 7938,C1(C)(CNC(c2nc(C(=O)OC)oc2)=O)CCCN1C(c1cnn(C)c1Cl)=O 7939,Nc1ccc(I)cc1S(=O)(=O)N1CCC(C2CCCCC2)CC1 7940,C(=O)(CC(P(C)(C)=O)P(C)(C)=O)NC1CC(NC(c2cc(C)nn2C)=O)C1 7941,C(=O)(C1=CC(C)(C)C1)NCC1CN(C(c2cnc(C)nc2)=O)CC1C 7942,C(=O)(C(C)(C)C(=O)NCC1CN(C(c2cn(C)nc2C)=O)C1)OCC 7943,CC1(C)CCCN(C(C2CC(N=[N+]=[N-])C2)=O)C1C(=O)NC1CCCSC1 7944,c1(CNC(c2cnc(C)s2)=O)ccc(C(=O)NCC2(F)CCOCC2)nc1 7945,C1(O)(CCNC(CSc2n(C)nnn2)=O)CCN(C(C2(C#N)CCC2)=O)C1 7946,C(C1=CCN(C(c2cnc(-c3ccco3)s2)=O)CC1)NC(C1(C=C)CCC1)=O 7947,C1(C(N(C)Cc2c(C)cco2)=O)C2CC3C(C2NC(C2CCC(F)C2)=O)C13 7948,C(=O)(C1=CC2CCCC12)NCCC1CN(C(=O)CCc2ccco2)C1 7949,CC(CC(N)=O)C(=O)NCC(C)CNC(C1(C(F)(F)F)CC=CCO1)=O 7950,c1(C(N2CC(CNC(CC3(CC)CC3)=O)CC2(C)CC)=O)ccn2nncc2c1 7951,N1(C(CCC#C)=O)CC2OCC(NC(=O)C(C)OCC)C2C1 7952,c1(C(N2C3CCC2CC(C(N2CCC(O)C(F)C2)=O)C3)=O)c(F)cc(Cl)cc1Cl 7953,N(C(=NCc1ccoc1)NCc1ccccc1-c1ccc(F)cc1)CC(C)(C)C 7954,C=C(Br)CCC(=O)NCC(CCOC)NC(=O)C(C)SC 7955,C(N=c1ccnc(CO)[nH]1)C12OCC(CNC(C3CCC(C)CC3)=O)(C1)C2 7956,c1(C(=O)NCC2(OC)CCCC23CCC3)ccc2c(c1)C(C)(C)CCN2 7957,c1(CC(=O)NC(CCN(C)C)C(=O)OC(C)(C)C)c(C)nn(C)c1C 7958,c1(-c2c(C(N(CCC(C)NC(C3CC3(C)C)=O)C)=O)c[nH]n2)ccccc1Br 7959,C(=O)(C(C)(O)CC(C)C)NC(C(=O)NC(CC)CCCO)CO 7960,c1(C(N(CC(C)(C)NC(C2C(CCC)C2)=O)C)=O)cnsc1C 7961,N#Cc1ccc(Cl)nc1NC(C1C2CN(C(C3CC3(F)F)=O)CC12)=O 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8160,N1(C(CN(C2CC2)CC)=O)CC2(C1)CN(C(=O)CCC1CCCO1)C2 8161,Cc1c[nH]c2ncc(C(=O)NCC3(CNC(=O)CN4CC5CCC4C5)CC3)cc12 8162,C=CC(C)(C)C(=O)NC(C)CCCNC(C1(CC)CCCCC1)=O 8163,C12(NC(=O)CCF)CCCC1CN(C(c1ccc(-c3ccsc3)nc1)=O)C2 8164,c1(C(=O)NC2CCC(NC(C3(C(C)C)CC3)=O)C2)cccnc1C(=O)NC1CC1 8165,c1(C(=O)NC2C(CNC(=O)CCF)COC2)ncccc1C1CC1 8166,c1(OC)ncc(C(=O)NCC(CNC(=O)CCc2csc(=N)[nH]2)OC)cc1C 8167,C1(C)(C(=O)NCC2CC(NC(c3n(CC)ccc3)=O)C2)CCC(=O)N(C)C1 8168,CC1CN(C(=O)COC2CCC2)CCCN1C(C1C2COCC12)=O 8169,C1(N(C(Cn2nnc(=N)[nH]2)=O)CCO)CCN(C(=O)CC2CC(OC)C2)CC1 8170,c1(CC)nc(NC(C2CN(C(=O)CN(C)CC3CCCC3)C2)C)cc(C)n1 8171,C1(NC(c2coc(Cl)n2)=O)CCC2(CC1)CCN(C(c1ccc(I)c(O)c1)=O)C2 8172,C(C)(N=c1[nH]c(=N)[nH]c(=NCC(C)C)[nH]1)c1ccc(F)cc1.c1(CC)ccccc1 8173,c1(C(=O)NC2C(NC(C(C)C3CC3)=O)CCC2)cccc(-n2ccnn2)c1 8174,C1(CC)CC1N=c1nc2sccc2c(Nn2cc(-c3ccccc3Cl)nn2)[nH]1 8175,N1(C(c2cnc(CCC)s2)=O)CC(NC(=O)C(C)(CC)CO)C(C2CC2)C1 8176,CC1(C)CN(C(c2ccc(F)c(F)c2Br)=O)CCC1NC(C1CC1CF)=O 8177,Cc1nnc2n1C(C(=O)N1CC(C)(NC(C3CCc4nccn4CC3)=O)C1)CC2 8178,C1(C(=O)NC(C(=O)OCC)CC)CN(C(C2(Cl)CCC2)=O)CC12CC2 8179,C1(NC(C=CCCC)=O)CCC2(CCN(C(C3(C)CCCC3O)=O)C2)C1 8180,C1(O)(CNC(c2n(C(CC)C)ncc2)=O)CCN(C(C2CCCOCC2)=O)CC1 8181,Cc1cnn(C)c1CC(=O)NCC1CCCN(C(c2cnn(C3CCC3)c2)=O)C1 8182,C1(NC(=O)CBr)CCC(NC(C2(n3cccn3)CC2)=O)C1.C(C)N 8183,C(C(C(=O)NCc1cc(C)no1)C(C)(C)C)NC(C(C)(C)SC)=O 8184,c1(OC)nc(C)cc(C)c1NC(N1CCCC(C(C)=O)C1)=O 8185,C(C)(C)(CCCC(=O)Nc1cnn(C)c1C)NC(CCn1ccc(C)n1)=O 8186,C12(C(=O)NC3CCN(C(CC(C=C)C)=O)C3C)CCC(CC1)C(C)O2 8187,C1(CCNC(=O)CN2CCCC2)(OC)CN(C(=O)C(n2cc(Cl)cn2)C)C1 8188,c1(SCC(=O)NCC(C)NC(c2ccc(OCCF)cc2)=O)ccc(O)cc1 8189,N1(C(CC=C=C)=O)CCC2(CC1)CN(C(c1cc(F)cnc1Cl)=O)CCO2 8190,N1(C(=O)NC2CN(C3CCCCC3)C2)CCC(C2CCCC23OCCO3)C1 8191,c1(CC)c(C(C(=O)NCc2nnn(C)n2)N(CC(C)C#N)C)cccc1C 8192,N1(c2ccnc(NC(c3ccncc3Cl)C)n2)CC2CC1CS2=O 8193,N1(C(C(Cn2cncn2)NC(COCCSC)=O)=O)CCCN(C(C)C)CC1 8194,Cc1ccnc(C(N2CCN(CCNC(C3(C)CCCC3C)=O)CC2)=O)c1O 8195,CC(C)(C#CC(=O)N1CC(O)C(C)(C)C1)CNC(C1CCC(=O)N1)=O 8196,Cc1cc(C(=O)NCC2CC2CNC(=O)CC2CCCOC2)cc(N)c1 8197,c1(NC(CNC(C(N2CCC(C)C2)=O)=O)=O)c[nH]c2cccc(Cl)c12 8198,N1(C(CCC#N)=O)CCN(C2CCCC2NC(=O)CC(O)CC2CC2)CC1 8199,c1(COC)cc(C(N2CC=CC2C(=O)NCC(n2ccnn2)C)=O)n[nH]1 8200,C1(CCCC)(C(N2CCC(C(=O)OC)C2)=O)CN(C(C2CCC2C(=O)OC)=O)C1 8201,c1(C(=O)NCC2CCC(CC(=O)OC)CC2)cc2cccc(Br)n2c1 8202,C1(C(=O)NC(C)CC(=O)N(C)CCOCCCO)CC2CC(=O)C1O2 8203,C1(NC(=O)Nc2ccccc2)CCN(C(c2ccc(F)s2)=O)C1 8204,c1(C(N2C(CC(N3CCCC(F)C3)=O)COCC2)=O)ccc(Cl)c2cc[nH]c12 8205,C1(CC(=O)NCC2(NC(C3CCC4(CCC4)O3)=O)CCCC2)CCC2(CCC2)O1 8206,C(=O)(CCC(=O)NCCC1COCCN1C(=O)Cn1cc(C2CCC2)nn1)NC 8207,C(C(C)(C)N=c1[nH]nc(C#N)s1)N(C)C(c1cc2c(=O)[nH]ccn2n1)=O 8208,C12(CC)CCCC1CN(C(C1CC3(CO1)CN(Cn1ccncc1=O)C3)=O)C2 8209,N1(C(c2c(N)nccc2)=O)CCC2(CNC(C3(C(F)F)CCCO3)=O)CCCC12 8210,c1(C(=O)OC)cc(C)cnc1NC1CC(C)N(C(c2cnn(C3CCC3)c2)=O)C1 8211,C(CC(C)C)(C(=O)N1CCC(C(C)CO)CC1)N(C(CSCCC(C)C)=O)C 8212,N1(CC(=O)NC(CC)C)CCC2(CC1)CN(C(c1ccccc1F)=O)CC(C)O2 8213,C1(C(=O)NCCCC(=O)N(CCCN(C)C)CCC)CC(=O)OC1(C)C 8214,C(=O)(C1CCCc2scnc21)N(CC(CO)(CO)NC(=O)C=Cc1ccoc1)C 8215,c1(C(C)=O)cc(C(=O)NC2COCCN(c3ccnc(C)n3)C2)ccc1[N+](=O)[O-] 8216,c1(C(N2CC3(C2)CN(C(C2C=CCN2)=O)C3)=O)cc(C(F)(F)F)ccc1O 8217,C1(N(C(C2CCN(CC(C)C)C2)=O)C)CN(C(=O)CCCC2CC2)CC1O 8218,C1(CNC(c2c(C)cc(C)s2)=O)CCC12CCN(C(C1CCCOC1)=O)CC2 8219,N1(C(c2cc([N+](=O)[O-])sn2)C(=O)NCC2CC2)CCOc2cccc(F)c2C1 8220,N1(C(c2c(COC)cc[nH]2)=O)CC=CC1(CNC(C1CCC2(CC2)C1)=O)COC 8221,c1(C(=O)NCCN(C(c2sc(C)cc2Br)=O)CC)cnc(OC(C)C)cn1 8222,Cc1ccc(-n2cc(CCCNC(C3(CO)CC3)=O)nn2)cc1Cl 8223,c1(C(N(CCOC)CCNC(C2CN(c3nncs3)C2)=O)=O)cc(CO)n(C)n1 8224,Cc1c[nH]nc1C(=O)NC(C)CC(C)NC(=O)C(c1cncnc1)C 8225,C(=O)(C1=CCCCO1)NCCN(C(C1(O)CCN(C(=O)OC(C)(C)C)C1)=O)C1CC1 8226,c1(NC(C2CCC(c3cc[nH]n3)O2)=O)c(F)ccc(Br)c1F 8227,C1(CCC(=O)NC2CCCC2CNC(C2CC(=O)N2)=O)CCCCO1 8228,C(=O)(CC(C)CNC(C1C=CCCN1C(=O)CSC(C)(C)C)=O)OC 8229,c1(C(N2CC(OC)(CNC(=O)C(C(C)(C)C)NC(C)=O)C2)=O)cnc2nccn2c1 8230,Cc1cn(C)nc1C(N1CCC(CNC(=O)CC2CCC(C(F)(F)F)O2)CC1)=O 8231,C(=O)(C(C)(C)c1cccnc1)NCCN(C(C)C)C(c1nocc1Br)=O 8232,C1(NC(c2c(OC)csc2)=O)C2CC(O)C1N(C(=O)C=CC1C(C)C1(Cl)Cl)C2 8233,c1(C(=O)NCCCCCCNC(C2N(CC)CCC2)=O)[nH]c(=N)ccc1C 8234,CN1CCN(C)C(CN(C=O)Cc2ccc(-c3cccc(Cl)c3)o2)C1 8235,C1(C(N2CC(NC(C(c3cncnc3)C)=O)C(O)CC2)=O)CC2CC1CC2(F)F 8236,N1(C(c2c(CC)con2)=O)CC=CC(C(=O)NCC#CC2CC2)C1 8237,c1(Sc2nnc(NC(Cn3ncc(C#C)c3)=O)s2)ccc(Cl)c(F)c1 8238,c1(-n2cc(C3N(C(CSC(C)(C)C)=O)CCC3)nn2)ncc(Cl)cc1Cl 8239,CC1COCC(C(=O)NC(C)(C(=O)N(C2CCN(CCF)C2)C)C2CCC2)O1 8240,C1(C(=O)NCCN2CC(=O)NCC2)C2CCC(C2)C1NC(C1CC(=C2CCC2)C1)=O 8241,c1(C(C(=O)Nc2c(C(=O)OCC)c[nH]n2)(C)C)ccc(Cl)cc1Cl 8242,C(=O)(C(CNC(C1OCC2CCCC12)=O)CC(C)C)NC(CC)C(F)(F)F 8243,C(=O)(CCCC(C)(C)NC(=O)C(C)C(C)C)N(CC#CC)C 8244,c1(Cc2ccc(CNC(C3N(OC)CC(F)C3)=O)o2)ncnc2cc(Br)ccc12 8245,C=CCC(CC=C)C(=O)N1CCCC(C)(NC(=O)CCOC(C)C)C1 8246,Cc1ccc(CCNC(=O)CCOCCCNC(C2CCOC2)=O)nc1 8247,CC1CCC(NC(=O)CCCN2CCCC2)CN1C(=O)CN(C)CCO 8248,O=S(=O)(CCn1cc(-c2cccs2)nn1)c1ccccc1F 8249,C1(CNC(C(F)=CCC)=O)CC(NC(c2coc(-c3ccsc3)c2)=O)C1(C)C 8250,C(CC(C)(C)C(F)(F)F)NC1(N(C)C(=O)NC(C)C)CCCC1 8251,NC(CCNCc1csc(C(F)(F)F)n1)C(F)(F)F 8252,C(CCC(C)(C)NC(=O)CC1CCC(C)C1)NC(CSc1nc(C)[nH]n1)=O 8253,C(CS(=O)(=O)CC(=O)NC(C1CC(NC(=O)CN2CSCC2=O)C1)C)OC 8254,N1(C(C2(C)CC(C)C2)=O)CCN(C)C(CNC(C2(C)CCCS2)=O)C1 8255,C(=O)(C1=NN(C2CC2)C(=O)CC1)NC1C(CNC(c2cc(OC)n[nH]2)=O)C1 8256,C1(NC(CCC=C)=O)CC2CCCC(C1)N2c1cc(SC)ncn1 8257,C1(NC(CC2CC(SC)C2)=O)C=CCN(C(c2ccc(C)cn2)=O)C1 8258,CCCCC(C(=O)NCC1CCCN(C(c2ncccc2CO)=O)CC1)C(C)C 8259,C(CCCCCCCO)=CC(=O)NC1CN(C(C(C(C)C)OC)=O)CC12CC2 8260,C1(NC(C(CC)NC(c2ccn(C)c2)=O)=O)CN(CC)CC1C 8261,c1(C(N2CCCC(O)(CNC(C(C(C)C)C#N)=O)C2)=O)sc2cccnc2c1Cl 8262,N1(C(C(C)O)=O)CCCC(C2CCCN(CCCOc3cccc(Cl)c3)C2)C1 8263,C1(C(=O)NCC=CCNC(C2(CC)CCOC2)=O)CC2(C1)CC(C)C2 8264,C1(C(N2CC(C(C)OC)C2)=O)(CCNC(=O)C(C)C2CC2)CCCC1 8265,c1(NCC(=O)NC2(F)CC(NC(CCSC)=O)C2)cccnc1C(=O)OC(C)=O 8266,c1(OC)cc(OC)cc(NC(=O)N(C)CC2CCN(CC(C)O)CC2)c1 8267,C1(NC(CN(C(COC)=O)C)=O)CC(F)CN(C(=O)C(F)(F)CO)C1 8268,c1(CCNC(C(N2CCC(C(N)=O)CC2)c2cn(C)nn2)=O)cccc(F)c1 8269,C1(CNC(C2(CCC=C)CC2)=O)CC2CC1CN2C(=O)COC(C)CC 8270,c1(C(=O)NC2CC3(C2)CN(C(=O)COCC2CC2)C3)cc2cccc(F)c2s1 8271,CN1CCC(=CC(=O)NCC2CCN(C(=O)CC3CCC(=O)N3)C2)CC1 8272,C(=O)(C(C)(C)C(F)F)N(CC(C)(C)NC(C1CC12CC2)=O)C 8273,c1(C(=O)NC2C(C)CN(C(C3(F)CC3)=O)CC2C)ccc2ccccc2n1 8274,N1(C(C2CN(C(c3c(C)nsc3C)=O)CC2C)=O)CCCc2occc2C1 8275,C1(NC(CCSC)C)Cc2ccccc2CN1C(=O)OC(C)(C)C 8276,C12(CNC(COCCCOCC)=O)CC(NC(C3COCCO3)=O)(C1)C2 8277,C1(C(N2CC3C(NC(c4cc5cn[nH]c5cn4)=O)(C3)C2)=O)CC2CCCC(C1)C2 8278,Cc1ccsc1C(=O)NCC1C=CC(NC(=O)C(O)CC2CCCC2)C1 8279,c1(CCOC)ccc(-c2nc(C3CCCC(Cn4cncn4)C3)n(CF)n2)cn1 8280,C(C(CC(F)(F)F)NC(C1(O)CC1)=O)NC(c1nc(CC(C)C)sc1)=O 8281,N1(C(C2(COC)CCCO2)=O)CCC(n2cc(C3CCCCC3O)nn2)CC1 8282,N1(C(CCN(CCC)C)=O)CC2CCC2(CC(=O)N(c2ccsc2)CC)C1 8283,c1(C(=O)OC)cncc(-n2cc(CONC(c3ccnnc3O)=O)nn2)c1 8284,N(C(=NCCC(C)SC)NCC(=O)OC(C)(C)C)C1CC(OCC)C12CCC2 8285,Cc1ccc(CCC(=O)NCC23CC(CO2)N(C(C2CCC(C)C2)=O)C3)cc1C 8286,C1(C#N)(C(=O)NCC(C)NC(C2N(C(C)=O)CCC2)=O)CCCOC1 8287,C1(CC(=O)N(CCC(C)C)C)C(NC(C2(Cl)CC2C(C)=O)=O)CC1O 8288,N1(C(c2n(CC#C)cnn2)=O)CCC(C)C1C(=O)NC(C)(C)C#CCC 8289,c1(CC)ccc(C)c(C(N2CCC(CCNC(C3SCC=C3C)=O)CC2)=O)c1 8290,c1(C(=O)NC2C(CNC(c3ccc(O)cc3)=O)C2)cccc(Cl)c1[N+](=O)[O-] 8291,C1(CC(=O)NC)CCCN1C(C1(C(=O)OC(C)(C)C)CCC1)=O 8292,c1(OC(F)F)ncc(CN2CCOCC2Cn2cccn2)cc1F 8293,N12CCC(C)C1C2=O.c1(NS(Cc2c(C)ccs2)(=O)=O)ccccc1SCCO 8294,Cc1cnc(-c2cn(CCNC(C3C4CC5C(C4=O)C35)=O)nn2)c(C)c1 8295,c1(C(N2CCC(CC)C2CNC(C2CC2(C)C)=O)=O)ccc(F)c(Cl)c1 8296,N1(C(c2cc(C3CC3)ccn2)=O)CC2OCCN(C(c3sccc3Cl)=O)C2C1 8297,N1(C(CCOCC)=O)CCC(O)C1C(=O)N(CC(C)(C)OC)C 8298,C(CC(CC)(CC)NC(c1ccnc(OC)c1)=O)NC(C(C)OCC=C)=O 8299,N1(C(c2ccc(CNC(C(CCCC)F)=O)o2)=O)CCC2(CCCOC2)C1 8300,c1(C(=O)NCC2(NC(c3ocnc3C3CC3)=O)CC2)cnc2c(c1)CCOC2 8301,C1(CNC(=O)NC(C(C)c2ccccc2)(C)C)CC(C)(C)CO1 8302,C12(CNC(C(c3ccn(C)n3)C)=O)CC(CCO1)N(C(=O)CN1CCSCC1)C2 8303,C(=O)(C(C(=O)N1CC2CCCC1C2c1cn(CCOC)nn1)C(C)(C)C)OCC 8304,c1(C(N(C2CCCC(NC(=O)CCc3cn(C)cn3)C2)C)=O)ccnc(CO)c1 8305,c1(C(=O)NCC2C3CN(C(CCC(=O)NCC)=O)C(C3)C2)csc2c1CCCC2 8306,N1(C(C2(OC)CC(C)C2)=O)CCN(C(=O)CCn2nc(C)cc2C)CC12CCC2 8307,C(=O)(CS(=O)(=O)NC(=O)CC1CCOCC1)NCC1(O)CN(CC)C1 8308,C1(CNC(CC2(C)CC2(Cl)Cl)=O)C2CN(C(c3ccc(N(C)C)nc3)=O)CC12 8309,N1(C(C2OCCN(C)C2=O)=O)CCC2(CCC2)C(NC(c2ncccn2)=O)C1 8310,c1(OC)c(C(N2CCCC(CNC(=O)C(O)P(C)(C)=O)C2)=O)cccc1Cl 8311,C1(C(=O)NC(c2ccc(O)nc2)C)CC(NC(C2(C)CNC(=O)C2)=O)C(O)C1 8312,c1(C(=O)NC2CCN(C(CCCCNC(N)=O)=O)C2)ccc(N)cc1C(F)(F)F 8313,C1(CNC(C(C)OCCC#C)=O)CN(C(=O)Cc2csnc2C)CCC1(F)F 8314,C(=O)(CC(C)(C)C#N)NC(C(C(C)C)NC(=O)CCc1ncc[nH]1)C 8315,N1(C(C(C(C)C)SC)=O)CC2(CCCN(C(=O)C(c3nc(C)cs3)C)C2)C1 8316,N1(C(COCCOCCOC)=O)CCOC(C(C)NC(c2ccnc(S)c2)=O)C1 8317,C1(NC(C(C)N(C(=O)CC2CCOC2)CCC)=O)CCc2n[nH]cc2C1 8318,C(=O)(CC(C)(C)CC(=O)NCC(F)CNC(c1ccc(C)nc1OC)=O)OCC 8319,N12CC3(CCN(C3)CC1=O)C2.c1(-n2ccc(C)n2)cccc(-c2nn[nH]n2)c1 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8338,CCCCC(CC)CC(=O)NCCCC(C)(C)C(=O)NCC(C)(O)COC 8339,c1(OC)cc(OC)cc(CC(=O)NCCCOCCN(C2COC(C)C2)C)c1 8340,c1(C(=O)NCC(C=C)(F)F)ccncc1-c1cccc(CNC(C)=O)c1 8341,c1(C(=O)NC(C2CCCN2C(=O)CSc2cnc[nH]2)C)ccc(C(F)(F)F)cn1 8342,CN1CCC2CN(C(C3CN(C(c4ccc(O)cc4O)=O)CCS3)=O)CC2C1 8343,c1(C(=O)NC2CC(C(=O)NC(CCCC)CO)OCC2)ccc(=NC)[nH]c1 8344,CCC(O)C(C)C(=O)NCCC1(OC)CN(C(C2CC2F)=O)C1 8345,CC1(C)Cc2[nH]nc(C(N3CCC(O)(CCNC(=O)C(F)C4CCC4)C3)=O)c2C1 8346,CCC(C(=O)NCCCCCN(C(=O)C(C)c1cccs1)C(C)C)C(C)C 8347,N1(C(=O)OC(C)(C)C)C(CCNC(c2c[nH]nc2C(F)(F)F)=O)COC1(C)C 8348,C1(C(N2C(COc3nn(C(C)(C)C)c(C4CC4)c3)CCC2)=O)CC(C2CCC2)C1 8349,C1(C(=O)NCc2nc(-c3cccc(C(F)(F)F)c3)no2)CCCCCCN1 8350,n1(CC)cc(C(=O)NCC2CC(NC(C3CC3C3CC3)=O)C2)c(C(C)C)n1 8351,c1(CC(=O)NCC2CC(NC(C(c3n(C)ncc3)(C)C)=O)C2)c(F)cccc1F 8352,c1(C(=O)NCCCCCN(C(C(COCC)C)=O)C)cc(OC)n(C)n1 8353,Cc1cc(C(=O)NC2CC(CCNC(C3(O)CCC(C)CC3)=O)C2)nc(C)n1 8354,c1(C(N2CC(O)(CNC(C3CC4CCC3O4)=O)C2)=O)cc2n(n1)CC1(CC1)C2 8355,N(C(=NCC(=C)C)NC1CC12CC2)C(C#C)CC.c1(C2NCC2)ccccc1 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8392,C=CCC(CC=C)C(=O)NCC1COCC1NC(C12CCC(CC1)CO2)=O 8393,c1(C(N(CC(N2C(CO)CC2C)=O)CC#C)=O)cncc(CO)c1 8394,c1(COCC)ccc(CO)o1.C1(=O)C(CNC2CCOC2c2cnn(CC)c2)N1 8395,C1(C(N2C(Cc3n(C)ncc3)CCC2)=O)C2COC(C)(C)OCC12 8396,C(=O)(C1CS(=O)(=O)c2ccccc21)N(CCN(C(C(CC)C#N)=O)C)C 8397,C1(=CCNC(C2CC=CCC2)=O)CCN(C(c2cccnc2C(F)(F)F)=O)CC1 8398,C(=O)(C1=C(Cl)CCOC1)NCC1C(C)CN(C(=O)C=Cc2cccn2C)C1 8399,C12(C(=O)NC3(CC(=O)NCC4(C5CCC5)CC4)CCC3)CCC(CC1)CO2 8400,c1(CNC(N(C2CCC2O)CC)=O)csc(C2CCCO2)n1 8401,C(C(O)C(=O)NCC1CCC1C(=O)NCCC1CCCCO1)=CC 8402,CC(C)CC(C)(O)c1cn(C2(C(=O)NCC3CCCC3(F)F)CC2)nn1 8403,N#CC1(C(=O)NCc2nc(C(N3CCC(C(F)F)CC3)=O)co2)CCCOC1 8404,C1(NC(Cc2c(C)cc(C)s2)=O)CCN(C(=O)CCC(C)(C)C)C(C)C1 8405,C(=O)(C1=CC2C=CC(C1)C2)NC(CC(C)C)C(=O)N1CC(CO)CC1CO 8406,c1(C(N2C3CCN(C(COCCCOC)=O)CC3C2)=O)cnc2c(c1)CCCO2 8407,CCCC(C(O)C(=O)NCCC(C)C(=O)OC)NC(C1CC1C(F)(F)F)=O 8408,Cc1noc(N)c1C(=O)NCC(C)C(=O)NC(c1cncc(F)c1)C 8409,c1(C(N2CCCC(CNC(C(C)OCC=C)=O)C2)=O)c(OC(F)F)cccc1Cl 8410,c1(N(CCC(N2CCOCC(N3CCCC3)C2)=O)C(C)=O)nc2ccccc2s1 8411,c1(C(=O)NC(CNC(C(C)SC)=O)C(C)C)cc(C)cc(O)n1 8412,N1(C(c2n(C)ccc2)=O)CC(OC)C2(CC2)C1.c1(CNC)nc(C(=O)O)cs1 8413,c1(OC)ccccc1C(C)C(=O)N(CC(C)CNC(c1nocc1C)=O)C 8414,N1(C(C(=O)N(C(C)CO)CC)C)CCC(C(=O)OC)CC1.c1(CSC)ccco1.N 8415,C(=O)(CS(=O)(=O)CCOC)N1CCNC(=O)NCC1.CCC(C)C(=O)C(=O)OCC 8416,N1(C(CCN(CCCCC)C(C)C)=O)CC(NC(=O)Cc2ccccc2)C(O)C1 8417,C1(n2cc(CNC(C3(Cl)C(C)(C)C3)=O)nn2)CCN(C(C2CCOC2=O)=O)CC1 8418,C12(NC(Cc3cn(CC)nn3)=O)CCCC1CN(C(C1(C(F)F)CCCO1)=O)C2 8419,C1(CC(=O)N(C(C)C(=O)NC(C(C)(C)CO)C2CC2)CCC)CCC(=O)NC1 8420,C1(CNC(C2CC3C=CC2C3)=O)CC2(CC2)CN1C(=O)COc1ccc(Cl)nc1 8421,Cc1cc(S(=O)(=O)NC(C(=O)O)c2cscn2)sc1C 8422,CCCCCC(F)C(=O)N1CC(OCC(=O)NCC(CC2CC2)CO)C1 8423,C(=O)(CC(C)P(C)(C)=O)N1C(C(C)NC(C2(N3CCCCC3=O)CC2)=O)CCC1 8424,O=S(=O)(N(CC(O)C1CC1)C1CC1)N1CCN(CC(F)(F)F)CC1 8425,N1(C(C)=O)CC(NC(=O)C(C(C)C)n2cnnc2Cc2nnc(C)o2)C(C)C1 8426,c1(C(=O)NC2(CC=C)CN(C(C3CCCCC3C)=O)C2)ccc2ccnn2c1 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8589,C12(C(=O)NC(C)C(CO)NC(c3cnco3)=O)C3C4C1C1C2C3C41C(N)=O 8590,c1(NC(CC(N)C23CC(C2)C3)=O)ccc2c(c1)OCCNC2 8591,Cc1cc(C(=O)NC2CCOCC2C(=O)NCCC2CC(C)(C)C2)nnc1C 8592,c1(N2CCN(C(=O)CC3C=CS(=O)(=O)C3)CC(O)C2)ncc([N+](=O)[O-])cc1F 8593,CC1CN(C(C2(C)CCCOC2)=O)CCC1CNC(=O)C1=CCSC1 8594,C1(CC)CN(C(c2cc(Cl)ccn2)=O)CCC1NC(C1CC(=O)N(CC)C1)=O 8595,C1(NC(C(C)SC)=O)CN(C(=O)C(C)CC2CCC2)CC(F)(F)C1 8596,CC(CS(C)(=O)=O)C(=O)N1CCC(NC(c2ccn(CCO)c(=O)c2)=O)C12CC2 8597,CCC(CNC(=O)CN(CC(C)C)C(=O)C=CC1CCCC1)C(C)C 8598,C(=O)(C1CSc2ccccc21)N(C1CN(C(=O)CCCn2cccc2)C1)C 8599,N1(C(Cn2nc(C)oc2=O)=O)CCc2sccc2C1CNC(C1CC12CCC2)=O 8600,N1(C(CN(C)C(c2ncccc2N)=O)=O)CCC2CC2C1 8601,CCCCCCN=c1cc(N(C)Cc2ccc(-c3ccncc3)cc2)nc(C)[nH]1 8602,c1(C(=O)NC(c2cccc(Cl)c2)CNC(CSCCC)=O)ccc(C)nc1OC 8603,C1(CNC(CN(C2CCC2)C(C2C(C)CCOC2)=O)=O)CC2(CCO1)CC2 8604,CCCCCC(CC)C(=O)N(CC(O)CN(C(=O)Cc1nc[nH]n1)C)C 8605,C1(NC(CCC(=O)OC)=O)CN(C(c2cc(Cl)ccc2C)=O)CC1C#N 8606,Cc1cn2cc(C(=O)NC3CCC(NC(C4CSCCS4)=O)CC3)ccc2n1 8607,c1(C(N2CC3C(CNC(c4cc(CCC)[nH]n4)=O)C3C2)=O)nc(C)ncc1Br 8608,N1(C(C(CCCC)F)=O)CCC2(CC1)CC2C(=O)NCC(C)(C)OCCO 8609,c1(CN(c2nc(C)c(F)cn2)C2CNC2)ccc2nn(C)cc2c1 8610,C(C)(CC(=O)NC1(C)CC(C(=O)NCC2(CN(C)C)CCC2)C1)OC 8611,c1(C(=O)NCCCOCCNC(C(C)O)=O)cncc2c(O)nccc12 8612,C1(C(N2CC(O)C2)=O)(NC(C=CCN(C)CC)=O)CCSC1 8613,C(C(C)(C)CNC(C1CCC(=O)O1)=O)NC(C1C(COC)C1)=O 8614,C#CC(CNC(=O)CSCCNC(c1cc(F)c[nH]1)=O)CC1CC1 8615,c1(CC)[nH]nc(C(=O)NC(c2cn(Cc3ccncc3NC)nn2)C)c1F 8616,C(=O)(CCCCCCCCS(C)(=O)=O)NCC=C1CCN(C(CCC#C)=O)CC1 8617,N1(C(C2CC(=O)NC2)=O)CCC(O)(CNC(C2CCC3CC23)=O)CC1 8618,C(=O)(C(Cc1cn[nH]c1)NC(=O)CN1CCCC1)N(C)CCc1cccs1 8619,N1(C(CN2CC(=O)N(C)C2=O)=O)CC2CC1CN(C(=O)CCC(F)F)C2 8620,c1(CN2CCOCC(NC(C(CCC)O)=O)C2)cc(F)c(Cl)cc1O 8621,c1(C(N2CC3CCCC(C2)N3C(c2cccs2)=O)=O)cc2c(cn1)OCCO2 8622,c1(CCC(N2CC(CNC(CCOCCN(C)C)=O)C2)=O)sccc1Br 8623,CCCC(C(=O)OC)C(=O)N1CCC(C)(NC(c2oc(C(F)F)cc2C)=O)C1 8624,C1(CNC(c2c(C)cno2)=O)CCC2(CCC2)CN1C(=O)CCC1CC1(F)F 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8643,c1(N(C)Cc2ccc(OC)c(OC)c2)ncnc2c1nnn2CC#N 8644,n1(CC)cc(Cl)c(C(N2CC(NC(c3cccnc3O)=O)C(SC)C2)=O)n1 8645,CC1CCCC1(c1nnnn1C)NCCc1cnc(Cc2ccccc2)s1 8646,O=S(=O)(c1cc2ccccc2s1)NCC1(O)CCCN(Cc2ncccc2Cl)C1 8647,C1(NC(c2ccc(COC)o2)=O)CN(C(=O)C(=O)NCCC(N)=O)C2CCCC12 8648,C(c1ccc(F)c(F)c1)=CC(=O)N(CC(C)NC(=O)C1=CS(=O)CCC1)C 8649,CC(C)(F)C(=O)NC1COCC1C(=O)NCC[Si](C)(C)C 8650,CCCC(C)CC(=O)NCCCCC(C)NC(c1ccn(C(C)C)n1)=O 8651,C1(CCC(=O)NCC(CSC)OC)CCCCN1C(=O)CCCC1CC1 8652,Cc1cnc(NCCc2ncccc2C)c(S(=O)(=O)NCC2CCSC(C)C2)c1 8653,n1(CC(=O)NC2C(C)CCN(C(C34CCC(C3)C4)=O)C2)ccc(=O)c([N+](=O)[O-])c1 8654,C1(CNC(c2ccc(Cl)cc2)=O)CN(Cc2cc(Br)no2)CCO1 8655,S(=O)(=O)(c1ccc2nc(O)oc2c1)N1CCCN(C(C#CC)=O)CC1 8656,C(CCC(C)(C)C)NC(c1c(CNC(C(C)=C(C)C)=O)n[nH]c1)=O 8657,Cc1ccc(C(=O)NC2CC3CC2N(C(=O)CN2CCC(C)CC2)C3)c(O)n1 8658,N1(C(C(C)C2CC2)=O)CCCC2(NC(c3cncc(F)c3)=O)CC2C1 8659,c1(C(C)=O)c(C)[nH]c(C(=O)NCC2(O)CC(NC(=O)CCC3CC3)C2)c1C 8660,N1(C(=O)Nc2cccc(-c3c(Cl)cc(C)c(F)c3)c2)CCc2c(O)noc2C1 8661,c1(C(N2CC(F)(CNC(c3ccc(CO)o3)=O)C2)=O)cc(F)c(Br)cc1F 8662,N1(C(C(C(COCC)C)C)=O)CCc2sc(CNC(=O)COC(C)C)nc2C1 8663,CN1CCOCC1C(=O)NC1CC(NC(c2cnn(CCF)c2)=O)CC1O 8664,c1(C(=O)NCCCOCCN(C(COC(C)=O)=O)C)coc(-c2ccccc2)c1 8665,C1(C(N2C(CCNC(COC)=O)CCC2)=O)CCC(F)(F)CC1 8666,C#CCCCC(C)C(=O)NCC(C(=O)NC1CC(O)C(F)C1)N(C)C 8667,CCCS(=O)(=O)CC(=O)NCCCC(C)NC(C1(CC)CCOCC1)=O 8668,c1(CN2CCC(CC(=O)Nc3c(OC)ccnc3)C2)ccnc(Cl)c1Cl 8669,C(CCN=c1[nH]c2cc(Br)cnc2s1)N(C(CC(C)C1CC1)=O)CC1CCCC1 8670,C1(C(C)=O)CC(CC(N2CCN(C(=O)C(F)=C3CCC3)CC2)=O)C1(C)C 8671,C1(CNC(Cc2c(SC)cccc2)=O)CCC2(CN(C(=O)CC3CN(C)C3)C2)O1 8672,CC(C)(C)CC(O)C(=O)NC(CCOCCO)C(N1C2CCC1CC(O)C2)=O 8673,C1(NC(=O)CC2CCS(=O)(=O)C2)CC2(C1)CC(CNC(=O)NCC1CCCC1)C2 8674,N1(C(CCNC(C)=O)=O)CCCC2(C1)CN(C(C1C(C#N)C1(C)C)=O)C2 8675,C12(CNC(c3cc(C)sc3)=O)CCC(CC1)N(C(C1CC1C1CCCO1)=O)C2 8676,C(=O)(CS(=O)C(F)(F)F)N(CC(C)N(C(CNC(C)=O)=O)C)C 8677,C(N=c1[nH]c(=NCCCc2nccs2)[nH]c2cccc(F)c12)c1cc(CC)on1 8678,n1(CC(=O)NCC#CCNC(C2(C)CCOCC2)=O)cnc([N+](=O)[O-])c1 8679,C1(C(=O)NCC2(COC)CN(C(c3ccco3)=O)C2)C2CCCCC12 8680,C1(C(N2CCC(C)(CNC(c3cnc(NC(C)=O)s3)=O)C2)=O)CC(C)CC(C)C1 8681,N1(C(COCCCC(C)C)=O)Cc2nccn2CC(NC(=O)C2CC2)C1 8682,C12(CNC(C(C)SC)=O)CC(NC(=O)C(C)Sc3ccc(Cl)cc3)(C1)C(C)O2 8683,C(=O)(C1CCc2c[nH]nc21)NC1CC2CN(C(c3cc(C)[nH]n3)=O)CC1C2 8684,N1(C(CC=CC=C)=O)CC2COCCC2(NC(c2ccc3c(c2)CCC3=O)=O)C1 8685,C1(NC(C2=C(C)OCC2)=O)CC12CCN(C(=O)Cc1ccc([N+](=O)[O-])cc1)CC2 8686,Cc1cc(C(N2C3CCC2CC(CNC(=O)Cc2cnc[nH]2)C3)=O)c(F)cc1F 8687,N1(C(C=CC)=O)CCN(CCSCC)C(C)CC1C.c12ccc(Cl)cc1N2 8688,C(C(=O)N=c1ccn(CC2CC2)[nH]1)C1CN(C(CCCCC=CC)=O)CC12CC2 8689,N1(C(c2c(CC)cccn2)=O)CCN(C(c2cccc(N)c2C(F)F)=O)CC1C 8690,C1(C(N(C2CCC2)CC#C)=O)CC2CCC(C1)N2C(=O)Cc1ccon1 8691,c1(C(=O)NCC(CC=C)NC(=O)C(n2ccnc2C)C)nc(C)ccc1OC 8692,c1(C(=O)NC2C(C(=O)NC(c3cnc[nH]3)C)COC2)cnn(C)c1Cl 8693,CC1=C(C(=O)NCC2CCCCN2C(c2cccc3nonc23)=O)CCCC1 8694,c1(C(=O)NC23CC(CNC(C4C(OC)CCC4)=O)(C2)C3)nnc(S)n1C 8695,C1(Oc2c(C)cc(N)cc2)(NC(CCCO)C)CCCS(=O)(=O)C1 8696,C#CCCCCCC(=O)NCC1(CNC(C2CC2=C)=O)CC1(F)F 8697,C12(C(N3CCC(C(C)NC(C4COC(=O)N4)=O)CC3)=O)CCC(CO)(CC1)CC2 8698,c1(C(N2CCC(NC(C(C=CCCC)O)=O)C(O)C2)=O)cnc2n1CCOC2 8699,O=S(=O)(c1ccc2c(c1)CC2)NC1CCc2ccccc21.c1(O)ccc(Cl)c(Cl)c1 8700,N1(C(c2c(C)ccs2)=O)CC(NC(c2cncc(N)c2)=O)C(c2ccnn2C)C1 8701,c1(CN2C(C(N(C3CC3)CC)=O)CC3(CC3)C2)cc(OC)c(O)c(Br)c1 8702,c1(OC)ccc(C(=O)NC(C)CC(C)NC(c2cncnc2)=O)cc1C(F)F 8703,N1(C(C(C)=CC)=O)CCC2(NC(=O)CC3CS(=O)(=O)C3)CCCCCC12 8704,N(C(=NCCOC)NCc1ncccc1NC(=O)OC(C)(C)C)CCOCC 8705,C1(NCc2[nH]c(=N)sc2)CCCCC1C(=O)NCc1ccccc1N1CCCC1 8706,N1(C(=O)NCCC(=O)OCC)CCC2CN(C(=O)Nc3ccc(F)c(Cl)c3)CC12 8707,C12(NC(C3N(CC)CC3)=O)CC(C1)N(C(=O)CCn1cc(Cl)cn1)C2 8708,C1(NC(c2ccc(SC)s2)=O)CC2CC(NC(=O)C=Cc3cc[nH]n3)CC2C1 8709,c1(-n2cc(C(N(C(C)CCNC(C3CC(C#N)C3)=O)C)=O)nn2)ccccc1Cl 8710,c1(OC)cnc(C(N2CCCCC2CCCNC(=O)Cc2c[nH]nc2C)=O)cn1 8711,C1(NC(COCC=C)=O)CN(C(C2CCCC(=O)N2C)=O)CCC12CCC2 8712,C1(C2CCCN(C(C3CC(F)C3)=O)C2)(NC(C(C)NC(=O)CC(C)(C)C)=O)CC1 8713,c1(C(=O)NCCC(C)N(C(c2occ(C)c2)=O)C)ccc(=NCC2CC2)[nH]c1 8714,c1(OCCN(C)C)ccccc1C(=O)NC1C2CC1N(C(=O)CN1CCCC1)C2 8715,c1(OC)ccc(C(N2CCC(CN(C(=O)Cc3cscc3F)C)C2)=O)c(O)c1 8716,C=C1CCC(C(N2CCCCC2C(=O)NC(C)C)=O)CC1 8717,C1(NC(CCN(CC(=O)OC(C)(C)C)C)=O)CC(SCc2cccs2)C1 8718,C1(C(=O)NCCN(C2CCCCCC2)C(=O)CN2CC=CC2)CC2CCC(C1)O2 8719,N1(C(C23N(C(C(C(=O)OC)C)=O)CC(C)(C2)C3)=O)CCC2(CC1)CSC2 8720,c1(OC(C(=O)NC(C)CNC(C2CC(CF)C2)=O)C)ccc2c(c1)CCCC2 8721,N1(C(CC(C)(C)n2cc(C(n3cccc3)(C)C)nn2)=O)Cc2ccccc2C1 8722,c1(OC)cc(C(=O)NCCC(O)CNC(=O)C(C)(C)C)ccc1[N+](=O)[O-] 8723,C(=O)(C1=CS(=O)CCC1)N1CC(C(=O)NCCSc2cocn2)C1 8724,CC(N=c1cccc(S(=O)(=O)NCCC23CCCC2C3)[nH]1)c1cnsc1 8725,C1(O)(CNC(CC=C(C)C)=O)CCN(C(=O)C(C#N)C2CC2)CC1 8726,N1(c2nnc(-c3nnn(C)n3)n2C)CCc2cc(F)cc(F)c2C1.c1(CCC)ccccc1S(C)(=O)=O 8727,N1(C(CNC(=O)C2CC2)=O)CCN(C(=O)C(O)C2CC2)CC2(CC2)C1 8728,C(CN=c1[nH]c2c(c(=NC(C)c3cn(C)nc3C)[nH]1)CCC2)(C1CCCC1)OC 8729,c1(C(N(CCn2cc(C(N(C(C)C)C)C3CC3)nn2)C)=O)c([N+](=O)[O-])cnn1C.CCS 8730,N1(Cc2cn(C(C)CNC(=O)CSC3(C)CCCCC3)nn2)CCS(=O)(=O)CC1 8731,c1(CCC)noc(CCC(=O)NC2CCCC2NC(C2CC2C)=O)n1 8732,N1(C(C=C2CCN(C)C2)=O)CC2CC(C1)CN(C(C1CC(=O)N(C3CC3)C1)=O)C2 8733,C(N=c1nc2ncn(C)c2c(NCC2(CO)CCCO2)[nH]1)c1nnn(CC)n1 8734,c1(SCn2cc(C3N(C(CC(COC)C)=O)CC=C3)nn2)cn(C)c(C)cc1=O 8735,c1(C(N(C(C)CN(C)C(C2CCOC2)=O)C)=O)cc2c(nn1)OCCS2 8736,c1(C(N2CCC(NC(=O)CC3(C(F)(F)F)CC3)C2)=O)cc(-n2ccnc2)ccn1 8737,c1(C(=O)NCC(CNC(C2C(=C)C2)=O)O)cc2cc(Br)ccc2c(OC)n1 8738,C1(NC(c2cccc(CC)c2)=O)CCCN(C(=O)CSc2cnn(C)c2)C1CC 8739,c1(CNC(CSCC=C)=O)ncoc1C1CN(C(=O)CCOC(C)CC(C)C)C1 8740,C1(NC(=O)CN2CC=CC2)COC2(CCN(C(C3CC34CCSCC4)=O)CC2)C1 8741,CC(C)C(O)C(=O)NC(C1CCCCN1C(=O)CNC=O)C 8742,Cc1ccc(F)c(C(=O)NCC(C)CN(C)C(C23CCC(C2)OC3C)=O)c1 8743,c1(C(=O)NC2CCC(N(C(c3ccc(OC)nn3)=O)C)C2)cc(F)c(F)cc1Cl 8744,c1(OC)ccc(C(N2CCN(C(C3CCC(OCCC(C)C)C3)=O)CC2)=O)cc1 8745,Cc1nc(O)c(Br)cc1C(=O)NCCC(C)NC(=O)Cc1ccc(O)nc1 8746,C(=O)(C(F)(CC)C(=O)OC)NCC1C(NC(c2c(CC)occ2C)=O)CC1 8747,c1(SC)ccc(C(=O)NCC(C(C)C)NC(=O)Cc2cnc(C)[nH]2)c(Cl)c1 8748,N1(C(c2nc(CC)sc2)C(=O)NCc2nnn(C)n2)CCOC(C2(C)N=N2)C1 8749,CCCCC(CNC(=O)C(C1CCOC1)OC)NC(=O)CSC(C)(C)C 8750,N1(C(C2CC(SC)C2)=O)CC=C(CNC(=O)CCNC(=O)CC(C)C)CC1 8751,c1(NC2CCN(C(C=CCC)=O)CC2CC)c(Cl)cccc1[N+](=O)[O-] 8752,c1(N2CCCC(OCCCOC)C2)nc(=N)[nH]c(=NCC(=O)NC2CCC2)[nH]1 8753,Cc1sncc1C(=O)N(C(C)CCNC(=O)CC1(C)CC1)C 8754,N1(C(C2=CCN(C(C3CN(C)C(=O)CC3)=O)C2)=O)CC2(C1)NC(=O)NC2=O 8755,c1(C(=O)NCC(C)(O)CNC(=O)Cn2ccsc2=N)ccc2c(c1)CCCO2 8756,c1(N2CC(CC)SCC2)nc(=NCC(C)C(C)(C)C)[nH]c2c1CSC2 8757,Cc1nnccc1C(N1CC2CC1C2C(=O)NCCc1ccncc1)=O 8758,c1(C(=O)NC2CC(CNC(=O)C3=COCCO3)CC2O)nsc2c(Cl)cccc12 8759,C1(NC(=O)C2CC2)COCCN1CCNC(C1C(C)(CC)C1)=O 8760,c1(CC(=O)NCC(C(C)C)NC(C2CC(N(C)C)C2)=O)ccc(Cl)nc1 8761,c1(NCCCN(c2ccccc2Cl)CC)cc(Cl)nn(C)c1=O 8762,Cc1ccnc(C(=O)NC2(C3CCCN3C(C3CCCN3C)=O)CC2)c1 8763,C(=O)(C1=NNC(=O)CC1)N(CC(=O)NCCCn1c(C)ncc1)CC(C)C 8764,N1(C(c2ncc(OC)s2)C(=O)NC)CCC(c2nccs2)CC1 8765,CCC(CC(F)F)C(=O)NCC(C)CNC(c1c[nH]c(=N)o1)=O 8766,CC(O)CCCCCC(=O)N1CCC(C(=O)NOC2CC3CCC2C3)C(C)C1 8767,CC(C)CCC(N)C(=O)NCC(c1ccco1)N1CCCC1 8768,C#CCCC(O)C(=O)N1CCCC1C(C)NC(=O)CCc1cncn1C 8769,C1(NC(C(C(C)C)c2cccnc2)=O)CN(C(=O)Cc2cccs2)CC12CCC2 8770,C1(C(N(CC(C)(C)NC(c2c(CC)nco2)=O)C)=O)CCCCC1(F)F 8771,C1(CNC(=O)Cn2cnnn2)CN(C(c2cccc(-c3nc[nH]n3)c2)=O)CCO1 8772,C(=O)(CC1=CCCC1)NCC(CC)NC(c1ccccc1NC(C)(C)C)=O.C(N)(=O)N 8773,C1(CC)(CNC(C2OCCC2NC(=O)OC(C)(C)C)=O)CCCO1 8774,CC(C)(C)C(O)CC(=O)N1CC(CNC(c2ccc(C(F)(F)F)[nH]2)=O)C1 8775,C(=O)(C1Cc2c(Cl)cccc21)N(C1CCCN(C(c2nnc(CC)o2)C)CC1)C 8776,C1(NC(c2c(CCC)nns2)=O)CCCCCC1NC(=O)C(C)(C(C)C)OC 8777,CN1CCCCC1CC(N1CC(C(=O)NOCCc2ccccc2)(CO)C1)=O 8778,C1(NC(NCc2nc(C3CC3)n[nH]2)=NCc2c(C)cccc2)CC(C)OC(C)C1 8779,c1(C(N(CCNC(C2(C)CCN(C)C2)=O)CC)=O)c(Cl)ccc(O)c1N 8780,Cc1cc(F)ccc1CC(=O)NCCC(C)N(C)C(c1cccc(F)c1O)=O 8781,Cc1ccn(C(C)(C)C(=O)NC2(C)CC(NC(=O)C(C3CCCOC3)OC)C2)n1 8782,c1(C(=O)NCCN(C(=O)CC2CC3CCC(C2)C3)CC)nc(C)ccc1OC 8783,c1(C(=O)NC2C(C(N3C(C(=O)OC)CC3)=O)OCC2)cccc(F)c1O 8784,Cc1cnc(NCc2c(C)cccc2C)c(S(=O)(=O)N2CCC(C3CCC3)C2)c1 8785,C1(C(N(C)CC2CN(C)C2)=O)CN(C(=O)C(C2(O)CCCC2)F)CCO1 8786,N1(C(C2C(C)(C)C2(F)F)=O)CC2(C1)C(NC(C1(n3cncn3)CC1)=O)CCS2(=O)=O 8787,C1(C(=O)NC(C(N2CCCC(OCC)C2)=O)C)CCC2(CCC2)C1 8788,N1(C(C2C(C(N)=O)COC2)=O)CC(F)CC1CNC(=O)OCC1CCOCC1 8789,C(=O)(C1SCCc2ccccc21)N1CC(C(C)NC(=O)CC2(C)CC2)C1 8790,C1(N(C(=O)CCCCC2CC2)C)CCCN(C(c2cccc(F)c2N)=O)CC1 8791,c1(C(N2CC3C(CNC(C(C)c4cccs4)=O)C3C2)=O)coc2cccc(O)c12 8792,c1(C(N2CCCC3(NC(C=CCCC)=O)C(C2)C3)=O)cc2c(cc1O)CCCC2 8793,CC(C)C(O)C(C)C(=O)NCC12CC1CN(C(=O)Cc1cnn(C)c1)C2 8794,c1(C(N(CC(=O)N(C(C(N)=O)C2CC2)C)CCC)=O)ccc(N)cn1 8795,C1(c2cn(C3C(NC(c4cn(CCC)nn4)=O)CCC3)nn2)(OC)CCCOC1 8796,N1(CCN(C(=O)CCN2CCOCC2)C)CCN(C(C2(C)CCCC2O)=O)CC1 8797,c1(C(=O)NC(C2OCCN(C(C(C=C)CC)=O)C2)C)cc(N)cc(F)c1 8798,Cc1ncc(NC(C2CC(C)(NC(=O)CC3COCCO3)C2)=O)c(C)c1C 8799,c1(CC(=O)NC2C(C)CN(C(=O)C3=CCSC3)C2)cccc2cnccc12 8800,c1(C(=O)NCCOCCOCCNC(C2(O)CCOC2)=O)ccc2c(c1)CCO2 8801,C1(CNC(c2n(CC)c(O)nc2)=O)CN(C(C2CCCCC2)=O)CC2(CCC2)O1 8802,c1(C(=O)NCCC(CNC(C2(CN(C)C)CC2)=O)O)cccc2ccn(C)c12 8803,N1(C(c2c(C)cno2)=O)CCCCC(CNC(=O)Cc2cn(C)nc2C)C1 8804,c1(C(N2C(CC(=O)Nc3c(C)cnc(Cl)c3)CCC2)=O)ccc2ncccc2c1 8805,C(=O)(C(O)CCC(F)(F)F)NCC1CC(NC(CC(=O)NCC)=O)C1(C)C 8806,C1(C(=O)NC(c2c(C)cccn2)C)CC2(CC(NC(=O)Cn3nccn3)C2)C1 8807,C(CCF)(C(=O)N1CCCC1C)NC(CCOC(C)=O)=O 8808,Cc1nc(C2CCN(C(=O)NC3COC(C)C3)CC2)nc2c1CCCC2 8809,C1(CC)CCCN(C(=O)CC(C)(C)C2CC2)C1C(N1CC2(CC2)CC1CO)=O 8810,Cc1onc(CN2CCCC2)c1C(=O)NCC1CCN1C(C1CC(C)(CO)C1)=O 8811,C1(C(=O)NC2CN(C(c3ccc(CC)s3)=O)CC2C)CCC2(CCCC2)CC1 8812,C1(C(C)C)CCCC(C(=O)N(C)CCN(C)C(c2cc(O)nn2C)=O)C1 8813,C(=O)(C1Cc2c(Cl)cccc21)NCCN(C)C(c1cnc(CCC(F)(F)F)s1)=O 8814,c1(C(N2CC(CNC(C(C)(C)OCC)=O)CC2(C)C)=O)ccnc2[nH]ncc12 8815,c1(C(N(CCC)CCNC(C2CC2(F)Cl)=O)=O)nc(C)c(C)nc1C 8816,N1(C(C(C)(C)C2CCCO2)=O)CCC(O)(CNC(=O)CC2CSC2)C1 8817,CC(C)CC(C)(CO)NC(=O)C(C)C(C)NC(c1c[nH]nc1C(C)C)=O 8818,N1(C(CCSc2n(C)nnn2)=O)CCN(C(C2(C)COC2)=O)CC1CCO 8819,N1(C(C=C(C(=O)N(CCC)CCC)F)=O)CCC(C)C1CSC 8820,c1(C(N(CCCC(=O)NC2CCSCC2)C)=O)ccc2[nH]nc(Cl)c2c1 8821,N1(C(C)=O)CCC(N(C)C)CC1.N12CCCCC1c1nnc(o1)CS2(=O)=O 8822,c1(C(N2CC3C(CNC(c4cc(C)oc4)=O)(C3)C2)=O)cc([N+](=O)[O-])oc1C 8823,c1(C(C(=O)NC(C)(C)CC)N(C(C#C)C2CCC2)C)cnc(C)nc1 8824,C12(C(=O)NC3(C)CN(C(=O)CC4(O)CCOCC4)C3)CCCC1(C(=O)NC1CC1)C2 8825,N1(Cc2cccc(C(=O)NCC(C)C#N)c2)C(=O)CN(C)C1=O 8826,c1(C(=O)NC(CC(=O)NC(CCCC)C)CC2CC2)cccc(C)c1F 8827,c1(C(N2CCC(NC(c3cnc(C)nc3)=O)C2C)=O)cc2c(Cl)cccc2[nH]1 8828,C1(NC(COCCC)=O)CC2CCC(C1C)N2C(c1cc(C)n(CC)n1)=O 8829,C(C(=O)NOCC1CC1)C(C)(C)CNC(C1COCC1C(N)=O)=O 8830,C(C1CCCN1C(c1cc(F)c[nH]1)=O)=CC(=O)NCC1(CC(N)=O)CC1 8831,C(=O)(CC(C)CC(=O)OC)NC(CC)(CN(C(=O)C#CC(C)(C)C)C1CC1)CC 8832,n1(CCC)ccnc1C(F)(F)C(=O)N1CC(NC(=O)C(F)CN(CC)CC)C1 8833,c1(C(=O)NC2(C)CC(NC(COCCN(C)C)=O)C2)cc(O)nc(Cl)c1 8834,C(C(=O)N1OC2CCC1CC2)(C1C(C)=NNC1=O)NC(c1ccc(C)c(O)c1)=O 8835,Cc1cccc(F)c1C(=O)NCCNC(=O)C(C)(C)N(S(C)(=O)=O)C.C12CC1N2 8836,C1(O)(C(=O)NCC=C=C)CCN(CC(C)CO)CC1 8837,c1(NCc2scc(CC)c2)ccc(SC)cc1.C1(C)C(=O)N1C(C)C 8838,C(=O)(C(F)CC(C)(C)NC(c1ncccc1O)=O)NC(CC)C(C)C 8839,C1(C(N2CCN(C(C)=O)CC2c2cnn(C)c2)=O)CCc2cnc(C)n2C1 8840,C(=O)(C1=Cc2ccccc2C1)NCC1(C)CN(C(c2cnc(O)s2)=O)CCO1 8841,C1(C(N(CCCNc2cnn(CO)c2)C)=O)C=CCC(CC(=O)N)C1.C(C)(C)(C)O 8842,c1(C(=O)NC2CN(C(C=COCC)=O)CC(O)C2)[nH]c2c(c1C)CCCC2 8843,C=CC(C)(C)CC(=O)N1CCN(C(c2[nH]ccc2C2CC2)=O)CC1CF 8844,c1(C(=O)NCCCN(C(COCC(=O)NC)=O)C(C)C)cscc1SC 8845,C1(CN(C)C(c2cnn(CC(F)F)n2)=O)COCCN1C(=O)CC(Cl)Cl 8846,Cc1cc(C(N2CC(NC(c3cc(C(=O)C(F)(F)F)c[nH]3)=O)C2)=O)nn1C1CC1 8847,c1(NC2C(F)CCN(C(c3ccc(OC)c(C)c3)=O)C2)ncc2sccc2n1 8848,Nc1nc(C(N2CCC(CCNC(C3CCCCC3)=O)C2)=O)ccc1[N+](=O)[O-] 8849,C(=O)(C(CC(C)C)NC(C1CC1OC(C)=O)=O)NCC(C(=O)OCC)(F)F 8850,c1(C(N2C(C(=O)NCC34CC(CCO3)C4)CC2)=O)coc2ccccc12 8851,n1(CC)ccc(C(=O)NCC2(F)CCN(C(=O)C(c3ccnn3C)O)C2)cc1=O 8852,Cc1cc(C(N2CCCCC2CNC(=O)C(C)(C)C2CC2)=O)cc([N+](=O)[O-])c1Cl 8853,c1(OC)ccc2cc(CN3CCC4CN(C(c5ccco5)=O)CC34)c(O)nc2c1 8854,C1(CN(C(CNC(CC)=O)=O)C)CCN(C(c2coc(C(C)C)n2)=O)C1 8855,C(=O)(C1CSc2ccccc21)NC1CCC(CNC(c2ncncc2F)=O)CC1 8856,c1(C(CNC(c2cnc(CC)s2)=O)NC(C2CCN(C)C2)=O)ccc(F)cc1F 8857,n1(CC)ccc(=NC(=O)C2C3CC4C(C3NC(c3sc(F)cc3C)=O)C24)[nH]1 8858,Nc1ccc([N+](=O)[O-])c(C(N2CCCCC(NC(=O)CC3CCCO3)C2)=O)c1 8859,N1(C(C2C(C(=O)OCC)CC2)=O)CCN(C(=O)CCc2n[nH]c(=N)s2)CC1C 8860,C1(C(=O)NC(CNC(CCOCC#C)=O)C)CNC(=O)CC1C 8861,n1(CC)nnc(C(N2CCC2CNC(=O)CNc2nccs2)=O)c1C 8862,c1(NC(=O)Nc2c(OC)ccc(SCC)c2)c(C)cccc1C#N 8863,C(=O)(C(CC)C(=O)N1CC(C(=O)NCC2CC3(CC(OC)C3)C2)(OC)C1)OCC 8864,CC1CN(C(=O)CCCC#N)CC(C)N(C(c2cc3sccc3[nH]2)=O)C1 8865,C1(C2CCCN(C(c3ccsc3S(C)(=O)=O)=O)C2)(NC(CC(C)OC)=O)CC1 8866,CN1CCN(C(C2C=CC=CC=C2)=O)CC1C(N1CCC2CC12)=O 8867,C(=O)(CCCCCSC)NC(C1CCOCC1)C(=O)N(CCCCO)CC 8868,C1(NC(CCC(CC)OC)=O)(CNC(C2CCCN2N=O)=O)CCC(F)(F)CC1 8869,c1(C(N2CCN(C(c3[nH]cc(C#N)c3)=O)CC2CCO)=O)nccc2nn[nH]c12 8870,c1(C(=O)NC2C(CNC(c3c(C)nns3)=O)CCC2)ccc(F)c(F)c1N 8871,C1(NC(C=CCCC)=O)CCCN(C(C2CC3(CSC3)C2)=O)C1 8872,C1(NC(C(C)Cc2ccc(F)cc2)=O)CC2CC(NC(c3ccsc3)=O)C2C1 8873,C1(CNC(C(CC=C)CC)=O)CN(C(=O)CCC(=O)OCC)C2COCC2O1 8874,C1(NC(CC(C)C)=O)CCCC(NC(=O)CC2CCC(=O)C2C)C1 8875,c1(NC(C)=O)ccc(F)c(C(N2CCC(C)(NC(C3CC(=C(F)F)C3)=O)C2)=O)c1 8876,c1(C(N2C(C(=O)NC3COCC3O)CSCC2)=O)ccc2sccc2c1O 8877,C1(CNC(CNC(=O)OC)=O)N(C(=O)CCCC(C)(F)F)CCCC1(C)C 8878,C1(COCC(=O)NCC2(OCC)CC2)CCCC1 8879,C1(C(=O)NC(C)C2CC2)CCN(C(=O)C2=NOCC2)C(C)(C)C1 8880,c1(C(=O)NCC2CC(CNC(C(C)(C)C(N)=O)=O)OC2)c[nH]nc1S(N)(=O)=O 8881,c1(C(CCC)C)nc(-c2cc(C(F)(F)F)ns2)n(Cc2cncc(F)c2)n1 8882,N1(C(C(C)=C(CC)C)=O)CC(C(=O)NCCC2(C)CC2(F)F)C(C(C)C)C1 8883,C1(NC(NCc2sccc2)=NCC2CCCO2)CCCC12CCC2 8884,C(C(C)(C)C#CC(=O)NC(C)CN(C)C(C)C)NC(Cc1ccc(OC)cc1)=O 8885,O=C1OC(C(=O)NCC2CCN2C(=O)Cc2cn[nH]c2)Cc2ccc(Cl)cc21 8886,Cc1ccc(C)c(CC(=O)N(C(CNC(c2cncc(C)c2C)=O)C2CC2)C)c1 8887,c1(C(=O)NC2C(C(=O)OC)CCCC2)c(C(F)(F)F)oc2ccccc12 8888,N1(C(=O)CCOC2CC2)CC(S(=O)(=O)N2CCN(C(C3CCCSC3)=O)CC2)C1 8889,C1(CC(=O)N(CCC(=O)NCC(c2ccsc2)C)CC#C)CCCC(=O)N1 8890,S(=O)(=O)(c1ccc([N+](=O)[O-])cc1OC)N1CC(C(=O)OC)C(N)C1 8891,C(C(C(C)(C)C)NC(c1c[nH]nc1C1CCOCC1)=O)NC(CC1(C)CC1)=O 8892,c1(CCC(=O)N(CC(C)NC(C2CC2(Br)Br)=O)C)cncnc1 8893,c1(CN2C(C(N3CC(F)(F)C3)=O)CNCC2)ccc(Br)c(O)c1 8894,N1(C(C2C(OCC)CC2)=O)CCC(CNC(=O)C(CN(C)C)CC)C(C)(C)C1 8895,C(=O)(C(CO)C(C)(C)C)N(CC(C(N1C2(CC(COC)C2)CC1)=O)C)C 8896,N1(C(C=CCC)=O)CCC(CC)C1C(=O)N(CC1CC1)OC 8897,CCCC(C(=O)NCCn1cc(C(N2CCC(N(C)C)CC2)=O)cn1)NC(N)=O 8898,N1(C(c2c(CCC)cccc2)=O)CCC2(CCCCN(C(=O)C3CCCS3)C2)C1 8899,N1(C(c2cc(CC)nc(O)c2)=O)CC2CN(C(=O)CN(C)S(N)(=O)=O)CC2C1 8900,C1(CC(=O)N(C)CCNC(=O)CC2(C)CCC2)COCC1(C)C 8901,C1(C(N(C(C)=O)Cc2cccc(SC)c2)=O)CCN(C(=O)C(C)C)C1(C)C 8902,Cc1nnc2c(C(N3CCC(CNC(C4CCC4)=O)C34CCC4)=O)cccn12 8903,CC(C)(N=[N+]=[N-])C(=O)NC1CCC(CNC(=O)Cc2cc[nH]n2)C1 8904,C=CCCCC(=O)NC(CC1CC1)C(=O)NC1CCCC1 8905,C1(O)(CC(N2C(Cn3cc(CNC(C(CC)OC)=O)nn3)CC2)=O)CCCN(C)C1 8906,C(c1c(F)ccc(Cl)c1F)=CC(N1CC2C(NC(CC(C)C(F)F)=O)(C2)C1)=O 8907,c1(CC)cc(=NCC(CC(C)C)NC(=O)CCNS(C)(=O)=O)[nH]cn1 8908,N1(C(CCCC(CC)CC)=O)CCOC2(CCN(C(=O)CSC(F)F)CC2)C1 8909,C(=O)(CC(=O)NCc1nc[nH]n1)NC(C1(C(=O)NC2CC2)CC1)C 8910,Cc1cncc(CC(=O)NCC(C2CCN(C(=O)C=CC(C)C)CC2)C)c1 8911,N1(C(C(CCC)C)=O)CCN(C(c2n[nH]c(C)c2F)=O)C(CC(C)(C)C)C1 8912,C(=O)(C1CCCn2ncnc21)N1C(C(=O)NC2CN(C(C)=O)C2)CC2COCC21 8913,N1(C(C2CC(C)=C(C)CC2)=O)CCC(C)N(C(=O)C(c2cnn(C)c2)C)CC1 8914,C1(CC(=O)NCCC2(OC)CN(C(c3c(C)nsc3C)=O)C2)CCC(F)(F)CO1 8915,C1(N(CCC)C(C2CC2C2CC2)=O)CCN(C(c2ncn(C)c2C)=O)CC1 8916,c1(CNC(C(C)N(C)C(C2(F)CC=CCC2)=O)=O)cnccc1Cl 8917,C1(O)(CC(=O)NC2(C(=O)NCC(=C)CC)CC2)CCCOC1 8918,C1(F)(CNC(C2CCC(CC)O2)=O)CCN(C(c2sc(C)cc2OC)=O)C1 8919,C(C1CCOCC1)=CC(=O)N(C(C)C(=O)Nc1cnn(CC)c1C)CC 8920,C1(C)(C(=O)NCC2CN(C(c3c(CC)onc3)=O)CC2O)CCCCC1(F)F 8921,C1(NC(c2c(C)ccnc2)=O)CN(C(c2ccc(Br)nc2)=O)CC1C#N 8922,CC(C)(C)C(C)(C)C(=O)N1CCC(C2CC2)(NC(c2nc(=O)n(C)[nH]2)=O)C1 8923,CC(C)CC(CNC(C1(C)CCOCC1)=O)NC(C1C(C(F)F)C1(C)C)=O 8924,c1(C(N(C)CC2OCCN(C(c3cc(C)c(C)o3)=O)C2)=O)cccc(=S)n1O 8925,N1(C(CSCCCC)=O)CC2CCC1CN2C(C1(CCCC)CCCC1)=O 8926,c1(C(=O)NC2COCC2NC(C2CCCOC2)=O)ccnnc1S 8927,N1(C(c2nc(CCCC)sc2)=O)CC2CCC1C(CNC(=O)C(CO)N(C)C)C2 8928,C1(O)(C(=O)NC(C)COc2ccccc2Cl)CCN(C(c2ccccn2)=O)CC1 8929,C1(C(N(CC=CC(NOCC2CC(=C)C2)=O)C)=O)C2CCC(C2)C1C 8930,c1(CN2C3CN(C(=O)OC(C)C)C(C3)C2)ccc([N+](=O)[O-])cc1F 8931,C1(CC(=O)NCCCCCN(CC)CC)CN(C(=O)C(C)OC)CC1C 8932,N1(C(C2CC(=O)N(Cc3ccccc3)C2)=O)CCn2cccc2C12CC2 8933,N1(C(C(n2cc(Cl)cn2)C)=O)CCC(CCNC(C2CN(C3COC3)C2)=O)C1 8934,c1(C(=O)NCCC2N(C(Cc3cnc(C)s3)=O)CCC2)ccccc1F 8935,C1(CO)CCC(C2CC2)CC1.c1(C(CNC(=O)OC(C)(C)C)CC(=O)O)ccccc1 8936,N1(C(c2cnc(Cl)s2)=O)CCCC(NC(=O)CSCc2ccc(F)cc2)C1 8937,c1(C(=O)NCCC(C)NC(=O)Cc2c(Cl)cccc2Cl)coc2c1C(O)CCC2 8938,c1(C(=O)NC2CC3(CN(C(C4(N=[N+]=[N-])CC4)=O)C3)OC2)cc(Cl)cc2c1CCC2 8939,c1(C(N(CCCC(=O)OC)C(=O)CCNC(C)(C)C)C)c(Cl)cnn1C 8940,CCC(CC(F)F)C(=O)NC1CCN(Cc2ccnc(-c3ccccc3)n2)C1 8941,c1(C(=O)NCc2csc(C(=O)NC(C(F)(F)F)C3CC3)c2)cnncc1O 8942,N1(C(C2(C#N)C(C)C2)=O)CCC2(CC1)CN(C(=O)CCNC(=O)C=CCl)C2 8943,C(CC)(C(C)(C)O)NC(C(C)=CC=C)=O.C1CCC(=O)N1C 8944,C1(C(=O)Nc2ccccn2)CC2(C1)CC(N=c1ncn(C3CC3)[nH]1)CCS2(=O)=O 8945,c1(CC(=O)N(C2CN(C(C3COCCO3)=O)CCC2O)C)ccc([N+](=O)[O-])cc1 8946,C1(C(=O)NCC2(NC(C(C)C3CCOC3)=O)CC2)CC(=O)c2ccccc2O1 8947,C1(NC(c2c(CNC(C(C)N=[N+]=[N-])=O)cco2)=O)CC12CCOCC2 8948,c1(CNC(C2CC23CN(Cc2ccnc(Cl)c2)C3)=O)cc(Br)ccc1O 8949,C1(C(N2CC(NC(c3n[nH]c(CC)c3Cl)=O)C3(C2)CC3)=O)CC=C(C(C)C)CC1 8950,CCC(C)(COC)C(=O)NC1CC2C(NC(=O)CCc3ccnc(C)c3)C2C1 8951,c1(C(=O)NCCC(C(C)C)NC(C2(OC)CCSC2)=O)c(C)c(C)cc(C)c1C 8952,N1(C(CSCC#C)=O)CCC(CC(=O)NC(C2CCCCO2)(C)C)C1 8953,C1(CC#C)(C(=O)NC(c2ccco2)C)CCN(C(=O)C(C)C2CC2)C1 8954,N1(C(C2C=CCN(C(CC3CC(CC)C3)=O)C2)=O)CC2CCCC2(CO)C1 8955,N1(C(C2C(OCC)CC2)=O)CC2CCC(C1)N2C(=O)CCc1ccon1 8956,Cc1cc(=O)ccn1CC(=O)NC1(CCNC(c2cc(=O)c(C)c[nH]2)=O)CCC1 8957,C(C)(CCCCCO)NC(C1N(C(CCc2onc(C)n2)=O)CC=C1)=O 8958,C12(C(=O)NC3C(NC(C=C(C)c4cccs4)=O)COC3)CCN(CC1)S(=O)(=O)C2 8959,N1(C(c2c(OC)cncc2)=O)CC2CC(NC(C3CCN(C)C3)=O)CC1C2 8960,C(=O)(CCCC(=O)C(C)OC(=O)C=Cc1ccc(O)c(O)c1)OC 8961,CCC(C)C(C(=O)NC1CCOCC1C)N(C(=O)CC(=O)NC1CC1)C 8962,Cc1[nH]nc2ncc(C(=O)NCC3(F)CCN(C(C4CC(N(C)C)C4)=O)C3)cc12 8963,N1(C(C(C)NS(CCC)(=O)=O)=O)CCC2CCC12CNC(=O)CNC(=O)C1CC1 8964,CC1(C)CC(CNC(=O)CNC(=O)OC(C)(C)C)CN1C(=O)CCS(C)(=O)=O 8965,c1(C(CC)NC(=O)NCc2ccc(Cl)nc2C)cccc(S(N)(=O)=O)c1 8966,C1(C(=O)CBr)COCCC1n1cc(CNC(=O)OC2COC2)nn1 8967,c1(C(=O)NCC2(F)CC(NC(c3cnns3)=O)C2)ccc([N+](=O)[O-])cn1 8968,c1(C(=O)NC2CN(C(C=CC)=O)C(CC)(CC)C2)cc(Cl)cc(Cl)c1OC 8969,CC1CCN(C(C2CC23CCCC3)=O)C1CNC(=O)CSc1cccc(F)c1 8970,CC(F)(F)CC(=O)NCC1CC1CNC(c1cnc(Cl)[nH]1)=O 8971,C1(NC(Cc2cc(C)no2)=O)CC(C)CN(C(C2CC(C)(C)CN2C)=O)C1 8972,CC(CO)(CO)C(=O)NC1CN(C(=O)Cc2nc(Cl)cs2)CC1O 8973,c1(OC)cccc(C(N2CC3C(C(N4CCOCC4C(C)C)=O)C3C2)=O)c1Br 8974,C(=O)(C(C)CC(=O)N(CCC(N1CC(N=[N+]=[N-])C1)=O)C)OC 8975,C1(CC(=O)NC2C(CC)N(C(c3cc4n(n3)CCC4)=O)CC2)CCS(=O)(=O)CC1 8976,C1(C(=O)NC(CC(=C)Cl)C(=O)OC)CCOC2(CCCC2)C1 8977,c1(C(N(C(C)CCNC(c2cnc(Cl)[nH]2)=O)C)=O)ccc(C(F)F)cc1F 8978,c1(N2CCN(C(C(=O)NCC(COC)(C)CO)=O)CC2)ccc(F)cc1OC 8979,CC1(C(=O)NC2CN(C(=O)C(F)(F)C3CC3)CC2C(F)F)CCCS1(=O)=O 8980,C1(NC(CC(n2ccc(C)n2)C)=O)CN(C(C2CC(=C3CCC3)C2)=O)CC1(C)C 8981,C1(S(C)(=O)=O)CN2CCN1C2=O.C(C)(C(=O)OC(C)(C)C)NC(C1CCC1)N 8982,C=CC(C)(CC)C(=O)N(C)CCOCCN(C)C(c1cc(O)cc(F)c1)=O 8983,C(=O)(C(C)C(O)C(C)CC)NC1(C)CCN(C(C2(C#C)CCCCC2)=O)C1 8984,c1(CC)ccc(OC)cc1C(=O)NC(C)C(C)NC(c1cnn(CC)c1C)=O 8985,C(=O)(CC1OCc2ncccc21)NC(C)CNC(C1C2(CC2)C12CC2)=O 8986,C1(CC)(NC(=O)C(O)C2CC2)CCCN(C(=O)CN(c2ccc(Cl)cc2)C)C1 8987,Cc1ccc(C=CCC(N2CC(NC(=O)CSC3CC3)C(C(F)F)C2)=O)cc1 8988,C1(C)(N(C)C)CCCN(C(C2CCC3(CC3)N2C(C2CC3(CCC3)C2)=O)=O)C1 8989,c1(-c2c(C)noc2)nc(-c2ccccn2)nn1Cc1ccc(Cl)cc1 8990,C1(NC(CCOCC#C)=O)COC2(COC)CC1C2.C12CN(C1)C2=O 8991,Cn1nccc1C=CC(=O)NCC1CCC(C(N2CC(O)C(O)C2)=O)CC1 8992,C1(C(=O)OCC)(NC(C2CC(NC(=O)CC3CSC3)C2)=O)CCOC1 8993,CC(=O)CCCC(C)C(=O)N1CCC(NC(C2SC3C=CC2CC3)=O)C(F)C1 8994,C1(CC(N2CCN(C)C(c3ccccc3)C2)=O)CCN(C(C)(C)C)C2(CC2)C1 8995,C1(CCCC)CN(C(=O)CN(C)C(C)=O)CCN1C(=O)C(C1CC1)OC 8996,CCC(CC(=O)NCC(C)(C(C)C)NC(c1cc(CO)[nH]n1)=O)c1ccccc1 8997,C(=O)(CCS(=O)(=O)C1CCCC1)NCC(CC)NC(C1CC(OC)C(OC)C1)=O 8998,C1(CNC(CSCC)=O)CCN(C(=O)CCn2cc(Br)c(C)n2)C12CC2 8999,Cc1nc2ncccc2cc1C(=O)NCC(O)CN(C)C(c1nsnc1O)=O 9000,c1(OC)ccc2[nH]c(C(N3CCC(CNC(=O)CCc4cnc[nH]4)C3)=O)cc2c1 9001,Cc1coc(CN(C(C2CCCC2O)C(=O)NCCC#N)Cc2ccco2)c1 9002,C=C(C)C(O)CC(=O)N1CC=C(CNC(=O)C(CO)NC(N)=O)CC1 9003,c1(C(N(C)CC2(N(C)C)CC2)=O)c(Cl)nn(C)c1Cl 9004,C1(NC(c2ccc(OC)cc2Br)=O)CC2CCCC(C1)N2C(=O)C(C)O 9005,c1(C(N2CC(C)C(NC(c3cccc(Cl)c3)=O)C2)=O)ccc2c(c1)CCCCS2 9006,C#CCCC(C(=O)N1CCC1C(C)O)NC(c1cnccn1)=O 9007,C1(C(N2C(CNC(c3c(C)cccc3Cl)=O)C=CC2)=O)CC2CCCN2C(=O)N1 9008,N1(C(C(CC(C)C)NC(N)=O)=O)CCC2CCC(NC(=O)CCc3cnn[nH]3)C12 9009,c1(C(=O)NCC2C(NC(C(C(C)C)SCC)=O)CC2)ccnc2[nH]c(O)nc12 9010,C1(CC(=O)NCC2(O)CN(C(CC(C)c3cccnc3)=O)C2)NC(=O)CNC1=O 9011,C(C)(CN=C(NCC(F)F)N1CCC(C(N)=O)CC1)C1CCC(C)CC1 9012,c1(C(N2CC(CNC(CCN(C(C)=O)C)=O)C2)=O)cnc2cc(Br)ccn12 9013,c1(C(=O)NCC2C(CNCc3ccc(NC)cc3)C2)occ2c1CCC2 9014,C1(C(=O)NC2C(C)(C)C(=O)NC2)CCN(C(=O)C(F)(F)c2ccccc2)O1 9015,CC1=Nc2ccccc2C12CCN(C(C1CC3(CC3)CN1C)=O)CC2 9016,c1(OCC=C)ccc(Cl)c(CNC(=O)NCC2(O)CC=CC2)n1 9017,c1(CC)nc(C)n(C)c1C(=O)NCC1CC2CCC1N2C(c1c(C)noc1C)=O 9018,C1(C(=O)NC(C(=O)NC(CN(C(C)C)C)C)Cn2cncn2)CCCSC1C 9019,c1(CC(=O)NCC2(F)CN(C(CSC(C)C)=O)C2)ccc(OC(C)C#N)cc1 9020,C(CC(CNC(=O)COCCOC)OC)NC(CC=CCC)=O 9021,C1(NC(c2cc(C(=O)OC)nn2C)=O)CN(C(c2ncncc2F)=O)CC12CC2 9022,N1(C(C2C(C)CC2)=O)CC(NC(=O)COc2ccon2)C(F)C1 9023,c1(C(N2CCC(C3N(C(COC)=O)CC3(C)C)CC2)=O)cc(F)cnc1O 9024,c1(C(C)OCC)nc(C)c(C(=O)NCC(C2CC2)NC(=O)CCCC2(C)N=N2)s1 9025,Cc1ccc(NC(=O)C(F)CC2CN(C(c3cocn3)=O)C2)cn1 9026,C12(C(=O)NCC(C#C)OC)CC(CN(C(=O)CN(C)C3CC3)C1)C2 9027,C(CCC(=O)N1CCC(N(C(=O)CCC=C)CCO)C1)=CCC=C 9028,N(C(=NCC)N1CCN(C(C)=O)C(C)(C)C1)C(C#C)(CC)CC 9029,C1(F)(CNC(CCN(CCCCC)C)=O)CCCN(C(C2CC3CC3C2)=O)C1 9030,C(=O)(C(C(C)C1CCCC1)N1CCCC1)NCCCSC 9031,c1(C(=O)NC(CC(C)NC(C2CCCC(C(F)(F)F)C2)=O)C)cc(N)ccn1 9032,Cc1cccc2[nH]cc(CC(=O)N(C)CCNC(C3CC4(C3)CC(C)C4)=O)c12 9033,c1(C(=O)NCc2cc(Cl)cc(Cl)c2Cl)ccc(S(=O)(=O)NC2CC2)o1 9034,Cc1nc2cc(C(N3CC4CC(NC(c5cccc(Cl)c5C)=O)C4C3)=O)[nH]c2s1 9035,S(=O)(=O)(c1ccc(C(=O)NC2CCN(C(C34CC(C)(C3)C4)=O)C(C)C2)cc1)NC 9036,C(c1c(C)nn(C)c1Cl)=CC(N1CCC(CCN)(OCC)C1)=O 9037,C(N=c1[nH]c(=NCc2cc(C(F)F)n[nH]2)c2ccccc2[nH]1)C1(C(N)=O)CC1 9038,c1(C(N2C(C3(NC(C4C(C)(C)CC4)=O)CC3)CCC2)=O)cc2cccnn2n1 9039,C1(O)(C(=O)OCC)CCN(C(=O)CCN2CCN(CCO)CC2)CC1 9040,c1(C(N(C(CCNC(Cc2c(C)ccc(C)c2)=O)C)C)=O)ncc(Cl)c(N)c1Cl 9041,c1(C(=O)NC2CCC(C(=O)Nc3ccc(F)c(O)c3)C2)cnc2ncccn12 9042,c1(C(C)C)ccc(CSCc2cnn(C)c2)cc1OCC(F)F 9043,N1(C(CCCC(C)=O)=O)CC2CC(NC(C3C4CCC3(C)C4(C)C)=O)CC1C2 9044,C1(C(=O)NCC2C(CNC(c3ccn(C)n3)=O)C2)C2CCN1CC2 9045,C1(NC(CC2CCC(C)(O)CC2)=O)CN(C(=O)C(C)(C)F)CCC12CCC2 9046,c1(C(C)C)ccc(O)c(C(=O)N(C2CN(C(C3CC4C(C3)C4(F)F)=O)C2)C)c1 9047,Cc1cc(NC(=O)CN2C(=O)CNC2=O)ccc1NC(=O)CP(C)(C)=O 9048,CC1CN(C(c2ccc(C#N)c(O)c2)=O)CCCN1C(=O)C(F)C(C)(C)O 9049,C1(CC)CCN(C(=O)C=CC2CCCC2)C1C(=O)NCC1(C(C)(C)O)CC1 9050,C12CC3CC3N1C2=O.c1(COC(C2CCN(C3CCCCC3)C2)=O)ccccc1 9051,c1(N2CC(c3ccccc3)(CC)OCC2)nc(=NCc2cc[nH]n2)[nH]c2cc[nH]c12 9052,c1(C(=O)NC2C(CNC(=O)C=Cc3ccncc3)CCC2)ncc(Cl)cc1Cl 9053,C#Cc1ccc(F)c(C(N2CCCC2CN(C)C(C2CCCCC2(C)C)=O)=O)c1 9054,n1(CC(N2CCOCC(CNC(C3C4COCC34)=O)C2)=O)cc2ccccc2n1 9055,N1(CC(c2nnnn2C)(C)NCCc2cc(CC)no2)C(=O)CCCC1=O 9056,C1(CNC(C2(C(=O)OC)CC2)=O)CCCC1C(=O)N(C)CCn1cncn1 9057,c1(C(=O)NCC(C)(C)CNC(C2CC(C(=O)O)C2)=O)ccnc(-n2cccc2)c1 9058,c1(NCC)cccc(C(=O)NCC(C)N(C)C(C2CC3(CC3)CO2)=O)c1 9059,C1(NC(c2c(CC)scc2)=O)C2CC3CN(C(c4c[nH]c(Br)c4)=O)C1C3C2 9060,N1(C(c2cc(C)no2)C(=O)NCC2CCCO2)CCCC(c2ccc(F)cc2)C1 9061,CN1C(=O)CCCC1C(N1CC(C2CC2C(N2CC(OC(=O)N(C)C)C2)=O)C1)=O 9062,C1(OC)CC2(C1)CC(C(=O)NCC(C)(CC(C)C)NC(c1nc(C)oc1C)=O)C2 9063,n1(CC(N2C(COCC)CCCC2)=O)cc(I)cc(N)c1=O 9064,CC1(CNC(=O)CCCCC2CC2)CN(C(C2NC(=O)OC2C)=O)CCO1 9065,c1(OC)c(C(=O)NCC2CCN(C(=O)Cc3csc(=N)[nH]3)C2)[nH]c2ccccc12 9066,N1(C(C(C)N(C(c2cccc(C)n2)=O)C2CC2)=O)Cc2cnn(C)c2C1 9067,C(C(C(=O)NCCS(C)(=N)=O)NC(=O)C=NOC)OCC 9068,C(=O)(CC(C)C(C)C)NCC(CNC(C1N(CCCC)CCCC1)=O)C 9069,N1(C(C2CN(C)C2)=O)CCC(NC(c2cnc(C(F)F)nc2)=O)C(F)C1 9070,c1(C(=O)NCC2(CNC(C(C)=C3CCC3)=O)CC2)nc2cccnc2s1 9071,C1(NC(C(C2CCC2)OCC)=O)CN(C(C2CC(O)CN2C)=O)CC1CO 9072,c1(OCCC)ccc(CCCC(=O)NC2(COC)CCCCC2)cc1 9073,c1(C(N2CCCC(CNC(CCc3onc(C)n3)=O)C2)=O)c(C)oc(C)c1C 9074,C(CNC(=O)CCCOC1CCOCC1)(C(C)(C)C)NC(Cc1c(C)cco1)=O 9075,C(c1ccc(F)c(F)c1)=CC(=O)NCCC1C(C)(C)CCO1 9076,CCC(C)(CO)C(=O)NCC(O)CCNC(=O)CC1(C)CCCCC1 9077,c1(NC(C)=O)ccc(C(=O)NC2(C)CN(C(c3nnn(C)n3)=O)C2)c(Cl)c1 9078,N1(C(C=C=C(C)C)=O)C(C(=O)NCC(=O)NC(C)(C)C)CCC12CC2 9079,N1(C(C(CC)OC)=O)CCC=C(CNC(C2CC(=O)N(CC)C2)=O)C1 9080,Cc1ccc(Cl)c(OC(C)C(=O)NC(C)(C)CCNC(=O)C(O)CC)c1 9081,c1(CCC(=O)NCC(CC)NC(c2cnn(C)c2)=O)ccccn1 9082,O=S(=O)(OC1CC2OCCC2C1)c1c[nH]ccc1=NC1CNC1 9083,N1(C(c2c(CC)non2)=O)CC=C(CNC(=O)CCC2CC(OC)C2)CC1 9084,c1(C(C)=O)cccc(C(=O)NCC(CO)NC(c2cnc(Cl)[nH]2)=O)c1 9085,C1(NC(C(CC)=CC)=O)CC2CN(C(=O)C(C)Oc3ccc(SCC)cc3)CC12 9086,CC1(C)C(NC(C2CC=CC2)=O)CCN1C(=O)Cc1cc(-c2ccccc2)on1 9087,C=CCN=c1[nH]cc(C(N2CCN(C(N)=O)CC2)=O)s1.C1(=O)CNCCN1 9088,C1(C(N2CCCC(NC(C(C(C)C)(C)O)=O)CC2)=O)CCC2CCCCN12 9089,C1(NC(C(N2CCN(C)CC2)C)=O)CC(C)CN(C(=O)CCc2cnn[nH]2)C1 9090,C(c1ccco1)=CC(=O)NC(C(=O)NCCCOCC(C)C)C1CCOC1 9091,CN1CCN(C(c2cc(C3CC3)ccn2)=O)c2ccc(O)cc21 9092,Cc1cc[nH]c(=N)c1C(=O)NCC1CC1CNC(=O)CC1CCCC1 9093,N1(C(COC2CN(C(C)=O)C2)=O)CCC(CCCNC(c2cnc(Cl)s2)=O)CC1 9094,c1(C(=O)NCc2nnc(C)o2)ccc(CNC(=O)Cn2cnnc2O)cn1 9095,Cc1scc(C(N2CC(OC3CCOCC3C(=O)NOC3CCOCC3)C2)=O)c1C 9096,C(=O)(C(CC(C)C)NC(C)=O)NCCNC(c1ccc(CC)o1)=O 9097,c1(NC(=O)NC2N(C(CNC(c3nc(C)sc3C)=O)=O)CC2)cc(Cl)ccc1C 9098,CC(C)(CC(F)F)C(=O)N1CCCC(O)(CNC(C2(C)CC2(F)F)=O)CC1 9099,O=C1CCN(Cc2nnnn2C2CCCCC2)C(=O)N1Cc1c(F)cncc1F 9100,C1(NC(c2cc(C)[nH]n2)=O)C2CC3CN(C(c4ccnnc4)=O)C1C3C2 9101,C(CC(C(=O)NCc1nc(C)c(C)[nH]1)NC(=O)C(C)C(F)F)OCC 9102,c1(C(C)C(=O)NC2CC2NC(C2COC2)=O)ccc(C(F)(F)F)cc1 9103,C(=O)(CC(C)C(C)(C)NC(=O)Cc1ccnn1C)NC(C)CCC1CCCC1 9104,n1(CC(=O)NCCN(C(c2c(CC)c(F)ccc2)=O)C)nnc2ccccc2c1=O 9105,C1(CCOC)CCN(C(=O)CCN(C(=O)CN(C)C)Cc2ccccn2)CC1 9106,C1(C(=O)NCc2c(CCNC(C3CCN(C)C3)=O)ocn2)CCC2(CC2)C1 9107,c1(NC(CCNC(=O)NC(CO)CCO)=O)csc(O)n1 9108,Cc1c(C(=O)NCCCN(CCO)C(C2COCCN2C)=O)c[nH]c1C#N 9109,C(=O)(CC(O)CC(C)C)N1C(C(N2CCC(COC)C2)=O)CC(OC)C1 9110,C1(C2(NC(COCC=C)=O)CC2)CCCCN1C(c1cnn(CC(C)C)c1)=O 9111,C1(C#N)(C(N2CC(C)C(NC(C3(CF)CCC3)=O)C2)=O)CC2C=CC1C2 9112,C1(NC(C(CC(C)C)N(C(=O)C(C)n2ccnc2)C)=O)CC2(C1)CC21CCC1 9113,C(=O)(CCCCN=[N+]=[N-])NC(C(=O)NCC(C#C)CC)COC(C)C 9114,N1(C(C)(C)C)CCCC(C(N2CCC2CF)=O)C1 9115,c1(C(=O)NC2CCCC(NC(CCCOC(C)C)=O)C2)ccnc(S(N)(=O)=O)c1 9116,N1(C(C(C(C)C)NC(N)=O)=O)CCC(F)(C(N2CCC3(CCO3)C2)=O)CC1 9117,C1(C(=O)N(C)Cc2cncn2C)(C2CC2)CCCO1.CN(CCO)C 9118,C1(C(=O)NCCCN(C(C(C)c2cncs2)=O)C)Cc2nccnc2C1 9119,C1(C(=O)NC)CCN(C(=O)C(CCN(C)C)NC(c2cnsn2)=O)C1C 9120,N(C(=NCCCCl)NCc1cccc(F)c1)Cc1c(C)cc(C(=O)N(C)C)cc1 9121,C(N=c1[nH]c(=NCC(F)F)[nH]c2cccnc12)C1C(C)(C)OCCO1 9122,Cc1ccc(C(N2CCOC(CC(N3CCN(CCO)C(C)C3)=O)C2)=O)nc1C 9123,Cn1ccc2ccc(C(=O)NCC3(O)CC(NC(C4CC(CCO)C4)=O)C3)cc12 9124,CC1(C)CN(C(=O)CSC(F)F)CC1N=c1cc(Cl)nc(C(F)(F)F)[nH]1 9125,C1(N(C(C2CC(C(=O)OC)C2)=O)C)CCC(NC(=O)C(N2CCOCC2)C)CC1 9126,CCC(CNC(=O)CCC(C)(C)[N+](=O)[O-])N=c1[nH]c2ccc(F)cc2s1 9127,CC1(C(=O)NCC2CCCCN(C(C3CCSCC3)=O)CC2)CCCCNC1=O 9128,C1(N=[N+]=[N-])(C(=O)NCc2cc(C)n(C)n2)CCN(C(=O)C(O)Cn2cncn2)C1 9129,Cc1ccnc(CNC(C23CC(NC(=O)OC(C)(C)C)C2C3)=O)c1 9130,c1(CC)cnoc1C(=O)NC1CC(O)(CNC(=O)CC(C)F)C1 9131,C1(NC(C2CC3(CC(=C)C3)C2)=O)CCC2CC1CN2C(=O)C(c1cnn(C)c1)=O 9132,c1(COC)cc(C(N2CC(CNC(C3(NC(C)C)CC3)=O)C(C)C2)=O)ccc1F 9133,C(CNC(C1(C#N)CC1(C)C)=O)(CC(C)C)NC(Cc1n(C(C)C)ncc1)=O 9134,CC(=O)C(C)(C)CC(=O)N1CCC(C(=O)NCC(C2CC(C)(C)C2)O)CC1 9135,N1(C(CC2(C(=C)F)CCC2)=O)CCN(C(=O)Cc2cccc(C)c2)CCC1C 9136,C1(C(=O)O)CC(F)CN(Cc2ccc(OCBr)cc2)C1.C123CC(C1)(C2)CN3 9137,c1(C(=O)NC23CC(C(=O)O)C(C2)C3)ccc2c(c1)nc(O)n2C1CC1 9138,Cn1ccc(C(=O)NC(C2CCN(C(c3cn(CC(F)(F)F)cn3)=O)C2)(C)C)c1 9139,c1(C(=O)NCCCN(C(C2C(C)C2)=O)CCO)cc(F)c2ncccc2c1 9140,CC(C)(O)C(F)C(=O)NCC1CCN1C(=O)CC1CCC2(CCC2)O1 9141,C1(C(C)NC(=O)CONC(=O)C2CC(C(N)=O)C2)CC2CCC1C2 9142,Cc1nc(C(=O)NC(C)CCCCNC(c2ocnc2C2CC2)=O)[nH]c1C 9143,C1(OC)CN(C(=O)CC2CCN(C)C2=O)CC1C(=O)NCC1CCC1(F)F 9144,N1(C(c2c(C(C)C)nn(C)c2)=O)CC(CNC(=O)CN(C)C2CC2)C(C)(C)C1 9145,N(C1CCc2ccc(F)cc21)C(=O)C(F)(F)c1csnn1 9146,N1(C(C2C(C3C(C)C3)C2)=O)CCC2(CCCC2NC(C2CCCO2)=O)CC1 9147,CC(CNC(c1ccnn1Cc1ccccc1)=O)(CO)NC(=O)CC1CCCO1 9148,N1(C(CC(CC)C(C)C)=O)CCC2CCN(C(C3CCOC3C3CC3)=O)CC12 9149,c1(C(=O)NCC(CC)(C)NC(C2CS(=O)C2)=O)nc(Cl)c(Cl)s1 9150,C=C(C)CC(C(=O)NCC=CCCC)NC(C1CCOC(C)(C)C1)=O 9151,c1(NCC=C=C)ncccc1S(=O)(=O)N1CC2CC3CC2C1C3 9152,c1(C(=O)NCCC(C)NC(C2CC2C2CCC2)=O)ccnn(C)c1=O 9153,N1(C(C2N(C(c3cc(OCCOC)n[nH]3)=O)CCC(O)C2)=O)CC(O)CC(C)(C)C1 9154,N1(C(c2c(NCCCC)cccc2)=O)CCN(C(c2cnc(Cl)cn2)=O)C(C)C1 9155,c1(CC)cc2c(NC(C)COC(c3cccc(Cl)c3)C)ncnc2s1 9156,C1(CCNC(=O)Cc2cc[nH]n2)CC(F)(F)CN1C(c1cc(Cl)c(Cl)s1)=O 9157,C12(NC(c3c(C)occ3)=O)CCCC1N(C(c1ccc(C3CCC3)cc1)=O)CC2 9158,C(=O)(CN=c1cc[nH]cc1)NCC(c1ccccc1)NC(c1c(C)cnn1C)=O 9159,C12(CNC(C3CC34CCCC4)=O)CCC(CC1)CN2C(=O)COCC1CCCO1 9160,c1(OC)ccc(NC(C2CC2NC(c2cnc(O)cc2O)=O)=O)cc1C#N 9161,C#CCC(CC#C)C(=O)NCC(F)CNC(C1(O)CCCCC1)=O 9162,c12ccccc1C2c1nnnn1-n1cccn1.C1(N(C)C)(CC#N)COC1 9163,Cn1cnn(CC(=O)NC2CCOCC2C(N2CCCC2CCO)=O)c1=O 9164,c1(C(N(CC(C)(C)NC(c2c(C)ccnn2)=O)C)=O)[nH]c2cc(F)ccc2c1C 9165,c1(C(=O)NCC2C(C(=O)NCc3c(OC)cccc3)CCC2)ccc(C)cc1O 9166,C1(OC)(CNC(N2CCCC2C(F)(F)F)=O)CCCCC1 9167,N1(C(C(CC)OC)=O)CCC(O)(C(C)NC(=O)CN2CCC(O)CC2)CC1 9168,c1(C(=O)NC(CN(C(=O)CC2COCCO2)CC)C)cnc(OC)c(Br)c1 9169,c1(C(=O)NC2C(CNC(C3(CC)CC(C)(C)C3)=O)CC2)nsc2ccc(C)cc12 9170,c1(C(N(C2CCN(C(C3CCCC3(C)C)=O)C2)C)=O)ncc(F)cn1 9171,Cc1cc(C(=O)NCC2CC(C)CN(C(C3(C)SCCCS3)=O)C2)c(O)nn1 9172,c1(C(=O)NCCCNC(CC2C=NN(C)C2=O)=O)cc[nH]c(=N)c1[N+](=O)[O-] 9173,N1(C(C2(C)N(C(C(CC)N(C)C)=O)CCC2)=O)CC2CC1CN2C(C)=O 9174,c1(C(=O)NC(CNC(c2nc(C)oc2C)=O)C)ccc(F)c2cccnc12 9175,c1(C(=O)NCC(C2CC2)NC(C(CSC)OC)=O)cc(C(F)(F)F)nn1C(C)C 9176,c1(C(=O)NC(c2cc(F)ccc2F)CC(=O)OC)ccc(C(N)=O)c(Cl)c1 9177,c1(C(=O)NCCN(C)C(C2CCCCS2(=O)=O)=O)c(F)cc(OC(F)F)cc1F 9178,N1(C(c2c(Cl)cc(C)s2)=O)CCC2(CCCC2NC(c2coc(C#N)c2)=O)C1 9179,c1(OC)cccc(C(=O)NC2CN(C(=O)C(C)n3ccnc3)CC2C)c1 9180,Cc1ccn(C)c1C(=O)N(CC(C)CNC(c1nn(C(C)C)cc1Br)=O)C 9181,C(=O)(CCC(=O)NC1(CF)CCN(C(c2cnoc2CSC)=O)C1)NCCC 9182,C1(C(=O)NCCCNC(C(C(C)(C)C)O)=O)CC(=O)c2cc(Cl)ccc2O1 9183,C1(C(N(CCC(C)NC(CC2CC(=C)C2)=O)C)=O)COCC1(C)C 9184,C(CC(CC)C(=O)N1CCN(C(c2cc(C)c(Cl)s2)=O)C(C2CC2)C1)=CC 9185,c1(C(N(C)CC2(NC(COCCCCC)=O)CC2)=O)ccnn1CCCC 9186,c1(C(N2CCCC(NC(C(CC)F)=O)(CC)C2)=O)nnn2ccccc12 9187,c1(C(N(C2CCN(C(=O)CC3CCC3=O)CC2)CC)=O)cccc2ccccc12 9188,C1(NC(C=C(C)C)=O)CC2CN(C(C3CCS(=O)CC3)=O)CCN2C1=O 9189,CC(C)CC(C(=O)N1CCC(CNC(c2nnn(C)c2N)=O)C(O)C1)C(C)C 9190,N1(C(=O)NCc2ccc([Si](C)(C)C)s2)CCn2c(cc3ccccc23)C1 9191,c1(C(=O)NC2CN(C(CCN3C(C)CCCC3)=O)CC2O)ccn2nnnc2c1 9192,CC(F)(F)CCC(=O)N(CC(=O)NC1CCC12CCCC2)C1CCC1 9193,C1(C(N)=O)C2CC1N(C(C1(n3cc(Cn4ccnc4)nn3)CCOCC1)=O)C2 9194,C1(NC(CC2CC(OC)C2)=O)CN(C(=O)C(C)CC2CCC2)CC1CC1CC1 9195,c1(C(=O)NC(C)CCNC(c2cc(Cl)ccn2)=O)nn(C)cc1S(N)(=O)=O 9196,c1(C(=O)NCC2N(C(CCOC(C)C)=O)CCC2)nn(C)cc1S(N)(=O)=O 9197,Cc1cc(C(N2CCC(O)(CNC(C3(O)CCOCC3)=O)CC2)=O)cc(C)n1 9198,C1(F)(CNC(Cc2ccc(CCCC)cc2)=O)COCCN(C(=O)CCC#N)C1 9199,C1(C(=O)NC(CNC(C2(OC)CCSCC2)=O)C(C)C)CC2(C)CC1CO2 9200,C1(CNC(=O)CSC(F)F)CN(C(C2CC2Br)=O)CC1O 9201,c1(OC)cc(N)c(C(=O)NC2CCCC(N)CC2)cc1Cl 9202,C1(C(=O)NCC2N(C(C(C)(C)n3cnnn3)=O)CCC2)CC1C1CCCC1 9203,N1(C(c2cc(C(C)(F)F)on2)=O)CC2CC1CN2C(C1CCCCO1)=O 9204,c1(C2(C(=O)NCC(CC=C)NC(C3COCCO3)=O)CCC2)ccccc1C#N 9205,Cn1ncc2c(C(=O)NC3(CNC(c4sc(Cl)nc4Cl)=O)COC3)cc(Br)cc12 9206,CC1CN(C(C2CCCS2)=O)CC2(CCN(C(c3ccn(CC#N)n3)=O)C2)O1 9207,N12CCC3(CC1)CCN3CC2=O.N1(C(C=CC)=O)CCN(S(=O)(=O)CCCC)CC1 9208,C1(CNC(C2CCCCN2C(C23CC(F)(C2)C3)=O)=O)CCC(O)CC1 9209,N1(C(C(CC)=CC)=O)CC(NC(C2CC3C=CC2C3)=O)CC(F)C1 9210,CN1C(=O)CN(CC(N2CC(CNC(=O)CC3CCCOC3)CC2(C)C)=O)C1=O 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9888,N1(C(c2cccc3ccn(C)c32)=O)CCOC2(CCN(C(C3CC3(Cl)Cl)=O)C2)C1 9889,N1(C(C)=O)CCOC(C(N2CCC(NC(=O)CCc3ncc(C)[nH]3)C2C)=O)C1 9890,CC1(C)CCCCC1(C)NC(=O)NCC1CCC(=O)NC1=O 9891,CCC(CN(C(c1cc(C)co1)C(=O)NC(C)(C)C)C)CC 9892,Cc1noc(C)c1C(=O)NCC12CC1CN(C(=O)Cc1cccc(C(F)(F)F)n1)C2 9893,C=CC1(C(N2CCCC(OC3CC3)C2)=O)CCN(C(C2CC3CC(=O)C2O3)=O)C1 9894,c1(SC)ccc(C(N2CC(NC(c3ncn(C)c3C)=O)C(C(F)F)C2)=O)c(Cl)c1 9895,N1(C(C(C)CO)=O)CCC2(CCCCC2NC(c2cc(F)cc(Cl)c2)=O)CC1 9896,Cc1nn[nH]c1CCNC1CCC(Cc2ccncc2)C1 9897,N1(C(C(CC)OCC)=O)CC2CCC(C1)C(NC(c1c(C)nn(C)c1Cl)=O)C2 9898,C1(CO)CCC(CNC(c2nnnn2CCCF)CC2CCOC2)CC1 9899,CC1CCCCC1(CNC(=O)CCC(=O)c1ccccn1)NC(c1cnsc1)=O 9900,c1(NC(=O)NC(C(CN(C)C)(C)C)c2nnnn2C)ccc(Cl)c(P(C)(C)=O)c1 9901,c1(C(=O)NC2CCC2CNC(C2C(F)(F)C23CCC3)=O)cc(C2CC2)ccc1F 9902,c1(C(=O)NCC(O)Cc2nn[nH]n2)ccc2c(c1)CCCC2 9903,c1(CC)cccc(C(N2CC(O)(C(F)C(=O)N(C3CC(O)C3(C)C)C)C2)=O)c1 9904,NC1CCCC2CN(CC(=O)NC3CCN(c4nncs4)CC3)CC12 9905,C1(C(N2CC(C(CC)C)C2)=O)CCCN(C(c2sccc2CO)=O)C1C 9906,c1(OC)csc(C(N2CCC(F)(CNC(C3(C)CCCS3)=O)C2)=O)c1OC 9907,c1(C(=O)NCC2(C(C)NC(c3cc(C(C)=O)oc3)=O)CC2)cc(C)ccc1C 9908,C(=O)(C(CC(C)C)CC(C)C)NC1C(CNC(CCc2ccc(C)o2)=O)CC1 9909,n1(C(C)C)c(O)nc(N(CCCNC(C2CCN(C)C2=O)=O)CCOC)cc1=O 9910,c1(NC(c2c(C)nc(CC)o2)=O)ccc(NC(c2cncc(C)n2)=O)c(C)c1 9911,CCC(CC(C)C)C(=O)NCC1CCC(NC(=O)Cn2nnnc2C(C)C)CC1 9912,CC(CCN(C)C)C(=O)NC1CCCC1C(N1CCC1(C)CCO)=O 9913,c1(C(=O)OCc2c(C)ncn2C)cc(S(=O)(=O)N(C)C)ccc1F 9914,N1(C(c2cc(C)c(Br)o2)=O)CC2(COC(CNC(c3ccncn3)=O)C2)C1 9915,N1(C(C2(Br)C3COCC23)=O)CC2(C1)CN(C(C1(C3CCC3)CC1)=O)C2 9916,N1(Cc2ccc(OC)c(-c3ccncc3F)c2)CCCC2(C1)OC(=O)NC2=O 9917,C1(OC)CCCCC1C1CCN(Cc2cccc(C3CCCNC3)c2)C1 9918,C#CC1(C)CCCN(C(=O)C(CCSC)NC(=O)COC(C)C)C1 9919,Cc1ncn(C)c(=O)c1C(=O)NCC1(NC(=O)C(N2CCCC2)C2CC2)CCC1 9920,CN=c1[nH]cc(C(=O)NCC2(NC(=O)C(C)=C3CCCC3)CCOC2)o1 9921,C1(NC(=O)Cc2cn[nH]c2)CC12CCN(C(c1ccc(O)cc1Cl)=O)CC2 9922,N1(CC)CCN(C(=O)C(C)CNC(=O)C(F)C(C)(F)F)CC1C 9923,CC1=C(C(=O)NCC(C2CCOC2)NC(c2cc(CF)on2)=O)CCC(C)(C)C1 9924,C(=O)(CCCCCC(=O)N1CC(NC(=O)C(C)=C2CCC2)C(C2CC2)C1)OCC 9925,c1(C(=O)NC2CCC(NC(COCCOC)=O)CC2)c(C)ccc(Cl)c1O 9926,N1(C(c2cc(C)nn2CC(F)F)=O)CCC(F)C(NC(C2CCCC2)=O)C1 9927,Cc1c(C(N2CC(CCNC(=O)C(C)(C)C)OC(C)C2)=O)[nH]c2c1C(=O)CCC2 9928,N1(C(c2ccc(CC)c(CC)c2)=O)CC2CCN(C(c3cccn3CC)=O)C2C1 9929,C1(CNC(=O)C=C2CC2)CC(F)CN1C(=O)CCC1CCCO1 9930,N1(C(C=C(C)Cl)=O)CCN(C(c2cccn(C)c2=O)=O)C(C(C)(C)C)C1 9931,CCCCC(C(=O)NCCN(C(=O)C=C1CC1)C)NC(=O)OC(C)(C)C 9932,C1(C(=O)NCCNC(C(COC)OC)=O)CC2CC1CO2 9933,c1(C(N2C(C)(CNC(=O)CC3(O)CCCOC3)CCC2)=O)cccc(N=[N+]=[N-])c1 9934,Cc1[nH]nc(C(F)(F)CO)c1C(=O)NCCOCCNC(=O)C=Cc1ccoc1 9935,C(=O)(CC(C)C(F)F)NC(CC)(C)CCNC(c1n[nH]cc1C)=O 9936,N1(C(C(C)=CC)=O)CC2C3CCC(C2C1)N(C(=O)Cc1ccc(C)c(Br)c1)C3 9937,S1(=O)(=O)c2ccc(cc2)C=CC(=O)N1CC(C)O.C(C(C)(C)O)OC(C)C 9938,C1(NC(C2CC3CCC(C2)C3=O)=O)CC2CN(C(=O)C(F)CC3CC3)CC2C1 9939,CC1CCC(C(N2CC(CO)CC2CO)=O)CN1C(=O)Cc1cc[nH]c1 9940,N1(C(c2cc(C(C)C)no2)=O)CCC(C(N2CCCCC(C)CC2)=O)CC1(C)C 9941,N1(C(CNC(CC)=O)=O)CCC(C2CCN(C(=O)CCCC(F)F)CC2)CC1 9942,C1(C(=O)NC2(C)CCC(C)C2)CC2(CC(NC(C3(O)CC4CCC3C4)=O)C2)C1 9943,c1(C(=O)NCC2(F)CC(NC(CC3CC(=O)NC3)=O)C2)csc2nnsc12 9944,C1(NC(C2C(=C)CC2)=O)CCC2CC1CN2C(c1c[nH]ccc1=O)=O 9945,C1(C(=O)NCc2c(CC)n[nH]c2)CCC(C)(C)N(C(C23CCC(C2)C3)=O)C1 9946,C1(CC)CN(C(=O)Cc2cccc(C)c2Cl)CCC1NC(c1ncc(C)cn1)=O 9947,N12C3CCC1CN(CC3)C(=O)Nc1c(cccc1)N(CC)C(=O)C2.C(C)(C)OC 9948,C12(CNC(=O)CC3CC3)CCCC1N(C(=O)CN1CCCCC1)CCC2 9949,C=C1Cn2c(C(=O)NCC3(C)CCN(C(=O)C(=Cc4c[nH]cn4)F)C3)nnc2S1 9950,CCC(C)CC(C(=O)Nc1ccc(OC)cc1C)NC(=O)CC1(O)CCOCC1 9951,C(C)(C(C)(C)CO)NC(C1C(CNC(C2(CC)CCCC2)=O)CCC1)=O 9952,Cc1nn(CC(N2CCC(NC(=O)COCC3CCOC3)C2C)=O)cc1[N+](=O)[O-] 9953,C1(NC(c2cnsc2)=O)CC2CCC1N2C(=O)COc1ccc(Cl)nc1 9954,c1(C(=O)NC(c2cncnc2)C)cccc(CNC(C2CCC3(CC3)C2)=O)n1 9955,C(=O)(C1=CCC(C)(C)CC1)NC1CC(CNC(c2c(C)[nH]nc2C(F)F)=O)C1 9956,N1(C(CCCOCCC)=O)CC(C)CCC1CNC(=O)CNS(=O)(=O)CC 9957,N1(C(C(C)C#N)=O)CC(F)(F)CC1CNC(c1ccc(C(F)(F)C(F)F)cn1)=O 9958,C(CCCC(CO)NC(c1ccc(F)cc1)=O)NCc1c(C(=O)OCC)scc1 9959,N1(C(C2(F)CCN(C(CC(C)n3cccc3)=O)C2)=O)CC2CCC1C(O)C2O 9960,C=CCN=C(NC1CCn2c(C)cnc2C1)N1CCCC(Cc2ccccc2)C1 9961,Cc1cc(C)n(C(C)CC(=O)NCCC(C)NC(=O)CSCc2ccccc2)n1 9962,C(=O)(CC(=O)N(CCNC(C1(C2CCCCO2)CC1)=O)C1CC1)NCC#C 9963,N1(C(c2c(CC)cccc2)=O)CCCC(NC(c2cnc(S)nc2)=O)C1CC 9964,C(=O)(C1=CC2(CCOC2)C1)NCC1(CC(C(=O)CCCn2cncn2)=O)CC1.NC 9965,c1(C(N2CC(NC(CCC=CC)=O)C(O)C2)=O)ccc2sncc2c1 9966,CCC(CC)(C(=O)NCC1(O)CC(NC(=O)C(n2nccc2C)C)C1)OC 9967,C(=O)(C1=CC2CCCCCC12)NC1CC(F)(CNC(c2ccc(C)o2)=O)C1 9968,N1(C(C(C)OC2CCCCC2)=O)CC(C2CCCN(C(=O)C=CS(C)(=O)=O)C2)C1 9969,Cc1cc(C(=O)NCCC(C)NC(=O)C(C)C#N)n[nH]1 9970,N1(C(CN(C2CCCCC2)C)=O)CC(F)(F)CC1(C)CNC(c1csc(Cl)n1)=O 9971,c1(CNC(c2cc(C)ncc2)c2nnnn2-c2ccccc2Cl)cc(Cl)cc(Br)c1 9972,c1(C(N2CC(CNC(C3(CF)CCC3)=O)C3(CC3)C2)=O)cnc2n1CCCC2 9973,C1(NC(C(CC)(C)F)=O)CN(C(=O)CCCOc2cccc(C)c2)CC1(C)C 9974,CCC(C)(C)C(O)C(=O)N1CCC(NC(=O)Cc2scnc2C)C1 9975,N1(C(CCOCCOC)=O)CCCC12CCN(C(C1CCCCC1C)=O)CC2 9976,c1(OC)ccc(C=CC(=O)NCC2CN(C(C3OCCC3C(C)C)=O)C2)nc1 9977,C(=O)(CC1CCC(=O)c2ccccc21)NCCNC(C(C)C1CCC1)=O 9978,c1(C(N2CC3(CC(CNC(C4(CC)CC4)=O)OC3)C2)=O)cnc2c(c1)CCCO2 9979,c1(C(=O)NC(CCNC(C2N(C(C)=O)CCC2)=O)C)cccc(Br)c1 9980,CC(C(=O)N(C1CN(C(c2nn(C(F)F)cc2Cl)=O)CC1O)C)C(C)(F)F 9981,CCCC(CCC)C(=O)NC1CCC(C)N(C(C2(c3ccccc3Cl)CC2)=O)C1 9982,C1(C(=O)OCC)C(NC(=O)NCc2cc(C(F)(F)F)n(C)n2)C2CCCCCC12 9983,N1CCC2(C=C(C(=O)N)C2)C1.CC1(C)CCCC(N2CCC2C2CCOCC2)C1 9984,C(CCCC(=O)N1CCC1CNC(C1(F)CCCOC1)=O)N(C)C 9985,c1(C(=O)NCC(CC=C)NC(=O)CC(C)N(C)C)c(OC)cccc1C 9986,c1(C(=O)NCC(CC)NC(c2cc(O)ncn2)=O)ccnn2ccnc12 9987,N1(C(C2(COC)COC2)=O)CC(C(N2CCCCCC2)=O)C(C2CC2)C1 9988,c1(N(C)Cc2ccncc2F)cccc(S(=O)(=O)NC2CSC2)n1 9989,C1(C(N2CCC(C)(NC(=O)CCCC(N)=O)CC2)=O)CC(F)(F)C12CCC2 9990,c1(CCC)cccc(C(C)C)c1NCCN1CCC1C1CCCCO1 9991,C(=O)(CS(=O)(=O)C(C)(C)C)NC1C(C)CN(C(c2scnc2C(C)(C)C)=O)CC1 9992,c1(CC(=O)NCCOCCN(C(CC(=C)C)=O)C)ccc2c(c1)ncn2C 9993,N1(C(c2ccc3nc(C)oc3c2)=O)CCc2ccccc2C1CNC(=O)C1CC1 9994,C1(CNC(=O)C(N2CCOCC2)C2CC2)CC(O)CN(C(C23CCC(CC2)O3)=O)C1 9995,N1(C(C2(CC)COC2)=O)CCCCC1C1(NC(=O)CN2CC(C)(C)C2)CC1 9996,c1(C(=O)NC2CC(NC(c3ccccc3O)=O)C2)cc2ccc(Br)cn2c1 9997,N1(C(CCNS(C)(=O)=O)=O)CCCC1C1(OCCNC(=O)Cn2nccn2)CC1 9998,C1(C)(CNC(C(CC)N(C)C)=O)CCCN1c1nccc(-n2ccnc2)n1 9999,Cc1cnccc1C(C)C(=O)N1CC(CNC(=O)CC2CCOC(C(C)C)C2)C1 10000,c1(C(N(C(C)C(=O)O)CCF)=O)ccc(CNC(C23CC(C2)NC3=O)=O)cc1 10001,C(CCCC(C)N(C1CCCCC1)C(c1ccccc1)=O)NC(C(C)CC1CC1)=O 10002,c1(C(C(=O)N(C(C)CNC(=O)C2=COCC2)CC)C)ccc(C(F)F)cc1 10003,C(=O)(C1=NOC(CNC(c2ncsc2C)=O)C1)N(C1CCN(CC)C1)C 10004,C(CCSC)(C(=O)NC(c1nccc(C)n1)C)NC(c1cc(OC)ns1)=O 10005,C(=O)(CC(C)(C)C(=O)NC1COCCC1NC(c1cc(CC)c(C)s1)=O)OCC 10006,c1(CC(=O)NCCC(O)CNC(C2(CO)CCCC2)=O)ccc(Cl)cc1Cl 10007,N1(C(C(C=CC)O)=O)CCC(c2ccccc2CNC(C2(SC)CC2)=O)CC1 10008,N1(C(CCC2CCN(C(C3(OC)CCOC3)=O)CC2)=O)CC2C(C1)C2(F)F 10009,C1(CNC(c2cn(C3CC3)cn2)=O)C2CN(C(c3c[nH]cc3Br)=O)CC12 10010,C1(NC(CNC(c2nncc(OC)c2)=O)=O)C2C=CC(C2)C1CO 10011,c1(C(=O)NC2C(CNC(CC(C)c3ccncc3)=O)C2)nnc2n1CCCCC2 10012,n1(CCC(=O)N(CCOC)CCNC(C2CCC=CC2NC)=O)cccnc1=O 10013,CCC(CC1CCCC1)C(=O)NCCNC(=O)CNC(=O)Nc1ccc(Cl)cc1 10014,CS(=O)(=O)C(CNC(=O)C=CC1CCOCC1)CNC(C1(F)CC=CCC1)=O 10015,n1(CC)nnc(C(=O)NCC(C)(C)C(=O)NC(c2ncn(C)n2)C)c1C 10016,C1(C(=O)NCc2c(C(=O)NCC(C3CCC3)OCC)n[nH]c2)CCCCC1C 10017,N1(C(Cc2c(C)ccs2)=O)CCOC(CCC(N2CCC(C(F)F)CC2)=O)C1 10018,N1(C(CN(C(C=C)=O)C(C)=O)=O)CCN(C(=O)Cc2c(C)noc2C)CC1C 10019,C1(C(=O)N(CC(C)O)C)(CNC(C2C(C(=O)OC)C2)=O)CCCC1 10020,N1(C(C2(C)CCC2)=O)CCC2(CCCN2C(=O)CS(=O)C(F)(F)F)C1 10021,c1(COC)nc(CNC(=O)C(=O)NC(c2ccccc2)c2ccco2)cs1 10022,c1(CC)cccc(CC)c1CC(=O)N(C)CC1CCCN1C(C1CCOC1C)=O 10023,N1(C(c2c(CC)nco2)=O)CC2OCCN(C(=O)C(C)C(O)C(C)C)C2C1 10024,CC1(CNC(C2CC(O)C(F)C2)=O)CCN(C(=O)CCn2cnccc2=O)CC1 10025,Cc1cc(C(N2CC(CCO)OC(C)C2)=O)cc2cccnc12 10026,N12CCCC(C1)N(C(=O)C(C)C)C1(CC1)C2=O.C(C(C)C)NC(C)=O 10027,CC1(CNC(c2ccnc(S)c2)=O)CN(C(c2cccc(Cl)c2Cl)=O)CCO1 10028,C1(C)(CC)C=C(C(=O)NC2CC2NC(C2(C(=O)OC)CC2)=O)C1 10029,C1(C2(C(N)=O)CC2)CCCCN1C(C1CCCOC1)=O.c12sccc1CNC2=O 10030,c1(C(=O)NC(C2(CO)CC2)C)ccc(F)cc1O.c12ccc(cc1)CNC(=O)C2 10031,C1(C(=O)NCCNC(=O)OCC)CC=CCN1C(c1ccsc1C)=O 10032,C(=O)(CCCCCCCC1CC1)NC(C)CNC(c1c(Cl)cnn1C)=O 10033,c1(-c2cc(C(N(CCCNC(CN3C(C)CC3)=O)C)=O)on2)cccc(F)c1 10034,C1(C)(CNC(C(C(C)C)OCC)=O)CCN(C(=O)C(C2CCCCC2)F)CC1 10035,O=C1CCC(C(=O)NC2CC3CCC2N3C(C2(O)CCOC2)=O)=NN1 10036,N1(C(=O)C(O)C2CCCC2)CCC2(CC1)CCN(c1nc(O)c3c[nH]nc3n1)C2 10037,C(C#CC(=O)N(C1CC(C(=O)OCC)C1)C)NC(C=CCCC)=O 10038,CC1(C)CN(C(=O)CC2(CO)CC2)CC1NC(C1(C)CCCS1(=O)=O)=O 10039,C1(NC(c2c(CC)onc2C)=O)CCCN(CCOc2ccc(Cl)cc2Cl)CC1 10040,C(CO)(C(C)(C)C)NC(CC1CC(C(=O)Nc2c(OC)ccs2)C1)=O 10041,C(C(C)C(=O)N(C)CCC1CN(C)C1)NC(CCOC(C)=O)=O 10042,CCCCC(C)CCC(=O)NCCNC(=O)C(c1ccccc1)n1cccn1 10043,C1(CNC(COCC#C)=O)CCC2CN(C(c3ccncc3CC)=O)CCC2C1 10044,C1(=CC(N2CC(NC(=O)C(F)=C3CCC3)CC(C)C2)=O)CCOc2ccccc21 10045,c1(CC)ccc(C(C)C(=O)NCC(O)CNC(=O)CCc2cncs2)cc1 10046,c1(CC(=O)NC(CNC(c2c(CC)n[nH]c2)=O)C2CC2)cc(C)ccc1Br 10047,c1(CC(=O)NC2CN(C(c3cc[nH]n3)=O)C3CC23)ccc2c[nH]nc2c1 10048,N1(C(c2c(C)cc(CNC(CC3ON=C(CC)C3)=O)o2)=O)C2CCC1CC(F)C2 10049,C#CCCCC(C(=O)NCCSC)N1CCC(CCn2cccn2)C1.OC 10050,C(CCCCC(=O)N1CCC(N(C)C(c2ccnc(C3CCC3)c2)=O)C1)OCC 10051,c1(NC(C)=O)cccc2c1CCCN2C(C1OCCC1C(C)C)=O 10052,C1(NC(C)=O)CCC12CN(C(C1CCC(C(N)=O)CC1)=O)C2 10053,Cc1nc2ccc(C(=O)Nc3cc(Cl)cnc3OC(F)F)cc2n(C)c1=O 10054,C1(C)(OC)CCCN(C(C2(F)CCN(C(=O)CCCCC3CC3)CC2)=O)CC1 10055,c1(-n2cc(CCCC)nn2)cccc(C(=O)OC)c1.C(C(=O)N(CCSC)CC)N 10056,C(=O)(C(C)(F)C(=O)N1CCCC(C)C1)OCC.C1CO1 10057,N1(C(c2cc(C)c(O)cc2)=O)CC(F)(F)CC1(C)CNC(C1CCC1(C)C)=O 10058,N1(C(c2nc(C(N)=O)sc2)=O)CC(CNC(C2CS(=O)C2)=O)N2CCC1C2 10059,CC1(C)CC(NC(c2ccc(C(C)(C)C)o2)=O)CC(O)C1 10060,c1(C(=O)NCC2CCC(CNC(C3CC34CCOC4)=O)CC2)ccc(F)c(Cl)c1 10061,c1(C(N2CC3C(NC(C4CCC(C)O4)=O)(C3)C2)=O)cc2c(Cl)cncc2s1 10062,CS(=O)c1ccc(CC(=O)NCC(O)CNC(c2conc2C2CC2)=O)cc1 10063,C1(NC(CCC2CCCN(C(c3c(CC)occ3)=O)C2)=O)CNC(=O)C12CC2 10064,CCCC(O)CC(=O)N(CC(O)CN(C)C(c1nc(C)ncc1Br)=O)C 10065,C1(COC)(NC(=O)CC2CCCN2C)CCN(C(=O)C=C(C)C)C1 10066,c1(C(=O)NC2CC3(C(N4CC(N5CCC5)C4)=O)COC2C3)cn2ccccc2n1 10067,CC(CCC(C)(C)C)C(=O)N1CC(C2CC2C(=O)NCC2CC3CCC2O3)C1 10068,C(c1ccc(F)c(OC)c1)=CC(N1C2CC(NC(CCCCOC)=O)C2CC1)=O 10069,N1(C(C(C)NC(CC)=O)=O)CC2CC1CCC2NC(=O)C(C)=C1CCC1 10070,c1(CC(N2CC(CNC(C3C(=C)C3)=O)C(F)(F)C2)=O)nc2nc(C)cc(C)n2n1 10071,C#CCC(CC(=O)NC1CCCCCC1)NC(c1cccc(C)c1C)=O 10072,C(C(C)(C)C(=O)NC(CNC(C1(c2ccccc2)CCCO1)=O)C1CCC1)SC 10073,c1(N(C)C)ccc(F)c(C(=O)NCCCCn2cc(-c3cccnc3F)nn2)c1 10074,N1(C(c2c(C)cc(SC)o2)=O)CCC(C)C(NC(C2OC(C)CC2C)=O)C1C 10075,N1(C(c2c(C)oc(C)c2Br)=O)CCN(C(=O)C(C)N(C)C)CC(C)(F)C1 10076,N1(C(c2c(C)noc2C2CC2)=O)CCCC(CC(=O)NC2(CC(C)=O)CC2)C1 10077,c1(C(N2CC(F)(CN)C2)=O)cccc(C2CC2)c1.C1(C=O)CC(n2cnnc2)C1 10078,C1(C(=O)NC(CC)CN(C)C(C2(OC(C)C)CCCC2)=O)CCC(F)(F)C1 10079,c1(C(N2CCC(CNC(CCC)=O)C(F)(F)C2)=O)cc([N+](=O)[O-])cc(Br)c1C 10080,Cc1ccc2nnc(C(=O)N(C)CCNC(C3(C)CCOC(C)C3)=O)n2c1 10081,N1(C(CC2CN(C(c3ccc(CC)s3)=O)CC23CC3)=O)CCn2ncc(C)c2C1 10082,C1(C#N)(CC(=O)N(CCCNC(=O)C(C)CC2CC2)CC)CCOCC1 10083,C(=O)(C(CC(C)C)NC)N(CCN(C(=O)C(O)C1CC1)Cc1ccccc1)CC 10084,C1(F)(C(=O)NCCCN(CCCCNC(C=C(C)C)=O)C)CCCC1 10085,c1(-n2cc(C3(N(CC(C)C)C)CCC3)nn2)ccnc(Br)c1.N12CCCC1C2=O 10086,N#CC1CN(C(c2cc(Cl)ccc2Cl)=O)CCN1C(c1cnnc(Cl)c1)=O 10087,CCCCC(O)CC(=O)NCC1CCC(C(=O)NCC2CC2CC)O1 10088,C1(NC(CC2(C)N(C(CC(=O)NCC)=O)CC2)=O)C2CCC1CC2 10089,C(C(F)(F)C(=O)NCCC1CCN(C(=O)CC2CCNC2=O)CC1)N(C)C 10090,N1(C(CCC2C(C)(C)C2)=O)CCN(CCNC(C2CC(=C3CCC3)C2)=O)CC1 10091,N1(C(C=COCC)=O)CCCC(N(C(=O)CCOCC2CCCO2)C)C1 10092,N1(C(Cn2ccc(C)n2)=O)CC2(C1)CN(C(=O)Cc1ccnc(F)c1)CC2CO 10093,c1(OC)ccc(-c2nc(C)c(C(C)NC(c3nnnn3C3CC3)C3CC3)s2)cc1 10094,c1(OC)cc(C)cnc1C(=O)NC1(C(=O)O)CC(OC)C1 10095,N#Cc1c(F)cc(C(=O)NC2CC(CNC(=O)C3=CSCCO3)C2)cc1F 10096,C12(CNC(C(C)=CC)=O)CC(CO1)N(C(=O)Cc1ccccc1CC#N)C2 10097,C(C(C)(C)CCC#N)N(CCCCOC)Cc1cccc(Br)c1 10098,Cc1ccc(CN(C)C(C2(NC(=O)Cc3ccnc(O)c3)CC(O)C2)=O)cc1 10099,N1(C(CC(CC)SC)=O)CCC2(CC(NC(c3csc(O)n3)=O)C2)C1 10100,C(=O)(C1=C(CCl)N(CC2CC2)C(=O)NC1c1ccc(-c2ccccc2)o1)OCC 10101,C(=O)(C#CC1CCOC1)NCC1C(C(=O)NC2C(C)(C)C2(C)C)CC1 10102,C(=O)(C1=CN(C)S(=O)(=O)N=C1C)NCC(CN(C(C(C(CC)O)(C)C)=O)C)(C)C 10103,C(=O)(C(CN=[N+]=[N-])NC(c1nnc(C(C)CCCO)o1)=O)OCCN1CCN(C)CC1 10104,CCCC(C(=O)NCCCN(C(C)C)Cc1csc(C(C)C)n1)OC 10105,N1(C(CC(=C)Br)=O)CC2CCCC2(NC(=O)CCc2ccccc2Cl)C1 10106,Cc1cc(P(C)(C)=O)oc1C(=O)NC(C)CNC(c1cc(C2CC2)cs1)=O 10107,N1(C(C2(CSC)CC2)=O)CCC2(C1)CN(C(c1n[nH]c(C)n1)=O)C2 10108,N1(C(C=C(COC)C)=O)CC2ON=C(CNC(c3csnc3Br)=O)C2C1 10109,C1(NC(CCC#CC)=O)CC2(NC(c3scnc3COC)=O)COC1C2 10110,C1(C)(CCNC(C(C)O)=O)CCN(C(c2ccc(-c3cccnc3)cc2)=O)C1 10111,c1(C(=O)OC)cccc(C(N2CCC(NC(=O)CC3CC(SC)C3)C2C)=O)c1 10112,Cc1ccc2c(CCC(=O)N3CC(N(C(=O)CCCS(C)(=O)=O)C)C3)c[nH]c2c1 10113,C1(C)(CCC(=O)NCC(CNC(C(C)=C(CC)C)=O)O)CC1(F)F 10114,C=C(C)CCC(=O)NCCC1CC(NC(=O)C(F)(F)c2nc(C)cs2)C1 10115,N1(C(CCCCNC(Cc2ccc(C)nc2)=O)=O)CCN(C)C(CO)C1 10116,N1(C(c2c(C)cccc2O)=O)CC2(C1)CN(C(=O)CN1CCC1C)CC2CO 10117,C1(C(N2CC=C(C)C2)=O)(C(C)C)CCN(C(=O)CCC2CCC2)C1 10118,CC(C)CC(O)CNC(=O)CCCCN(C)C(C1(CO)CCCCO1)=O 10119,c1(C(N2CCCCC2C2CCCC2O)C(=O)NCC)cc(Br)ccc1F 10120,CC1(C)C(c2cccc(Cl)c2)CCN1C(c1nn(CC(F)(F)F)cc1Cl)=O 10121,c1(C(=O)NC2CC(NC(c3c(CC)nccn3)=O)C2)nc(C2CC2)ncc1Cl 10122,CN1CCCC1(C)C(=O)NCCOC1CN(C(=O)CC2CCCS2(=O)=O)C1 10123,C(=O)(C#CC1CCCO1)OCC(=O)NC1CC1 10124,C1(C(=O)NCCCCNC(C(C)CN2CCOCC2)=O)Cc2ccc(F)cc2O1 10125,C1(CN(C)C(c2cc(C(F)(F)F)ns2)=O)CCCCN1C(c1csc(Cl)n1)=O 10126,c1(C(=O)NCCCCCN(C(c2ccc(CC)nc2)=O)C)ccc(C)c(N)c1 10127,c1(C(=O)NCC2N(C(c3ccsc3)=O)CC(C)(C)OC2)cnnc2ccccc12 10128,C1(NC(c2c(C)nns2)=O)CCCN(C(=O)CC2CCN(C)C2)C1C 10129,c1(C(=O)NC(C2C3CNCC23)C(=O)OC)csc(Cl)c1OC 10130,c1(OC)ccc(O)cc1C(=O)NCC1CCCC(NC(C2CC(F)C2)=O)C1 10131,c1(C(N2CC(N(C(c3c(C)nccc3)=O)C)C(F)C2)=O)cc(C2CC2)nnc1O 10132,c1(CC(=O)N(C2CCN(C(c3c(CC)cco3)=O)C2)CC2CC2)cncnc1O 10133,n1(-c2cn(C)nc2)nc(OC(F)(F)F)nc1-c1cnco1.C1CCC1 10134,CC(CCN(C(=O)CCc1nncs1)C)NC(C1CC1CN(C)C)=O 10135,Cc1cccc(N2CCC(NC(=O)C(=O)Nc3n[nH]c(Br)n3)C2)c1 10136,N1(C(c2cn(CCO)nn2)=O)CCC2CN(C(C3CC(C4CCC4)C3)=O)C2C1 10137,C1(N2CCCCC2)(C(=O)NC)CCN(C(C2C3CC(=O)CC32)=O)CC1 10138,c1(C(=O)NCC(CN(C(c2ncc(C)c(C)c2)=O)C)C)ccc2ccnn2c1 10139,C1(C(N2CC(OC)(CNC(=O)C(C)C3CCCC3)C2)=O)COC(=O)N1C 10140,N1(C(C2CC(SC)C2)=O)CC(NC(c2csnc2C)=O)CC12CCCC2 10141,CC(=O)CCCC(=O)NCC1C(O)C(O)CN1C(c1c[nH]nc1Br)=O 10142,C1(NC(c2c(C(C)C)nns2)=O)CN(C(=O)C2=CSCCO2)CCC1CO 10143,N1(C(c2cnn(C)n2)=O)CC(NC(=O)C(F)(F)C2(O)CCC2)CC12CCOCC2 10144,CCC(C(=O)NCC1(CCNC(=O)Cc2ccncc2Cl)CC1)C(F)(F)F 10145,C12(NC(=O)COc3ccon3)CCCN(C(C3(CO)COC3)=O)CC1C2 10146,N1(C(CCC=CC)=O)CC2CC1C2C(N1C(C)CC1(C)C)=O 10147,C1(C2CN(C(=O)C(F)(F)C3(O)CCCC3)C2)(NC(c2ccc(CF)cc2)=O)CC1 10148,c1(C(=O)NC(c2cccc3cc[nH]c23)CC)cnn2cc(-c3nn[nH]n3)cnc12 10149,c1(C(N(CC(CN(C(=O)CC2CCCC2)C)O)C)=O)cc(P(C)(C)=O)cs1 10150,CC1CC(C(=O)NCCC(=O)NCC(C)S(C)(=O)=O)=NO1 10151,c1(N(C(CNCCC(=O)N(CC)CC)=O)C)cc(Br)c[nH]1.C(C)(=O)O 10152,c1(C(=O)NCC(CNC(CCCOCC=C)=O)O)ccc(S(=O)(=O)C(F)F)cc1 10153,Cc1cccc2c(C(=O)NC(C)CN(C)C(C34CCCCC3C4)=O)n[nH]c12 10154,c1(C(=O)NC2CC(F)(CNC(C3(C4CCCO4)CCC3)=O)C2)cc2cn[nH]c2cn1 10155,c1(C(=O)NCCC2(NC(C3C(C)(C)C3(C)C)=O)CCC2)ccccc1[N+](=O)[O-] 10156,CC1C(=O)CC2CCC1N2C(=O)NNc1nccs1 10157,Cn1cc(SCC(=O)NC2(CNC(=O)C(C)(c3cccs3)SC)CCOC2)cn1 10158,c1(C(=O)NCC2(F)CC(CNC(C(F)=C(C)C)=O)C2)cccc(Br)c1C 10159,c1(C(N2C(CNC(C(C(C)C)C)=O)CC(O)C2)=O)cc(=O)n(C)cc1Br 10160,c1(NC(c2ccc(-c3ccc(Br)s3)s2)=O)ncccc1OCCF 10161,C(=O)(C(O)C1=CCCCC1)N1C(C2(NC(CC(=O)NCC)=O)CC2)CCC1 10162,CCC(C)(CS(C)(=O)=O)C(=O)NCC(CNC(=O)CCOCC(F)F)C(F)(F)F 10163,c1(C(=O)NCC2(F)CC(NC(C(CC)N(C)C)=O)C2)cc2c(C#N)cccc2[nH]1 10164,N1(C(COCC#C)=O)CC(C2CCCN(C(C3(CC)CCCO3)=O)C2)C1 10165,N1(C(Cc2c(C)nc[nH]2)=O)CCC(CO)C(NC(C2(C(C)C)CCC2)=O)C1 10166,CN1CCC(C(=O)NC2COCC2CNC(=O)Cc2cccnc2Cl)CC1=O 10167,c1(C(N(CCC(C)NC(=O)C(C)(C)C)C)=O)ccc2c(c1)OC(C)(C)OC2 10168,CC(C1OCCc2ccccc21)NCc1csc([N+](=O)[O-])c1 10169,O=C(C(CCC1CCC1)NC(C1CC=CC(O)C1)=O)NCc1ccc(O)nn1 10170,N1(C(Cc2c(C)scc2)=O)CCC(C(=O)NCCC(F)=C(F)F)C1(C)C 10171,C1(NC(C(C)Nc2cccnc2)=O)COCCN(C(C2C3COCC23)=O)C1 10172,N1(C(c2ccc(CNC)c(C)c2)=O)CC=CCC12COC2 10173,C1(CNC(CNS(N)(=O)=O)=O)CC2(CCC2)CN1C(c1cccc(C2CC2)n1)=O 10174,n1(C(C)C)nccc1S(=O)(=O)N(C)CCOC(=O)OC(C)(C)C.C1CCN1 10175,N(C)(S(=O)(=O)N(C)CC1CC1)CC#C 10176,c1(C(C(=O)NCC=CCl)NC(CN(C)CC)=O)cnn(C)c1 10177,C1(c2nc(C)[nH]n2)CCN(N2CCCC(CO)(CO)C2)CC1 10178,N1(C(CCn2cc(CC3C(C)(C)C(O)C3)nn2)=O)CCOCC2(CC2)C1 10179,C1(CNC(CN(C2CC2)CC)=O)CN(C(c2cscc2OC)=O)C2CC12 10180,C(N=c1[nH]c(N(C)Cc2ccc(Br)cc2)nc2c1CCCCC2)c1cc(C)sc1 10181,C(=O)(CS(=O)(=O)CCO)NC1CCCC(NC(c2cncc(SCC)n2)=O)C1 10182,N1(C(C(COC)CC(C)C)=O)CC(C)OC2(CCN(C(=O)CCCSC)CC2)C1 10183,C1(C(N2CC(NC(c3c(COC)noc3)=O)C2)=O)CCCCC12OCCO2 10184,c1(OC)ccc(C)cc1C=CC(N1CCC(NC(=O)C(C)(C)SC)C(F)C1)=O 10185,c1(N2CCCC(NC(=O)C(C)CCC(C)(C)C)C2)ncnc2ccc(OC)cc12.CO 10186,C(CC(C)C(=O)NC1CCC(F)(CNC(c2c[nH]nc2C(C)C)=O)C1)OC 10187,Cc1nsc(NC2CC2)c1C(=O)NCC1CC(O)CN1C(=O)CC(C)F 10188,C(CC(C)C(F)(F)F)NC(C1(CF)CCN(C(c2cccc(C)c2)=O)C1)=O 10189,C1(CNC(CSCCC)=O)CC(C(=O)NCC2C3CCCCCC23)=NO1 10190,N1(C(C(C2CN(C(=O)CC3CC=CC3)C2)OC)=O)CC(OC)C(C)(C)C1 10191,C1(NC(C2C(CC)CCC2)=O)CC2(CCN(C(C3(C)CCN(C)CC3)=O)C2)C1 10192,C1(NC(C2(OC)CCSC2)=O)CCN(C(=O)C(c2c(C)noc2C)C)CC1CO 10193,c1(C(N2CCC(O)(CNC(C3C(CCOC)C3)=O)C2)=O)ccc([N+](=O)[O-])o1 10194,C(=O)(C(C)(O)C(C)C)N(CCC(=O)NC1C2CCCC12)CC 10195,C=C(C)CCCC(=O)NCC1(O)CCCN(C(c2cc(COC)on2)=O)C1 10196,C1(NC(C(C)OCC)=O)CCN(C(=O)Cc2ccc(C(C)=O)s2)CC1(C)C 10197,CC(C)C(C(=O)NC(CNC(=O)Cn1cnnn1)C(C)(C)C)NC=O 10198,c1(CC)[nH]nc(C(=O)N(CC(=O)N(C2CCCCC2C)C)C)c1C 10199,N1(C(=O)OC(C)(C)C)CCCC(Cn2cc(CC(=O)NC)nn2)C1 10200,N1(C(=O)NCc2ncc(CC)o2)CCCCC1CCNC(C)=O 10201,c1(CN(C(CNC(c2ccc(OC)nc2Cl)=O)C)C)cccc([N+](=O)[O-])c1 10202,N1(C(CNC(CCCC2(NC(N)=O)CCC2)=O)CO)CCC(OC2CC2)CC1 10203,CC(C(=O)NCc1cnsc1)F.C1CCCC2CN1C2 10204,Cc1ncc(CNC(=O)COc2ccc(-c3ccccc3)nc2)cc1Br 10205,C(=O)(C1CCc2ccccc21)NC1(C(=O)NCC(c2cnc[nH]2)C)CCCC1C 10206,C1(C(=O)NC(c2ccns2)C)(CC)CCCN(C(c2cnn(C(C)C)c2)=O)C1 10207,C#CCCCCCC(=O)N1CC(C2CN(C(C3CCCOCC3)=O)C2)C1 10208,Cc1cc(C(=O)OC(C(=O)Nc2ccc(N(C)C)c(F)c2)C(C)C)ncc1N 10209,c1(NC(C(CCC)C)CO)ccc(S(=O)(=O)NCc2cc(C)c(Br)cn2)cc1Br 10210,c1(C(=O)NCCC2CCCN(C(C3CC(F)C3)=O)C2)nccc2n[nH]cc12 10211,c1(C(N(CCN(C(c2cncc(N)c2)=O)CC)CC)=O)cn(C(C)C)cc1C 10212,N1(C(CC(C)OC)=O)CC2(CCN(C(=O)C(C)Sc3ccc(N)cc3)C2)C1 10213,c1(NC(C2(C)CCN(C(C3CC3F)=O)CC2)=O)sc2c(c1C#N)CCCC2 10214,C1(C#N)(C(=O)NC2CCCN(C(C(CCC)=CCC)=O)CC2)CC2CCC1CC2 10215,C(=O)(C(CC)(CC)OCC=C)NCC=CCNC(C(CC=CCC)C)=O 10216,c1(NC(=O)NCc2cccc(-c3cccc(OC)n3)c2)ccc2sc(O)nc2c1 10217,c1(C(N2CCC(C)C2C(NCP(C)(C)=O)=O)=O)cnn2c1CCC2 10218,O=C1CC2(CCCN(C(=O)C3=NOC(CO)C3)CC2)N1 10219,CC(CN(C)C)C(=O)N1CCCC1C(C)NC(=O)N(C)C 10220,C(=O)(C(CNC(C1CC1(F)Cl)=O)C(C)C)N1CCC(C(=O)NC)C1C 10221,C1(CNC(CSC)=O)CN(C(c2cc(C(C)(C)C)nn2C)=O)C2(CCC2)C1 10222,CCCC(CCC)CC(=O)NC1CN(C(C2CCCOCC2)=O)CC1OC 10223,C(C1c2ccccc2CN1C(=O)C(C)=CC(C)(C)C)NC(C(C1CC1)OC)=O 10224,c1(N(C2CCN(C(c3cnc(SC)s3)=O)C2)C)ncnc2sc(C(F)(F)F)nc12 10225,S(=O)(=O)(c1ccc(CC(=O)NCC2CCCN2C(=O)C(C)C(C)O)cc1)NCC 10226,n1(CC(=O)NCCCN(C(=O)CC2(O)CCC2)C)ncccc1=O 10227,c1(C(N2CC(O)CC(NC(CC(=O)NCC)=O)C2)=O)cnn2cc(OC)ccc12 10228,N1(C(C2CC(C)N2C(c2c[nH]nc2C(F)F)=O)=O)CCN(C)C(C2CC2)C1 10229,C1(N(C(C(=O)Nc2ccccc2)=O)CCCO)CC2CC1CN2 10230,c1(C(=O)OCC)ccccc1NC(C1CC1CNC(=O)CCc1ccn(C)c1)=O 10231,CC(CNC(C1(F)CCN(C(c2ccc(Cl)cn2)=O)CC1)=O)CC(F)(F)F 10232,C1(C(=O)NCC(CNC(Cc2c(C)n[nH]c2)=O)C)CCCN(C(C)C)C1 10233,c1(N2CCOCC(CNC(c3nc(CCC)sc3)=O)C2)nnc(C)c(C)c1C#N 10234,c1(NC(C2CCC(NC(C3N(C)CCCC3)=O)C2)=O)ccc(O)c(Br)c1 10235,CN1CCCC1C=CC(=O)NC1(C(=O)N(C2CSC2)C)CC(F)C1 10236,C12(CNC(c3ccccc3)=O)CCC1CN(C(c1ccc(=O)n(CCO)c1)=O)C2 10237,C1(CC(=O)NCc2nccc(OC)n2)(CO)CCN(C(C2CCOCC2)=O)CC1 10238,N1(C(Cc2cn(CC)nc2)=O)CC(C(=O)NCC2CC=CC2)C(C(C)C)C1 10239,C1(OCC)CC(NC(=O)NCCNS(=O)(=O)c2c(C)noc2C)C12CCCCC2 10240,c1(OC)nsc(OC)c1C(C)NC(C1(n2cc(F)cn2)CC1)=O 10241,C1(O)(CC#C)CCN(CC2(CC=C)CCOC2)CC1 10242,C12(CC)CCCN(C(N(CCCCCC=C)C=O)=O)CCC1C2.C(C)(C)(C)ON 10243,C1(C(=O)OC)CCOC1C(=O)NCCN(C)C(C1CC(C(C)C)C1)=O 10244,C(CCCC(=O)N1CC2C(C)C2C1)NC(COCC)=O 10245,CCS(=O)(=O)CC(=O)N1CCC(CN(C)C(c2cccc(OC)c2OC)=O)C1 10246,c1(C(N2CCC(O)(CNC(C(C)(C)OCC)=O)C2)=O)cc(Cl)c(OC)cc1C 10247,C(=O)(C(C)(C)CS(C)(=O)=O)NCCCC(C)NC(=O)C(O)CC(N)=O 10248,C(=O)(CC(C(C)C)SCCOC)N1C(N(C(=O)C(=O)NCC2CC2)CC)CCC1 10249,C(=O)(C(C)CC(C)C)N1CC(OC)C(NC(=O)C(F)(F)CN(C)C)C1 10250,Cc1cnc(Cl)[nH]c1=NCC=Cc1ccc(NC(=O)CC2CC(F)C2)cc1 10251,N1(C(c2c(Cl)ncc(C)c2)=O)CC2CCN(C(c3cc(Cl)c(Cl)cn3)=O)C2C1 10252,c1(C(C)=O)cc(NC2CCN(C(=O)CCC(C)CN(C)C)CC2)ccc1[N+](=O)[O-] 10253,N1(C(C(C)SC)=O)CCOC2(CCN(C(c3cccc4c3OCC4C)=O)CC2)C1 10254,c1(C(N(CC(CN(C(c2c(C)noc2N)=O)C)O)C)=O)cc(Cl)ccc1Cl 10255,N1(C(CCC2C(C)C2)=O)C2CCC1CN(C(c1csnn1)=O)C2 10256,Cc1cc(C(=O)NCC2CN(C(=O)COCCF)CC2C)c2c(C)nn(C)c2n1 10257,c1(C(=O)NCC(C2N(C(C(CC)CC)=O)CCCC2)(C)C)cnc2ccnn2c1 10258,N1(C(C(C)N(C(c2nsnc2O)=O)C2CC2)=O)CC23CCC2(COC3)C1 10259,c1(NC(C2(C)CCN(C(c3ccc(CF)cc3)=O)C2)=O)ccc(F)c(O)c1 10260,Cc1nn2c(C(N3CC4CC4(NC(=O)C(C)C(=O)OC(C)(C)C)C3)=O)c(C)nc2s1 10261,CCC(Cc1cccc(C)c1)C(=O)NCC(C(C)C)NC(=O)C(Cl)=CCl 10262,C(=O)(C(C(=O)N1CCCC(CNC(=O)CCCC)C1)OC)OCC.C(C)(=O)OCOC 10263,C(=O)(CC(C)C(F)(F)F)NC(C(NOC)=O)=O.C1CCN1CCO 10264,C1(CCNC(CCC#CC)=O)CN(C(C2CC3CCC3C2)=O)CCS1(=O)=O 10265,C1(C(=O)NC2(CCC)CC2)C(C2CC2)CCN1C(=O)COCCCF 10266,C1(NC(c2ccc(CS(=O)(=O)N(C)C)cc2)=O)CCCN(CCCCF)C1=O 10267,N1(C(CC2(C(=C)F)CCC2)=O)CCC(C(=O)NCC(Cl)C(C)(F)F)C(C)C1 10268,N1(S(CC)(=O)=O)CCC(C(=O)NC(C2CN(C(=O)C=CCOC)CCO2)C)CC1 10269,C(=O)(CCC(=O)NCCCCCCNC(C1CC1(Br)Br)=O)NCC 10270,C1(NC(CC2CN(C(C)=O)C2)=O)CN(C(c2cc(Cl)ccn2)=O)C2(CCOC2)C1 10271,c1(C(N2C(C)C(NC(c3cccc(N)c3)=O)CC2)=O)cc2ncccc2s1 10272,C1(NC(c2cc(CNC(C(C)(C)OC)=O)nn2C)=O)CNC(=O)C12CC2 10273,C#Cc1ccc(C(N2CCCC2CCC(N2CCOCCC2C(N)=O)=O)=O)cc1 10274,c1(CC(N2CCC(Cc3cn(CCO)nn3)C2)=O)ccc2c(c1)CCO2 10275,C(=O)(C(CC(C)C)C(C)C)NCCN1CCN(C(c2c(N)ccc(C)c2)=O)CC1 10276,Cc1c(CN2CC3(CCN3C(c3cc(Cl)cnc3Cl)=O)C2)[nH]c2ccccc12 10277,N1(C(N2CCC(CNC)C2)=O)CCCCC1CC(C)C 10278,C1(CC)CN(Cc2cccc(-c3ccccc3)n2)CCN1C(C1CC1F)=O 10279,Cc1ccc(C(=O)NCC(=O)NCC(C2CC2)NC(=O)C=CSc2nc[nH]n2)s1 10280,N1(C(C=Cc2cnc(C)s2)=O)CCCC12CCN(C(=O)C(C)CC(C)(F)F)C2 10281,CC(CC(=O)N(C)CC1CCCCN1C(C1CCCO1)=O)C(F)(F)F 10282,N1(C(c2ccn(CCCC)n2)=O)CC(NC(=O)CN2CCCCCC2)CC(F)C1 10283,c1(C(=O)NC2(CNC(C3=CCC(C)(C)CC3)=O)CC2)cc(Cl)cc2c1NCCC2 10284,N1(C(c2cc(CC)nc(O)c2)=O)CC2(CCN(C(=O)C(C)NC(=O)NC)C2)C1 10285,C1(CCN(C(CCSCC(=O)OC)=O)CC)C(C)CCCN1C(=O)C1=COCCC1 10286,c12cnn3c(cccc13)NC2=O.C1(C(=O)O)(C(=O)O)C2CCC12 10287,C1(C(N2CCC(CCOC)(NC(CC=CC)=O)C2)=O)CC2COCC2C1 10288,C1(C(=O)NCC(CCC)OCC)CCC2CCC1N2C(c1ccccn1)=O 10289,N1(C(Cc2c(C)oc(-c3ccsc3)n2)=O)CCc2nncn2CC1 10290,CC(C)C(C(=O)NC1(C)CN(C(C2CCC(=O)C2)=O)C1)c1cccc(Cl)c1 10291,c1(C(=O)NC(CN(C(CCc2ccc(C)nc2)=O)C)(C)C)nc(C)n(C)c1C 10292,c1(CC)cc(C(N2CC(NC(=O)CS(=O)CC)C(C)C2)=O)nn1CCO 10293,c1(C(N(OC)Cc2cnn(C)c2)=O)ccc(C(=O)O)cc1Cl 10294,C12(CNC(c3cncc(COC)c3)=O)CCC(CC1)CN2C(=O)CC1CCC1 10295,c1(CC)ccoc1C(=O)NCCN(C(c1ccc(SC)o1)=O)CC1CC1 10296,c1(CNCC2(C(=O)O)CCSC2)ncnc(O)c1F 10297,N1(C(C(C2CCCO2)SC)=O)CCC(N(C(=O)CCOC2CCC2)CCO)CC1 10298,N1(Cc2ccc(-c3nncc(C(C)=O)c3)s2)CCC(C)(O)C(C)(O)C1 10299,N1(C(c2nccc(C)c2O)=O)CCC2(CCC2)C(NC(C2CCCSC2)=O)C1 10300,C1(N(C(C2CC(=C)C2)=O)C)CCC(n2cc(CCc3nn[nH]n3)nn2)CC1 10301,S(=O)(=O)(c1ccc(NC(=O)NC2(C(=O)O)COC(C)(C)C2)cn1)NC(C)(C)C 10302,N1(C(CCCCCOC)=O)CC(NC(=O)COC2CCOC2)CC12CCC2 10303,N1(C(c2c(CC)c[nH]c2)=O)CC2=C(C1)CN(C(C13C4C5C1C1C3C4C51CO)=O)C2 10304,c1(OCC)cc(C(=O)NCC2CC(CNC(=O)CN3CCCCCC3)C2)ccn1 10305,C(=O)(C(C)(C)C(C)(C)O)NC(C(=O)N(CCCCCC)C)CC(F)F 10306,Cn1c(C(N2CCCCC2CCC(=O)NC2(C(C)(F)F)CC2)=O)cnc1Cl 10307,C(=O)(CCCC(=O)N1CCC(C(F)(F)F)C(OC)C1)NCCC 10308,C1(NC(c2c(CC)nc(C)nc2)=O)CN(C(=O)Cc2ccnn2C)CC12CCC2 10309,N1(C(CN(C)C2CC2)=O)CCN(C)c2ccc(NC(=O)OC(C)(C)C)cc21 10310,Cc1c(C(=O)NCC2CCN2C(c2cc(N(C)C)ccn2)=O)cnn1C(C)(C)C 10311,C(=O)(N=S(=O)(c1ccc(F)cc1F)C(F)F)C1(C)CCN(C)C1 10312,C1(CC=C)(NC(c2csc(CC)n2)=O)CN(C(=O)C(F)CC2CCCC2)C1 10313,N1(c2nc(OC)nc(C)c2)CCOC2(CCCN(C(C3CCCCC3C)=O)C2)C1 10314,Cc1ccc(C(=O)NCC(N2CCN(C(=O)C3=NOCC3)CC2)C(F)F)c(F)c1 10315,C1(COC)(NC(=O)CN2CCS(=O)CC2)CCN(C(C2(Cl)CC2(F)F)=O)C1 10316,C12(C(=O)NC(C3(C)C(C)CCC3)c3ccccc3)CC(CO1)N(c1cnccn1)C2 10317,c1(C(N2CC(OC)C(NC(C3C(Cl)(Cl)C34CC4)=O)C2)=O)cccc(F)c1F 10318,c1(C(C(=O)NC(C)CN(C(=O)Cn2cc(C(F)(F)F)cn2)C)C)cccc(Cl)c1 10319,C(=O)(CCCCCc1ccccc1)NC1C(CNC(c2c(CC)cc[nH]2)=O)C1 10320,N1(C(C2CC(N(C)C(C34CC(CO)(C3)C4)=O)C2)=O)CCC([N+](=O)[O-])CC1 10321,C(=O)(CCCCCC#N)N1CC(C(=O)NCC(C)C2CCC2)N(C)CC1 10322,C1(CNC(CS(CC)=O)=O)COCCN(C(C2CC(N3CCCC3)C2)=O)C1 10323,C(CS(=O)C(F)(F)F)Cc1cn(C(c2nnn(C(C)(C)C)n2)OC)nn1 10324,C1(NC(C(C2CCC2)OC)=O)COC2C(NC(c3cc([N+](=O)[O-])n[nH]3)=O)COC12 10325,C(=O)(CCC(C)(C)C)N1CC(C)C(CNC(c2cn(CCCF)nn2)=O)C1 10326,c1(C(N(C(C)CNC(C2COC3COCC23)=O)C)=O)cnc2cc[nH]c2c1 10327,N1(NC(CCCC(C)(C)CCc2c(C)oc(C3CC3)c2)=O)CC2CCC2(CO)C1 10328,N(C1CCCn2ccnc21)C(C(CCNC(c1c(C)cn(C)n1)=O)O)=O 10329,c1(C(=O)NC(CC=C)CNC(=O)C=Cc2scnc2C)cccc(S(C)=O)c1 10330,N1(C(C(CSC)C)=O)CCC(O)(CNC(c2c(C)coc2C)=O)C1 10331,Cc1nsc(C)c1C(=O)NCC1CC(C)N(C(=O)COCCCC(C)C)C1 10332,Cn1nnc(C(=O)NCCOCCNC(=O)CCCc2ccccc2)n1 10333,C12(NC(c3c(CCCC)ocn3)=O)CCN(C(c3cc(CF)on3)=O)CCC1C2 10334,N1(C(CSCCC(C)C)=O)CCCC2(NC(c3cncc4ccsc34)=O)CC2C1 10335,c1(N2CC(C)(NC(CCCNc3ccc(OC)cc3)=O)C2)ccc2nnnn2n1 10336,CC12CCC(C(N3CCOC(CNC(=O)CSC4CC4)C3)=O)(CO1)C2 10337,C1(CNC(CCC=CC(C)C)=O)CC2(CO1)CN(C(C1(C3CC3)CC(=O)C1)=O)C2 10338,c1(C(N2CCC(C)(NC(C3C4COCC34)=O)C2)=O)cccc2c1OCCN2 10339,c1(C(N2CCCCC(NC(c3scc(OC)c3)=O)C2)=O)cnc2c(n1)CCCC2 10340,c1(C(N(C)CC2N(C(C(C(CC)C)O)=O)CC(F)C2)=O)cc(C)cc(C)c1C 10341,N1(C(C2N(C(C3C(C)C4CCC3C4)=O)CC(F)(F)C2)=O)CC(=O)N2CCCC2C1 10342,c1(N(C(CNC(CCN(CCC)C)=O)C)C)ccc(C(=O)OC)c(C)n1 10343,C1(CNC(CN(C)C2CC2)=O)CCCC(NC(C2(O)CCOCC2)=O)C1 10344,C(=O)(C(C)C(C)S(C)(=O)=O)N1CC2C(CNC(CCCCC(C)C)=O)C2C1 10345,N(C1CCc2cccnc21)C(C1(C)CCN(C(C2N(C)CCCCC2)=O)CC1)=O 10346,C(=O)(NN=Cc1cccnc1)c1c(CN=[N+]=[N-])cc2ccccc2c1 10347,N1(C(c2c(C)ncnc2)=O)CCC2(CC1)COC(CNC(=O)C(C)C(C)C)C2 10348,C(=O)(N1CCC(C(=O)NC2(C)CC(O)(CO)C2)O1)c1ccc(CC)s1 10349,c1(CNC(C2CC(N(C(COCCC=C)=O)C)C2)=O)cc(CC)no1 10350,N1(C(CCC=C=C)=O)CC2(C(=O)NC3CN4CCC3C4)CCC1CC2 10351,c1(OC)cc(OC)cc(C(=O)NC2CCCC2CNC(C2CC(OC)C2)=O)c1 10352,C1(NC(c2c(OC)noc2C2CC2)=O)CCC(C)N(C(=O)C(O)CC(N)=O)C1 10353,CC#CCC(C(=O)NCCC(=O)NC(C)(C)C)NC(c1cc(CC)n(C)n1)=O 10354,Nc1cc(C(=O)NCC2(NC(=O)CCn3ccnn3)CC3CCC2C3)cc(F)c1 10355,c1(OCCC)cccc(C(c2nnnn2C)NCC(C2CCC2)C2CC2)c1 10356,CC1(C2CCCN(C(=O)CC3CCCC(N(C(=O)Cc4ccsn4)CO)C3)C2)CC1 10357,c1(CC)cc(N)ccc1C(=O)NCCC(O)CNC(=O)CCC1CCCOC1 10358,N1(C(c2c(C)nn(C3CCC3)c2)=O)CCC2(CCC2)C(NC(C2CC(O)C2)=O)C1 10359,n1(CC(=O)NCCC(C)NC(=O)CCOC2CCOC2)cnccc1=O 10360,c1(OC)ccnc(O)c1C(=O)NC1CCCCN(C(C2C3CC(=O)CC23)=O)C1 10361,N1(Cc2onc(CCC)n2)CC(C)(C)OC2(CCCOC2)C1 10362,N1(C(COCC(C)C)=O)CCC(N(C)C(C2CC3(CC(=O)C3)C2)=O)C(C)C1 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10381,c1(CC(N2CC3CC(NC(C4(F)CCCC4)=O)C(C3)C2)=O)ccc2nsnc2c1 10382,CCC(C)(C)CCCC(=O)N1CCC(N(C)C(C2CC3CCC3C2)=O)C1 10383,CN1CCC(c2nnc(COC(c3ocnc3C(F)(F)F)=O)o2)CC1 10384,c1(OC)cnc(C(=O)N(C)CCN(C)C(c2n[nH]cc2CC(C)C)=O)c(OC)n1 10385,C(C#Cc1ccccc1)N1CCN(C(=O)CC2(O)CCOC2)CC1 10386,C1(CC)CN(C(C2CC(O)CN2C)=O)CCC1NC(C1CCCN1C1CC1)=O 10387,c1(C(=O)NCC2C(NC(c3ccn(CCC)n3)=O)C2)cccc2c1OCC2C 10388,CC(C)CC(=O)C(=O)N(CCCCC(=O)NC(C)CCCCO)C 10389,N1(C(CCNC(C)=O)=O)CCC2(CC1)OCCCC2NC(=O)CSc1ccoc1 10390,C1(CNC(c2cc(C)on2)=O)C2CN(C(=O)C(C)(C)N3CCOCC3)CC12 10391,C1(OC)CCC1C(=O)NCCOCCNC(=O)CC1(C)CCC1 10392,C(CCF)(C(=O)N(CCNS(N)(=O)=O)CCO)NC(CCC1(C)CC1)=O 10393,C#CCCCCCCC(=O)N(C(C(=O)NCC1CCC(=O)N1)C1CC1)C 10394,C(=O)(CC(O)CC(C)C)NCC(C)NC(c1onc(CC)c1C)=O 10395,N1(C(CC2(COC)CC2)=O)CC(NC(c2ccc(-c3cscn3)cc2)=O)C(O)C1 10396,N1(C(c2cn(CC(CC)O)nn2)C(=O)NCCC#N)CCOC(C2(C)N=N2)C1 10397,C1(CC(=O)NC2CC(C(C)NC(CCOCCOCC)=O)C2)CCNC(=O)C1 10398,C(c1ccc(CN(C)Cc2cc(Br)ccc2Cl)cc1)=CC(=O)OC 10399,CC(C(=O)N1CCCCC1CCCNC(C1(C)C=CCCC1)=O)C(C)O 10400,CCCCS(=O)(=O)CC(=O)NCC1(C2CC2)CCN(C(C2CCS(=O)(=O)C2)=O)C1 10401,c1(CN2CCC(C#N)(C(C)(C)O)C2)cc(Br)cc(F)c1O 10402,S(=O)(=O)(c1c[nH]c(C(N2CC(NC(=O)C(C)N(C)C)C(C3CC3)C2)=O)c1)NC 10403,CC1CCCCN1CCC(=O)NCC1CCN(C(=O)C(c2ccccc2)=O)C1 10404,N1(Cc2c(OC)cco2)CCC2(CC1)CC2NC(c1ccc(C2CC2)s1)=O 10405,C1(C(=O)NC2CC(OC3CCC3)C2)CC2CN(C(C3CCC3)=O)CC2C1 10406,C1(C(N2CCN(C3CN(C(c4ccc(=N)[nH]c4)=O)C3)CC2)=O)CC(C2CC2)=NO1 10407,C1(O)(CCNC(C(C)c2ccon2)=O)CCN(C(c2cc(O)cs2)=O)CC1 10408,c1(C(=O)NCC(C)(CC)NC(CC(CC)C(F)F)=O)c(F)ccc2occc12 10409,c1(C(c2n(CCOCC)nnn2)NCC2CCCOC2)ccc2c(c1)COCC2 10410,C(=O)(C1CCCc2sc(=N)[nH]c21)N1C(CNC(CNC(CC)=O)=O)CC(F)C1 10411,C(=O)(C(CCS(C)(=O)=O)OC)NC1CCN(C(CSCC#C)=O)CC(O)C1 10412,C1(C(Cc2nnnn2C)NC(c2ncnn2C)CC)CCC(F)(F)CC1 10413,C1CN=C2C=C(N=C(COC)N2)N1.CCS(=O)(=O)NCCCSCC1CCCC1 10414,C12(NC(CNC(N)=O)=O)CC1CN(C(=O)CC(F)(F)Cl)C2 10415,c1(C2N(CC)CC2)ccc(Cl)cc1.C12CNCC1n1cc(nn1)-c1csc2n1 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10433,c12cnn3ccc(nc13)[nH]2.c1(C(=O)OCC)c[nH]nc1C(=O)N(C1CNC1)C 10434,c1(C(=O)NC2CC3CC2N(C(=O)CN2CCCCCC2)C3)cnc2scnc2c1 10435,N1(C(CN)=O)CC2CN(C(C3C(Sc4ccccc4)C4C=CC3C4)=O)CC(C1)O2 10436,Cc1cnc(C(=O)NCc2cccc(NC(=O)C(CC#N)c3ccccc3)c2)nc1 10437,C#Cc1ccc(CN=C(NCC2CCCO2)NCC2CCCS2)cc1 10438,c1(CN2C(C(=O)Nc3ccsc3)CNCC2)ccc([N+](=O)[O-])c(F)c1 10439,N1(C(c2nnn(CC)c2C)=O)CCCCC(N(C)C(C2CCCSC2)=O)C1 10440,N1(C(C(CCC)CCC)=O)CC2(C1)CN(C(C1CCC(=O)N1C(C)=O)=O)CCO2 10441,C(CCCCCS(N)(=O)=O)NC(=O)OC(C)(C)C.c12cccc(c1)CN(C=O)C2 10442,C(CN=c1nc(OC)cc[nH]1)C1CCC(NC(Cc2cc(OC)nc(C)c2)=O)C1 10443,Cc1nc(C(N2CC3CC2C3C(=O)NC(c2cnccn2)C)=O)cn1C 10444,N1(C(C)C(=O)NCc2ccncc2)CCN2C(C)COCC2C1 10445,c1(C(N(CC(CC)NC(C2C3CCCC23)=O)CC)=O)csc(-c2ccccc2)n1 10446,C(=O)(CCC(C)(C)[N+](=O)[O-])NC1C(C)CCN(C(c2c(C)cccc2)=O)CC1 10447,C(=O)(C(O)CC(C)C)N1C(COC)(CNC(C2(C)CC2(F)F)=O)CCC1 10448,C1(CNC(C(=O)NC(C(CC)C2CCC2)=O)C)CCN(C(C)CN(CC)CC)CC1 10449,Cc1cc(NC(=O)NCCF)cc(SCCO)c1 10450,C(=O)(C(CC(C)C)C(N)=O)NC(CC)CNC(c1sc(F)cc1Cl)=O 10451,C=CCC(CNC(c1cn2c(n1)CCC2)=O)C(=O)NC(CN(C)C)CO 10452,C(=O)(C(C)C1=CCCC1)NC(CN(C(=O)CCC(=O)c1ccccc1)CC)C 10453,C1(CC)CCN(C(=O)C(C#N)C(C)C)C(C(N2CC(F)(F)C2C2CC2)=O)C1 10454,C1(CNC(C(C)=CC)=O)CCN(C(C2CCn3cc(C)nc3C2)=O)CCC1(F)F 10455,Cc1cccc(OCC(=O)NCC(C)N(C(=O)C(F)C2CCOC2)C)c1 10456,c1(CNC(C2(C)CC=CCO2)c2n(CC=C)nnn2)cc(OC)c(OC)c(Cl)c1 10457,Cc1ncc(CCNC(=O)C(C2CCN(C(c3csc(C)n3)=O)C2)C)s1 10458,c1(C(=O)NCC2(O)CN(C(=O)CCc3ccc(F)nc3)C2)cncc(Cl)n1 10459,N1(C(C(C)(C)Cl)=O)C2CC1CN(C(C1(c3ccccc3F)CC1)=O)C2 10460,c1(OC)ccc2c(c1)C(C(=O)NC1(C)CN(C(=O)CCOC3CCCC3)C1)CC2 10461,N1(CCC(C2(CC(C)C)COC2)=O)CCC(N=c2nc(C3CCCC3)[nH]s2)CC1 10462,C1(CNC(c2c(OC)n[nH]c2)=O)CN(C(C2(F)CC=CCC2)=O)CCN1C 10463,C(c1ccncn1)=CC(=O)NC1C(NC(CNS(NC)(=O)=O)=O)CC1 10464,c1(COCC)cn(CC2(CC(N3CC(CC(=O)OC)C3)=O)CC2)nn1 10465,C(=O)(C1(C)CCn2ccnc21)NCC(C)CN(C)C(c1csnc1Cl)=O 10466,C1(C(=O)Nc2cncc(C(N)=O)c2)CCOCCN1C(=O)Cc1ccoc1 10467,C(=O)(CCCS(C)(=O)=O)N1CC2C(CNC(c3snc(C)c3N)=O)C2C1 10468,C=CC1(O)CCN(C(=O)Cc2ccc(F)cc2I)C1 10469,c1(CCNC2C(N3CCN(C)CC3)CCC2)c2c(nn1C)CCC2 10470,c1(C(=O)NCCCC(=O)N2CCC(c3nc[nH]n3)C2)ccc([N+](=O)[O-])o1 10471,Cc1cc(C(=O)NC2CC(NC(=O)CC3CSC3)C23CCC3)cc(Cl)c1 10472,C1(C(=O)NCCC2N(C(CNS(CCOCC)(=O)=O)=O)CCC2)CCC(C)(C)C1 10473,C1(C(N2CC(C)C(NC(CSCCOC)=O)C(C)C2)=O)CCc2nnnn2CC1 10474,Cc1cc(=NCC(C)CNC(=O)C=C2CCSCC2)[nH]c(CO)n1 10475,C(=O)(C(C)S(=O)(=O)CCC)NC(CCCC)CNC(c1n[nH]c(CC)c1Cl)=O 10476,N1(C(C(COC)O)=O)CC=CC(NC(C2(C(F)(F)F)CCCCC2)=O)C1 10477,C1(NC(c2cn(CCNC(CC3CC(C)OC3)=O)nn2)=O)(CO)CC2(CCC2)C1 10478,Cc1cccc(C(=O)NCC2(CNC(C3(C(F)F)CCCO3)=O)CC23CCC3)n1 10479,C#Cc1cnc(C(N2CCOCCC2C(=O)NCC(C2CCC2)OC)=O)c(C)c1 10480,C1(CC(=O)NC2CN(C(=O)CCc3nncs3)C2)COC(=O)C1 10481,C(c1ccc(C(F)F)o1)=CC(=O)NCC(N(C(C=C(C)Cl)=O)C)C1CC1 10482,C(=O)(C1=CC2(CN(C(=O)C(C)(O)C3CC3)C2)OC1)NCC(N(C)C)C1CC1 10483,c1(NC(N(c2c(C)ccc(C)c2)CCC#N)=O)nc2cccnc2s1 10484,c1(OC)cnccc1C(=O)NC1CCC1CNC(=O)C(O)c1ccsc1 10485,C(=O)(CC(O)CNC(=O)C=CC1CC1)N(CC(O)CO)C(C)C 10486,c1(CC)cccc(F)c1C(N1CCN(C(c2ccc(OC)c(N)c2)=O)CC1C)=O 10487,c1(C(N(CCN(C)C(c2csc(C3CC3)n2)=O)C)=O)c(N)ccc(F)c1F 10488,c1(C(N(C(C)CNC(=O)CC2(C)CC2)C)=O)cc(F)c(F)c(O)c1F 10489,C(CCC(C)(C)C(=O)NC(C)C(=O)NO)NC(Cc1ccn(CC)n1)=O 10490,Cc1ccc(C#N)c(NC(N2CC(N3CCOCC3)C(O)C2)=O)c1 10491,N1(C(C(CC)OC)=O)CCN(C(c2sc(OC)nc2Cl)=O)C(CF)C1 10492,Cc1cc(C(=O)N(CC)CC2CCCN2C(c2sc(C)c(C)c2C)=O)ncc1F 10493,C1(NC(CC(C)(C)NC(CCN(C)CC)=O)=O)CCCCC1(C)O 10494,N1(C(C2CCC(C)(C)O2)=O)CCCC2CN(C(c3csc(Cl)c3)=O)CCC12 10495,c1(C(N(CCN(CCOC2CCC(CC)CC2)C)C)=O)cc(C)nc(C)n1 10496,N1(C(c2cccc(NC(C)=O)c2)=O)CC2CC(NC(C3CCS(=O)(=O)N3)=O)C1C2 10497,CCCCC(C(=O)N1CCC(n2cc(Cc3cn(C)c(C)n3)nn2)CC1)N(C)C 10498,C1(C(N2CC3C(NC(c4ccc(=O)oc4)=O)C3C2)=O)COc2ccc(O)cc2O1 10499,Cn1cnc2[nH]c(=NCC3CCCN(C(=O)CSCC(F)(F)F)C3)nc(O)c12 10500,C(=O)(CCC(O)C(C)(C)C)N1CCC(C(C)(C)NC(CNC(COC)=O)=O)CC1 10501,N1(C(CN(CCC#C)C)=O)CC2CCC(NC(c3sc4ccsc4c3C)=O)(C2)C1 10502,c1(OC)ccc(COCC(O)CNC(C2(c3ccccc3)CC(C)C2)=O)cc1 10503,c1(C(=O)NCC(CO)NC(c2ccc(C(C)(C)C)nc2)=O)ccc(Cl)c(F)c1 10504,Cn1cc(SCC(N2CCCC2CCC(=O)NCc2cc[nH]n2)=O)cn1 10505,CCCC(CN=c1cccc(S(=O)(=O)NC2CCc3nc(C)cn3C2)[nH]1)OC 10506,C1(CC(=O)N(CCOCCNC(c2c(C)csc2)=O)C)CCCC(=O)N1 10507,CCC(CC(F)(F)F)N=c1[nH]c(=NC(C)CC(C)(C)OC)[nH]c2ccsc12 10508,C1(C(=O)NCCCOCCNC(C(C)C2=CCCC2)=O)CCC2(CC1)CC2(F)F 10509,C1(C(=O)Nc2ccc(-c3c(C)ncs3)cc2)CCCC12CCOCC2 10510,CC(C)CN=C(NCC1(COC)CCC1)NCC(c1cn(C)nc1C(F)F)(C)C 10511,CC(CO)C(=O)NCCOCCCN(C)C(c1cnn(C)c1)=O 10512,C=Cc1ccc(C(=O)NCC(C)(O)CNC(=O)COCCc2ccccc2)cc1 10513,C(CC(C)(C)N=c1[nH]nc(C(C)(C)C)o1)NC(C(C)CSC(F)(F)F)=O 10514,n1(CC(=O)NCC2N(C(COC)=O)CC(C)(C)C2)c(=O)nc(O)c2ccccc12 10515,c1(OC)c(F)cc(F)c(C(N2CCN(CC3(CNC)COC3)CC2)=O)c1F 10516,c1(C(N2CCC(OCc3ccccc3)C2)C(=O)NCC)cc(Cl)nn1C 10517,c1(C(C)NC(c2cn[nH]c2)=O)nocc1C(=O)NCC1(F)CC1 10518,c1(C(=O)NC)ccc(CNC(c2ccc(C(C)(C)C)cc2)C)cc1 10519,c1(C(N2CC(NC(C3C(CC(C)C)C3)=O)C(O)C2)=O)ccc(=O)n2c1CCC2 10520,N1(C(C=C(C)C(C)(C)C)=O)CCC(C2(NC(C3CC4CC4C3)=O)CCC2)CC1 10521,C1(C(=O)NC2(CCCC)CC2)CN(C(=O)C(C)OCCOC)CC1(C)C 10522,Cc1ccccc1C(=O)NC(CCN(C)C)C(=O)N1CC(C)C(F)C1 10523,c1(CNC(NCC2CC(CC)C2)=NCCF)nnc2c(=O)[nH]ccn12 10524,c1(C(N2CCCCC2COC)C(=O)NC(CC)C)ccc(C)c(OC)n1 10525,CC1CN(C(C2CC23CC(C)(C)C3)=O)CCC1NC(C1CC2(CCCO2)C1)=O 10526,CC1CC=C(C(=O)NCC(C)(CO)NC(=O)CN2CSCC2=O)CC1 10527,c1(OC)nc(N(CCN)Cc2c(F)cccc2F)ncc1F 10528,N1(C(Cc2nc(C)sc2C)=O)CC2CCCC2(NC(C2CCOC2(C)C)=O)C1 10529,N1(C(c2n(OC)cnc2C)=O)CC(C)CN(C(c2nn(C)c(C)c2Cl)=O)C(C)C1 10530,c1(OC)ncc(NC(C2(F)CCN(C(c3cc(O)ncc3Br)=O)CC2)=O)cc1F 10531,C1(CC(=O)NC(c2cnc(C)s2)C)(NC(c2cocn2)=O)CCCCC1 10532,CC(=NO)C1CC(C(=O)NCC(C2CCN(C(=O)CNC=O)CC2)(C)C)C1(C)C 10533,c1(CC(N2CCN(C(c3n(C=C)nnc3)=O)CC2)=O)ccc(Br)c(O)c1 10534,N1(C(c2c(C)cc[nH]2)=O)CCC2(CC1)CC2CNC(c1cnc(S)[nH]1)=O 10535,c1(C(=O)NC2CC(C)CN(C(=O)C=Cc3cccs3)C2)cncc(P(C)(C)=O)c1 10536,N1(C(=O)CC2CCCCN2C(=O)CC2(O)CCOC2)CCOC2(CCC2)C1 10537,N1(C(C2CCCC(OC)C2)=O)CCCC(NC(c2cc(Cl)cnn2)=O)C1C 10538,C(C)(CN=c1[nH]cncc1C)NC(C(c1ccc(C)cc1)C)=O 10539,c1(C(=O)NCCC(C)NC(c2c(C3CC3)cccc2F)=O)cn2cccnc2n1 10540,C(=O)(C(O)CCS(C)=O)N(C(C)C)CCN(C)C(c1ncc(F)cc1N)=O 10541,C(C(=O)NCCN(C(C1CCC12CCC2)=O)C(C)C)(C(F)(F)F)OC(C)=O 10542,C#CCC(O)C(=O)N1CC(C(=O)NCCCCC2CC2)C(F)C1 10543,N1(S(CCCC)(=O)=O)CCC(C(=O)NCCc2nccs2)(CO)CC1 10544,c1(C(C)NC(=O)C(C2CN(C(=O)CCC3(C)N=N3)C2)N(C)C)ncc(F)cn1 10545,C1(C(=O)NC2CCCC(CNC(=O)C3=CCCSC3)C2)CCc2ccccc2O1 10546,C1(C(=O)OC)CC(C(=O)NC(C)CCNC(C23COCC(C2)C3)=O)C1(C)C 10547,C1(C(CC(C(=O)N(CC)CC2CC(=C3CC3)C2)C)=O)(C(=O)OCC)CCCCO1 10548,C(C)(c1cccnc1)=CC(=O)NCCCC(C)(C)NC(CCC(=O)NC)=O 10549,c1(C(N2C(C(C)NC(c3c(C)nc(C)o3)=O)CCC2)=O)ccc(C)c(Cl)c1 10550,N1(C(C)=O)CCN(C(=O)NC2(c3cc(F)ccc3F)CCC2)C2CC12 10551,N1(C(c2ccc(CC)o2)=O)CCC(O)(CC(=O)NCC(c2ccncc2)C)CC1 10552,C1(OC)COCCC1CC(=O)N(CCCNC(=O)CNC(=O)NC1CC1)CCO 10553,Cn1cc2cccc(-c3nc(C(=O)NCc4cccc(Br)c4O)cs3)c2n1 10554,CN1CCC(C(C)(O)CN(C=O)Cc2cnn(-c3cccnc3)c2)CC1 10555,CC(C)CC(CNC(c1ccc(Cl)o1)=O)NC(=O)C(C)OCC1CC1 10556,CCC(C)(C)C(O)C(=O)N1CC(C(=O)NCc2nocc2C)C(C2CC2)C1 10557,C1(C)(CNC(C(=O)NCCOC)=O)CC(OC)CN1C(c1sccc1OC)=O 10558,c1(OC)ccc(F)cc1C(=O)Nc1ncc(C(N)=O)s1 10559,N1(C(CC(COC)NC(C2(C#N)CCCC2)=O)=O)CC(O)CC(O)C1 10560,N1(C(Cc2ccc(OC)cc2Cl)=O)CC(=O)N2CCCC2C1 10561,N1(C(=O)NCCN(CC=C)C)CCCC(C)(OC(C)=O)CC1 10562,C1(NC(C2C=CCN(C(c3n(C)c(=O)ccc3)=O)C2)=O)CC2(CCCCC2)C1 10563,c1(CN2CCN(C(CC(C)C)=O)C3C2C3)cc(Cl)c(Cl)cc1Cl 10564,CCC(CC)C(C)C(=O)N1CC(C)(CNC(c2c(C)cccc2C)=O)CC1(C)C 10565,N1(C(c2ccc(CO)[nH]2)=O)CC2(CCCN2C(=O)COc2cccnc2)C1 10566,c1(-n2cc(C3OCCN(SCCCC(=O)NCCO)C3)nn2)c(Cl)cc(F)cc1Cl 10567,N1(C(C=Cc2ccc(OC)cc2)=O)C2CCC1CN(C(c1cnncc1C)=O)C2 10568,N1(C(c2c[nH]c(=N)s2)=O)CCCC2C(NC(c3ccc(C4CCC4)cc3)=O)C12 10569,C=CCCCC(C(=O)N1CC(F)C(F)C1)NC(C1CC2CCC2C1)=O 10570,N1(C(c2ccc(Cl)o2)=O)CCCC2(CCC(NC(C3(C4CC4)CCC3)=O)C2)C1 10571,N1(CCCCNC(C(C(C)C)OC)=O)CCCN(C(c2csc(C)c2)=O)CC1 10572,Nc1cc(C(=O)NC2CC(CNC(C3CC(O)C3)=O)C23CCC3)cc(F)c1O 10573,C1(CC)CN(C(=O)C(C2CCOCC2)C)CCN1C(c1occc1Cl)=O 10574,N1(C(C2CCC(C)(CC)O2)=O)CC2CCC(CNC(c3ccc(C)s3)=O)C2C1 10575,c1(CNC(C2N(C(C=COCC)=O)CC(C)C2)=O)cc(F)cnc1Cl 10576,Cc1cc(S(C)(=O)=O)cc(C(=O)NC(C)C(C)(C)NC(=O)CC(O)C(C)C)c1C 10577,C1(C(=O)NC2(C)CC(=C)C2)CCCN(C(=O)C(C)=C2CC2)C1 10578,C(=O)(CC(C)C(F)F)N(CCN(C(CC1N(CC)CCC1)=O)C)C(C)C 10579,C1(NC(C=CCCC)=O)CCCC(NC(c2cncc(Cl)c2C)=O)CC1 10580,N1(C(CC)=O)CCOCC(NC(C2C(C)CCN2C(=O)OC(C)(C)C)=O)C1 10581,CN1CCN(C(c2ccc(-c3cnn(C)c3)o2)=O)C(CNC(=O)C2=COCC2)C1 10582,C1(NC(c2cnc(C)nc2)=O)CC12CCN(C(=O)CC(C)CF)CC2 10583,c1(C(N2CCC(NC(CC(C)n3cccn3)=O)C2C)=O)[nH]cc2c1CCCC2 10584,CCCCCC(C)CC(=O)NC(C1(C(=O)NC2CN(C)C(C)(C)C2)CC1)C 10585,CC1CCCC(CC(N2CC(OCCNC(C3(O)CCOC3)=O)C2)=O)C1 10586,c1(C(=O)NC2CN(C(C3C(NC(C)=O)CCCC3)=O)C2)c(Br)nc2n1CCC2 10587,N1(C(C(c2scc(C)n2)C)=O)CC2(CCN(C(c3cccc4sccc34)=O)C2)C1 10588,c1(C(N(C)CC2CCN(C(CNC(=O)OC)=O)CC2)=O)ncc(N)nc1C 10589,C1(C(N(CCCNC(CCCCC=C)=O)C)=O)Cc2ccc(F)cc2C1 10590,C#CC1(C(=O)N(C)CC2CC2(F)F)CCN(C(=O)CS(=O)(=O)CC)CC1 10591,c1(C(=O)NC2(CCNC(c3coc(C(F)(F)F)n3)=O)CC2)ccc2ncnn2c1 10592,CC1C(C)N(C(c2cccnc2CNC(=O)Cn2cc(CO)nn2)=O)CCN1C 10593,N#Cc1ccccc1OCC(N1CCC(CCNC(c2csnc2Cl)=O)CC1)=O 10594,N1(C(c2n(C)ccn2)=O)CC(NC(c2cc(F)ccc2Cl)=O)C(F)(F)C1 10595,CC(C)CC(CNC(C12CC(F)(C1)C2)=O)C(=O)NC(C)CS(C)(=O)=O 10596,Cc1cc(NCCOCC(=O)NC2CN(C(C3CCC(C)C3)=O)C2)on1 10597,CC1CN(C(=O)CC2(O)CCOCC2)CC(C)N(C(=O)CSc2nncs2)C1 10598,N1(C(Cc2cc(C)on2)=O)CC(NC(c2csc(C3CCCO3)n2)=O)CC1CO 10599,N1(C(C(CC)O)=O)CCCC12CCN(C(=O)C(O)COCc1ccccc1)C2 10600,n1(CC)nc(C)c(C(N2CC(N3CCN(C(c4cnn(C)n4)=O)CC3)C2)=O)c1Cl 10601,c1(OC)cc(CCOC(=O)C=CC(c2ccc(F)cc2)=O)cc(OC)c1O 10602,C1(C(=O)NC(C2CN(C(=O)C=C3CCOCC3)C2)C)CC12CCCCC2 10603,Cc1ccc(S(=O)(=O)N(C2Cc3ccc(Cl)cc3C2)CCO)cc1 10604,c1(C(N2C(CCCNC(C(C)SC(C)C)=O)CCC2)=O)cc2n(c1)CCSC2 10605,Cc1cc(C)c(C(=O)NC2CC2CNC(c2nc(-c3ccccc3)sc2C)=O)o1 10606,c1(C(=O)NCCC(CNC(=O)CC2CC3CCC2O3)OC)nnccc1C 10607,c1(C(=O)NCCC(CNC(c2nsnc2O)=O)OC)cc2ccncc2[nH]1 10608,C1(C(=O)NCC2(O)CCN(C(=O)CN3CCC(CO)CC3)C2)CC12CC(F)(F)C2 10609,N1(C(CC(C)SC)=O)CC(NC(c2cccc(C3(F)CC3)c2)=O)C(C)C1 10610,CC(C)(C)C#CC(=O)N1CCN(C(=O)C(=C2CCCCC2)F)C(C(F)F)C1 10611,C1(C(N2C(CN(C(=O)CC3CC4C=CC3O4)C)CCC2)=O)NC(=O)C2CC12 10612,Cc1nc(C2CC2)[nH]c1C(N1CCC(NC(C2SCCCS2)=O)CC1)=O 10613,C1(CC(=O)NC2CC(NC(C3N(CCC)CCCC3)=O)C2)CCC(=O)NC1=O 10614,CCCCC(CN=c1[nH]c(Cl)nc2c1CCC2)NC(C1(O)CCCCCC1)=O 10615,CC1(C)CCC(C(=O)NCC2(C)CC2(F)F)CN1C(C1CCC(=O)O1)=O 10616,C1(NC(=O)COc2cccc(F)c2)CN(C(C2(C(F)F)CCC2)=O)CCC1F 10617,Cc1ccc(CNC(=O)C=CCC2(NC(=O)C(C)CC#N)CCC2)cn1 10618,c1(CNC(=O)C(c2cccnc2)N2CCCCC2)c[nH]nc1C1CCOCC1 10619,N1(C(C2N(C(Cc3n(CC)ncc3)=O)CCC2)=O)CC(OC)C(OC)C1 10620,C1(C(=O)NCCC(C)NC(CCC(=C)C)=O)CCC(=O)N(Cc2ccccc2)C1 10621,C(=O)(CCCCC(N)=O)N1C(CC(N2CCCC(C)C2)=O)C(C)(C)CC1 10622,c1(C(C(=O)NC(CC(C)NC(C(Br)=C(C)C)=O)C)O)cccc(C)c1 10623,C1(C2CCN(C(C3CCC4(CC4)C3)=O)C2)(NC(c2cn(C)c(=O)cc2)=O)CC1 10624,c1(C(=O)NCCN(C2CCCCC2)C(C2CC(C)C2(C)C)=O)cc2c(s1)CCC2=O 10625,c1(C(=O)NC2(CC(=O)NCCC34CC(CO3)C4)CCCC2)ccc(Cl)cc1O 10626,C1(C2CN(C(C34CCCC3C4)=O)C2)(NC(CCCn2c(C)ncc2)=O)CC1 10627,C(=O)(C(CC)CC(C)C)NCc1cc(C(=O)NC(CCC(=C)C)C)on1 10628,c1(C(=O)NCC2N(C)C(=O)OC2)nn2ccccc2c1CNc1nccs1 10629,C(=O)(CCN(CCO)C(c1cocn1)=O)NCCN(C)C 10630,C1(NC(c2c(CCC)cccc2)=O)COC2C(NC(=O)CC3CN(C)C3)COC12 10631,CCCCC(C)C(=O)N1CC(C(C)NC(=O)C(c2cnn(C)c2)O)C1 10632,Cc1ncnc(C(=O)NC(C)(C)CC=CC(N2CCOC(C(C)C)C2)=O)c1C 10633,c1(C(N2CCN(CCNC(C(CC)(C)CC)=O)CC2)=O)cnn2c1CN(C)CC2 10634,C1(C(=O)NCCOCC)CC=CCN1C(C1CCC1(OC)OC)=O 10635,c1(C(=O)NCC2(CCNC(=O)CCc3cn[nH]c3)CC2)ccc(C(=O)O)cc1 10636,Cc1nc(C)c(CCC(=O)NC2CN(c3ccnc(CO)n3)CC2(C)C)c(O)n1 10637,C(=O)(CCC1=NNC(=O)CC1)N1CC(NC(C(CCCCC)O)=O)CC1(CC)CC 10638,N(C(=NCCN(S(C)(=O)=O)C)NCc1ccsc1C)Cc1cccc(C)c1 10639,c1(C(C(=O)NCC(=C)CCNC(c2ocnc2C)=O)(C)C)ccc(Cl)c(Cl)c1 10640,Cc1ccc(O)c(CNC(=O)CC2CCCN(C(=O)CC#N)C2)c1 10641,c1(C(=O)NCC(CC=C)NC(c2c(C(F)F)cnn2C)=O)cc(C#N)ccc1Cl 10642,C1(C(=O)NC2CC(NC(c3cnc(SC)n3C)=O)CC2O)CCCCN1N=O 10643,c1(-c2nc(CNC(=O)NCCCc3ccnc(C)n3)sc2)c(Cl)cccc1Cl 10644,CC1CN(C(C2CCCN(CCC3(O)CCCCC3)C2)=O)CC(C)O1 10645,C1(C(=O)Nc2cnc(OC)nc2)CC2(CCN1C(=O)Cc1ccccc1C)CC2 10646,c1(C(=O)NCCCC(C)NC(Cc2cn(C(C)C)nc2)=O)cc2sccc2s1 10647,N1(C(c2cc(CCC)n(C)n2)=O)C2CCC1CN(C(=O)C(O)CCC(C)C)CC2 10648,n1(CC(C(=O)NCCN(CC)Cc2ccc(C)cc2)C)cnc2ccccc12 10649,c1(C(N2CC(NC(c3ccc(C)cc3F)=O)C(C)C2)=O)ccc(Br)c2cc[nH]c12 10650,Cc1ccc(C)c(C(N2CC(F)(C(=O)NC(C)Cn3cc(C)cn3)C2)=O)c1 10651,C(=O)(C(CC)CC(C)C)NCCNC(c1cn(CC(OCC)OC)nc1)=O 10652,c1(SC)ccc2ccccc2c1.N12CCC(C1)c1cn(nn1)CC1(CC1)C2=O 10653,C1(C(N2CCCC2CNC(C23CC4CC(CC2C4)C3)=O)=O)CCOC2(CCC2)C1 10654,c1(C(=O)NC2CCN(C(C(N3CCSCC3)C)=O)C2)nnn2c1CCCC2 10655,c1(NC(C23C(CN(Cc4ccc(SC)s4)C2)C3)=O)ccc2c(c1)COC2 10656,c1(C(N(C2CC(NC(=O)C(=O)C(C)(C)C)C2)C)=O)cc(F)cc2ccoc12 10657,N1(C(C2C(OCC)C2)=O)C(CO)CSCC1c1ccccc1 10658,c1(C(N2C(CNC(CCC(=C)C)=O)CC3CC32)=O)c(OC)cnc2ccccc12 10659,c1(CNC(C(C2(O)CCC2)NC(c2cccnc2S)=O)=O)ccc(CO)nc1 10660,C(=O)(CCCCC(=O)NC(C1CCN(C(=O)CC2CCOC2(C)C)CC1)C)NC 10661,c1(C(=O)NC2CC2)cccc(CC(=O)NC2(CCC3CCCC3)CC2)c1.COC 10662,C1(C(=O)NC(CCC)(C)CO)CCC(C)(C)N(C(c2cc[nH]c2C)=O)C1 10663,C12(NC(c3cc(C)c(C)o3)=O)COCCC1CN(C(=O)Cc1[nH]cnc1C)C2 10664,c1(C(N2CCC(c3ccccc3Br)C2)=O)ccnc2ncnn12 10665,C=CCC(C)(C)C(=O)N1CCN(C(=O)C(C2CCC2)OC)C(C2CC2)C1 10666,N1(C(CSCC)=O)CCC(CC)(NC(=O)CCCCCSC)CC1 10667,CCC(C)(C#N)C(=O)N1CC2(NC(c3cc(-c4ccccc4)c[nH]3)=O)CC1C2 10668,c1(OCC)cccc(C(c2nnnn2CCCCc2cnc(COC)s2)N)c1.SC 10669,Cc1oc(C(=O)NC2C3CC2N(C(=O)CCCN(C)C)C3)cc1S(C)(=O)=O 10670,N1(C(C(c2ccccc2)C)=O)CCC2(C1)CN(C(C1(F)CCCOC1)=O)C2 10671,C1(C(NOCC#C)=O)CCC(CNC(=O)CCc2cccs2)C1 10672,N1(C(CC=C)=O)CCCC2CN(C(=O)C(C)C=Cc3ccccc3)CCC12 10673,C12(NC(C3N(C(C)=O)CCC3)=O)CCN(C(c3c[nH]nc3C3CC3)=O)CC1C2 10674,c1(C(=O)NCC2(CCNC(C(C)(C)OCC)=O)CC2)cc(C#N)no1 10675,c1(CNC(C2CCCCS2)=O)ccccc1-n1cc(CN2CCCC2=O)nn1 10676,C1(n2cc(CCC(C)O)nn2)CON(C(=O)C(C)C(F)F)C1 10677,C1(CNC(=O)CC(F)F)CC2(CO1)CN(C(c1cc(-c3ccncc3)on1)=O)C2 10678,c1(CNC(C2CCN(Cc3scnc3Cl)C2)=O)cc(-c2cccnc2)no1 10679,Cc1oc(Br)cc1C(=O)N(C1CCN(C(C2CC(F)C(=O)N2)=O)C1)CCO 10680,N1(C(=O)CCc2nc[nH]n2)C2CCC1C(F)C(NC(C1(CCNC=O)CC1)=O)C2 10681,N1(C(Cn2cc(C(=O)OC)nn2)=O)CCCC2(CCN(C(=O)C(C)C3CC3)C2)C1 10682,C(=O)(N=c1[nH]c(Cl)ncc1O)C1N(C(c2c(OC)cccn2)=O)CC2(CC2)C1 10683,C(=O)(C(O)C(F)F)N(CCN(C(C)C)C(c1ccc(N(C)C(C)C)nc1)=O)C 10684,c1(OC(C)C)cnc(C(=O)N(C)CC2CCN(C(=O)C(F)C3CCC3)C2)cn1 10685,C(=O)(NN(C(=O)C(CC(C)C)SC)C(=O)NOC)NC 10686,CCCCCC(O)C(=O)NCCC1CCCN(C(C2CC(F)(F)CS2)=O)C1 10687,C=CCCC(C(=O)N1CC(C)(C)C1COC)NC(C1(C)CCC2CC2C1)=O 10688,c1(C(=O)NC2(C)CCN(C(C(CC#C)CC#C)=O)C2)cc2ccc(Cl)c(F)c2[nH]1 10689,C1(NC(c2cc(C(F)F)ccn2)=O)CCN(C(C2C(Cl)(Cl)C23CC3)=O)CC1F 10690,c1(SC)nc(N(C)CC2CCN(C(c3cnc(C(N)=O)cn3)=O)CC2)ncc1C 10691,N1(C(c2c(C)cco2)=O)CCC2CC(CNC(C3(C(F)F)CCC3)=O)CCC2C1 10692,Cc1onc(C(=O)NCC2CCCC(NC(C3CC(C)(C)C3)=O)C2)c1[N+](=O)[O-] 10693,Cc1ccc(C)c(C(c2nnnn2CCCOCC2CC2)NCC23CCCC2C3)n1 10694,CN1CCCC(C)(C(=O)N(C)CC2(O)CCN(C(=O)CCc3cncs3)C2)C1 10695,C(=O)(CCN=C(NCC1(S(C)=O)CC1)NC1CCC(NS(C)(=O)=O)CC1)N(C)C 10696,OCC(Cc1cccc(F)c1)CN=c1[nH]c2c(F)c(F)c(F)cc2s1 10697,c1(C(=O)NC2CC3CN(C(c4c(C(C)C)ocn4)=O)C2C3)nccn2ccnc12 10698,N1(C(C(Cn2cccn2)NC(CC2(C)CC2)=O)=O)CCCC(F)(F)CC1 10699,N(C(=NCCCCl)NCCCN1CCCC1)CC(C1CCOCC1)(C)C 10700,c1(OC)cc([N+](=O)[O-])ccc1CNC(=O)C=Cc1ccc(Cl)cc1F 10701,C(=O)(C(C)(C)CC#N)N1C(CN(C(=O)Cc2cnc[nH]2)C)COCC1 10702,C1(OC)(CNC(=O)CC2CCC2)CCN(C(=O)CC(N2CCCS2(=O)=O)C)C1 10703,CS(=O)c1ccccc1-c1cccc(NCc2ccn(-c3ccccc3)n2)n1 10704,c1(OC(C)C)ncccc1C(=O)NCC1CCC(C2OCCO2)CC1 10705,C1(N(C)C(=O)NCc2ccncc2)CCN2CCCCC12 10706,c1(C(N2CCC(NC(c3cncnc3)=O)CC2C2CC2)=O)cc([N+](=O)[O-])ccn1 10707,C=C1CC2(C1)CC(C(=O)NC1CCN(C(=O)C=Cc3cncs3)CC1C)C2 10708,C(=O)(C(C)(C)C1CCN(C(c2cnn(CC)c2)=O)C1)NC(c1ccccc1)CC 10709,C1(OC)CCN(Cc2csc(C3OCCO3)n2)C(C)C1.c12ccc(cc1)o2 10710,C1(C(N(CC=C)C(C)C2CC2)=O)CN(C)CCN1C(=O)Cc1cn(C2CC2)nn1 10711,C1(O)(CCNC(C(CC)OCC)=O)CCN(C(c2cnccc2Br)=O)C1 10712,c1(C(N2C3CC(CC(NC(c4n(C)ccc4)=O)C3)C2)=O)coc2cc(O)ccc12 10713,c1(CC(C)C(=O)NCC2CCC(NC(=O)C(F)(F)CO)C2)ccc(F)cc1 10714,C(=O)(C1CCCc2ccnn21)N1CC(C2CN(C(CS(C)(=O)=O)=O)C2)C1 10715,Cc1nnc(CN(CC(N2CCCC(CNC(=O)CC3CCOC3)C2)=O)C)n1C 10716,C(=O)(C1=C(F)CN(C(C2CCCC(=O)C2)=O)CC1)NC(c1csnn1)C 10717,C1(NC(CCN(CCC)C)=O)CC2CC1CN(C(c1ccnn1CC1CC1)=O)C2 10718,C(=O)(CCCC(C)(C)C)NCC(CC=C)NC(=O)C(=Cc1ccco1)C 10719,C#Cc1cn(C)nc1C(=O)NC1CCC(CC(N2CCCC2C)=O)C1 10720,CC1(F)CCCCN(C(=O)C(C)(C2CCC2)NC(c2cccnc2O)=O)C1 10721,C#CCCCCC(=O)NCC1(CNC(c2ccncc2C)=O)CC1(F)F 10722,N1(C(C2COCCN(C(=O)C3=C(Cl)CCC3)C2)=O)CC2CSCC(C2)C1 10723,N1(C(C2C(C(C)C)OCC2)=O)CCCC2(C1)CN(C(c1ccc(N)cc1F)=O)C2 10724,c1(Sc2cn(C)nc2)ccnc(Cl)n1.C1C(=O)NC2CC2CNC(=O)CS1 10725,Cc1cnn(CCCNC(=O)C=CCN(C(=O)CCCC2CC2)C)c1 10726,CCC(C)CC(=O)NC1CCCC1C(=O)Nc1ccc(NC(C)=O)cc1 10727,C(=O)(C(O)CCC(F)(F)F)N1CC(CNC(c2c(C)cccn2)=O)N(C)CC1 10728,CCC(CC)(C(=O)NCCC(O)CNC(=O)Cn1cc([N+](=O)[O-])cn1)C(C)C 10729,N1(C(CCOc2cc(C)on2)=O)CC2(CC(NC(=O)C3=CCCCO3)C2)C1 10730,CC1OCCC1(C)C(=O)NC1CCOC(C(=O)NCc2ncc(Cl)cn2)C1 10731,C(CCN=c1[nH]c(=NCCC(C)F)[nH]c2c1COCC2)N(C(C)=O)C 10732,CCCC(CC)C(=O)N1CC(NC(c2cc(Cl)cc(Cl)c2)=O)CC(F)C1 10733,c1(OC)ccc2ccnc(C(C)NC(=O)N(c3ccccc3)CC#N)c2c1 10734,c1(C(N2C(CNC(c3cc(CCC)on3)=O)C=CC2)=O)n[nH]c2c1COC2 10735,N1(C(C(C(C)C)F)=O)CCCN(C(=O)COC(C)(C)C)C(c2ccccc2)C1 10736,C(CC(C)C)(C(=O)N1CC2CC(C1)C2NC(c1snnc1C)=O)NC(C)=O 10737,CCC(O)C(C)C(=O)NCC1CCCN1C(=O)CN1CCCC(C(=O)OC)C1=O 10738,C(=O)(C1=COCCO1)NCC(C(C)(C)C)NC(c1c(Cl)cncc1Cl)=O 10739,C1(NC(CCCC(C)C)=O)CC2(CCCN(C(=O)C3=NOC(C)(C)C3)C2)C1 10740,N1(C(Cn2c(C)cc(C)n2)=O)C2CCC1C(NC(c1ccsn1)=O)C2 10741,N1(C(C(C)(C)c2ccno2)=O)CC2CC(NC(c3csc(F)c3)=O)C(C2)C1 10742,C12(C(=O)NCCC3OCCN(C(C(CCSC)O)=O)C3)CCC(CC1)C2(C)C 10743,Cc1ccc(C(=O)NCC2CC(C(=O)NCCC(=O)N3CCCC3)=NO2)cc1F 10744,C1(C(=O)OC(C)(C)C)(NC2CC3CC3C2)CCOCC1 10745,N1(C(C2(OC)CC(c3cn(CCC(=O)OC)nn3)C2)=O)CC2COCC2(C)C1 10746,C1(C(F)F)CC(=O)N(C(C)(C)CO)C(C(CSCC=C)=O)CCN1 10747,c1(CSCC(=O)N(C(CNC(CCC(=C)C)=O)C)C)nc2ccccc2[nH]1 10748,C1(n2cc(CC(C(=O)NCC(COC)C(=O)OC)(C)C)nn2)CCc2nn[nH]c2C1 10749,C1(C(N2CC=CC(NC(c3c(C)oc(CO)c3)=O)C2)=O)CCCC1P(C)(C)=O 10750,c1(N2CC3C(CNC(C(C)Cc4ccco4)=O)C3C2)ncnc(Cl)c1Br 10751,C1(NC(C(F)=C(C)C)=O)CC2CCC1C1CN(C(=O)C=CC3CCCC3)CC21 10752,N1(C(CC2N(C(c3cc(C)c(C)nn3)=O)CC2)=O)CCCC(O)(C2CC2)C1 10753,C(c1ccc(C)cc1C)=CC(=O)NCC1(C)N(C(CC=C(C)C)=O)CCC1 10754,N1(C(c2c(CC)nccn2)=O)CCCN(C(=O)C(O)CC(F)(F)F)C(C)C1 10755,c1(C(=O)NCC2C(C)CCN2C(c2nnsc2C(F)F)=O)ccc(OC)cc1F 10756,C#Cc1ccc(C(N2CCN(C(=O)NC(C)(C)C)C(C(=O)OC)C2)=O)cn1 10757,Cc1cc(=O)n(C)cc1NC(=O)C(N)COC(C)(C)C 10758,C1(NC(c2ccn(CCCC)n2)=O)CC(O)CN(C(c2ccc(CF)cc2)=O)C1 10759,N1(C(CCOC)=O)C2CC=C(C(=O)NC(c3cc(C)on3)C)C1CC2 10760,c1(C(C(=O)NCC(CC(C)C)NC(c2sccc2F)=O)C)c(F)cccc1F 10761,C(C(CC(C)C)C(=O)NCC1COCC1NC(c1cc(C(=O)OC)no1)=O)OC 10762,S(=O)(=O)(c1ccc(N2CCOC(C)(CCO)C2)c(Cl)c1)NC(CCC=C(C)C)C 10763,S(=O)(=O)(c1cc(C)c2ccc(Cl)cc2n1)N1C(CC)C(C(=O)O)CCC1 10764,C1(CC)COCCN(C(=O)C(=O)NCCn2cc(C(C)(C)N(C)C)nn2)C1 10765,c1(C(N2CC(NC(C3(SC)CC3)=O)C(F)C2)=O)ccc2nc(O)[nH]c2n1 10766,C(CCN=c1[nH]c2c(c(=NCCN3CCOC3=O)[nH]1)COC2)SCC(C)C 10767,c1(CC)noc(C)c1N(C)C(N1CCC(C2CCCCN2C(=O)C2CC2)C1)=O 10768,Cc1nc(C(=O)NCCC(C)N(C)C(C2CC2C#N)=O)c2n1CCCC2 10769,N1(C(CCCOCC=C)=O)CCN(C(=O)C(O)CC)C(CC(=O)NCC)C1 10770,C1(NC(=O)CCCc2cccc(Cl)n2)CN(C(=O)CC(F)(F)Cl)CC12CC2 10771,N1(C(C(CC=CC)NC(=O)CC2NC(=O)NC2=O)=O)CCCC(O)(CO)C1 10772,c1(C(=O)NCC(C)CNC(C23CC(C(F)F)(CO2)C3)=O)ncc2ccccn12 10773,C1(CNC(CC(=C)Br)=O)CCCC2(CCN(C(=O)C(C)CN(C)C)CC2)O1 10774,CCCCC(O)C(=O)NCc1cc(C(=O)NC2CCN(C(C)C)CC2)no1 10775,N1(C(C(C)(C)NC(=O)NCC)=O)CCCC(CNC(=O)C(C)c2ccsc2)CC1 10776,c1(CC)c(C(N2CCC(NC(=O)COCC(F)(F)F)C(F)C2)=O)cccc1F 10777,c1(C(N(CCCNC(CC(CC)C)=O)CCO)=O)ncnc2cc[nH]c12 10778,S(=O)(=O)(c1ccc(=NCCc2ccc(OC)nc2)[nH]c1)NC(CCSCC)C 10779,Cc1cnc(C(N2CCC(NC(C3CCC(C)O3)=O)C23CC3)=O)c(C)c1 10780,CC1=NNC(=O)C1CC(=O)NC(CNC(=O)C(C)N1CC(C)C1)C(C)(C)C 10781,c1(C(=O)NCC(C)NC(c2cccc(C(C)=O)c2)=O)cccc2c(C)cccc12 10782,C(C1CN(C(c2cc(C)c(O)nn2)=O)CC1C(=O)NCCC(O)C1CCC1)=CC 10783,c1(COC)ccc(C(=O)N(CC(C)NC(=O)COCC2CC2)CC)cc1F 10784,c1(CC)noc(COCC(=O)NC(C)(C)CNC(=O)CN2CC(C)C2)n1 10785,C=CCN=C(NCC1CCN(C(=O)OC)C1)N1CCCC2(CCSC2)C1 10786,C=CC(C)(C)CC(=O)NC(C1CCN(C(=O)CCS(C)=O)C1)(C)C 10787,C1(C(=O)NCC(C)N(C(C(=O)NCCC)=O)C)CCS(=O)(=O)C1(C)C 10788,c1(C(=O)NCCC(C)N(C(CN2C(C)CC2)=O)C)nn(C)cc1N 10789,C1(CC)CCN(C(=O)CC(C)(C)O)C1CNC(c1cc(C)ncn1)=O 10790,C1(CN(C)C(C2(O)CCSCC2)=O)CC(F)CN1C(c1ccc(C(F)F)o1)=O 10791,c1(COC(c2ccc(OC3CCOCC3)cc2)=O)cc2c(s1)CCOC2 10792,C1(OC)CN(C(=NCCCCl)NCCNc2ccc(SC)cc2)CC1O 10793,Cc1c(C(F)(F)F)n[nH]c1C(N1CC(CNC(c2cccc(N)n2)=O)CC1C)=O 10794,c1(C(=O)NC(c2cccc(C)c2)CNC(C(C)(C)SC)=O)nc(Cl)ccc1N 10795,FC(F)C(F)(F)CCN=c1[nH]c(N2CCOCC2)nc(=NCCc2cnn[nH]2)[nH]1 10796,c1(NC(c2cn(CCOCCNS(C)(=O)=O)nn2)C)ccc(Cl)cc1C#N 10797,C1(CNC(=O)CCCn2ccnn2)CC2(CC2)CN1C(=O)COCC1CCC1 10798,C1(C(C)C)C(NC(c2cnn(C)c2N(C)C)=O)CCN1C(c1cnn[nH]1)=O 10799,C(=O)(C1=CCCC1C)N1C(CO)CC(NC(c2n(CC)c(O)nc2)=O)C1 10800,C1(C(N(CC(=O)NCCn2nccn2)C2CCC2)=O)Cc2nccn2C1 10801,C(=O)(CC(C)CC(C)(C)C)N1CC(NC(c2c(C)ccc(C)c2)=O)C(F)C1 10802,c1(NC(N(C(C(CC)C)C)C2CC2)=O)c(F)cccc1F 10803,c1(N2CC3(C(C(=O)Nc4c(C)ccc(I)c4)C3)C2)ncnc2c(C)csc12 10804,S(=O)(=O)(c1ccc(Cl)cc1)CC(=O)NC(C)CCNC(=O)C(C)OC(C)(C)C 10805,C(=O)(CCN(OC)C(=O)c1coc2c1COC2)N1CC(COC)(OC)C1 10806,c1(C(C)C)nc(C(=O)NCC(F)(F)C(F)F)n(-c2cccc(Br)c2)n1 10807,c1(CC)csc(CN(C(CC2(C)CCOC2)C(=O)NC2COC2)C)n1 10808,C12CC(c3ccccc3)(C1)NC(=O)C(=O)N2.C(=O)(CC(C)C1CCCO1)OCC 10809,c1(CCC(=O)NC2CCCC(C(=O)NCC(C)(C)C(N)=O)C2)ccc(F)c(F)c1 10810,Cc1cccc(OCC(=O)Nc2ccccc2CNC(=O)CC(C)(C)C#N)c1C 10811,c1(OC)c(Cl)ccc(C(=O)NCCC2CCC(NC(=O)C(O)CSC)C2)c1F 10812,c1(C(N(CCC(C)NC(c2cnoc2C2CC2)=O)C)=O)cc(F)cc2nn[nH]c12 10813,c1(C(N(CC(C)NC(=O)C(F)(F)c2cscn2)C)=O)cn(C)nc1Cl 10814,Cc1c(C(=O)NCCC2CCCCN2C(C2CN(C)CCO2)=O)cnn1C1CC1 10815,C1(C)(CC(=O)N(C2CC(NC(=O)C(O)Cc3cnc[nH]3)C2)C)CCCO1 10816,CC(C)(C)C(=O)N1CCCC1C1(C(=O)NCCC=CBr)CC1 10817,C(CC(C(=O)NC(c1ncc(F)cn1)C)NC(c1ccoc1Cl)=O)=CC 10818,N1(C(=O)NCC2(CC(F)F)CCCO2)CCC(C2(O)COC2)CC1 10819,C1(CNC(c2cc(OC)ns2)=O)CN(C(C2(c3cc[nH]n3)CC2)=O)CCN1 10820,C1(CNC(CCCOC(C)C)=O)CC(C)(C)CN1C(=O)CC1(O)CCCOC1 10821,C1(C(C)C)CN(C(C2CC2(C)C(F)F)=O)CC1C(=O)N(C)Cc1cnn[nH]1 10822,N1(C(c2csc(Br)n2)C(=O)NCC(=C)C)CCC(CO)(COC)C1 10823,C1(NC(CC=CCC)=O)CC(O)CN(C(=O)C(=O)Nc2ccccc2)C1 10824,N(C1CCSc2ccc(F)cc21)C(c1c(Cl)c(OC)cc(OC)c1)=O 10825,c1(NC(C2(C(=O)OCC)CC2)=O)ccc(NC2CCC(CO)(OC)CC2)c(O)c1 10826,CCCCC(C)CCC(=O)NCC(CC)N(C)C(C1CC(F)(F)C1)=O 10827,c1(C(=O)NCC2N(C(CC(=C)C)=O)CCC2C)cc([N+](=O)[O-])sn1 10828,CC1CC2(CC(C(=O)N(C(C)(C)CC(=O)N3CC(c4ncccn4)C3)C)C2)C1 10829,CC1CCN(C(c2cc(Cl)cs2)=O)CCN1C(=O)CC1OCCCC1(C)C 10830,C1(CNC(C2CC2CF)=O)CN(C(=O)Cn2ccnc2)CC12CC2 10831,C(=O)(CCC(CC)NC(=O)C(C)(C)C(C)O)NCC1(CCC=C)CC1 10832,Cc1ccc(NC(=O)Cn2cc(C3CC(NC(C45CCC4CC5)=O)C3)nn2)cc1 10833,N#Cc1ccc(C2CC2NC(=O)NCc2ncc[nH]2)cc1 10834,C1(NC(CS(CC)(=O)=O)=O)CCC2CCN(C(=O)Cc3ccco3)C1C2 10835,C1(N(CCC)C(c2cc(C)co2)=O)CCN(C(=O)CSCC2CCCCO2)CC1 10836,C1(C(N2CC(CCOC)C2)=O)CC(C)(C)CCN1C(c1cccc(C)n1)=O 10837,Nc1c(C(=O)NC2CC(CCNC(=O)CN3CCCC3CO)C2)cc(F)cc1Cl 10838,c1(CC(C(=O)C(C(N2CCSCC2)C)=O)O)ccc(F)cc1.C1(N)CC(N)C1 10839,c1(NC(=O)Cc2cc(F)cc(Br)c2)ccc(OCC(F)F)cc1F 10840,c1(OC)cc(C)cc(C(=O)NCC=CCNC(c2cnc(C)nc2CO)=O)c1N 10841,C(=O)(C(C)(C)C(F)(F)F)NC1CN(C(c2nc(CC)sc2N)=O)C(C)(C)C1 10842,Cc1cc(C(=O)NC(C)(CNC(C2CC2C(N)=O)=O)C(C)C)cc(C)c1C 10843,Cc1cc(C(=O)NCC2(CNC(=O)CC3COC(=O)C3)CCC2)n(CC(F)F)n1 10844,N1(C(C(CC)=CC)=O)CCC(C)C(NC(c2cc(Cl)cc(Cl)n2)=O)C1 10845,C1(CC(=O)OC)CC(C)(C)CN1C(=O)NC(C1(n2cccn2)CC1)C1CC1 10846,C1(NC(CCNC(N)=O)=O)CCCCC1NC(C1(CO)CC(F)(F)C1)=O 10847,C(=O)(C(=O)CCCC)N1CCC(N(C(CC=CC=C)=O)CC2CCCO2)CC1 10848,C1(N(C)C(c2ncoc2C2CC2)=O)CCCC(NC(=O)C=Cc2cncn2C)C1 10849,c1(C(N2C3CC(NC(c4c(C)[nH]cc4)=O)CC2CC3)=O)nncc2c1CCCC2 10850,C1(C(N(C2CC3(CC3)C2)C)=O)CC2CC1CN(C(C1CC1C1(C)COC1)=O)C2 10851,C1(C(=O)OC)CCC2(CCC2)N(C(=O)CCC2CCOC2=O)C1 10852,C1(OC)CCC2(CCN(C(C3CC4C=CC3N(C(=O)CC(C)OC)C4)=O)C2)C1 10853,C1(n2cc(C3CCN(C(c4nc(C)oc4)=O)CC3)nn2)CC(C)CCC1O 10854,c1(SC)nc(C(N2CCCC2c2cn(CC3CCCC(=O)N3)nn2)=O)c2n1CCCC2 10855,C(=O)(CS(=O)C(F)(F)F)N1CCC(CNC(CCOC)=O)C1(C)C 10856,Cc1cc(OCC(=O)NC2CC(NC(C3CCOC(=O)CC3)=O)C2)ccc1Cl 10857,C(=O)(CCC[N+](=O)[O-])NCC1N(C(C(Cc2c(C)noc2C)C)=O)CCCC1 10858,C1(NC(CC2N(CC)CCC2)=O)CC2CC1CN(C(c1cc(C(N)=O)c[nH]1)=O)C2 10859,Cc1nn(C)c2c(N3CCC4(CC4)C3)nc(=NCC3CC3C3CC3)[nH]c12 10860,C(N=c1[nH]c(C(F)F)nc2ccccc12)C1CN(c2c3ncn(C)c3ncn2)C1 10861,c1(NC(CC(C(C)C)CCO)=O)ccc2c(c1)CCO2.C(=O)(C(C)(O)C(F)(F)F)N 10862,C1(NC(C(C)NC(=O)NCC)=O)C=CCN(C(c2cc(OCC)n[nH]2)=O)C1 10863,C1(n2cc(CNC(C(C)=C(C)C)=O)nn2)CCN(C(=O)CCc2cccs2)CC1 10864,C1(NC(=O)Cc2ccc(O)cn2)CCCCCCC1NC(=O)CCc1ncc[nH]1 10865,c1(CC(N2C(CNC(C(C(C)C)(C)O)=O)COCC2)=O)cccc2c1OCCO2 10866,N1(C(CN(C(C)=O)C)=O)CCC(C2N(C(=O)CC3CC3(C)C)CC2(C)C)CC1 10867,N1(C(C(c2c(C)n[nH]c2C)C)=O)CCCN(C(c2cnns2)=O)C(C)C1 10868,C1(C(N2CC(CNC(=O)CSC)C(C(F)(F)F)C2)=O)(COC)CC=CCC1 10869,c1(OC)cc(C(=O)NC(C)C(CO)NC(=O)C(C)Sc2nncn2C)on1 10870,N1(C(C(C)SC(C)C)=O)CC(C2CC2)(C(=O)NC2C3CCCC23)C1 10871,C12(C(=O)NC3CC(C)N(C(=O)CCC4CCCC4)C3)CC(C)(CCO1)C2 10872,CCC(C)CCC(O)CC(=O)N1CC(F)(c2cn(Cc3nc(OC)cs3)nn2)C1 10873,C1(C)(CC)CCC(NC(=O)C(=O)N(c2ccccc2)CCNS(C)(=O)=O)C1 10874,c1(CC(N2CC=CC(NC(c3cncc(C#C)c3)=O)C2)=O)cn2cc(C)sc2n1 10875,C1(CN(C(CCN(CC(F)(F)F)C)=O)CC2CC2)CCN(C(=O)OC(C)(C)C)C1 10876,Cc1cccc(C(=O)NCCC(C)NC(c2ccc(C3CCCCC3)cc2)=O)c1 10877,C(CCCCC(=O)NC1CC(CCNC(=O)CCc2cnc(C)s2)C1)NC(C)=O 10878,N1(C(C(C(C)C)F)=O)CC2CCCC(NC(c3csnc3Cl)=O)C2C1 10879,CC(C)CC(C(=O)NC(C)CCN(C)C)ONC(=O)COC1CC1 10880,c1(CN2CC(C(N(CC)Cc3ccncc3)=O)SCC2)cnc(Cl)c(Cl)c1 10881,CCC(F)(F)CC(=O)N1C2CCC(C2)C1CNC(=O)C(C)Oc1ccccc1 10882,C1(C(N2CCC(NC(c3n(C)nnc3)=O)(CO)C2)=O)CCc2nccn2CC1 10883,c1(C(=O)NCC2C(CNC(C=C(CC)CC)=O)C2)cc(F)ccc1Br 10884,c1(SC(C(=O)NCC2CC(NC(C(c3cnccn3)C)=O)C2)C)ccccn1 10885,C1(O)(C(N2C(C(N3CCCCC3CO)=O)CC2)=O)CCOCC1 10886,c1(OCC)ncccc1C(=O)NCC1CC(O)(CNC(=O)COC)C1 10887,Cc1ccc(C(=O)NCCOC(C)(C)CNC(c2nccnc2C)=O)c(Cl)c1 10888,c1(NC(CN(C(=O)CC2CCCS2(=O)=O)CC)C(=O)OC)ccc2nn[nH]c2n1 10889,N1(C(CC(C)F)=O)CCC(C)(C)CC1C(=O)NCc1cncc(C#N)c1 10890,C(c1ccccc1Cl)=C(C)C(=O)NC1CC(C)N(C(=O)CCn2ccc(=N)[nH]2)C1 10891,c1(CC(=O)NCC2C=CC(NC(=O)C=CC(=O)NC3CC3)C2)cc(F)cc(Cl)c1 10892,S(=O)(=O)(c1cc2c(Br)cncc2s1)NCCC1CCN(C(C)=O)CC1 10893,C1(C)(CC)CC(C(=O)NCC2N(C(=O)C3=C(C)OCC3)CCC2(C)C)CCO1 10894,C12CCN(CC1)C2=O.C1(NC(COCc2nnc(C)s2)=O)CC12CC(O)C2 10895,c1(CC)cnc(N2CCCC2CCC(=O)NCc2cc(OCC)ccn2)c(Cl)c1 10896,CCC(C)C(CC(=O)N1CC(S(C)(=N)=O)C1)NC(C1CCC1C)=O 10897,C(=O)(CCCCC(=O)N1CC(CNC(=O)CN2CCCCC2)CC1C)OC 10898,c1(C(=O)NCC(CCC)NC(=O)CCN(C)CC)c(C)coc1CC 10899,c1(C(C(=O)NC2CCC2)N(Cc2cncs2)CC2CCCO2)ccc(F)cc1Br 10900,CC(C)C(C(=O)NC1CC1)N(CCC(C)N(C)C)C(C1CCC(=O)C1)=O 10901,N(C1COc2ccc(Cl)cc21)C1(c2n(CCSC)nnn2)CCN(OC)CC1 10902,c1(CNCCC2(OC)CN(C(C(CCC)O)=O)C2)nc(C)nc2sc(C)c(C)c12 10903,c1(NC(=O)CC2CCCO2)ncc(F)cn1.C12CCC(C1)CNC2=O 10904,c1(-c2nc(C(=O)Nc3cc(CCC)no3)c(C)s2)cccc(I)c1F 10905,C1(NC(=O)NCCn2cc(CN3CCC(=O)NC3=O)nn2)CNC(=O)CC12CCC2 10906,N1(C(c2cn(C)nn2)=O)CCCC(CCNC(=O)CCC2CCC2)CC1 10907,c1(OC)ccc(C(=O)O)cc1CN1CCC(O)C(C(=O)Nc2nc(C)ccc2F)C1 10908,C12(CNC(c3n(C(C)C)cnc3)=O)CC1CN(C(=O)Cn1cc(C#N)cn1)C2 10909,c1(CN2CC3(N(C(c4cc(F)c(F)cc4I)=O)CC3)C2)cc(Br)cc2[nH]ccc12 10910,Cc1nc2ccc(C(N3CC(NC(=O)C(C)C#N)C(n4ccnn4)C3)=O)cc2o1 10911,CCC(C)(COC)C(=O)NC1CC2CC1N(C(c1ccc(C(C)(C)C)cc1)=O)C2 10912,N1(C(c2cncc(NCC)c2)=O)CCC(NC(C2(CCCF)CC2)=O)C(CO)C1 10913,C1(CC#C)(C(N2CCCC2CC(=O)NC)=O)CCN(C(=O)C(COC)COC)C1 10914,c1(CC)ncc(C(=O)NCC2CCCC2NC(c2cc(OC)n[nH]2)=O)o1 10915,N1(C(c2c(C)nccc2Cl)=O)CCCC(NC(=O)C=Cc2ccsc2)C(F)C1 10916,N1(C(C(C)C2CCOC2)=O)CCC2CCC(C1)N2C(c1cc(=O)cc[nH]1)=O 10917,c1cc(F)cc(F)c1OC.C12CN(CC1(F)F)C(=O)c1ncsc1C(=O)N2.CC 10918,N1(C(CC(=O)NCC#C)=O)CCC(C(=O)NCCCC(C)(C)O)C12CCC2 10919,N1(C(CC(C=C)C)=O)CC(C)N(C(=O)C2=NOCC2)CC1C 10920,N1(C(C2=C(C)OCCC2)=O)CCC2(CNC(C3CCC(O)CC3)=O)CCCCC12 10921,c1(N(C(Cc2cn(CC(=O)O)nn2)=O)C(C2CCC(O)C2)=O)ccnc(O)c1Br 10922,C1(NC(CC2(NC(C)=O)CC2)=O)C(C)CN(C(c2nccn2C(C)C)=O)CC1C 10923,CCCCC(F)C(=O)NC1CCCCC1C(N1CCC(C(CC)CC)C1)=O 10924,c1(C(=O)NC2CC3(C2)CC(NCc2ncco2)C3)noc2ccc(Br)cc12 10925,c1(NC(c2sc(C)cc2Br)c2n(C(CC)C)nnn2)ccc(C(N)=O)cc1Cl 10926,Cc1cc(C(=O)NC2CC3CN(C(=O)C(F)(F)CO)CC23)cc2nn[nH]c12 10927,CCCC(C(=O)NC(C)CCNC(c1nn(CC)nc1Br)=O)NC(N)=O 10928,CN(C)S(=O)(=O)N1CCCC1NC(=O)CNC(=O)CC(=O)Nc1nccs1 10929,C(=O)(C(O)C1=CCCCC1)NC(C(=O)NCc1c(C)cnn1C)CC1CCCC1 10930,c1(C(=O)NCC2C(NC(c3cccc(O)n3)=O)C2)cc(Br)ccc1[N+](=O)[O-] 10931,c1(N(CC(N2CCC(O)(CN)C2)=O)C)ccc(NC(c2scc(C)n2)=O)c(Cl)c1 10932,c1(C(=O)NC(C(C(C)C)C)CNC(c2ccn(C)n2)=O)cc2ccc(O)cc2[nH]1 10933,C1(CCNC(C2CN(C)C(=O)C2)=O)CN(C(c2cccc(Cl)c2F)=O)CCCO1 10934,c1(C(N2C(C3CCN(C(C(C)NC=O)=O)C3)CCC2)=O)cccc(=O)n1C 10935,n1(CCC)c(C(N2CCC(NC(=O)C(O)C(F)F)C23CC3)=O)cc2ccccc12 10936,C(=O)(CCCn1cc(CCOCCN)nn1)N(CC(CN(C)C)O)C 10937,C1(CN(C(C2(Cc3ccc(Cl)cc3)CC2)=O)CC)CCN(C(=O)C(O)CF)CC1 10938,C(=O)(CC=CC(C)(C)C)N(CCN(C(C1C(C)C1)=O)C)C 10939,c1(C(N2C(C3(O)CN(C(c4ccn(CCC)n4)=O)C3)CCC2)=O)ccc(=N)[nH]n1 10940,C(N=c1[nH]c(=NCC2CCCSCC2)[nH]c2c1CC(C)CC2)c1[nH]c(=NC)sc1 10941,C1(N(C(CCN(C(C(COC)O)=O)C2CC2)=O)C)CCCC(C)C1C 10942,N1(C(CCOCC#C)=O)CC2CCC1CN2C(C1CCCC(C)CC1)=O 10943,S(=O)(=O)(c1ccc(N(C(C)COCc2cccc(C)c2)C)cc1Cl)NCCOC 10944,C(=O)(CCCCC(N)=O)N1CCC(NC(c2c(C)ccc(OC)c2)=O)(CF)C1 10945,C(=O)(CCCC(C)(F)F)N1CC(N(C(=O)C=Cc2ccnn2C)C)C(C)(C)C1 10946,c1(C(=O)NC(C)CCNC(=O)C=CC2CC2)c[nH]c2cccc(Br)c12 10947,c1(C(N2CC3CN(c4nccnc4F)CC3C2)=O)c(F)c(F)cc(F)c1F 10948,C(=O)(CP(C)(C)=O)NC1(CCNC(CCc2n(C)ncc2)=O)CCCC1 10949,c1(N(c2ccccc2)CCCOC)nnc(-c2ccc(C)nc2)n1CCC#N.CS 10950,c1(C(=O)NCC2(C)CCN(C(c3nocc3C(C)(C)C)=O)C2)cc2c(s1)CCC2 10951,N1(C(C2(COC)CC(=C)C2)=O)CC=C(C(=O)N2CCC(CC)C2)C1 10952,c1(SCC)c(C(=O)N(C(=O)C(O)CC)c2ccccn2)cccc1Br 10953,C1(NC(C(CCCC)O)=O)Cc2ccccc2C1NC(C1(CC)CC1)=O 10954,C1(O)(CN(C(C(C)=C2CCCC2)=O)C)CCCN(C(C2CN(C3CC3)C2)=O)C1 10955,C1(C)(C(N2CCC(C(N3C(CC(C)(C)C)CC3)=O)(CO)C2)=O)CC2(CCC2)C1 10956,N1(C(CCOCC)=O)CCC2(CC1)COC(CNC(C1(C)C=CCC1)=O)C2 10957,c1(CCC(=O)NCCSC(CO)C(=O)O)nc(-c2cccnc2)no1 10958,N1(Cc2n(C)nc(C3CC3)c2)CCC(CNC(=O)Cc2ccccc2O)C(O)C1 10959,c1(C(N(C(C)CNC(c2cccc(O)c2)=O)C)=O)cccc2nsnc12 10960,C(=O)(C1Cc2ccccc21)NC(CCC=C)C(=O)NC1CCC2(CC1)N=N2 10961,Cc1ccc(SC(C)C(=O)NC2C=CCN(C(=O)CC3CCC(=O)NC3)C2)cc1 10962,N1(C(CCC(=O)NC(C)CCN(C)C(C2CCC2C)=O)=O)CCc2sccc2C1 10963,c1(COC)nc(C)c(C(=O)NCCC(C(C)C)NC(c2n[nH]cc2C(C)C)=O)s1 10964,C1(NC(C2N(CC)CC2)=O)C2CCC1N(C(=O)Cn1ccc(Br)cc1=O)C2 10965,c1(OC(C)(C)C)c(F)cc(C(=O)OCC2CN(c3ccccc3)C(=O)O2)cc1F 10966,n1(CC)cc(C2CCC(NC(=O)N(C3CC(O)C3)C(C)C)C2)cn1 10967,C1(C(=O)NC2(C)CC(NC(c3cc(Cl)ccc3Cl)=O)C2)CCC2(CCC2)O1 10968,c1(SC)ncc(C(F)(F)F)c(N(C(c2cc(C)cc(F)c2)=O)CC2CCNC2)n1 10969,S(=O)(=O)(c1ccc(N(C)CCOc2ccccc2)c(C#N)c1)NCCSCC=C 10970,N1(C=O)CCC(C(F)C(=O)NCC)C1.C1(=O)CC2(CC2)OC(=O)C12CC2.OC 10971,c1(CCC(=O)N(C2CCC(NC(c3ncoc3C3CC3)=O)C2)C)ccc(F)nc1 10972,O=C(C#CC1CCCO1)N1CC2(CCN(C(C3(C(F)(F)F)CC=CCO3)=O)C2)C1 10973,Cc1noc(C)c1S(=O)(=O)NCC1CCN(C(c2ccc(Cl)s2)=O)C1 10974,c1(OC)cc2c(cc1C(=O)NC(C)(CNC(=O)CN(C)C1CC1)CO)CCC2 10975,c1(C(=O)NC(CC)Cn2cncn2)c[nH]nc1CCNC(C1(C)CC1)=O 10976,c1(CNC2C(C(N3CCC(Br)CC3)=O)CCC2)c(F)ccc(Cl)c1F 10977,C#CC1CN(C(=O)C(C2CCCO2)NC(=O)C=CCCC(C)C)CCN1C 10978,C(c1ccccc1Cl)=C(C)C(=O)NCC1(CNC(=O)CCCCN(C)C)CC1 10979,c1(C(CC(N2CC(CNC(CN(C)CC)=O)OCC2)=O)C)ccc(C)c(OC)c1 10980,C(C)(C)(CCCNC(=O)CC1C=CCC1)n1cc(C(COC)(C)O)nn1 10981,c1(C(N2C3C(NC(c4occc4Cl)=O)CC(C3)C2)=O)cccc2occc12 10982,C(=O)(CCCCCN=[N+]=[N-])N1CC(C)N(C(C2(CCC)CC2)=O)C(C)C1 10983,C1(CNC(CC2N(C(C3CC(C(C)C)C3)=O)CC2)=O)CNC(=O)CO1 10984,c1(OCC(N2CC(C)C(NC(C3C4CC5C(C4)C35)=O)C2)=O)ccc(Cl)c(Br)c1 10985,C12C(C3CC3)CCN1C(=O)CCCOC(OCC)c1cn(nn1)C2.C(C)(C)OC 10986,c1(C(=O)NC(CC(C)NC(C(C)=C2CCCC2)=O)C)c(C)nc(C(C)C)nc1S 10987,N1(C(CC=CCCCCC)=O)CCC2CCC(C1)N2C(=O)COCCC 10988,N1(C(c2cc(CNC(C3(COC)CC3)=O)sc2)=O)CCCC1C1CCCO1 10989,Cc1nccnc1C(C)OC(c1csc(-c2ccccc2)c1)=O 10990,Cc1nnc2n1CC(C(=O)NCCN(CCCN(C)C)C(=O)Cc1cocn1)C2 10991,N1(C(c2cnc(CC)[nH]2)=O)CC(C(F)F)CC1CNC(=O)CCCN(C)C(C)C 10992,C(=O)(C(C)C(C)(C)C)N1CCC(CC(C)NC(c2c(COC)nn(C)c2)=O)CC1 10993,N1(C(c2cn(CCN(C)C)nc2)=O)CCC2(CC1)CC2NC(c1cscc1F)=O 10994,c1(C(C(=O)NCCC(=C)CNC(c2cnc(N)cn2)=O)CC)cccc(Cl)c1 10995,C(C)(CNC(=O)CCn1cccc1)(C(C)C)NC(COCCCOC)=O 10996,c1(C(=O)NCC2C(NC(c3c(C)nn[nH]3)=O)CCC2)cnn(CC(F)F)c1C 10997,c1(C(C(=O)NC2CCN(CC(=O)NC)CC2)NC(CCC#C)=O)c(C)cccc1Br 10998,C1(C(N2CCC(O)(CCNC(CCc3nc(C)sc3)=O)C2)=O)CC12CC(C)(C)C2 10999,c1(C(N(CCCCCC)CCNC(=O)C(C2CC2)C2CC2)=O)n[nH]c(C)c1Cl 11000,N1(C(CSCC)=O)CCC(CNC(C2CC2C2CC2C)=O)C12CC2 11001,C=CC(C)(C)CC(=O)N(C(CC(F)F)C(=O)N1CCC(OC2CCC2)C1)C 11002,c1(C(N2CC(C)(CCC(=O)NC3CN(CCC)C3)C2)=O)cc2ccccn2n1 11003,N1(C(c2nc(C(C)=O)sc2)=O)CCC(C2CCN(C(=O)COCCO)C2)CC1 11004,c1(CCC(N2C(C)CCC(NC(C=C(C)Cl)=O)C2)=O)ccc2ocnc2c1 11005,c1(CC)ccc(C(=O)NCCN(C(C2CC23CCOC3)=O)CC)cc1C(F)(F)F 11006,N#Cc1cc2c(n(CNCc3nc4ccccc4n3C(F)F)c1=O)CCC2 11007,C1(NC(CC(=O)OC)=O)C2CCCC1CC(NC(C1CN3CCN1CC3C)=O)C2 11008,N1(C(C2CCN(C(CCC)=O)CC2)=O)CCN(C(C2CNC(=O)C2)=O)C2CCC12 11009,C1(n2cc(-c3cn(CC)nc3)nn2)CCCN(C(C2CCC(=O)CC2)=O)C1 11010,c1(NC(C2N(Cc3c(C)noc3)CCC2)=O)cc(Br)ncc1F 11011,C1(c2n(CC)nnn2)(NC2CCCC(C)O2)CCN(c2cccc(C)n2)CC1 11012,c1(C(N2CCC(CCNC(C3(COC)COC3)=O)C2)=O)ccc(C(C)C)nc1O 11013,C1(C(=O)NC2C(NC(c3cccc(C(F)F)c3)=O)COC2)CS(=O)(=O)CC12CC2 11014,C1(NC(c2nnn(-c3ccccc3)n2)=O)CC2(CCCCN2C(C2CCO2)=O)C1 11015,Cc1c[nH]cc(C(N2CC(NC(=O)CSc3cn[nH]c3)CC(O)C2)=O)c1=O 11016,C1(C(=O)NC(C=C)CO)(CC)CCN(C(=O)CC2CCCCN2C)C1 11017,c1(CC)onc(C)c1C(=O)NCC1(O)CN(C(=O)CCn2c(C)nccc2=O)C1 11018,CC1(NC(=O)CCF)CCN(C(=O)C(C)(C)c2ncco2)C1 11019,C#CC1(NC(N2CC(C(=O)NC)(CC)C2)=O)CCCCC1 11020,c1(CC)cnoc1C(=O)NCCN(C(c1cc(C(C)(F)F)n[nH]1)=O)CC 11021,c1(CC(=O)NCC(O)CNC(c2csc(-c3ccoc3)n2)=O)ccc(F)cc1 11022,CC1(O)CCC(NC(C2CC(F)(F)CN2C(=O)CC23CCCC2C3)=O)CC1 11023,c1(OC)cccc(S(=O)(=O)N2CCC3CCC(C2)N3C(=O)Cc2ccn(C)n2)c1 11024,N(C1CCc2c(F)cc(Br)cc21)C(c1nc2ccc(C)cc2s1)=O 11025,c1(CN(C)C)cc(C(=O)NC2CCC(CNC(=O)C(F)CC3CC3)CC2)ccn1 11026,C(CCCC(=O)NCCC(C)N(C)C)NC(C(N1CCOCC1)C)=O 11027,C1(CNC(c2ccc(SCC)cc2)=O)CC(F)(F)CN1C(=O)C(C)S(N)(=O)=O 11028,C1(C(=O)NCC2CC3CCC(C2)S3)C2CCCCCCC12 11029,Cc1cccc(Cl)c1CC(=O)NC1CC(CNC(=O)C=C(Cl)Cl)C(O)C1 11030,C1(C(N2CCC(C)(O)CC2)=O)CC2(CCC2)CN1C(=O)CSCC(F)F 11031,c1(N2CCN(CC(C)(C)NC(C(CCC)(C)C)=O)CC2)nc2cc(C)ccc2o1 11032,C1(C(=O)NCC2CCC2(F)F)CCCN(C(c2ccc(O)nc2)=O)CC1 11033,C1(C(=O)NC2(C)CCCN(C(c3cc(O)cc(=O)o3)=O)C2)CCC(C2CC2)CC1 11034,C1(CC)CN(C(=O)CNC(=O)CCc2csnn2)CC1F 11035,CN1CC=C(CC(=O)N2CCCCC(N(C)C(C3COCCN3C=O)=O)C2)CC1 11036,C12(c3onc(C)n3)CCC(CC1)N2C(=O)C(c1cccc(O)c1)C 11037,c1(OCC)cnc(C(=O)N(C)CC2CCN(C(c3ccn(C(C)C)n3)=O)C2)cn1 11038,c1(C(=O)NCC2(F)CCCN(S(CC)(=O)=O)C2)cnc2[nH]c(C)nc2c1 11039,C1(C(=O)NC2(CN(CC)CC)CC2)COCCN(C(=O)C=Cc2ccnn2C)C1 11040,c1(C(N2C(C(C)N)CCCC2)=O)ccc2c(c1)C(=O)OC2(C)C 11041,O=C1CCc2cc(C(N3CC(N4CCCC4=O)C3)=O)c(F)cc2N1 11042,c1(NC(COC)CCOC)nc2ccccc2nc1N1CCCC(C)(CO)C1 11043,c1(CNC(CCC2N(C)CCC2)=O)ncccc1C(N1CCCC2CC12)=O 11044,C1(C(N(CC(=C)C)CC)=O)CC=CCN1C(=O)Cc1csc(C)c1 11045,C12(NC(=O)Cc3sccc3Cl)CCC(CN(C(c3coc(Br)c3)=O)C1)C2 11046,c1(OC)nc(C)ncc1C(=O)NCC1CC2(CC2)CN1C(C1CCCS1(=O)=O)=O 11047,Cc1cc(C(=O)NCC(C2CCCC2)NC(c2ccccc2F)=O)c(O)nn1 11048,CC(C)C(C)(CNC(=O)CC1CCCC(C)O1)NC(=O)C1=CCCC1 11049,C1(C)(CNC(C2CCC(CC)O2)=O)CCCN1C(=O)CCc1ccccc1Cl 11050,C1(C2CN(C(C3CCC(=O)N(C(C)C)C3)=O)C2)(NC(CCN(C(C)=O)C)=O)CC1 11051,C1(COC)CC(O)CN1C(=O)C(C1CN(C(=O)C(C(C)C)NC(=O)OC)C1)SC 11052,c1(C(=O)NC(C#C)CC2CCOC2)ccc(-c2ccc(Br)cc2)n1C 11053,C(=O)(C1Cc2ccc(Cl)cc21)N1CC(OCCNC(C2CC3(C2)CC3(F)F)=O)C1 11054,C(c1ccc(Cl)cc1)=CC(=O)NCC1CC(OC)CN1C(=O)CCc1cnoc1 11055,Cc1nc(CCC(N2CCC(CCNC(c3ncoc3C3CC3)=O)C2)=O)cs1 11056,Cc1cc(Cl)c(Cl)cc1CNC(=O)COC1CCC(=O)NC1=O 11057,c1(N2CCC(C(C)NC(=O)COc3ccccc3)C2)cc(C(F)(F)F)nc(Cl)n1 11058,N1(CC=C(C)Cl)CC=CC1CF 11059,c1(OC)cc(C(=O)NC2(C)CCN(C(=O)C(C)NC=O)C2)cnc1O 11060,c1(C(=O)CNC(c2cccs2)=O)cc(Cl)ccc1OCC1CCCO1 11061,C1(C)(NC(C(CCN(C)C)NC(c2coc(CO)c2)=O)=O)CC2CCC1C2 11062,c1(C(N2C(CC#C)CCCC2)C(=O)NCC2(C#N)CCC2)ncc(C)cc1C 11063,C12(CNC(C(CNC(=O)COCC3CCOC3)N(C)C)=O)CC(C)(CCO1)C2 11064,N1(C(C(CC)=CC)=O)CCC(N=[N+]=[N-])(C(N2CC(n3cccn3)C2)=O)C1 11065,N(C1CCOc2c(F)cccc21)C(=O)Nc1ccc(S(=O)(=O)CF)cc1 11066,N1(C(c2c(C)[nH]nc2CO)=O)CCOC2(CCN(C(=O)C(C)NC(C)(C)C)C2)C1 11067,N1(C(CCCC#N)=O)CCN(C(C2CCCS2(=O)=O)=O)CC1CC1CC1 11068,C#CCC(C)(C(=O)N1CCN(C(C)C)C(=O)C1)NC(=O)CCCCCF 11069,C1(C(N(C2CCOCC2)C)=O)CC2C=CC1N(C(=O)CC(=O)OC(C)(C)C)C2 11070,CC1(C)C(NC(CC2(C(=O)OC)CCC2)=O)CC1CNC(C1CCOCC1)C1CC1 11071,c1(C(=O)NC2C(CNC(C(COC)N(C)C)=O)CC2)cnn2ccn(C)c12 11072,C1(C)(OC)CCN(C(c2cc(-c3c(Cl)cccc3Cl)on2)=O)CC1 11073,CCC(C(=O)NCC1(C(C)(C)O)CN(C(=O)CNS(N)(=O)=O)C1)NC1CC1 11074,N1(C(C(OC)OC)=O)CCC(CCC2CCCN2C(c2cnns2)=O)CC1 11075,n1(CC)nc(C(N2CCCC2CC(=O)NC2CCC(O)CC2)=O)c(C)n1 11076,C(=O)(C1=CCCSC1)NC1C(CNC(c2ccc(CNC(C)=O)cc2)=O)CCCC1 11077,C(=O)(CCC(=O)N(CC)CC)N1CC(OCC)(CO)C1.C1(CC(=O)N)CCCN1C 11078,N1(C(CC(CNC(=O)CSCCCN=[N+]=[N-])OC)=O)CCN(C)CC1C 11079,C(=O)(C#CC(C)(C)O)N1CCCC(NC(C(CC)(C)C)=O)C1 11080,C12(C(N3C(CC)CC(C)C3)=O)COCC1CN(C(C1CC1(C)C)=O)C2 11081,C(=O)(C(O)CC(C)C)NC1(CCNC(CNC(CCC(C)C)=O)=O)CCC1 11082,c1(NC(C2SCCN(C(c3cccc(OC)n3)=O)C2)=O)ccc2scnc2c1Br 11083,N1(C(C)=O)CCN(c2cccnc2C(N)=O)CC1(C)C 11084,C1(CNC(c2c(C)c(F)ccc2)=O)CCCCN(C(=O)Cc2n[nH]c(=N)s2)CC1 11085,C1(C(=O)NCC(C)OCC#C)C2CC3C(C2NC(C2(CO)CCOC2)=O)C13 11086,C1(C)(CNC(CCC(C)(C)F)=O)COCCN(C(c2ccncc2Cl)=O)C1 11087,N1(C(C2(C)CSC2)=O)CCC(C(C)(C)NC(c2ccc[nH]2)=O)CC1 11088,C(=O)(CN=S(C)(C)=O)N1C(CN(C)C(C2CC2c2ccncc2)=O)COCC1 11089,N1(C(c2cnc(COC)s2)=O)CC=CC(NC(C2C(C)C2C)=O)C1 11090,CCC(CO)CCNC(=O)CC1(C)CCN1C(=O)CC1CCC(=O)C1 11091,N1(C(C)CN2CCN(Cc3ccccn3)CC2)CCCC(C(=O)O)C1 11092,C1(CNC(c2c(C)cco2)=O)C(C2CC2)CCN1C(c1ncc[nH]c1=O)=O 11093,c1(CC)nnc(CC)s1.C1(C2COC2)C(=O)N1CC 11094,C=CCCCC(C(=O)NC(C=C)C(F)(F)F)NC(=O)CCNC(C)=O 11095,C1(CC(=O)N(C(C)C(=O)NC2C3CCCC23)CC)CCCC(C)O1 11096,c1(C(=O)NCC2CCC(NC(C3C(CCC)C3)=O)CC2)nccc2cccnc12 11097,C1(NC(C(CC)CC)=O)CCN(C(C2CC2C)=O)C(c2ccccc2)C1 11098,CC(C)(CNC(c1nn[nH]c1C(F)(F)F)=O)CNC(=O)C(c1cncnc1)O 11099,Cc1cc(C(N2CCOC(C(=O)Nc3cc(I)ccc3F)C2)=O)cc(C)n1 11100,C1(NC(C(=O)NC2CC(C)OC(C)C2)=O)CCCCC12CCCC2 11101,N1(C(c2cc(C(=O)OC)no2)=O)CCC(C(C)NC(=O)C=C2CCC2)CC1 11102,c1(C(N2CC(CC(C)NC(=O)CSC(C)(C)C)C2)=O)nc2c(s1)COCC2 11103,N1(C(c2cnn(CC)c2CC)C(=O)NCC)CC2(CC=CC2)C1C(C)C 11104,c1(SC(CNC(c2ccncc2CNC2CCCCC2)=O)CO)ccc(F)cc1 11105,N#CC1CCN(C(C2CCOC2CNC(C2CCCC2O)=O)=O)CC1 11106,c1(C(=O)NC2C3CN(C(C4CCCN(C(CC)=O)C4)=O)C2C3)cnc(F)c(C)c1 11107,N1(C(C(CC=C)C)=O)CC(NC(=O)Cc2ccoc2)CC(C)C1 11108,N1(CC)OCC(NC(C2C3CC3CN2C(c2ccccc2OC)=O)=O)C1=O 11109,c1(C(N2CCC3(NC(c4cc(C)c(C)[nH]4)=O)C(C2)C3)=O)nc2c(s1)CN(C)CC2 11110,C1(CNC(Cc2c(C)cccc2)=O)CC2(CO1)CN(C(c1c(C)n[nH]c1C)=O)C2 11111,C1(O)(C(C)NC(CSCC(C)=O)=O)CCN(C(=O)CCc2nc[nH]n2)CC1 11112,c1(CC(C=C)O)cn(CC(F)CCNC(=O)C(C)(C)OC2CCCC2)nn1 11113,C1(NC(CC2(C)CCOC2)=O)CCCCC1CC(N1CCC(n2ccnn2)C1)=O 11114,c1(C2C(CNCCNC(c3n(C(CC)C)ncc3)=O)C2)ccccc1Cl 11115,N1(C(c2cc(CC)[nH]n2)=O)CCC(CNC(=O)C(C)SC)C(C)C1 11116,c1(OC)ccc(Br)cc1CC(N1C(C(N2CC(F)CC2C(N)=O)=O)CC2CC12)=O 11117,N1(C(CC(C)N(C(C(C(=O)OCC)CC)=O)C)=O)CC2(C1)NC(=O)NC2=O 11118,c1(C2CC2NCC(=O)N(c2ccccn2)C(C)=O)cccc(F)c1 11119,N1(C(C=Cc2ncn(C)c2)=O)C2CCC1CN(C(c1cc(C3CC3)sn1)=O)CC2 11120,c1(OCCNC(C2N(C(CC#C)=O)CCCC2)=O)ccc(Br)c(Cl)c1 11121,CCC(C)CC(=O)NC1CC(CNC(=O)CSCc2ccc(Cl)s2)C1 11122,c1(CC)ncccc1C(N1CCC(CC(C)C)CC1)C(=O)NC(C)C(=O)NC 11123,N1(C(CCSC)=O)CCN(C(C23CCC(N=[N+]=[N-])C2C3)=O)C(C)C1C 11124,c1(C(=O)NCC(C)NC(c2ccccc2N(C)C)=O)cc(C#N)no1 11125,c1(OC)ccc(CC(=O)NCC2C=CCN2C(c2conc2C)=O)cn1 11126,c1(C(=O)NCC2(OC)CN(C(c3ncsc3C(F)(F)F)=O)C2)occ2c1CCC2 11127,C(=O)(C(C)C(C)(C)C)NCC1C(OCC)CN(C(=O)COc2cccc(F)n2)C1 11128,Cc1ccc(C(=O)O)c(-n2cc(-c3ccns3)nn2)c1.C12CCCN(C1)C2 11129,N1(C(c2c(C)n[nH]c2C)=O)CCN2C(=O)C(NC(=O)CC(C)(C)C)CC2C1 11130,c1(Cc2n(-c3c(C)cccc3)nc(-c3ccncc3)n2)cccc2cnccc12 11131,N1(C(C(CC)(CC)CO)=O)CCC2CCN(C(=O)CC3CC4(CCC4)C3)CC2C1 11132,C1(O)(C(C(=O)NOCCOCC2CCC2)NC(CN(C)C)=O)CCCCC1 11133,c1(C(N2CCC(C)N(C(c3ccco3)=O)CC2)=O)c(S(C)(=O)=O)cnn1C 11134,c1(O)cc(Cl)ccc1Cl.C1(C(=O)NC2CN(CC)C2)(NC(C(C)O)=O)CCOCC1 11135,c1(C(N2C(C)C(NC(=O)C(=O)N=S(C)(C)=O)CCC2)=O)cn2c(n1)C(C)CCC2 11136,N1(C(CCC=CC)=O)CCCCCC(NC(=O)C(C(C)O)N(C)C)C1 11137,Cc1ccc(CC(=O)N(CCCCCNC(C2(F)CCOC2)=O)C2CC2)cc1 11138,C1(CNC(CC(=C)C)=O)CN(C(c2ccc(C(C)C)nc2O)=O)CCCO1 11139,C1(CNC(c2cncc(OC)n2)=O)CCCN(C(=O)CN2CCCC2C)CC1 11140,c1(C(=O)NC23COC(CNC(C4(O)CCC4)=O)(C2)C3)cc([N+](=O)[O-])cnc1O 11141,C1(CC(=O)NC(C(C)(C)NC(c2cnc(CCCC)s2)=O)C)CC(=O)NC1=O 11142,N1(C(CCC(C)(C)NC(=O)Cn2cnnc2O)=O)CC2CC(C1)C2(C)C 11143,c1(OC)ccc(C)c(C(=O)NCC2(CCCNC(=O)C=C(C)C)CCCC2)n1 11144,O=S(=O)(c1cccc(F)c1)NCCO.C1(N)CC2(CCOCC2)C1 11145,c1(OC)cc(C(=O)NCC2CCC2NC(c2cc(Br)n(C)n2)=O)ccc1C 11146,c1(C(N2CCC(N(C(=O)CC3CCC(=O)N3C)C)C2)=O)ccc([N+](=O)[O-])c(Cl)c1 11147,c1(C(N2CCC(CC)C2C(=O)NCC2CC(C(C)C)C2)=O)ccc2n[nH]cc2c1 11148,c1(CNC(=O)NCCOCCNC2CC2C(=O)OC(C)(C)C)cccc(Cl)c1Cl.C 11149,c1(N2CC3CCN(C)C3C2)nc(=NCc2nccc(O)n2)[nH]c2ccsc12 11150,c1(C(N(C2C(O)CCN(C(c3nc(C)oc3C)=O)C2)C)=O)cccc2c1OCC2 11151,C(=O)(C(CC(N)=O)NC(C1C=CC1C(=O)OC)=O)NC(c1scc(C)n1)C 11152,Cn1cnn(CC(=O)NC2CCCC(NC(=O)CS(C)(=O)=O)C2)c1=O 11153,C1(c2scc(C)n2)COCCN1N1CCC(CCC(N)=O)CC1 11154,c1(C(N(C)CCN(C)C(C2(N(C)C)CCCSC2)=O)=O)coc2ccccc12 11155,c1(C(N)=O)cnn2ccc(NC(=O)CCn3c(O)nc4ccccc34)cc12 11156,c1(CC)cc(N(C)CC2(CNC(=O)C(C3CCOCC3)O)CC2)nc(CC)n1 11157,C1(C(N(CC(C2CC2)OC)C)=O)C2CCCC2CN1C(=O)Cn1ccccc1=O 11158,N1(CC)CC(NC(C2(NC(c3ncncc3Cl)=O)CC(O)C2)=O)CC1=O 11159,n1(CC(=O)NC2CC3CC2CN3C(c2ccoc2C2CC2)=O)nc(O)ccc1=O 11160,CCC(CNC(C1CC(=O)N(C2CC2C)C1)=O)(CC)c1ccccc1 11161,Cc1c(C(=O)N(CCC(=O)NC(CO)CCF)C2CC2)ccn1C 11162,c1(CC)cc(C(N2CCC(NC(=O)CN3CCC(C)(C)C3)C2C)=O)ccn1 11163,CCC(C(=O)N(C1(C(=O)NCC(F)Cl)CC1)C)C(C)C 11164,c1(CC(=O)NC(C(C)NC(c2c(CC)ocn2)=O)(C)C)ccc(F)c(Cl)c1F 11165,CC1(C)C(C)(C)C1(F)C(=O)NCC1CCCN(C(c2nnc(O)nc2O)=O)CC1 11166,c1(C(C)N(C(C2CC3CCC2CC3)C(=O)NCC2CC2)C)nc2ccccc2s1 11167,C(CCN(C)C(c1ccns1)=O)(C(C)(C)C)NC(c1cccc(COC)n1)=O 11168,Cn1nnc2cccc(C(=O)NCC3C=CCN3C(C3CCCO3)=O)c12 11169,c1(CCC)noc(CCC(=O)NC2CCN(C(=O)C=C(C)C(F)F)C2)n1 11170,C1(CNC(c2occ(C)c2)=O)CC(C)N(C(c2cn(C(C)C)cn2)=O)C1 11171,C(C)(CCC(C)(C)C)NC(c1nnnn1CC(F)F)C1CC(=C)C1 11172,CC(C)P(=O)(CC(=O)NCC1(C(C)(C)O)CN(C(=O)C(C)(C)F)C1)C(C)C 11173,C1(O)(CNC(CC2(N(C(CC3(OCC)CC3)=O)C)CC2)=O)CCCC1C 11174,CCCCC(CNC(=O)COC1CC1)NC(=O)C(C)Oc1cccc(C)c1 11175,CC(=O)C(C)CC(C)C(=O)N(C)CCNC(c1n[nH]c2c1CCC2)=O 11176,c1(C(N(C)C)=O)cccc(F)c1-c1cncc(NC(c2ccncc2F)=O)c1 11177,c1(C(N(C)CC2CC(F)CN2C(=O)C=C2CC2)=O)cccn2nnnc12 11178,c1(C(C)N(C)C(=O)N(C)CCC2CCCO2)cnn(C)c1 11179,Cn1nnc2ccc(C(N3CC(NC(c4ccc(=O)oc4)=O)C4(CC4)C3)=O)cc12 11180,N1(C(C2(SC)CCC2)=O)CCN(C(C2CCCCS2)=O)C(c2nccn2C)C1 11181,c1(C(=O)NCCC2(CNC(CN(S(C)(=O)=O)C)=O)CC2)nnc2ccccc2n1 11182,c1(OCC)cccc(C(=O)NC2(C)CCN(C(c3n[nH]c(C4CC4)n3)=O)C2)c1 11183,c1(C(C(=O)N(CCN(C(C(C)C2CCC2)=O)C)C)C)ccc(Cl)c(Cl)c1 11184,N1(C(C(C=C=C)C)=O)CC2CCN(C(c3nc4ncc(C)cn4n3)=O)C(C2)C1 11185,N1(C(CCC2(NC(COCCOC)=O)CCC2)=O)CCC(CO)C(C)(C)C1 11186,Cc1cccc(C(C(C)C)N(C(=O)Cn2cc(C(C)(C)S(C)(=O)=O)nn2)CCO)c1 11187,C(C(CCC(=O)O)CC(F)(F)F)NC(C(CC=C)F)=O 11188,N1(C(CC(COC)C)=O)CCCC(C)(NC(=O)CCCc2ccc(Cl)cc2)C1 11189,N1(C(C2CCC(C(=O)OC)C2)=O)CC2CC(C)N(C(c3ccsc3Cl)=O)C2C1 11190,c1(CC)cc(C(=O)NCC2(C(N3CC(O)C3)=O)CC(C)(C)C2)c(C)o1 11191,C1(C(=O)NCC2(F)CC(CNC(C3CCCO3)=O)C2)Cc2ccccc2S1 11192,CCC(C#N)C(=O)NC(CNC(c1cnn(C(C)C)c1C1CC1)=O)CC(C)C 11193,C(=O)(CCS(=O)(=O)C(F)(F)F)NCC1(F)CN(C(c2n(C)ncc2C2CC2)=O)C1 11194,CC1COCCC1NC(=O)C(C)N(C(=O)CC=C(Cl)Cl)C1CC1 11195,C1(NC(COCCCCC)=O)CN(C(c2cnc(CC)s2)=O)CCC1CO 11196,CC(C)CC(C(=O)N1CC(C(=O)NCCc2ncon2)CC(C)C1)C(N)=O 11197,CC(C)(C)C(CNC(=O)C(O)CC1CCOCC1)NC(=O)C=Cc1ccc[nH]1 11198,C(=O)(C(O)CCCNC(=O)C(C)c1cc[nH]n1)NCC(COC)(C)CO 11199,N1(Cc2cc(C)n(C)n2)CCC2(CCN(C(=O)C(O)CC(C)C)C2)C1 11200,N1(C(C2C(=C)C2)=O)CCC(CO)(CNC(=O)Cn2cccnc2=O)C1 11201,c1(NC(C2C3(CN(C(CC(CC)C)=O)C3)C2)=O)cc(F)c([N+](=O)[O-])cc1F 11202,c1(C(=O)NCC(CC)NC(C2(O)CCOC2)=O)ccsc1C(F)F 11203,c1(NC(N2CCCC(O)(c3ccc(Cl)cc3)C2)=O)ccc(S(=O)(=O)CC2CC2)cc1 11204,N1(C(Cc2c(C)ccnc2)=O)CC2CCC1C(NC(c1nc(C)n(C)n1)=O)C2 11205,C1(CNC(c2ncn(C(C)(C)C)n2)=O)CC2CCC1N2C(C1(C)CCC(=O)C1)=O 11206,C(=O)(C1CCCc2ncccc21)NCC(CN(C(c1c(C)onc1CO)=O)C)C 11207,c1(C2N(C(C3N(c4ccnc(OC)n4)CCCC3)=O)CCC2)ccc(Br)cc1F 11208,CC12CC(C1)C(=O)N2C(C1CCC1F)=O.c1(-c2cscn2)ccccc1.C 11209,C(N=c1cc[nH]cc1S(=O)(=O)NC(C)(C)C1CC1)c1cnc(CC)s1 11210,N1(C(C(C2CCCC2)NC(C2NC(=O)CC(C)C2)=O)=O)CCC2CCC(C1)N2C 11211,C1(C(=O)NCCC(C)N(C(C(C)OCC#C)=O)C)CC12CCOCC2 11212,CC(CN(C)C)CCC(=O)N1CCN(C(c2ncc(F)cc2F)=O)CC1 11213,N1(C(C(C)N(CCC)C(C2CCCCS2)=O)=O)CC2(COC(=O)C2)C1 11214,c1(NC(C)=O)ccc(C(=O)NC23CCN(C(=O)OC(C)(C)C)CC2C3)c(C)c1 11215,c1(C(N(CCNC(C2N(C(C)=O)CSC2)=O)C2CC2)=O)cnc(C2CC2)nc1C 11216,C1(C)(CNC(C(c2cccnc2)C)=O)CCCN1C(c1cccc[n+]1[O-])=O 11217,c1(C(=O)NCC(C)NC(=O)C(c2ccc(Cl)cc2Cl)O)nccc2[nH]ccc12 11218,c1(C(=O)NCC(C)NC(C(c2cc3ccccc3o2)C)=O)ccc2c(c1)CCO2 11219,C(=O)(CC(CNC(c1csc(F)c1)=O)OC)NC(c1ncc[nH]1)CC 11220,Cc1nc(N2CCC(C)C(NC(=O)Cn3nnnc3C3CC3)C2)cc(C#N)n1 11221,N1(C(C2(C)COC2)=O)CC(C(N2CCCCC2CCCO)=O)C(C)(C)C1 11222,C(=O)(CC1OCc2ccccc21)NCC1CN(C(C(CCOC)C)=O)C(C)C1 11223,Cn1c(=N)[nH]c2ccc(C(N3CCCC4(NC(=O)CCC(N)=O)CC4C3)=O)cc12 11224,C1(CC(=O)NC(CC)CSC)CCCN1C(c1csc(NC(=O)C2CC2)n1)=O 11225,c1(CC(c2c(C)c(Cl)sc2Cl)Nc2cc(Cl)ccc2Cl)cnc2cccnc2c1 11226,c1(C(N(CCCCNC(C2CC2C2CCCO2)=O)C)=O)ccncc1Br 11227,C1(NC(C(CSC)C)=O)CC2CN(C(c3cc(-c4ccncc4)on3)=O)CC12 11228,N1(C(C(Cc2cn[nH]c2)NC(c2cc(OC)no2)=O)=O)CCOCC1CC(C)C 11229,CC1(C2(C(N3CCC(CCC(=O)N4CC(C(F)(F)F)C4)C3)=O)CC2)CC1 11230,N1(C(C(C)(C)NC(=O)C(F)(F)F)=O)CC2CN(C(C3CC(=O)C3)=O)CC2C1 11231,C1(N=[N+]=[N-])(C(=O)NCC(CCC)OC)CCN(C(=O)CCCCC2CC2)C1 11232,N1(C(c2nc(C)nc(O)c2)=O)CC2CCN(C(c3cc(C(F)F)n(C)n3)=O)CC12 11233,c1(CNC(C2N(C(C(C)NC=O)=O)CC=C2)=O)cccc(C#N)n1 11234,C1(N(C)C)CCN(C(C2CCCCCN2C(=O)CCCn2ccnc2)=O)CC1O 11235,c1(C(N(C2CCN(C(=O)CSC(F)(F)F)C2)CC#C)=O)nccn1CC 11236,N1(C(=O)CCC2OCCO2)CCCC2C1CCN2C(=O)CC1CCC1 11237,C(CC(F)(F)Cn1cc(C)nn1)NC(C1(CCCC)CC1)=O.C(C)(CC)O 11238,N1(C(CC(C)(C)N(C)C(C2CC(=O)CC23CCC3)=O)=O)CCC2(CC=CCO2)C1 11239,N1(C(c2cncc(C)n2)=O)CCC2CN(C(c3nc(C4CC4)cs3)=O)CC2C1 11240,C1(C(=O)NCCCN(C(=O)CC2CCCCO2)C)(CC)CCOCC1 11241,c1(C(C(=O)N(C2CCN(C(C3CC=CCO3)=O)CC2)CC#C)C)ccccc1C 11242,S(=O)(=O)(c1cccs1)N(CCCO)C.C12CCN(CC1)C(=O)C(=O)NCC2 11243,N1(C(CC(=C)C)=O)CC(NC(=O)CCc2cc(Cl)no2)CC(C)C1 11244,c1(C(N2C3CN(C(C4C(CCC)C4)=O)C(C3)C2)=O)ccc(Br)c2cn[nH]c12 11245,c1(C(=O)NC(CC(N2C(C)CCC(C)C2)=O)CC2CC2)c[nH]c2nccc-2c1 11246,N1(C(C(C)=C(C)C)=O)CCC(NC(c2cc(C)cnc2Cl)=O)CC1C 11247,C1(CC(N2CCC(N(C(COCCOCCOC)=O)C)C2)=O)CCCS(=O)(=O)C1 11248,c1(NCc2c(N)ncc(Br)c2)ccc(S(=O)(=O)NC2CCC=CCC2)c(Br)c1 11249,Cc1cc(C)cc(C=CC(=O)NC(CNC(=O)CCC(C)(C)F)CC(C)C)c1 11250,CC(C)(CCCF)C(=O)NCc1ncc(C(=O)NOCC(F)(F)F)cn1 11251,N1(C(N(CCOC)Cc2ccco2)=O)CCN2CC(O)CC2C1 11252,N1(C(C(CC)NC(N)=O)=O)CC(C(F)(F)F)CC1CNC(=O)C(COC)CC 11253,N1(C(c2cnc(C)o2)=O)CC(NC(c2ccc(CC(C)(C)C)cc2)=O)CC1C 11254,C(=O)(CC(C)(O)COC)N(CCC(C)(C)NC(C=CC=CC)=O)C 11255,C1(C(=O)NC(C)CCF)CN(C(=O)CC#N)C2(CCC2)C1 11256,c1(OC)ncc(C=CC(N2CC(NC(C3CCCS3)=O)C3(CC3)C2)=O)cn1 11257,C(c1sc(Cl)nc1Cl)=CC(N1CCC(N(C(=O)Cc2cccnc2)C)C1)=O 11258,Cc1onc(Cl)c1C(=O)NC1CCN(C(c2ccc(C#N)s2)=O)C1 11259,C1(C(N2CCC(C(C)(C)NC(C(C)NS(C)(=O)=O)=O)CC2)=O)CCCCC1(F)F 11260,N1(C(CCc2cc(OC)c(Cl)cc2)=O)CCCC2(CCN(C(=O)CC3CC3)C2)C1 11261,CC1CC=C(C(=O)N2CCC(CN(C)C(c3cccc(O)c3F)=O)C2)CC1 11262,Cc1cc2nc[nH]c(=NCC(C(C)(C)C)NC(c3cc(O)nc(C)n3)=O)c2[nH]1 11263,C1(C(N(CCCCNC(c2c(C)ccc(Cl)c2)=O)C)=O)CCCC2CCCN12 11264,Cc1cc(NC(C2CC(NC(=O)Cc3cc(F)ccc3F)C2)=O)nc(Br)c1 11265,C1(CN(C(C(C)O)=O)C)CCCN(C(=O)C=CCN2CCC2)C1 11266,c1(CC(=O)NC2CN(C(C3CCN(CCO)C(=O)C3)=O)C2)ccc(O)c(Br)c1 11267,c1(CCC(=O)N(C(C)CNC(C2CCC2(C)C)=O)CC)cccc(C(F)(F)F)c1 11268,c1(NC2C(C(=O)Nc3c(OC)cc(F)c(F)c3)C2)ncnc2c(C)cccc12 11269,CC1=C(C(=O)N(CCCCCNC(=O)C(F)C2CCOC2)C)SCCO1 11270,N1(C(C2(O)CCCN(C(C)=O)C2)=O)CC2CN(C(c3c[nH]c(=O)cn3)=O)CC2C1 11271,c1(C(C)C)cc(C(N2CCN(C(C3(C)CC3Br)=O)CC2C)=O)nc2ncnn12 11272,Cc1cc(O)ccc1CNC(C12CC(NC(=O)OC(C)(C)C)C1C2)=O 11273,c1(C(=O)NCC23C(CN(C(C(CC)COC)=O)C2)CC3)cnc2[nH]cnc2c1 11274,C1(OC)CC(OC(C)(C)C)CN(C(C2CC(CC(F)F)C2)=O)C1 11275,CC(C)C(O)C(C)C(=O)N1CC(C(=O)NC2CC(C3CC3)C2)CCC1C 11276,N1(C(COCCC)=O)CC(N(C(=O)CNc2cccnc2)C)C(C)(C)C1 11277,C1(C)(CNC(C2(CC=C)CC=CC2)=O)CCCN(C(=O)CN2CCCCCC2)C1 11278,C#CCC(C)(CNC(=O)N(C)CCc1ccc(OC)cc1)CO.N1(CC)CCOCC1 11279,CC(CC(C)(C)C)C(=O)NCC12CCC(C1)N(C(C1(C(F)(F)F)CCC1)=O)C2 11280,N1(C(C(C)C2CC2)=O)CCCC(CN2CCN(C(C3(F)CC=CC3)=O)CC2)C1 11281,N1(C(C23C(NC(C(C)CO)=O)CC(CC2)C3)=O)CC2OCC(CO)C2C1 11282,C1(C(N2CCC(COC)(NC(=O)Cc3cncnc3)C2)=O)CC2C(C1)C2(F)F 11283,C(=O)(C(C(C)(C)C)OCC)N(CCCNC(C12CCCC1(C(N)=O)C2)=O)CC 11284,N1(CC(N2CCC(C3CCCN3C(C34CSCC3C4)=O)C2)=O)CCC(F)CC1 11285,c1(N2CC(C(C)C)OCC2)nc(NC2CC2C(F)(F)F)c2cnn(C)c2n1 11286,c1(CCC)ccc(CNC(c2nnnn2CC)c2ncco2)cc1 11287,C1(NC(c2c(CC)nc[nH]2)=O)(CC)CCN(C(c2ccoc2C2CC2)=O)CC1 11288,Cc1[nH]c(C(=O)NC(CCN(C(=O)C(N)=O)C)C(C)C)c(C)c1C 11289,CC1OC(C)C(C(=O)NC2(CCCCNC(=O)CC3CC(F)(F)C3)CC2)C1C 11290,c1(C(N2CCCC(N(C)C(c3ccsc3)=O)CC2)=O)cc(N)cc(O)c1F 11291,N1(C(C2C(COC)C2)=O)CCCC(CO)C1.C12CC(CO)N(C1)C(=O)OC2=O 11292,CC(C)C(CNC(=O)CSC(F)F)C(=O)NCCc1ccon1 11293,N1(C(c2cc(OC)n(C)n2)=O)CC(C)(C(N2CC3C4CCC(C4)C23)=O)CC1(C)C 11294,O=C(C#CC1CCCCO1)NC1CCC2CCN(C(=O)CCC3CC3)C1C2 11295,Cc1cn2c(n1)CCC(C(=O)NC1CC(CNC(c3ccc(C)s3)=O)C1)C2 11296,C1(N(C(=O)C=CC2CCC2)CCNC(c2cc(C3CC3)on2)=O)CCCCCC1 11297,N1(C(CC=CC)=O)CCC(N(C(=O)CCCNC(c2ccsc2)=O)C)CC1 11298,Cc1ccnc(CNC(C2COCCN(C(c3ccncc3)=O)C2)=O)c1F 11299,C1(C(N2CCN(C(=O)C=C3CCSCC3)C(C3CC3)C2)=O)CC2CCC(C1)C2 11300,c1(C(N(C)CCNC(c2ccsc2Br)=O)=O)ccc2sc(=N)[nH]c2c1 11301,N1(CC(=O)Nc2c(C(=O)NCCCC3CCCCC3)scc2)CCS(=O)(=O)CC1 11302,Cn1nc(C(F)F)nc1CNC(=O)Cn1cc(C(C)(C)C(=O)O)nn1 11303,C#CC1(C(=O)NCCC2(C)CCCC2)CCN(C(C2CCC(N(C)C)C2)=O)CC1 11304,CC1(C)CCCN(C(=O)C2=CCCOC2)C1C(N1CCNC(=O)C1)=O 11305,C(=O)(CCCCCCC=C)NCC1N(C(c2cc(C#C)cc(N)c2)=O)CCC1C 11306,C12(NC(c3ccc(OCC)cc3)=O)CCCC1CN(C(c1occc1F)=O)C2 11307,n1(C2CN(C(c3cn(C)c(C(=O)O)c3)=O)C2)cnc2ccccc12 11308,c1(C(N2C(C3(NC(CCC=C(C)C)=O)CC3)CCC2)=O)ncc(Cl)cc1O 11309,Cc1cc(CN=C(NC2CC23CCC3)NC2CC2)c(C)n1-c1ccc(F)cc1 11310,C=CC(C)(O)CC(=O)NCc1cc(C(=O)NC(C)COCCOC)no1 11311,C(=O)(C1CCc2snnc21)N1C(CNC(C(CC)OCC)=O)CCCC1 11312,C1(OC)CC2CCC1CC2C(=O)NC1CCC(C)N(C(C2CCC(C)O2)=O)C1 11313,C1(NC(C23CC(C)(C2)C3)=O)CCC2CC1CN2C(=O)Cc1ncncc1Cl 11314,C(C)(C)(CC(=O)N1CCCCC1C)N(C(C1C(C)C1C)=O)C1CC1 11315,c1(C(=O)NCCN(C(C)C)C(c2cc(Cl)cn2C)=O)nc2n(c1Cl)CCCC2 11316,N1(C(CC)=O)CCC(NC(C2CCCN(Cc3ccccc3)C2)=O)C12CC2 11317,N1(C(c2ncoc2COC)C(=O)NCC=C)CCOC2(CCCSC2)C1 11318,c1(N2C(C3(NC(c4ccoc4Br)=O)CC3)CCC2)ccc([N+](=O)[O-])cc1 11319,CC(C)CC(C)C(=O)NCC(C)NC(c1c(Br)cnn1C)=O 11320,C(C)(CCC(F)(F)F)(c1nnnn1C(C)(C)C)NCC(COC)(O)CO 11321,C1(NC(C=NOC)=O)C2CC3CN(C(=O)CCCCCF)C1C3C2 11322,CCC(CNC(c1cscc1C)=O)(CC)NC(c1ccc(-c2cscn2)cc1)=O 11323,N1(c2nccc(=NCc3n(C)cnc3)[nH]2)CCC2(COC(C)(C)C2)C1 11324,Cc1ccc(C2CCCCC2)n1CC(=O)NC(C1CN(CCN(C)C)C1)C 11325,CCCC(C(=O)NCC(C1CC1)NC(c1cn(C)cc1C)=O)C(C)C 11326,N1(C(CCC=CC(C)C)=O)CC2(CCCC2)C1 11327,CCC(COC)C(=O)NC(C)CC(C)NC(c1ccn(CC)n1)=O 11328,O=C(CCc1ccco1)NCCN(C(=O)Cc1nc[nH]n1)CC1CC1 11329,C(CCS(=O)(=O)N1CC(N2CCC(C(c3nc(C)on3)C3CC3)CC2)C1)N(C)C 11330,CCC(CC)C(=O)NCC(=O)NCCCC1(NC(=O)C(C)C(C)O)CC1 11331,CC1=C(C)CC(C)(C(N2CC(F)(CNC(C3CC4CCC(C3)S4)=O)C2)=O)CC1 11332,n1(CC(C(=O)NCCCNC(c2scc(C(C)=O)c2)=O)(C)O)c(C)cccc1=O 11333,Cc1ncc(F)c(N2CCC(C#N)(NC(c3n[nH]c(C)c3C)=O)C2)n1 11334,C1(NC(c2n[nH]cc2-c2ccccc2)=O)CC2(C1)CN(C(C1CCCCO1)=O)C2 11335,c1(C(=O)NC2CN(C(=O)C(F)(F)c3nccs3)CCC2F)cccc2nccn12 11336,N1(C(C(F)=CC)=O)CCCCC1CCNC(=O)C(C)(C)c1ccccn1 11337,c1(CC(=O)NCC(C)(C2CC2)NC(C(CCC)OC)=O)ccc2ocnc2c1 11338,CCC1c2ccsc2CCN1C(c1cc(F)ncc1F)C(=O)NC(C)(C)C 11339,C(C(C)C(C)C(=O)N(CC(C)NC(c1cc(O)ccc1N)=O)C)OC 11340,Cc1cc(CCC(=O)NC2CC(CCNC(=O)CCn3cnnn3)C2)cc(C)c1 11341,Cc1cc([N+](=O)[O-])cnc1C(N1CCC(C2(NC(c3csc(O)n3)=O)CC2)C1)=O 11342,CN1CCCC1C=CC(=O)NCCN(C(=O)C=Cc1cscn1)C1CC1 11343,c1(CCC(=O)N(C(CC)C)CC)ccc(OC)c(OC(=O)C(C)=CC(C)(C)C)c1 11344,C1(C(=O)NCC2(C)N(C(c3cccc(CC)n3)=O)CCC2)C(C)OC(C)C1C 11345,C(CO)(C(=O)NCc1cc(C(N2CCC(c3nc[nH]n3)C2)=O)co1)N(C)C 11346,c1(C(N(CC(CC)NC(CC(=C)I)=O)C)=O)n[nH]c(C)c1O 11347,Cc1cc(Cl)cnc1C(N1CC(O)(CCc2cn(C3CCCCC3)nn2)C1)=O 11348,Cc1cc(F)c(CC(N2CCN(c3ncccn3)C(=O)C2)=O)cc1F 11349,c1(N(C(C2CCC(CC)O2)=O)C)cc(F)ccc1SC 11350,CCC(CC(=O)NCCC1CC(C)C1)N(C)C(c1cnsc1C)=O 11351,c1(CNC(Cc2cn(CC)nn2)=O)ncccc1CNC(C1CNC(=O)C1)=O 11352,c1(OC)cc(CC(=O)NC2CCC2NC(=O)CCc2ncc[nH]2)cc(F)c1 11353,C=CC1OCCC1C(=O)NCCOC1CN(C(=O)CC(O)CN(C)C)C1 11354,C=CC(C)(C)CC(=O)NC1CCC(CNC(c2cc(C3CC3)ccc2F)=O)C1 11355,c1(NC(=O)NC(c2ccnn2C)C)cc(C(=O)O)c2n1CCOC2 11356,NS(=O)(=O)c1cc(C(=O)NC2CC(F)CN(C(C3CC=CCO3)=O)C2)ccc1F 11357,Cc1ccc(C(=O)NCCN(CC(C)O)C(c2coc(Br)c2)=O)o1 11358,c1(C2(CNC(=O)CCSC3CC3)CC2)cccc(Cl)c1.C12CC(F)(C1)CNC2=O 11359,C1(c2cn(Cc3ccc(C)o3)nn2)COCCN1C(=O)Cc1cn[nH]c1 11360,c1(OC)cc2[nH]ncc2cc1NC(=O)CC1CCN(C(c2cncnc2)=O)C1 11361,c1(NC(=O)OCC)ccc2c(c1)OCCO2.C12CCCC1C(=O)OC2 11362,Cc1cnccc1C(=O)NCC1CC2CC2N1C(c1cc(C)n(C(C)C)n1)=O 11363,c1(C(N2CC(O)(CNC(C3CC(O)C3)=O)C2)=O)ccc(Cn2cncn2)nc1 11364,N1(C(=O)CCC2CC2(F)F)CC(O)C(O)C1CNC(C1(C(N)=O)CCC1)=O 11365,C1(C(N2C(CNC(Cc3cccc(OC)n3)=O)C(C)CC2)=O)CC(=O)CC(=O)C1 11366,N1(C(C2CCC(=C)CC2)=O)CCC2CCN(C(=O)C(C)SC(C)C)CC2C1 11367,c1(C(N2CC(NC(c3ccc(CO)o3)=O)CC(C)C2)=O)cc2c(cn1)OCCO2 11368,c1(C(=O)N)nc(C)n(C)n1.c1(CC(CCc2cccnc2)NC(C)=O)ccccc1 11369,C(C#CC(F)(F)F)NC(C(C1CCN(C(=O)OC)C1)F)=O 11370,c1(NC2CCC(SCCCC=CC)C2)ccc(S(=O)(=O)N(C)C)cc1C#N 11371,c1(C(=O)NC2CCCN(C(C3C4CCCC34)=O)C2)ccc2c(c1)C=CS2(=O)=O 11372,c1(-n2cc(Cn3cnc(C(=O)OC)n3)nn2)cccc(OCc2ccccc2)c1 11373,Cn1c(C(N2CCOC(C3CN(C(=O)C=CCO)C3)C2)=O)cnc1O 11374,C(N=c1cc(C)nc[nH]1)C1CN(C(C(C(C)C)NC(COC)=O)=O)CC1(C)C 11375,C(CCC(C)C)(C(=O)N1CCC(O)C(C)C1)NC(CCN(CC)CC)=O 11376,c1(NC(C2CC(C)CN2Cc2cncc(O)c2)=O)ccc(C(N)=O)c(F)c1 11377,C1(C(N2CC(N(C(=O)CC(O)c3ccccc3)C)C2)=O)CC2COCC(C1)C2 11378,c1(C(=O)NCC(CO)NC(c2ccc(C3(C)CC3)cc2)=O)cccc([N+](=O)[O-])c1 11379,Cc1c(Cl)ccnc1C(N1CCC(CF)(NC(=O)CCc2ncc[nH]2)C1)=O 11380,c1(CNc2cc(C(C)(C)C#N)c(F)cc2)nc(O)c2ccccc2n1 11381,n1(CC(=O)NC(C)CCO)cc(C(N2CCOCC2)C2CC2)nn1 11382,Cn1nccc1C(N1CCC(c2ccccn2)C1)C(=O)NC1(C)CC1 11383,N1(C(=O)Nc2n(C)c(=O)on2)CCN2C(=O)COCC2C1 11384,C(N=c1[nH]cnc2cc(C)[nH]c12)C1CC(NC(=O)CN2CCCC2=O)C1 11385,N1(C(CNC(C(CC)C)C#N)=O)C2CCC1C(NC(=O)C(F)(F)F)C2 11386,c1(C(N(C2(CC(NOC3CCN(C)CC3)=O)CC2)C)=O)cccc2[nH]ncc12 11387,C12(C(N(CC(CN(C(C3CCN(C)C3=O)=O)C)O)C)=O)CCC(CC1)CO2 11388,C1(CC(=O)NCC(CO)OC)CN(C(c2snnc2C)=O)CC12CC2 11389,Cc1cc(C)c(C(N2CC3(CC3C(=O)NC(c3cncnc3)C)C2)=O)c(C)c1 11390,C1(NC(COCCCC)=O)C(C)CCN(C(=O)CCc2ccn(C)n2)C1C 11391,N1(C(C2(COC)CCCC2)=O)CCCC2(C1)CN(C(C1CN3CCN1CC3)=O)C2 11392,Fc1cccc2cccc(CNCc3cc(F)cnc3Cl)c12 11393,Cc1ccc(C(=O)NCC=CCNC(=O)C(=Cc2c[nH]cn2)F)cc1F 11394,C(C(C)C(=O)NCCN1CC(CF)C1)N(C(C1CC(O)(CC#C)C1)=O)C 11395,C(C(C)(COC)C(=O)N1CCC(NC(=O)C(O)C2CC2)C(CO)C1)OC 11396,N1(C(C2C(C(=O)OCC)C2)=O)Cc2ccnn2CC1C.C1(=O)CCCC(C)(C)N1 11397,Cn1cnc(CNC(C2(C3CCCN3C(=O)C=CC(c3cnn(C)c3)=O)CC2)=O)n1 11398,C1(CNC(C2(COC)CCCC2)=O)CC(C)(C)CN1C(=O)C1CC1 11399,c1(C(=O)NCC(CCCC)NC(=O)C2=CCCC2(C)C)ccc(Cl)c(C)c1N 11400,C(=O)(CCC(F)(F)c1ccc(Br)cc1)N(CC(C)(C)CO)C 11401,S(=O)(=O)(c1cccc(F)c1C)N1CCN(C2CN(C(C=COCC)=O)C2)CC1 11402,C1CCCCCC(=O)N1.c1(CNC(CN(CCC)C)=O)csnc1C 11403,C1(CNC(=O)COC2CCCNC2=O)CCNC2(CC2)C1 11404,CN1CCCC1CCC(=O)Nc1cc(C(=O)NOCC(O)CO)on1 11405,c1(C2(C(N(C3CN(C(=O)CCc4cn(C)cn4)C3)C)=O)CC2)ncccc1F 11406,C1(C(C)C(=O)N(C2(C(=O)NC(C)C(=O)NC3CC3)CC2)C)CCC(=O)N1 11407,c1(OC)ncc(Cl)cc1C(=O)NC1CCN(C(=O)C(C)C(F)F)C1 11408,C#Cc1cccc(NC(c2cccc(C)c2C)C)c1.c12ccccc1O2 11409,N1(C(C)=O)CCN(C(C2(F)CCN(C(C3CCCN3C)=O)C2)=O)CC1 11410,C#Cc1cc(COC(=O)Cc2ccc(C=O)[nH]2)cc(C(F)(F)F)c1 11411,c1(NC(c2ccoc2)=O)ccsc1C(=O)NCCF 11412,c1(OCC(=O)NCC(C2CC2)NC(Cc2c(C)ccnc2)=O)cc(Cl)ccc1C 11413,C=C(C)C1OCCC1C(N1CCC2(CC2NC(c2cccnn2)=O)C1)=O 11414,N1(C(c2cc(OC)ncc2)=O)CCC(C2CC2)(NC(=O)CC2CC23CC3)C1.C1CC1 11415,c1(OCC)ccccc1NC(=O)C(N1CCC(C)(NC(C2CCN2CC)=O)C1)=O 11416,N1(C(CC2N(C)CC=CC2)=O)CC2(CCCC2NC(c2ccc(=N)[nH]n2)=O)C1 11417,c1(NC(C2CCOCC2)COC)ccc(S(=O)(=O)N(C2(C)CCOC2)C)cc1F 11418,C(=O)(C(CC)C(=O)OC)NCCN(C(c1nccc(CC)c1)=O)C(C)C 11419,CC1=C(C(=O)NC(C)C(C)NC(c2cc3c(C)cccn3c2)=O)C(=O)OC1(C)C 11420,C1(C)(NC(C2(C(C)(C)OC)CC2)=O)CN(C(=O)Cc2cnc(C(C)C)o2)C1 11421,N1(C(COCc2c(C)ncs2)=O)CC2(NC(C3CCC(=O)N3)=O)CC1C2 11422,c1(C(C(=O)NCCC2(NC(C3CC34CCC4)=O)CC2)(F)F)ccccc1F 11423,c1(CNC2CC(CC(=O)NCc3cccc(C(=O)OC)c3)C2)c(I)ccnc1Cl 11424,C1(C(=O)NCC(C)(C)OC)CN(C(=O)C(O)CSC)CCC1(C)C 11425,N1(C(COCCCOC)=O)CCOCC1CNC(c1conc1C(C)C)=O 11426,C12(C(=O)NC(CC(=O)NC(C)C)C)CCC(CN(C(=O)C(CO)N(C)C)C1)C2 11427,N1(C(C=CCN(C)C)=O)CCOC(CNC(=O)C(C)(C)c2ccccc2)C1 11428,n1(CCN(C)C)cc(C(=O)NC2CC2NC(c2cn(CC(F)(F)F)nn2)=O)nn1 11429,C12(C(=O)OC)CCC1(C(=O)OC)CN(C(=O)COC1CN(C(C)=O)C1)C2 11430,c1(SCC)ccc(CC(=O)NC(C)Cn2cc(-c3cnn(C)c3)nn2)cc1 11431,CCC(C)CC(C(=O)NCc1cccnc1)NC(c1cc(C(C)=O)[nH]n1)=O 11432,N1(C(CNC(CNC(C2C(=C)C2C(=O)OC)=O)=O)=O)CCC(C(C)C#N)CC1 11433,N12CCCC3(C1)CN(C3)C(=O)C1C(C1)C2=O.c1(COC)ccnc(C(=O)OC)c1 11434,C(C)(C)(CCCC(=O)N1CC(CC(C)C)C1)NC(c1cc(COC)on1)=O 11435,CCC(C(F)(F)F)NC(=O)C(=O)N(C1CCC1O)C 11436,N#CC1CCCCCN1C(=O)NCCO 11437,n1(CC)ccc(C(N2CCCC2CCNC(C2CN(CC(C)C)C2)=O)=O)n1 11438,CC1CN(C(C2(C)CCCN2)=O)CCCN1C(c1cc(Cl)ccn1)=O 11439,C1(C(=O)NC2CC(CCNC(c3cc(-c4cccnc4)[nH]n3)=O)C2)CCC(F)C1 11440,C(=O)(C(C)(CC)CCC(C)C)NC(CN(C(c1ccc(F)cc1)=O)CC)C 11441,C1(C2(O)CCC2)(C(=O)NCC(c2ccccc2)NC(c2ccc(C#C)o2)=O)CC1 11442,Cc1cc(C(=O)NC2CCCC(NC(c3ccsn3)=O)C2)ncc1S(N)(=O)=O 11443,C1(CC)CC(C)CN1C(c1c(Br)ncn1C)C(=O)NCCOC 11444,N1(C(CCC(C)C)=O)CCC2(CC1)CCN(C(C13CCCCN1CCC3)=O)C2 11445,CC1(C)CCc2c1n[nH]c2C(N1CCC(NC(=O)CCC(N)=O)CC1C1CC1)=O 11446,N1(C(Cn2cc(C(=O)NC)nn2)=O)C2CCCC1CC(NC(C1CCOC1)=O)C2 11447,N1(C(C(C2CN(C(c3c(NC)nccc3)=O)C2)OC)=O)CC2CCC1C(CO)C2 11448,c1(C(N(C2CC2)CC2N(C(CCCCC)=O)CCC2)=O)cc2c(C)cccc2[nH]1 11449,Cc1nc(C#N)c(NCCC(=O)NCCN(C2CCCCCC2)C(=O)CCF)o1 11450,N1(C(C2(CC=C)CC2)=O)CCC(F)(C(=O)NC(c2nc(C)no2)CO)C1 11451,N1(C(C(CNC(c2cc(C(C)C)on2)=O)CC2CCCC2)=O)CCCCCC1C 11452,C1(NC(c2csc(C(F)F)c2)=O)CC(NC(c2ccc[nH]2)=O)C12CCC2 11453,c1(CC)cc(C(=O)N(CCn2cc(C(C)(C)N(C)C)nn2)CC)c(C)nn1 11454,CCC(CC)(CC(=O)OC)NC(c1ccc(Cl)cc1C(F)(F)F)C(=O)OC 11455,N1(C(C(=O)NCCC(C)(C)NC)=O)CCC(C2CCC2)CC1 11456,c1(C(N(c2ccc(Br)cc2)C(C)C)=O)cc(Br)c2[nH]c(=N)sc2c1 11457,N1(C(C(C(C)C)OCC)=O)CCC(O)(C(C)NC(=O)CCOCC(F)F)CC1 11458,C1(C(N(C2CCCN(C(c3ccc(C(N)=O)o3)=O)C2)CC)=O)CC(=O)N(O)C1 11459,C1(C(=O)NCC(CCC)NC(c2cnns2)=O)(CC)CCOCC1 11460,C(=O)(C1Cc2ccccc21)N(C)CC1N(C(CCC=C=C)=O)CCOC1 11461,C1(C(=O)NC(C)CF)CN(C(c2cncc(N(C)C)c2)=O)CCC1(F)F 11462,N1(C(c2ccc(C(=O)OC)cn2)C(=O)NCc2ccco2)CCC2CN(C)CC12 11463,C1(OC)CN(C(=O)C=CC2CCCC2)CC1NC(C1CCN1S(C)(=O)=O)=O 11464,c1(CN(C(C2CC(CCNC(=O)CCCc3ncco3)C2)=O)CC)cccnc1 11465,c1(C(N2C3(CNC(C=CCC)=O)CCC2CC3)=O)ccc(Br)c(F)c1C 11466,C#Cc1ccc(C(=O)NC2(C(=O)NCc3ncn(C)n3)CCSC2)cc1 11467,C1(COC)(CNC(c2nocc2C)=O)CCN(C(C2CCC(C)(C)C2)=O)C1 11468,C#Cc1ccc(C2CC2C(N2CCN(C(=O)C(C)CC(C)C)C(CC)C2)=O)cc1 11469,n1(CC(CC)CC)nc(-c2ccc(C(C)C)cc2)nc1C1CCC(=O)N1C1CC1 11470,C(=O)(C(F)C(C)(C)O)NCC(C)N(C(=O)CSCCC#N)CC 11471,C12(CNC(c3c(CC)nc(C)nc3)=O)CCCC(CN1C(=O)CS(C)(=O)=O)C2 11472,c1(C(=O)OC)sc(C(N2CC=CC(NC(C3(OC)CCCOC3)=O)C2)=O)cc1N 11473,Cc1cc(Br)cc(C)c1NNC(=O)Cc1ccnc(F)c1F 11474,c1(C(N(CCCCCNC(C(n2ncc(C)c2)C)=O)C)=O)cncc(C)c1O 11475,Cc1cccc(F)c1C(N1CCC(C)(CNC(=O)CC(F)(F)Cl)CC1)=O 11476,N1(C(CC(C)(C)O)=O)CCC(NC(=O)CCNC(=O)CO)C(F)C1 11477,C1(C(N(CCOC)CCNC(c2coc(CF)n2)=O)=O)CC2OC(C)(C)OC2C1 11478,N(C1CCc2cccnc21)C(C1C(C(C)(F)F)C1)=O.C1(c2ccoc2)C(=O)N1 11479,c1(CCNC(=O)CC2CCCC2O)cc(C(=O)Nc2csc(Cl)c2)no1 11480,S(=O)(=O)(c1ccc(N(C)CCC2CC2)cc1Br)N(C(C)CN)C 11481,C1(CCNC(=O)CO)(NC(CC2CN(C)C2)=O)CCCC1 11482,C1(CN(C(COCCCC)=O)C)CCCC(NC(=O)CS(N)(=O)=O)C1 11483,c1(C(=O)NCC(CN(C(c2c(CC)nc(C)o2)=O)C)O)cccc(F)c1C 11484,c1(OC)cc(C(=O)N(CCC(C)NC(=O)C(O)Cc2cn(C)cn2)C)[nH]n1 11485,c1(C(=O)NC2CCC3CC2CN3C(=O)C#CC2CC2)cc(O)nc2cnccc12 11486,CCCCC(CNC(c1n[nH]c(C)c1Cl)=O)NC(=O)CCCC1CCCC(=O)N1 11487,c1(OC(C(=O)NC2CC(NC(c3cc(CC)on3)=O)C2)(C)C)c(F)cccc1F 11488,C1(N2CCN(CCOC)CC2)COC2(CCN(C(C3CCCO3)=O)CC2)C1 11489,N1(C(C2(CCC=C)CC2)=O)CCC2(C=C(C(=O)N3CCOC(C)CC3)C2)C1 11490,c1(C2C(C(N3C(CNC(c4coc(O)n4)=O)CC3)=O)C2)ccccc1 11491,C1(NC(CC(CNC(c2ccnn2CCF)=O)O)=O)CCCCCCC1O 11492,c1(CC)nc(C)c(C(=O)NCCN(C(=O)C(C)C2CCC2)Cc2ccccc2)s1 11493,C1(CC)CC(C(=O)NC(CNC(=O)CC2CCOCC2)C(C)(C)C)CCO1 11494,Cc1ncc(C(N2CCCC(C(N3CCN(C)C(C(C)C)C3)=O)CC2)=O)c(=N)[nH]1 11495,N1(C(c2ccnc(OC)n2)=O)CCCC2C1CCCN2C(c1cc(C)n(C)c1)=O 11496,CCCC(CCC)C(C)NS(=O)(=O)Cc1ccc(F)cc1Cl 11497,N1(C(CN(C)C2CC2)=O)CCCC(O)(CNC(c2ccnnc2O)=O)C1 11498,c1(C(=O)NCC(C2CC2)SC)occc1CNC(C1CC1Cl)=O 11499,C1(C)(C(=O)NCC2C(C(N(CC(=O)NC(C)C)C)=O)CCO2)CCC(=O)CC1 11500,N1(CCC)CC(C(=O)NCCCCCCNC(c2ccsc2C)=O)CC1=O 11501,CC1CN(C(C2CC2C(F)F)=O)CC1NC(C1CCC(N2CCCC2=O)CC1)=O 11502,C(=O)(CC1=CCOCC1)NC1(n2cccn2)CCN(C(C(C)C)=O)CC1 11503,C(C)(CCCCNC(C1CCCC1(F)F)=O)NC(Cn1ccc(C(=O)OC)n1)=O 11504,N1(Cc2nccc(C)c2)CC(C(=O)Nc2ncc(C(N)=O)cc2Br)CC(F)C1 11505,CN1N=C(CC(=O)N2CCCCC(N(C)C(C3CC4(CCCO4)C3)=O)C2)CC1=O 11506,N1(C(c2cc(CC)ncc2)=O)CCCC(F)(C(=O)NCC(C)OCCOC)C1 11507,CC(C(C)(C)NC(c1cc(CO)[nH]n1)=O)NC(c1cnn(CC(F)(F)F)c1)=O 11508,C(CC1=CCN(C)CC1)NC(C(C1CCN(C(CSCCC(C)C)=O)C1)C)=O 11509,C1(CNC(CC2CCC(=O)NC2)=O)(NC(C2CCC2)=O)CC2CCC1CC2 11510,c1(C(=O)NC2C(C)N(C(=O)C(O)CCN(C)C)CC2)c[nH]c2cnccc12 11511,N1(C(c2c(C)scc2)=O)CC2CC2(NC(=O)CCc2cncc(O)c2)C1 11512,C1(N(C(C(C)OC)=O)C)CCC(CNC(=O)COCc2ccc(OC)nc2)CC1 11513,C12(C(N(C)CC3CCN(C(C4C(C)(C)OC4(C)C)=O)C3)=O)CCCC(C)(C1)OC2 11514,C1(O)(C(=O)NCC2C3CN(c4nccc(C(C)=O)n4)CC32)CCCC(C)(C)CC1 11515,O(NC(=O)CC1(CNC(=O)COC(C)C)CC1)CC(C)C 11516,Cc1cn2c(CC(=O)NC(C)C(C)(C)NC(C3CCCCC(=O)N3)=O)csc2n1 11517,C1(NC(c2ccc(Br)s2)=O)CN(C(C2C=CC=CC=C2)=O)CC12CC2 11518,c1(C(=O)NC2CCC(C(=O)Nc3cnccn3)CC2)cnc2ncccn12 11519,Cc1ccc2ccccc2c1NCC1CC(F)(F)C1 11520,C1(NC(C2CN(C(C)=O)C2)=O)CN(C(C2(C)CC2(C)C)=O)CC1c1ccnn1C 11521,c1(OC)cccc(CC(=O)OCCC2CSCCN2C(=O)CC2CCOC2)c1F 11522,c1(C(=O)Nc2c(C#N)nc(C)o2)n[nH]c2cc(C(=O)NC(C)C)ccc12 11523,Cc1ccnc(C)c1CNC(c1coc(CNC(C2CC(F)C2)=O)c1)=O 11524,C(C(C)CC(=O)NC1CC(NC(c2coc(-c3ccccc3C)n2)=O)C1)OC 11525,c1(C(C(=O)N(CCCC)C)=O)cccc(N)c1.C1(SC)CCCCC1CCC(C)C 11526,N1(C(C=CC=CCC)=O)CCC(C(F)CNC(C2CC2[N+](=O)[O-])=O)CC1 11527,c1(C(=O)NCC(CCCC)NC(=O)C(F)C2CCC2)cnc2c(C)cccc2c1 11528,N1(C(Cc2nc(C)c(C)[nH]2)=O)CCC2CCCC12CNC(c1ccc(F)s1)=O 11529,N1(S(=O)(=O)c2ccc(NCc3ccns3)nc2)C2CCC1c1ccccc12 11530,C1(F)(C(N(CCO)CC)=O)CCN(C(=O)C(C2(O)CCCC2)F)C1 11531,C(=O)(NNc1cc(Cl)nc(C2CC2)n1)NC(c1cc(Cl)nc(Cl)c1)C 11532,C1(NC(c2cc(Cl)c(Cl)cn2)=O)CC2(C1)CC(NC(C13CC(CO1)C3)=O)C2 11533,N1(c2cc(C)[nH]c(=NCCC3CCCN3)n2)CC2(C)CN(C)CC2(C)C1 11534,C1(CNC(c2c(C)nc[nH]2)=O)(NC(c2cnc(O)n2C)=O)CC(F)(F)C1 11535,C1(NC(c2cccc(OC(F)F)c2)=O)CCN(C(C23C=CC(CC2)C3)=O)CC1 11536,C1(C(=O)NCCN(C(=O)OC)C)COCCC1NC(c1ccccc1C)=O 11537,N1(C(C=CC)=O)C(CNC(=O)C(c2ccc(Br)cc2)OC)CC2CCCC12 11538,C#Cc1cc(F)c(C(=O)NC(C(C)NC(=O)CC(=O)NCC)C(C)C)cc1F 11539,C(=O)(C1CCCc2ncccc21)N(CCCCC(O)C1CCC1)C 11540,Cc1cncc(-n2cc(CONC(C3C(C)=NOC3C)=O)nn2)c1 11541,C(C(CC(=O)NCC1CCC1NC(c1cccc(=O)o1)=O)CC(C)C)NC(C)=O 11542,Cc1ccc(C(=O)NC2(CO)CCN(C(=O)C(C)(O)C3CCC3)C2)cc1Cl 11543,C1(NC(C(CC(=C)C)C)=O)(CNC(=O)CCC2CCC2)CC2CCC1CC2 11544,c1(OC)cc(C(=O)NCCCNC(=O)CSC(C)(C)C)c(F)cn1 11545,N1(Cc2nnc(CC)o2)CCCC(NC(=O)CCCOC(C)C)C1C 11546,C(C)(C(CC(=O)NCC1CC(CN=[N+]=[N-])C1)NC(=O)C(C)c1cc[nH]n1)OC 11547,C12(CNC(C34CC(C(C)(C)C)(C3)C4)=O)CC(CN1C(C1(C#N)CCOC1)=O)C2 11548,c1(NC(CN(C)Cc2cccc(F)c2)=O)nc(Cl)c(C#N)n1C 11549,CC1(C2(C)CC2C(=O)O)CC1.N12CCOCC1c1cn(nn1)CC(F)(F)CC2 11550,C12(NC(=O)CC=CCNC(=O)C(O)c3ccsc3)CC(CO)(C1)C2 11551,CC(C)(CCNC(C1CNC(=O)N1)=O)NC(=O)CCCc1ncco1 11552,c1(C(N2C(CNC(c3cnc[nH]3)=O)CCCC2)=O)cc2ccc(Cl)cc2c(=O)o1 11553,C1(CNC(=O)COCC2CCCCC2)CC2(CCC2)CN1C(=O)C1=COCCC1 11554,C(=O)(CCCCCN(C1CC2CC2C1)Cc1ccccc1)NC(C)(C)C 11555,c1(NCCc2n(C)c(Br)nn2)[nH]c(=NCC(Cl)(Cl)Cl)nc2c1cnn2C 11556,Cc1nn(C)c(C(=O)NCC(C)NC(C2CC2c2cnn(CCN(C)C)c2)=O)c1Cl 11557,N1(C(C(COCC)OC)=O)CCC(N(C(=O)COCC(C)C)C)CC1 11558,c1(OC)cnc(CNCCN(C2CCCC2)C(=O)C=Cc2ncc[nH]2)nc1 11559,c1(C(N2CC(NC(CCCOCCC)=O)C(OC)C2)=O)cc(=O)cc(Cl)[nH]1 11560,c1(OC)nccc(C(N2CCN(C(=O)C(Cl)(Cl)Cl)C(C(C)C)C2)=O)c1F 11561,CC(C)CC(C(=O)N1CCCC1CCc1ccccc1)NC=O 11562,c1(CC(C)C)c(C(=O)N(C2CCC(NC(C34CCC3CC4)=O)C2)C)cnn1C 11563,N1(C(C(C)SCC)=O)CCC2CN(C(c3cnc(C)o3)=O)CC2C1 11564,Cn1nc(Cl)cc1C(=O)NCC1(CNC(C2CC(F)C2)=O)CCCCC1 11565,C1(C)(NC(C(=Cc2ccco2)C)=O)CCCN(C(c2c(Cl)n[nH]c2C2CC2)=O)C1 11566,c1(C(=O)NCCC(C)NC(C2CCCC(=O)CC2)=O)c[nH]cc(Cl)c1=O 11567,Cc1ccc(C(C)(F)F)cc1C(N1CC(C)(NC(=O)C(c2ccnn2C)C)C1)=O 11568,CC1(C)CC(=O)OC1CNC(C1C=CCN(C(C2CCSCC2)=O)C1)=O 11569,C(CC(O)CC(=O)NC1C=CCN(C(=O)C(C(C)C)NC(N)=O)C1)SC 11570,C(=O)(C(CCCOC)NC(=O)CC(CN(C)C)CC)NCCc1ccn(CC)n1 11571,C1(C(=O)NC2C(O)CCN(C(CCNC(=O)NC)=O)C2)CC2CCCCCC12 11572,CCC(C(=O)NCC1(OC)CN(C(=O)CCc2cnc(O)[nH]2)C1)OC 11573,Cc1[nH]c(C(=O)NC(c2ccc(F)cc2F)C)c(C)c1C(=O)NCC1CCCO1 11574,N1(C(CC2(C)CC2)=O)CC(C)(C)OCC1CNC(=O)Cc1sccc1C(=O)CO 11575,N1(C(CC(CC)CC)=O)CCC2CN(C(=O)CC34CCC(CC3)C4)CC2CC1 11576,c1(CC)ncc(C(=O)NCC2CC(F)(F)CN2C(=O)CN2CC3CC3C2)c(O)n1 11577,N1(C(CNC2C(NC(C3C(C#N)C3)=O)CCO2)=O)CCCC2CCCCC12 11578,N1(C(c2ccc([Si](C)(C)C)s2)C(=O)NCCCC)CCC2(C1)NC(=O)N(C)C2=O 11579,c1(SC)ccc(CC(=O)NCCCC2CCN(C(C3CCC(=O)N3)=O)CC2)cc1 11580,C1(CC(N2CC(CCNC(c3[nH]c(C)nc3C)=O)(OC)C2)=O)CCCNC(=O)C1 11581,Nc1cc(Cl)nc(Cl)c1C(N1CC2(NC(=O)C=C3CCCC3)CCC1C2)=O 11582,Cc1ccc(C=CC(=O)NC(C2(O)CN(C(c3cnc(Cl)[nH]3)=O)C2)C)cc1Cl 11583,C1(O)(CNC(CC(CC)c2ccccc2)=O)CCN(C(c2ccc(=N)[nH]n2)=O)CC1 11584,C(=O)(C1CCc2ccccc21)N1CC2C(C(=O)NC(CC=C)C)(CCC2)C1 11585,C(=O)(CCCCN1CCOCC1)N(CCNC(C(CC)O)=O)C(C)C 11586,c1(CNC(c2nnnn2C2CCC2)C2(OC)CC2)cc(Cl)nc(Cl)c1 11587,C1(C(=O)Nc2c(CC)ncnc2CC)CCc2nncn2C1 11588,C1(CC=C)(C(=O)NC(C)CCC(=O)OC)CCN(C(=O)CSC(F)(F)F)C1 11589,N1(C(c2ccc(=NC)[nH]c2)=O)CCC2CC2(NC(c2c(CO)noc2C)=O)CC1 11590,CCC(CC)C(=O)NCC(C)NC(c1cnn(C(C)(C)C)c1C(F)(F)F)=O 11591,C(=O)(C1=C(Cl)CCCC1)NC1(C(N2CC(S(C)(=N)=O)C2)=O)C(C)(C)C1 11592,c1(C(=O)NC2CC(NC(c3c[nH]c(=NC)s3)=O)C2)cccc(S(=O)(=O)C(F)F)c1 11593,C1(C)(NC(C=CC(C)NC(COC)=O)=O)CCC(C)=C(C)C1 11594,O=C(CCC[N+](=O)[O-])NC1(CNC(=O)C(=O)Nc2ccccc2)CCCC1 11595,c1(C(C(=O)NCCCCCN(C(c2c(COC)nn[nH]2)=O)C)C)ccc(F)cc1 11596,C(CCCCCCCCCCCCC)NC(c1scc2c1OCCO2)CCC=C 11597,C=CC1CN(C(c2n[nH]c(C)c2C)=O)CC1NC(c1ncoc1C1CC1)=O 11598,c1(C(=O)NC2(CCCNC(C(C)n3cnnn3)=O)CC2)ccc(Br)nc1N 11599,N1(S(CC)(=O)=O)CCC(C(=O)NC(C)CCN(C(=O)CN(C)C(C)=O)C)CC1 11600,N#CC1(CC(N2CCCCCC2CNC(=O)C(F)n2cccn2)=O)CCOCC1 11601,CC1(C)CN(C(c2ccc(C#N)o2)=O)CC(CNC(C23COCC2C3)=O)O1 11602,C(CN(C)N1CCC(CCN2CCCC2)CC1)c1ccc(OC)cc1 11603,c1(C(N2CCC(C)(C(N3CCC(CF)CC3)=O)C2)=O)ccc(Br)cc1S(C)(=O)=O 11604,N1(C(c2cc(C(C)(C)C)no2)=O)C2CCC1C(NC(c1ccc[nH]1)=O)C2 11605,c1(CSCC(=O)NCC(C)CNC(=O)C(C)O)ccc(Cl)cc1Cl 11606,c1(CN(CC(=O)N(C(C)CNC(C2CCO2)=O)C)C)ccc(Cl)s1 11607,O=C1Nc2ccccc2CC1CC(N1CC2CC(CO)CC(C2)C1)=O 11608,C(=O)(C(F)C1=CCCCC1)N1CC(C)N(C(=O)C=Cc2cccn2C)CCC1 11609,CC(C)CCCCCC(=O)N1CCCC1CCNC(C12CCC1C2)=O 11610,C(=O)(CCCCCN(C)C)N(CC(=O)NC(C)CCO)C1CCC1 11611,c1(C(N2C(CNC(c3cn(CC)nc3)=O)CCC2)=O)cc(Cl)ccc1OC 11612,C(=O)(CC1=CCOCC1)NCCC(C)NC(c1ncc(OC)cn1)=O 11613,CCCCC(O)CC(=O)NCC1CN(C(=O)CNC(N)=O)CCCO1 11614,c1(C(=O)NC2C3CCN(C(CSCC#C)=O)C32)cnc2cc(C)nn2c1 11615,c1(C(=O)NC(C(C(C)C)NC(c2cc(CC)ncn2)=O)C)cnc(O)cc1C 11616,CC12CC(C(=O)NC3CN(C(c4ccc5cnnn5c4)=O)CC3F)(C1)C(C)(C)O2 11617,CCC(O)C(F)(F)C(=O)N(CC(C)(C)Nc1ncnc2[nH]ccc12)C 11618,C(=O)(C1CCc2c(Cl)cccc21)NC1CC(CCNC(c2cc(=N)[nH]cc2)=O)C1 11619,c1(C(N2CC(CNC(c3cncc(OCC)c3)=O)C2)=O)cc2c(Cl)cccc2s1 11620,CCC(C(=O)N(C1C2CN(C(=O)CN3CCN(C)C(=O)C3)CC12)C)C(C)(C)CC 11621,c1(OC)cccc(F)c1CC(N1CC(C)(NC(=O)CCCCCNC(C)=O)C1)=O 11622,N1(C(=O)NCC#CCN(C)C)CCC(C2CCCCC2)C1 11623,C1(c2onc(C)n2)CCC(C)N1C(=O)NCc1ccc(-c2nnco2)cc1 11624,N1(C(c2c(C)con2)=O)CC(NC(=O)C(C)(C)c2cscc2Cl)C(O)C1 11625,N1(C(=O)Nc2c(C)ncc(C)c2)CCC2(CC1)OC(C)(C)NC2=O 11626,C(=O)(CC(C)C(F)(F)F)N1CCC(CNC(CC(=C)Br)=O)C(O)C1 11627,c1(C(=O)NC(CC(C)Nc2ncnc(Cl)c2F)C)cc2ccoc2cc1F 11628,C(N=c1cc[nH]c(=NCCCc2cccc(C)n2)[nH]1)c1c(CC)nn[nH]1 11629,c1(OC)cc(C)cc(C(=O)NCCOCCNC(C2(S(N)(=O)=O)CCCC2)=O)c1O 11630,C(=O)(C1=C(Cl)CCCC1)NCC(C)(F)CNC(=O)COCC1CCCO1 11631,Cc1nc(C)c(C(=O)NC(C2CCCCC2)CNC(c2ccnc(Cl)c2)=O)[nH]1 11632,C1(NC(C(CO)OC)=O)CCOC(CNC(c2ccc(C(F)F)cc2)=O)C1 11633,C(CC1=CCN(C(C2CCCC23CCC3)=O)CC1)NC(C1CCC2CC2C1)=O 11634,N1(C(c2[nH]cc(CC(C)C)c2)=O)CC2(CCN(C(c3cc(=N)[nH]c(=N)[nH]3)=O)C2)C1 11635,N1(c2cc(N3CC(C(=C)C)OCC3)ncn2)C2CCC1CC(=O)NC2 11636,N1(C(c2cnn(C)c2C(C)(F)F)=O)CC2CN(C(=O)Cn3ccnn3)CC2C1 11637,Cc1sc(Cl)c(C(=O)N(CCCCN(C(=O)CN2CCCC2=O)C)C)c1C 11638,CCC(C)(C(=O)N(CCCCCNC(=O)C(CC#N)c1ccccc1)C)OC 11639,N(C1CCNc2ccc(Br)cc21)C(c1ccc(F)c(CO)c1)=O 11640,c1(CC(=O)NC2(CO)CCN(C(C=C3CCC(C)C3)=O)C2)cccc(Cl)c1F 11641,Cc1ccc(=N)[nH]c1C(=O)NCC(CO)NC(=O)CCn1cncn1 11642,C1(CC(C)C)CC(=O)N(C)CC(=O)N1.CCC1=NOC(CC(=O)OCC)C1 11643,C(=O)(CC(F)(F)C(C)C)NCC(CNC(C(COCC)C)=O)CO 11644,CP(C)(=O)c1cc(F)ccc1NC(=O)COCc1ccc2ccccc2c1 11645,c1(C(N(CCCN(C(CC2(COC)CCCC2)=O)C)C)=O)ccc(C)n(C)c1=O 11646,C(CCN=C(NC1CSC1(C)C)N1CCC(CC(C)C)CC1)SC 11647,C(=O)(C(C)C(=O)N1CCOCC1)NCc1onc(CC(=O)NC)n1 11648,CC(C)C(C(=O)N(CC(O)CN(C(=O)C(C)Cc1ccccc1)C)C)NC(N)=O 11649,C1(C(N(C2CCCN(C(c3csc(C)c3N)=O)CC2)C)=O)CCc2cnnn2C1 11650,c1(CC(=O)NC(C(C)C)Cn2cc(-c3ncoc3C3CC3)nn2)ccc(Br)cc1 11651,C1(C(=O)NC2C(CO)CCN(C(c3cnc(C)o3)=O)C2)CC2(CCCCC2)C1 11652,N1(C(Cc2ccc(C)o2)=O)CC2CC(NC(C3CC3CF)=O)CC(C2)C1 11653,c1(NC(=O)NC)cccc(C(=O)NCc2cc(Br)ncc2F)c1C 11654,N1(C(C2(C(=O)OC)CC2C)=O)CCC(NC(C2CCCC(F)C2)=O)C(F)C1 11655,N1(CCNC(C(C)(C)OC(C)C)=O)CCCN(C(=O)CC2CNC(=O)O2)CC1 11656,c12ccc(c(F)c1)OC(=O)CN2.c1(CC)ccc(C(C)(C)OC(F)F)cc1 11657,C1(CNC(C2(C(C)NC(=O)C=C3CCCCC3)CC2)=O)CC12CCOCC2 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11676,C1(O)(C(N(CCCN(C(C2CC(=C)C2)=O)C)C)=O)CCCC(C)(C)CC1 11677,N1(C(c2c(CC)noc2)=O)CC2(CCCC2NC(=O)C(c2ccccc2)C)C1 11678,CCCC(CC(=O)NCc1ccc(CO)o1)NC(c1c[nH]c(C#N)c1C)=O 11679,c1(C(N2CCN(C(C(CC)SC)=O)CC2CF)=O)coc2c(F)cccc12 11680,C=CCCC(C(=O)NC1(C)CC2CCC1C2)NC(=O)C(O)CC 11681,Cc1n[nH]c(C)c1CC(N1CC2C(NC(c3ccn(C)c3C)=O)C2C1)=O 11682,Cc1cc(F)ccc1C(c1ccccc1)NC1(C)CCOC1=O 11683,CN=c1nc(C(=O)N(C2CCN(C(=O)C(C)N(C)C)C2)C)cc(C)[nH]1 11684,Cc1ccn2nc(C(=O)OC3CCN(N4CCNCC4)CC3)nc2n1 11685,C(C(=O)NCCN(CCOC)C(c1cccc(C(F)(F)F)c1)=O)(C(C)C)SC 11686,N1(C(C2(CC)CCC2)=O)CC(C(=O)NOCCNC(=O)NC(C)C)C(O)C1.OCC 11687,C=CCC(CNC(c1cnc[nH]1)=O)NC(=O)CC1COCC1O 11688,N1(C(Cc2ccc(C)cc2C)=O)CC2CC(C)N(C(=O)C3=CCCC3C)C2C1 11689,C1(C(N2C(CC(=O)NCCC(C)OC)CCCC2)=O)CC(C)(C)CN1C 11690,C1(NC(Cc2cn(C(C)(C)C)nc2)=O)CC(NC(=O)C2=CCC2)C(O)C1 11691,C1(C(=O)NC(C)CC2CCCCC2)CCN(C(=O)CCC2CC2(C)C)C1 11692,Cc1ccc(OCCCNC(=O)NCCC2CCCS2(=O)=O)cc1C 11693,CN1CCOC2CN(C(C3CC(C)(NC(=O)CC4CCCOCC4)C3)=O)CC12 11694,c1(OCC)ccc(CNC(=O)NC(C)Cc2n[nH]c(=N)o2)cc1 11695,CCC(C)(C#N)C(=O)NCCCN(C(=O)CSCC(N)=O)CCO 11696,CC(CC(=O)N1CC(O)(C(C)NC(=O)C=CS(C)(=O)=O)C1)C(F)(F)F 11697,c1(C(C)C)ccc(N(CCC(=O)NCc2ccccc2)C(c2nc[nH]n2)=O)cc1 11698,C1(F)(C(=O)NC(CC(=O)NC)C)CCN(C(c2cscn2)=O)C1 11699,c1(C(=O)N(C2CCN(C(=O)CCF)CC2)C2C(C)C2)nn(C)c(NC(C)C)c1Cl 11700,C(=O)(C1CNC(=O)c2ccccc21)NCCN(C)Cc1ccc(F)c2ccccc12 11701,N1(C(C(C(C)(C)C)n2ccnn2)=O)CCCC(NC(=O)CCS(C)(=O)=O)CCC1 11702,N1(C(c2nocc2C)C(=O)NC(CC)C)CCC2(CCc3ccccc32)C1 11703,CCS(=O)c1ccccc1CC(=O)NCC(OC)OC 11704,C1(C2N(C(Cc3c(C)cc[nH]3)=O)CCC2)CCN(C(C2CC(F)(CF)C2)=O)CC1 11705,C1(COC)(CNC(C2(c3ccno3)CC2)=O)CN(C(C2CCO2)=O)C1 11706,c1(OC)cccc(CNC(=O)C(c2n[nH]c(C)c2Br)N(C)CC2CCSC2)c1 11707,N1(C(Cn2c(C)cc(C)n2)=O)CCC2C(C1)CN2C(C12CC(C)C1C2)=O 11708,N1(C(C(CC#C)(C)NC(=O)C(C2CCCCC2)C)=O)CCCC2OCCC2C1 11709,c1(C(=O)NCC2(C(N(CCC(C)C)C3CC3)=O)CC2)ccc2[nH]ccc2c1 11710,N1(CC(=C(Cl)c2ccccc2F)C)c2ccc(Cl)cc2NC(=O)C1C 11711,N1(C(C2(OC)CCN(C(C3CC4(CCC4O)C3)=O)C2)=O)CCOCC2(CC2)C1 11712,c1(SC)c(C(N2CCC(NC(C3CCC(C)(C)O3)=O)C2C)=O)cnn1C 11713,c1(CNC(C(C2(O)CCC2)NC(c2ccc(CO)s2)=O)=O)ccc(O)nc1 11714,CC1CC(O)CCN(C(=O)Nc2ccccc2CON2CCCCC2)C1 11715,C12(C(=O)NCC3(C)CCN(C(C(C=C)O)=O)C3)C3C4C1C1C2C3C41C(=O)OCC 11716,C1(NC(Cc2nc(C)sc2)=O)C2CC1N(C(C1(Sc3ccccc3)CC1)=O)C2C 11717,C1(C(=O)NCC(CNC(=O)C=Cc2cnc[nH]2)F)CC2(C1)CC1(CC1)C2 11718,C1(C(N(C2(C(=O)NCc3nc(CC)[nH]n3)CC2)C)=O)CCC(C2CC2)C1 11719,c1(NC(c2n(CC)nnn2)C23CCCC2C3)ccc(OC(C)C)cc1 11720,CC1(C)CC(NC(c2cccc(C(F)(F)F)c2)=O)CN1C(=O)CCN1CCCC1 11721,C(=O)(C(C)CC(C)(F)F)NC(CC(C)C)(C)CNC(=O)C(F)(F)c1cscn1 11722,CC1CCOC1CNC(=O)C(C1CCC1)NC(c1sccc1CO)=O 11723,c1(CC(=O)NC23CCC(CNC(C4CC(O)C4)=O)(C2)OC3)ccc2sccc2c1 11724,C(=O)(CCCCCO)NCC12N(C(C3C(OC)CCC3)=O)CC(C1)C2 11725,c1(C(N2C(C)C(C)N(C(c3ccc(Cl)cn3)=O)CC2)=O)ccc2nn[nH]c2c1O 11726,C12CCCC(C1)NC2=O.c1(C(N2CC(CC(C)(C)OCC)C2)=O)sccc1OC 11727,c1(OC)cc(C(N2CC3(C2)CN(C(=O)C(O)CC2CCCC2)C3)=O)c(F)cn1 11728,c1(-c2cn(CC(C)NC(C3CC(C)OC3=O)=O)nn2)ccc(N)c(Cl)c1 11729,C(CS(=O)(=O)CC(=O)N1CCC(C)N(C(c2n[nH]c(C)c2C)=O)CC1)OC 11730,c1(SC)cc(C(=O)NCCN(CC(C)O)C(c2ccn(CCOC)n2)=O)co1 11731,C1(C2CCC2)(C(=O)NCC(CN(C)C(c2ccn(C3CC3(F)F)n2)=O)O)CCC1 11732,C(=O)(CCCCN(C)C)NC(C)C(CO)NC(C1CC=CCC1)=O 11733,N1(C(C=CC(c2cccnc2)C)=O)CC2C(CNC(C3CN(C)CCO3)=O)C2C1 11734,N1(C(C(CC)OC)=O)CCCCC1C(C)(C)CNC(C1(N(C)C)CCOCC1)=O 11735,C1(=O)C(C(C)C)N(C)CCN1.C(COC)=CC 11736,C=C=CC(C)C(=O)N(C)CCC1CCCCN1C(c1n[nH]cc1Br)=O 11737,c1(C(N2C(CNC(C(CCN(C)C)O)=O)CCC2)=O)c[nH]c2cccnc2c1=O 11738,N1(C(c2cc(C)c(C)[nH]2)=O)CC(C2CCCCN(C(=O)Cc3ccccc3)C2)C1 11739,Cc1ccc2cc(C(=O)NC(C)Cc3cc(Br)ccc3F)cnc2c1 11740,CC(C)(C)CN(C(C1(CNC(=O)CC2CC=CC2)CC1)=O)C1CC1 11741,C(=O)(CCCC(=O)NCCC(O)CNC(=O)Cc1cncn1C)N(C)C 11742,N1(C(COCCC#C)=O)CCN(C(c2nnc(C)cc2O)=O)C2CCCCC2C1 11743,c1(CC)nc(=N)[nH]cc1C(N1CCCCCC1CNC(C1CNC(=O)N1C)=O)=O 11744,N1(C(c2c(CC)cncc2)=O)CCCC(C)(NC(=O)CC2COC(C)(C)C2)C1 11745,c1(CC(N2CC(NC(C3C(C(C)C)CCO3)=O)C2)=O)cc2ccccc2cc1O 11746,CC(C)CCCC(C)C(=O)N1CCC(CC(=O)NCCC2(CO)CC2)C1 11747,N1(C(CCSCC)=O)CCC(NC(C23CCC(CC2)CO3)=O)C(F)C1 11748,C1(CC(=O)NC(c2c(C)ncs2)C)CCN(C(c2n[nH]c(C)c2C)=O)C1(C)C 11749,C1(NC(c2csc(Cl)c2)=O)CCN(C(=O)Cc2cc(Cl)ccc2O)CC1O 11750,c1(CC)cccc(S(=O)(=O)N2CCN(C(c3cc(C)c(Br)s3)=O)C(CC)C2)c1 11751,c1(C(N2CCC(C)(NC(CC3C(C)CCCC3)=O)C2)=O)cc(F)cc2nc[nH]c12 11752,c1(OC)ncnc(C)c1C(=O)NCCCOCCNC(=O)C(C)(C)c1cscn1 11753,C12(C(=O)NC3COCCN(C(=O)CC4CSC4)C3)CC=CCN1CCC2 11754,C1(C(=O)NC2CC(NC(CCSCC)=O)CC2O)CCN(C(=O)C2CC2)CC1 11755,c1(C(CC2CC2)=O)cccc(CC(=O)OC(C(C)=CC)=O)c1 11756,C1(NC(C2C(C)(C)CCO2)=O)(CO)CCCN(C(C2CC(n3ccnn3)C2)=O)C1 11757,C1(C(=O)NC2CC(CNC(c3c(C)ncs3)=O)CC2O)CC12CCS(=O)(=O)CC2 11758,CC(C)CC(CO)NC(C1C(CO)CCN1C(=O)CC1(CSC2CC2)CC1)=O 11759,O(NC(=O)C(COCC)NC(=O)CCC1CCOCC1)CC(CC)C 11760,c1(C(=O)NC23CC(NC(c4cccnn4)=O)(C2)C3)ccc(=O)n2c1COCC2 11761,N1(C(CCN(C)C)=O)CC(C(=O)N(C2CCSC2)C)C(F)(F)C1 11762,Cc1ccc(C(=O)NCC(C)CC(=O)NC(c2ncccc2F)C)cc1O 11763,C(CC(=O)N1CCN(CCO)CC1)(C(F)(F)F)NC(CCC(C)(C)OC)=O 11764,CC(C(O)C(F)F)NC(C1(N(C(=O)CCOC2CCCC2)C2CC2)CCCC1)=O 11765,c1(C(N2CCN(C(C(CCC)=CCC)=O)C3C2C3)=O)ccc(S(N)(=O)=O)c(Cl)c1 11766,N1(C(CC(C)(C)OC)=O)CC2(CCC(CNC(=O)C(C)(C)c3cc[nH]n3)O2)C1 11767,C1(NC(C=C(C)Cl)=O)CN(C(c2c(C)ccn2C)=O)CC1O 11768,N1(C(CCC2(C#N)CCC2)=O)CC2(CCN2C(C2CC(C3CC3)=NO2)=O)C1 11769,N1(C(C(CC)C(=O)OC)=O)CC2(CCC(NC(C3CCCOCC3)=O)CC2)C1 11770,C1(NC(C(CO)NC(N)=O)=O)CCCN(Cc2ccccc2)C1 11771,CC1CN(CCS(C)(=O)=O)CCC1NC(C1CCCN1C)=O 11772,c1(C(=O)NCC2CCCN(c3nccc(CO)n3)C2)cnc(O)c(C(F)(F)F)c1 11773,C1(NC(COCCCC)=O)CCN(CCNC(=O)CN2CC3CC3C2)CC1 11774,C(=O)(C1=CCN(C(c2cc[nH]n2)=O)C1)NC(c1ncc[nH]1)C 11775,C(=O)(CC(C)(C)NC(C1(C(C)(F)F)CC1)=O)N(CC(COC)O)C 11776,C1(O)(CC(=O)NC(C)CNc2cc(O)nc(O)n2)CCCN(C)C1 11777,c1(CC(C)NCC=Cc2ccc(C(=O)OCC)o2)cc2cnccc2o1 11778,c1(CC)nn(C)c(C(N2CCSC(C(N3CCOC(SC)C3)=O)C2)=O)c1Cl 11779,C(=O)(CCC(=O)OC(C)(C)C)N(CC(CN(C(=O)CN1CC(=O)NC1=O)C)O)C 11780,C(=O)(C1=CCN(C(c2cnc(Cl)n2C)=O)C1)N1C(C)(C(C)C)CC1 11781,N1(C(c2ccc3c(n2)NCC3)=O)CCCC2CN(C(C3(F)CCC3)=O)CCC12 11782,N1(C(C(C)OC)=O)CC(CNC(=O)C(c2ccc(C)cc2)C)C2(CCC2)C1 11783,Cc1cc(C(N2CC(NC(=O)C(F)F)C(F)C2)=O)c(C)n1-c1ccc(Br)cc1 11784,C1(N(C(C(C=C)O)=O)C)CCC(CNC(=O)C(COC)N(C)C)CC1 11785,C(CCCc1cccs1)(c1ccccc1)NC(C(n1cc(C2(O)CC2)nn1)C)=O 11786,CCC(O)CC(=O)NC(C)(C(=O)N(C)CC1CCCC2CC12)C1CCC1 11787,CCC(C)(O)C(=O)NCC1(F)CCC(CNC(=O)C=C(C)Cl)C1 11788,c1(C(N2CC(CC(=O)N(CCCCCC)CC)(OC)C2)=O)ncn2c1CCC2 11789,CC1Cn2nccc2CN1C(=O)C1=CCN(C(C2(C)CCCC2O)=O)C1 11790,CCC(CC(=O)N(C1CCCCC1CC)C)N(C(=O)CN(C1CCC1)C)C 11791,C1(NC(c2cnc(O)s2)=O)CCN(C(=O)CC2CC2C2CC2)C1C1CC1 11792,c1(NC(N2C(CCNC(C3C4CCOCC34)=O)CCC2)=O)cnccc1CO 11793,c1(C(=O)OC)cnc(C)nc1N1CCC(NC(c2cnn(C)n2)=O)C(O)C1 11794,N1(C(C(C)(C)OC)=O)CC2(CCCN(C(=O)CC3CCCC(=O)C3)C2)C1 11795,c1(C(N2C3C(NC(c4c(C)cc(C)nc4)=O)C(C3)C2)=O)ccc2nc(S)[nH]c2c1 11796,c1(CC(=O)OC)cccc(CN2CC3CC3(C(N3CCC(C#N)C3)=O)C2)c1 11797,c1(CC)cc(F)ccc1C(=O)NC(C)C(C)NC(C1(C2CC2)CC1)=O 11798,c1(C(N(CC(CN(C(C2(CC=C)CCCC2)=O)C)O)C)=O)cnc(CO)nc1C 11799,CC1CCN(C(c2n[nH]cc2Cl)=O)C(CNC(c2cc(-c3ccco3)on2)=O)C1 11800,N1(C(c2c(C)nc(Cl)s2)=O)CCc2sc(C(=O)NCC3COC3)cc2C1 11801,N1(CC)CCC(C(=O)NC2CCCCC2CNC(c2cnsc2C)=O)CC1 11802,C(CN=C(NC(C)COC)NC1CC2(CC2)C1)OC 11803,C1(C(N(CC2=CCSC2)C)=O)C2CCC(C2)N1C(C1(C)CCC1)=O 11804,N1(C(c2cnn(CCC)c2C)=O)CCC2C(CCCN2C(=O)C(C)C(=O)OC)C1 11805,C(CNC(c1ccccc1N(C)C)=O)(C(C)C(C)C)NC(Cc1cnc(C)s1)=O 11806,c1(C(N(CCN(C(=O)Cc2noc3ccccc23)C)C)=O)nc2c(s1)COCC2 11807,C1(NC(C(C)(O)C2CCC2)=O)CC2(C1)CC2C(=O)NCC1=CCCOC1 11808,c1(C(N2CC(n3cc(CNC(CC)=O)nn3)C2)=O)cc(Cl)cn1C 11809,C(C(=O)NC(C)(C)C)(C(C)CC1CC(F)(F)C1)N(C1CCCC1)CC 11810,c1(C(=O)NC2C(NC(C(C)CN(C)C)=O)CCCC2)ccc2c(O)ncnc2c1 11811,CC1(C(=O)NCC2CC(O)(CNC(=O)CNC(C3CCC3)=O)C2)CCOCC1 11812,C#Cc1cncc(C(=O)NCCC(C)(C)NC(c2cncn(C)c2=O)=O)c1 11813,Cc1cc(C(N2CCOC(CC(=O)NC(c3ncccc3F)C)C2)=O)c(C)s1 11814,Cc1ncsc1CC(=O)NCC1CC1CNC(=O)Cn1cncc1C 11815,c1(C(=O)NC2CCCC(NC(c3ncc(C)c(Cl)c3)=O)C2)cc([N+](=O)[O-])cn1C 11816,n1(CC(=O)NC2C(NC(Cc3c(C)n[nH]c3)=O)COC2)nc(C)n(C)c1=O 11817,C(=O)(CCCCCC(C)(C)C)N1C(CN(C(C(CCOC)(C)C)=O)C)COCC1 11818,c1(NC(c2cnc3n2CCC3)c2n(CCCF)nnn2)cnc(OCF)c(Br)c1 11819,C1(NC(CSCC(=O)OCC(C)C)=O)CN(C(=O)CCOC(C)C)CCC1C 11820,N1(C(c2c(C)nc[nH]2)=O)CC2CC(NC(c3cc(N)ccn3)=O)C(C2)C1 11821,C1(C(=O)NCC2OCCN(C(C(CC)NC(N)=O)=O)C2)Cc2ccccc2N1C 11822,c1(CNC(=O)NC2(C(=O)O)C(C)C2)cc(Cl)cc(Br)c1 11823,N1(C(C2(CCNC(CCC(C)OC)=O)CCCC2)=O)CCSCC(C)C1 11824,N1(C(c2cc(C)nc(O)c2)=O)CC(CNC(c2nccnc2Cl)=O)OC(C)(C)C1 11825,N1(C(c2c(CC)ocn2)=O)CCCC2(C1)CN(C(c1c(C)noc1C(C)C)=O)C2 11826,Cc1nc(C(=O)NCC2C=CC(NC(=O)C(O)CC3CCOCC3)C2)sc1C 11827,N1(CCOC)CCOC2(CCN(C(C3CCC4CCCCN34)=O)CC2)C1 11828,Cc1ccccc1NC(C1COC(=O)C1)=O.N12CCOCC1CC(=O)NCC2=O 11829,N1(C(c2c(OC)cccn2)=O)CC23CCCC2(C1)CN(c1ncncc1Br)C3 11830,c1(CCS(N)(=O)=O)cccc(NC(=O)NCC2C3CCCCC23)c1 11831,CCCC(C)CCNC(c1nnnn1CCCF)c1cn[nH]c1 11832,N1(C(CCC=C)=O)CC(CC(=O)Nc2cnccc2CO)C(C)C1 11833,Cc1c(F)cc(C(N2CC(NC(c3ccc(CO)cc3)=O)C(C#N)C2)=O)cc1Br 11834,N1(C(C2(SC)CC2)=O)CCC(C2CCN(C(=O)CCC(C)C)C2)C1 11835,Cc1ccc(=O)n(CC(N2CC(NC(c3cc(C(C)(C)C)n[nH]3)=O)CC2C)=O)n1 11836,N1(C(CC=C(C)C)=O)CC(C2CCN(C(=O)CCOCC(C)C)CC2)C1 11837,CCCCCCC(F)C(=O)N(C1CCN(C(C2CC2(F)F)=O)C1)CC 11838,c1(NC(C2CN(C(=O)Cc3ncccn3)CCN2)=O)ncc(Br)cc1Br 11839,N1(C(c2cccc(COC)c2)=O)CC2CCCC2(Nc2nc(C)cc(C)n2)C1 11840,C#Cc1ccc(CC(=O)NCCC2(CNC(C3CC3C3CC3C)=O)CC2)cc1 11841,C(=O)(C1=CC2CCCC12)N1CC(N)C(C)C1.c1(C2(C(=O)OC)CC2)cc(C)ccc1C 11842,CC(C)CC(=O)C(=O)NCCOCC(N1CC(CO)C(F)(CO)C1)=O 11843,C(=O)(CS(=O)(=O)C(C)(C)C)N1CC(C(N)=O)(CNC(Cc2c(C)nc(C)s2)=O)C1 11844,Cc1c(C(=O)NC(CNC(C2(n3cc(Cl)cn3)CC2)=O)CO)ccn1C 11845,C1(C(N(CCN(C(CC2C(C)=NOC2=O)=O)C)C)=O)SC2C=CC1CC2 11846,n1(CC)nc(C(N2CC3CC3(NC(C3CCCC3(C)C)=O)C2)=O)cc1O 11847,CCC(c1cccc(Cl)c1)=CC(=O)NC1CCC(CNC(C2CNC(=O)N2)=O)C1 11848,C(=O)(C(CC(C)(C)C)NC(C1CC(=O)CCO1)=O)NC1CCC(C)(OC)CC1 11849,C(CN=c1nc2[nH][nH]cc-2c(O)n1)N(C(c1ccccc1S(C)=O)=O)CC 11850,C1(NC(COCCCOC)=O)CCCC2CN(C(=O)C(C)CS(C)(=O)=O)CC12 11851,N1(C(c2n[nH]c(CC)c2F)=O)CCCC2(CCCN(C(=O)CCOC)C2)C1 11852,C1(NC(c2c(CC)nn[nH]2)=O)CC=CCC1C(=O)NC(C(C)C)C1CC1 11853,C1(C(N2CCC(N(CC#C)C(C3COCCO3)=O)C2)=O)CCCCC1(C)C 11854,c1(C(CN(C2CC(CO)C2)C)O)ccc(Cl)cc1 11855,C#CC(C)(C)C(=O)NC(C1CN(C(=O)C=CCN(CC(F)(F)F)C)C1)C 11856,c1(C(C)(C)C)c[nH]c(C(=O)NC(CNC(=O)CC2CCCCO2)CO)c1 11857,c1(NC2(C)CC(NC(c3cnn(COC)c3C)=O)C2)cc(=O)n(C(C)C)c(O)n1 11858,N1(C(c2c(C)ncn2C)=O)CC2OCCN(C(C3CCN3C)=O)C2C1 11859,Cc1cc(CN2CCC(C)(NC(c3cc(C)n(C)n3)=O)C2)c(C)s1 11860,N1(C(C(C)NC(CC)=O)=O)C2CCC1CN(C(c1c(C)nc(C)n1O)=O)C2 11861,Cn1cc(Br)cc1C(=O)NCCC1CN(C(c2cncnc2C2CC2)=O)C1 11862,c1(C(=O)NCCN(CC(C)O)C(=O)C=CC2CC2)ncoc1C1CC1 11863,c1(C(=O)NCCN(c2[nH]cnc3nc(Cl)cc2-3)CCC)cc(F)cc2nn[nH]c12 11864,C1(CC(=O)NC(C(=O)OCCC)C)CC(C)N(C(=O)CC2CCCC(=O)C2)C1 11865,Cc1cc(F)cnc1C(N1CCCC1CN(C)C(C1(C(F)(F)F)CCC1)=O)=O 11866,N1(CCNC(C2C=CCC2)=O)CCCN(C(=O)Cc2csc(C3CC3)n2)CC1 11867,N1(C(=O)C2=CCCO2)CC2CCCN(C(C3C=CCCC3)=O)C2C1 11868,N1(C(C2(C)CCN(Cc3c(OC)ccc(Cl)c3)CC2)=O)CCCC(S(C)(=O)=O)C1 11869,c1(CCC(N2CCCC(n3cc(COC(=N)O)nn3)C2)=O)ncc(Br)cn1 11870,C(=O)(C1=CCCC1C)N(C(C(=O)NCc1cc(COC)n[nH]1)C)C1CC1 11871,N1(C(C(CCCC)(C)F)=O)CCC2(CCN(C(c3c(C#N)cnn3C)=O)CC2)C1 11872,c1(C(=O)NCC2N(C(CC3C(CC)C3)=O)CC2)cccc(Br)c1N 11873,C1(N(C(CC2(COC)CC2)=O)C)CCCN(C(c2c(C)ccn2C)=O)C1 11874,N1(C(C(=O)N(C)C)=O)CCC2CCN(C(c3coc4ccccc34)=O)CC12 11875,CCC(C)(CNC(=O)C(C)CN(C(=O)Cc1csc(C)n1)C)OC 11876,N1(C(C2CCN(C(C)=O)CC2)=O)Cc2[nH][nH]c(=NC(=O)C3CC3F)c2C1 11877,C(=O)(C(F)(F)C(O)c1ccccc1)NCC(C)NC(=O)CSC1CC1 11878,C1(C(N2C(CC)C(NC(=O)CN(CC)CC)CC2)=O)CC2(CC(OC)C2)C1 11879,C(=O)(C1=C(F)CN(C(C2CC(n3ccnn3)C2)=O)CC1)N(C1CC2CC2C1)C 11880,N1(C(c2cc(C)[nH]n2)=O)CC2(NC(=O)CN3CCCS3(=O)=O)CCC1C2 11881,CC(Cc1ccc(Cl)cc1)CC(=O)N1CCC1CNC(C1CSC1)=O 11882,Cc1ccc(NC(=O)CSCC(N2CCC3C(CC2)C3(F)F)=O)c2ccccc12 11883,N1(C(C2(C#C)CC2)=O)CC(NC(c2coc(C)n2)=O)CCC(O)C1 11884,c1(C(CNC(CC2(C)CN(C(C3CNC(=O)C3)=O)C2)=O)=O)ccc(Cl)cc1 11885,N1(C(=O)C(C2CCOCC2)O)CC2CCCC2(Nc2cc(Cl)ncn2)C1 11886,C1(F)(C(=O)NC(C(=O)O)C2CCCC2)CN(C(=O)OC(C)(C)C)CC1C1CC1 11887,CC1COc2c(C(N3CCC34CN(C(=O)COCC3CC3)C4)=O)cccc21 11888,C(=O)(CC(=O)N(CC(C)C(=O)NCCCC(=O)NC)C)OCC 11889,C12(CNC(C(C)OCc3ccncc3)=O)CCCCC1N(C(=O)C(C)O)CC2 11890,N1(C(C(CC)C(F)(F)F)=O)CCC(C2CCN(C(=O)CCn3cnnn3)CC2)C1 11891,c1(CN(c2nnc(N3CCN(C(C)(C)C)CC(C)C3)n2C)CC)ccc(F)cc1Cl 11892,CC1(C)CC(CNC(=O)C(F)=CC2CC2)CN(C(=O)CN2CC3CC3C2)C1 11893,Cc1ccncc1C(=O)NCc1cn(CCNC(=O)Cc2ccns2)nn1 11894,C=CC(CC)CC(=O)N1CCN(CCCNC(C2(S(C)(=O)=O)CC2)=O)CC1 11895,N(C(=NCCCF)N1CCCC(S(C)(=O)=O)C1)C1(c2c(C)nccn2)CC1 11896,c1(NC(=O)CCc2ccc(C(N3CCSCC3)=O)[nH]2)cc(Br)cc(I)c1 11897,C1(CCNC(CC2(C)OCCO2)=O)CCCN(C(c2cnc(Cl)s2)=O)CC1 11898,c1(C(C(=O)NCC2CCC(NC(=O)Cc3cnns3)C2)(F)F)ccc(F)cc1F 11899,C=CCC(CC)C(=O)NCC(=O)OC.C12(CCN(C)C1)C(=O)N2C 11900,Cc1cncc(C(N2CC(NC(c3cc(-c4cnn(C)c4)[nH]n3)=O)C(F)C2)=O)n1 11901,c1(C(=O)NC2C(C)CN(C(c3cccn(C)c3=O)=O)C2)cccc2c1CCCC2 11902,c1(C(N2CCCC(CCNC(C(CC)CO)=O)C2)=O)ccc2nonc2c1 11903,C1(CNC(CC(=O)NCC)=O)CCN(C(=O)CN(c2ccnc(Cl)n2)C)CC1 11904,c1(CNC(c2cn(C(C(=O)NCC(=O)NC)C)nn2)C)ccc(C(F)(F)F)cc1 11905,N1(C(C(C2CCCO2)NC(=O)CC2CCCC23CC3)=O)CCS(=O)(=O)CC1 11906,C1(C(=O)NCC2CCN(C(C3CCO3)=O)CC2(F)F)CCC2(CCCC2)CC1 11907,N1(C(CCCC#CC)=O)CCC2(CCC2NC(=O)CCc2nncn2C)CC1 11908,n1(CC)c(N(C(C)C2CC2)Cc2cccc(CO)c2)nnc1-c1ncc[nH]1 11909,C1(CNC(C(C)NC(N)=O)=O)CCN(CC2(C#N)CCC2)C1 11910,N1(C(COCCCC#C)=O)CCC(C2N(C(=O)C=C(C)C)CC2(C)C)CC1 11911,C(=O)(C1=C(C)CCCC1)NCC12N(C(C(CCCC)O)=O)C(CC1)CC2 11912,C(=O)(C=CS(F)(F)(F)(F)F)N1CCN(C)CC(CC(=O)O)C1 11913,c1(CNC(COCC(=C)C)=O)ocnc1C(=O)NC(C)Cc1cccnc1 11914,N1(CCC)CCc2cc(C(C)NC(C)CSC)ccc21.ON 11915,C1(NC(C2C(CC)C2)=O)CCN(C(c2cc(F)ccc2F)=O)C1(C)C 11916,CCCC(C(=O)NCCN1CCC(NC(=O)C2=CCCC2)CC1)S(N)(=O)=O 11917,CC1OC2CCC1(C(=O)NCC(C1CCCC1)NC(c1cc(Cl)cs1)=O)C2 11918,c1(OC)ccc(C(=O)NCC(C(C)(C)C)NC(c2ccsc2)=O)cc1C(F)F 11919,C1(C#N)(C(=O)NCC(C2CCCC2)NC(C(C2CCOCC2)C)=O)CC=CC1 11920,C(=O)(CCCCCC(C)(C)C)NCC(CNC(CN1CC(CC)C1)=O)O 11921,C#CCCCC(=O)NCc1ccc(N2CCN(C(=O)CSCCC)CC2)cc1 11922,C1(C(N2C(C(C)(C)NC(=O)CC3CCCC(O)C3)CCC2)=O)CC(S(C)(=O)=O)C1 11923,C12(C(=O)NCC3C(C(=O)NCc4nc(C(F)(F)F)cs4)CCC3)CCCN(CC1)C2 11924,N1(C(=O)CC2CCCO2)CCN(C(c2cnc(O)o2)=O)C(c2ccccn2)C1 11925,C1(CNC(C2N(CC)CC2)=O)CN(C(=O)Cn2cc(CC3CC3)nn2)CCCO1 11926,c1(OCC=C)ccc(CCNC2CC(=O)N(c3ccccc3Cl)C2)cc1 11927,C1(C(=O)NC2C3CN(C(=O)CN4CCCC4)CC23)CCc2ncc(Br)n2C1 11928,C#CC(CSc1cc(COC)nc(C)n1)CC(C)(C)C 11929,C1(C(=O)NCC(C(C)C)NC(c2c(C)snc2)=O)CCCN(C(=O)C2CC2)C1 11930,C1(O)(CNC(COCC)=O)CCN(C(=O)C=C2CCCCC2)C1 11931,c1(OCC)cc(C(=O)NC(C)C=CC(=O)N(CCCOC(C)C)C)[nH]n1 11932,c1(OCC(=O)NCC2(CNC(C3N(N=O)CCC3)=O)CC2)ccccc1[N+](=O)[O-] 11933,c1(N2CC(O)(CCNC(C=COCC)=O)C2)ncc2cccnc2n1 11934,N1(C(C2CCC(C)C2)C(=O)NCc2ccccc2)CC2C(=O)NC(=O)C2C1 11935,C1(NC(C2ON=C(CC)C2)=O)CC2CCCC(C1)N2C(c1nonc1CC)=O 11936,c1(C(N2CCC(CC=C)(NC(C3COC(C)C3)=O)C2)=O)cc([N+](=O)[O-])cnc1O 11937,N1(C(c2c(CC)noc2)=O)CCC2(CC1)CN(C(=O)NCc1ncc[nH]1)CCO2 11938,N1(C(COC)=O)Cc2ccccc2CC1NCC(C)(C)CNC(=O)C(=O)N(C)C 11939,C1(CNC(C=CCCC)=O)C2CN(C(c3ccc(I)cn3)=O)CC12 11940,c1(COC(c2cc(Nc3ccc(F)cc3)on2)=O)ccccc1C(F)(F)F 11941,N1(C(C=COCC)=O)CCCC(CN(C(=O)CCCCN2CCCCC2)C)C1 11942,c1(-c2cn(CC(=O)N(CCC)C(C)C)nn2)ccc(C(=O)NC(C)C)nc1 11943,c1(COC(c2sc(OC)c(Br)c2)=O)c(F)cc(F)c(O)c1F 11944,c1(C(=O)NC2CCN(C(C3CCN(C4COC4)C3)=O)C2)ccc2c(c1)NCC2 11945,N1(C(CCCCC=C)=O)Cc2ccnn2CC(NC(c2ccsc2)=O)C1 11946,N(C1CCc2cc(Br)ccc21)C(=O)Cn1cc(COc2cccc(CO)c2)nn1 11947,Cc1ccc(C)c(C(=O)NC2CCN(C(=O)CSc3ccccn3)CC2F)c1C 11948,c1(-c2nc(C(CC)CC)n(-c3cnnn3C)n2)ccc2ncccc2c1 11949,c1(OC)ccc2c(C(=O)NC(C3CCCCN3C(c3ccns3)=O)C)n[nH]c2c1 11950,CCC(CC)C(=O)NCCCCC(C)NC(=O)C(C1CC1)Oc1ccccc1Cl 11951,C1(NC(=O)CC2CCCCCO2)CC2CCC(C1)N2C(C1(CC(F)(F)F)CC1)=O 11952,O(N1CCC(c2nc(COC(=O)OC(C)(C)C)nn2-c2cccnc2)CC1)CC 11953,c1(CN=C(NCC(CCCC)CO)NC(C)C2CC2)ccc(S(=O)(=O)N(C)C)cc1 11954,CC1(C)CC(C(=O)NC2(c3cc[nH]n3)CC2)(CO)C1.C1(C=O)CCC(F)(F)C1 11955,c1(OCCCC(C)NC(C(N2C(C(=O)OC)C(C)CC2)=O)=O)ncc(Cl)cc1Cl 11956,CC1Oc2c(F)cccc2C1NC(=O)C(N1CCCC(O)(C(N)=O)C1)=O 11957,CC1(C)CC(C(N2CC(Cc3ccco3)C2)=O)N(C(=O)CC2CCC=CCC2)C1 11958,C(CCC(=O)NCC1(C(N2CC(CC)C2)=O)CC=CC1)=CCC=C 11959,C1(NC(CN(C(C2CC(C(N)=O)C2)=O)C2CC2)=O)CCn2nnnc2C1 11960,CC(C)CC(F)C(=O)N1CC(CNC(c2csc3nnsc23)=O)C1 11961,c1(C(N(CC)CC2CCN(C(C3CNC(=O)N3)=O)CC2)=O)cc2n(n1)CCO2 11962,c1(SC2C(C(=O)NCC(C3CCCCC3)NC(C)=O)C2)ccccc1 11963,CCCCC(C(=O)NCC1(O)CCN(C(=O)Cc2cnccc2Cl)CC1)C(C)C 11964,C(=O)(C(C)(C)C1=CCN(C(=O)C(C2CC2)C2CC2)C1)NCC(C(CC)C)CO 11965,n1(CC(=O)NCC(C)(CNC(=O)CCOC2CCC2)OC)nc(C)nc1C 11966,O=C(C1=CC2(CCOC2)C1)NCC1CCN(C(c2cc(=O)cc[nH]2)=O)C12CC2 11967,c1(N(C)Cc2ncccn2)nc(N2CCCC(CC(F)F)C2)nc2c1ncn2C 11968,c1(-c2cncc(Sc3ccc(F)c(C)c3Cl)c2)ccc2c3c(cccc13)C(=O)N2 11969,O=S(=O)(c1cc(Br)cc(Br)c1)N1CCn2cccc2C1CO 11970,c1(C(=O)NCCC2(O)CN(C(C(CC#C)C)=O)C2)cc(NC(C)=O)cc(Cl)c1 11971,C1(C(=O)NC(c2ccc(C)cc2)CC)Cc2cccc(C)c2O1 11972,C1(NC(C)=O)CCC(NC(=O)C(C)NC(C2CCC2)=O)CC1.C12(CCC1)C(=O)N2 11973,c1(NC(=O)Nc2cn(C(C)(C)C)cn2)cc(C(F)(F)F)ccc1O.C12CN(C1)C2 11974,c1(C(=O)NC(CNC(C2(C#C)CC2)=O)CC(C)C)ccc(Cl)c(C(F)F)c1 11975,CC1(C)CC2(CC(C(=O)NCC(O)CNC(=O)CP(C)(C)=O)C2)C1 11976,S(=O)(=O)(c1ccc2c(c1)CCCO2)N(CC=C)Cc1cccc(Br)c1 11977,C(=O)(C(CC(C)C)OC)N(C1CCC(NC(C2(CC)CC(C)(C)C2)=O)CC1)C 11978,N1(C(C2(C(=O)OC(C)(C)C)CCCOC2)=O)Cc2ccccc2C(C(=O)O)C1 11979,Cc1cc2sc(C(=O)NCC(C)NC(=O)C(C#N)C(C)C)cc2s1 11980,CC(C)(CNC(=O)CC(C1CCC1)C1CCC1)N=c1[nH]nc(C#N)s1 11981,c1(OC)ccc(O)cc1NC(=O)CCC(C)NC(=O)C(C)(C)C(C)O 11982,CCC(O)(CC)CCNC(C1CC(NC(c2c(C)n[nH]c2C)=O)C(O)C1)=O 11983,c1(C(N2CCCC(NC(C(CC=C)C)=O)C2)=O)cccn2c(CC)nnc12 11984,C1(NC(C2(C(=O)OCC)CCO2)=O)CCCCC1NC(=O)C1=NOCC1 11985,N1(C(C2CCC(C)O2)=O)CC2CCCC(N(C(=O)CCOCC3CC3)C)C2C1 11986,C1(NC(C2CC3CCC2C3)=O)CCCC(CC(N2CCC(F)CC2)=O)C1 11987,CC(C)C(Br)C(=O)c1cnn(C2CCN(C)CC2)c1 11988,C1(c2n(-c3c(CC)cccc3)nnn2)(NC(C)CC(C)C(F)F)CSC(C)(C)C1 11989,N1(C(c2c(N)cncc2)=O)CC2(CCCC2NC(=O)COCC(F)F)C1 11990,C(=O)(C(C)S(C)(=O)=O)NCC1(CNC(c2n[nH]c(C)c2Cl)=O)CC(F)(F)C1 11991,C12(NC(C(CC#CC)NC(=O)C(COC)OC)=O)CCC(CC1)C2(C)C 11992,c1(C(=O)NC(CN(C(c2ccc(OC)c(F)c2)=O)C)C)csc2c1CCC(C)C2 11993,c1(OCC(=O)OC)cccc(C(=O)NCC2(O)CN(C(=O)CCC(C)C)C2)c1 11994,C(CC(C(=O)NC1CC(CNC(=O)OC(C)(C)C)C1)c1ccccc1)=CC 11995,c1(N2CCCC(NC(=O)C(F)CC3CCCCC3)CC2)ncnc2cccnc12 11996,N1(C(CC2(C)CCC2)=O)CCC(C)(C)C1C(=O)Nc1cccc(CO)c1 11997,c1(C(N2CCC(NC(c3nn(C)c(Cl)c3)=O)C2)=O)c(F)cncc1Cl 11998,C(=O)(C(O)CC(F)(F)F)N1CC(CCCCNC(c2ccc([N+](=O)[O-])o2)=O)C1 11999,c1(CNC(C=NOC)=O)ccccc1CNC(C1CC(=O)N(c2cn[nH]c2)C1)=O 12000,C(=O)(CCCCCC(C)C)N1CC(CC(N2C(CC)CCC(C)C2)=O)OCC1 12001,c1(OCC)nc(N2CCCC2CNC(C23CCCC(C2)OC3)=O)ncc1Cl 12002,C1(C(=O)NC2CN(C(c3c(C(C)C)ocn3)=O)CC2C)CCC2(C1)CC2(F)F 12003,CC1(C)CN(C(=O)C(F)F)CCC1NC(=O)CCc1ccc(F)cc1Cl 12004,N1(C(C(C)(C)OC)=O)CCC(C2CCN(C(c3cn(C)nc3C3CC3)=O)CC2)C1 12005,CC1(C)CN(C(=O)Cc2cnc[nH]2)CC1CNC(c1c[nH]cc(Br)c1=O)=O 12006,c1(C(N2CCCC(C(N(C(CC(CC)C)C)C)=O)C2)=O)cccn2cncc12 12007,C(=O)(C1=CCC(C)CC1)N1CCN(C(c2ccc(C)cc2F)=O)CC1 12008,Cc1cc(C)n(CC(=O)NCc2cc(C(=O)NCc3noc(C)n3)co2)n1 12009,c1(CC2N(C(COC(COCCC(C)C)=O)=O)CCC2)ccc(Cl)c(Br)c1 12010,C(=O)(C(C(C)(C)C)NC(C1CCN(C(=O)C=Cc2cncs2)C1)=O)OC 12011,C1(NC(c2c(SC)cccn2)=O)COC2(CCN(C(C3(C#N)CCCO3)=O)C2)C1 12012,C(=O)(C1=C(F)CN(C(C2COCCO2)=O)CC1)NCC(C(C)O)C 12013,C(C(=O)N1CC(NC(C2CCCN2S(C)(=O)=O)=O)C2(CC2)C1)(C(C)(C)C)OC 12014,C12(C(N(CC#C)C)=O)C(NC(=O)C=C(C3CC3)C3CC3)C3CC1C2C3 12015,CC1C(NC(=O)C(C)(C)COC(C)C)CC2CCC1N2C(c1cc(C#N)c[nH]1)=O 12016,C(C(C(=O)N(C1(C2CC2)CC1)C)NC(C1CCC(=O)O1)=O)N(C)C 12017,C1(C#N)(C(N2CCC(CN(C)C(c3ccnc(CO)c3)=O)CC2)=O)CCCC(=O)C1 12018,C1(NC(c2cnc[nH]2)=O)CCN(C(=O)CSc2ccccc2O)C2CC12 12019,Cc1[nH]nc2c(C(N3CCCCC(NC(C4(C)CCCOC4)=O)C3)=O)cccc12 12020,C1(C(=O)NC2CCC(NC(CCc3cc(C)on3)=O)C2)CCC2(CCCCC2)C1 12021,c1(SC)cc(C(=O)NCC2(NC(C3C=CC(C(F)(F)F)C3)=O)CCC2)ccc1N 12022,Cc1ccc(F)c(C(N2CC(CNC(=O)C(C3CCOCC3)C)C(O)C2)=O)c1 12023,C(=O)(C#CC1CCOCC1)N1CCC(C(N2CCCC(CC(C)C)C2)=O)C1C 12024,c1(C(=O)NCCCCCN(C(=O)CC2(C)CC2(Cl)Cl)C)cc([N+](=O)[O-])cnc1N 12025,N#Cc1ccc(N2CCCC(NC(=O)NC(c3ccccn3)CCO)C2=O)cc1 12026,N1(C(CC=C)=O)CCCN(C(=O)C(c2ccc(OC)c(F)c2)C)C(CC2CC2)C1 12027,c1(CC)cccc(C(=O)N(C)CC2(NC(c3cc(C4CC4C)on3)=O)CC2)c1F 12028,Cc1cc(C(=O)NCCn2cc(C(=O)NC(C)CS(C)=O)nn2)ccn1 12029,C1(N(C(C(COC)N(C)C)=O)C)CN(C(c2cn(C)nn2)=O)CC1O 12030,C(C(=O)CCC(=O)N=c1ccn(CC(C)C)[nH]1)OCCOC 12031,C#Cc1ccc(C(N2CC3CC3(C(=O)NC(c3nnc(O)n3C)C)C2)=O)cc1 12032,CCC(C)CCCC(=O)N1CC=CC1C(=O)N(C)CC1CN(C)CCO1 12033,c1(OC)ccc(CCC(=O)N(C(C)CCNC(=O)C=CC(=O)NC2CC2)C)cc1C 12034,C1(O)(C(C)NC(=O)CCCOC2CCOCC2)CCN(C(=O)Cn2ccnn2)C1 12035,C1(C(=O)Nc2c(F)ccc(C)c2F)CC2CCC(C1)S2(=O)=O 12036,Cc1cc(=O)n(CCC(=O)NC23CC(NC(=O)CSc4n[nH]c(=N)s4)(C2)C3)cn1 12037,N1(C(Cn2c(C)ncc2)=O)CCOC(CCNC(C2CC(F)C(=O)N2)=O)C1 12038,c1(C(=O)NC(C)CNC(c2nscc2Br)=O)ccnc(OCCO)c1 12039,c1(CC)c(C(N2CCC(COC)(NC(c3sccc3OC)=O)C2)=O)cccc1F 12040,C1(CCOC)(NC(=O)CCNC(N)=O)CCN(C(c2cc(F)cc(Cl)c2)=O)CC1 12041,c1(OC)c(NC2CCCC(NC(=O)C=Cc3cnccn3)C2)ncnc1Cl 12042,Cn1cncc1C=CC(N1CCOCC1C(=O)NCCc1ccco1)=O 12043,N1(C(c2c(CC)cns2)=O)CC(O)CC1C(=O)NC(COC)CC 12044,C1(NC(CCCC)=O)CC2(CCN(C(=O)C(C(C)C)N(CC)CC)CC2)C1 12045,c1(NC(CCC(=O)NC2(CC=C)CCN(C(=O)CCF)C2)=O)ccc(Cl)c(Cl)c1 12046,CCCC(O)C(=O)NCCCN(CCCNC(=O)CCCC#N)C 12047,N(C(=NCc1ccc(C)cc1)NC1CCOCC1)C(C#C)CN(C)C 12048,C1(OC)C(OC)CN(C(=O)C(C)C2CC2)C1CNC(c1nc(Cl)sc1C)=O 12049,C1(OCC)COCCC1NC(C1CCN(C(C)C(=O)Nc2nccs2)CC1)C 12050,C1(NC(CCC=CC)=O)CC2(CCC(CNC(c3cc(CCC)on3)=O)CC2)C1 12051,Cc1cncc(CNc2cncc(NC(=O)C3CC3)c2)c1 12052,C1(OC)CC(CNC(=O)C=Cc2ccnn2C)N(C(c2cc(C)on2)=O)C1 12053,c1(C(=O)NC(C2CN(C(CC(C)SC)=O)C2)C)ncnc(C)c1C 12054,C(=O)(C(=O)CC(C)C)N1CCC(C(C(=O)N(C)CC2(OCC)CCC2)C)CC1 12055,C1(C(N2C(CCNC(c3cccc(=O)o3)=O)CCCC2)=O)CC12CC(F)(F)C2 12056,C12(C(CNC(=O)CC3CCCOC3)NC(CCC3CC(C)C3)=O)CCC(CC1)C2 12057,N1(C(CCNC(C(C)(C)C)=O)=O)CCC(CCNC(C2(O)CCC2)=O)C(F)(F)C1 12058,CC(C)(C)C(C(=O)NCC(O)CF)NC(c1ccc(CC#N)cc1)=O 12059,C1(CC(=O)Nn2c(Cn3ccnc3)ccc2)CCCCN1CC1CCC(C(N)=O)O1 12060,c1(C2(C(=O)NC(COC)CC3CCCCC3)CCCC2)ccc(OC)cc1 12061,c1(C(=O)NCCN(C(C)C)C(C2(C(=O)N(C)C)CC2)=O)cc(C(F)F)ccn1 12062,C(=O)(C#CC1CCOC1)N(C1CN(C(CC(C)(C)OC)=O)CC1(C)C)C 12063,N1(C(CSCC=C)=O)CC2(CNC(C3(C)C=CCC3)=O)CCC1CC2 12064,c1(C(=O)NC2(C)CN(C(=O)Cc3ccsc3)C2)nc2n(c1Br)CCC2 12065,c1(C(N2CCCC(NC(c3ccco3)=O)(CO)C2)=O)c(F)cc(F)c(O)c1F 12066,CC(CC(C)(C)C)C(F)C(=O)N1CCC1CNC(=O)CC1CNC(=O)O1 12067,C1(NC(c2c(C)nccn2)=O)CCC2(CC1)CN(C(=O)C(C)S(N)(=O)=O)CCO2 12068,c1(OCCCC)ccc(S(=O)(=O)N2CC(c3ccccc3)C3(CCC3)C2)cc1 12069,CC(CC(=O)NC1CCCCC1NC(=O)CC(F)F)S(=O)(=O)c1ccc(F)cc1 12070,C(=O)(C1CCc2nccn21)NCCN(C(c1cccc(CC)c1)=O)C 12071,Cc1cc(C(=O)NC(CNC(c2ccc(CC(N)=O)cc2)=O)C2CC2)ncn1 12072,c1(C(c2n(CC(=C)C)nnn2)NCCc2ccno2)ccc(C(OC)OC)cc1 12073,c1ccc(F)c(Cl)c1.N1(C(C)=O)CC(C)(n2c(=O)ccc(=O)[nH]2)C1.C1CC1 12074,c1(C(N2CC3(C(NC(C4CCC(C)CC4)=O)CC3)C2)=O)cnc2ncc(Cl)cn12 12075,Cc1nnccc1C(N1CC2CC1C2C(=O)N(C)CC1(N(C)C)CC1)=O 12076,N1(CC)CCCC(C(=O)NCC(C)(C)CCNC(C2CC(O)CN2C(C)=O)=O)C1 12077,c1(OC)ccc2onc(CC(=O)N(C)CCN(C)C(c3c[nH]c(=N)o3)=O)c2c1 12078,C1(CNC(CC2(C)CC2)=O)CCCN(C(c2ccc(-n3cnnc3)cc2)=O)CC1 12079,c1(C(N2CC3CN(C(=O)Cc4cc(Cl)ccc4Cl)CC32)=O)cc(Cl)c(Cl)cc1F 12080,N1(Cc2cc(C)n(CCC)c2C)CCS(=N)(=O)C(C)(C)C1 12081,c1(C(=O)NCCCOCCNC(c2c(C)ccnc2O)=O)cc2c[nH]cnc-2n1 12082,C1(NC(CC(C)CNC(C2(F)CCC2)=O)=O)CCC(=O)N(C)C1 12083,C1(=O)C(C(CC)CC)N1.C(C)(C(=O)NC)N(CC(C)C)CC=C 12084,N1(C(c2c(OC)cnnc2OC)=O)CC2ON=C(CNC(c3ccco3)=O)C2C1 12085,N1(C(Cc2scc(C)c2)=O)CC(CNC(C2CC(=O)N(O)C2)=O)CC(C)C1 12086,C(C(F)(F)CN(C(=O)C(c1ccoc1)NC(=O)CSC)C)OC 12087,n1(CC(=O)NCC(C)N(C(CCC(C)SC)=O)C)c(=O)cnc2ccccc12 12088,c1ccc2cc(C3(N(C4CC4)CC4CC4)CCC3)ccc2c1 12089,C1(COC)CN(C(C2CCCC3(CC3)C2)=O)CCN1C(c1cnn(C(C)C)c1)=O 12090,c1(C(=O)NC2C(NC(=O)CSCc3ncc[nH]3)CCC2)cccc[n+]1[O-] 12091,N1(C(C2(C)CC(C)C2)=O)CCC(O)(C(N2CCC(Oc3ccccc3)CC2)=O)C1 12092,c1(C(C(=O)NCC2C3CN(C(=O)CC4CC(F)(F)C4)CC23)=O)ccc(O)c(Cl)c1 12093,N1(C(CC=C)=O)CC(C(=O)N(CC2=CCSC2)C)C2(CCC2)C1 12094,C1(NC(C(C(C)C)O)=O)C2CC3C1C3C2C(=O)NCc1ccccc1F 12095,c1(C(N2C(C(C)(C)NC(C(C)=CC)=O)CCC2)=O)ccc(C(F)(F)F)cn1 12096,c1(CC(=O)NC(C)(C)CNC(=O)CC2CC3(CC3)C2)c[nH]c2ccccc2c1=O 12097,c1(OCCC)cccc(CC(=O)NCCCCCN(C(=O)C(C)CO)C(C)C)c1 12098,N1(CC)CCCC(C(=O)Nc2scnc2C(=O)NC(C2CCOC2)CSC)C1 12099,CC1(C)C2CC(C(=O)NC3(CNC(=O)Cn4ncnn4)CCOC3)CC12 12100,N1(C(C2CC(NC(C=C(C)C3CC3)=O)C2(C)C)=O)CCN2CCCC2C1 12101,n1(CC(N2CCC(NC(CC3C(C)=NOC3=O)=O)C2)=O)cc2ncccc2n1 12102,c1(CNC(=O)NCCCC2CNCCO2)ccc(C(F)F)cc1Cl.C(C(F)(F)F)O 12103,C1(O)(C(N)=O)CCCN(C(c2cc(C(N)=O)cs2)C(=O)NC2CCCC2)C1 12104,C1(CC)C(NC(C2CS(=O)C2)=O)CCCN1C(c1ccc(C)c(C)c1)=O 12105,CC1CCc2c(C(N3CCCCC3CNC(c3cccc(=O)n3C)=O)=O)n[nH]c21 12106,CC(C)C(C(C)NC(c1cscc1Cl)=O)NC(c1ncoc1-c1ccon1)=O 12107,CCCS(=O)(=O)C(C)C(=O)NCC1CN(C)CCN1C(c1cc2occc2[nH]1)=O 12108,c1(C(=O)NC23CCN(C(=O)CNS(=O)(=O)C4CC4)CC2C3)n[nH]c2c1CCCC2 12109,C1(CNC(CCc2cc(C)no2)=O)CCN(C(c2cc(Cl)c(Cl)n2C)=O)CC1C 12110,N1(C(c2c(C)n[nH]c2)=O)CC(NC(c2conc2C2CCCC2)=O)CC(C)C1 12111,c1(C(N2CCOCC2C2CCOC2)C(=O)NC2CC2)cccc([N+](=O)[O-])c1 12112,N1(C(CCS(C)=O)=O)CCC2(CCCN(C(=O)C3Cc4ccc(Cl)cc43)C2)C1 12113,C1(C(=O)NCCCCCCn2cc(-c3cncc(F)c3)nn2)(CC)CCCOC1 12114,C1(C(=O)NCCC#C)COC2(C1)CN(C(=O)C(C)OC)C2 12115,c1(C(N2CCC(O)(CNC(CCC(C)OC)=O)C2)=O)ccnc(C)c1C 12116,C1(NC(C2CCC(O)C2)=O)CC2(CCN(C(C3(F)CC=CCC3)=O)CC2)C1 12117,C(=O)(C1=NN2CC(C)CN=C2N1)NCCN(CCOC)C(c1cccc(=O)o1)=O 12118,n1(CCC)cc(C(=O)N(CCNC(=O)CC2OCCC2C)C(C)C)nn1 12119,c1(C(=O)NC(CC)CNC(=O)C(C)SC(F)(F)F)ccc([N+](=O)[O-])s1 12120,N1(C(C(C)(C)N(C)C)=O)CC23CCCCC2(C1)CN(C(=O)C(O)CC(N)=O)C3 12121,Cc1ncnc(C)c1CC(=O)NCC(C)CN(C)C(c1occc1CN(C)C)=O 12122,c1(C(N(C2CN(C(CCCN(C(C)=O)C)=O)C2)C)=O)ccc([N+](=O)[O-])s1 12123,C1(NC(C2CCC(CC)O2)=O)CC(OC)CN(C(=O)Cc2ccns2)C1 12124,Cc1nc2cc(C(=O)NC(CNC(=O)CN3CCCCC3=O)CO)c(F)cc2[nH]1 12125,C=CCC(C(=O)N1CC(CSC)C1)NC(c1ccnn1CCC)=O 12126,Cc1cc(C(=O)NC2CC(CNC(C3CC3(C)C(C)C)=O)C2)c(F)cc1Cl 12127,c1(CC)cc(C(=O)NC2CCC2NC(c2cc(N)c(F)cn2)=O)cc(O)n1 12128,C1(COC)CC(F)CN1C(c1cccnc1OC)=O.c12ccc(o1)CNC2=O 12129,C1(CC)CCC(N=c2ccc(Br)c(S(=O)(=O)NC(c3cccs3)C)[nH]2)CC1 12130,N#CC1(CC(N2CC=CC2CNC(C2CCCCS2)=O)=O)CCCCC1 12131,CC1(C)CC(CNC(C2CSCN2C(=O)CC=C(Cl)Cl)=O)CCO1 12132,C1(NC(C23N(C(CN(CCOC)C)=O)CCC2C3)=O)CN2CCC1(C)CC2 12133,C(=O)(C(C)(C)CO)NCC(=O)Nc1cn(C)nn1 12134,N1(C(C(CC=C)CC)=O)CC(NC(C2CC(C)(C)C2)=O)CC2(CCC2)C1 12135,N1(C(CCn2c(C)cc(C)n2)=O)CCC2CC1CN2C(C1CCCS(=O)(=O)C1)=O 12136,Cc1cc(C)c2[nH]c(=NCC(C)NC(=O)Cc3c(F)cccc3Cl)sc2c1 12137,C1(CCOC)(NC(=O)C(=Cc2cnc[nH]2)C)CCN(C(C2(C)CC=CCC2)=O)C1 12138,c1(CCC(=O)NC(CN(C(=O)C(C)CC(F)F)CC)C)c(C)ncnc1O 12139,N1(C(COCC=C)=O)CC2C=CC1C(C(=O)NCC(CO)C(C)CC)C2 12140,N1(C(=O)CCOc2ccc(F)cc2)CCN(C(=O)Cn2ncnn2)C2CCCC12 12141,c1(CC(=O)N(CC(C)NC(=O)CC2SC(=N)NC2=O)C)ccc(O)nn1 12142,CN1CCC(C(=O)NCC=CCC(=O)NC2(C3CC3)CCCC2)CC1=O 12143,C1(CC)CCCC1C(=O)N(CC(C)CNC(c1csc(C)c1)=O)C 12144,Cc1ccc(F)c(N)c1C(=O)NC1CC(C)(CNC(C2CCCN(C)C2)=O)C1 12145,Cc1sc(C)c(C(N2CCC(C)C(NC(c3cnc[nH]3)=O)C2)=O)c1C#N 12146,c1(CC)nc(-n2cccc2)sc1C(=O)NC1CN(C(c2cnoc2C)=O)CC1C 12147,CN=c1[nH]c(=NC(C)c2cccc(S(N)(=O)=O)c2)[nH]c(=NCC(C)N(C)C)[nH]1 12148,c1(C(=O)NCC2C(CNC(C3(CCN(C)C)CC3)=O)C2)ccc2c(c1)COC2=O 12149,N1(C(CNC(=O)OC)=O)C2CCC1CC(CCNC(=O)Cc1ccnn1C)C2 12150,Cc1occc1C(=O)OCc1cn(C(c2ccccn2)C)nn1 12151,Cc1[nH][nH]c2ncnc(=NCC3(CNC(C4C(C)C4C)=O)CCC3)c1-2 12152,c1(C(C)C)nc(C(=O)NCC(C)(C)NC(c2cc(C(N)=O)no2)=O)cs1 12153,N1(C(C2(C#C)CCC2)=O)CCCN(C(=O)CCC2CC2(F)F)CC1 12154,N1(C(c2ccc(Cl)cc2F)C(=O)NCC2CC2)CC=C(c2cccs2)CC1 12155,C(=O)(CC1COc2ccccc21)NC1C(CNC(CC2(C=C)CCOCC2)=O)C1 12156,c1(C(=O)NCCCC2(NC(=O)CCNC(N)=O)CC2)cnc(-c2ccco2)s1 12157,c1(CCNC(N2CCCC2C2CCCC2O)=O)cccc2n[nH]cc12 12158,C(C(=O)N1CCC(n2cc(-c3ccc(Cl)s3)nn2)C(O)C1)(C(C)(C)C)SC 12159,C1(CNC(Cn2c(=N)scc2)=O)CN(C(=O)CSC(F)(F)F)CCO1 12160,N1(C(C(CCSC)O)=O)CCC(CNC(=O)CCc2ccnn2C)CC1C 12161,c1(C(C(=O)NCCSC)N(C)Cc2c(C(=O)OC)cccc2)ccc(F)cc1Cl 12162,CC1CN(c2cc(C(F)F)ncn2)CCC1NC(C1CCC2CC2CC1)=O 12163,C1(C(N2CC(NC(C3CC(C)(C)C3)=O)C(C(F)F)C2)=O)CCn2c(O)nnc2C1 12164,C1(CC(=O)OC)CS(=O)(=O)CCN1C(=O)C(=O)N=S(C)(C)=O 12165,c1(CC)ccc(C(=O)NC(C)CN(C(=O)CN2CCNC(=O)C2)CC)c(Cl)c1 12166,C1(C(N2CC(c3ncccn3)C2)=O)C2CN(C(=O)CSc3ccccn3)CC12 12167,CC1(NC(c2cnn(CCNC(c3ccccc3C#N)=O)c2)=O)CCC(O)CC1 12168,Cc1noc(C)c1CNC(C1CCN(C(C2CCC(O)C2)=O)CC1)=O 12169,C1(NC(C(CC)Oc2ccccc2Cl)=O)CCCC12CN(C(c1cc[nH]c1)=O)C2 12170,C1(C(=O)NC2(CO)CCN(C(C34CC(C3)C(C(F)F)O4)=O)C2)CCS(=O)(=O)CC1 12171,C1(CNC(C2C(C)OC(C)C2C)=O)CCC2(CN(CCOC3CCCCC3)C2)O1 12172,C(c1ccc(C(=O)O)cc1)=CC(N1C(C(=O)OC)CC1)=O.c1cc(C(=O)O)co1 12173,N1(C(c2cn(CCOC)nn2)=O)CCN(C(c2c(C)ncn2O)=O)CC2(CC2)C1 12174,CCC(C(=O)OC)C(=O)NC1CCCCN(C(C2OC(C)CC2C)=O)C1 12175,N1(C(c2cn(C3CC3)cn2)=O)CCC2(C1)CN(C(C1CC=CC(O)C1)=O)C2 12176,N1(c2nnn(C)n2)CC2CC1CCC2NC(=O)C(C)(C)n1cnnn1 12177,CC1CCCc2nc(C(=O)N(CC(O)CN(C(=O)Cc3csc(S)n3)C)C)cn21 12178,c1(NC(C2N(C(CCOC)=O)CC(F)C2)=O)ccc(F)c(C(=O)OC)c1Br 12179,C12(CNC(c3c(COC)cc[nH]3)=O)CCC(CC1)N2C(=O)CC1(C(=O)OC)CC1 12180,C1(CNC(C(=O)N(c2ccccc2O)C)=O)CC2CN(C(c3nncn3C)=O)CC12 12181,c1(-n2c(CCCCSC)nc(-c3ccc(F)cc3)n2)ccc(F)c(Cl)c1 12182,C=C(C)C(CC(=O)N1CC(OCCNC(=O)C(c2cnn(C)c2)C)C1)OCC 12183,N1(C(c2cnc(C(C)C)o2)=O)CCC2(CCC(NC(=O)C(C)n3cncn3)C2)C1 12184,N1(C(C(CCC)C#N)=O)CC2CCC1C1CN(C(c3cccnc3)=O)CC21 12185,C12(C(N3C(c4ccc(C)o4)CCCC3)=O)CCC(C)(CC1)O2 12186,c1(CS(=O)(=O)NCCSCCOC)cccc(OCCSC)n1 12187,N1(C(CC2N(C(c3cnc(C)s3)=O)CCC2)=O)CC(C)CC(C)(C)C1 12188,N1(C(c2c(CNC(c3cnc(CC)s3)=O)ocn2)=O)CCCN(C)CC1 12189,c1(C(=O)NC(CCOC)CNC(=O)C=CC2CCCC2)cnc[nH]c1=N 12190,c1(NC(CCC=CCC=C)=O)ccc(NC(=O)C(O)P(C)(C)=O)cc1C 12191,N1(C(c2ccn(C)c2)=O)CC2CC3CC2C1C3NC(=O)C1=CC(O)CCC1 12192,c1(C(C)C)nc(Cl)cc(=NCC(C)NC(=O)CC2CC(F)(F)C2)[nH]1 12193,N1(CC(=O)CC2CC2)CC23COCC2(COC3)C1 12194,c1(OC)ccc2cc(C(=O)NCCCOCCNC(=O)C(C)OC(C)C)[nH]c2c1 12195,c1(CC(=O)N(CC)CC2CCCN2C(=O)CC2OCCCO2)ccc(F)c(C)c1 12196,CS(=O)(=O)c1ccc(CC(=O)NC2CC2(C(=O)O)C(=O)O)cc1 12197,C1(C(=O)NC(CCC)CCC)CCCCN(C(=O)CCc2cc(C)no2)C1 12198,c1(C(=O)NCCCN(C(c2cc(COC)sc2)=O)C2CC2)nccn2nccc12 12199,c1(SCC(=O)NCCN(C(=O)C(C)(C)OC)CC)ccccc1CSC 12200,N1(C(c2c(CC)noc2)=O)CCC2(NC(c3occ(C)c3C)=O)CCCCCC12 12201,C1(C(=O)NC2C(C(=O)NCC3(OCC)CN(C)C3)CCOC2)C2CCC(C2)C1C 12202,C12(CNC(c3cc(C)c(F)cn3)=O)CCC(CN(C(=O)C#CC3CC3)C1)C2 12203,C1(C)(C(=O)NC(CC(C)C)CNC(C2(C#N)CCCCC2)=O)CC(C(C)C)=NO1 12204,C1(N(C(=O)C(C2CCCC2)SC)CCOC)CCN(C(C2CS(=O)(=O)C2)=O)CC1 12205,C1(NC(CCSCC(N)=O)=O)CCN(C2CCN(C(C3CC=CCO3)=O)C2)CC1 12206,Cc1cccc(Br)c1C(=O)NC1CN(C(c2ncoc2C)=O)CC1C#N 12207,c1(NC(C2CN(c3ncnc4ccsc34)CCO2)=O)ncc2c(Br)cccc2n1 12208,CC(C(=O)OC(C)(C)C)N(C(C(C1CC1C1CCOC1)N(CC#N)C)=O)C1CC1 12209,C(=O)(C(F)CCC)NC(c1ccccc1)CNC(CCOCC#C)=O 12210,N1(C(C(CC)OC)=O)CCC(CC(N2CC(C(C)C)C2)=O)C1(C)C 12211,CC(C)(C)C#CC(=O)NCC1CCCCC1C(=O)NOCCC(F)F 12212,c1(OC)ccc(NC(=O)NC(C)CO)c(C(=O)N(C2CCCCCC2)C)c1 12213,c1(C(N(C(CN(C(Cc2cncc(C)c2)=O)C)C)C)=O)cnc2c(c1)nnn2C 12214,CC1CCN(C(=O)C(c2ccc(F)c(F)c2)(C)C)CCN1C(C1CCCOC1)=O 12215,C(C(C)C(F)F)NC(CCN(C(C(C)=C(C)C)=O)CCCO)=O 12216,N1(C(CCC(C)C)=O)CC(O)(C2(CNC(c3cccc4ccnn34)=O)CC2)C1 12217,Cc1c(C(=O)N(CC(C)(C)NC(=O)C=CCO)C)[nH]c2c1CCCC2 12218,C(=O)(CC1=NNC(=O)C1)N1CCN(C(c2c(C)oc(C(C)C)n2)=O)CC1CO 12219,N1(C(C2(C=C)CC2)=O)CC(NC(=O)C(C)C=Cc2ccc(C)cc2)C2(CCC2)C1 12220,CC(CF)CC(=O)NCCCC1(NC(c2nccnc2N)=O)CC1 12221,Cc1nscc1C(=O)NC(C1CCN(C(=O)CC2CCCN2C(C)C)C1)(C)C 12222,CC1CC2CN(C(=O)C(=O)NCC3CCC(C4CC4)CC3)CCN2C1 12223,Cc1nc(=NCc2ccc(CNC(C34CCC(C)(CO3)C4)=O)c(F)c2)[nH]cc1Br 12224,c1(N2CCC(CCNC(Cc3ccn(CC)n3)=O)CC2)nc(Cl)ncc1Cl 12225,C1(C(=O)NC2(CO)CN(C(c3ccc(C)c(Br)c3)=O)C2)CCn2ccnc2C1 12226,Cc1cn2cc(NC(c3cscc3-c3cccc(CO)c3)=O)ccc2n1 12227,CC(CC(=O)NCC1(C(C)(C)O)CN(C(=O)C(C2CCCCC2)O)C1)P(C)(C)=O 12228,[N-]=[N+]=NC1CCN(C(=O)C(C2CCC2)NC(=O)C2CC2)CC1 12229,c1(OCC)ccc(CN(c2ccc(C(=O)N(C)C)c(C)c2)C)cc1OC 12230,C(=O)(CCN(OC)C(=O)CS(=O)C(C)C)N1C(CC)CC(F)C1 12231,N1(C(c2ccc(C)c(C)n2)=O)CCC2(CCCN(Cc3cn[nH]c3)C2)C1 12232,C12(NC(C(c3cccc(Cl)c3)CC)=O)COC(C)(C1)C2 12233,c1(CC(=O)NCC(CC)(CC)NC(C2CNC(=O)N2)=O)c[nH]c2ccc(C)cc12 12234,C1(CNC(Cc2cc(C)on2)=O)CCC(NC(=O)Cc2ccccc2Br)CC1 12235,C1(CC=C)(NC(C2CC(CC)CO2)=O)CCCN(C(C2C3CC4C(C3=O)C24)=O)C1 12236,C1(NC(CN(CCCCCC)C)=O)CCCCCC1NC(C1(CO)CC1(F)F)=O 12237,C=C(Br)CC(C)(C)C(=O)NC1CCCN(C(C2(C#N)CCOC2)=O)CC1 12238,C1(NC(c2nc(CCC)oc2)=O)CCC(C(=O)NC2C(C)CCC2C)CC1 12239,C1(CC(=O)NC2C3CN(C(C4CCN(C(C)=O)CC4)=O)CC32)CCC2(CC1)CC2 12240,N1(C(=O)CC2CCCC3CC23)CC(C2CC2)(C(N2CCCC(CO)CC2)=O)C1 12241,c1(CC)cnc(C)c(NC(=O)C(CCNC(=O)CP(C)(C)=O)OC)c1 12242,c1(NC(c2c(C)cccn2)C)ncccc1S(=O)(=O)NC1CCCC(O)C1 12243,c1(C(N2CC3(CCCCN3C(c3ccns3)=O)C2)=O)cc2cc(F)cc(F)c2[nH]1 12244,C(=O)(N=c1cc2ccccn2[nH]1)C1C(C(N2CCSCC2C2CC2)=O)OCC1 12245,C(CCN=c1ccnc(Cl)[nH]1)NC(c1coc(C2CCOCC2)n1)=O 12246,CCC(C)(C)C(=O)N(C)CC1CCN(C(c2cnc(SC)nc2)=O)C1 12247,C#Cc1cccc(C(N2CC(CC=C)(NC(C3CCCC3(C)C)=O)C2)=O)c1F 12248,N1(C(CC#N)=O)CCC2CCN(C(=O)CCn3ccnc3)CC2C1 12249,C1(C(N2C(C)C(NC(c3cc(O)nn3C)=O)CCC2)=O)CCc2cnn(C)c2C1 12250,N1(C(C(C)N(CC)CC)=O)CCOCC1CNC(=O)COCc1ccc(C)cc1 12251,C(CC(F)F)(C(=O)N1CCCC2(CC2)C1)N(C(=O)CC1CCCSC1)C 12252,c1(SC)ncc(N)c(C(=O)NC2CCC(NC(C3CC3C)=O)C2)n1 12253,N1(C(C(c2ccccc2)NC(C)=O)=O)CCC(C)(NC(=O)CC2(O)CCC2)C1 12254,Cc1oc(Cl)nc1C(=O)N(C(C)CCNC(=O)Cc1ccccc1O)C 12255,C12(C(N3C(C#C)CCC3)=O)C(NC(C3CCC(N(C)C)C3)=O)C3CC1C2C3 12256,C1(C)(CC)CCC(C(=O)N(C2(CC(=O)NC(C)(C)CCO)CC2)C)O1 12257,C1(CC(C)C)COCC1(c1nnnn1C1COC1)Nc1cnn(C(C)(C)C)c1 12258,CN1CC(C(N2CCCC(NC(=O)CCCc3ccsc3)C2)=O)CC1=O 12259,C(=O)(C1Cc2c(Cl)cccc21)NCC(C)(CO)NC(c1c(C)ncc(N)c1)=O 12260,c1(CC(C)N(C=O)CC(c2ccc(Cl)cc2)O)ccc(C#N)cc1 12261,C1(NC(c2c(CC)nn(C)c2)=O)C2CC3CN(C(=O)CC4CN(C)C4)C1C3C2 12262,c1(C(N(CCOC)CCNC(c2cccnn2)=O)=O)c(O)ncc(Br)c1C 12263,N1(C(C(=O)NCC2COC(C)(C)O2)=O)CCOC(C(F)F)CC1 12264,C(C(=O)N(CCC(=O)N1CCCC1C(O)CO)OC)(C1CCCC1)OC 12265,Cc1cc(C(=O)NC(C(N2CCCC2CF)=O)C2CC2)sc1C 12266,C1(NC(C2CCCC(O)C2)=O)CCCN(C(c2cc(C3CC3)cs2)=O)CC1 12267,C1(NC(C(c2ccccc2F)(C)C)=O)CCN(c2nnc(C(N)=O)s2)CC(O)C1 12268,N1(C(c2c(CC)[nH]cc2)=O)CCCC(NC(c2nccc3[nH]ccc23)=O)C(F)C1 12269,Cc1ccc(OCC(=O)NCC2CCCN2C(=O)Cn2ncccc2=O)c(C)c1 12270,c1(C(CNC(=O)CC2CC3(CCC3)C2)NC(C(CC)CC)=O)ccc(F)cc1F 12271,C1(NC(C(=O)NCCCOC(C)=O)=O)CCOCC1 12272,C1(CNC(COC)=O)CC2CCC1N2C(c1cc(C)cc(C)n1)=O 12273,N1(C(C2(CC)CCC2)=O)CCOC(C)(CNC(=O)CC2CC(=O)NC2=O)C1 12274,Cn1c(N(c2nccc(C(F)(F)F)n2)CCC#N)nnc1C1CCC(=O)NC1 12275,N1(CC)CCC(O)C(F)(F)C1.c12ccccc1CNC(=O)C2 12276,CCCCC(C(=O)NCCn1cncn1)NC(c1cn[nH]c1)=O 12277,S(=O)(=O)(c1cnc(Cl)cc1C)N1CC(NCc2c(OC)c(O)ccc2)C(C)C1 12278,CCCC(CC)CCC(=O)NC1CC(CNC(=O)C(CCC(N)=O)NC(C)=O)C1 12279,c1(CNC(N2CCC(C(N(C)C)=O)C2)=O)ccc(N2CCCS2(=O)=O)cc1 12280,Cc1cc(C(=O)N(C2CC(C(=O)NC(C(F)(F)F)C3CC3)C2)C)n[nH]1 12281,N1(C(CN2CCC(C(=O)O)C2=O)=O)CC2(CCN2C(c2ccc([N+](=O)[O-])[nH]2)=O)C1 12282,CC1(CNC(c2cc[nH]n2)=O)CCN(C(c2c(Br)cnn2C2CCC2)=O)C1 12283,S(=O)(=O)(c1ccc2c(c1)CCCC2)CC(c1ccnc(OC(F)(F)F)c1)=O 12284,C1(CNC(C=CC)=O)CCC2(CN(C(=O)C(c3ccccc3)N3CCCC3)C2)O1 12285,C1(C(NOCC=CC)=O)CC12CCN(C(=O)C(CCC)CCC)CC2 12286,c1(C(=O)NC2CCC(NC(C(CCC)O)=O)C2)cccc2ccc(C)nc12 12287,c1(C(N2CC(O)(C3CC3)C2)=O)cc2c(F)c(Cl)ccc2[nH]1 12288,c1(OC(=O)NOC2CN(Cc3cc(Br)co3)C2)ccccc1 12289,N1(C(c2ccc(C(C)(C)C)[nH]2)=O)CCCC(CCNC(c2ccc(C#N)s2)=O)C1 12290,N1(C(=O)CCN2CCCCC2)CCN(C(c2cn3ccnc3s2)=O)C2COCC12 12291,c1(SC)nc(C)c(C(N2CCCC2)=O)s1.C1(C)C(=O)NC(=O)CCNC(=O)N1 12292,C1(CCC)CN(C(c2cnns2)=O)CCN1C(=O)CN(C(c1cccs1)=O)C 12293,Cc1ccc2nc(SCC(N3CC4CCN(C(=O)C(C)CO)CC4C3)=O)[nH]c2c1 12294,c1(COC)nc(OC)cc(NC23CCC(CC2NC(=O)CCCCCF)C3)n1 12295,C(CCC(=O)N(C)CCN(C)C(c1cc(-c2cccs2)[nH]n1)=O)OCC 12296,N1(C(C(C)SC(C)C)=O)CCC(C)(C)C1CC(=O)NCC1CCCCC1 12297,C1(CC#C)(C(=O)NCC2CC2NC(=O)CCCc2nc(C3CC3)no2)CCCC1 12298,N1(CCC(=O)NCC2(CN(C(C(CC)C)=O)C)CC2)CCCCC1C 12299,N#Cc1ccccc1CS(=O)(=O)Nc1cccc(C(=O)Cn2cccn2)c1 12300,N1(C(C2(SC)CCC2)=O)CCC(O)(C(C)NC(=O)COC2CC(F)(F)C2)CC1 12301,C(c1cncn1C)=CC(=O)NCC1(CN(C(C(C)OCC(F)(F)F)=O)C)CC1 12302,c1(C2(C)C(C(=O)NCCNC(c3c(OCC)nccc3)=O)C2)ccc(F)c(F)c1 12303,CC1CCOCC1NC(=O)NC1(Cc2ccccc2Cl)CCCCC1 12304,c1(N(c2ccc(N)cc2)CCNC(N(CCOC)C)=O)ccccc1Cl 12305,c1(OC)cc(N)c(Cl)cc1C(N1CC2CC(NC(c3ccc(F)cc3)=O)C1C2)=O 12306,CCC(C(=O)NCCOCCNC(c1ccc(N)c(Br)n1)=O)C(C)(F)F 12307,C(=O)(CC(O)CC(C)C)N1CCC(C(C(=O)NC(C(=O)OC)(C)CO)F)C1 12308,c1(C(=O)NC2CCN(C(=O)C3=COCCC3)CC2O)cnc2ccc(F)cc2c1 12309,c1(CCC(N2CCC(NC(C(CCSC)O)=O)C2(C)C)=O)nc2cnccc2[nH]1 12310,CCC(C)(C)C(O)C(=O)NC1(C(=O)NCC2CCC(C)(C)CO2)CCOCC1 12311,CCC(C)C(O)C(=O)N1CCCC(C)(CNC(=O)C(C2CCCCC2)C)C1 12312,c1(C(=O)NCC(C(C)C)NC(C2(C)CSC2)=O)cc2cc(F)c(F)cc2[nH]1 12313,C1(NC(COCc2onc(C)n2)=O)CN(C(=O)Cn2cncn2)CC1F 12314,CCC(CC(=O)NC1CC(CCNC(c2cc(Cl)ns2)=O)C1)C(C)(C)C 12315,C(=O)(C(CC)(CC)C(=O)O)Nc1c(C(=O)OCC)cc(OCC)cc1.C(=O)OC 12316,c1(C(=O)NC(CNC(c2cc(C)nnc2)=O)C2CCC2)cc([N+](=O)[O-])ccc1N 12317,CCC(CC(F)F)C(=O)N1CC(NC(N)=O)CC(NC(=O)CCOC)C1 12318,N1(C(CN(CCCCCC)C)=O)CC(CNC(C2(CO)CC2(F)F)=O)C(O)C1 12319,N1(C(C23CC(NCc4c(C)ncs4)(C2)C3)=O)CCN2C(=O)COCC2C1 12320,c1(C(=O)NC2CCN(C(c3c(C)ccnc3C)=O)CC2O)cccc2c1COC2 12321,c1(C(=O)NC2C(CNC(C(CCC)CC)=O)CC2)cc(C)c(Br)c(C)c1 12322,c1(C(=O)NCCCN(C(c2c(C)csc2Cl)=O)C2CC2)cc2c(nn1)CCCC2 12323,C1(NC(=O)CCCCC2CC2)CC2CC1N(C(c1csc3nnsc13)=O)C2 12324,c1(C(N2CC(C(N(C(C=C)C3CC3)C)=O)C(F)(F)C2)=O)ccc2nccn2c1 12325,C1(C2CCN(C(=O)C(=C3CCCCC3)F)CC2)(NC(c2cnsc2)=O)CCC1 12326,N#CC1CCCN(C(=O)C(=O)NCc2cc(O)ncc2Br)C1 12327,N1(C(c2cc(OC)n[nH]2)=O)CC2COCCC2(NC(=O)Cn2ccc(C3CC3)n2)C1 12328,c1(C(N(CC(CC)NC(=O)C(C2CC2)OC)C)=O)cc([N+](=O)[O-])n[nH]1 12329,N1(C(C(C)CC2CC2)=O)Cc2ccccc2CC1CNC(=O)C(C)C(C)(F)F 12330,N1(C(C(F)=CCC)=O)CC2(CCC2)CC1CNC(c1c(C)nn(C(C)C)c1C)=O 12331,C1(C(=O)NC2CCCN(C(C=C(C)CN3CCOCC3)=O)C2)CC2CCC(C1)S2 12332,C1(CN(C(C2(SC)CN(C(=O)CSC(F)(F)F)C2)=O)C)CCCCC1O 12333,C1(C2CC2)(C(N(C2CCN(C(c3cc(-c4cccnc4)n(C)n3)=O)C2)C)=O)CCC1 12334,C1(OC)CCC(C(=O)N(C(C)(C(=O)NC(C)CC(C)C)C2CC2)C)CC1 12335,N1(C(C(C)C(F)F)=O)CCC(C)C(N(C)C(c2cc(C(F)(F)F)ccc2F)=O)C1 12336,O=C(CC(F)(F)C(F)(F)F)NC1CCCCC1NC(C1(c2ncco2)CC1)=O 12337,C#Cc1ccc(CC(N2CCN(C(C)=O)C(CS(C)(=O)=O)C2)=O)c(F)c1 12338,C=CC1(C(=O)NC(C)CN2CCCC2)CCN(C(C2OCCC2(C)C)=O)CC1 12339,N1(C(CCC#CC)=O)CC(NC(=O)C=CC(c2ccc(F)cc2)=O)CC12CCCC2 12340,N1(C(CSCCCC)=O)CCC2(CC1)OCCC2NC(=O)CSc1n[nH]c(O)n1 12341,C1(NC(=O)CN2CCC2)CC2(CCCCN2C(C2CCc3nnnn3C2)=O)C1 12342,c1(C(N(C2CCN(C(c3ccc(C4CC4)nc3)=O)CC2)C)=O)cc(N)nc(Cl)c1 12343,N1(C(CCC=C=C)=O)CCCC(O)(CCNC(=O)CCN2CCC(F)C2)C1 12344,C1(NC(c2ccn(CCC)n2)=O)CCC12CN(C(=O)CCOCC)C2 12345,CCCC(C(O)C(=O)Nc1cccnc1C)NC(c1c[nH]ccc1=O)=O 12346,Cc1cc(Cl)c(C)c(C(=O)NC2CC2CNC(=O)C(C)OC2CCCC2)c1N 12347,C12(NC(c3cc(C)c(Cl)cn3)=O)CCCC1CN(C(C1CN(C(C)C)C1)=O)C2 12348,CCC(CC)C(C(=O)NC(C1CCCN1C(=O)CNS(=O)(=O)CC)C)OC 12349,N1(C(C(C)=C2CCC2)=O)CCN(CC(=O)N(CC(F)Cl)C)CC1 12350,N12CC(C)(C1)OCC2=O.C1(CC(C)C)(C(=O)N(C(C(N)=O)C2CC2)C)COC1 12351,N1(CC2(C(=O)NC(c3ccn(C)n3)C)CCC2)CCN(C(N)=O)CC1 12352,N1(C(c2cc(C)no2)C(=O)NCC(F)F)CCc2cc(C#N)ccc2C1 12353,c1(-n2c(SCCCn3ncc(C)c3)ncc2)ccc(C(N)=O)cc1 12354,Cc1nc(Br)ccc1C(N1C2CN(Cc3cc(Cl)ccn3)CC12)=O 12355,N1(C(C2N(C(C(C)NC(=O)C3CC3)=O)CCSC2)=O)Cc2cncnc2C1 12356,c1(OC)cc(C(N2CCC(NC(=O)C(Cl)=CCl)CC2C)=O)ccc1[N+](=O)[O-] 12357,C1(c2cn(COC3CCC(C4CC4)NC3)nn2)(NC(CC2(C)CC2)=O)CC(F)(F)C1 12358,n1(C(C)C)ncc2cc(C(N)=O)cnc12.c1(C23CC(C2)NC3)c(F)cccc1F 12359,C(=O)(C(CC(C)(C)C)OC)NCCN(C(=O)CC1CC1(C)C)CCC 12360,N1(CCSc2ccc(C(c3cn(C)nc3)(C)C)cc2)CCCCCCC1 12361,C1(NC(C2C(CC)C2)=O)CCCCCCC1NC(=O)CCc1cnc[nH]1 12362,c1(C(N(CC(CC)C)C)=O)coc2c1CN(C(C1CC1C(F)(F)F)=O)C2 12363,C(=O)(C(O)C(C(C)C)OC)NC(CNC(C(CC)N(C)C)=O)COC 12364,C(N=c1[nH]c(N2CCCC(C(N)=O)(N(C)C)C2)nc(=N)[nH]1)C1(OC)CCCCC1 12365,C1(F)(C(N2C(C)(c3ccc(C(F)(F)F)cc3)CCC2)=O)CC2CCC1C2 12366,C1(N(C(c2c(C)nccc2)=O)C)CN(C(C2CC3C=CC2C3)=O)CC1(C)C 12367,c1(OC2CN(C(=O)NCC)C3CC23)nc(C)cc(C)c1C(=O)OC(C)(C)C 12368,Cc1ccsc1CCCC(=O)NCC(CO)NC(=O)CN1CCCC1 12369,C12(CNC(CS(=O)(=O)NC)=O)CCCC1CN(C(c1cc(C)co1)=O)C2 12370,Cc1csc(=O)n1CC(=O)NC1C2CC1N(C(=O)C=Cc1cncs1)C2 12371,c1(C(=O)NCC2N(C(C(C=C)(C)C)=O)CC2)ccc2cnccc2c1 12372,C(CCC(=O)NCCc1cn(CC2(COC)CCC2)nn1)CNCCOC 12373,Cc1cnn(C)c1C(=O)NC(C)C(C1CCCCC1)NC(c1ccsc1)=O 12374,C1(C(=O)NCCN(C(c2cc(C(=O)OC)nn2C)=O)C)CC12CCc1ccccc12 12375,N1(C(c2ccc(OC)s2)=O)CC(NC(C2CCN2C2CCCC2)=O)CC12CCCC2 12376,N1(C(C2(CCNC(C3CC(C)(C)OCC3)=O)CC2)=O)CCCC(C)(O)CC1 12377,c1(C(=O)NCC2CN(C(C3C(C)OCCO3)=O)C(C)(C)C2)c[nH]c2ccccc12 12378,C(=O)(C1=NNC(=O)C1)N(CCCCC(=O)NCCC1CC(C)(C)CO1)C 12379,O=C(C1=CCCOCC1)NC1CN(C(c2cc(Cl)ns2)=O)CCC1O 12380,CC1CC(NC(c2cn(CCF)nn2)=O)CN1C(=O)CCC(F)F 12381,N#CCCCCCC(=O)NC1CC2CCC1CC2NC(C1CCS(=O)(=O)CC1)=O 12382,C=CC1CCCC(NC(C2CC(C)(NC(=O)C=CC(C)(C)C)C2)=O)C1 12383,N1(CC)CCN(C(c2nc(Cl)cs2)C(=O)Nc2ccc(Cl)cc2F)CC1(C)C 12384,C(=O)(CCCC(=O)N1CCC(C(C)NC(=O)CC2CCC(C)(C)CC2)C1)OCC 12385,c1(SC)ccccc1C(N1CCC(NC(c2ccc(CN(C)C)[nH]2)=O)C1C)=O 12386,N1(C(C2CCCN(C(C)C)C2)=O)C2CCCC1CN(C(=O)C(C)CC(N)=O)C2 12387,C1(CN=C(NC(C)C)NC2CCCSC2)CC2(CC2)S(=O)(=O)N1 12388,Cc1ccc(C=CC(N2CCC3(CC3C(=O)NCC3(CC(N)=O)CC3)C2)=O)cc1 12389,C(=O)(C1CCOc2c(F)cccc21)NC(CC(C)NC(C1CC2C=CC1C2)=O)C 12390,C1(C(=O)NC2C(NC(=O)Cn3cc(C4CCC4)nn3)COC2)CCCOCC1 12391,Cc1cccc2c1c(CNC1CC(NC(=O)C(O)C(C)C)C1)cn2C 12392,N1(C(C2CC(=C)C2)=O)CCN(C)C(C(=O)NC2(C(=O)OC)CCCO2)C1 12393,c1(C(N(C2CCN(C(=O)COc3ccccc3)C2)C)=O)c(N)cnn1C 12394,c1(C(N(CCC(C)NC(c2ccc([N+](=O)[O-])cc2)=O)C)=O)cc2c(ccn2C)[nH]1 12395,C(=O)(CC(CC)C(C)C)NC1C2(CN(C(c3nc(CC)sc3)=O)C2)CC1 12396,C(N=c1nc2c(ncn2C)c(NCc2ccoc2C)[nH]1)C1(CCC)CC1 12397,c1(C(=O)NCCCNC(CC(CCC)(C)O)=O)cc(S(=O)(=O)CC)cnc1O 12398,Cn1cc(C(O)C(N2CCC(OCCCNC(=O)Cc3cccnc3)C2)=O)cn1 12399,c1(OC)cc(C)ccc1OCC(=O)NCCC(C)NC(=O)C(C)S(N)(=O)=O 12400,CC(C)C(C(C)NC(c1c[nH]nc1-c1ccncc1)=O)NC(=O)CSCC(N)=O 12401,N1(c2nnc(C)s2)CC2(C1)SCCC2NC(C1CC(=O)N(C(C)C2CC2)C1)=O 12402,CC1NC(=O)CCC1NC(=O)C1=NOC(CNC(C2COCC(C)O2)=O)C1 12403,C1(N2CCC(N(C(=O)CC3CCCCCC3)C3CC3)C2)CCC(=O)NC1=O 12404,C12(NC(COCCCC)=O)CCN(C(c3ncn4c3CCC4)=O)CC1C2 12405,c1(CC(=O)N(CC(C)N(C(C(CCC)OCC)=O)C)C)cc(F)cc(Cl)c1 12406,N1(CC(C)C)N=C(C(=O)N2CCCN(C(=O)C(C)N(C)C)C(CO)C2)CCC1=O 12407,N#CC1(C(=O)NC2CC(CCNC(=O)C=C(Cl)Cl)C2)CC2(CC2)C1 12408,Cc1c(C(=O)NC2CC(NC(C3(F)CCOC3)=O)C2)[nH]c2ccc(C(C)C)cc12 12409,Cc1cnc(C=CC(=O)NCCCC(C)NC(c2sc(C)cc2OC(F)F)=O)[nH]1 12410,N1(C(c2ccnc(F)c2)=O)CCC(F)(F)C(CNC(C23CCCC2C3(F)F)=O)C1 12411,Cn1nc(C(N2CC(O)CC2(C)C(=O)NOCC(O)C(C)(C)C)=O)ccc1=O 12412,C1(CNC(C2(C)CC=CCC2)=O)CC12CCN(C(C13CC(C(F)F)(C1)C3)=O)CC2 12413,c1(NC(C23CC(C(N4C5CCCC4COC5)=O)(C2)C3)=O)cccc2n[nH]cc12 12414,c1(OC)cccc(N2CC3CCC2C(NC(C2CC(=O)N(C)C2)=O)C3)c1[N+](=O)[O-] 12415,CP(C)(=O)c1ccnc(C(N2CCCN(C(c3cccc(Cl)c3N)=O)CC2)=O)c1 12416,c1(C(N2C(CNC(c3cnc(C)s3)=O)CC(O)C2)=O)cccc(CO)c1C 12417,C1(NC(COCCSC)=O)CCCC1CNC(=O)CCC1CCN(C)C1 12418,Cn1cc(C(N2CC3CC3(C(=O)NC3CNC(=O)C3)C2)=O)n(C)c1=O 12419,CCC(C)C(C)(O)CNC(C1CCC(C2CC2)N1C(c1cccc(O)c1F)=O)=O 12420,c1(-c2ncc(C(N(C(C)CO)Cc3ccccc3)=O)s2)ccccc1Cl 12421,N1(C(CCSc2ccc(C)cc2)=O)CC2(CCC2NC(=O)CC2CNC(=O)C2)C1 12422,CC(=O)CCCC(=O)N(C)CC1CCN(C(=O)COCc2ccnc(O)c2)C1 12423,N1(C(C(C)OC2CCCCC2)=O)CCC(CNC(C2(CO)CC2)=O)C12CCC2 12424,C12(C(=O)NCC(CSC)OC)CC(C(=O)NCCCl)(C1)C2 12425,C1(O)(CCNC(C)=O)CCN(C(=O)C(Cc2ccccc2)n2cnnc2)C1 12426,c12cccc(c1)NC(=O)NC2.N1(CC(C)C)CCC(NC2CC2)C1 12427,C1(CC(=O)NC(Cn2cncn2)C(=O)NCC2CC2Cl)CNC(=O)O1 12428,CC#CCC(CO)NC(C1(CNC(C2C(C#N)C2(C)C)=O)CCCC1)=O 12429,C(=O)(C(C)(C)C(C)(C)C)NC1C(C(=O)NCCC(C)(C)OC)CCCCC1 12430,C(=O)(N=c1[nH]onc1C1CCCCC1O)C1(C(O)CNc2ccc(Br)nc2F)CC1 12431,N1(C(C)=O)CCN(C(=O)C(Cc2ccco2)NC(=O)Cc2coc(C)n2)C(C)C1 12432,C1(CC=C)(NC(c2cc(COC)on2)=O)CCN(C(C2CSCCS2)=O)C1 12433,C1(CC(=O)NCCCC=CC)C(NC(c2csnn2)=O)CC1O 12434,c1(OC)ccc(-c2ncc(-c3cn(Cc4ccco4)nn3)s2)cc1 12435,C1(NC(CSc2n(C)ccn2)=O)CCC2(CC1)CCN(C(=O)CC1CC1(C)C)C2 12436,N1(C(C(CN=[N+]=[N-])NC(C2CC2OC(C)(C)C)=O)=O)CCn2nncc2C1 12437,CC1OC2(C(=O)NC3C=CCN(C(c4c(F)cccc4F)=O)C3)CCC1CC2 12438,c1(C(N2CC(C)C(CNC(c3cc(Cl)no3)=O)CC2)=O)ccc2ncccn12 12439,C1(CCNC(C(c2cccnc2)NC(CCN(C)C)=O)=O)CC1C1CC1 12440,c1(NC(CCOC)C)ncccc1S(=O)(=O)N1CCCCC2(CCCC2)C1 12441,c1(C(=O)NC2CC(CNCCC(=O)OC)C2)c(N2CCCC2)cccc1Cl 12442,N1(CC(C)(C)NC(C(CC2CC2)OC)=O)CCN(C(C23CCCC2C3)=O)CC1 12443,C=CC1(CC(=O)NC2(CC(C)(C)C)CC2)CN(C(C2CC(C)(C)CO2)=O)C1 12444,C1(C(=O)OC)CC2CC2N1N1CC(NC(=O)OC(C)(C)C)C(F)(F)C1 12445,C(CCOCCOC)(C(=O)NCCN(C(=O)C1=CCCC1)CCOC)OC 12446,C=CC1(C(=O)NC(c2nn[nH]n2)C2CC2)CCN(C(=O)C=CCC)C1 12447,c1(C(N(CCCNC(CC(N2CCCCC2=O)C)=O)C)=O)ncccc1Br 12448,CC1CCC(C)(C(=O)N(CC(C)CNC(=O)C(O)Cc2ccccc2)C)C1 12449,c1(C(=O)NCC2CC(NC(c3cc(SC)c(C)o3)=O)C2(C)C)ccc(N)cc1Cl 12450,CC1C(C(=O)N(C2CCOC2=O)C)CCCN1C(c1ccc(F)cc1)=O 12451,c1(N2CCC(CC=C)C2)cc(Br)ccc1S(=O)(=O)N1CCOCCC1 12452,C1(NC(c2n(CC)ncc2Cl)=O)CC2CCC(C1C)N2C(=O)C(C)S(=O)CC 12453,c1(C(N2CC3C(CCNC(=O)CSC(F)(F)F)(CC3)C2)=O)cnc2cc[nH]c2c1 12454,N1(C(c2c(CC)nccc2)=O)CCCC(C)(C(=O)Nc2cc(Br)cnc2Br)C1 12455,CON(C)C(=O)CN(C)N1CCOC(COC(F)F)C1 12456,c1(OC)cccc(C(C)NC(=O)NC(C(O)CO)C2CC2)n1 12457,CC1CSCCN(C(c2cnn(CCNC(=O)CC3CC(F)C3)c2)=O)C1 12458,CC1CC(CNC(C2(F)CCCCC2)=O)CN1C(=O)CCc1cnn[nH]1 12459,C(CC(O)C(=O)N1CCCC(NC(c2cnnn2-c2ccccc2F)=O)C1)SC 12460,c1(OC)ccnc(NC(C2(C)CCCN2C(c2cc(O)cc(F)c2)=O)=O)c1I 12461,C1(C(N2C(C(C)NC(c3ccc(Cl)cn3)=O)CCC2)=O)OCC2COCCC12 12462,C1(C(N2CC(c3cn(CCC=C=C)nn3)(C(=O)OC)C2)=O)CC2C=CC1C2 12463,C1(NC(c2c(CC)scc2)=O)CC2CCC(C1)N2C(=O)C(C(CC)CC)OC 12464,CC(C)C(CN(C)C)C(=O)NC1CCN(C(=O)CCC2CC2)CC1O 12465,C(CSC)(CC(=O)N(C)CC1CN(C)CCO1)NC(CCN(CCC)C)=O 12466,C(CC(C)(C)C(=O)NC1CCC(CNC(=O)COc2ccc(Cl)cc2C)C1)OC 12467,N1(C(C(C(C)C)SC)=O)CCC(C)C(NC(c2cc(C(C)(C)C)n[nH]2)=O)C1 12468,N1(C(=O)C2=CSCS2)CCC2(CC1)CN(C(C1CC3(CCCC3)CO1)=O)C2 12469,C1(NC(c2ccc(CC)cc2O)=O)CC(NC(c2ccoc2)=O)C12CCOCC2 12470,CC1COC2(C1)CN(C(C1CC3CC1CC3NC(C1CC3(C1)CC31CC1)=O)=O)C2 12471,C1(CC(=O)NC(C(=O)OCC=C)(C)C)C2CCCC2N1C(=O)CCc1cnoc1 12472,N1(C(CC=C(C)C)=O)CCC2(CC1)CN(C(C1C3CCC1CC3)=O)CC(C)O2 12473,C(CC(C)C)(C(=O)N1CCCC(NC(c2c[nH]c(C#N)c2)=O)C1)NC(=O)OC 12474,C(C(C)(C)CNC(C1(OC(C)C)CCC1)=O)N(C(=O)CCc1conc1C)CC 12475,c1(-c2scc(C)c2)nc(C(=O)Nc2cccc(F)c2C(N)=O)ccc1F 12476,Cc1nc(NC(=O)Cc2ccc(C(F)(F)F)cc2)cnc1Cl.C12CC1CNC2=O 12477,O=C1CN(CC(N2CCC3CC23C(=O)Nc2cnccc2CO)=O)CCN1 12478,CC(C)C(O)C(C)C(=O)N1CC=CC1(C)C(=O)N(C1(C2CC2)CC1)C 12479,Cn1nc(C(=O)NCC2CC(NC(=O)C(c3ccc(Cl)cc3)(C)C)C2)ccc1=O 12480,c1(CC)n[nH]cc1C(=O)NCCC1CCN(C(=O)C(O)C2CCC2)C1 12481,Cc1cccc(C)c1C(N1CCN(C(c2cc(O)ccc2Cl)=O)C2CC12)=O 12482,c1(CNC(=O)C2=CC(C)(C)C2)cc(C)ccc1OC.C=C1CC2(C1)C(=O)NC2 12483,C=CCC(C(=O)NC1COCC1CNC(=O)C(C(C)(C)C)NC(N)=O)C(C)C 12484,CC1CC(NC(c2csnc2Cl)=O)CCN1C(C1CN2CCC1CC2)=O 12485,C1(C)(CNC(CS(=O)(=O)NCC)=O)CC(F)(F)CN1C(c1cc(C(C)=O)on1)=O 12486,c1(C(=O)NCC2C(C)(C)C(NC(=O)Cn3nccn3)C2)ccnc2ccnn12 12487,c1(C(=O)NCC2(C)CC(NC(C3COC(=O)O3)=O)C2)cc(Cl)cc([N+](=O)[O-])c1 12488,c1(C(=O)NCCCC2N(C(c3c(C)ccs3)=O)CCC2)ccccc1OC1CC1 12489,CC1=C(C(N)NC(C2(n3cccn3)CCNCC2)=O)NC1 12490,C1(C2CCN(C(c3ccc(Cl)cc3)=O)C2)(NC(c2cn3c(n2)CCC3)=O)CC1 12491,CC(C)CC(CNC(c1cscc1Cl)=O)C(=O)NCCNC(=O)N(C)C 12492,C1(N(C(c2cc(CC)on2)=O)C)CCCN(C(=O)CC2C=CCC2)C1 12493,c1(C(=O)NC2C(CNC(Cc3cnc(C)s3)=O)CC2)cc(F)c(C)cc1O 12494,C1(C)(C(N2CCC(CCNC(C3(C(=O)NC)CCC3)=O)C2)=O)CCCCO1 12495,N1(C(CSCCOC)=O)CCC2(CC(C(=O)N(C)Cc3ccc(F)cc3)C2)C1 12496,N1(C(CCC(=O)OCC)=O)CCC(CO)(CNC(c2cncnc2CC)=O)CC1 12497,c1(OC)c(C)cc(C(=O)NCCC2CCC(NC(=O)C(O)P(C)(C)=O)C2)cc1C 12498,CC1CCc2nc(Cl)nc(N3CCCCC(NC(c4coc(Cl)c4)=O)C3)c2C1 12499,N1(C(C2N(C(C)=O)CSC2)=O)CCC12CN(C(=O)CN(C1CCCC1)C)C2 12500,C1(CC)CN(C)CCCN1C(C1COCC1NC(=O)C(F)C(C)(F)F)=O 12501,CC(C)CC(=O)NC(c1nocc1C(=O)NCC1CCN1C(C)(C)C)C 12502,Cc1cc(C(F)F)n2ncc(C(=O)NCC(C(C)C)NC(=O)C3=CCCC3)c2n1 12503,C1(C(N(C)CC2CC(F)C2)=O)CC2C=CC1N(C(C1CC=CC1)=O)C2 12504,C1(C(N(CCNC(=O)CNC=O)CC)=O)CCn2ncnc2C1 12505,N1(C(C2NC(C)C2)=O)CCCC2(CCC2)C1.CC1=C(C=O)CCC1 12506,c1(SC)c(C(=O)NC2CCC(NC(=O)C(N3CCCCCC3)C)C2)cccc1F 12507,c1(CC(C)NC(=O)C(N2CCC(N(c3ccccc3)C)C2)=O)ccccc1Cl 12508,C(=O)(C1CCc2cc(F)ccc21)N1CCC(CN(C(C2=NOC(C)C2)=O)C)CC1 12509,N1(C(C(=Cc2cccnc2)C)=O)CCCC(C)(NC(=O)COC(F)F)C1 12510,N1(C(C2N(CC)CCOC2)=O)CC2(C1)CN(C(=O)CC1CCCC1)CC2CO 12511,C1(NC(C2C3COCC23)=O)CN(C(=O)C=CCF)C2(CCC2)C1 12512,c1(CCNC(C=C(CNC(CCCOC)=O)C)=O)cccc(C)n1 12513,C1(NC(CC2CCC(=O)N2)=O)CN(C(=O)Cn2cnccc2=O)CC1CC1CC1 12514,c1(OC)c(Cl)cc(C(=O)N(CCC(C)NC(c2cc(C)oc2C)=O)C)cc1Cl 12515,N1(C(C(c2ccc(OC)cc2)CC)=O)CC(NC(c2occc2C)=O)CC(C)C1 12516,C(=O)(C(C)(C)C)NC(C)C(=O)NC(C1CCCC1)CNC(=O)C=Cc1ncco1 12517,c1(NC2CN(C)CC2O)ccc(S(=O)(=O)N2CCC3(CCOC3)CC2)cc1Cl 12518,CC1CC(NC(C2(C)CCN(C)C2=O)=O)CCN1C(c1cnc(F)c(Cl)c1)=O 12519,C(c1ccc(C)c(Cl)c1)=CC(=O)NC1CCCC(NC(CC=C=C)=O)C1 12520,N1(CC(=O)NC2CC(CCNC(C3(CO)CCCO3)=O)C2)CCCNC1=O 12521,c1(C(=O)NCC23C(CN(C(C4CC(=O)N4)=O)C2)C3)ccc([N+](=O)[O-])c(C(F)(F)F)c1 12522,CC(CCc1ccncc1)N=c1[nH]c2c(c(=NCCCCOC)[nH]1)COC2 12523,N1(C(C(C)C)=O)CCCCC(C(=O)NC(=O)C(C)Sc2ccccc2)C1 12524,CCCCCCCCC(=O)NC1CC1NC(c1ccc(C(C)(C)C)s1)=O 12525,C(=O)(C1=C(Cl)CCOC1)N1CC(NC(c2c(C)nccc2)=O)C(C(F)(F)F)C1 12526,N1(C(CC(C)O)=O)CC(CNC(=O)CC2C=CCC2)C(F)(CO)C1 12527,C1(NC(CN(C)C(N)=O)=O)C2CCC1N(C(=O)Cc1cncc(F)c1)C2 12528,N1(C(c2c(C)noc2)=O)CCC2OCCN(C(c3cc4cccn4cn3)=O)C2C1 12529,n1(CCCC)nnnc1C(c1ccncc1)NCCSCC1CCCC1 12530,N1(C(C(=Cc2ccc(Br)o2)C)=O)CC(NC(=O)C(C)C)C2(CCC2)C1 12531,c1(NC(C(C2CCN(Cc3cc[nH]c3)CC2)C)=O)cc(Cl)ccn1 12532,N1(C(CN(CCOC)C)=O)CCC(NC(C2CCCN2C(C)C)=O)C(F)(F)CC1 12533,N1(C(CC2CC(C)N(C(=O)CC(C)(C)C3CC3)C2)=O)CC2C3CCC(O3)C2C1 12534,c1(OC(C)C(=O)NC(C)CC2CN(C(C3CSCN3C)=O)C2)ccc(F)nc1 12535,N1(C(c2cc(C)oc2C)=O)CCC(NC(=O)Cn2ccnn2)C(CO)CC1 12536,c1(C(=O)NCC2CC(NC(=O)CSc3ccccn3)C2)cc2ccccc2o1 12537,C1(C(N(C)Cc2c(CNC(CSC)=O)cccc2)=O)CCOCC1(C)C 12538,C1(NC(c2cc(C)ncc2C)=O)CC2CN(C(C34CC(CO)(C3)C4)=O)CC2C1 12539,c1(N(C)CC2CCCN(C(C3(C)CC=C(C)CC3)=O)C2)nc2cc(C)ccc2o1 12540,CC(C)(CCNC(c1c[nH]nc1Cl)=O)C(=O)NC1C2CCC1CC2 12541,C1(OC)CC(NC(=O)C=CBr)CN(C(=O)CC2CCSCC2)C1 12542,C(=O)(CCCC(=O)N(C)C)N(CC)CC1CCCC1NC(=O)C=Cc1ccsc1 12543,Cc1cc(F)sc1C(=O)N(CCCCCCNC(c1ccn(C)c1)=O)C 12544,CC1(C(=O)NCC2CC(NC(c3cccc(CF)c3)=O)C2)CC2CC2C1 12545,Cc1ccc(C(=O)NC(C)CCNC(=O)C(C)(C)c2nccs2)s1 12546,N1(C(CCc2c(C)cccn2)=O)CCC(CNC(C2CCCOC2)=O)C(C)C1 12547,C=CCC(CC(C)C)C(=O)NCCCC(N1CC(O)CC1CN(C)C)=O 12548,C#Cc1ccc(C(=O)NCC(C)(C)CNC(C2CCC3CC2CO3)=O)nc1 12549,N1(C(C(CN(C)C)N(C)C)=O)CCCC(CC(=O)NCC2CC(C)(C)CO2)CC1 12550,C(C1=NOC2CN(C(c3cc4ccc(F)cc4o3)=O)CC12)NC(CC(C)C)=O 12551,CC1CN(C(=O)C(C)(C)C(C)NC(=O)C2=COCCC2)CCS1=O 12552,C(=O)(C(C)(C)C(C)(F)F)NCc1c(C(=O)NC(CC)C(C)(F)F)n(C)nc1 12553,c1(C(=O)NCC#CCNC(c2cc(CC)nnc2C)=O)cnc2ccnn2c1C 12554,N1(C(c2ccc(C)nc2C2CC2)=O)CCOC2(CCN(CC3CCC3)CC2)C1 12555,C1(C(=O)NC2CC(CNC(C3CC4(CCC4)C3)=O)C2)CC12CCCOC2 12556,C1(NC(CC(C)c2cnn(C)c2)=O)CC2CC1CN(C(C1C=CC=CC=C1)=O)C2 12557,CC1(C#N)CCN(C(=O)C(C2(O)CN(C(c3c[nH][nH]c3=N)=O)C2)F)C1 12558,N1(C(=O)OC(C)(C)C)CCCCCC1N=c1ccc(Br)n[nH]1 12559,CC1CN(C(=O)Cc2nc(C3CC3)n[nH]2)CC1NC(=O)CC1CC1 12560,CON1CCC(C(N2CC=CC(NC(C3CC4(C3)CC4(F)F)=O)C2)=O)CC1 12561,C1(C(=O)NC2CC3(C(NC(c4c(C)nc(CO)s4)=O)C3)C2)COC2CCCCC12 12562,C(=O)(C(C)(C)C(C)O)NCCn1cc(C(N(CCCC)CCOC)=O)nn1 12563,c1(COC(C)C)ccc(C(=O)NCC2(C)CCCN2C(C2CC(C)=NO2)=O)cc1 12564,N1(C(C(C2(C)CC2)NC(CCCSC)=O)=O)CC2CCC(C1)C2C#N 12565,C#CCC(C(=O)NCCCSC)N(C(=O)C(=Cc1cn[nH]c1)C)C 12566,C1(SC)CCN(C(=O)CCOC2CN(C(=O)C(C)CCN(C)C)C2)C1 12567,CN1CCN(C(C2CCCC2)=O)C(C2CC2)C1.c1(CN2C(=O)C2)sccc1CO 12568,C(=O)(C(C)S(=O)(=O)C(C)C)NCC(CNC(C(CC)(CC)CC)=O)C 12569,C1(OC)(CNC(=O)N(C(C)C)Cc2cccc(N3CCCCC3)c2)CCCSC1 12570,c1(CC(=O)NCCN(C(c2cnccc2Cl)=O)CC)ccc(OC)c(C)c1 12571,C1(C)(N(C)C)CCCN(C(=O)COCCNC(=O)Cc2ccnn2C)C1 12572,N1(C(C2N(C(C(=Cc3cn[nH]c3)C)=O)C(C)CC2)=O)C2CCC1COC2 12573,CC1CCCC(O)(C(=O)NCCNC(c2ccc3cc[nH]c3n2)=O)CC1 12574,c1(C(=O)NC2C(NC(c3c(C)cco3)=O)CC2)cc(F)c(F)c(O)c1F 12575,c1(C(=O)NCC(C)NC(C(CC)n2cncn2)=O)cnc(C)n1C 12576,CCCCC(S(=O)(=O)NC(=O)C(c1ccc(Br)nc1)(C)C)c1ccccc1 12577,CC(C)CC(C)(CNC(c1cc(Br)n[nH]1)=O)NC(c1ccc(Cl)o1)=O 12578,Cn1cc(C(F)=CC(=O)OCC(C2CCC(F)C2)=O)cn1 12579,N1(C(c2c(CC)ncs2)=O)CCCC(CO)(NC(=O)CSCC(=O)OCC)C1 12580,N#Cc1ccc(NCCCNC(c2ccc(CC3CCC3)cc2)=O)c([N+](=O)[O-])c1 12581,c1(C(N2CCN(C(=O)Nc3cccc(C)c3)C3C2C3)=O)nncc2c1CCCC2 12582,N1(C(c2c(SC)cc(F)cc2)=O)CCN(C(=O)CC2COC(C)(C)C2)CCC1C 12583,c1(CNC(CC=C)=O)nc2c(s1)CCN(C(=O)CS(=O)(=O)N1CCOCC1)C2 12584,C1(F)(C(=O)NCC2CC(NC(Cc3cnc(C)o3)=O)C2)CCCOC1 12585,C(CCC(=O)NC1CCC(NC(=O)C(C)(O)C2CCCCC2)C1)N(C(C)=O)C 12586,c1(OC)nc(Cl)ccc1C(N1CCC(NC(c2ncccc2C)=O)CC1C)=O 12587,N1(C(CCCn2cc(CC(C)(C)CO)nn2)=O)CC2CC2(CN2CCCC2)C1 12588,CCCCCC(CC)C(=O)NCc1c[nH]nc1C(=O)NCC(=O)OCC 12589,N1(C(c2cc(OCC)n[nH]2)=O)CCC2(C(=O)NC(C3CCOC3)C)CC2C1 12590,N1(CC(=O)NC2C3CC2N(C(c2snc(O)c2Cl)=O)C3)CCCCCCC1=O 12591,c1(C2(CN(C(F)CF)C3CC3)CCCC2)ccc(Cl)cc1 12592,C=C(C)C(C)(C)C(=O)NC1COCC1NC(=O)CCC(=O)c1ccncc1 12593,N1(C(C(CC)OC)=O)C2CCC1CC(CNC(c1n[nH]cc1C(C)(C)C)=O)C2 12594,C(=O)(N1CCCc2ccnn21)C1C2(CCN(C(c3cc(OCC)no3)=O)C2)C1 12595,CC(C)CC(C)(CNC(c1c[nH]ccc1=O)=O)NC(C1CN(C)CC(C)O1)=O 12596,C(N=c1nc2c(c[nH]1)COCC2)C1(NC(c2ccc(C)c(F)n2)=O)CCCC1 12597,C1(NC(C23CCC(F)(CC2)CC3)=O)CN(C(C2CC3CC3C2)=O)C2CCCCC12 12598,C(CCS(=O)(=O)c1ccc(F)cc1)NC(=O)NCC1(C)CCCC1O 12599,c1(CC(=O)N(C2CC(NC(c3cccs3)=O)C2)C)cccc(N2CCCCC2)c1 12600,C=CCC(C)(C)C(=O)NCC(C)(C1CC1)NC(c1ccnc(S)c1)=O 12601,C1(NC(Cn2c(C)ccn2)=O)CS(=O)(=O)C2CN(C(=O)CC3CCCOC3)CC12 12602,Cc1nn(CC(=O)NC2CCCC2CNC(c2cncc(N)n2)=O)cc1[N+](=O)[O-] 12603,C1(C(N2CCC(O)(C(C)NC(=O)COCCF)C2)=O)CS(=O)(=O)CC(=O)N1 12604,c1(NCC2C(C)CCN(C(=O)C(C)(C)CF)C2)ncnc2cnccc12 12605,C1(C(N(C)CCNC(c2ccc3c(c2)OCC3)=O)=O)C2C3CC4C1C1C2CC3C41 12606,N1(C(c2c(C)cnnc2)=O)CCC2(CC2)CC1C(=O)NCc1ncn(C2CC2)n1 12607,C1(C)(CNC(CC=C)=O)CN(C(c2coc(COC)n2)=O)CC1C 12608,N1(C(c2ccn(CC)c2C)=O)CC2(C1)CN(C(c1cc(C(F)F)[nH]n1)=O)C2 12609,C(=O)(C(F)(F)CCC(=O)NCCc1cnc2n1CCCC2)OC(C)(C)C 12610,CC(CC(F)(F)F)C(=O)N1CC2(CC2)CC1CNC(=O)CC12CCCC1C2 12611,C1(NC(c2c[nH]nc2Br)=O)CN(C(c2cc(CO)[nH]n2)=O)CC1O 12612,c1(NC(COC(C(C(C)C)CC2CCCCC2)=O)=O)cccc2c1nc(O)n2C 12613,Cc1csc(C(=O)N(C)CCOCCNC(=O)C(N2CCN(C)CC2)C)c1Cl 12614,c1(C(=O)OC(C)C(=O)N2CC(CC3CC3)C2)cc(Br)cs1 12615,N1(C(CCCc2ccc(CCC)cc2)=O)CCCC2(NC(=O)CCOCC)CC12 12616,N1(C(C2(C3N(C(c4cc(C(C)C)[nH]n4)=O)CCC3)CC2)=O)CCC(C)(C#N)CC1 12617,C1(C(CNC(CSC)=O)(C)O)CCCN(C(c2cnc(C3CC3)[nH]2)=O)C1 12618,c1(C(N(C)CCN(C)C(C2CCC3C2C3(F)F)=O)=O)cc2ccccc2[nH]1 12619,C12(CNC(=O)NC3CC(C)(C#N)C3)CCC(N=[N+]=[N-])(CC1)C2 12620,C1(C(=O)NCCCOC=C)CC12CCN(Cc1cc(O)c(O)c(O)c1)CC2 12621,Cc1ccn2ncc(C(N3CCN(C(=O)CN(C)C)CC(CO)C3)=O)c2n1 12622,N=c1[nH][nH]c2cc(C(N3CC4CC3C4C(N3CC4CC4C3)=O)=O)ccc12 12623,CC(C)(CCCO)NC(C1CSCCN1C(C1CC(=O)C1(C)C)=O)=O 12624,c1(C(=O)NCCN(CCC)C(c2c[nH]nc2S(N)(=O)=O)=O)cc2n(n1)CCOC2 12625,C1(C(=O)NCC(C)(C)NC(CN(C2CC2)CC)=O)CCCC(F)C1 12626,c1(C(=O)NC2CC(N(C)C)C2)ccnc(CNC(C2(N3CCCC3)CCC2)=O)c1 12627,c1(NC(CC)=O)cncc(C(N2CC=CC2CNC(=O)C=C2CCC2)=O)c1 12628,CN1CC(CNC(=O)CC=CCNC(=O)CC2CCC(C#N)C2)CC1=O 12629,C12(NC(C3OCCN(C(C)C)C3)=O)CC(CNC(=O)C(C)C(F)F)(C1)OC2C 12630,N1(C(COCCCOC)=O)CC2C(NC(=O)CNS(=O)(=O)N(C)C)C2C1 12631,C1(CNC(NC(C#C)CCC)=NCCC=C)CCC2(CCOCC2)O1 12632,C(=O)(CC1=CCOCC1)NC(COC)CC(=O)N1CC(OCCSC)C1 12633,C(C(=O)NCCC1(C)CCOC1)(C(C)(C)O)NC(C1CCC(CC)O1)=O 12634,c1(C(=O)NCC(C2CCCC2)OC)cc(CNC(=O)CCCc2cnn[nH]2)on1 12635,CCCCCCCC1CN(C(=O)CCCn2cc(C(C)(C)CO)nn2)C1.C1C(=O)O1 12636,C1(NC(COC2(C)CCCC2)=O)CCN(C(C2CN(C3CCC3)C2)=O)C1C(C)C 12637,N1(C(C2C(C)C2(F)F)=O)CC(NC(=O)CONC(=O)OC(C)(C)C)C(C(F)F)C1 12638,C1(C(=O)NC(c2n(C(C)C)ncn2)C)CCN(C2COC2)CC1 12639,C(C(O)CC(=O)NC1C(CNCCNC(c2ccccc2F)=O)C1(C)C)N(C)C 12640,O=C1CCC(C(=O)NCCOC2CN(C(c3ccccc3C(F)F)=O)C2)CN1 12641,c1(C(N2CCC(NC(c3cnc(C)s3)=O)(CO)C2)=O)cn(C)c(C)cc1=O 12642,Cc1cc(F)sc1C(=O)NC(C1CCN(C(C2CC2(C)C)=O)C1)C 12643,N1(c2ccc(CC)nc2OC)CCN(C(C)=O)CC(C)(C)C1 12644,c1(C(N(C2CN(C(c3cnc(C(C)O)s3)=O)CC2O)C)=O)nccc2ccsc12 12645,Cc1cc(Cl)c(NC(c2cc(F)c(Cl)cc2O)=O)cc1O 12646,CC(C)(C#CC(=O)NCC(C)(O)C1CC1)CNC(=O)CN1CCOC1=O 12647,C1(C(=O)NCC2(NC(c3cn(CCOC)nn3)=O)CC(OC)C2)CCCCC1F 12648,CC1COc2ccc(C(N3CC4CN(C(=O)CC5=CCCC5)CC4(C)C3)=O)cc21 12649,Nc1c(F)ccc(F)c1C(=O)NCC1CCCC1NC(=O)CN1CCOCC1 12650,C(=O)(CCCCCC(C)O)N(CC(CNC(C(C)NC(C)=O)=O)O)C 12651,Cc1cc(Cl)c(Cl)cc1C(=O)OCc1ncoc1C(C)C 12652,C(N=c1[nH]c(NC2CCCn3ncnc32)nc2ccccc12)c1cc(C)ncn1 12653,S(=O)(=O)(c1cnccc1COCC(C)C#N)N(CCOC)Cc1ccc(Cl)cc1 12654,c1(CNC(=O)C(c2sncc2Br)N2CCCC2C2CC2)ccccc1 12655,N1(C(CCCCCN(C)C(c2cncnc2)=O)=O)CC2CCC1C(CO)C2 12656,c1(C(=O)NC2(CC=C)CCN(C(=O)CC(C)OC)C2)cc(C)cc(Br)c1 12657,C1(C(N(C)CC2(O)CN(C(=O)C=Cc3cc[nH]n3)C2)=O)COCCN1C 12658,c1(C(N(CC(CC)NC(=O)CCC2CC=C(C)CC2)CC)=O)cccc(C)c1F 12659,N1(C(C(c2ccn(C)c2)C)=O)CC2CCCC(N(C(=O)CN(C)CCO)C)C2C1 12660,c1(NC(C)=O)c[nH]c(C)c1C(=O)NCC=C1CCN(C(=O)C=C2CC2)CC1 12661,CN1CCCC2CN(c3cc(C(=O)O)c4c(c3)CCCC4)CCC12 12662,CCN=c1[nH]cc(C(=O)NC2CC(Cn3cc(CCC4CCCC4)nn3)C2)s1 12663,N1(C(CCn2ccc(C)n2)=O)CCC(C)N(C(=O)CC2COCC2O)CC1 12664,C(=O)(C1=C(Cl)CCOC1)N1CCCC(C)C1CN=c1[nH]nc(Cc2ccccn2)o1 12665,N1(C(C(C)(C)SC)=O)CCN(C(c2n[nH]c3c2CCC3)=O)C(C2CCC2)C1 12666,c1(C(N(CCCC(=O)NCC(C)N(C)C)C)=O)c(O)cccc1F 12667,c1(C(=O)NC(C)CN(C)C(c2ccc(N)cc2)=O)cc2ccc(O)nc2s1 12668,N1(C(c2cccc(N)c2Br)=O)CCOCC(F)(CNC(c2cnc[nH]2)=O)C1 12669,CCC(CN=c1cc(NCC(N2CCCCCC2)C)nc[nH]1)OC 12670,CC#CCCC(=O)NCC(C1CCOC1)NC(=O)Cc1cnn(C)c1C(F)F 12671,C1(NC(CC2C(OC)COCC2)=O)COC2(C1)CN(C(C1(C)CS(=O)(=O)C1)=O)C2 12672,c1(C(N2CC(OC)C(CNC(=O)C(C)CC3CCCC3)C2)=O)cc2n(n1)CCO2 12673,CC(C)CCC(C(=O)NCC(C)(O)CO)NC(c1cn(C)cn1)=O 12674,c1(NC(CC)=O)ccc(C)c(C(=O)NCCc2ncc(Br)cn2)c1 12675,C1(NC(C2CC(C)OC2)=O)CCCC12CCN(C(=O)CCC(C)(F)F)CC2 12676,c1(CCC(=O)NCC(C)(CO)NC(C2(OC(C)=O)CC2)=O)nnc(S)n1C 12677,N1(C(Cc2ccc(C(CC)=O)cc2)=O)CCC2(C1)CN(C(c1ccsc1)=O)C2 12678,c1(C(N2CCN(C(C3CCC(=C)CC3)=O)C(C)C2)=O)cc2ccccc2nc1O 12679,c1(NC2CC(CNC(CCC(=O)N(CC)CC)=O)C2)ncn(C)c(=O)c1Br 12680,Cc1cnn2ccc(C(N3CCC(C(C)NC(=O)CP(C)(C)=O)C3)=O)nc12 12681,C1(SC)CN(C(c2cc(C)ccc2Cl)C(=O)NC2CCCC2)C2(CCC2)C1 12682,N1(C(C(CC)O)=O)CCC(C2(NC(=O)Cn3cccn3)CCC2)CC1 12683,C(=O)(C(O)P(C)(C)=O)NCC(CN(C)C(c1cncc(C(F)(F)F)c1)=O)(C)C 12684,N1(C(C(CCOC)OC)=O)CC(CO)C2(C1)CN(C(=O)CN1CCS(=O)CC1)C2 12685,C(=O)(C(CNC(=O)CC(F)(F)F)C(C)(C)C)NCc1cn(CC=C)nn1 12686,CC(C)S(=O)(=O)c1cccc(C(=O)NC2COCC2CNC(=O)CN(C)C)c1 12687,c1(C(=O)NC23CC(CNC(CC4CCCN(C)C4)=O)(C2)C3)ccc(F)cc1Cl 12688,C(=O)(C(F)(CNC(C1CCC(C)O1)=O)C(C)C)NCc1onc(COC)n1 12689,Cn1cc(-c2n[nH]cc2NC(c2nc(C3CC3)cs2)=O)cn1 12690,C(CCCCC(C(=O)NCC1CCOC1)N1CCn2cccc2C1C)OC 12691,O=S(=O)(c1ccccc1N1CCc2sccc2C1)N1CC(OCC(F)F)C1 12692,C(=O)(CCCC(F)(F)F)N1CCC(C)C(NC(=O)C(c2ccccc2F)(F)F)C1 12693,C1(CC)CN(C(C2CC(C(C)(C)C)C2)=O)CCN1C(=O)Cn1nc(O)ccc1=O 12694,c1(C(=O)NCC(C)CNC(=O)C(O)C2CCC2)cccc(S(=O)(=O)CF)c1 12695,C12(C(=O)NC3CCN(C(Cc4cn(CC)nc4)=O)CC3O)CC1Cc1c[nH]nc12 12696,C(N=c1[nH]c(=NC(C)c2nc[nH]n2)[nH]c2ccc(Cl)cc12)C1(COCC)CC1 12697,c1(N(C)CCOC(F)F)nc(=NCc2cc(Br)ccc2C)[nH]c2c1CSC2 12698,Cn1cc(C=CC(=O)NCCC2(C(=O)NCC3CC3C3CC3)CCC2)nn1 12699,C1(C(C)NC(C(CC)NC(N)=O)=O)CCN(C(=O)CCCC2CC2)CC1 12700,C1(COC)(CNC(=O)CCC2CCOCC2)CCN(C(C2CC(=O)N(C)C2)=O)C1 12701,C#CCC(C)(C)C(=O)NC(CNC(=O)C(C)n1ccnc1)CCOC 12702,C1(NC(c2[nH]c(=N)sc2)=O)CN(C(=O)C=CBr)CC12CCS(=O)(=O)CC2 12703,C=C(F)CN=C(NCc1cccc(NC)c1)NC1CC(=O)N(c2ccccc2)C1 12704,N1(C(C(C2(O)CN(C(C(C)OC(C)=O)=O)C2)F)=O)CCc2ncn(C)c2C1 12705,c1(C(=O)OC)c(NC(=O)CCC(C)(C)OC)sc2c1CCC(C)C2 12706,C(=O)(C(C(F)(F)F)C(F)(F)F)N1C(C(N2CC(C)(C)c3c2cccc3)=O)CSC1 12707,C(=O)(C(C)(C)C(O)C(C)C)NC1CC=C(C(=O)NC2N(C(C)=O)CCC2)C1 12708,S(=O)(=O)(c1ccncc1)N1CCC(C)(C(=O)Nc2c(N(C)C)cccc2)C1 12709,C1(NC(c2cnoc2C2CC2)=O)COCCC1NC(C1CC1C(F)(F)F)=O 12710,CCC(C(=O)NC(CNC(c1cc(C2CC2)ns1)=O)Cc1ccccc1)NC(C)=O 12711,C1(C2CN(C(=O)C(Br)=C(C)C)C2)(NC(CC2ON=C(CC)C2)=O)CC1 12712,c1(C(=O)NCC(CC)NC(c2cc(N(C)C)ccn2)=O)ncc(N)cc1C 12713,c1(C(=O)NC(c2nocc2C(=O)NCCCC2(C)CC2)C)cccnc1O 12714,c1(C(N2CC=CC(NC(c3ccc(COC)s3)=O)C2)=O)nc(C2CC2)ncc1Cl 12715,C1(NC(C2C(C)N(C)CC2)=O)CCC12CN(C(=O)CCCc1ccccc1)C2 12716,C(CC(=O)N=c1cc[nH]cc1)N1C(C)CC(c2ccc(OCC)cc2)C1 12717,C1(CCNC(c2cnn(CCC)c2C)=O)CCN(C(=O)CN(C)CCO)C(C)C1 12718,C1(C(N2C(C)CC(NC(C3CC3C3CC3)=O)CC2)=O)CCCCC1N=[N+]=[N-] 12719,CCCC(C)(C)CC(=O)N1CC2CCC2(CC(=O)NCc2cc(C)ncn2)C1 12720,c1(C(=O)NC(CNC(C(F)=CC)=O)CC(F)(F)F)cc(=O)n2nccc2[nH]1 12721,CN=c1ncc(-c2nc(C(N3CC4CCC(C3)O4)=O)cs2)c[nH]1 12722,C1(NC(c2cnn(C3CCC3)c2)=O)CN(C(c2ccsc2Cl)=O)CCC1CO 12723,N1(C(Cc2scc(C)c2)=O)CCC(C)(NC(c2coc(C(F)(F)F)c2)=O)C1 12724,C1(NC(C2CC(C)(C)C2)=O)CC(NC(c2coc(Br)n2)=O)C12CCOCC2 12725,N1(CC2OCC(CO)C2)CCc2cc(C(F)(F)F)ccc2C1 12726,C(=O)(CC(O)CC(C)C)NCC(CCC)C(=O)NC1C=CC(C(=O)OC)C1 12727,C(=O)(C1c2c[nH]nc2CN1C(=O)CCCn1ccnc1)NCC(N1CCCC1)C 12728,c1(C(=O)NCCOCCC(=O)N(C(C)CC)C)ccc(C(F)F)o1 12729,c1(NC(C)=O)ccc(Cl)c(C(=O)NCC(C)NC(=O)C(c2ccccc2Cl)O)c1 12730,c1(C(=O)NC2CC(C)(NC(c3ccnc(C)n3)=O)C2)cc(N)c2ncccc2c1 12731,c1(C(=O)NCC2N(C(C3C(=C)C3)=O)CCC2)cc(F)cc(Br)c1Cl 12732,C(=O)(C1=CCC(NC(=O)CCC2(C#N)CCC2)C1)NCC(=O)NCCC 12733,C1(CNC(=O)NCC2CCC(C(=O)OC)C2)CCCC(C)(C)CC1 12734,N1(C(C(CCC)O)=O)CCC(C(F)(F)F)CC1CNC(c1nn(C)cc1SC)=O 12735,Cn1ccn2ncc(C(N3CC4C(NC(=O)C=Cc5cc[nH]c5)C4C3)=O)c12 12736,C1(NC(C(CSC)O)=O)CC2CC1CC2C(=O)NC(CCO)C(C)(C)C 12737,C=CC(CC)CC(=O)Nc1c[nH]nc1-c1cnn(C)c1.C12CN(CC1C=C)C2=O 12738,c1(C(N2C(C)CC(CNC(=O)C=Cc3cc[nH]c3)C2)=O)cnc2n1CCS2 12739,Cc1nn(C)c2ncc(C(=O)NCCCC(C)NC(c3nc(=O)n(C)[nH]3)=O)cc12 12740,C(=O)(C1Cc2ccc(Cl)cc21)NC(CCCC)CNC(c1cc(C2CC2)[nH]n1)=O 12741,C(=O)(C(C)(C)C1CCCO1)N(CCCN(C(=O)Cc1cccnc1)C)C 12742,c1(OC)cc(C(=O)NC2CN(C(C3CC34CCCCC4)=O)C2)c2ccccc2c1 12743,c1(CCC(=O)NC(C)CNC(C2(CC3CCC3)CC2)=O)ccc(Br)s1 12744,C(=O)(C1=CCCC1P(C)(C)=O)N1CC(C)C(CNC(=O)C(C)(C)CSC)C1 12745,c1(NC(=O)NCCN2CC(F)C(F)(c3ccccc3)C2)ccc([N+](=O)[O-])cc1O 12746,C(=O)(C(CNC(=O)CC1CCOC1)N(C)C)N1CC(OC)C1 12747,N1(C(C2(CC)COC2)=O)CCC2(CC1)CC2C(=O)NOCC(O)CO 12748,c1(C(=O)NCC2CCC(NC(c3c(CC)non3)=O)C2)nccc2c1NCCC2 12749,N1(C(c2cc(Br)ccn2)=O)CCOC(CNS(=O)(=O)CCBr)C1 12750,C(=O)(C1=Cc2ccccc2C1O)N1CC(O)(CNC(c2cncc(CC)c2)=O)C1 12751,CC1(C(=O)NCCN(C(=O)CSC2CC2)Cc2ccccc2Cl)COCCO1 12752,C(=O)(C(C)C(F)(F)F)N(CC=CC(=O)N(C)Cc1c(CC)noc1)C 12753,CC1(C)NC(=O)CC1C(=O)NCC1(CNC(C2(C)CC3C=CC2C3)=O)CC1(F)F 12754,CCC(CC)CC(F)C(=O)N1CCC2(CC(NC(=O)CC3(C(F)(F)F)CC3)C2)C1 12755,C#Cc1ccc(C(=O)NC(CCN(C)C)C(=O)NCc2nnc(C)n2C)cc1 12756,C=C(Br)CC(=O)NC(CO)C(C)NC(=O)C=Cc1cnc[nH]1 12757,c1(OC)cscc1C(=O)NC(CNC(C1CC1c1ccccc1)=O)C(C)C 12758,CCCC(CCCNC(C1CC1(F)F)=O)NC(=O)CCCCc1ccccc1O 12759,c1(CC)ncc(C(N2CC(C(=O)NCc3nn[nH]c3C3CC3)C(C)C2)=O)cn1 12760,C1(F)(C(=O)NCC2(F)CC(CNC(CC3(C)OCCO3)=O)C2)CCCCC1 12761,CCCC(CC)CCC(=O)N(C1CCN(C(=O)CC(C)N(C)C)CC1)CCCC 12762,CC1=CCC(C)(C(=O)NCCC23CCC(C2)N(C(c2csc(C)c2N)=O)C3)CC1 12763,N1(C(c2c(CC)con2)=O)CCC(C2CC2)(NC(C2CC2(F)F)=O)C1 12764,C1(NC(c2nc(CC)oc2C)=O)COC2(CNC(=O)C(C)C3CC3)CC1C2 12765,C1(CCN(C(=O)C(O)Cn2cncn2)C)CCCCN1C(=O)CCC#N 12766,c1(C(=O)NCCN2CCCN(C(C3C(OC)C3)=O)CC2)cccc2c1ncn2C 12767,Cc1cccnc1CN1CCC1CNC(c1ccc(CO)s1)=O 12768,c1(OC)ccc(C(=O)NCc2cc(C(F)(F)F)nn2C)c2cccnc12 12769,C1(O)(CNC(c2cc(OCC)n[nH]2)=O)CCN(C(=O)CC2CCCC2O)C1 12770,C1(C(=O)NCc2ncc(C)nc2)CC12CCN(C(=O)CCc1cncn1C)CC2 12771,C1(NC(c2ccc(Cl)cc2)=O)CN(C(=O)C(O)Cc2cnc[nH]2)CC1CC1CC1 12772,CCC(CC(=O)NC1CCN(C(C2CC23CCCCC3)=O)C1(C)C)CC(F)(F)F 12773,c1(C(=O)NC(C)C(C)NC(c2c(F)cncc2Cl)=O)cc(F)cc2cc[nH]c12 12774,C1(N(C(COCC(=C)C)=O)C)C2CN(C(C3(C(C)C)CNC(=O)C3)=O)CC12 12775,N1(CC)CCN(CC(=O)NCC(CO)NC(=O)Cc2ccco2)CC1 12776,N1(C(C=CCNC(c2c(C)con2)=O)=O)CCC2CC2C1 12777,c1(C(=O)NCC(CC(=O)Nc2c(C)noc2)C)cnc(C)c(C)c1 12778,C(=O)(C(C)CCC(C)(C)C)N1CCC(NC(c2ccc(C)cc2)=O)(CF)C1 12779,c1(N(C)Cc2c(C)ccnc2)nc(N(C)CC2CC(F)C2)nc2ncn(C)c12 12780,c1(C(=O)NC2(C)CC2)cn2c(n1)CCN(C(=O)Cn1cc(S(C)(=O)=O)cn1)CC2 12781,C(=O)(C1=CS(=O)CCC1)N(CC(C)NC(c1ncccc1F)=O)C 12782,C1(C(C)(C)CNC(=O)CNC(N)=O)CCCCN1C(=O)C=Cc1ccco1 12783,C(=O)(CCC(=O)NC1CC(c2ccccc2)(CNC(=O)C=CS(C)=O)C1)NC 12784,Cc1cnc(C)c(C(=O)NCC(C)CN(C)C(c2sc(F)cc2Cl)=O)c1 12785,CC1CCC(O)(CN(C)C(C2CCN(C(c3ns[nH]c3=O)=O)C(C)C2)=O)CC1 12786,c1(NC(C2C(Nc3ncc(SC)cn3)C2)=O)c(C)ccc(I)c1C 12787,c1(OC)nccnc1CNC(C1(F)CN(C(=O)CC2CCCNC2=O)C1)=O 12788,C1(NC(=O)CN2CCSCC2)CCCC(NC(c2cccc(C(F)F)c2)=O)CC1 12789,C1(C#N)(C(=O)NC(CCC#C)C(=O)O)CCc2ccccc2C1 12790,c1(N(C)CCc2ccc(F)cc2)nc2cc[nH]c2c(=NCC2(C)CC3(CC3)C2)[nH]1 12791,O=C(C1=C(Cl)CCOC1)N1CCCC2CC12 12792,C(C)(CCCCNC(=O)CCC1CCC1)NC(CSCCC)=O 12793,C1(C(=O)NCC2N(C(CCc3c(C)noc3Cl)=O)CC2)CC1C1(C)CCOCC1 12794,C1(O)(CNC(C2(N(C)C)CC2)=O)CCN(C(c2cc(Cl)ccc2F)=O)CC1 12795,c1(C(=O)NCC=CCNC(C2(CCC)CCOCC2)=O)cccc2oc(C)cc12 12796,CCC(C)(CNC(c1ccc(C(C)=O)[nH]1)=O)C(=O)NCC1CC(=O)N(C)C1=O 12797,CC(CNC(=O)CC=CCNC(=O)CCn1ccnc1)CN1CCCC1 12798,C(=O)(C(C)(C)C(F)(F)F)NC1C(NC(c2cccc(SCCC)c2)=O)C1 12799,CCS(=O)(=O)CCNC(C1(CNC(C2CC2(F)Cl)=O)CC(=C)C1)=O 12800,c1(C(=O)NC(CNC(CS(=O)(=O)NC)=O)C2CCC2)nn(C)c(Cl)c1Cl 12801,c1(CNC(C(CCOC)NC(=O)CSC(F)F)=O)cccc(F)c1F 12802,C1(C(=O)NCCN(CC(C)O)C(c2[nH]nnc2C2CC2)=O)CC(F)C(=O)N1 12803,c1(CNC(=O)Cc2ccc(CC3(F)CCNCC3)cc2)ncnc2ccccc12 12804,N1(C(C(N2CCOCC2)C)=O)CC2CC(NC(=O)C=Cc3cccnc3)CC1C2 12805,c1(C(=O)NCCCN(C(=O)Cn2nnc(=O)[nH]2)C)ccc(SC)o1.C(=O)(NC1CC1)N 12806,C1(C(N2CCC(CCN(C)C)C2)=O)CN(C)CCN1C(c1ccccc1Cl)=O 12807,C1(O)(C(N(c2cccc(C)c2C)CCC#N)=O)CCCC(C)(C)CC1 12808,c1(C(N2CCC(NC(c3ccc(OC)nc3)=O)C2C)=O)cc(Cl)cc2c1OCC2 12809,C1(C(=O)NC)CCN(C(C2COC(CNC(C3CN(C(C)=O)C3)=O)C2)=O)C1C 12810,C1(NC(CCCCC=C)=O)CN(C(=O)C(CC)N2CCCC2=O)CC(F)(F)C1 12811,N1(C(CCCc2[nH]c(=N)sc2)=O)CCC2CCCN(C(=O)CCCC(F)F)C2C1 12812,c1(C(N2CCC(CNC(CC(CC)C3CCC3)=O)CC2)=O)nnc2ccccn12 12813,C(C(C)N=c1nc(N(C)Cc2cc(F)ccc2F)c2sccc2[nH]1)c1ccc(C)s1 12814,N1(C(CCCC(C)NC(c2c(OC)n[nH]c2)=O)=O)CCCC12CCOC2=O 12815,N1(C(C=CCN(CC)CC)=O)CC(NC(c2nccc(OC)c2N)=O)CC(F)C1 12816,CC1CCCCC1(CNC(c1ccc(=O)n(C)n1)=O)NC(=O)CCNC(=O)CO 12817,C(CN=C(NCC(C)(C)OC)N1CCc2c(F)ccc(F)c2C1)OCC=C 12818,N1(C(CS(CC)=O)=O)CC2CCC1(CNC(=O)C#CC(C)(C)C)CC2 12819,N1(C(c2cc(CCOC)on2)=O)CC(C)CN(C(=O)CC2CCSC2)CC1C 12820,C1(CC=C)(NC(c2nncs2)=O)CCN(C(=O)C(CO)N(C)C)C1 12821,C(=O)(C#CC1(C)CCCO1)N(CCCCN(C)C(C1(C)CC1Br)=O)C 12822,c1(C(N(C)CC2CCN(C(Cc3c(C)ccs3)=O)CC2)=O)csc2ccncc12 12823,N1(C(c2cc(CC)oc2C)=O)CC2CCC1CN2C(=O)CCC1CCN(C)C1 12824,Cc1nnc2n1C(C(=O)NCCCC(C)NC(c1sccc1Cl)=O)CC2 12825,Cn1cc(Cl)c(C(=O)NCC(C)(O)CNC(c2ccc(OCC(F)F)cn2)=O)n1 12826,CC1(C)CC(C(=O)NC2CC3CCCC3C2)CN(C(=O)CCN2CCCCC2)C1 12827,C1(NC(=O)CCCn2cccn2)CS(=O)(=O)CC1NC(C12CCCN1CCC2)=O 12828,N1(C(C(CCSC)NC(C2CN(C)CC(C)O2)=O)=O)CCn2nccc2C1 12829,C(=O)(C(F)CCC(C)(C)C)NCc1c(C(=O)Nc2c(C)csc2)nco1 12830,CC1ON=C(C(=O)NC(C2CCCN2C(c2csnn2)=O)(C)C)C1C 12831,CCCCCC(O)CC(=O)NC1CCCC1NC(C1(CO)CC1)=O 12832,C1(C)(CNC(C(CC)Sc2nc(=N)[nH][nH]2)=O)CCN(C(=O)OC(C)(C)C)CC1 12833,CCC(CC)CC(F)C(=O)NCCC1(O)CCN(C(C2OCCC2CC)=O)CC1 12834,c1(C(=O)NCC2C(Nc3nccc(C)n3)CCCC2)ccc(C)c2c1CCC2 12835,N1(C(c2c(OCC)scc2)=O)CCN(C(C2CCC(CN(C)C)C2)=O)C(CC)C1 12836,c1(OC)ccc(C(CNC(=O)Cc2nnc(C)n2C)NC(=O)C(O)C(C)C)cc1 12837,C1(O)(COC)CN(C(C2CCC2CNC(=O)C(C)c2ccco2)=O)C1 12838,CCC(C(=O)NCc1cc(Cn2cc(Cl)cn2)cs1)c1ccccc1 12839,Cn1nc(C(=O)Nc2nnc(Cn3ccccc3=O)s2)c2ccccc2c1=O 12840,C1(CN(C(CCOC)=O)C)CCCCN1C(c1sccc1OC)=O 12841,C(C1CCCCCC1)=CC(=O)NCC1(F)CN(C(CCC(=C)Cl)=O)C1 12842,C=CC1CN(C(c2cnc(C)c(CC(C)C)c2)=O)CC1NC(=O)C#CC1CC1 12843,CC(C)CC(O)C(C)C(=O)NCC1CN(C(=O)CN(S(=O)(=O)c2cccs2)C)C1 12844,CC1CCCC=C1C(=O)NCC1CCC1NC(c1ccn(C(C)(C)C)c1)=O 12845,c1(C(=O)NCC2N(C(CC(c3scc(C)c3)O)=O)CCC2)c(C)coc1C 12846,C(=O)(C1=NOC(CNC(=O)CCOCC)C1)NCC(=C)F 12847,N1(C(C)C(=O)NCCC2CC(NC(C3(C4CC4)CC3)=O)C2)CCCCC1=O 12848,c1(C(C)C)ccoc1C(=O)NC12CC(NC(=O)C(F)C3CCCC3)(C1)C2 12849,c1(CNC(C(C)O)=O)ccc(CNC(C2CCCN2Cc2cccnc2)=O)cc1 12850,c1(CC)nc(Cl)c(F)c(=NCCCCNC(=O)C(Cc2ccccc2)CC)[nH]1 12851,c1(C(N2C(CNC(C(CSC)O)=O)CC(C)(C)C2)=O)ccc2oc(=N)[nH]c2c1 12852,N1(C(C(C2CC(C)(C)C2)OC)=O)CCC2(CCC(NC(=O)CC(F)(F)F)C2)C1 12853,C=CCCC(CC(C)C)C(=O)N(CC(C)NC(C1CCOC(C)C1)=O)C 12854,c1(C(=O)NC(CCCC=C)c2ccccc2)[nH]cc2c1CCCC2 12855,N1(C(C2(F)CN(C(C(C)OCCC=C)=O)C2)=O)C2CCC1CC(=O)NC2 12856,c1(C(N2C(CN(C(CN(C)CCO)=O)C)COCC2)=O)cc(O)c2ccoc2c1 12857,C(=O)(C#CC1(C)CC1)NC(C)C(=O)NCC(CNC(=O)C(C)(C)C)(C)C 12858,c1(C(=O)NC2CC3CCC2(NC(c2ccon2)=O)C3)cc2ccccn2c1 12859,c1(C(C)(C)C(=O)NCCC2(NC(C3CC4CC4C3)=O)CC2)ccc(F)cc1 12860,C1(S(C)(=O)=O)(N(C)Cc2conc2C(F)(F)F)CC1C(F)(F)F 12861,CC(C)(C)CCCC(=O)NCC1CCN(C(=O)CC2CCOC(C(C)(C)C)C2)C1 12862,C1(C(N(C(C)C2CC2)CC)=O)CC2CC2N1C(=O)CCOCC1CC1 12863,N12CCC(N=C3NC(=NC4=C3COC4)N3CCSC(C3)C1)C2.C1CC2CC1C1CC21 12864,c1(COC)nn[nH]c1C(=O)NC(C)C(C)NC(=O)CNc1nccs1 12865,c1(SC)cccnc1C(=O)NCC1CC2CC2N1C(=O)CCc1cscn1 12866,C1(NC(C(C(C)(C)C)O)=O)CC(N=c2ccnc(Cl)[nH]2)C1(C)C 12867,c1(C(=O)NCC(CNC(CNC(=O)NC)=O)O)c(Br)nc2n1CCCC2 12868,N1(C(CCCN(C(C)C)C)=O)CCN(C(C2COC(=O)N2C)=O)C(C)C1 12869,N1(C(C(C)OCC(C)C)=O)CCC(C2CCN(C(C3CCCCN3C)=O)CC2)C1 12870,C1(CNC(CC(CCC)O)=O)CN(c2ccc(C(C)=O)c(C)n2)CCC1(F)F 12871,N1(C(c2n(CC)nnc2)=O)C2CCC1CC(N(C(=O)CN(C1CCSC1)C)C)C2 12872,c1(CCCNC(c2cc(CNC(C3CCCO3)=O)[nH]n2)=O)ccc(F)cc1 12873,c1(C(N2CC(C)C(CCNC(c3ccncc3Cl)=O)C2)=O)cncc2nc[nH]c12 12874,c1(OCC(=O)NCC(CC)N(C(=O)C(F)C2CCC2)C)ccc(Cl)cc1C 12875,N1(C(CCSCC)=O)CCCC2(CCCCC2NC(=O)CC2(O)CCOCC2)C1 12876,C1(C(=O)NCCOC2CN(C(c3ncsc3C3CC3)=O)C2)CCCC2(CCC2)C1 12877,C1(CN(C(=O)CN2CCCC2=O)C)CCCN(C(=O)C(CO)NC(N)=O)C1 12878,CC1C(=O)CC1C(=O)NC(C)(CNC(=O)Cc1cn(C)cn1)CO 12879,C(C(C(C)(C)C)NC(=O)CCCN1CCCC1)NC(C1CC(OC)C1)=O 12880,N1(C(C2(C)COCCO2)=O)C2CCC1CN(C(c1ccc(C(F)F)nc1)=O)C2 12881,Cc1cc2[nH]c(C(=O)NCC3(O)CN(C(C4CC5CCC4O5)=O)C3)cc2o1 12882,C1(C(=O)NCC2C3CN(C(COCCCC#C)=O)CC32)CCC(S(N)(=O)=O)CC1 12883,C1(NC(C(C)(COC)NC(C(C)OCCOC)=O)=O)CCOC12CCCC2 12884,N1(C(C2N(C(C(CCCC)F)=O)C(C)C2)=O)CCC12CCCCC2 12885,C(=O)(C(CC)CC=C)NC(CCCCNC(c1cc(CCCCC)[nH]n1)=O)C 12886,N1(C(c2n(C)cnn2)C(=O)NCC(F)F)CCOC(c2cn(C)cn2)C1 12887,Cc1cc(NC(N2CCCCC2C(C)CN(C)C)=O)cc(N)c1 12888,Cc1cc2ccccc2nc1C(=O)NC1CC(C)(NC(=O)C2=CCS(=O)(=O)C2)C1 12889,c1(CN2C(C)CCC(C(=O)OC)C2)cccc(C#N)c1OC 12890,C1(C(N2CCCC(C(=O)Nc3cnn(C(F)F)c3)C2)=O)CCCC2(CC2)C1 12891,N1(C(Cc2c(C)nsc2)=O)CCC(F)C(NC(c2ccnc(C(F)(F)F)n2)=O)C1 12892,C#CC1CN(C(=O)C(=Cc2cnc[nH]2)C)CCN1C(C1Cc2nc(C)cn2C1)=O 12893,N1(C(C(Br)=C(C)C)=O)CC2CN(C(c3cccc4cncn34)=O)CC2C1 12894,C1(NC(CCC(=O)OC)=O)CC(O)CN(C(=O)C(F)(F)c2cnnn2C)C1 12895,N1(C(C(CC)NC(N)=O)=O)CC(CNC(=O)CCCF)C(n2cccn2)C1 12896,c1(C(=O)NCC(C2CCCN(C(c3ccc(Cl)cn3)=O)C2)(C)O)cccc(Cl)c1 12897,C1(C(C(=O)OCCCCCC)CC)CCN(c2ccccc2)CC1 12898,Cn1nc(C(=O)NOCC(N2CC3CC2(CO)C3)=O)cc1O 12899,N1(C(c2cncc(C#C)c2)=O)CCC2CCCC12CNC(=O)C(C)(C(C)C)OC 12900,CCCC(C)(CC)C(=O)NCC1CC(C(=O)Nc2cncc(C(N)=O)c2)=NO1 12901,C1(C(C)C)CN(C(=O)CCc2ccncn2)CC1C(=O)NCCc1cccnc1 12902,CCC(CC(=O)N(CCCC(=O)N1CC(CS(C)=O)C1)C)C1CC1 12903,c1(C(N(C2CN(C(C(C(C)C)N3CCC3)=O)C2)C)=O)cc2c([nH]1)CCC2 12904,C1(CCCCCC)CCCC1(c1nnnn1C1CC1)NCc1cocn1 12905,CC12CN(C(=O)COC(F)F)CC1(C)CN(C(N)=O)C2.C12Cc3cccc(c3O1)O2 12906,c1(OCC)ccc(CNC(=O)NC2CCN(C(=O)C(F)n3cccn3)CC2)cc1 12907,CC(CCCCNC(c1cc(Cl)cnn1)=O)NC(=O)C(C1CCCCCC1)O 12908,c1(NC(CCC)CC(F)F)ncccc1S(=O)(=O)NC(CCC)CC(C)C 12909,C(CC(C(C)(C)C)NC(c1ccc(F)c(F)c1)=O)N(C(C1(C)CC(C)C1)=O)C 12910,O=C(C1=CCCN(CCn2ccc3ccccc23)C1)NCCc1ccncc1 12911,C1(NC(C2CCN(CC)C2)=O)CCC2(CC1)CCN(C(=O)C1=NOCC1)C2 12912,C(=O)(C(O)CC(N)=O)NCC1(C(C)(C)O)CN(C(C2(OC)CCC(C)C2)=O)C1 12913,C#Cc1ccc(CCC(N2CC3(NC(=O)COCC=C)CCC2C3)=O)cc1 12914,CC(C)CC(O)C(=O)N1CC(O)CC1CNC(C1C2(CC2)C12CC2)=O 12915,C(=O)(C(CO)C(C)(C)C)N1C(C(=O)NCCN2CC(CF)C2)(COC)C=CC1 12916,CC(C)CC(CNC(c1cccc(=O)o1)=O)C(=O)N(C)CC1CC1 12917,C1(NCc2ccc(OC)cc2)CCC(C)N(C(=O)CSc2ccccc2)C1 12918,C(C(=O)N(C)CC1CCCOC1)(C(C)(C)C)NC(c1c(CC)ocn1)=O 12919,CC1=C(C(=O)NC2CN(C(c3nn(C)c(Cl)c3Cl)=O)CC2F)SCCO1 12920,C1(CC(N2CCC(CN(C)C(c3ncn(C)n3)=O)C2)=O)CCC(=O)C1C 12921,N1(C(c2ccc(C)c(F)c2)=O)CCN(C(=O)C(C)(O)C(C)C)CC(CO)C1 12922,CCC(O)C(F)(F)C(=O)N1CCOCC(C(=O)NCC#CC#CCO)C1 12923,N1(C(C=C(CC)CC)=O)CCC2CCC12CNC(c1ccc(O)c(Br)c1)=O 12924,c1(C(=O)NC2CCCN(C(c3[nH]cc(CC)c3)=O)C2C)cc2c(s1)CCSC2 12925,C1(NC(CC2N(C(C=C(C)C3CC3)=O)C3C2CCC3)=O)CCc2n[nH]cc2C1 12926,c1(C(N2CC3CC2CN3Cc2cccc(Br)c2Br)=O)cc(Cl)cnc1Br 12927,C1(Br)(C(=O)NCC(C)NC(c2cc(C(N)=O)c[nH]2)=O)C(C)C1C 12928,C(O)(C1CCCc2ccccc21)C1CN(C(C(CC)Oc2ccccc2)=O)C1 12929,C1(C(=O)NCC(O)CC2CCCC2)CC2CC2N1C(C1CCCCO1)=O 12930,Cn1nc2c(c1C(N1CC(NC(=O)CSC(C)(C)C)C3(CC3)C1)=O)COCC2 12931,C(=O)(CC(C)(C)C(F)F)N1CCC(C(C)C(N2CC(CO)C(O)C2)=O)C1 12932,c1(C(N(CC(C)O)CCNC(C(CC=CC)C)=O)=O)cc2cc(C)cc(C)c2[nH]1 12933,C1(CNC(C(=Cc2cccs2)C)=O)C2CCC(C2)N1C(=O)CNS(N)(=O)=O 12934,C12(NC(Cc3c(C)con3)=O)CCC(c3nn[nH]n3)(CC1)CC2 12935,N1(C(C(C)NC(COC)=O)=O)CCC(CO)(NC(=O)CN2CC=CC2)CC1 12936,n1(CCCOC)cc(C(=O)N(CCCCNC(c2cc(C)no2)=O)C)cn1 12937,Cc1[nH]c(C)c(C(=O)NC(CNC(C2C(C)C2C)=O)C2CCC2)c1C 12938,C#CCC(C(=O)NCC(O)CN(CC(C)C)C)NC(=O)COCC=C 12939,c1(C(=O)NCC(C)(CO)NC(=O)CSC2CC2)cccc(OC(F)F)c1 12940,N1(C(C2(NC(c3ccc(C)n3C)=O)CCCC2)=O)CCOC(C)(C)CC1 12941,Cc1cc(=NCc2cnc(C)o2)[nH]cc1S(=O)(=O)N(C(C)C)CC1CC1 12942,c1(C(N2CCN(C(c3ccccc3)=O)C(CC3CC3)C2)=O)cc([N+](=O)[O-])n[nH]1 12943,c1(NC(=O)NC2C(C)(C)C2)cccc(CN2CCOCC2)c1 12944,C(C)(CCC(=O)NCC1(CCNC(=O)Cc2cc[nH]n2)CC1)OC 12945,c1(C(N2CCN(C(c3c(CC)onc3)=O)C(CC#N)C2)=O)ccc2ccoc2c1 12946,C1(N(C(C(=O)NC)c2nc[nH]n2)C)CCCC1(C)C 12947,C1(NC(=O)NCC(C2CCOCC2)(C)C)CC2(C1)CC(F)(F)C2 12948,c1(C(=O)NC(C=CC(=O)NC2(C)CC(=C)C2)C)cc(C)ccc1O 12949,C1(C(=O)NC(CC(=O)NC)C)CNC(=O)CN1C(C1CC2(CCO1)CC2)=O 12950,Cc1cc(NCCC(C)NC(C2(O)CCCC(C)(C)C2)=O)n2ncc(C)c2n1 12951,C#Cc1c[nH]nc1C(=O)NCCN(C)C(C1CCC(NC(C)=O)CC1)=O 12952,C(CCC#N)(C(=O)O)NCc1nc(-c2ccc(C)o2)sc1 12953,C1(C(N(C)CC2CCCN(C(c3cc(CO)on3)=O)C2)=O)CC2(CCCC2)CO1 12954,C1(C(C)C)CC(CNC(=O)N(C)Cc2ccno2)CCO1 12955,c1(CNC(C(C)O)=O)cn(CC2CCCN2C(c2cc(C(F)F)on2)=O)nn1 12956,N1(C(C(CCCC)C)=O)CCCC2CN(C(=O)COC)CC12 12957,c1(NC2C(CC)CN(C(=O)CCC(=O)N(C)C)CC2)ncnc2sc(C)nc12 12958,C=CC1(C(N2CC(CNC(c3cnccc3OC)=O)C2)=O)CCOCC1 12959,c1(C(N(C(C(=O)NCCn2ncc(C)c2)C2CC2)C)=O)cn(C)nc1C 12960,CCCCC(F)(F)C(=O)NCCCC1CN(C(C2Cc3nccn3C2)=O)CCO1 12961,c1(C(=O)NC2CC(C)(C)N(C(C3COC(=O)O3)=O)C2)cccc([N+](=O)[O-])c1 12962,c1(NC(C(C2CCN(C(c3sccc3Cl)=O)C2)C)=O)ccc2c(c1)OCC2 12963,N1(C(C(CCCNC(C2CCC3CC2CO3)=O)O)=O)CC=CC12CCCCC2 12964,N1(C(C(c2ccc(C)cc2)(C)C)=O)CCN(CC(F)(F)F)CC1(C)C 12965,N1(C(C=C(C)C(C)C)=O)CC2CCCC2(NC(=O)CNS(=O)(=O)c2cccs2)C1 12966,C(C(CC(C)C)NC(=O)C(C)O)NC(CCCN(CCC)CCC)=O 12967,N1(C(C2C(C)(C(C)C)C2)=O)CC(C)CN(C(C2CCSC(C)C2)=O)CC1C 12968,C(=O)(C1CC(NC(N2CCOCC3(CCOCC3)C2)=O)c2ccccc21)OC 12969,c1(C(=O)NC2CCCN(C(C3(CC(C)C)CC3)=O)C2)cccc2c1NCC(C)C2 12970,c1(C(=O)NCC2N(C(C(C)C3CCCC3)=O)CCCC2C)nccc2occc12 12971,c1(C(N(CCCNC(C2CCC(C(F)(F)F)CC2)=O)C)=O)ncn2c1COCC2 12972,C12(C(=O)NCc3c(Cn4cc(CNC=O)nn4)nco3)CCN(CC1)C2 12973,c1(C(N2CCCN(C3COC(C)(C)OC3)CC2)=O)cc(O)nc(Cl)c1C#N 12974,c1(C(c2nnnn2C2CCC2)NCc2ccc(C)s2)ccc(C)c2cccnc12 12975,N1(C(C2C(C)(C)C2)=O)CCC(COC2CCN(C(=O)CN3CC4CC4C3)C2)CC1 12976,Cc1cnc(NC(C)CC(C)C)c(S(=O)(=O)N2CC(CO)C3(CC3)C2)c1 12977,c1(SC)cc(N2CC(CN(C(=O)CC3SC(=N)NC3=O)C)C2)nc(SC)n1 12978,N(C)(C1CCCc2ccccc21)Cc1c(OC)cccc1Br 12979,C1(NC(CSC)=O)(CNC(C23COC(CF)(C2)C3)=O)CC2CCC1C2 12980,C1(OC)CCCCC1CNC(c1ncoc1CNC(=O)C=C=C(C)C)=O 12981,c1(C(=O)NC(CNC(COCCCCC)=O)(C)C)cc(N)c(C)cc1Cl 12982,N1(C(C2CC(C(=O)OC)C2)=O)CC(NC(c2ccc(C(C)(C)C)s2)=O)CC(C)C1 12983,N12CCCN(CC1C)C(=O)c1cc(ccc1Cl)C2=O.C1(OCCCC)CCCC1 12984,c12cc(Cl)ccc1OC2.N1(C(C)=O)CCC(NC(=O)Cc2cc(N(C)C)no2)C1 12985,c1(C(C)(C)C)nnc2n1CC(NC(=O)C(=O)N(c1ccc(O)cc1)CCO)CC2 12986,Cc1cc(C)c(C(=O)NC2CC3(C2)CN(C(=O)CC2CC(F)C2)C3)c(S)n1 12987,C#Cc1ccc(OCC(=O)NCC2(F)CCCN(C(=O)CCC=C(C)C)C2)cc1 12988,c1(C(C)NC(=O)NCC2(c3cccc(Cl)c3)CCOCC2)nc(Cl)ccc1Cl 12989,N1(C(C2(OC)CCCCC2)=O)CCC(C)C(NC(c2cc(F)ccc2Cl)=O)C1 12990,C1(C(=O)NCCCSCC)C(NC(c2cc(C(F)F)[nH]n2)=O)C1(C)C 12991,CC1CC(NC(=O)CC=CC(C)(C)C)CN1C(c1cc(N2CCOCC2)ccn1)=O 12992,N1(C(C2CC(NC(C(COC)(C)OC)=O)C2)=O)CC2CCCCC2C1C 12993,C(=O)(C(F)C(=O)NC1(C)CC(NC(=O)CC2CC2(C)C)C1)OCC 12994,c1(CC)sc2ccccc2c1Cl.C(C)(C(F)(F)F)OC(N(C(=O)CS)C)=O 12995,CC1CCCCC1(C)C(N1CCC(c2cn(Cc3cnn(C)c3)nn2)C1)=O 12996,N1(C(c2cc(CO)on2)=O)CCC2CCN(C(C3CC4(C3)CC4(F)F)=O)CC2C1 12997,Nc1ncc(C(N2CCCCC(NC(C3CC4(CC4)C3)=O)C2)=O)cc1Cl 12998,C1(NC(C(CCC)NC(C)=O)=O)CN(Cc2ccn(C)n2)CC(F)(F)C1 12999,c1(C(=O)NC2C(NC(c3ccc(N(C)C)cn3)=O)C2)cnc(O)c(F)c1 13000,Cc1ccc2nc(N3CCCC(NC(=O)CN(C)C(N)=O)C3C)sc2n1 13001,c1(C(=O)NC2C(NC(C(C(C)O)NC(C)=O)=O)CCC2)cc(C)c(=O)n(C)c1 13002,N1(C(c2c(CC)scc2)=O)CC2(C)CN(C(=O)C=CC=C(Cl)Cl)CC2(C)C1 13003,Cc1csc(=O)n1CC(N1CCN(CC(C)(C)F)CC1)=O 13004,C1(CC(=O)NC2CN(C(=O)C=Cc3ccccn3)CC2OC)(CC)CCOCC1 13005,C1(NC(CNC(CNC(C)=O)=O)=O)COC2(CCN(C(c3ccoc3)=O)C2)C1 13006,c1(COCC(=O)NCC(C2CC2)NC(C2(CC3CC3)CC=CC2)=O)ccccc1 13007,Cc1ncc(C=CC(=O)NCCCCCNC(c2ccc(C(N)=O)o2)=O)c(O)n1 13008,C(c1cccnc1)=C(C)C(=O)NCc1ccc(C(=O)NC2CC(O)C2(C)C)nc1 13009,c1(C(=O)NC2CC(C)(NC(C3C(C)OC(=O)N3)=O)C2)cc(NS(C)=O)ccc1F 13010,CCC(O)C(F)(F)C(=O)N1CCCC(C(=O)NC2COCC2CO)C1 13011,CCCCC(O)C(C)C(=O)N1CC(O)(C(C)(C)CNC(=O)Cc2cnoc2)C1 13012,C1(CCNC(c2cn(CC)nn2)=O)CN(C(c2cnc(=N)[nH]c2)=O)CCO1 13013,c1(OC)cc(CC(N2CC(CNC(=O)CCc3cnc(O)[nH]3)CC2C)=O)ccn1 13014,c1(C2(C)CCN(C(=O)NC(C(=O)OC)C)C2)cc(Cl)ccc1Cl 13015,c1(OC)ccc(Br)c(CN=C(NCc2ccco2)NCC2(F)CCOC2)c1 13016,Cc1nc(-c2ccccc2)ncc1C(=O)NC1CN(C(C2CCCC(O)C2)=O)C1 13017,c1(C(N(CCCNC(C2CC2(C)C)=O)Cc2ccccc2)=O)snc(O)c1Cl 13018,C(C(=O)N1CC2C(C(=O)NC(C)(CO)C3CCC3)C2C1)(C(C)(C)C)N(C)C 13019,Cc1cnc(C(C)NC(=O)C=CC(C)(C)NC(=O)CCCNC(=O)C2CC2)s1 13020,c1(CC)n[nH]c(=NC2CC3CN(C(=O)Cc4cc(C(F)(F)F)co4)CC23)o1 13021,N(C1CCOc2ccc(F)cc21)Cc1ccc(-c2ccc(N)c([N+](=O)[O-])c2)s1 13022,C(=O)(CC(C)CC(C)C)N1CCC(C(N(CCN(CC)CC)C)=O)(CO)C1 13023,C1(NC(c2c(Cl)cn(CCC)n2)=O)CCC12CN(C(=O)C(C1CCCCC1)O)C2 13024,C(C(O)CCNC(=O)C(CO)NC(c1ncsc1NC)=O)OC 13025,N1(C(CC2CC(=C)C2)=O)CCN(CC(=O)NCC(=O)Nc2cn[nH]c2)CC1 13026,N1(C(CSCC(C)C)=O)CCC2(C1)CN(C(=O)C(N1CCC(C)C1)=O)CCO2 13027,N1(C(c2cc(CCOC)on2)=O)CCC2(CCCN2C(=O)CP(C)(C)=O)C1 13028,N(C1CCc2cccnc21)C(N(C)Cc1ncc(Br)cc1Cl)=O 13029,c1(C(=O)NC(CCNC(CCn2ccc(C)n2)=O)C)cnn2cc(C#N)cnc12 13030,C1(CNC(c2ccc(-c3cc[nH]n3)s2)=O)CCC(NC(C2(CF)CCC2)=O)CC1 13031,C12(CNC(CN(C(COC)=O)C)=O)CC1CN(C(C1(F)CC1(Cl)Cl)=O)C2 13032,N1(C(c2cc(C(CC)C)no2)=O)CC(F)(F)CC1CCNC(=O)CCSC 13033,c1(C(C(=O)NCC2(NC(CCOCCC)=O)CCCC2)(F)F)ccccc1OC 13034,N1(C(C2CCCN(C)C2)=O)CCC(CNC(C2CC(=O)N(O)C2)=O)C12CC2 13035,C1(CN(C(CN(C)CC)=O)C)COCCN1C(=O)CCCc1csc(C)n1 13036,c1(NCCn2c(C)cc(C)n2)ncccc1S(=O)(=O)N1CCn2ncc(Cl)c2C1 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13054,C(C)(CCC(=O)N1CC(C(F)Cn2cc(CC3CCCC3)nn2)C1)OCC 13055,c1(NC(c2ccc(NC(C)=O)cc2)=O)n[nH]c2c1CN(Cc1cc(Br)c(C)s1)C2 13056,N1(C(c2cnc(C)[nH]2)=O)CCC(C2CCCN(C(c3nc(C)c(C)s3)=O)C2)C1 13057,N1(C(Cc2cc(OC)c(F)cc2)=O)CCN(Cc2ccc([N+](=O)[O-])s2)CC12CC2 13058,C(=O)(C(C)(C)CC(F)F)NCC1CC(OC)CN1C(c1ccc(Cl)c(Cl)c1)=O 13059,C1(O)(COC)CCN(C(=O)C(C)(C)CNC(=O)C(C)OCC(C)C)CC1 13060,c1(CC(NC(=NC)NCC23CCN(CC2)C3)CCC)cccc(Br)c1.O 13061,Cc1cc(=NCC2CC(C)(C)CCO2)[nH]c(N2CC(C(F)(F)F)C(S(C)(=O)=O)C2)n1 13062,C=C(F)C1(CC(=O)NC(C)(C)C(C)NC(C2CC2(C(C)C)CC)=O)CCC1 13063,C1(N(C(CC)=O)C)CCCCN(C(C23CC(c4ccc(OC)cc4)(C2)C3)=O)C1 13064,N1(C(C2CN(C)C(=O)C2)=O)CCCOC(CCNC(c2c[nH]cc2C2CC2)=O)C1 13065,c1(NC(C)=O)ccc(C2CC2)c(Cl)c1.c12cnn(c1)CCNC2=O 13066,c1(C(C)C)ccc(OCC(N2CC(NC(C3(CCF)CC3)=O)C(O)C2)=O)cc1 13067,c1(CNC2CCC(N(C(=O)C=Cc3cccs3)C)C2)cc(F)ccc1F 13068,C1(CC(N2CCC(N(C(=O)C=CCOC(C)(C)C)CC)C2)=O)CC(C2CC2)C1 13069,N1(C(c2ccc(C#N)c(Cl)c2)=O)CCC2(CCN(c3ncc4cn[nH]c4n3)C2)C1 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13155,C1(C(=O)NCC2(C)CC3(CC3)C2)(CNC(CC)=O)CC12CCC2 13156,N1(C(C(C=C)C)=O)CC2CCCC2C1C(N1CCC(C)(CN(C)C)C1)=O 13157,CON(C)C1CN(C(=O)CC2CCCCN2C(=O)COCCCF)C1 13158,C1(CNC(CC2(COC)CC2)=O)CN(C(c2cc[nH]c(=N)c2)=O)C2CC12 13159,c1(OC)cccc(CC(N2CCCC2C(C)NC(=O)C=Cc2ccco2)=O)n1 13160,C(=O)(C1CCc2cc(Cl)ccc21)NCC1(NC(c2cn(CCC)nc2)=O)CCC1 13161,c1(NCC2(OC)CNC2)cnc2n1CCOC2 13162,N(C1c2ccccc2CC1NC(=O)C=C1CCC1)C(C1N(N=O)CCCC1)=O 13163,CC1(C)CC(C(N2C3CCC2CC(NC(C2CC2C(F)F)=O)C3)=O)CC(C)(C)O1 13164,c1(C(C)=O)cccc(OCC(N2CC(NC(=O)CCC3(C)CC3)C3CC23)=O)c1 13165,n1(CC(C)CO)cc(C2CCCN2C(=O)C=CI)nn1 13166,Cc1nccc(C(=O)NCc2cncc(C(=O)NC3CCN(C(C)C)C3)c2)c1N 13167,c1(CNC(c2c(OC)ccs2)=O)ccc(CNC(C2CCC(=O)N2C)=O)c(F)c1 13168,N1(C(Cc2ccc(OC)nc2)=O)CCN(c2ccccc2)C(C)C1 13169,C1(CNC(c2cc[nH]c2)=O)C2CCC1CN(C(=O)CC(O)c1ccccc1)C2 13170,N1(C(C(=Cc2ccccc2)C)=O)CCCC(C)(C(=O)NCC(C)(C)O)C1 13171,C=CC(CC)C(=O)N(C)CC1COCCN1C(=O)CCC1(C)CC1(F)F 13172,C1(C(=O)NC(CNC(C(CCSC)O)=O)(C)C)Cc2ccc(Br)cc2C1 13173,C1(CC)CN(C(C2CC(=O)N(CCOC)C2)=O)CCN1C(c1ccc(F)cn1)=O 13174,C(C(C(=O)N1CCCC1CCNC(=O)C(C)Oc1ccccc1)OC)OC 13175,C1(C(=O)NC2CCN(C(N3CCCC3)=O)C2)CCC(F)(F)CC1O 13176,N1(C(COC(C)=O)=O)CCC2CCN(C(=O)C3Cc4ccccc43)CC2C1 13177,c1(C(N2CC(C3(NC(CCC4CCC(=O)C4)=O)CC3)C2)=O)cc2cccnn2c1 13178,c1(C(=O)NCC(C)(C2CC2)NC(C2CCC2(F)F)=O)cc2c(nn1)CCOC2 13179,C1(C(N2CCN(C(C3CCC(C)(C)CC3)=O)C3C2C3)=O)CCCN(S(N)(=O)=O)C1 13180,C(CN=c1ccnc(N2CCN3CC(O)CC3C2)[nH]1)(C1CCCCC1)OC 13181,CCC(C)(CO)C(=O)N1CC(CNC(c2ccnnc2)=O)C(F)(F)C1 13182,CC1CC(C)(C(=O)NCC2CN(C(=O)CCCOc3ccccc3F)C2)CCO1 13183,c1(CC)cc(C(=O)NCC(C)(F)CNC(C2CCCCC2O)=O)ccc1C 13184,CC(CNC(=O)CNC(=O)CN(C)C)C(F)C(=O)NCC1CC1(F)F 13185,C(=O)(C(C)CS(C)(=O)=O)NC1CC(C)(NC(CC2N(C(C)=O)CCC2)=O)C1 13186,c1(OCCO)cccc(NC(=O)CC2CCN(c3ncc(Cl)cn3)C2)c1 13187,c1(OC(C)C)ncccc1C(=O)NCC1(CNC(C2OCCO2)=O)CC1(F)F 13188,CC1CN(C(c2ccc(C(F)(F)F)cc2Br)=O)CCN1C(c1ccnnc1)=O 13189,c1(C(N(CCC(=O)NC(C(C)SC)C)C2CC2)=O)ccnc(C)n1 13190,N1(C(CN(C)C(N)=O)=O)CC2(C1)C(NC(C1CCC3CCC1O3)=O)CCS2(=O)=O 13191,Cc1cc(C(N2CCC2CNC(c2cc(-c3ccco3)no2)=O)=O)cn1C 13192,c1(C(=O)NCC(c2ccc(OC)cc2)NC(CC=CCC)=O)cc(C)c(F)cn1 13193,c1(C(N2CC(NC(C3CC4CCCCC34)=O)(CO)C2)=O)cc(F)c(CO)c(F)c1 13194,c1(C(N2CC(C)CC(C)C2C)C(=O)NCCCSC)ccc([N+](=O)[O-])cc1OC 13195,C1(CC)CN(C(=O)CN2CCNC(=O)C2)CCN1C(=O)CC1CCCCC1O 13196,c1(C(N(C2CCN(C(C3CCCS3)=O)CC2)CC)=O)n[nH]c2c(C)cccc12 13197,c1(C(=O)NCC(C(C(C)C)C)NC(c2nsnc2O)=O)cc(F)c(F)c(F)c1F 13198,c1(CC(=O)NC2C=CC(CNC(C(C)(F)F)=O)C2)cccc2cnccc12 13199,C(=O)(C1=NOC2(CCC2)C1)NC(CNC(C1(C)CCC(=O)NC1)=O)CC(F)(F)F.C 13200,C1(C(N2CC(NC(=O)NC)C2)=O)C2CC(O)C1N(C(c1ccnn1C)=O)C2 13201,C(=O)(C(C)CS(C)(=O)=O)NC1CC(CCNC(COc2cc(C)cc(C)c2)=O)C1 13202,C=CCC(C)(C)CC(=O)NC1CC(NC(c2ncccc2Cl)=O)C1 13203,c1(C(=O)NC(C2CC(C(=O)Nc3ccsn3)C2)C)c[nH]nc1-n1cnnn1 13204,C1(NC(c2cn(CCNC(C3(CC4CCC4)CC3)=O)nn2)=O)CCCCC1O 13205,C1(NC(C2C=CCC2)=O)C=CCN(C(=O)CC(c2ccccc2)c2ncc[nH]2)C1 13206,CC1(C)CCC(O)(CNC(=O)CCCC2CN(C(=O)CN3CCOCC3)C2)C1 13207,C(=O)(CCCCCCn1cc(CSCC)nn1)N(C(c1ccncc1)(C)C)CC 13208,c1(C(=O)NC2CCC(CNC(c3cc(OC)no3)=O)C2)ccc(=O)n(C)c1 13209,CC1CN(C(c2ncn3c2CCCC3)=O)CC(C)C1NC(c1ccc[nH]1)=O 13210,CS(=O)(=O)CC(=O)NCC1(C(=O)Nc2cccc(CO)c2)CC12CCC2 13211,C1(F)(CNC(C(c2c(C)cccc2)C)=O)COCCN(C(=O)CSC(F)F)C1 13212,c1(C(N(C2CCN(Cc3ccsn3)C2)C)=O)cccc(C=O)c1Br 13213,C(CC(=O)NC1CCNC1(C)C)(C(F)(F)F)NC(N)=O 13214,N1(C(c2ccc(C)cc2F)=O)CCC2CN(C(=O)CC3CCCCO3)C2C1 13215,C#CC1C2CN(C(C3COCC3C(=O)O)=O)CC12 13216,c1(NC)ccnc(C(N2CC(CO)(NC(=O)CCC(C)c3ccccc3)C2)=O)c1 13217,C(=O)(CCCC(=O)NCCCC(C)(C)NC(C1CC2CCC1C2)=O)NCC 13218,N1(C(c2scc(C)c2)=O)CCC(N=c2cc(C)nc(S(C)(=O)=O)[nH]2)C(C)C1 13219,N1(CC(=O)NC(C)CCNC(=O)Cn2nnc(C3CC3)n2)CCC(N(C)C)CC1 13220,c1(C(=O)NCCOC2CCN(C(CN(C(C)=O)C)=O)C2)c(C2CC2)cccc1F 13221,c1(C(N2CC(C(C)NC(c3ncncc3Cl)=O)OCC2)=O)ccnc(C#N)c1 13222,Cc1cccc(CN(CC(C)C#N)Cc2ccc(OCF)cc2)c1C 13223,N1(C(C2CCC(C)(CC)O2)=O)CC=C(CC(=O)NCc2ccc(F)c(C)c2)CC1 13224,N1(C(C2N(C)CCN(C(c3c(OC)csc3)=O)C2)=O)CCCC(C)(C)CC1 13225,C1(CNC(c2nn(CC)nc2C)=O)(NC(C2CC(O)C2)=O)CCCCC1C 13226,c1(C(=O)NC2COCCN(C(C(CCSC)O)=O)C2)cc2ncccc2s1 13227,c1(C(=O)NC(C2CCN(C(C=CCC)=O)C2)C)c(C)cnn1C 13228,c1(CC(N2C(CNC(=O)Cc3ccno3)CCC2)=O)ccc2ncsc2c1 13229,C(CC(C)C)(C(=O)NC1(CNC(C2CCOC2)=O)CC1)OC 13230,C1(C(=O)NCC(CNC(C2CSC2)=O)OC)CC2CCC(C1)N2S(=O)(=O)CC 13231,C(C(C)C(=O)N(C1CCC1)C)N(C(CCNC(C)=O)=O)C 13232,C1(NC(C(CC=CCC)C)=O)C2CCC(C2)C1C(=O)NCC1CCC(C)C1 13233,c1(C(=O)NCC2C(CNC(C(C=C)(C)O)=O)C2(F)F)ccc(CC)c(Br)c1 13234,C1(C(N(C(C(C)C)C)C)=O)CN(C(c2coc3c2COC3)=O)CC(C)O1 13235,N1(C(c2cncc(SC)c2)=O)CC(NC(=O)CC2CNC(=O)C2)CC(C)(C)C1 13236,C1(C(C(C)C)NC(C(CC)F)=O)CCN(C(=O)C=Cc2cnccn2)CC1 13237,c1(C(=O)NCC(C)N(C(c2cnc[nH]c2=N)=O)CC)ccc(F)cc1OC 13238,C1(C(C)OC)CCN(C(=O)C=CC(C)NC(=O)C(C)C2CCCC2)CC1 13239,N1(C(C=CCC)=O)C2CCC1C(NC(c1cccn1C1CCCC1)=O)C2 13240,C1(SC)CN(C(=O)C(C)(C)n2cccn2)CC1NC(C1CCC1c1nc[nH]n1)=O 13241,N1(C(CC(CN(C)C)O)=O)CC(C(=O)NCC(C)(C)CCCO)C(F)(F)C1 13242,N1(C(C2CCC(C)N(C(=O)COCC(F)F)C2)=O)CCCN2CCCC2C1 13243,Cc1cnc2n1CCC(C(=O)OC(C)(C)C)C2.C1C(c2ccccc2)C(=O)N1 13244,CN1CCN(C(=O)Cc2ccnc(O)c2)C(CNC(C2CC3(CC3)CO2)=O)C1 13245,c1(CN2C(C(=O)NCc3ncc(Br)s3)CC(O)C2)c(Cl)ccnc1Cl 13246,C(=O)(CC(C)(C)C1CC1)N1CCC(C(C)N(C(c2ccc(C(C)=O)o2)=O)C2CC2)C1 13247,N1(C(c2cc(C(C)=O)[nH]n2)=O)C(CNC(=O)C(C)(C)C2CCC2)CC2COCC12 13248,c1(-c2ccc(OC)s2)n[nH]c(=NC(=O)N(c2ccc(Cl)cc2)CC2CC2)s1 13249,C(CCCC(=O)O)n1cc(CN(C(C(c2ccnn2C)C)=O)CCCO)nn1 13250,Cc1c(CC(N2CCOC(C(=O)N(C3CCCC3(F)F)C)C2)=O)cnn1C 13251,C(CS(=O)(=O)C1=CCC2CC2C1)N(C)S(=O)(=O)NCC(=O)O 13252,C12(C(=O)NCCN(C(C3CC3C(=O)OC)=O)CC)CCC(C1)C2c1ccccc1 13253,CC(C)CC(O)CC(=O)N1CCC(C(C)(C)CNC(C2CCOC2)=O)CC1 13254,C#Cc1c[nH]nc1C(=O)NC1CC1NC(c1ccccc1COC(C)(C)C)=O 13255,N1(C(CCCC)=O)CCC(NC(c2csc(-c3ccsc3)n2)=O)C(CC)C1 13256,c1(C(=O)NC2CC3(CN(C(C(C)CN(C)C)=O)C3)C2)nnc(O)c2ccccc12 13257,N1(C(C2CC=CC(NC(C3(CO)CCCCO3)=O)C2)=O)CC2C=CCC(C2)C1 13258,c1(C(=O)N)cn2ccnc2cn1.C1(C2CCC2)CCCN1C(C1CC1F)=O 13259,N1(c2n(CCC#C)c(C=C)nn2)CCc2c(NC(C)=O)cccc2C1 13260,Nc1ccc(C(N2CCCC2C2(NC(=O)C#CC3CCC3)CC2)=O)nc1C(F)(F)F 13261,C(C(O)CNC(C1CCCO1)=O)NC(CSCC#N)=O 13262,C1(NC(C=CC(C)NC(c2c(CC)[nH]cc2)=O)=O)(CO)CCCCC1C 13263,C1(C(=O)NC2(C(N)=O)CCOC2)CN(C(=O)CC2CCCC3CC23)CC1C(F)F 13264,CC1CC(=O)NC1C(N1CCC(CNC(c2ncoc2C(F)(F)F)=O)CC1)=O 13265,C1(O)(C(=O)NC(C)Cn2cc(C3CCCO3)nn2)Cc2ccccc2C1 13266,c1(NCC2(CNC(c3cncc(OC)c3C)=O)CC2)ncnc2cc(Br)ccc12 13267,C(=O)(C1CCCc2sccc21)NCC1(NC(C2CCN(C)C2)=O)CC1 13268,Cc1cccc(C(C)NC(=O)C(CCC2CCC2)NC(=O)C(C)c2cccs2)n1 13269,N1(C(CC(C2CC2)NC(C(CC(C)C)O)=O)=O)CC2CCOC(=O)C2C1 13270,c1(OC)cc2nn[nH]c2cc1C(=O)NCCCCNC(c1cnn(C)n1)=O 13271,C1(CC(=O)NC2CN(C(C)=O)C2)CCN(C(=O)Cc2ccc(C)s2)CC1 13272,c1(C(=O)NC(C2CC(NC(C3CC(SC)C3)=O)C2)C)ccnn1CCF 13273,c1(CC(=O)NCC2C(NC(C3(C)CC3)=O)CCC2)ccc2nonc2c1 13274,C1(C(=O)NC(C23CCC(CC2)C3)C)(NC(C2CCO2)=O)CCCCC1 13275,c1(C(N2CC3CC3(C(=O)NCc3cncs3)C2)=O)cc(Cl)c(O)cc1F 13276,C#Cc1ccc(C(=O)NCC2CCCC(NC(=O)Cc3ccoc3)C2)c(F)c1 13277,CC(C)C(F)(CNC(C1(CCN(C)C)CC1)=O)C(=O)NCC(C)(C)CN=[N+]=[N-] 13278,n1(CCC(N2C(C)CN(C(C3(CO)CCCO3)=O)CC2)=O)ccc2ccccc12 13279,C1(NC(C2(CCNC(CC(=O)OCC)=O)CCC2)=O)CC(C2CCCC2)C1 13280,C(CC1=CCN(C(c2ccc(F)c(F)c2N)=O)CC1)NC(C(CCC)=CCC)=O 13281,c1(N(CCC(N)=O)C)ncnc(N2CCC(OCc3ccccc3)C2)c1[N+](=O)[O-] 13282,c1(C(=O)OCC)nnn(C)c1CNCc1cscc1Cl 13283,C1(C(=O)NC(CC=C)C(=O)OCC)CNC(=O)CN1C(C1CC1C(F)F)=O 13284,n1(CC)ccc(CC(=O)N(CCC(=O)NCc2csc(O)n2)C(C)C)n1 13285,C1(C(=O)NCC2N(c3nc(C)cc(C)n3)CCN(C)C2)CCCC2CCCCC12 13286,Cc1ncccc1NC(c1c[nH]nc1CCCNC(=O)CC1CCCC(C)O1)=O 13287,c1(C(=O)NC(C)CN(C)C(C2NC(=O)CC2C)=O)ccc(N)cc1O 13288,C1(C(=O)NCCOCCC(=O)NC(CC)C2CC2)CCC1C#N 13289,c1(OC)cc(F)c(F)cc1-c1ccc(C(=O)Nc2nc(Cl)c(Cl)cc2Cl)nn1 13290,N1(C(=O)OC(C)(C)C)CC2(CCC2)CC1NCC(C1CCOC1)=O 13291,C1(CC#C)(C(=O)NC(CC(N)=O)C2CC2)CCN(C(c2ccnn2C)=O)C1 13292,c1(C(N2C(CNC(=O)C(F)C(C)C)CC(OC)C2)=O)cc(C)c(F)cc1N 13293,O=C1NCCCCC1C(=O)NCC12CC(CN1C(c1ncccc1Br)=O)C2 13294,N1(C(c2ccc(C3CCC3)cc2)C(=O)NCCOC)CCS(=O)(=O)C2(CCC2)C1 13295,N1(C(C(CC#C)C)=O)CCOC2CN(C(=O)Cc3cccc(OC)c3Cl)CC12 13296,C1(C(N)=O)CCC(NC(=O)CCC2CCOCC2)C1.C12CCN1C(=O)C2 13297,Cc1ncc([N+](=O)[O-])cc1NC(=O)CC1CCN(Cc2cc(F)c(F)c(F)c2)C1 13298,O=C(C#CC1CCOCC1)NC12CCCN(C(c3cc4n(n3)CCC4)=O)CC1C2 13299,c1(C(N(CCN(C(C2CC2F)=O)CC)CC)=O)coc2cccc(Br)c12 13300,C(CC)(CCCO)NC(C1(CC=C)CCCN1C(=O)C(C#N)CC)=O 13301,c1(OC)ccc2[nH]ccc2c1C(N1CCC(C)(NC(=O)C(CC(C)C)OC)C1)=O 13302,C(=O)(C(C)(C(C)C)OC)NC(CC=C)CNC(c1n[nH]c(C)n1)=O 13303,c1(OCCC(=O)N(CCNC(C(CC)O)=O)CCOC)ccc(C)cc1Cl 13304,C(c1ccccc1Cl)=C(C)C(N1CC(NC(=O)CC2(C)CCCO2)CC(F)C1)=O 13305,Cc1ccc(O)cc1C(N1CC(C)CC1C(=O)N(C1CC2CC2C1)C)=O 13306,c1(CC)nn(C)cc1C(=O)NC1CC(CNC(=O)C(C)(C)NS(C)(=O)=O)C1(C)C 13307,CC1(C)C(NCC(F)(F)C(F)F)C2CCCN(C(C3CC34CC4)=O)C12 13308,Cc1ccc2ccc(C(=O)NC3(CNC(C4CCCSC4C)=O)CCC3)nc2c1 13309,CC1CCN(C(C2CN(S(N)(=O)=O)C2)=O)CCN1C(c1ccn2ccccc12)=O 13310,c1(C(N2CC(C)(NC(C(CN(C)C)O)=O)C2)=O)ccn2ccnc2n1 13311,CC(CO)(C(=O)NC(C1CCCCC1)CO)NC(=O)CCC1CCOCC1 13312,N1(C(CC=C)=O)CCOC(Cn2cc(CC(c3ccccc3)O)nn2)C1 13313,c1(COC)cnc(NC(=O)NCC(c2ccccn2)C)nc1 13314,CC1CN(C(=O)CS(N)(=O)=O)CCC1N(C)C(c1cnc(C(F)F)nc1)=O 13315,C1(CC(=O)N(CC(C)NC(=O)CCCCCn2cnnn2)C)CCS(=O)(=O)CC1 13316,CCC(CC)C(=O)NC1CC(CO)N(C(=O)CNS(C)(=O)=O)C1 13317,CC1CC2CN(C(C3CC3(F)Cl)=O)CC2N1C(=O)C(O)CC(N)=O 13318,C1(OC2CN(C(c3ccon3)=O)C2)CCN(C(=O)NC23C=CC(CC2)C3)CC1 13319,C1(NC(c2ccnc(F)c2)c2n(CCCSCC)nnn2)CCCCCCC1 13320,CCC(C(=O)N(CC(C)O)CCNC(=O)CC1CCCO1)NC(c1ccco1)=O 13321,C1(C(N2CCCC2CNC(C23CC(F)(C2)C3)=O)=O)CCN(CC(F)(F)F)C(=O)C1 13322,C1(NC(C(C)OCC)=O)CN(C(c2c(Cl)csc2Cl)=O)CC1(C)C 13323,N1(C(c2cnn[nH]2)=O)CCC(NS(=O)(=O)CC2CCOC2)CC1 13324,CCCCCC(C)CC(=O)NCCC1(C(N2CC3CC2CS3=O)=O)CCC1 13325,C1(C(=O)NC2CCC(CNC(=O)CSC3CC3)C2)CC2(CCOC2)C1 13326,C(=O)CC(C)(C)N.C(=O)(C(C)(C)COC)NCC(=O)N(CCOC)CC 13327,CN(C)S(=O)(=O)N(C)CC(=O)NCCC1CCC(NC(=O)CC2(CO)CC2)C1 13328,c1(OC)cc(-c2csc(C(N3CCCC(CO)C3)=O)n2)c(NC(C)=O)cn1 13329,c1(C(N2C(C(=O)OC)C=CC2)=O)oc(CNC(c2nnsc2N)=O)nc1C 13330,C1(NC(c2ccnc(C)n2)=O)C2CC1CN(C(=O)CSc1ccccc1Cl)C2 13331,CC1CCC(CNC(=O)C(O)C(F)(F)F)CN1C(c1cnc[nH]1)=O 13332,CC(C#N)CCC(=O)N1CC(CNC(c2cc(-c3cnn(C)c3)on2)=O)C(O)C1 13333,C1(C)(C(=O)NC2CC(CN(CC)Cc3ccccc3)C2)C=CCCC1.C1C(=O)N1 13334,C1(NC(C2CC(=O)N(C3CC3)C2)=O)CCN(C(C2C(C(=O)NCC#C)C2)=O)CC1 13335,c1(C(=O)OC)cnc(N2CCC(OCCNC(=O)C(O)Cc3cnc[nH]3)C2)s1 13336,C1(C(=O)NCC(C(C)C)O)CN(C(C2CS(=O)C2)=O)CC1(C)C 13337,c1(C(N2CC(CCO)(NC(CSC(C)C)=O)C2)=O)nncc2ccccc12 13338,C(=O)(C(CO)C(C)C)NCC(C)N(C(Cc1cccc(C(C)C)c1)=O)C 13339,c1(OC)ccc(C(=O)NCCNC(=O)CC2CCCC(C)C2)nc1Br 13340,N1(C(CC=CCC)=O)CCCC2(CCCN2C(=O)N(c2cccnc2)CC)C1 13341,C1(NC(c2c(C)cns2)=O)CCC(CNC(c2csc(Br)n2)=O)CC1 13342,C1(NC(c2cncc(C)n2)c2n(C(CC)C)nnn2)CC(S(C)(=O)=O)C1 13343,CC(C)C(CN(C)C)C(=O)NC1CCC(CCC(=O)NCC2CCCC23CC3)C1 13344,Cc1c(C(=O)NC2CC(C(=O)NCC3COCC3(C)C)C2)ncn1C 13345,N1(C(C(C)OCc2ccccc2)=O)CC2(C1)SCCC2NC(=O)CCCC(N)=O 13346,CC1CN(C(c2cccc(F)c2)=O)CCC1C(=O)N(C)Cc1ccc(O)nc1 13347,C1(C(N(CC(CCC)O)C)=O)(CNC(c2c(C)cnn2C)=O)CC12CCC2 13348,C1(C(N2CCN(c3cncc4nccn34)CC2)=O)CC2(C1)CC21CCC1 13349,c1(C(N(C)CP(C)(C)=O)=O)cc(C(=O)O)c([N+](=O)[O-])cn1 13350,N1(Cc2c(OC)ccc(OC)c2)CCC(C2CCN(C)CC2OC)CC1 13351,N1(C(C(CC)NC(N)=O)=O)CC2CCC1C(C(N1CCC(Br)C1)=O)C2 13352,C12(CNC(C(CC)N(C)C)=O)CC1CN(C(C1COCCO1)=O)C2 13353,C1(C(N2CCC(NC(C3C(C#C)C3)=O)CC2C)=O)CSc2ccccc2O1 13354,c1(OC)ccc(F)cc1CCC(=O)N1CC(NS(=O)(=O)CC2C(C)(C)C2(F)F)C1 13355,C(C)(C)(CCCC(=O)NC(CO)CC(C)(C)C)NC(C(C)O)=O 13356,c1(CC(=O)NCCCC(C)NC(c2ccoc2)=O)cccc(OC(F)(F)F)c1 13357,N1(CC(=O)NC2CCC2NC(C2(CC(F)F)CC2)=O)Cc2ccccc2C1 13358,Cc1nc(O)nc(O)c1CC(=O)NC12CCCC1N(C(=O)C(F)(F)C(C)O)CC2 13359,N1(C(CC(CC)(C)C)=O)CCCN(C(c2ccc(OC3CCC3)cc2)=O)CC1C 13360,CC1CCC(CNC(=O)CCN(CCCO)C(C23CCC(C2)C3)=O)N1C 13361,C1(C(c2ccccc2)C(=O)NCCN(CCC(C)C)CCOC)CCCCCC1 13362,c1(C(=O)NCC(CC)NC(c2ccn(-c3cccc(F)c3)n2)=O)cccnc1C 13363,C12(C(=O)NCCCN(C(=O)CN3CCCS3(=O)=O)CC)CCCCC1C2(F)F 13364,c1(C(F)(F)F)nc(NCC2CCC3(CCC3)O2)cc(=NCc2ccc(Br)cc2)[nH]1 13365,N1(C(CN(C(C)C)C)=O)CCC(C(C)(C)CNC(=O)CC2NC(=O)NC2=O)CC1 13366,CC1CC(NC(=O)CC2CCC3(CC2)CC3)CCN1CCN1CCCCCC1=O 13367,CC(C)CC(C)(CNC(C1CC(=O)NC(=O)N1)=O)NC(C1CC(F)(F)C1)=O 13368,C1(C(=O)NC2CC(C)(NC(c3n(C)ccc3)=O)C2)CCC(=O)N1C1CC1 13369,C1(OCC(=O)NC2CC(NC(Cn3ncc(C(=O)OC)c3)=O)C2)CCCCC1C 13370,C1(NC(C2=C(C)CC2)=O)CN(C(c2csc(CO)n2)=O)CC(F)(F)C1 13371,CCC(CC(=O)NCC1(O)CCN(C(C2(COC)CC(C)(C)C2)=O)C1)CC(C)C 13372,C1(=O)CC(NC(C)=O)C(=O)NC1CC(O)(COC)CNC(=O)CCCC(C)=O 13373,N1(C(=O)OC(C)(C)C)CCC(CC(N2CC3CC3(CO)C2)=O)C(C)(C)C1 13374,Cc1cc(C)c(C(=O)NCCC2CN(C(C3CNC(=O)N3C)=O)CCO2)c(C)n1 13375,CCN=c1[nH]c(C)c(C(=O)NC(C2(CNC(=O)Cn3nc(C)oc3=O)CC2)C)s1 13376,c1(C(N2CC(C(=O)NC(CN(CC)CC)C)C(OC)C2)=O)ccc(C#N)n1C 13377,c1(C(N2CCC(NC(CC(CC)C)=O)C(F)C2)=O)cc2nc(C)ccc2o1 13378,c1(C(=O)NCC2CC3CN(C(C(C)=CC4CC4)=O)CC32)cc2ccc(F)cc2o1 13379,c1(C(=O)NCCCCCNC(C(C)OCC2CC2)=O)ccc(Br)cc1O 13380,C1(CC)CN(C(C2CN(C)CCN2C)=O)CCC1NC(c1cnc(C(N)=O)s1)=O 13381,N1(C(C(C)NC(C2CN(C)C2)=O)=O)CC(=O)NC(=O)C1C 13382,c1(OC(C)C)ccc(CCC(=O)NCC2CSCCS2)cc1 13383,CC1(C)OC(=O)NC1C(=O)NC1COCCC1NC(C1CC(F)(CF)C1)=O 13384,c1(C(C)NC(=O)NCCCCl)ccccc1C(=O)Nc1cc(O)ccn1 13385,c1(C(=O)NCC=CCC(=O)NC(COC)(C)C2CC2)ccn(C)n1 13386,N1(C(c2cccc(Cl)n2)C(=O)NC(CC)(C)C)CCC2(CC=CCO2)C1 13387,C1(F)(C(N2C(CN(C(=O)C=CC=C(Cl)Cl)C)COCC2)=O)C(C)(C)C1(C)C 13388,C(C(CC(C)C)NC(C1CC(=O)N(C)C1)=O)NC(C=CC=CC)=O 13389,c1(CC)onc(C(=O)NCC2C=CCN2C(=O)C(O)C(C)C)c1C 13390,c1(C(=O)OCC)ccc(C(=O)NCCNC(C2(C)CCOC2)=O)cc1 13391,C1(CNC(C(C)CC2CCCC2)c2nnnn2C2COC2)CCCCS1(=O)=O 13392,c1(CNC(=O)COCCCCCC)cccc(-n2cc(-c3ccncc3)nn2)c1 13393,N1(C(C(c2scc(C)n2)(F)F)=O)CC(NC(c2cc(Cl)ccc2O)=O)CC(O)C1 13394,N1(CCC)CCCC(C(=O)NC(C)(C)CNC(c2c[nH]c(=N)o2)=O)C1 13395,N1(C(C(C)N2CCC2)=O)CC(CNC(=O)Cc2ccc(F)nc2)CC1(C)C 13396,C1(Br)(C(=O)NCC(C)N(C(c2cc(CC)on2)=O)C)CC12CCC2 13397,c1(C(=O)NC(C(C)C)CNC(=O)COCC(F)F)cn(C)nc1C(C)(F)F 13398,Cc1ncn(CCNC(c2conc2C(C)NC(=O)CCC2CC2(F)F)=O)c1C 13399,C1(C(N(C2CC(NC(C(SC)SC)=O)C2)C)=O)CCCC2(CC2)C1 13400,c1(N2CC(CNC(=O)C(F)CC3CCCC3)OCCC2)nc2ccc(F)cc2o1 13401,c1(CC(=O)N(CCC(C)NC(COCC(=C)C)=O)C)ccc(S(=O)C2CC2)cc1 13402,C#CCC(C)(C)C(=O)N1CCOC(C(C)NC(=O)Cn2ccc(C)c2)C1 13403,CC(O)C(C(=O)NCC1CCCCN1C(c1coc(C(F)F)c1)=O)N(C)C 13404,c1(C(N2CCC(CN(C(CC3C(C)CCO3)=O)C)CC2)=O)cc(S(C)(=O)=O)cs1 13405,N1(C(CCCCSC)=O)C2CC1CN(C(=O)CCP(C)(C)=O)C2 13406,c1(CCC(=O)NCC(C)(C2CC2)NC(C2(F)CCCCC2)=O)nc2ccccc2[nH]1 13407,N1(C(c2ccc(CC)[nH]2)=O)CC2CC2(CNC(=O)CC2CCC(=O)N2C)C1 13408,c1(C(=O)Nc2nc(C(=O)OC)n(C)c2)ccc(OC)nc1NC(C)=O 13409,Cc1ccc2[nH]c(C(=O)NCCN(C(=O)COC(C)C)C(C)C)cc2c1F 13410,Cc1nc(N(C)CCOCCNC(=O)C(C)(C)CNC(N)=O)cc(Cl)n1 13411,C(=O)(CCCCC(F)(F)F)NC1CC(NC(c2cc(C3CCC3)[nH]n2)=O)CC1O 13412,c1(OC)ccc2c(c1)C(C(=O)NCCCNC(c1cnc(C(N)=O)cn1)=O)CC2 13413,C(=O)(CC(C1CC1)NC(=O)C=Cc1ccco1)N(C1CCOC1)CC 13414,N1(Cc2nnc(C(C)C)o2)CCCOC(CNC(c2occ3c2CCC3)=O)C1 13415,CC1CCN(C(C23CC(C)(C2)C3)=O)CCN1C(=O)C(Cc1ccccc1)N(C)C 13416,C1(NC(c2c(COC)noc2)=O)CC(CO)N(C(=O)CSCc2ccncc2)C1 13417,Cc1cc(NC(=O)C=Cc2ccccc2)ccc1NC(C1CCCC2CC12)=O 13418,C=CCCCCCC(=O)NCC(CCCC)NC(=O)CN1CCCCC1=O 13419,N1(c2n(CC=C)c(C3CC3CC)nn2)CCCC(n2ccnn2)CC1 13420,C1(NC(C(C)(F)CC2CCCC2)=O)CCCC2CN(C(=O)CC(=O)N(C)C)CC12 13421,C#CC1(C(=O)NCc2ccncn2)CCN(C(=O)C(=O)C2CCCC2)C1 13422,Cc1noc(C(=O)NC2CCC2CNC(c2cnccc2C(F)(F)F)=O)c1C 13423,c1(CC(=O)NCC(C(C)(C)C)NC(=O)CCNS(C)(=O)=O)c[nH]c(=N)nc1O 13424,C1(N(C(CCOCC#C)=O)C)CCN(C(=O)C=C(CCC)CCC)CC1C 13425,C(=O)(C(CCNC(=O)CCCCC1CC1)OC)N(C1CCN(C)C1)CCC 13426,C(=O)(C(C)OCC1CC1)NCC(=CC(=O)N(CC(C)N(C(C)=O)C)C)C 13427,C1(CC(=O)NCC(C2CCC2)NC(c2coc(O)n2)=O)(COC)CCCC1 13428,c1(C2(NC(C3(CNC(CCC(C)C)=O)CCCC3)=O)CC2)ccc([N+](=O)[O-])cc1 13429,NS(=O)(=O)CCCC(=O)NCCC1CCCCN1C(=O)CCN1CCCCC1 13430,N1(C(C(C)N(C)C(C2C3CCCCC23)=O)=O)CCC12CC(CO)C2 13431,C1(NC(CC(=O)NN2CCN(CCO)CC2)=O)C2CCC(C2)C1c1ccccc1 13432,C(=O)(C1=CS(=O)CCC1)N(CCC(C)NC(C1CN(S(CC)(=O)=O)C1)=O)C 13433,c1(C(=O)NCC2(F)CCN(C(CN3C(C)CCC3)=O)C2)nc2ncccn2n1 13434,c1(C(=O)NCC(CNC(c2ccon2)=O)OC)nc2ccccc2nc1O 13435,C1(SC)CN(C(=O)CCc2cncs2)CC1NC(=O)CN1CCCCCC1 13436,C(C)(C)(CC(=O)N1CCCC1CC(F)F)n1cc(CCN(CC)CC)nn1 13437,c1(C(N(C(C)CN(C(=O)CCCCc2cnc[nH]2)C)C)=O)cnc2ncccn12 13438,c1(CCC(=O)N(C)CC2CCN(C(=O)CCSC(F)(F)F)C2)cccc(O)n1 13439,C#Cc1cnn(CC(=O)NCC2CC2CNC(c2ccc[n+]([O-])c2)=O)c1 13440,C#CCC(C)(C)C(=O)NC1CCC(CNC(C2CCCOC2)=O)C1 13441,c1(C(N2CC(O)(CNC(c3cnn(C(F)F)c3)=O)C2)=O)ccc2cc[nH]c2c1Br 13442,c1(C(=O)NCCN(C(=O)CCC2CCCCC2)CC)nn(C)cc1SC 13443,C1(N2CCNC2)CCN(N2CCC(c3cccc(Cl)c3)C2)CC1.CS(=O)(=O)NC 13444,CC(C(C(=O)N(C1(C)CCCC1)C)N(C)C)C(C)(C)C 13445,C1(F)(C(N2CC(OC)C(OC)C2)=O)CCN(C(c2ccc(O)nn2)=O)C1 13446,c1(N2CC3CC(CNCCSc4cn(C)nc4)C3C2)nc(Cl)nc2ccccc12 13447,C=CCCCC(=O)NCCS(=O)(=O)Cc1cn(CCCN2CCCC2)nn1 13448,c1(C(N(C)CC2CCN(C(C3CCC(F)(F)C3)=O)C2)=O)cc2ccncc2s1 13449,c1(CC(=O)NC2CN(C(c3c[nH]nn3)=O)C3C2C3)cc(C)ccc1OC.CCOC 13450,C(N=c1[nH]c(=NCc2cc(F)ccc2C)c2[nH]ccc2[nH]1)c1cc(C)c(C)s1 13451,C(=O)(C(F)(F)C1=CCOCC1)NCC#CCNC(=O)COCC1CCOC1 13452,C(=O)(CC(C(F)F)NC(C1(n2cccc2)CC1)=O)N1CC(O)(CCC)C1 13453,c1(N(C)C)cccc(NC(=O)Nc2ccccc2OCCCn2ccnc2)c1 13454,c1(C(N(C(C)CN(C)C(C2(CF)CC2)=O)C)=O)nccc(Br)c1O 13455,c1(C(N(CCCCN(C(=O)CCc2ccn(C)c2)C)C)=O)csc(C(C)(F)F)n1 13456,C1(C(=O)NCCOCC(=O)N(C2CCN(C)C2)C)(OC)CC(C)(C)C1 13457,C(C(CC(C)C)C(=O)N1CC(n2cc(C(C)(C)O)nn2)C(O)C1)C1C(C)C1 13458,C1(C)(C(=O)NCc2c(C(=O)NCc3ncc(CC)s3)[nH]cc2)CCC2CC2C1 13459,N(C(=NCC1CCCO1)NC1CCN(c2ccc(F)cc2)C1)CC1(C)CCCS1 13460,c1(OC)ccc(C(=O)Nc2cccc(CNC(=O)C(F)(F)C(F)F)c2)c(C)n1 13461,CC(C)C(C#N)C(=O)N1CCC(NC(c2cnc(-c3cnccn3)s2)=O)C12CC2 13462,c1(C(=O)NC23CC(C(N(C4(C#C)CC4)C)=O)(C2)C3)cccc(O)c1 13463,CC#CC1CN(C(C2OCCC2NC(c2snnc2CC)=O)=O)C1 13464,C(CC1=CCN(C(C2(C)CC2C(F)(F)F)=O)CC1)NC(CC(CCC)O)=O 13465,N1(C(c2cnc(C)c(Cl)c2)=O)CC2CC1CCN2C(C1CCSC1)=O 13466,c1(C(N2CCC(N(C)C(c3ccccn3)=O)C2)=O)ccc(CO)nc1 13467,N1(C(C)=O)CCC(C)N(C(=O)CCOC(C)C)CC1 13468,O=C(C1=CCCSC1)NCCCCCCNC(C1COCC1C(F)F)=O 13469,C1(C(=O)NCCN(C(C)=O)CC)CCCCN1C(C1(C2CCC2)CC1)=O 13470,c1(C(=O)NCCCNC(C2C(CC)CCN2C(C)=O)=O)cc2cccnc2cn1 13471,C1(C(=O)NCc2nc(CC)[nH]n2)C=CCN(C(C2CCCC(=O)C2)=O)C1 13472,N1(C(C(C=C)CC)=O)CCN2CCN(C(c3c[nH]ccc3=O)=O)CC2C1 13473,N1(C(c2cc(OC)nc(Cl)c2)=O)CCOC2CCN(C(=O)C3=NNC(=O)C3)CC12 13474,C1(CCNC(Cc2c(C)n[nH]c2C)=O)CN(C(c2nn(C)cc2Cl)=O)CC(C)O1 13475,C1(N(C)C(C2CC2(C)C)=O)CN(C(=O)Cc2ccc(Cl)cn2)CC1(C)C 13476,c1(C(=O)NC2(C)CCN(C(Cc3c(C)occ3)=O)C2)ncnc2c1CCC2 13477,c1(OCC)ccc2nc(N3CC(CO)(NC(=O)C(C)CC(C)CC)C3)sc2c1 13478,c1(CNC(C(C(C)(C)C)O)=O)ccc2c(c1)CN(C(=O)C1=CCCOC1)C2 13479,N1(C(Cc2n(C)nnc2)=O)CCC=CC1C(N1CCOC(CC(N)=O)C1)=O 13480,N1(C(N(c2ccc(C)c(C)c2)C)=O)CCCc2ccc(Br)cc2C1 13481,CN1CC=C(C(=O)NCCC(c2ccccc2)N(C)C(C2CC3(CSC3)C2)=O)C1 13482,c1(C(N2CC(C(N)=O)(CNC(C(C)C3CC3)=O)C2)=O)ccnc2[nH]c(O)nc12 13483,c1(OC)ccc(-c2cncc(C(=O)N(C)CCN(C)C(C3CC3Cl)=O)c2)c(C)c1 13484,Cc1[nH]nc(Cl)c1C(=O)NCC1CC(NC(=O)CCc2cn(C)nn2)CCO1 13485,N1(C(C(CC)(C)OC)=O)CCOC2(CCCN(C(=O)C=CC3CCCC3)C2)C1 13486,c1(C(C)C)ccc(C2CCN(C(=O)CN3CCCCC3)CC2)cc1 13487,c1(CC(C(=O)N(CCOCCCN(C(CCC=C)=O)C)C)O)ccc(OC)cc1 13488,Cc1cc(=NC(C)CCC2CCCCC2)[nH]c(=NCC=CBr)[nH]1 13489,c1(C(=O)NC2CC(CNC(C3=CCCC3C)=O)C2)n[nH]c2c1CCSC2 13490,C1(C(=O)NCC2(C)CC(NC(C3(OC)CC3)=O)C2)CC(c2ccccc2)=NO1 13491,c1(C(=O)NC2C(CNC(C(OC)OC)=O)COC2)cc2ccccc2s1 13492,N1(C(C2CCSCC2)C(=O)NCCOC)C2CCC1CC(CO)C2 13493,C1(NC(C(N2CCC(C)(CCO)C2)c2ccncc2F)=O)CCC(F)(F)CC1 13494,CC(C)(O)C(C)(C)C(=O)N1CC2CC(NC(C3CCCC3)=O)C1C2 13495,C1(C)(OCC(=O)NCC2(CN(C(=O)CCCc3nncn3C)C)CC2)CCCC1 13496,C(=O)(CC(CC(C)C)NC(c1cc[nH]c1C)=O)NCCC(CC)O 13497,c1(C(=O)NCC(CNC(CCCCC=C)=O)O)cc2c(C(F)(F)F)cccc2s1 13498,C(=O)(C#Cc1ccccc1)N1CC2C(C(=O)Nc3cc(OC)ncc3Br)C2C1 13499,C1(CNC(CCN(C(C2(C(C)C)CCCC2)=O)CC)=O)CC(C)CC(C)C1 13500,CC#CCC(C)NC(C1(CCNC(=O)CC(Cl)Cl)CC1)=O 13501,c1(C(=O)NC2CC(CNC(C3C(C)CC(=O)N3)=O)C2)cc(N)cnc1Cl 13502,c1(C(N2CC(NC(=O)C(F)C3CCC3)(CO)C2)=O)cncc([N+](=O)[O-])c1 13503,C1(C(F)(F)F)(C(N2CC(OCC(N3CCOCC3)=O)(CO)C2)=O)CC2CC2C1 13504,C1(C(=O)NC2CC(NC(c3c(C)n[nH]c3)=O)CC2O)C(F)(F)C12CCC2 13505,c1(C(=O)NC2CN(C(C3C(COC)(COC)C3)=O)C(C)(C)C2)ccc2nccn2c1 13506,C(C1=CCCOC1)NC(C(c1cccs1)NC(c1cc(CO)on1)=O)=O 13507,N1(C(C2C(=C)C2)=O)C2CCC1C(CNC(=O)C(F)F)C2 13508,Cn1ccc(C(N2CC(O)(CNC(=O)C(O)c3ccsc3)C2)=O)c1C1CCC1 13509,C(C)(C)(CCNC(c1cnc(C(C)(C)C)o1)=O)NC(C1CC(CN(C)C)C1)=O 13510,c1(C(=O)NC2CC(F)(CNC(C(C)C3CCOC3)=O)C2)[nH]nc([N+](=O)[O-])c1Cl 13511,CC1C(NC(=O)CN2C(=O)CCC2=O)CCN1C(=O)Cc1ccccc1Cl 13512,N1(C(c2n(C(C)C)ncc2)=O)CCSC(C(=O)N(CCO)CCO)C1 13513,C#CC1(NC(C2CN(C(C3CCC3(OC)OC)=O)CCO2)=O)CC2CCCC12 13514,C12(CNC(C3C(OC)C3)=O)CC1CN(C(c1ccoc1C)=O)C2 13515,C(=O)(C(CC(C)CC)NC(=O)CCC1CCC1)NCC1(CCC=C)CC1 13516,N1(C(c2c(CC)n[nH]c2)=O)CC2CC2(CNC(=O)C(O)CC2CC2)C1 13517,n1(CCC)cc(S(=O)(=O)NC(c2ccc(O)nc2)C)cn1 13518,N1(C(c2c(C)nc[nH]2)=O)CC2CCCC1(CNC(C1CCCN1C)=O)C2 13519,N1(C(C(CC)O)=O)CCCC(N(C)C(c2ccnc(OC)c2)=O)C1 13520,CCCCCC(C)CC(=O)N(C1CC(NC(C2C=CCS2)=O)C1)C 13521,C(=O)(CC(C)(C)O)NC(C(N1CC(OCC(C)C)C1)=O)C1CCCC1 13522,Cc1cc(CCNC(=O)C(Cn2cncn2)NC(=O)CC2CCOC2C)n[nH]1 13523,C(=O)(C(CC(C)C)N(C(=O)C(C1(O)CCCCC1)(F)F)C1CC1)OC 13524,C1(C(N2C(C)CCN(C(C=C(C)C(F)F)=O)CC2)=O)CCc2ccc(F)cc2O1 13525,Cc1noc(C)c1CC(N1CCC(C)(CCNC(c2cnnn2C)=O)C1)=O 13526,c1(C(N2CCC(O)(C(C)NC(CCC)=O)C2)=O)ccc(Cl)nc1OCC 13527,C(=O)(CCC(=O)N1CCC(C(C)(O)CNC(=O)C(C)SC2CC2)CC1)NC 13528,C1(CN(C)C(C2(C)CCC2)=O)CCCN(c2nc(Cc3ccccc3)ns2)C1 13529,C1(C)(C(=O)NCC(N2CCCCC2)C)CN(C(=O)C=CCN2CCC2)C(C)(C)C1 13530,C1(N)(C(=O)Nc2cc(COC)c(OC)cc2)CCC(C)(C)CC1 13531,CC1CCC(NC(c2nn[nH]c2Cl)=O)CN1C(=O)CCCCc1ccccc1 13532,c1(OC)ccc(C(=O)NCCC2CCCN(C(=O)CCC(C)N(C)C)C2)c(N)c1 13533,Cn1nc(Cl)c(C(N2CC(C(F)(F)F)C(CNC(C3CCOC3)=O)C2)=O)c1Cl 13534,N1(C(C(CC(=C)C)C)=O)C2CCC1CC(N(C)C(c1ccc(Br)s1)=O)C2 13535,N1(Cc2c(C)scn2)CC2CN(c3nccc(-c4cccnc4)n3)CC12 13536,c1(C(=O)NC2C(C(=O)NCC3CCC3)CCCC2)cc(Br)cc([N+](=O)[O-])c1Cl 13537,CCC(CC(=O)NC1(CNC(C2CCCSC2C)=O)CCC1)c1ccccc1 13538,c1(C(=O)NC2CCN(C(=O)C=Cc3cc[nH]n3)CC2)ccc(Br)cc1[N+](=O)[O-] 13539,C1(C(=O)NC(C2CCN(C(Cc3c(C)nc(C)s3)=O)C2)C)CCCCC12CCC2 13540,C(=O)(C1CCCc2ncccc21)N(CCCNC(C1CC2(CC2)C1)=O)C 13541,c1(NC(C2CCN(Cc3cccc(-c4nn[nH]n4)c3)C2)=O)cc(Br)ccc1Br 13542,C1(NC(C2CC(=C3CCC3)C2)=O)C2CCC1N(C(c1cnccc1Cl)=O)C2 13543,N1(C(C(COCC)C)=O)CCN(C(c2cnn(C)c2C2CC2)=O)CC1C(C)C 13544,N1(C(CC2(CSC)CC2)=O)CC(NC(=O)C(C)C(C)O)CC12CCCC2 13545,N1(C(C2COCC(C)(C)O2)=O)CC2(CCC(CNC(C3(CCF)CC3)=O)O2)C1 13546,C1(NC(CCCCOC)=O)COC2(C1)CN(CCc1c(C)noc1C)C2 13547,N1(C(C2CC(CNC(CCCN(C)C)=O)C2)=O)CCCC(F)(CO)C1 13548,C1(NC(C(CC)(C)OC)=O)CCCCN(C(c2ccc(C)nc2N)=O)C1 13549,CONC(=O)C(=O)N1CC(F)CC1CN(C(=O)CN(C)C(C)C)C 13550,N1(C(C2C(C(C)C)OCC2)=O)CC2CC(NC(=O)Cc3ccc(F)cc3)C1C2 13551,N1(C(c2cn(C)nc2)=O)CCC(CNC(c2ccc3n[nH]cc3n2)=O)C12CCC2 13552,N1(C(C(CO)NC(C)=O)=O)CCn2nc(C(=O)N(CC(O)CO)C)cc2C1 13553,N1(C(CCC(C)OC)=O)CCC(NC(=O)CSc2ccncc2)C(F)C1 13554,CC(CF)CC(=O)NCC1CC1CNC(c1cc(-c2ccncc2)ccn1)=O 13555,N1(C(c2ncccc2F)=O)CCN(C(C2(C(F)F)CCOCC2)=O)CC1C(F)F 13556,c1(C(N(CCNC(=O)C(C)=C2CCC2)CC)=O)cnn(-c2ccncc2)c1C 13557,c1(C(N(C2CCCC2)CCCNC(C2C(C)(C)CC2)=O)=O)cc[n+]([O-])cc1 13558,c1(C(=O)NCC2C=CCN2C(=O)CC2CCCOCC2)ccc(F)cc1Br 13559,C(N=c1[nH]cnc2ccc(O)cc12)C1C(NC(c2n(CC)ccn2)=O)CCCC1 13560,n1(C(C)C)ccc(C(=O)NC(C)(C)C(=O)NC(C2CCC2)C)n1 13561,CC12COCC1CN(C(N1CCCC1C(O)C(F)F)=O)C2 13562,c1(CC(=O)NCC2N(C(CC(=O)NCC#C)=O)CCC2)cccc(C)c1Br 13563,N1(C(c2n(CC)ncc2Cl)=O)CCN(C(=O)CCc2ccoc2)C(C)CC1C 13564,C1(CC)CCCC(N=c2nc3scnc3c(NCc3c[nH]nc3C3CC3)[nH]2)CC1 13565,c1(C(=O)NC(CC)CN(C(=O)CSCc2cccnc2)C)cn(C)nc1C(C)C 13566,C1(NC(C(C)C=Cc2ccccc2)=O)CN(C(=O)CCCC2CCC2)CCC1C 13567,Cc1nn(C)c(Cl)c1C(=O)NCC1CC2CC1CN2C(=O)CC1CC2(CC2)C1 13568,Cn1nc(CNCCC(O)C(F)F)cc1NC(C1CCCCC1)=O 13569,C1(CNC(CSCCC)=O)(CNC(C2CN(c3nncs3)C2)=O)CC12CCC2 13570,N1(C(c2n(COC)ncc2)=O)CCC(C)C(CNC(c2nc(Cl)cs2)=O)C1 13571,N1(C(c2c(C)ccnn2)=O)CC2(CC(NC(C34CC3COC4(C)C)=O)C2)C1 13572,c1(C(N(CCNC(c2nn(C)c(C3CC3)c2C)=O)CC)=O)cc2n(n1)CCC2 13573,c1(CC(=O)N(CCNC(=O)CCn2cnnn2)CC)cc(Cl)ccc1Br 13574,c1(OC)[nH]c(=NC2CCCCCN(C(=O)C(=O)NC(C)C)C2)sc1C 13575,C1(CNC(C(=O)NCCOCCCC)=O)CN(C(=O)C=NOC)CC12CCC2 13576,N1(C(C2(C(=O)OC)CC2C)=O)CC2CCCN(C(=O)C(C(C)C)NC(N)=O)C2C1 13577,CC(CCCC(=O)NCc1ccnc(Cl)c1)NC(c1ccccc1C1CC1)=O 13578,C1(C)(C(=O)NCC2CC(NC(C3CC(C(=O)OC)C3)=O)C2)CCCNS1(=O)=O 13579,c1(N(C(=O)OC(C)(C)C)C2CC2)cnn(C)c1.C1(=O)CCN(C)CC1=O 13580,c1(CCC)[nH]ccc1C(=O)N(C1(CC(=O)NC2(CC(C)C)CC2)CC1)C 13581,c1(C(C(N2C(CNC(c3cc(I)on3)=O)CC2)=O)F)ccc(C(F)(F)F)cc1 13582,Cc1csc(=O)n1CCC(N1CC2CC2(NC(=O)COCCF)C1)=O 13583,C1(C(=O)NCC2OCCN(C(c3onc(CC)n3)C)C2)Cc2ccccc2O1 13584,N1(C(C2C3CCCCC23)=O)CC2C(c3cn(Cc4ncc(F)cn4)nn3)C2C1 13585,C1(N(C(C2CSC2)=O)CC)CCCN(C(c2ccc(O)c(Cl)c2)=O)CC1 13586,c1(CC)ncc(C(=O)NCC2(COC)CN(C(C3CC4C=CC3O4)=O)C2)c(O)n1 13587,C1(C(N2CCCCC2)=O)CCCN(C(=O)CN(CC2CCC2)CC2CC2)C1 13588,C1(OC(C(=O)NC(C(CO)SC)C)C)CCCN(C(=O)OC(C)(C)C)C1 13589,Cc1cc(C(=O)N(C)CC2CCN(C(=O)C#CC(=O)N(C)C)CC2)ccn1 13590,C1(NC(Cc2ccc(C)nc2)=O)CCCN(C(=O)CC(O)C(C)C)CC1 13591,C1(OC)CCC12CC(C(=O)NC1CC(CNC(=O)C3=CCCSC3)C1)C2 13592,c1(C(N2CCC(C(C)C(=O)NCC(C)(C)O)CC2)=O)ccc(C#N)cn1 13593,c1(C(=O)NCC2CC(NC(C3C(OCC)C3C)=O)C2)cnc2c(c1)nnn2C 13594,n12nc(cc1C)C(=O)NCCOCCCNC(=O)C2.C12(CC1)C(=O)N2.CC.SC 13595,Cc1coc(C)c1CNC(=O)C(C)N(C(c1ccccc1)=O)C1CC1 13596,N1(C(C)=O)CCCC1C(=O)NC(C1CCCN1C(=O)CC1CCCO1)(C)C 13597,c1(OC)cnc(Br)cc1C(N1CCN(Cc2cnn(C)c2)CC1CC#N)=O 13598,C1(C(N2CC(O)(CNC(c3c(C)cc[nH]3)=O)C2)=O)C2C(=O)OCC12Br 13599,c1(CC(=O)NC2CC(NC(=O)C(F)=CC3CC3)C2)noc2ccccc12 13600,Cc1cc(C(=O)NC2CCCC(NC(C3C4CCCOC34)=O)C2)cc2ccsc12 13601,C(c1ccccc1)=C(C)C(N1CC2CC2(C(=O)NCC2=CCCC2)C1)=O 13602,C1(CC(=O)NC2CN(C(c3cn(CCO)nn3)=O)C2)CC(=O)c2ccccc2C1 13603,C#Cc1ccc(NC(C2CC(F)(F)CN2c2cc(C(F)(F)F)ncn2)=O)cc1Cl 13604,C1(CNC(C2C(CC)OCC2)=O)CCN(C(=O)CN2CCNC(=O)C2)C12CC2 13605,CN1CCC(CCC(=O)NCCC2CCCN2C(c2cc(C3CC3)on2)=O)CC1 13606,N1(C(C2(SC)CN(C(c3c(CC)cccc3)=O)C2)=O)CC2CC(CO)C(C2)C1 13607,C1(NC(N(CC(C)C)CCn2cc(C(NCC)=O)cn2)=O)CCCC12CC2 13608,C1(NC(Cn2ncn(C)c2=O)=O)CCN(c2cc(C(F)F)ncn2)CC1O 13609,C(=O)(C(C)(CC)CCC)NC(CCNC(C1(CC#C)CCC1)=O)C 13610,n1(CCC)cc(C(=O)N(CC(O)CCNC(=O)CSCC(N)=O)CC)c(C)n1 13611,C(=O)(CCC(=O)NC)NC(C1CCC(C(N2CC(CSCC)C2)=O)C1)=O 13612,C=CC1CN(C(=O)CN(C2CC2)CC)CC1NC(=O)C(F)(F)C1CCOCC1 13613,C1(C(=O)NC(c2ncc(C)o2)C)CCC2(CC2)N1C(c1nn(C)cc1C)=O 13614,c1(C(=O)NC2C(NC(c3cccc(CC)c3)=O)CCCC2)cc(Cl)cc(F)c1N 13615,C1(C)(c2n(CC)ccn2)NC(=O)N(CC(O)COc2ccc3c(c2)CCC3)C1=O 13616,c1(CC2CCNCC2)cn(CC(=O)NONC(=O)C(F)n2ccnc2)nn1 13617,CCC(CC(C)C)C(=O)N(C)CC1CN(C(c2ccccc2C(N)=O)=O)C1 13618,CC1CCC(C(=O)N(C)Cc2nnnn2C)N1C(c1ccn(C)n1)=O 13619,N1(C(c2[nH]c(=NC)sc2)=O)CC(N(C(=O)C(C)SC(C)C)C)C(C)(C)C1 13620,C=CCCCC(C(=O)NCC(Cl)Cl)NC(=O)OC(C)(C)C 13621,Cc1ncc(C(=O)NC2CN(C(c3c(C)noc3C3CC3)=O)CC2C)cc1C#N 13622,CCCC(C(=O)N1CC(NC(C2(C3CCCCO3)CCOCC2)=O)C1)OCC 13623,c1(C(=O)NC(C)CNC(=O)C(c2cnn(C)c2)=O)c(F)ccc(C(F)(F)F)c1F 13624,N1(C(c2cnc(OCC)s2)=O)CCCC(O)(CNC(=O)C2=C(Cl)CCOC2)CC1 13625,Cc1cc(NC(c2ccc(CNC(c3cnns3)=O)s2)=O)c(O)cc1F 13626,c1(CC)ccnc(CNC(=O)CC2CC(NC(c3cc(OC)ccn3)=O)C2)c1 13627,C12(CNC(C3C(OC)C3)=O)CC1CN(C(C1CCN(C(=O)C(C)(C)C)CC1)=O)C2 13628,N1(C(CCC(C)C)=O)CCCC2C1CCCCN2C(=O)CCc1cccn1C 13629,C(=O)(C(F)C(F)(F)F)N(C1CCN(c2cc(CC)ncn2)CC1)Cc1sccc1C 13630,N1(S(=O)(=O)CC2CC2)CCCC2C1CCN2Cc1cc2ccncc2[nH]1 13631,C12(CNC(C=CC(C)(C)C)=O)CCC(CC1)CN2C(C1CC12CCC2)=O 13632,N1(C(CC(=O)OC)=O)CC(C(=O)Nc2c(CO)noc2C)CC12CCC2 13633,C1(CC)C(NC(=O)C(CO)N(C)C)CCN1C(c1ccncc1SC1CC1)=O 13634,CC1=C(C(=O)N2CC(CNC(=O)CN3CCSCC3)CC(C)C2)CCCO1 13635,CCC(CC(=O)N1CC2CN(C(c3c[nH]c(=NC)o3)=O)CC2C1)C(C)C 13636,N1(C(=O)CC2CCC3CC3C2)CC23CCCC2(C1)CN(C(C1CCC=CO1)=O)C3 13637,C1(CNC(Cc2nccc(C)c2)=O)C(C)CCCN1C(c1ccc(C)cc1F)=O 13638,C(C(C)(C(C)C)C(C)C)NC(CC1C(C)CN(C(=O)C=Cc2nccs2)C1)=O 13639,c1(C(=O)NC2CN(C(CCc3ccn(C)c3)=O)C3C2C3)ccc2cc[nH]c2n1 13640,c1(OC)cc(C(=O)NC2CCC(NC(=O)Cn3ncnn3)CC2)ccc1[N+](=O)[O-] 13641,c1(C(N(CCNC(CCC(N)=O)=O)C2CC2)=O)cc2c(O)ncnc2cn1 13642,c1(CC)nccnc1C(N1CCCC1(C)C(=O)NOCCOCCF)=O 13643,C(C(C)(C)C(=O)N1CCC1CNC(C1(C)CCC(C)C1)=O)OC(C)C 13644,c1(C(N(C(CNC(C2CN(C(C)=O)C2)=O)C)C2CC2)=O)ccc(C)c(Br)c1 13645,Cc1ccc(C#N)cc1C(N1CC2CC1CCC2NC(=O)C(F)(F)C(F)F)=O 13646,C1(NC(c2c(F)ccnc2F)=O)CCN(C(=O)CCc2cc[nH]n2)CCC1CO 13647,Cc1conc1CC(=O)N(CC(=O)N(C)Cc1cccnc1)CCO 13648,N1(C(CC2CC(OC)C2)=O)CC(CC(N2CCCC(CCF)C2)=O)CC1C 13649,c1(C(N(C(C)CCNC(C2SC3C=CC2CC3)=O)C)=O)cc2ccc(Cl)cc2o1 13650,c1(CCC)cc(C(=O)NC2CCCCC2NC(=O)CC2CC(C)(C)C2)cc(O)n1 13651,c1(C(=O)NC(C2CCCCN2C(=O)C(C)(F)F)C)ccccc1OCC(N)=O 13652,c1(SC)cccc(C(=O)NCCN(C(c2cnc(S)[nH]2)=O)C2CC2)c1 13653,c1(C(CNC(=O)CCn2cccn2)NC(CNS(NC)(=O)=O)=O)ccccc1Cl 13654,Fc1ccc(F)c(NCC2CCCC(C(F)(F)F)C2)c1F 13655,C(=O)(C(C)(C)C(N)=O)NCCC1C(C)CN(C(=O)COCc2cccnc2)C1 13656,c1(NC(C2C(C(=O)OC)C2)=O)ccc(C(=O)Nc2cnc(O)cc2C)cc1C 13657,Cc1cc(C(=O)NC2CCCN(C(C3CCN(C)C3)=O)C2)cc([N+](=O)[O-])c1O 13658,c1(OC)ccc(CC(=O)NC2CC(C)(NC(=O)CCc3ccccn3)C2)cn1 13659,C(=O)(C1=CC2(CCN(C(=O)CCSC)C2)C1)N(CC=C)CCN.C(CC)SC 13660,C1(CNC(Cc2scc(C)c2)=O)CCCN(CC(N2CCC2)=O)C1 13661,C(=O)(C(C)CC(C)CC)NCC(CCC)C(=O)NC1CCC(O)C(O)C1 13662,n1(CC(C)NCCCC(C)(C)CO)cnc2c(cnn2C)c1=O 13663,N1(C(c2c(CC)c[nH]n2)=O)CCC2C(C(=O)NC(c3noc(C)n3)CC)C2C1 13664,CN1C(=O)C(F)CC1C(N1CCCC1(C)CNC(=O)CCN1CCCCC1)=O 13665,CCCCCCCC(=O)N1CC(C)(NC(c2cccc(C3CCCOC3)c2)=O)C1 13666,C(=O)(C(C)CCCC)N1CC(CC(=O)NCC=CC)OCC1 13667,CCCC(O)(CCC)CC(=O)NC1CC(O)(CNC(C2CCC23CCC3)=O)C1 13668,N1(C(Cc2c(C)non2)=O)CC(NC(=O)CCC2CCCC2)CCC1C 13669,C=CC(F)(F)C(=O)NCC(O)CC(=O)N(C)CC1CCOC1C 13670,c1(C(=O)NCC2CCN(C(c3cn(CC)nn3)=O)C2)ccc2[nH]c(=N)sc2c1 13671,C1(CNC(c2n(C)c(O)nc2)=O)COCCN(C(c2csc(C#N)c2)=O)C1 13672,C1(C(N2C(C(=O)NC3CCCC3CF)CC(OC)C2)=O)CC2(CCC2)CO1 13673,N1(C(C2CN(C)C(=O)N2)=O)CCOCC(C(N2CCN(C)C(=O)C2)=O)C1 13674,Cc1nc(C2CC2)oc1C(=O)NCC(O)CCNC(C1(C)CC(F)C1)=O 13675,C1(CC#C)(C(=O)NCC(c2cccc(Br)c2)C)CCCNC1 13676,N1(C(CN2C(C)CCCC2)=O)CC(C(N2CC(CCO)C2)=O)C2(CCC2)C1 13677,N1(C(c2ccc(C)o2)=O)CCc2nc(CNC(=O)C(C)(C)c3cnc[nH]3)sc2C1 13678,c1(C(=O)NCC2(C(=O)NC(COC)C(C)C)CC(=C)C2)cnc(C)n1C 13679,Cc1cc(C)c(C(N2CCN(C(c3ccns3)=O)CC2C(C)C)=O)cc1N 13680,Cc1cc(C(=O)NCC23CCC2CN(C(c2sccc2C#N)=O)C3)nc(C)c1 13681,C1(C2CCCC2)(C(=O)NC(CCNC(c2nc(C(C)C)sc2)=O)C)CCNC1=O 13682,C1(CNC(C(C=C)C)=O)CN(C(=O)Cc2csnn2)CC12CC2 13683,O=C1CCC(S(=O)(=O)N(CCO)CC2CCCN(C(=O)C3=COCCC3)C2)CC1 13684,Cc1ncnc(O)c1C(=O)NC1CC(C)(NC(=O)CCc2cc(F)cc(F)c2)C1 13685,C1(CC)CC(C(N2CC(NC(c3cc(C(F)F)cc(F)c3)=O)C2)=O)CC(=O)N1 13686,Cc1cc(C(=O)NCC2(O)CCCN(C(c3cc(C(F)F)cs3)=O)C2)cnc1O 13687,C12(CNC(C3C(C(N)=O)C3)=O)CC(NC(c3scnc3Br)=O)(C1)C2 13688,C(c1cccc([N+](=O)[O-])c1)=CC(=O)NC1(C)CCN(C(C2(O)CCOC2)=O)C1 13689,c1(C(C(n2cc(C(C(=O)OC)(C)C)nn2)C)NC2CC3CC3C2)cccc(Cl)c1 13690,c1(OC)sccc1C(=O)N(C)CC=CC(C(C(C)N)C)=O.OC 13691,C1(CC(=O)NCCNC(C2CN(C(c3c(C)cco3)=O)C2)=O)CC(O)C1(C)C 13692,N1(C(CCCc2onc(C(C)C)n2)=O)CCN(C(C2CCC(O)C2)=O)C(C)C1 13693,C1(CNC(C2(C#C)CC(=O)C2)=O)CN(C)CCN1C(c1cc(CC)on1)=O 13694,C(C(CC(=O)NC1CCN(C(=O)Cc2ccn(C(F)F)n2)C1)C(F)(F)F)N(C)C 13695,Cc1cc(Cl)cnc1S(=O)(=O)N1CCSC(c2cnn(C(C)C)c2)C1 13696,c1(OC)ccnc(C2CCCN2CC(=O)NC2CCC(C)CC2)n1 13697,CCC(C)(O)C(=O)N1CC2CC2(C(N2CCC(CO)CC2)=O)C1 13698,N1(C(C(CC)C#N)=O)CC(CCNC(=O)C2CC2)C2(CC2)C1 13699,Cc1cc(CNC(=O)NCCc2c(Cl)cccc2Cl)nc(Cl)c1Br 13700,N1(C(c2ncc(C)s2)C(=O)NCCCSC)CCC(C(C)(F)F)CC1 13701,N1(C(CN(CC(C)C)C(=O)CC2CCCCC2O)=O)CC2OCC(CO)C2C1 13702,N1(C(CSCCOC)=O)CCC2(C1)CN(C(=O)Cc1ccnn1CC)CC(C)O2 13703,O=C(CCCNC(C1(CNC(=O)Cn2cnccc2=O)CC2(CC2)C1)=O)NO 13704,c1(CC(N2CC(CCC)N(C(=O)C(O)C(C)C)CC2)=O)coc2cc(O)ccc12 13705,c1(C(N(C)CC2CCN(C(CSCC)=O)C2)=O)cc(C(F)(F)F)cc(Cl)c1 13706,C1(C(=O)OC)CC2CNCC2N1S(=O)(=O)CC1CNC2COCC2O1 13707,Cc1cc(=NC(Cn2ccnc2)CCO)[nH]c(C(N2CC(C)OC(C)C2)C)n1 13708,CC1(C(N2CCOC3CC23)=O)CCN(C(=O)CC2(O)CCCC2)CC1 13709,C(C(C(C)C(C)C)NC(=O)Cc1cc(C)[nH]n1)NC(CCc1cccc(C)c1)=O 13710,CN1CC(C(=O)NCCC2(O)CN(C(=O)CSC(F)F)C2)C(c2cccnc2)C1 13711,C1(C(N2CC(C=C)(CC(=O)NC(C#C)(CC)CC)C2)=O)CCC(C#N)CC1 13712,CC(F)(F)C(F)C(=O)N1CCC(N(C(C2CCCCC2)=O)CC2CC2)C1 13713,C1(CNC(CCCOCCC)=O)CC2CCC1N2C(=O)C(N)=O 13714,CN1CCn2cc(C(N3CCCC4CN(C(C5(C)CC5)=O)CCC34)=O)nc2C1=O 13715,C(=O)(C(C)S(=O)(=O)C(C)C)NCCNC(C1N(CCCC)CCOC1)=O 13716,N1(C(c2c(CC)c(C(=O)OC)c(C)[nH]2)=O)CC2CC(NC(=O)CC3CC3)CC2C1 13717,CC1CC(NC(=O)Cc2sc(O)nc2O)CN(C(=O)C(C2CCOCC2)O)C1 13718,C1(NC(=O)Nc2scc(C(=O)OC)c2)C2Cc3cc(F)ccc3C12 13719,N1(C(C2(CC(=O)OC)CC2)=O)CCCCC(N(C)C(C2OCCC2(C)C)=O)C1.C1(C)CC1 13720,CCCCCCCCOCC(N1CCCC1CN(C(C1CCC(C)C1)=O)CC)=O 13721,C1(NC(COCCN(C)C)=O)CC2CCC1CN2C(=O)CCCn1cccc1 13722,c1(C(=O)Nc2c(OC(C)C)ccc(C#N)c2)ccc2c(c1)NCCC(=O)N2 13723,C1(C(=O)OC(c2ncc(-c3ccc(Br)cc3)o2)C)(C(F)F)CNC(=O)C1 13724,C(=O)(CCCCOC)NCc1c(C(=O)NC(C2CCCOC2)CC)scc1 13725,C1(NC(c2ncc(Cl)cn2)=O)CC12CCN(C(c1ccc3cc[nH]c3c1)=O)CC2 13726,c1(NC(C(=O)NC(C2CCN2C2CC2)C)=O)ccnc(Oc2ccccc2)c1 13727,C(=O)(C(Cc1cnc[nH]1)NC(C1CCOCC1)=O)NCC(=C)Br 13728,c1(C(=O)Nc2c(F)ccc(NC(CC)=O)c2)c2c(nn1C)CCNC2 13729,c1(C(=O)NCCNC(C2C(C(N)=O)C2)=O)ccnc2ccc(O)cc12 13730,c1(C(N(C(C)CNC(c2cnc(Cl)s2)=O)C)=O)ccc2c(c1)NS(=O)(=O)C2 13731,C(=O)(C#CC1CCCCO1)NCC(c1ccccc1)CNC(C1(CC=C)CC1)=O 13732,C1(C(=O)NCCC(C)NC(C=C(C)C2CC2)=O)(CO)CCOC1 13733,c1(CNC(N2C(N3CCCC3)(CC)CCC2)=O)sccc1S(C)(=O)=O 13734,c1(C(=O)NC2CCN(Cc3ccc(C)[nH]3)CC2F)n[nH]c2c1CS(=O)(=O)C2 13735,N1(C(COC)=O)CCCC2(CCCCC2NC(=O)C(CO)NC(N)=O)C1 13736,c1(NC(C2C3CN(C(c4ncccn4)=O)CC23)=O)cc(F)ccc1I 13737,c1(N2CCCC(OC)C2)ccc(Br)c(S(=O)(=O)NCC2(C(C)C)CC2)n1 13738,C(=O)(C#CC1(C)CCCO1)N(CCN(C(C1CC(C)(CC(F)(F)F)C1)=O)CC)CC 13739,C1(NC(CCC(C)SC)=O)CCCN(C(C2CCC(C)C(C)C2)=O)C1C 13740,C1(C(=O)NCC2(C(=O)NC(CC(=O)NCC)C)CC23CCC3)CC2CCCC2C1 13741,N1(C(C(=O)Nc2ccc(C)cc2C)C)CC=C(C(C)(C)C)CC1 13742,Cn1nc(NC(=O)NC(CNC(=O)C(F)(F)Br)C(C)(C)C)cc1C(F)(F)F 13743,CCCCCC(C(=O)N1CCCCC1CNC(c1cc(C)cc(O)c1)=O)C(C)C 13744,N1(C(c2c(C)cccc2Cl)C(=O)NCCC2(C)CC2)CCOCC12CCOC2 13745,C12(C(N3C(C)(CNC(CC=C)=O)CCC3)=O)CCC(C)(CC1)OC2(C)C 13746,N1(C(=O)NCCCCO)CCC(O)(Cc2ccccc2)C1.c12cncc(c1)OC2 13747,c1(N2C(C3(NC(c4cc(C)n(C)n4)=O)CC3)CCC2)ncnc2c1SCCC2 13748,C1(NC(=O)NCC2CN(S(CC)(=O)=O)C2)CCCN(CCOC(C)C)C1 13749,c1(C(C)C(=O)NCC(C)N(C)C(c2cc(-c3ccco3)no2)=O)cccc(Cl)c1 13750,N1(C(CC(CC)C)=O)CCN(C(C2CCC(CO)CC2)=O)C2CC12 13751,C1(NC(C(C)OC2CCOC2)=O)CCCC(NC(c2c(Cl)cnn2C)=O)C1 13752,C1(C2CCCN(C(=O)CN3CCCCCC3=O)C2)(NC(C(C)CC#N)=O)CC1 13753,C1(C(N(CC(CCC)O)C)=O)CCCN1NC(=O)c1c[nH]c2cnccc12 13754,C1(CCOC)CCN(N2CC3C=CCOC3C2)C1 13755,Cc1cc(C(N2CCC(O)C(NC(c3ccc(C)o3)=O)C2)=O)c(S(N)(=O)=O)s1 13756,N1(C(=O)NC(c2c(C)nns2)C)CC(C#N)(c2ccccn2)C1 13757,C1(NC(CN(CCC)C)=O)(CNC(C2(O)COC2)=O)CCCCC1C 13758,c1(N(CC(=C)C)C)nc2ccccc2nc1NCC1CCCN(C(C)CC)C1 13759,c1(NC(C=Cc2c(Nc3cc(OC)cc(F)c3)cccc2)=O)ncc2cn[nH]c2n1 13760,c1(N2CCCC(=C)C2)nc(=NCCC2CCCN2C)[nH]c2c1CC(C)CC2 13761,C=C=CCC(=O)NC(C(=O)NCc1cnn(CC)c1)C1(C)CC1 13762,c1(OC)cc(NCc2ncccc2Cl)ncn1 13763,C1(C(N2CCC(NC(=O)NC3CC4CC4C3)C2)=O)CCCNC1=O 13764,Cc1c(Cl)ccnc1C(=O)NC1CCC(F)(CNC(=O)C=C2CCC2)C1 13765,c1(C(N2CCC(C)N(C(=O)C=CC3CCOC3)CC2)=O)c(F)ccc2occc12 13766,N12C(=O)NC(C1=O)Cc1ccc(o1)C2.C1(OC)CCCC(C)C1 13767,N1(C(c2onc(COC)n2)C)CC(NC(c2cccc(Cl)c2C)=O)C(C)(C)C1 13768,C1(CN(C(C(Cc2ccc(OC)c(Br)c2)CN)=O)C)CCc2nccn2C1 13769,N1(C(c2ccc(OCC#C)cc2)=O)CC2CC1CCN2C(=O)CC(CC)C1CC1 13770,C(N=c1nc2sccc2c(NCC2C=CCC2)[nH]1)C1(OCC)CCCSC1 13771,Cc1noc2nc(C(N3CC(NC(=O)Cc4nnc(O)s4)CCC3C)=O)ccc12 13772,C=Cc1cc(C(N2CCC(NC(=O)CCSCCCC)C2CC)=O)cc(F)c1 13773,c1(CC2CCN(CC(N)=O)C2)ccc(C2CCNCC2)cc1 13774,c1(C(=O)NCC(CN(C(C2CCCCC2O)=O)CC)(C)C)cccc(C(F)F)c1 13775,C#CCC(CC(=O)Nn1cnn(C)c1=O)NC(=O)C(C)C(O)CCCC 13776,c1(C(=O)NC2CN(C(c3c(C)c(Cl)ccn3)=O)CC2O)cc(F)c(F)c(Cl)c1 13777,C1(CCNC(C=C(C)C(F)F)=O)(NC(=O)OC(C)(C)C)CC1(C)C 13778,C1(NC(CCC=CC(C)C)=O)CCCC(N(C)C(c2csc(C(N)=O)n2)=O)C1 13779,c1(C(=O)NCC(=O)NCC(CNC(=O)Cc2nnc(O)s2)OC)ccccc1C 13780,c1(CC(=O)CN2CCC3CC3C2)ccc(I)cc1.c1(C=O)ccccc1 13781,Cn1c(C(=O)NC2(CNC(c3ccc(N)c(CO)c3)=O)CC2)cc2sccc12 13782,C1(CNC(C(C)=C2CCCC2)=O)CN(C(=O)CCC2(C)N=N2)CCC1(F)F 13783,C1(NC(C2(C)CC(=C)C2)=O)CCCC(NC(c2cccc(C(=O)NC)n2)=O)CC1 13784,CC1(CC(=O)NCC2CCCN2N=O)CCN(C(=O)CC2CN(CCO)C2)C1 13785,C1(C)(NC(CCSCC)=O)CCN(C(C2CCCC2(C)C)=O)CC1 13786,CC1CN(C(c2cnns2)=O)CCC1C(=O)N(C)CCOCc1ccccc1 13787,c1(C(COCC)(C)N(C(C2CCCCC2)C(=O)OC)C)ccc(Br)cc1 13788,N1(C(CCOC)=O)CCC(C(C)NC(=O)C(c2cnn(C(C)C)c2)=O)C1 13789,C1(C(=O)OC(=O)CC)CN(C(C2CCCN2C(=O)C(C)C)=O)CCC1CC 13790,Cc1ccc(F)c(O)c1C(=O)NC1CC(NC(C2CCOC2C2CC2)=O)C1 13791,C(CCSC)(C(=O)NCC1(C(=O)OC)CN(C(c2scc(C)c2C)=O)C1)OC 13792,CCC(C)C(O)C(C)C(=O)N1CC(C(N2CC(N(C)C)C2)=O)C2(CC2)C1 13793,CC1CCC(F)(C(=O)NCC(C)(C)OCC(=O)NCCCCCCC2CC2)CC1 13794,c1(-c2nc(C(CCCC)O)n(CCN3CCCCC3=O)n2)cc(F)c(N)c(F)c1 13795,C(=O)(C(CO)C(C)C)N(C(CC(C)C)CNC(=O)C(=O)N(C)C)C1CC1 13796,C(=O)(CCCCc1cnn[nH]1)NCCCC1N(C(C(C)n2ccnn2)=O)CCC1 13797,C(C(CN=c1[nH]c(N2CCC(C)(C)CCCC2)nc2c1CCCCC2)OC)OC 13798,CC1C2CCN1CC(NC(c1cnn(CCC(=O)O)c1)=O)C2 13799,N1(C(c2cnn(C)n2)=O)CCC2C(NC(C34CCCC3(C(N)=O)C4)=O)CC12 13800,N1(C(Cc2ccn(C)n2)=O)CC2CC(C(=O)Nc3ccccc3C(F)(F)F)C1C2 13801,N(C1CCCn2ncnc21)C(C(C)NC(C1CN(C2COC2)C1)=O)=O 13802,N1(C(N=c2cc(CC(C)C)o[nH]2)=O)CCCC2CC(C)CCC12 13803,C(CC1=CCN(C(c2nc3cnccc3s2)=O)CC1)NC(CCN(C)CC)=O 13804,Cc1nc(NCc2cc(Cl)ccc2OC(F)F)cc(=NCc2ccnn2C)[nH]1 13805,C1(CNC(=O)NC2CCCC2CF)CCCN1c1ncccn1.OC 13806,c1(N(C(C2(C(C3(F)CC3)=O)CC2)=O)CCO)nc2ccc([N+](=O)[O-])cc2[nH]1 13807,N1(C(c2occ(C)c2)=O)CCCC(C2(NC(=O)C(O)Cc3[nH]cnc3C)CC2)C1 13808,n1(CC)ncc(C(=O)NC2CN(C(C3CC3(F)F)=O)CC2F)c1C 13809,C1(CCNC(C2(C(=O)OCC)CC2)=O)CCN(C(=O)Cn2cccn2)C(C)C1 13810,CC(O)C(C)(C)C(=O)N1C2CCC1C(CNC(=O)C(C)(C)Oc1ccccc1)C2 13811,c1(C(C)NCC(C)SC)[nH]nnc1C 13812,C1(C)(OC(CC)C(c2cccc(Cl)c2)C)CCC1(C)NC(=O)Oc1ccccc1 13813,c1(C(N(C2CC(C(N3CC4CCC3CC4)=O)C2)C)=O)cc(I)c(O)c(I)c1 13814,N1(C(C2C(C(=O)OC)CC2)=O)CCC(C)(NC(c2cccc(NC(N)=O)c2)=O)C1 13815,N1(C(c2c(SC)cnn2C)=O)CCC(CNC(c2ccc(=O)n(C)c2)=O)C1(C)C 13816,CCC(O)CC(=O)N(CC(=O)NC(c1cnc(C)s1)C)C1CCC1 13817,C(=O)(CC(=O)NCCC1(C(N2CCC(CCO)C2)=O)CC1)OCC 13818,Cc1cccc2cc(C(N3CC(NC(=O)CCF)C3)=O)oc12 13819,C(C(O)CC(F)(F)F)NC(C(C(C)C)NC(c1c(C)cc(C)o1)=O)=O 13820,Cc1[nH]c2ccc(Cl)cc2c1C(=O)NC1CC1NC(=O)C(C(C)(C)C)N(C)C 13821,C1(C(N2C(C(C)NC(c3c(C)cc(C)nc3)=O)CCC2)=O)CC(C(C)(C)C)=NO1 13822,N1(CCC)CCCCC1C(=O)NCCC(C(C)C)NC(=O)Cc1cc(C)[nH]n1 13823,C1(C)(C(=O)NCC(CNC(c2c(C)cc(CC)o2)=O)(C)C)CCC(C)=C(C)C1 13824,c1(C(=O)NC(CNC(c2cc(SCC)ncc2)=O)CC)ncnc2ccsc12 13825,c1(N(C)C2CC2)cc(-c2ccc(C(O)C(=O)O)cc2)cnc1O 13826,c1(C(=O)NCC(CO)NC(c2ccn(C)c2)=O)cccc(S(C)(=O)=O)c1 13827,C1(CNC(C(C(C)C)SCC)=O)(NC(=O)C(C)O)CCC(F)(F)CC1 13828,CC1CCN(C(C2CC(O)C2)=O)CCN1C(C12CC(C(F)(F)F)(CO1)C2)=O 13829,CC12CC(C(N3CCC(C)(CNC(c4cc(N)c(Cl)cn4)=O)C3)=O)(CCO1)C2 13830,N1(C(C(C)NS(CC)(=O)=O)=O)CCC2(CCCC2NC(c2cnoc2)=O)CC1 13831,c1(N2C(C3CCN(C(c4c(CC)c[nH]c4)=O)C3)CCC2)cc(Cl)nc(C(C)C)n1 13832,N1(C(COCC(=C)C)=O)CCC(CNC(C2CCS(=O)(=O)C2)=O)C12CC2 13833,N1(C(COC(C)=O)=O)CCC(C2(CNC(C3CC3F)=O)CCOCC2)CC1 13834,c1(CC)nc(C)c(CC(=O)NC2CC3(C2)CC(NC(C2CC2F)=O)C3)c(C)n1 13835,N1(C(C=C(COC)C)=O)CC(NC(=O)C(F)CC2CCCC2)C(C)(C)C1 13836,N1(C(c2cc(C)sn2)=O)CCC(O)(CCNC(C2(CO)CCC2)=O)C1 13837,N(C(=NCc1cccc(NC(c2ncc[nH]c2=O)=O)c1)NC1CC1C)C(C)C 13838,C1(C(N2CC3C(CNC(c4c(C)cccc4C)=O)C3C2)=O)CCC2CCCCN12 13839,c1(CC(=O)NCCN(C(=O)CC2CCNC2=O)C)cc(Cl)sc1Cl 13840,N1(C(CC2CC(CC)C2)=O)CCCC(CCNC(C2CC(OC)C2)=O)CC1 13841,C(=O)(C(C)CS(C)(=O)=O)N(CCNC(C(C1CCC(C)CC1)CC)=O)CC 13842,C1(NC(N2CC3C(CC#N)CC(C3)C2)=O)CCCC12CCOCC2 13843,C#Cc1cc(NC(C2CC(=O)C2C(C)(C)N)=O)ccc1C 13844,N1(C(C)=O)CCC(C)(C(=O)N(C)CC2CCCCN2C(c2cncn2C)=O)C1 13845,C1(NC(c2cc(CCOCC)on2)=O)CC(F)CN(C(=O)COCCOC)C1 13846,CCCCC(C(=O)N(CCCNC(=O)C(C)(C)c1cncnc1)CC)C(C)C 13847,N1(CC(C)N(C(=O)C=C2CCC2)C2CC2)CCCC(C)C1 13848,N1(CC(N2C(C(C)(C)CNC(c3cnsc3)=O)CCC2)=O)CCP(C)(=O)CC1 13849,c1(C(=O)NC2C(CC)CN(C(=O)CCc3cn[nH]c3)CC2)ncsc1S(N)(=O)=O 13850,N1(CCS(CC)(=O)=O)CCC(c2ncc(C(=O)O)s2)C1 13851,C1(C2(O)CCN(C)CC2)(C(=O)NC(CCCNC(CCC=C(C)C)=O)(C)C)CC1 13852,C(C)(C)(C(O)C(F)F)NC(CC1(NC(Cc2c(C)nn(C)c2)=O)CC1)=O 13853,Cc1nc2[nH]c(C(=O)NCCCCN(C)C(C3(C)CC4CC4C3)=O)cc2s1 13854,c1(-c2c(C(=O)Nc3ncc(C)cc3Br)ccnc2)noc2c1COCC2 13855,C12(CNC(C3C(CC)CCC3)=O)CCC(CNC(c3cc[nH]n3)=O)(CC1)CO2 13856,Cc1cc(C(N2CCN(C(=O)Cc3cnn(C)c3)C(CC(F)F)C2)=O)cc(O)n1 13857,N12CCC(F)(C1)C(=O)N(C)CCC2=O.C1(C(N2CCCC2)=O)CC2CCC1O2 13858,c1(CC)noc(CN(CCNC(=O)CCc2nc(C)no2)C2CC2)n1 13859,c1(-c2nc(C3C(C)(C)C3)nn2CCn2ccnc2)cncc2c(Cl)cccc12 13860,c1(C(N2CCCC(CNC(C=C(C)C(F)F)=O)C2)=O)cc2cc(C)c(C)cc2o1 13861,N#CC12CCC(C(=O)Nc3nc(=NCC4CCCO4)[nH]cc3C#N)(CC1)CC2 13862,c1(C(C(=O)N(CC(C)NC(C(Cn2ccc(C)n2)C)=O)C)(C)C)cccc(O)c1 13863,C1(C(=O)NCCC(C)O)CN(C(c2cccc(O)c2F)=O)C(C)(C)C1 13864,N1(C(c2nncc(C)c2)=O)CCC(C)C(NC(c2ccoc2)=O)C1 13865,CC1C(C(=O)N(C)Cc2ccnn2C)CCN1C(C1CCCC1)=O 13866,N1(C(CN(c2ncccn2)C(C2C(OC)CCC2)=O)=O)CCCC2C(O)CC12 13867,Cc1nn(C)c(C)c1C(=O)NCC(CC(C)C)NC(c1cccc(Cl)c1F)=O 13868,c1(CC(=O)NC2CCC(C)(CNC(C3(COC)CC3)=O)C2)c(Cl)ccc(O)c1Cl 13869,N1(C(c2n(C(CC)C)ncc2)=O)CC(NC(c2cnc(O)c(F)c2)=O)C2(CC2)C1 13870,N1(C(C2N(C=O)CCC2)=O)CCC(C=CC(=O)NC2(C(N)=O)CC2)CC1 13871,c1(OC)cc(C(=O)N(C(CNC(=O)C(C)=C(C)C)C2CC2)C)[nH]n1 13872,c1(C(=O)NC23CC(C(=O)NC4CC(=C)C4)(C2)C3)cc2cn[nH]c2cn1 13873,C(=O)(CC1=NN(C)C(=O)C1)NCC(C(C)C)NC(=O)C(C)P(C)(C)=O 13874,C(=O)(CC(F)(F)C(C)C)N1CCCC(N(C(C(CCCOC)C)=O)C)C1 13875,N1(C(C(C2CCOC2)NC(C(Cc2cnc[nH]2)OC)=O)=O)CC(C2CCCCC2)C1 13876,Cc1noc2nc(C3CC3)cc(C(=O)N(C)CCN3CCCCC3CC(O)CO)c12 13877,C(=O)(C(F)CCC(C)C)NC1CCC(CNC(c2c(C)oc(Cl)n2)=O)C1 13878,c1(C(N(C(C)C)CCN(C(=O)CCCCO)C)=O)ccc(C(F)F)c(F)c1 13879,c1(C(=O)NCCN(C(C(C(C)(C)C)SC)=O)C2CC2)ccc2c(c1)OCCC2 13880,N1(C(C(CCCC)(F)F)=O)CC2CN(C(=O)C(c3ccccc3C)C)CC(C1)O2 13881,C1(NC(C(C#C)(C)C)=O)CN(C(C2CC3(CC3)CO2)=O)CC1C=C 13882,C1(C(N2CCN(C(CNC(CCNC(C)=O)=O)=O)CC2)=O)CC2(CCCC2)CO1 13883,c1(C(C)(C)C)ccc(S(=O)(=O)N2CC3CC2CC3N2CCC(Cl)C2)cc1 13884,C1(C(=O)NC2C(CNC(CC(C)(C)OC)=O)CCCC2)CCC2(CC1)CC2(F)F 13885,C(=O)(N=c1cc[nH]cc1-c1noc(C2CCCC(C(N)=O)C2)n1)N.Cn1ccnc1 13886,C(CC1=CCCCC1)NC(c1c(CNC(C2(Cl)C(C(C)=O)C2)=O)ccs1)=O 13887,c1(C(N2CCN(C(C3CCSCC3)=O)C3CC23)=O)cc(Cl)c(F)cc1Cl 13888,C1(NC(c2c(C)nn(C(C)C)c2)=O)CCN(C(C2(C)CCC2)=O)CC1C 13889,C1(C)(C(N2CC3(C(NC(C(=O)N(C)C)=O)CC3)C2)=O)Oc2ccccc2NC1=O 13890,CC1CCc2[nH]c3ccc(C(N4CCN(C(=O)CCN(C)C)CC4)=O)cc3c2C1 13891,Cc1ccc(CC(=O)NCC2(C(=O)NC(CCO)C3CCCC3)CCC2)c(O)c1 13892,Cc1cc2ncn(CC(=O)NC(C)(C)CN(C)C(C3CC3(F)Cl)=O)c2cc1C 13893,c1(C(=O)NC2C(NC(CCc3cc(C)on3)=O)CC2)cn(C)nc1C(F)(F)F 13894,C1(C)(NC(c2c(CC)nccn2)=O)CCN(C(c2nccc(N)c2Cl)=O)CC1 13895,C1(C)(C(N(CC(CNC(C2C(OC)CCC2)=O)C)C)=O)CCC(=O)NC1 13896,N1(C(c2c(=N)[nH]cnc2)=O)CC2CCN(C(=O)CSCC(N)=O)CC12 13897,N1(C(c2ccc(C(C)=O)o2)=O)CC=CC(C(=O)N(CC(C)C(C)C)C)C1 13898,N1(CC)CCC(C)C(CSC)C1.N12CCCC1(CC)C(=O)NC1(CC1)CC2=O 13899,C(=O)(CC1=NN(C)C(=O)C1)NCC(C(=O)N1CC(O)(COC)C1)(C)CC 13900,c1(OC)cc(O)c(CN2CC3(CC(CC(=O)NC4CSC4)C3)C2)cc1Cl 13901,c1(CC(=O)OC)ccc(S(=O)(=O)N2CCC(C(=O)O)(C(F)F)CC2)cc1 13902,c1(COC)cnc(OC)c(C(=O)NCC#CCNC(c2coc(Cl)n2)=O)c1 13903,C1(c2n(CCC)nnn2)(NCC2(CC)CCCO2)CC(C)SC(C)C1 13904,C1(CNC(C2CC(SC)C2)=O)C=CCN1C(c1ncn(C)n1)=O 13905,N1(C(C23N(C(c4c(OC)cnnc4)=O)CC(CO)(C2)C3)=O)CCCC12CCOC2 13906,c1(-n2cc(CN3C(CCCO)CCC3)nn2)cc(Br)ncc1Br 13907,N(C(=NCC(C)OC)NCC1CCCCC1)Cc1ccc(CC)cc1 13908,c1(C(N2CC3C(NC(=O)CCOC4COC4)C3C2)=O)cc(Cl)ccc1Br 13909,CC1(C)CC(CC(=O)NCC(C)(CO)NC(c2cccnn2)=O)C1 13910,c1(C(=O)OC)cc(F)cc2c1CCN(C(C1CCC(C(=O)N(C)C)O1)=O)C2 13911,C1(C(N(CCCC)CCCC)=O)CCN(C(=O)c2ccc(CC)o2)O1 13912,Cc1cnc(C=CC(N2CCC(C3CCCCN3C(=O)C=CCF)CC2)=O)[nH]1 13913,N1(C(C=CC(=O)NC2CC2)=O)CCCCCC(NC(C2(C3CCC3)CC2)=O)C1 13914,C#CCCCC(C)C(=O)N(CCN(C(=O)CCc1cocn1)CC)CC 13915,C(c1ccccn1)=C(C(=O)N(CCOC)CCNC(C1CCOC1C)=O)C 13916,Cc1cc(C(=O)NCCC2C(C)CCCN2C(=O)C(F)=CC2CC2)cc(F)c1C 13917,O=C1CC2C(C(=O)NCc3csc(CNC(=O)Cn4nccn4)n3)C2C1 13918,C(=O)(C(C)C(C)(C)C)NC(CN(C(c1ccc(OCCC)s1)=O)C)(CO)CO 13919,N1(C(c2snnc2C)C(=O)NCC2(C(=O)OCC)CC2)CC2(CC2)CC1C 13920,CC1CC(C)(C(=O)NC2CCC2NC(c2cc(F)n(C)n2)=O)CCO1 13921,n1(CC(=O)NCC2N(C(c3cc(C(=O)OC)sc3)=O)CC2)nc(C)cc1C(F)F 13922,Cc1cc(=NCC2CN(C(c3cnn4c3CCC4)=O)CCCO2)c(C#N)c[nH]1 13923,c1(OCC)cncc(C(=O)NCC(COC)NC(c2cn(C)c(C)n2)=O)c1 13924,CCC(O)C(C)C(=O)N1CCC(=CCNC(=O)C=CC(=O)N(C)C)CC1 13925,N1(C(CCC#C)=O)CC(NC(c2cccnc2C)=O)CC12CCCCC2 13926,C(CC(CC)C(=O)NC1CCCCC1C(=O)N(C(C)CC)CCO)=CC 13927,c1(CNCc2ncc(OCCOC)c(C)c2)cc([N+](=O)[O-])nn1C 13928,C1(NC(C(c2cn(C)nc2)(F)F)=O)CCN(C(=O)CCOCC(F)(F)F)C1(C)C 13929,c1(CC)nc(C)c(C(=O)N(CC(C)(C)CNC(=O)CCn2nc(C)cc2C)C)o1 13930,CN1CCC(C(N2CCC2C(N2CCCC(CCO)C2)=O)=O)CC1=O 13931,CCC(C)C(O)C(C)C(=O)N(CCC(=O)NCC1CC1)CCCO 13932,c1(C(=O)NCC2CCCCCN2C(=O)COC2CCCC2)cc2c(nn1)CCC2 13933,N1(C(C2CCC(N=[N+]=[N-])C2)=O)CCC2(CC1)CN(C(c1ccncc1)=O)CCO2 13934,Nc1nccn2ncc(C(=O)NC3CCC(CNC(=O)Cc4ncc(Cl)s4)C3)c12 13935,C1(C(=O)OCCOCC(C)(F)F)CCCCN1O 13936,CC1(C)CC(C(=O)NCC2CCCCN2C(c2ccon2)=O)CC(C)(C)S1(=O)=O 13937,c1(C(=O)NC2CCC2NC(=O)C(O)c2cnc[nH]2)ccc2c(c1)CCCS2(=O)=O 13938,C1(CNC(c2csc(C)c2C)=O)CN(C(=O)CCC#N)CCC1C 13939,C1(C(N(CCN(C(C)C)C(c2ccc(CC#N)cc2)=O)C)=O)C2CC2C2CC12 13940,C1(CNC(c2cn(CC=C)nc2)=O)COC(C)(C)CN1C(=O)C(C)NC(C)(C)C 13941,c1(-c2cc(Br)no2)nc(-c2ccsc2)nn1C1CCC1 13942,C(=O)(C1=C(C(C)F)N(CC(=O)O)C(=O)NC1c1cc(Cl)c(F)cc1F)OCC 13943,N1(C(Cc2c(C)ccs2)=O)CCC(C)(NC(=O)Cc2nnn(C(C)(C)C)n2)C1 13944,c1(C(N2CCCC(NC(c3ccc(CF)cc3)=O)CC2)=O)cn2ccnc2cn1 13945,c1(-c2cn(C3CCC(C(N4CCC(C)(OC)CC4)=O)C3)nn2)ccc2cc[nH]c2c1 13946,C#Cc1ccc(CCCC(=O)NC2CCN(C(c3c[nH]c(=N)o3)=O)CC2C)cc1 13947,CC#CCCCC(=O)NC(C(=O)NCC1CCCC1CF)c1cccs1 13948,c1(C(N(CC(C)C)CCC)=O)occc1CNC(c1nccn1C(C)C)=O 13949,C(=O)(C(COC(C)C)NC(c1cn(C(C)(C)C)nn1)=O)N(C(C)SC)CC 13950,C(=O)(C1CCCc2nn[nH]c21)NCC(C)CNC(c1ncn2c1CCCC2)=O 13951,c1(C(=O)NCC2CCC(NC(C(c3cnn(C)c3)OC)=O)C2)ccc(O)nc1Cl 13952,Cn1c(C(=O)NCC(C2CCOC2)NC(c2cnc3n2CCS3)=O)cccc1=O 13953,CCCCC(C)CCC(=O)N1CCC(F)C(NC(c2nc(Br)c[nH]2)=O)C1 13954,c1(C(=O)NC(c2cnn(C)c2)C(=O)NC(c2ccccc2)C)n[nH]c2c1CCC2 13955,C1(CNC(C=Cc2n(CC)ncc2)=O)CCN(C(=O)C(C)(C)SC)CC1C 13956,Cc1cc(C(=O)N)cc(F)c1C.c1(C2(C(=O)CC3(O)CNC3)CC2)cccnc1Cl 13957,C(=O)(C(F)(CNC(=O)CC1CC(CC)=NO1)C(C)C)N1C(CC#C)CCCC1 13958,CC(C)C(CNC(C1C2CCCCCC12)=O)C(=O)NC(C1(O)CCC1)C 13959,c1(C(CC)CNC(=O)NCCc2csc(N(C)C)n2)ccc(OC)cc1 13960,c1(OCC(N2CCC(N3CCCC3=O)CC2)=O)ccc(Br)cc1OCC(F)(F)F 13961,C1(C(=O)NC(c2ccc(C)cc2)CNC(C2CC(=C)C2)=O)CCC2(CC1)CC2 13962,Cc1cnc(C)c(C(N2CC(NC(c3c[nH]nc3C(C)C)=O)CCC2C)=O)c1 13963,N1(C(C(COC)OC)=O)CCCC(NC(=O)CC2CSCCS2)CCC1 13964,C12CC(C1)CNC2=O.C1(C(=O)OC(C)(C)C)(CNCC(C)OC)CCC1 13965,CCCC(O)C(=O)NC(C(=O)N1CCC(N(C)CC)C1)C(C)C 13966,c1(NC(c2ccc(Br)s2)C)[nH]c(=NCC(C)Oc2ccccc2)nc2scnc12 13967,CCCCCCC(C)C(=O)NC1CC(C(=O)NC(C)Cc2nn[nH]n2)=CC1O 13968,Cc1c[nH]nc1C(=O)NC1CN(C(C2(C(=O)NC3CCOCC3)CC2)=O)C1 13969,N1(C(c2scc(C)c2)=O)CC2CCCC2(NC(=O)Cn2nc(C)n(C)c2=O)C1 13970,CC1(C)C(c2ccc(Br)cc2)CCN1C(C1CCN(C(=O)CN)CC1)=O 13971,c1(C(=O)NC2(C(=O)NCC(C)Cn3cccn3)CC2C)cc([N+](=O)[O-])n[nH]1 13972,C1(C(=O)NCC2CCN(CC)C2)CSCCN1C(=O)CSC(C)(C)C 13973,N1(C(C(C(CC)O)C)=O)CCOC2(CCN(C(=O)CC3CCCCCC3)C2)C1 13974,c1(C(=O)NCCCN(C(C(C)n2cccn2)=O)C)ccc(S(=O)(=O)CF)nc1 13975,c1(C(=O)NC2C(O)CCN(C(CCCCC#C)=O)C2)cc(Cl)cc(Cl)c1O 13976,n1(CC)nc(C2CC2)cc1S(=O)(=O)NC1C(C)C1C(=O)NC 13977,c1(C(=O)NCC2(O)CCCN(Cc3nc(CC)sc3)C2)c(F)cc(Cl)cc1F 13978,C1(C(N(C)CC2CCN(C)C2)=O)CC2(CCC2)CN1C(c1ccc(C#N)s1)=O 13979,CCC(C)CCC(=O)NCc1nc(C)c(C(=O)NCC2(CC)CCCC2)o1 13980,C(=O)(C1=NOC2(CCN(Cc3csc(Br)c3)C2)C1)Nc1cc(C)c(C#N)c(C)c1 13981,C1(C(=O)NCC(C(C)C)NC(c2csc(C(F)F)n2)=O)CC(=O)N(C)C1 13982,c1(C(=O)N(C)C)ccc2sccc2c1.N12CCOC(C1)C2C(C)C 13983,N1(C(c2ccc(C(C)=O)cc2)=O)CCC(F)CC1C(N1CCN(C)CC1CO)=O 13984,C(CC1=CCCCC1)NC(C1C=CCN(C(c2ccsc2Cl)=O)C1)=O 13985,C(=O)(C(C)(C)CF)N(C1CCN(C(C2CCN(C)C2c2ccccc2)=O)CC1)C 13986,c1(C(=O)NC2CC(CCNC(Cc3n(C)nnc3)=O)C2)ccc(N)cc1O 13987,c1(C(N2CC(CNC(CC3(OC)CC3)=O)C(O)C2)=O)cc(C)c(Cl)cc1F 13988,Cn1c(CN(C=O)Cc2ccc(N3CC=CC3)cc2)nnc1-c1ccccc1 13989,c1(NC2CN(C(C)=O)C2)[nH]c(=NC(C)c2cnc[nH]2)nc2sccc12 13990,N1(C(=O)Cn2cnnc2)CC2CC(N=c3ccnc(CO)[nH]3)CC1C2 13991,C(=O)(CC(C1CCC1)NC(=O)NC1CCN(C2CCOCC2)C1)N(C)C 13992,N1(C(CC(CC)c2ccc(C)cc2)=O)CCC2(CC1)CN(C(=O)CCC(C)=O)C2 13993,C(c1ccc(Cl)cc1Cl)=CC(=O)N(C1CCCN(C(C)=O)C1)C 13994,C(=O)(C(CCSC)NC(=O)C(CCC)N(C)C)NCCC1(C#C)CCC1 13995,C1(C2(NC(C34CC3CN(C(=O)C(C3CC3)SC)C4)=O)CC2)(OC)CCC1 13996,C1(C(N2CC(CCNC(C(CC)NC(C)=O)=O)C2)=O)CC2(CCC2O)C1 13997,C12(C(N(C)CC3CCN(C(C(C)OCC)=O)CC3)=O)CCC(OC)(CC1)CC2 13998,S(=O)(=O)(CCC(=O)NCC1COCCN1C(c1ncnn1C(C)C)=O)NC 13999,N1(C(CCSCC)=O)CCC(NC(c2ccc3cc(C)cn3c2)=O)C2(CCC2)C1 14000,N1(C(CCCc2c(C)ccs2)=O)C2CCC1C(CNC(=O)C=Cc1ncc[nH]1)C2 14001,c1(C(=O)NCC2CCC(NC(c3ccc(Cl)o3)=O)C2)cccc2cc[nH]c12 14002,Cc1c(Cl)cc(C(=O)NCC(C)NC(=O)CN2CCCC(C)C2)cc1Br 14003,c1(C(N2CCN(C(c3nc(CC)oc3)=O)CC2CC)=O)c(C)cc(Br)cc1C 14004,c1(CC)cc(C(=O)NC2CC(C(=O)NC3C=CCC3)C2)ccn1 14005,c1(C(=O)NCC23CC(NC(CN(CCC)C)=O)(C2)C3)ccc2cccnc2c1 14006,C1(C(=O)NCC(CC)N(C(C=C(CCC)C)=O)C)(CC)CCNC1=O 14007,N1(C(c2c[nH]c(=NC)o2)=O)CCCC12CCCN(C(=O)COCP(C)(C)=O)C2 14008,c1(C(=O)NCC(CNC(C2C(OC)CC2)=O)(C)C)cccc(SC)c1[N+](=O)[O-] 14009,C(CCCCNC(=O)CC(F)F)NC(=O)C=CCn1cncn1 14010,n1(CCC)cc(Cl)c(C(=O)NC(C)CN(C(c2cccc(F)c2)=O)CC)n1 14011,c1(OC)cc(C)c(C(=O)NCC2CCC3(CN(C(=O)CC(C)SC)C3)O2)c(C)c1 14012,C1(NC(C(CC=C)NC(=O)C(C)OCOC)=O)CC(C)(C)OC1(C)C 14013,C1(N(C(c2cc(CC)on2)=O)C)CCCC(NC(=O)CCCN2CCCC2)C1 14014,CCC(CC(=O)NCC(C)CN(C(=O)C(c1cccn1C)=O)C)C(C)(C)C 14015,N1(C(CC(C(C)OC)NC(c2c(CC)oc(C)c2)=O)=O)CC=C(C(C)(C)C)CC1 14016,C(c1ccc(OCC)c(Cl)c1)=CC(N1CC(NC(COCC)=O)C(C)C1)=O 14017,C12(NC(C(CC)N(C)C)=O)CC3CC(C1)CC(NC(C1C4CC4C4CC14)=O)(C3)C2 14018,C1(C(N(CC(=C)C)CC(=C)C)=O)CCCC(NC(c2ccc(C3CC3)nc2)=O)C1 14019,N1(C(c2n(C)ncc2Cl)=O)CC(O)CCC1C(=O)NCC1CC2(CC2)C1 14020,c1(OC)ccccc1C(CNC1CCN(c2ccc(C)cn2)C1)OC 14021,N1(C(C(CC=CC)C)=O)C(C(N2CCCC2C(O)CC)=O)CCC12CC2 14022,C1(CNC(C2CC(=C)C2)=O)CC(F)CN(C(=O)C(c2cccn2C)=O)C1 14023,Cc1cccc(C(=O)NCCC23CCC2CN(C(c2nocc2Br)=O)C3)c1O 14024,c1(C(=O)Nc2cn(C)nc2)coc2cc(N)c(-c3cnc4n[nH]cc4c3)cc12 14025,CC1=C(C(=O)OCC(F)(F)F)C(c2cc(C(C)C)cc(C)c2)NC(=O)N1C 14026,c1(C(=O)NC2CC(NC(=O)COCCOCCO)C2)ccc(F)c(O)c1F 14027,C(=O)(CCN=c1cc(NC2CC(C3CC3)C2)nc[nH]1)N(C)CCO 14028,c1(SCC(=O)NCC2(F)CC(NC(C3C4CC4C4CC34)=O)C2)cccc[n+]1[O-] 14029,N1(C(C(C=CC)O)=O)CCC2CC12C(=O)NCCCN1CCOC1=O 14030,N1(C(=O)CSc2n[nH]c(O)n2)CCN2CCNCC2C1 14031,C1(C(=O)NC2C(NC(C3(C)CCCC3)=O)CS(=O)(=O)C2)CCC(C2CC2)CC1 14032,N1(CC(=O)NC(CNC(CC=C)=O)C(C)C)C(=O)NC(C)(COC)C1=O 14033,c1(CC(=O)NCC(CNC(Cc2cnc(C)[nH]2)=O)F)ccc(Br)cc1 14034,c1(C(N2C(C(C)NC(=O)C(O)C3CCC3)CCC2)=O)cc2c[nH]cnc-2n1 14035,c1(OC)ccc(S(=O)(=O)N2CCCC(C)(C(=O)Nc3c[nH]nc3C#N)C2)cc1Br 14036,C(=O)(CCCC(F)(F)F)NCCCN1CCC(NC(C(NOC)=O)=O)C1 14037,C1(NC(CN(C(=O)OC)C)=O)(CNC(c2cnc[nH]2)=O)CCCCCC1 14038,c1(OC)ccc(CN2CCCC(C(C)NC(c3ccc(Cl)cc3)=O)C2)c(Cl)n1 14039,C(CN=C(NCC(=O)N(C)C)NCC1CCOC1)(c1ccc(F)cc1)N(C)C 14040,CCCC(C)(CC)C(=O)NC1CC(CCNC(=O)C(C)(CC)CC)C1 14041,C1(NC(C(CC)N(CC)CC)=O)C2CN(C(c3cccnn3)=O)CC12 14042,N1(C(C(CCCC)=O)=O)CCOC2(CCN(C(=O)C=Cc3cccs3)C2)C1 14043,CC1(NC(C2C3CCCCC23)=O)CCN(C(=O)CN2CCC(O)CC2)CC1 14044,Cc1cc(CC(=O)NCCN(C(C23CCCCC2C3)=O)CC2CC2)n(C)n1 14045,CCCCC(O)C(C)C(=O)N1CCN(C(=O)CC2CCSC2)CC1C(C)(C)C 14046,c1(C(=O)NC2C(NC(C3CN(C)C(=O)N3)=O)CCCC2)cccc(C(N)=O)c1F 14047,c1(NCC2C(C)CC=CC2)ccc2c(c1)COCC2 14048,c1(C(=O)NCC(C)NC(=O)C(=O)N(C)C)ccc(NC(=O)Cn2cnnc2O)cc1 14049,c1(CCC(=O)NCC2N(C(Cc3cn(CC)nc3)=O)CC=C2)cc(C)nn1C 14050,c1(CC(=O)NCC2C(NC(C(C)C3CCC3)=O)CCC2)ccc2nc(O)[nH]c2c1 14051,N1(C(C(COCC)NC(c2cccc(C)n2)=O)=O)CC(C)(C)C1COC 14052,Cc1cccc(C)c1C(O)C(=O)NC(C1CN(C(=O)CSC(F)(F)F)C1)C 14053,C1(CNC(=O)C(=O)NCC(=C2CCSCC2)c2ccccc2)CCCC(=O)N1 14054,c1(OC)c(F)ccc(-c2ccc(CC(=O)NC(C)C#N)cc2F)c1F 14055,c1(-c2nc(C(C)SCC)nn2-c2nc(C)nn2C)onc2cc(C)ccc12 14056,c1(NC(c2n(CCCC(=O)OCC)nnn2)(C)CCBr)ccc2c(c1)CCCS2 14057,c1(C(N(C2CC(NC(=O)CC3CCC3)C2)C)=O)ccc(OCC(F)(F)F)c(Cl)c1 14058,c1(CC(=O)NC2CC3CN(CC4(C(=O)N(C)C)CC4)C2C3)ccc(S(C)=O)cc1 14059,C1(NC(CCCCOC)=O)C2CC3C1C3C2C(=O)NCCN1CCOCC1C 14060,Cc1nc(CC(=O)NCCn2cc(C3(CCO)CC3)nn2)c(Br)s1 14061,c1(C(=O)NC(C2(O)CN(C(=O)CC3CCNC3=O)C2)C)ccccc1OCC(N)=O 14062,N#Cc1cnn(CC(N2CC3CC2CN3C(c2cnnc(O)c2)=O)=O)c1N 14063,c1(N(C)C)ncc(C(=O)NC(CC(N)=O)c2cn(CC3CCCO3)nn2)cn1 14064,C(c1cccc(O)c1)=CC(=O)NCC(C)(F)CNC(C1CCCN1C1CC1)=O 14065,N1(C(C(=O)NCC(=C)C)C(CC)CC(C)C)c2ccc(F)cc2CC1C 14066,CCCCC(C(=O)NC1CC2(C1)CN(C(c1cc(CC)[nH]n1)=O)C2)NC(N)=O 14067,C(=O)(CCCCCCC=C)NC(CC#C)C(=O)NCCCc1cccs1 14068,C1(NC(c2ccc(C#C)o2)=O)(CO)CCCN(C(=O)CCCc2ccccn2)C1 14069,c1(C(=O)NC2CCCN(C(CC(COC)C)=O)C2C)ccc2c(c1)C(=O)NC2=O 14070,c1(C(N2CC(NC(C3C(C)C3c3ccccc3)=O)C2)=O)nccnc1Cl 14071,C1(CNC(CC2ON=C(C)C2)=O)CCC(CN(C(=O)C(C)n2ccnn2)C)CC1 14072,N1(C(C(CC=C)OC)=O)CCCC(O)(CN(C)C(C2(O)CCCCCC2)=O)C1 14073,C(=O)(C(C)(C)C(N)=O)NCCCC(C)NC(=O)C(C)c1ccco1 14074,C1(CC)(NC(c2ccc(Cl)c(OC)c2)=O)CCCN(C(=O)CCc2cn[nH]c2)C1 14075,CC1CN(C(=O)CC(C)(C)O)CC2(CCN(C(c3ccc(=O)n(C)n3)=O)C2)O1 14076,c1(CC)cccc(C(=O)NC2C=CCN(C(C3(c4ccn(C)n4)CC3)=O)C2)c1 14077,c1(C(=O)NC(C2CCCN2C(=O)CN=S(C)(C)=O)(C)C)ncc2c(F)cccn12 14078,CC(C)C(C(=O)NCCCCC(C)NC(=O)Cc1cnns1)C1CCCCC1 14079,C1(CNC(=O)Cc2ccccc2CO)CN(C(c2cccc[n+]2[O-])=O)CC12CC2 14080,C12(NC(=O)CC34CCCC3C4)CCC(C(=O)NCc3cnsc3)(CC1)C2 14081,C1(NC(c2c(CC)noc2)=O)CN(C(c2cccc(N)n2)=O)CC(C)(C)C1 14082,C1(C2(O)CN(C(c3cccc(OC)c3)=O)C2)(CNC(C(COCC)C)=O)CC1 14083,C(=O)(CCCCNC(=O)Cc1cncc(C)c1)NCC#CC 14084,CCCCC(C)(F)C(=O)N1CC2(CCN(C(c3cocc3Br)=O)C2)C1 14085,c1(SCC)ccccc1-c1ccc(N2CCN(C(c3ncnn3C)=O)CC2)nc1 14086,C1(C(C)C)CN(C(c2ccc(Cl)nc2)=O)CCN1C(c1cn(CC2CC2)nn1)=O 14087,c1(C(=O)NCCC(CNC(c2ccc(CO)s2)=O)OC)cccc(C)n1 14088,N1(SCC)CCc2c(NC(c3ccc(F)cc3I)=O)cccc2C1 14089,C1(CNC(CC=C)=O)CN(C(=O)CN(CCC)C(=O)OC(C)(C)C)CCC1(F)F 14090,C12(C(=O)NC3C(NC(CCc4cn(C)nc4)=O)CC3)CCC(CC1)C(C)(C)O2 14091,c1(SC)ccc(C=CC(N2CC(CNC(c3cn(CCO)nn3)=O)C(C)C2)=O)o1 14092,CC1CCCCCCN1C(=O)C(C)N(C(=O)CCN1CCOC1=O)C1CC1 14093,Cc1c(C(F)(F)F)nc(Cl)nc1CN(C(C)Cc1ccc(Br)cc1)C 14094,N1(C(C(C=CC)O)=O)CCC(N2CCN(C(=O)C(c3ccnn3C)C)CC2)CC1 14095,CN1CCC(C(F)(F)F)(C(=O)NCC(O)CC2CCCC2O)C1 14096,c1(C(N2CCC(N)(CC(=O)OC)C2)=O)cc(Br)c(O)nc1C 14097,N1(C(c2cc(CC)c(C)s2)=O)CC(C)CCC1CNC(=O)COC(F)(F)F 14098,c1(NC(C(CC)NC(C)=O)=O)ccc(-n2ccnc2)cn1.C123CC(C1)(C2)NC3=O 14099,N1(C(c2n[nH]c(CC)c2C)=O)CCCCC(C(=O)NCC(c2cnn(C)c2)C)C1 14100,C#Cc1ccc(C(=O)NCCCNC(C2(C)CCC(=O)C2)=O)c(F)c1 14101,c1(C(C)(C)C)ccc(CNC(=O)CC2CCCC2NC(=O)CCNC(N)=O)nc1 14102,N1(C(C(C(C)O)(F)F)=O)CC2(C1)CN(C(C1(c3ccno3)CC1)=O)CCO2 14103,c1(C(C(=O)NCC(C)N(C)C(c2cnccn2)=O)(C)F)ccccc1F 14104,CS(=O)CCC(O)C(=O)NC1CC(CNC(c2cncc(F)c2Cl)=O)C1 14105,C1(C2(O)CN(C(=O)Cc3ccncc3Cl)C2)(CN(C(c2cnsc2)=O)C2CC2)CC1 14106,C(=O)(C(C)(C)C(O)C(C)C)NCC1(F)CCN(C(c2n(CC=C)ccc2)=O)C1 14107,CC1CN(C(=O)C=CC2CCCC2)CC(C)N1C(C1CCC(C2CC2)C1)=O 14108,c1(N(CCNCc2cccc(C)n2)C)ncnc(NC2C=CCN2C)c1C 14109,CC(C)C(C(C)NC(c1cc(Cl)n(C)n1)=O)NC(c1cc(C2CCC2)on1)=O 14110,Cc1nn(C)cc1C(N1CC(CNC(=O)CC2CC(C3CC3)C2)C1)=O 14111,C(=O)(C(CC(=C)C)NC(c1c[nH]nc1OC)=O)NCCCCCC=C 14112,C1(C(=O)Nc2cn(CC#C)nc2)CN(C(C2(NC(C)=O)CC2)=O)CCO1 14113,C1(O)(CCNC(=O)COc2ccccn2)CCN(C(=O)CC2CC2C2CC2)C1 14114,C=CCC(CC)C(=O)N(C1CN(C(c2ccnn2C)=O)CC1(C)C)C 14115,C1(CC(N2CCC(NC(C3(C)C(C)C3)=O)C2)=O)CCN(Cc2ccccc2)CC1 14116,C1(C(=O)OC)CC12CCC(NC(=O)Nc1ccc(F)cc1Cl)CC2 14117,CC(C)(C)C#CC(=O)NCC1CN(C(=O)C=Cc2ccsc2)CC1(F)F 14118,N1(C(C(CN(C(Cc2cc(C)sc2)=O)C)C)=O)CCC2(COC(=O)N2)C1 14119,N1(C(C(C)NC=O)=O)CC(O)(CCNC(=O)Cc2ccsc2)C1 14120,C1(NC(CCC=C)=O)CCCN(C(C2(COC)CCOC2)=O)C1 14121,C(=O)(C(C)(CC(C)C)NC(=O)OC(C)(C)C)N1C(CNC(C(C=C)(F)F)=O)CC1 14122,C1(C)(C(=O)NC(CC)(C)CNC(=O)CC2(CSC)CC2)CC(C)(C)C1 14123,N1(C(C(COCC)C)=O)CCC(CC(N)=O)(NC(=O)COCCN(C)C)CC1 14124,N1(C(c2ncc(C)s2)=O)CCC2(OCCO2)C(C(=O)O)C1 14125,Cc1nsc(CN(C(C(=O)NCc2cccs2)C2CCSC2)C)n1 14126,N1(CC(=O)Nc2c(OC)cccc2)CCCC(=O)C1C 14127,c1(OC)cc(NC(C2CC(NC(=O)CC3CC(OC)C3)C2)=O)cc(F)c1 14128,c1(C(=O)NC(CC)CNC(C2CCN2C2CCCC2)=O)ccc2ncccc2c1 14129,c1(OCC)cc(C(=O)NCCCCCN(C(c2c[nH]ccc2=O)=O)CC)ccn1 14130,c1(C(N(C)CCN(C)C(C2(C(F)(F)F)CCCC2)=O)=O)ccnc(OCCO)c1 14131,N1(C(CSCC(C)=O)=O)CCC(N(C)C(c2ccn(CCF)n2)=O)C1 14132,c1(CN(C(=O)CCOC2CN(C(c3ccco3)=O)C2)CC)cnn[nH]1 14133,N1(C(CNC(CC)=O)=O)CC2CC(N(C(=O)C(C)Cn3cccn3)CC)C1C2 14134,C1(S(=O)(=O)N2CCN(C(=O)CCCCSC)CC2)(CC=C)CC1 14135,N1(C(C(=O)Nc2cc(C)c(-n3cnnn3)cc2)=O)CC2CC(NC(N)=O)CC1C2 14136,C#Cc1ccc(NCc2ccnc(Br)c2)cc1C#N 14137,CC(C)C(O)C(=O)N1CC2CC1(CNC(=O)CC1CC3(CC3)C1)C2 14138,c1(C(C)N)cccc(S(C)(=O)=O)c1.n1(C(C)Cc2nc(C3CC3)n[nH]2)ccc(C(F)(F)F)n1 14139,C1(NC(c2c(OC)oc(C)n2)=O)CN(C(=O)CC2CCC(=O)NC2)CC1C1CC1 14140,C1(NC(c2c(O)ncc(NC(C)=O)c2)=O)CN(C(C)=O)CC2(CCC2)C1 14141,c1(C(=O)NCC2C(CNC(c3cccc(C#C)c3)=O)C2)ncc([N+](=O)[O-])cc1C 14142,c1(OC(CC)C(=O)NC(C)(C)CNC(=O)CC(C)c2ccco2)cccc(C)c1 14143,N1(CCNC(C2(C)CCCS2)=O)CCCN(C(C2(n3cccn3)CCC2)=O)CC1 14144,CC1(C)CC(NC(C2CSC2)=O)CCN(C(=O)COc2ccccc2)C1 14145,CC(O)C(C(=O)NN(C)CC1CCN(C(c2ncoc2C(C)C)=O)CC1)N(C)C 14146,C1(CC(=O)NC2CCCC(CNC(c3cccc[n+]3[O-])=O)C2)CCS(=O)(=O)CC1 14147,N1(CCCCC(C)Nc2cc(N(C)C)ncn2)C(=O)c2ccccc2C1=O 14148,N1(C(C(C)SC)=O)CCC(N(CCO)C(C2CC3C=CC2O3)=O)CC1 14149,N#CC1(C(=O)NC2CCCC(C(=O)NCc3ccncn3)C2)CC12CCC2 14150,Cc1cccnc1CCNC(=O)Nc1ccc(-n2ccnc2)nc1 14151,c1(C(N2CC(CCC=C)(C(N3CCCCCCC3)=O)C2)=O)ccc2[nH]ccc2n1 14152,Cc1ccc2c(C(N3CCN(CC(N4CCC(C)C4)=O)C(=O)C3)=O)cccc2c1 14153,C1(C(=O)NCCCc2onc(C)n2)CN(C(=O)CCCNC(=O)C2CC2)CCO1 14154,N1(C(C2N(C(C)=O)CCC2)=O)CCOCC(CNC(C2C=CCC2)=O)C1 14155,c1(CC)cc(CC(N2CCCC2C(C)NC(c2cn(C(C)(C)C)cn2)=O)=O)on1 14156,n1(CC(=O)NCC(CNC(CC)=O)F)cnc(-c2ccccc2)n1 14157,N1(C(CN(C2CC2)CC)=O)CCC(CNC(c2ccc(O)cc2F)=O)C(CO)C1 14158,Cn1cc(C#N)cc1C(=O)NC1CCN(C(c2coc3c2COC3)=O)CC1 14159,CCCC(CCCNC(C12CC(NC(c3cc(CC)cc(C)c3)=O)(C1)C2)=O)OC 14160,C1(NC(c2cc(CC)on2)=O)CC12CCN(C(=O)CNC(N)=O)CC2 14161,C(=O)(C1=CCSC1)C(C(CSC)NC(=O)C)=O.C(C(C)C(C)(C)C)NC 14162,C=CCC(F)(F)C(=O)NCC(C1(O)CCN(C(c2coc(C(N)=O)c2)=O)C1)C 14163,CC(CCNC(C1CN(C(c2cc(O)ccc2F)=O)C(C)(C)C1)=O)CC(C)(C)C 14164,CCCN(Cc1ccc(O)cc1)N1Cc2ccc(C(C)=O)cc2C1 14165,N1(C(C(C(C)O)C)=O)CC(NC(=O)CN(C)Cc2ccccc2)CC2(CC2)C1 14166,N1(C(CC(c2ccc(OC)cc2)C)=O)C2CCC(CO)C1CC2 14167,CCCC(C)(O)C(=O)N1CC(C(C)NC(c2ccc(=O)n(O)c2)=O)C1 14168,c1(C(N2CC(CCCCNC(C=COCC)=O)C2)=O)cc(C)c(C)nc1C 14169,C1(NC(COCC=C)=O)CC1C1CCN(C(C2CCc3nn[nH]c3C2)=O)CC1 14170,N1(C(CSCC=C)=O)CC2CCCN(C(=O)C(C)Oc3cccc(C)c3)C2C1 14171,c1(C(N2CCC(C)(C(=O)Nc3c(COC)cccn3)C2)=O)coc2ccccc12 14172,N1(C(CCC(=O)OC)=O)CCN(C(c2ccc(C)cc2Cl)=O)C(C(F)F)C1 14173,N1(C(C2N(C(c3ccc(C#N)cc3)=O)CCCCC2)=O)CCC2(COC(=O)N2)C1 14174,C1(O)(CC)CCN(C(c2cc(C(N)=O)co2)C(=O)NC(C)CC)C1 14175,c1(CNC(C2CCC3(CN(S(=O)(=O)CCCCl)C3)O2)=O)c(F)ccc(Br)c1F 14176,c1(NC(c2ncc(C34CCCCC3C4)o2)=O)ccc(N2CCOCC2)c(F)c1 14177,c1(C(=O)NCC(=C2CN(C(CC3CCC(OC)C3)=O)C2)F)cc(C)ncc1C 14178,N1(C(CNC(C(CC)C)=O)=O)CC2C(C(=O)NCc3ncc(Cl)cn3)C2C1 14179,c1(C(N2CC(C(F)(F)F)CC(CN)C2)=O)cc(C(F)F)nc2ccc(Cl)cc12 14180,c1(C(=O)NC2CN(C(CC3CC(N(C)C)C3)=O)C2)ccc(Cl)c(N)c1 14181,N1(C(C)=O)C=Cc2ccccc2C1CC(=O)NCCn1cc(C(C)(O)C(C)C)nn1 14182,c1(CC)ccc(C(=O)NC(C)CNC(=O)CS(=O)(=O)C2CC2)cc1[N+](=O)[O-] 14183,C1(C2CN(C(c3sccc3F)=O)C2)(NC(c2ccc(O)nc2Cl)=O)CC1 14184,CCCC(O)(CCC)CC(=O)NC(C)CN(C)C(C1CCn2nccc2C1)=O 14185,N1(C(C(C)(C)OCCC)=O)C2CCC1C(C(=O)NC1COCCN(C)C1)C2 14186,CC1CCCc2ncc(C(N3CCC(CO)(NC(=O)Cc4ccon4)C3)=O)n21 14187,C(CNC(C1(O)CC1(C)C)=O)(CC(C)C)NC(CCc1cnc(C)s1)=O 14188,C1(F)(C(=O)OC)CN(CC(c2ccco2)=O)CC1c1cccnc1 14189,c1(C(N2CC(C)(NC(C(CC(C)C)O)=O)C2)=O)coc2cccc(Br)c12 14190,c12cc(ncn1)C(=O)NCC1CCC(CC1)C2=O.C1(O)(CN)CCC(C)C1.CO 14191,C1(C(=O)NCCCNC(COCCCC)=O)CCCCC1F 14192,Cc1ccc2sc(C(N3CCC(CO)(NC(=O)C(=O)C(C)(C)C)CC3)=O)cc2c1 14193,C1(NC(C(C)(C)CO)=O)CN(C(c2n[nH]c3ccccc23)=O)C2(CCCCC2)C1 14194,N1(C(c2ccc(CSC)cc2)=O)CC2CC(C)N(C(C3CCC3CF)=O)C2C1 14195,N1(C(c2ccc(O)cc2)=O)CCC2(CCN(C(c3ccnc4ccnn34)=O)C2)C1 14196,O=C(C#CC1CC1)NCC1CCCC1NC(=O)Cc1cccc(C(F)(F)F)c1 14197,C1(C(CC)C)CCN(C(=O)C(C2(O)CCC2)NC(c2cccs2)=O)CC1 14198,C(=O)(C#CC1CC1)OC.N1(C(C=CC(=O)NC2NCC3(CC3)N2)=O)CCOCC1 14199,c1(CC)nc(C(C)C)ccc1C(=O)NCC(CC(C)C)NC(=O)COCC1CC1 14200,C(=O)(C(C(C)NC(C1CCC(C)=C(C)C1)=O)C(C)C)N1CC=C(C)C1 14201,C(C(C)(C)CNC(c1cc(C)ns1)=O)NC(CCOCC)=O 14202,C#CCC(C(=O)NC)NC(C1(CNC(=O)CCCSC)CC12CCC2)=O 14203,Cc1cc(C(N2C(CNC(C3CC34CCOCC4)=O)CC2)=O)ccc1[N+](=O)[O-] 14204,CON1CCC(C(=O)NC2(C)CC(C(=O)NC3CC(F)(F)C3(C)C)C2)CC1 14205,c1(C(=O)OC(C=CC(=O)OCC)C)cccn1Cc1ccccc1 14206,N1(C(C(CC2CC2)OC)=O)CCCN(C(=O)CN2CCCCCC2)C(C)C1 14207,c1(CC)nocc1C(=O)NCC=CCNC(C1(c2nc[nH]n2)CCC1)=O 14208,C#CCCCCCC(=O)N(CC(CC)NC(=O)Cc1cncn1C)C 14209,N1(CC(C)(C)NC(C(C2CCN(C(=O)C(F)F)CC2)C)=O)CC2CCCC2C1 14210,CC(C)CC(O)C(=O)NCC1CCCN1C(=O)C1=CCCCC1 14211,C1(C)(OC)CN(C(=O)NC(CC)(c2nnnn2C2CCC2)NC(=O)OC(C)(C)C)C1 14212,c1(C(=O)NCC(O)CCC2CC2)cccc(-c2ccccc2)n1 14213,c1(SCC(=O)NCC(C)NC(=O)C=CCN2CCCC2=O)nccn1C 14214,C1(CNC(C2C(NC(CSCCOC)=O)COC2)=O)CC2CCCC2C1 14215,N1(c2ccnc(OC)n2)CCOC2CN(C(c3ccn(C)c3)=O)CC12 14216,CC1CC=CCC1C(N1CC(NC(c2ccccc2C(C)(F)F)=O)C(F)C1)=O 14217,c1(OC)ccc(CC(=O)NC2CC(N(C(=O)CS(N)(=O)=O)C)C2)cn1 14218,c1(CC)cc(OC)ccc1N.c12ccc(cc1)N(CC)C(=O)C2N 14219,N1(C(CC2CC(OC)C2)=O)CCC2C(NC(=O)CC3CN(C)CC3O)CC12 14220,c1(OC)cscc1C(N1CCC(CCNC(C2CC2F)=O)C1)=O 14221,C1(C(=O)NCC2(C(C)NC(C3CC=CC3)=O)CC2)C=CCCC1 14222,c1(C(C)C)conc1CC(=O)NC(CNC(=O)C(C)CC1CC1)C(C)C 14223,c1(OC)cccc(-n2nc(-c3ccsc3)nc2-c2scnc2Cl)c1 14224,C=CCCCCCCCC(=O)N(CC)CC1CC(O)C1(C)C 14225,C1(N(C)C(=O)NCCCN(C)OC(C)(C)C)(Cc2nnn(C)n2)CCOCC1 14226,N1(C(CCCOCC=C)=O)CC(C(N2CCC(N3CC(O)C3)C2)=O)CCC1(C)C 14227,c1(OCC)ccc(C(=O)NCCN(C)C(c2ccccc2C2CC2)=O)cc1N 14228,N1(C(COCCOCC)=O)CCC(NC(=O)COCc2cccc(C)c2)CC1 14229,c1(C(C)NS(=O)(=O)Cc2noc(C3CC3)n2)cc2ccc(O)cc2[nH]1 14230,C=CCC(C)C(=O)NC1(C(=O)Nc2ccc(Cl)nc2)CCN(C(=O)C(C)SC)C1 14231,C(=O)(CC(C(F)(F)F)P(C)(C)=O)NCCC1CC(NC(c2c(C)[nH][nH]c2=N)=O)C1 14232,CCCCCCC(CC)NC(=O)C(C1CCCN(C(=O)CC(C)CC)C1)(C)C 14233,C#Cc1ncc(F)cc1NC(=O)NCC(c1ccc(Cl)cc1)CO 14234,c1(OC(c2nc(C(=O)OCC)n(C)n2)=O)cc([N+](=O)[O-])ccc1SCC 14235,c1(OC)c(Cl)ccc(C(N2CC=CC2C(=O)NCCN2C(=O)CSC2=S)=O)c1F 14236,C(c1nc2ccccc2o1)=CC(=O)NCC1(F)CCN(C(C(C)OCC)=O)CC1 14237,N1(C(C(CC)c2ccccc2)=O)CC2(CC(NC(c3c(C)ncn3O)=O)CO2)C1 14238,Cc1[nH]c(=N)sc1C(=O)NC1CCCC1(O)C(F)(F)F 14239,CC1CN(C(c2nn(C)cc2Cl)=O)CC1CNC(C1(C)CC=CCC1)=O 14240,C1(Cc2cn(CCCCSC)nn2)CCCC(C)C1 14241,C(=O)(C1=NNC(=O)CC1)N(CCCNC(c1cc(C)cc(C)c1)=O)CC 14242,c1(CC(=O)NC2C=CCN(C(c3c(C(=O)OC)cco3)=O)C2)cc(F)ccc1C 14243,N1(C(CC(CCC)C)=O)CCC2(CCCN(C(=O)CCS(C)=O)C2)CC1 14244,c1(CCC(=O)NCCCN(C(=O)C(C)C2=CCCC2)CC)nc2ncccn2n1 14245,c1(N2CCN(C(C34CCCN(CC3)C4)=O)CC2)ncnc2sc3ccccc3c12 14246,N1(CC(C(=C)Br)O)CCN(C2(C(N)=O)CCCC2)CC1 14247,C(C#Cc1ncccn1)NC(=O)Nc1cc(C(F)(F)F)ccc1Br 14248,C1(CC)CC(CC(N2CC(NC(=O)C(=O)OC(C)(C)C)C2)=O)CCO1 14249,N1(C(C2C(C(=O)OC)C2(F)F)=O)CCOC(C)(CNC(=O)COC2CC2)C1 14250,Cc1cc(=NC(=O)NCC2COc3ccc(O)cc3O2)c(C2CC2)c[nH]1 14251,c1(N(C(=O)CN(C(c2c[nH][nH]c2=N)=O)C2CC2)C)ccccc1O 14252,N1(C(c2c(C)nn[nH]2)=O)CCC(F)C(NC(c2cc(Br)ncc2Br)=O)C1 14253,c1(Cc2ccccc2-c2nn[nH]n2)csc2ccccc12.C12CCN1C2=O 14254,c1(C(N(C2CCN(Cc3cnn(C)c3)C2)CCC)=O)ncoc1C 14255,c1(OC(CC)=O)ccc(OCC)cc1C(N1CCCCC1CCO)=O.C1C(=O)N1 14256,N1(C(c2c(CC)nn(C)c2)=O)CCCC(F)(C(N2CCCC2(C)CO)=O)C1 14257,c1(CN2CCC(C(C(=O)Nc3cncc(OCC)c3)C)CC2)cc(F)cnc1Cl 14258,C1(NC(C2CCN(C)C2)=O)C2CN(Cc3ncc(Br)s3)CC12 14259,c1(CC(N2CCC(C)(NC(C=Cc3ccc(C)o3)=O)C2)=O)cccc([N+](=O)[O-])c1 14260,c1(NC(C2CCN(C(c3ccncc3)=O)C2)C)ncc([N+](=O)[O-])c(=N)[nH]1 14261,N1(C(Cn2cnc(=N)[nH]2)=O)CCC2CCN(C(=O)CC=C(Cl)Cl)CC2C1 14262,O=C(C1CCCc2c[nH]nc21)NC1CN(C(c2cc(F)c(F)cc2O)=O)CC1F 14263,Cc1cnc(Cl)c(C(=O)NC(C2CCN(C(c3ccco3)=O)C2)C)c1 14264,c1(C(=O)NCC2(CNC(CC(COC)C)=O)CCCCC2)cnn2ncccc12 14265,C1(C(=O)NCCC2CN(C(=O)CC3CC3)C2)CCC(CC(F)(F)F)CC1 14266,C1(C(=O)NC2CC(CNC(c3nc(C)oc3C)=O)CC2O)CC2OC1C1CC21 14267,c1(C(N(C(C)CNC(=O)Cc2cc(C3CC3)on2)C)=O)ncc(C#N)cc1F 14268,c1(OCC(=O)N=CC(O)C(=O)OCC)cccnc1OC 14269,n1(CC=C)cc(C(=O)NC2(C(N3CC(C)(OC(C)=O)C3)=O)CCC2)cn1 14270,C1(CNC(C2C(C)(C)C2(C)C)c2n(C(C)C)nnn2)CC(F)(F)C(=O)N1 14271,N1(C(C2N(C(CC(CC)O)=O)CCC=C2)=O)CC2CCCC(O)C2C1 14272,C(=O)(CC(C)CC(C)C)NCC(C(=O)N(C(CC)CO)CC)C(C)C 14273,N1(C(c2ccnc(C)c2N)=O)CCCC(C)(C)C1C(=O)NCCC(C)C(F)F 14274,O(S(=O)(=O)c1cccc2c1OC(C)C2)c1c(OC)cccc1C(=O)O 14275,CC1(C)OC2CC(C(=O)NCC3CN(C(=O)Cc4nnc(O)s4)CC3O)CC2O1 14276,Cc1n[nH]c(C)c1CC(=O)NC1CCC(CNC(c2cnsn2)=O)C1 14277,CCCC(=O)NCC(=O)NCC(F)CNC(=O)Cn1cccn1 14278,C1(CNC(c2cccc(SC)c2)=O)CN(C(c2cnns2)=O)CCC1C(F)(F)F 14279,N1(C(C(CCCC)(C)F)=O)CCC2(CCC(NC(C3CCCC3OC)=O)C2)C1 14280,N1(C(C(C(C)C)NC(C)=O)=O)CCC2CCC(NC(=O)CC3(C)CC3)C1C2 14281,c1(OC)cccc(OCC(N2CCC(NC(c3occc3Br)=O)C2)=O)c1[N+](=O)[O-] 14282,C#Cc1cncc(C(=O)NC2C=CCCC2C(=O)Nc2ccc(O)cc2CC)c1 14283,N1(C(c2c(C)sc(O)n2)=O)CCC2(CC1)CC(NC(c1ncoc1C1CC1)=O)C2 14284,N1(C(C2C(=C)C2)=O)CCC(C)(C)C1CNC(c1scc(C)c1Br)=O 14285,C1(NC(C2CCCC2)=O)COCCN(C(=O)CC(O)Cc2ccccc2)C1 14286,C1(C(=O)NC(CC)CNC(=O)CN2CCCCC2)CCC2(CCC2)OC1 14287,c1(C(=O)NC2CC(F)(CNC(CSCC#C)=O)C2)cc(S(=O)(=O)CC)ccc1F 14288,CC1CC(c2cn(CCN3CCNC3=O)nn2)CCN1C(C1CS(=O)(=O)C1)=O 14289,N1(C(c2cnn(CCF)c2)C(=O)NC2CC2)CCN(c2ccc(Cl)cc2)CC1 14290,Cc1n[nH]c(C)c1CO.C12CN(CC1C(F)F)C(=O)c1ccn(n1)CC(=O)N2C 14291,c1(C(N2C(CN(C(=O)CC3(C)CCCC3)C)COCC2)=O)cccc(S(C)=O)c1 14292,N(C1c2ccccc2CC1NC(=O)C(O)P(C)(C)=O)C(C(CCSC)OC)=O 14293,c1(OC)c(C(=O)NC2CC(C)CN(C(c3cnc(Cl)c(Br)c3)=O)C2)cccc1Cl 14294,C1(CNC(c2c(C)nc(CNC(C(CC)O)=O)o2)=O)CC12CCCCC2 14295,N1(C(CCC=CC(C)C)=O)CCN(C(C2CCCN2C2CCOCC2)=O)CC1C 14296,N1(C(C(C)=C2CC2)=O)CCC2C(CCCN2C(=O)Cn2cnnn2)C1 14297,C(S(=O)CC(=O)N1CCC(C(=O)NCc2nc[nH]n2)CC1)c1ccc(CC)o1 14298,C1(NC(CC(=C)C)=O)CN(C(=O)C(C)Oc2cc(C)ccc2Cl)CC(F)(F)C1 14299,Cc1c(C(=O)NC2CC(C)CN(C(C3CCC(C)CC3)=O)C2)cccc1F 14300,C1(NC(c2occ(C(=O)OC)c2)=O)C2CC(CN(C(c3csnn3)=O)C2)C1CO 14301,CCCC(C(=O)NCC(C(C)C)NC(c1cn(CC(=O)N(C)C)nn1)=O)N(C)C 14302,N1(C(C2CC3C(C)(C)C3C2)=O)CC2=C(C1)CN(C(c1cnoc1C1CCC1)=O)C2 14303,N1(C(c2ccc(CC)o2)=O)CCN(C(CNC(C2CC2C)=O)C(F)F)CC1 14304,Cc1ncc(C#N)cc1NC(=O)C(O)CCNC(C1C2CCCCCC12)=O 14305,N1(C(C2=CCN(C(c3c(C)n(C)cc3)=O)C2)=O)CCC(O)C(C)(C)C1 14306,CC1(C)CC(NC(C2CN(C(c3ccccc3)=O)CCS2)=O)CC(C)(C)O1 14307,C1(C(=O)NCCCN(C(=O)Cc2nn(C)cc2Br)CC)CC2CC(=O)C1C2 14308,N1(C(Cc2ccc(C)cc2Cl)=O)CCC(CNC(c2ncc(C)s2)=O)C12CCC2 14309,Cc1cc(F)c(C(=O)N(CCN(C)C(C2CCCC3CC23)=O)C(C)C)cc1F 14310,C1(C#N)(C(=O)NCC(CNC(c2c(NC(C)=O)cccn2)=O)OC)CCCCC1 14311,c1(C(=O)NCC(C)NC(C2CC3CC3C2)=O)ccncc1I 14312,C1(C2CCC2)(C(=O)NCc2cnc(NOC(c3cn(CC)nc3CC)=O)s2)CCC1.O 14313,c1(CN2CC3N(C(c4c(OC)ccc(F)c4)=O)C(C3)C2)cccc(F)c1C#N 14314,C1(CNC(CCOCCC)=O)CC(F)(F)CN1C(=O)Cc1ccn(C)n1 14315,c1(OC)cccc(CC(N2CC(NC(C3CC4(CC4)C3)=O)C(SC)C2)=O)c1F 14316,N1(C(C(C)=C(C)C)=O)CC2CC3CC2C1C3NC(=O)Cc1ccoc1 14317,Cc1ccccc1C1(C(N2CCC(C(=O)NC3CC3Cn3cnnn3)C2)=O)CC1 14318,C1(NC(C=CCCC)=O)CCOC12CCN(C(C1CC3COCC3C1)=O)CC2 14319,C1(CNC(C(COC)O)=O)CC2(CO1)CN(C(=O)CN(C)C)C2 14320,c1(-c2cn(C(N3CCN(CC(C)O)CC3)CC)nn2)cc(C)nc(C)c1 14321,c1(C(=O)NCC(C)N(C(=O)Cc2cn(C)nn2)C)ccc2ncnn2n1 14322,Cc1nnc2n1CC(C(=O)NC(CNC(c1nccn3cnnc13)=O)C(C)C)C2 14323,C1(C(N(C2CN(C(C=C(CC)CC)=O)CC23CC3)C)=O)CC(=O)N(C)C(=O)N1 14324,C#Cc1cccc(C(=O)NCCOC2CN(C(=O)COc3ccc(F)nc3)C2)c1 14325,c1(C(=O)NCC(C)CN(C(=O)C2=CCCC2C)C)cc2c([N+](=O)[O-])cccc2[nH]1 14326,C1(CCC)(NC(C2OCCO2)=O)CCCN(C(=O)CC2CCCCC(=O)N2)C1 14327,C1(NC(c2cc(C(=O)OC)ncc2)=O)CC(N=c2[nH]nc(CO)s2)C1(C)C.C1CC1 14328,C12(CNC(C34CC(CC(C)O3)C4)=O)CN(C(=O)C=CC3CC3)CC1CCO2 14329,C1(OC)CCC(CC(=O)NCC2CC(C)N(C(=O)Cc3cccnc3Cl)C2)CC1 14330,C(=O)(C1=CC2(CCN(C(=O)CC3COC(=O)C3)C2)C1)NC(CC#C)CC#C 14331,C1(C(N2CC(COC)(CNC(=O)Cc3cnoc3)C2)=O)CCC(C)(C)O1 14332,C12(CNC(c3c(C)nsc3)=O)CCCC1CN(C(=O)CCc1ccccc1)C2 14333,c1(C(CC)NC(=O)C(=O)Nc2nc(C)c(Br)cc2Br)nc2cc(Cl)ccc2o1 14334,C1(CC(=O)NC(c2noc(C)n2)CC)CN(C(c2ccnc(O)c2)=O)CCC1C 14335,C(c1c(C)noc1C)=CC(=O)NC(c1sc(C(=O)OCC)c(C)n1)C 14336,c1(C(N2CCC(O)(C(C)NC(c3nnc(C)s3)=O)C2)=O)csc2cccnc12 14337,c1(C(C(=O)NCC2CC(O)(CNC(=O)C3=CCC3)C2)=O)cc(F)cc(Cl)c1 14338,CCCC(C(=O)NCCN(c1ncnc(=N)[nH]1)CC)S(N)(=O)=O 14339,c1(CCC(=O)NC2CC3CC(NC(C4C(=C)C4)=O)C2C3)nc2ccccc2[nH]1 14340,c1(C(N2CC(N(C)C)C(C)(C)C2)=O)coc2c1CN(C(C1CCCC(O)C1)=O)C2 14341,C1(C)(CNC(=NCCOC)NCC2CCOC2)Cc2ccccc2C1 14342,C1(NC(CCCC(C)=O)=O)CCN(C)C12CCCN(C(C1CCC(=O)N1)=O)C2 14343,Cc1cc(C(N2CCC(O)(CNC(=O)C(F)(F)C(C)O)C2)=O)ncc1C#N 14344,CCC(O)C(F)(F)C(=O)NC(C)CNC(=O)CCCSC(C)(C)C 14345,C1(NC(c2c(OC)n(C)nc2)=O)CC2(CCN(C(C3CCCN3C)=O)C2)C1 14346,N1(C(C(C)O)=O)C2CCC1CN(C(C1CCN(CC(F)(F)F)CC1)=O)CC2 14347,N1(C(c2c(CC)cc(N)cc2OC)=O)CC2CCCC(NC(=O)C(C)Br)C2C1 14348,C(C(=O)NC1C=CC(C(=O)NCCc2c[nH]nc2O)C1)(C(C)C)OCC 14349,C1(C(=O)NC2(C)CC2)C2CC1N(C(C1OCCOC1c1ccccc1)=O)C2 14350,c1(OC)ccc(Br)c(CN2CCCC(C(=O)NCC3CCC(C)(C)CC3)CC2)n1 14351,Cn1nnc2cc(C(N3CCC(C4CCCN4c4ccnc(Cl)n4)C3)=O)cnc12 14352,Cc1cc(N)n2ncc(C(=O)NCC=CCNC(=O)COc3ccccc3)c2n1 14353,CC(C)CC(C)(O)C(=O)NC1CCC1C(=O)NC1CCCC(CO)C1 14354,c1(C(=O)NCCN(C(c2cnc(C(C)C)nc2)=O)C(C)C)cc(F)cc(N)c1F 14355,C1(NC(CC=C)=O)CC(C(=O)Nc2cnccc2CC)C1(C)C 14356,O=C(C(O)C(F)(F)F)N1CCOCCC1C(F)F 14357,CCC(C#N)C(=O)NC(C(=O)NCc1ncc(C)s1)C1CC1 14358,c1(C(N(CC(CC)(C)OC)C)=O)cc(S(N)(=O)=O)c(C)o1 14359,c1(-c2nc(CC3ON=C(C)C3)sc2)c(F)cccc1Cl.N12CCCC(C1)C2=O 14360,C=C(CNC(c1nnnn1CCSC)(C)COC(C)C)C1CCOCC1 14361,C1(N(C)C(c2cncc(N3CCCC3)n2)=O)CCCN(C(c2csnn2)=O)CC1 14362,c1(CNC(C2C(c3ccc(C)o3)C2)=O)cccc(N=c2cc[nH]cc2)c1 14363,N1(C(c2c(C)cc(SC)o2)=O)CC2CC(NC(C3CCCC3(C)C)=O)C2C1 14364,C1(CNC(C(CSC)O)=O)CCN(C(c2noc3c2COCC3)=O)CCC1(F)F 14365,C1(OC)CCN(C(=O)N(C(C)C)Cc2ccccc2)CC1.C12CCCN1C2 14366,N1(C(CC(C)N(C(C(CCCC)O)=O)C)=O)CC2(CCCCCC2)C1 14367,O=C(C(O)C1CN(C(=O)C(=O)NC2CC2)C1)NCC(O)CO 14368,C1(C(=O)NCCC2N(C(CSCCCC)=O)CCOC2)CCC(C)=C(C)C1 14369,N1(C(c2n(CC(C)C)ncc2)=O)CCCC2(CCC(NC(C3(C)CC3)=O)C2)C1 14370,C(=O)(C1=NOC2(CCC2)C1)N(CCCC(=O)NCCOCC(C)(C)O)C 14371,CC1=CCC(N=c2ccc(Br)c(S(=O)(=O)NC3CCC4(CC4)C3)[nH]2)CC1 14372,C(c1cc(Cl)c2c(c1)OCO2)=CC(=O)NC.CC1(C(=O)NCC2CC2)CCCNC1=O 14373,S(=O)(=O)(c1ccc(Cl)cc1)NC(C(=O)NC(c1ccc(C(F)(F)F)cc1)C)CO 14374,c1(OC)cc(C(N2CC(C(=O)NC3CCC(C(C)O)CC3)C(C)C2)=O)nn1C 14375,c1(C(N(CC(CO)(CO)NC(C(C=CC)O)=O)C)=O)cc(Cl)cc2cccnc12 14376,C12(NC(CC(C=C)C)=O)CC(CNC(c3cnn(C)c3)=O)(C1)OC21CCOCC1 14377,C(=O)(CC(C(F)(F)F)NC(=O)CCn1ccc(C)n1)NCCC1ON=C(C)C1 14378,Cn1ncc2cccc(C(N3CCC4CN(C(c5ccnc(O)c5)=O)CC34)=O)c12 14379,CC1(C#CC(=O)NCCc2ocnc2CNC(=O)CC2CCC3CC23)COC1 14380,S(=O)(=O)(c1cnn2ccc(=NCC(C)(C)C(O)C(C)C)[nH]c12)NC(CCC=C)C 14381,c1(C(N2CC(NC(c3cc(CC)ncc3)=O)C(O)C2)=O)oc2ccccc2c1Cl 14382,c1(C(C)C)cccc(F)c1C(=O)NC1CC(NC(C2C3CC4C(C3)C24)=O)C1 14383,C#CCCCCC(=O)NC(Cn1cccn1)C(=O)NC(C)(C)C#CC 14384,c1(C(=O)NCc2c(C(=O)NCCS(CC)=O)nco2)cnc(O)cc1C 14385,Cc1cc(=O)n(CCC(N2CCC(NC(c3cnns3)=O)C2C(C)(C)C)=O)cn1 14386,C=CCC(CO)NC(C1(C2CCCN2C(=O)CCC2CCC(=O)C2)CC1)=O 14387,C1(CN(C)C(C23CSCC2C3)=O)CCN(C(C2CC23CCC3)=O)CC1 14388,C1(C(C)CNC(=O)C(=O)NCC2CC2)CCCN(C(=O)C=CC2CC2)C1 14389,C1(CNC(CCCC#C)=O)COC(C)(C)CN1C(C1CCC(F)(F)C1)=O 14390,C=CC(CCC)CC(=O)NCCC1CCCN(C(C2(C(C)C)CCC2)=O)C1 14391,c1(C(=O)NCCNC(c2c(C)c3c(s2)ccs3)=O)cc2c(s1)CC(C)CC2C 14392,c1(NCCC(C)S(C)=O)nc2ccccc2nc1NCCCCCN(C)C 14393,n1(CC)c(SCC(C)C(=O)N(C)C(=O)OC)nc2ccccc12 14394,N1(CCN(C(c2c(CC)c[nH]n2)=O)C)CCN(C(=O)C(O)C2CC2)CC1 14395,c1(C(N2CC(NC(CCSCC)=O)C(C)CC2)=O)nn2c(c1C)OCCC2 14396,CCC(CC)(CC)C(=O)N1CCC(N(C(=O)Cc2csc(C3CC3)n2)C)C1 14397,C#Cc1ccc(C(=O)N(C2CCCN(C(c3ccn(C4CCC4)n3)=O)C2)C)nc1 14398,C(CNC(c1cccn(C)c1=O)=O)(CC(F)(F)F)NC(C(=Cc1cccs1)C)=O 14399,c1(NC2CCN(C(C)=O)CC2)nc2c(c(=NCC34CCCCC3C4)[nH]1)CSC2 14400,c1(OC)ccc(S(=O)(=O)NCC2CCC(CSC)CC2)cc1 14401,C(CCC(N)=O)(C(=O)NCc1cc(C2CC2)n[nH]1)n1cc(CCN(C)CC)nn1 14402,N(C1CCCn2ncnc21)C(C1C2CN(C(=O)C3=C(Cl)CCCC3)CC21)=O 14403,CN1N=CC(CC(N2CC3C(CNC(=O)Cc4nnc(S)n4C)C3C2)=O)C1=O 14404,CC1(C=CC(=O)NCC2CCC(NC(=O)CCc3cncs3)C2)CCOCC1 14405,c1(C(=O)NC(C)CNC(=O)COC(F)(F)F)nc(OCCO)ccc1Cl 14406,N1(C(CCC(=C)C)=O)CCC(NC(c2ccc(OC(F)F)cn2)=O)CC1C1CC1 14407,C(c1ccc(Br)cc1)=CC(=O)NC(C)CCCNC(=O)CP(C)(C)=O 14408,N1(C(COCc2cc(C)no2)=O)CCCC1(C)CNC(c1nccs1)=O 14409,c1(SC)nc(N2CCC(NC(c3cccnc3O)=O)CC2)c(Br)c(C)n1 14410,C(=O)(C(O)(C(C)C)C(F)(F)F)NC1CCCC(NC(c2cc(OC)ncn2)=O)C1 14411,CC1CC(NC(c2cccc(Br)c2)=O)CCN1C(=O)CC1CCCCN1C 14412,C#CC1CCC(C(=O)NCCN(C(=O)C(C)N2CC(C)C2)CCOC)CC1 14413,C12(C(N3CC4C(CC(=O)NCCc5ccc(O)cc5)C4C3)=O)CCCC1OCC2 14414,C1(O)(C(C)NC(CSCCC)=O)CCN(C(C2C=CC=CC=C2)=O)CC1 14415,c1(C(N(CC)CC2CCCN2C(=O)CSCC(C)C)=O)scc(Cl)c1Cl 14416,C1(NC(C(CSC)C)=O)CCCN(C(c2ccccc2OC2CCC2)=O)CCC1 14417,Cn1[nH]nnc1=NCCCC(C)(C)NC(C1CC(c2cccc(F)c2)(F)C1)=O 14418,c1(C(=O)NC2C3CCN(C(C(C=C)O)=O)C32)ccc(C)c(C)c1 14419,c12ncc(s1)C(=O)NCC(CNC(c1cscn1)=O)OC2=O.CCOC 14420,N1(C(c2ccc(Cl)cc2)C(=O)NCCC#N)CCCN2CCCCC12 14421,c1(C(N2CCC(N(C(CSCCC)=O)C)C2)=O)cc2c(nn1)CCCC2 14422,Cc1nn(C)c(C(=O)NCC(CO)NC(=O)CNC(N)=O)c1I 14423,c1(C(N2CC(CCC)C(NC(=O)CCC=CBr)C2)=O)cc(C)cc(O)n1 14424,C(=O)(C(C)(CC)CC)NCc1ccc(C(N(CC=C)CC)=O)o1 14425,Cc1ccc(NC(C)C)c(C(=O)NC23CC(NC(=O)CCc4ccoc4)(C2)C3)c1 14426,N1(C(C2(CC(C)C)CC2)=O)CCN(C(=O)CNC(=O)Cc2cc(C)nn2C)CC1 14427,C1(N(C)CC)(C(=O)NC2CC(CCNC(=O)C(C)OCCF)C2)CCC1 14428,c1(NCC2CC(CN=c3[nH]nc(C(C)C)o3)OC2)ccnc2[nH]nnc12 14429,c1(CCC(c2cc3c(cn2)OCC3)=O)nc(O)c2c3c(sc2n1)CCC3 14430,N1(C(C2C(C)CCC2)=O)CCCCC(Cn2cc(CCc3ccccc3)nn2)C1 14431,O=S(=O)(c1ccc2nc(N3CCC(O)C(F)C3)ccc2c1)N1C2CCC1CC2 14432,c1(CC(=O)NC(C2CCN(C(c3cncnc3)=O)CC2)C)ccccc1S(C)=O 14433,C1(n2c(COC(F)(F)F)nc(-c3ccc(OC(C)C)cc3)n2)C(C)CCCC1C 14434,N1(C(c2c(OC)nc(C)nc2)=O)CCCN(C(c2ccc(F)cc2C)=O)CC1C 14435,c1(N2CCC(CC)(OC)C2)cc(=NCCc2cnc3ncccn23)[nH]c(CC)n1 14436,CCCC(CCC)CC(=O)N1CCOCC1CNC(=O)C(C)(CC)CO 14437,CONC(=O)CNC(=O)CCC1CC(NC(c2coc(C(N)=O)c2)=O)C1 14438,C1(OC(C)C)CC(=O)N(CCC)C1CCC(C)C 14439,C1(NC(c2cc(C3CC3)cs2)=O)CCN(C(C2CCCCS2(=O)=O)=O)CC(O)C1 14440,N1(C(c2c(CC)sc(=N)[nH]2)=O)CCN(C(=O)COCc2ccnc(O)c2)C2CC12 14441,C1(C(N(C)CCc2cccs2)=O)CCN(N2CCN(Cc3cncn3C)CC2)C1 14442,CC(CC#N)N=c1cc[nH]cc1S(=O)(=O)NC1(NCCn2ccnc2)CCCCC1 14443,N1(C(c2ccc(Cn3cc(CNC=O)nn3)o2)=O)C(CO)CCC12CCC2 14444,c1(C(=O)NC(COC)CNC(=O)C(C)(COC)OC)cc(C)c(O)c([N+](=O)[O-])c1 14445,c1(CNC(CCNC(C=C(C)C)=O)=O)cccnc1C(F)(F)F 14446,c1(C(=O)NCCN(C(=O)C(C2CCCO2)OC)CC)cnn(CC(F)F)c1 14447,C(=O)(C(C)CC(C)C)N1CCC(N(C(C(C(=O)OCC)F)=O)C)CC1 14448,c1(C(=O)NC23CC(C(N(C(CC)CO)CC)=O)(C2)C3)cc(Br)cc(F)c1F.N 14449,N1(C(C(C)n2cncn2)=O)CC2C(N(C(=O)CCCN(C)C)C)C2C1 14450,c1(CN2CCC(NC(c3cc(OC)cc(OC)c3)=O)CC2)ccc(Cl)c(C)c1F 14451,N(C(=S)N1CCC1c1ccccc1)c1ccc(C)o1.c12ccc(cc1)N(C)C2 14452,Cn1cc(C(=O)NCC23CC2CN(C(c2ccnn2CC2CCC2)=O)C3)c(Cl)n1 14453,CCC(C)(COC)CNC(=O)CONC(=O)C=Cc1cncs1 14454,C(C)(C)(CC(=O)NC(C)CC(C)NC(=O)CCCCc1cnc[nH]1)OC 14455,C1(C(N2CC(NC(C(CC)(C)O)=O)C(C)C2)=O)CC(c2cccnc2)=NO1 14456,C1(OC)CN(C(c2ccn(-c3ccc(Nc4cnn(C)c4)cc3)n2)=O)CC1O 14457,c1(C(=O)NC2(CO)CCN(C(C(COC)O)=O)C2)cc(F)c(SC)cc1N 14458,C1(CC)C(C(=O)Nc2ccccc2OC)CCN1C(c1cnn(C(C)C)c1)=O 14459,N1(C(C(F)(F)C2(OC)CCC2)=O)CCC(NC(=O)C2=CCCCC2)CC(C)(C)C1 14460,N1(C(C(C)OC2CCCCC2)=O)CCC(C)C(NC(=O)C(C)(C)CO)C1 14461,CCC(CC)C(=O)N(C)CC1CN(C(c2ncn(C(C)(C)C)n2)=O)CCO1 14462,c1(CN(C(C(C)OCC2CC2)=O)C)cnn2c1CN(C(c1cc(Cl)no1)=O)CC2 14463,N1(C(Cc2c(C)non2)=O)CCC2CCN(C(C3CC(C)(C)CN3C)=O)CC12 14464,C1(CNC(C(C)Oc2cccc(F)c2)=O)CN(C(=O)CCC2CC2)CCS1(=O)=O 14465,C#Cc1cccc(C(=O)NC2CCN(C(C3CC=CC3)=O)C(C3CC3)C2)c1Cl 14466,c1(N(CC(C)C(C)(C)C)C)nc2c(c(=NC3COC(C)(C)C3)[nH]1)COCC2 14467,C(C(CO)(CO)NC(c1cncnc1)=O)N(C(C1C(OC)C1)=O)C 14468,c1(C(=O)Nc2ccc(OCC(=O)NCC)cc2)c(C#N)cnn1C 14469,C1(NC(C(CC(=O)OC)C)=O)CC2CCC1CC2NC(=O)CC1(CS(C)(=O)=O)CC1 14470,c1(C(=O)NC23C(CN(C(CC4C(C)(C)CC4)=O)C2)C3)cccc2c1OCCO2 14471,C1(C(N2CC(CNC(c3cc(OC)no3)=O)(COC)C2)=O)CCCCN1C(C)C 14472,C(CC(C)(C)C(=O)N1CCCC(CN(C(=O)Cc2csc(Cl)c2)C)C1)OC 14473,C1(C(N(CC(C)C#N)C)=O)CCCCCC1NC(C1CCC(F)CC1)=O 14474,N1(C(C)=O)CCCC(C(=O)NCC2CN(C(c3cnnn3C)=O)CCO2)C1 14475,N1(C(C(CC=CC)CC)=O)CCCN(C(=O)CCC)C(C)C1 14476,N=c1cc[nH]cc1C(=O)NCC(O)CNC(c1ccnc(OCCO)c1)=O 14477,C1(O)(CNC(Cc2cncc(C)c2)=O)CCCN(C(c2nn(C)c(C)c2Cl)=O)C1 14478,c1(CC(=O)NCCN2CCN(C(c3c(CC)onc3)=O)CC2)c(C)nc(O)nc1C 14479,Cc1nc(CNC(C2CC2c2ccco2)C)sc1C(=O)O 14480,Cc1c[nH]cc1C(=O)N(C)CCOCCN(C)C(C1CC1C(C)O)=O 14481,C12(CNC(C=CC)=O)CC(NC(=O)CC(CC)SC)(C1)C(C)(C)O2 14482,C1(N)(CC)CCCN(C(=O)C(N2CCCC(N3CCC3)C2)=O)C1 14483,CCCC(CC)CCC(=O)NC1CCC2CCN(C(=O)Cc3coc(C)n3)C1C2 14484,CCCCS(=O)(=O)NCC(=O)NC1CC1NC(c1ccc(C(F)(F)F)cn1)=O 14485,C(=O)(C(CC(N)=O)NC(c1cc(C)n(C)c1)=O)NCCCOCCCC 14486,c1(C(CC)C)nc(-c2coc(C)n2)n(C(C)C(C)(C)C)n1 14487,N1(C(CSCC=C)=O)CCCN(C(C2(C3CC3)CC2)=O)CC1c1ccccc1 14488,N1(C(CN2C(C)CCC2)=O)CC=CC(NC(C2CC2C)=O)C1 14489,N1(C(C(CC(C)C)(F)F)=O)CCOC2(CCC(NC(=O)C(C)(C)CF)CC2)C1 14490,C1(NC(c2c(C(C)O)cccc2)=O)CCN(C(C2CC(O)C2)=O)C(C)C1 14491,C1(C2CCCOC2)(NC(C(CC2CCCC2)NC(C(C=C)OC)=O)=O)CC1 14492,c1(C(N2CC(NC(C3C(CC)OCC3)=O)C(C)C2)=O)cncc(N=[N+]=[N-])c1 14493,c1(OCCOC)ccc(C(=O)NCC(O)CN(C(=O)C#CC2CC2)C)c(Cl)c1 14494,C1(C(=O)NC2(CF)CCN(C(c3scc(C(C)=O)c3)=O)C2)CCCC1S(C)(=O)=O 14495,c1(C(N(C(=O)CC2CC=CCC2)C(C)C)=O)cncc2nc[nH]c12 14496,C=Cc1ccccc1NC(=O)CC(=C)C 14497,Cc1c(C(=O)NC2CC2NC(=O)CCC2CCCC2)cc(-c2ccccc2)n1C 14498,N1(C(CC2(OC)CCC2)=O)CCN(C(c2cccc(F)c2O)=O)C2(CC2)C1 14499,N1(Cc2ccccc2)CCC2CCN(NCc3nc(CC)[nH]n3)CC12 14500,C1(O)(C(C)NC(COCCNC(c2c(C)scc2)=O)=O)CCCCC1 14501,C1(C(=O)NCCN(C(=O)CC2(C(F)F)CC2)C(C)C)CCC(C(F)(F)F)O1 14502,CC1CN(C(C2CC3CCC2C3)=O)CCC1CNC(c1cnn(C(F)(F)F)c1)=O 14503,c1(CC(N2CC3(CC(CNC(C(C)(O)C4CC4)=O)C3)C2)=O)csc2ccccc12 14504,Cc1cc(C(=O)N(CCC(=O)NC2CC2(C)C(F)F)C(C)C)c(C)[nH]1 14505,N1(C(C(C2CC2)SC)=O)CC2(C(=O)N(CC3=CCSC3)C)CC1CO2 14506,N(C1CC2(CN(C(=O)C=C3CC3)C2)n2ccnc21)C(C1C(=O)NCC1)=O 14507,C1(C(=O)NCc2nc(CNC(=O)OC(C)(C)C)oc2)CCc2nnc(O)n2C1 14508,Cc1cccc(OCC(=O)NCCC(C)N(C(=O)CCCC#N)C)c1 14509,CCCCC(C(=O)N1CCN(C(c2cc(C(C)(C)C)oc2C)=O)CC1CC)N(C)C 14510,c1(C(C(C)C)Nc2c(O)ccc(C#C)c2)ccc2ccccc2c1 14511,C(=O)(C(C)S(N)(=O)=O)N1CC(O)(CNC(c2c(C)n(-c3cnn(C)c3)nn2)=O)C1 14512,C(=O)(CC1C(=O)Nc2ccccc21)NCC1N(C(CC(C)(C)CC(F)F)=O)CC1 14513,C1(C2CCNCC2)(C(=O)NCC(Cc2ccccc2C(F)(F)F)CO)CCC1 14514,C(=O)(C(C)CC(C)(F)F)N(C(CCNC(CC(C=C)(C)C)=O)C)C 14515,C1(C(=O)NC(C)CC2CN(C(c3cccnc3N)=O)C2)CCCN2CCCCC12 14516,C(=O)(CCCCC(N)=O)N1CCC(CNC(CN2CCCC(N(C)C)C2)=O)CC1 14517,CC1OC2(C)CC1(C(=O)NCC1CCCC(NC(C3C4COCC34)=O)C1)C2 14518,c1(CC)nc(N2CC=CC(NC(c3ccccc3C(F)F)=O)C2)[nH]c(=N)n1 14519,CCC(C)(C)C(C)CC(=O)NC1CC2CCC1(NC(=O)CN(CC(C)(C)C)C)C2 14520,c1(SC)cscc1C(N1CCC(NC(C2CC(SC)C2)=O)C1)=O 14521,c1(C(C(F)(F)F)N(C(N2CC(F)(F)C2)=O)Cc2ccc(C)o2)ccc(O)cc1 14522,C1(NC(C(CCC)C)=O)CC2(CCN(c3cc(Cl)nc(CC)n3)CC2)C1 14523,C1(C(N)=O)CCC(CCC(=O)NCC2CCN2C(c2ccsc2Cl)=O)O1 14524,c1(OC)ccncc1CC(=O)NC1COCCC1NC(c1csc(C(C)C)n1)=O 14525,c1(C(N2CC3(CCN3C(c3cc(Cl)sc3Cl)=O)C2)=O)cc2n(c1)CCOC2 14526,N1(C(CC=CCC)=O)CCCC(OC(N2CCC2C)=O)C1 14527,c1(C(=O)NCC2C=CCN2C(c2cnc(O)s2)=O)coc2c(Cl)cccc12 14528,C1(NC(C2(C(=O)NC)CCC2)=O)CCC(Nc2ncncc2I)CC1 14529,c1(CNC(c2c(C)n[nH]c2)=O)ccc(C(C)NC(c2c[nH]nc2C(C)C)=O)cc1 14530,C1(C(=O)NCc2c(CNC(c3n[nH]c(C)c3O)=O)cccc2)CC12CCCCC2 14531,C(=O)(C(CCC=C)NC(=O)C(c1cnn(C)c1)=O)NC(C#C)CC1CCCC1 14532,C1(CNC(=O)C=Cc2cn[nH]c2)(NC(C2SCCCS2)=O)CC2CCC1C2 14533,c1(CC)ccc(C(=O)OCC(=O)CCC2CC2)cc1[N+](=O)[O-] 14534,O(NC(=O)C(CCC1CC1)NC(=O)C(C)CC)CC(=O)OCC 14535,CCC(CC)N(CCC(=O)NC(C1CN(C(=O)Cc2cn[nH]c2)C1)C)C 14536,c1(C(N(C2CCN(C(CSCC=C)=O)C2)C)=O)cc(C)nc(N2CCCC2)n1 14537,C1(NC(c2c(C)ncs2)=O)CCCOC12CCN(C(=O)CC1CC=CCC1)CC2 14538,N1(C(CCCCC#N)=O)CCN(C(=O)Cc2noc3ccccc23)CC(CO)C1 14539,C1(NC(C2C(CCC)C2)=O)C=CCCC1C(=O)NCc1cn(C(C)C)nn1 14540,CC1CN(C(=O)CCCC2CN(C(=O)CN(C)C)C2)CC1NC(=O)OC(C)(C)C 14541,C1(CNC(C(COC)(F)F)=O)CN(C(=O)C(C)N(C)C(C)=O)C2(CCC2)C1 14542,C(=O)(C(C)(C)CC(C)C)N1CCN(C2C(NC(C=NOC)=O)CCC2)CC1 14543,N1(C(CCC(C2CCCC2)OC)=O)CCCC1CC(C1C(C)C1C)=O.C(C)OC 14544,C(=O)(C(C)(C)C(F)F)NC1CC2(C(NC(c3cc(COC)cn3C)=O)C2)C1 14545,c1(NC(C)=O)cccc(NC(=O)CC(c2cn(C)nc2C(F)(F)F)C)c1 14546,C1(NC(C2CC(N(C)CC)C2)=O)CCCC(NC(c2cncc(F)c2)=O)CC1 14547,C12(C(=O)NCC3(C)CCCOC3)CCCC1CCN2C(=O)CCS(C)(=O)=O 14548,C1(NC(C2(CC)CCC2)=O)CN(C(=O)C(C)Oc2cccc(C)c2)CC1C1CC1 14549,c1(C(=O)NCC2N(C(C(C)(C)OC(C)=O)=O)CCC2)cccn2nccc12 14550,C=C(Cl)C(C)(C)C(=O)N(C)CCOCCNC(c1cc(OC(C)C)nc(C)c1)=O 14551,Cc1c(C(=O)NCc2ccsc2C(=O)NCC2CCN2C(C)(C)C)cccc1F 14552,c1(C(N(C)CCNC(c2ccc(N)c(Cl)c2)=O)=O)nsc2ccccc12 14553,c1(C(=O)NCCCCCNC(CC(=O)OC)=O)cccc(C)n1 14554,O=C(CCC(CF)CF)N1CCC(CO)C(NC(C2(c3ccno3)CC2)=O)C1 14555,C(CCN(C)C(=O)NC(C1CCC1(C)C)=O)(C(C)(C)C)NC(C)=O 14556,N1(C(c2ccc(C)n2C)=O)CCCC2C1CCCN2C(=O)C(F)F 14557,c1(C(=O)NCC2COCCN(C(C(CC(=O)OC)C)=O)C2)cnn2ccncc12 14558,c1(C(N2CC(CNC(CSCCOC)=O)C2)=O)nc(N(C)C)nc(=N)[nH]1 14559,C1(NC(C(C)NC(=O)CC(F)(F)F)=O)CC(O)CN(C(=O)OC(C)(C)C)C1 14560,Cc1ccc(C)c(C(N2CCN(C)C(C(N3CCC(OC4CC4)C3)=O)C2)=O)n1 14561,c1(CC(N2CC(O)(CNC(CC3CC(=C)C3)=O)C2)=O)ccc(N(C)C(C)=O)cc1 14562,c1(OCC(N2CCC(NC(=O)C=CSc3nc[nH]n3)C2)=O)cccc(Cl)c1 14563,CCCN=C(NCCCN1CC(C)CC(C)C1)N1CCC(COC)C1 14564,c1(C(=O)NC2CN(C(c3c(CC)cc(C)cc3)=O)CC2C)cc(C)n(C)c(=O)c1 14565,C1(C)(CC)CC(C(N2CC(N(C(=O)CCc3cc[nH]n3)C)C2)=O)C1 14566,c1(C2(C(=O)NCCCC(C)NC(C3(C(C)C)CCC3)=O)CC2)cccc(Cl)n1 14567,C1(O)(CCNC(C2CCCN(C(C)C)C2)=O)CCCN(C(=O)COCCF)C1 14568,c1(C(=O)NCC(CNC(CCCCC#C)=O)(C)F)ccc2cccnc2n1 14569,CC(C)CC(C)(CNC(C1CC1C(C)C)=O)NC(C1(CCF)CCOCC1)=O 14570,C1(C(=O)NCCCC(C)(F)F)(CNC(CCOC(C)=O)=O)CC2(CC2)C1 14571,N1(C(CCCCC)=O)CC2CCC(C1)N2C(=O)CC1(O)CCOCC1 14572,C(=O)(C1SCCc2sccc21)N1CCOCC(CNC(C=CCOC)=O)C1 14573,N1(C(CCCOCC)=O)CCN(C(C2(CN(C)C)CCCC2)=O)CC1C1CC1 14574,c1(C(=O)NC2CN(C(C3CCCCO3)=O)C2)cc([N+](=O)[O-])c2nsnc2c1 14575,c1(N(C(NN(C2CCCCO2)CCCC)=S)C)cc(CC)c(Br)nc1Br.CC 14576,CC(C)CCCCCC(=O)N1CCC(O)(C(C)CNC(=O)C2=CC3C=CC2C3)C1 14577,c1(C(N2CC(C)C(CNC(c3ccccn3)=O)CC2)=O)c[nH]c2cc(O)ccc12 14578,Cc1cc(Br)cnc1C(N1CCCC1CC1CC1)C(=O)NCCC#N 14579,C(=O)(C(C)C(=O)NC1CC(C)(NC(=O)CCc2ccc(C(F)(F)F)nc2)C1)OC 14580,c1(CCC)ccc(C=CC(=O)N(CCC(C(C)C)NC(=O)C(O)CCC)C)cc1 14581,Cc1ccc(F)c(CNC(C2CCC(NC(c3cnc(Cl)c(Cl)c3)=O)C2)=O)c1F 14582,C(=O)(C(F)C(F)(F)F)NC(C1N(C(c2cc(SC)ncc2)=O)CCC1)C 14583,CCC(CC)(CCNC(c1c(C)coc1C(C)C)=O)NC(=O)CCCSC 14584,N1(C(COC)=O)CC(C)(C)CCC1CNC(=O)CS(=O)(=O)CC1CCCO1 14585,Cc1cnccc1C(C(=O)NCC(C)C)N(CC(N1CCCCC1)C)C 14586,N1(C(c2nc(C)oc2)=O)CC(NC(c2cc(C)c(Br)o2)=O)CCC(O)C1 14587,c1(C(N(CC=CC(=O)NCC(CC)(C)Cl)C)=O)ccc(F)cn1 14588,N1(C(C(=O)N(C(CCCC)CO)CC)=O)C(C(N2CCC(O)C2)=O)C2CC(F)C1C2 14589,C1(NC(CC=CCC)=O)CCC(C(=O)NCCC(Cl)Cl)C1 14590,C#Cc1cccc(C(N2CC(C#N)(CNC(=O)OC(C)(C)C)C2)=O)c1Cl 14591,N1(C(=O)Nc2cncc(C(C)(C)C)n2)CCCN(C(=O)C2=CCC2)CC1CO 14592,N1(C(C(N2CCNC2=O)C)=O)CC2(CC(NC(c3cncnc3)=O)c3nccn32)C1 14593,C(=O)(CCC(F)(F)F)N1CC(NC(CN2CC(C)(C)C2)=O)C(CC2CC2)C1 14594,C1(C(=O)OCC)CCCC(C(=O)N(C)CCN(C(c2ccnc(C)c2)=O)CC)C1 14595,CC1CCC2(CN1C(=O)NCCCn1ccccc1=O)OCc1ccccc12 14596,C#CCCN=C(NCCC(CCC)NC)NC1CCN(S(C)(=O)=O)C1 14597,C1(NC(c2n(CCC)ncc2)=O)CCN(C(c2cc(Br)n(C)c2)=O)CC1 14598,N1(C(c2sccc2CO)=O)CCN(C(=O)C=CC2CC2)CC1 14599,CC(C)(C(=O)NCC(O)CNC(c1csc(CO)n1)=O)C1CCCC1 14600,C(=O)(C(CC(F)F)NC(=O)C=NOC)N(CCSC)CC 14601,c1(C(N2CC(C)(NC(C(=O)OCC)=O)C2)=O)c[nH]c2cc(OC)ccc12 14602,c1(C(=O)NCCN(C(c2ccc(C(C)C)o2)=O)CC)n[nH]cc1I 14603,C=C1CC2CC1CN2C(=O)CC1CC(C)N(C(c2cnn(C)c2C=C)=O)C1 14604,n1(CC)nc(C)c(CNC2C(Cn3cc(C4CC=CCC4)nn3)C2(F)F)c1C 14605,c1(CN2CCC(O)C(O)C2)ccc2nn[nH]c2c1 14606,C=C(C)C1CCC(C)(O)C(NCCc2ccc3c(c2)CCO3)C1 14607,N(C(=NCC(C)C)N1CCCCC(C)(F)C1)CC1(OCC)CCC1 14608,C1(NC(C2C(N)CCC2)=O)CCCC(F)(F)C1 14609,c1(C(=O)NCC2CCN(C(C(C)SC)=O)C2)sc2ccccc2c1Br 14610,CC(C)CC(C)(C(N)=O)NC(c1ccc(CNC(C2CCC(=O)O2)=O)nc1)=O 14611,Cc1cc(=O)oc(C)c1C(=O)NCCCCCN(C)C(c1c(C)cnnc1O)=O 14612,C1(NC(C2(OC)CC2)=O)CCC2CCN(C(c3c(C(F)F)cccc3N)=O)C1C2 14613,C12(CNC(C=COCC)=O)CCCCC1CN(C(c1ccc(SC)o1)=O)C2 14614,CC1CCC=C1C(=O)NCCC(C)N(C)C(c1ccc(O)c(CO)c1)=O 14615,C1(C#N)(C(N2CC(C(C)NC(c3cc(C4CC4)no3)=O)OCC2)=O)CCOCC1 14616,Cc1ccnc(NC2CC(O)(CNC(c3ccn(O)c(=O)c3)=O)C2)c1[N+](=O)[O-] 14617,Cc1cnc2n1CCN(C(=O)C(C)(C1CC1)N(C(=O)CCc1cn(C)nn1)C)C2 14618,C(=O)(C1=CC2CCCC12)NC12CN(C(CN(CCC)C)=O)C(CO)(C1)C2 14619,c1(OC)ccc(CN2CCN(CC(C3CCC(=O)NC3)=O)CC2)cc1 14620,C(c1cncc(O)c1)=CC(=O)NCC(CNC(c1cc(OC)ncn1)=O)O 14621,CCC(CC(=O)NCCC(C)(C)OC)N(C)C(C1CCCC(CF)C1)=O 14622,CC(C)C(F)(F)CC(=O)NC(C)(CNC(c1ccc2n[nH]cc2c1)=O)C1CCC1 14623,CC1(C)C(NC(C2CC(F)(F)C2)=O)CC1CC(=O)NCC1CCC(F)(F)C1 14624,Cn1nccc1C(=O)NCC(O)CNC(c1cc(-c2ccncc2)[nH]n1)=O 14625,CC1CC2(CC(NC(C3CC(C)N3C(c3ccc(O)c(F)c3)=O)=O)C2)C1 14626,C=C1CC(C(C(=O)NCCCC2CC2)N(CC(C)C)CC2CCOC2)C1 14627,N1(C(c2cnc(CC)s2)=O)CCCC(C2(NC(c3csc(C)n3)=O)CC2)C1 14628,c1(COCCOCC)cc(Cl)cnc1NC(CN(C(C(C)OC)=O)C1CC1)=O 14629,c1(C(c2nnnn2-c2ccccc2)(C)NCc2cc(Br)co2)ccc[n+]([O-])c1 14630,N1(C(C(CC)n2cncn2)=O)CC(NC(=O)CC2CCN(CCF)CC2)C(O)C1 14631,C(=O)(C(C)C(=O)NCC1CC1)OC.C1C(O)C(=O)N2CCC(C2)O1 14632,C(C)(C(=O)OC(C)(C)C)NC(=O)NCC1(CCN(C)C(C2(CC)CC2)=O)CC1 14633,c1(CC(=O)NC2CC(NC(=O)Cc3cnn(C(F)F)c3)C2)ccc([N+](=O)[O-])cc1 14634,C1(C(N2CC3C(CN(C(Cc4cc(C)on4)=O)C)C3C2)=O)CC2OC(=O)OC2C1 14635,C12(C(N3C(CC(NOCC(N)=O)=O)CCC3)=O)CCCC1C2(F)F 14636,Cc1ccc2nc(C(N3CC(O)CC3CNC(C3(C)CC=CCC3)=O)=O)cn2c1 14637,C(=O)(CC(CC)C(C)(C)C)NCCCCNC(CC(C=C)CCC)=O 14638,N1(C(c2cn(CCC)nn2)=O)CC2=C(C1)CN(C(c1ccc[nH]1)=O)C2 14639,C(CNC(C1CC2(CSC2)C1)=O)(CC(F)(F)F)NC(C=NOC)=O 14640,CC(C)(C)C(CO)C(=O)N1CCCC1CCNC(=O)CC1C=CCC1 14641,n1(CC(=O)NC2C3CC(NC(C4CC4[N+](=O)[O-])=O)CC23)ncccc1=O 14642,C(C)(CO)(C(=O)N1CCCC(N(C(=O)CCC2CCCC2)CCO)C1)OC 14643,C1(CCC(C)(C)NC(c2ncn(CC)c2)=O)CCCCN1C(=O)Cn1ccnn1 14644,N1(C(c2ccc(C#C)cn2)=O)C2CCC1CN(C(c1ncc(C)cc1OC)=O)C2 14645,C12(COC)CC(CNC(C3C=CCC3)=O)(CN1C(c1ccccc1CC#N)=O)C2 14646,C1(NC(c2scc(COC)c2)=O)CN(C(=O)CC(C)F)C2(CCCC2)C1 14647,C1(OC)CCCCC1NC(=O)C(C1CCN(C(C2CCNC2=O)=O)CC1)C 14648,c1(C(N(C2CCCCC2)CCNC(C=CC(C)(C)SC)=O)=O)cn2c(n1)CCCC2C 14649,CN1C(=O)CCCC1C(=O)NCC(c1ccccc1)CNC(=O)C#CC1(C)CC1 14650,C1(N(C(C(C(C)OC)O)=O)C)CCCN(C(=O)CN2CCC(C(N)=O)CC2)CC1 14651,N1(C(C2(C(=O)OC)CC2)=O)C2CCC1CN(C(c1c(C)c[nH]c1CC(N)=O)=O)C2 14652,c1(C(N2CCN(C(c3c(C)nc(CO)o3)=O)CC2C)=O)cc2cc(Cl)ccc2[nH]1 14653,C#CCCCC(=O)NCCCN(C(=O)CC1C(=O)NN=C1C)Cc1ccccc1 14654,C#Cc1cc(C(N2CCCCC2CC(=O)NCC(C)O)=O)ccc1C 14655,C1(CC(=O)NCCN(C)CC)CN(C(c2cn3c(n2)CCC3)=O)CCC1C 14656,C1(NC(C(c2cccc(F)c2)(C)O)=O)CCCN(C(C2CC2F)=O)C1 14657,c1(NC2(CNC(CC(c3ccc(C)cc3)C)=O)CC2)ccc([N+](=O)[O-])cn1 14658,c1(C(N(C(C)CNC(C2CCN(C3CC3)C2=O)=O)C)=O)c(F)cncc1Br 14659,c1(C(=O)NC(CC)(C)CNC(C2(CCN(C)C)CCC2)=O)cc(C#N)c[nH]1 14660,C#Cc1cccc(NC(C2(NC(=O)COC(C)CC)CC2C)=O)c1 14661,c1(CC)ccc(C(N2CC(NC(c3ncccc3C)=O)C(SC)C2)=O)c(Cl)c1 14662,CCC(C)(CC)C(=O)NCC(C)(CO)NC(c1cnc(C(C)OC)s1)=O 14663,S(=O)(=O)(c1cccc(=NCc2c[nH]nc2-c2cccs2)[nH]1)NC1C(CC)CCC1 14664,c1(OC)ccncc1C(=O)NCC1(CNC(c2cc(F)cs2)=O)CC1 14665,C1(OC)CC(C)CN(C(=O)CC(C)CNC(C2CCOC2(C)C)=O)C1 14666,c1(CC)ccoc1C(=O)NCC1CCCC1NC(=O)CNC(=O)NC 14667,CC1CN(C(c2ccnnc2O)=O)CC1NC(C1(Cl)CC1(F)F)=O 14668,C#Cc1cnn(C)c1C(N1CCC(O)(c2nc(C)no2)C1)=O 14669,C1(C(=O)NCC(CC(C)C)NC(=O)COC2CCOC2)CCc2nnn(C)c2C1 14670,N1(C(C(C)(C)CC#N)=O)CC2CC(NC(=O)Cc3cccc([N+](=O)[O-])c3)CC1C2 14671,c1(C(=O)OC)cc(NC(C(C(C)C)N(C)CC)=O)ccc1Cl 14672,c1(C(=O)NCCC2(NC(CCC)=O)CC2)ccc(Oc2cccc(C)c2)nc1 14673,C1(C(=O)Nc2cc(-n3cc(C(C)(C)N(C)C)nn3)ncc2)C2C(=O)OCC12Br 14674,N1(C(C(C=C)OC)=O)CCCC1(C)C(=O)NC(c1ccccn1)C 14675,C1(C(N2C(CNC(COc3cn(C(C)C)nc3)=O)CC2)=O)CC1C1CC1C 14676,c1(C(=O)NCC(C2CC2)NC(=O)C=CBr)cc(Cl)ccc1F 14677,CC(C(=O)N1CCN(C(=O)CCC2CC2)CC1CCO)C(C)(C)C 14678,C1(C(=O)NCCC(c2cccc(F)c2)C)CCCCC1NC(C1CCCO1)=O 14679,c1(CC)cccc(C(=O)NC2CC(N(C)C(c3ccc(C(F)F)o3)=O)C2)c1O 14680,c1(C(N2CCCC(C(C)=O)C2)=O)cc(F)ncc1NS(C)(=O)=O 14681,c1(C(=O)NCCC2(OC)CN(C(c3c(CC)csc3)=O)C2)cc(C)ncc1C 14682,C12(CNC(C(CC)N(C)C)=O)CCC(CC1)N2C(c1nncn1CC)=O 14683,Cc1sc2ncnc(NCC3CCCC(NC(=O)CCCNC(N)=O)C3)c2c1C 14684,N1(C(CN(C(=O)OCC)C)=O)CCN(C(c2sc(C)cc2Cl)=O)CC1CC1CC1 14685,c1(C(N(C(CC)CC(=O)NCCc2ncon2)C)=O)ccc([N+](=O)[O-])[nH]1 14686,S(=O)(=O)(c1cnc(C(=O)O)c(Cl)c1)NCC1(OCC)CN(C)C1 14687,C(=O)(C(CC(C)(C)C)NC(c1cscc1C)=O)NCC(CC(=O)OC)O 14688,N1(C(CCOCCN(C(C2CC(C)(CC)C2)=O)C)=O)CCN(C)C(=O)C1C 14689,CCC(C)CCC(O)CC(=O)NCCC(C(C)C)NC(=O)C(C)(C#N)CC 14690,C(C1CCCN1C(=O)Cc1cccs1)=CC(=O)NCC(O)C1CCC1 14691,N1(c2nnc(-c3c(F)ccc(N)c3)o2)CCCC2(CC=CCO2)C1 14692,N1(C(c2cnc(C)o2)=O)CCCN(C(=O)C=CC2CCOC2)CC1C 14693,c1(C(N(CCC(C)NC(C2CC(N(C)C)C2)=O)C)=O)cc(CO)[nH]n1 14694,CC1(CNC(=O)C(O)c2ccsc2)COCCN(C(c2cc(C#N)c[nH]2)=O)C1 14695,c1(C(N2CCOCC(NC(=O)CC3CCCC4CC34)C2)=O)cnc2occc2c1 14696,C#CCC(C)(C(=O)NCC1(N(C)C)CCCC1)NC(=O)C(C)N1CC(C)C1 14697,c1(CC(=O)NCCCCCNC(C2CC2C(F)(F)F)=O)cc(O)cc(Br)c1 14698,Cc1nn(C)c(C)c1CC(N1CCC(O)(C(C)NC(c2c(Cl)nsc2Cl)=O)C1)=O 14699,C(C1CN(C(C2OCCC2C)=O)CC1C(=O)N(C)Cc1cscn1)=CC 14700,C(C(C(F)(F)F)OC)NC(c1scc(CNC(C(C)OCCCC)=O)c1)=O 14701,C1(C(=O)NC(C)CNC(C2CC2c2cncn2C)=O)C2C3CCC(C3)C12 14702,C(=O)(C1=CCC(C)(C)CC1)NC1CN(C(c2ccn(C)c2)=O)C(CO)C1 14703,C(=O)(C(C)C(O)C(C)C)NC(CNC(CN(C1CC1)CC)=O)Cc1ccccc1 14704,c1(OC)cc(C(=O)N(CCC(C(C)C)NC(C2(F)CC2)=O)C)c2c(c1)CCCC2 14705,c1(CCC(=O)NCCN(C(=O)CSCc2ncccn2)CC)ccc(Cl)cc1 14706,c1(OC)ccc(OCCN2CCCC2CNC(c2nccc(Br)n2)=O)cc1 14707,Cc1c(C(N2CC(NC(=O)C(C)(C)O)C(C3CC3)C2)=O)[nH]c2c1CCCC2 14708,C1(C)(C(=O)NC(CC)CNC(=O)Cn2cnc(=N)[nH]2)CCC(C)(C)CC1 14709,N1(C(c2cccc(F)c2)=O)CCC2(CCN(C(=O)OCc3ccccc3)CC2)C1 14710,C#CC1(C(=O)N(C(CCO)C(F)F)C)CCN(C(c2c[nH]cc2C)=O)C1 14711,CC1=C(C(=O)NCC2(C)CCCN(C(C3COC4COCC34)=O)C2)SCCO1 14712,C1(NC(C2(C)C(C(=O)OC)C2)=O)CC(NC(=O)CC2CCOC2(C)C)C(O)C1 14713,C(c1ccc(C2CC2)cc1)=CC(=O)NC1CCCCC1NC(C1(CCF)CC1)=O 14714,c1(C(=O)NC2C(OC)CN(C(C(C)OCOC)=O)C2)ccn2cncc2c1 14715,CC1=C(CC(=O)N(C)C(c2ccccc2)C2CCOCC2)c2ccccc2C1 14716,C(=O)(CCCC(C)(C)C)NC1CCC(N2CCN(C(COC)=O)CC2)C1 14717,CC1(C)CC(NC(c2cccc(C(N)=O)n2)=O)CN1C(c1cnnc(O)c1)=O 14718,C(=O)(CC(C)(C)C(=O)N(C1C2CN(C(=O)CNC(C)=O)CC12)C)OCC 14719,N1(C(C(C)NC(CC)(C)C)=O)CCOC(C)(CNC(=O)CN2CC(C)(C)C2)C1 14720,C1(NC(CC2N(C)CCC2)=O)CC2(C1)CC2NC(=O)CCC1CCCCCC1 14721,CC(C)(C)CC(O)C(=O)NCCCCCNC(C1CCCCC1C(C)(C)C)=O 14722,c1(OC)nccc(C(=O)N(C)CCNC(C2CCCN2C)=O)c1Br 14723,C(=O)(CCCC(CC)NC(C1CCCO1)=O)NC(CC=C)(C)CC=C 14724,N1(C(CNC(CC)=O)=O)CC(CNC(=O)Cc2ncccc2C)CC1(C)C 14725,Cc1cc(C(N2CCOC(C(C)NC(C3(C#N)CC3C(F)(F)F)=O)C2)=O)nn1C 14726,C(=O)(C(F)(F)C(C)(C)O)NCC(C1CCN(C(=O)C=CI)CC1)(C)C 14727,N1(C(CC(CC(C)(C)C)O)=O)CCc2sccc2C1CNC(C1CC(F)(F)C1)=O 14728,c1(C(N(C)CC2CCCN(C(C3CC(C)C3)=O)C2)=O)cc(F)cc(Cl)c1N 14729,C(C)(C)(CCC(=O)NCCN(SC(F)F)C)NC(CNC(CC(C)C)=O)=O 14730,C(c1ccc(OC2CN(C(C3CCN(C(C)=O)C3)=O)C2)cn1)=CC(=O)NCCO 14731,N1(C(CN2CC(=O)NCC2)=O)CCC(C2CC2)C1CNC(c1ccn(C(F)F)n1)=O 14732,CC(O)(CC(=O)N1CCCCC1CNC(c1cc(Br)sn1)=O)C(F)(F)F 14733,C1(CNC(c2n(C(C)C)ncc2)=O)CN(C(=O)CN2C(=O)CCC2=O)C2CC12 14734,c1(CONC(=O)CC2CCCCN2Cc2ncc(Br)cc2I)cc(F)ccc1Br 14735,S(=O)(=O)(c1ccc(C)cc1)N(CC(=O)NCC(CCCC)NC(=O)C=CSC)C 14736,c1(NC(N2CCOC(C(F)F)C2)=O)ccc(-c2cnco2)cc1 14737,N1(S(=O)(=O)c2sccc2I)CC2CN(S(=O)(=O)c3ccccc3)CC(C1)O2 14738,c1(C(=O)NC(C(C)NC(c2ccc(CO)cn2)=O)(C)C)cn2c(n1)CCCC2 14739,Cc1cc(N2CCCC(CCF)C2)ncc1S(=O)(=O)N1CCOCCC1C(C)C 14740,c1(OC)cncc(CCC(=O)NCc2ncoc2CCNC(=O)C(CC)OC)c1 14741,N1(C(c2c(N)nccn2)=O)CCC2(NC(=O)C3=CCCCC3)CC2C1 14742,C1(C(=O)OCCOC2CCCCO2)(CC)CCNC1=O 14743,C#CC1CC2CCC1N(C(=O)CC(C)NC(=O)C(=O)C(C)CC)C2 14744,CC(C)C(F)C(=O)NC(Cc1ccoc1)C(=O)NC1CC2(CCC2)C1 14745,C(=O)(C(O)CCCN(C)CCOC)NC.c12ccc(nc1)[nH]c2=O 14746,C(CC(=O)NCc1cccc(F)c1F)(C(F)F)NC(CC(C=C)C)=O 14747,C1(CCC(=O)NC23C(CN(C(C(C=C)(F)F)=O)C2)C3)CCc2ccccc2C1 14748,C1(S(N)(=O)=O)(C(=O)NC(CCCC)CNC(=O)CNC(=O)C2CC2)CCCC1 14749,N1(C(C2C(C)OCCC2)=O)CCOC2(CCN(C(=O)Cc3cnccc3Cl)C2)C1 14750,N1(C(c2c(C)nc(CNC(C3CC(C)CO3)=O)o2)=O)CCN(C)CC1C1CC1 14751,N1(C(C2C=CC(NC(C(CN(C)C)O)=O)C2)=O)CCC(O)CC1C1CC1 14752,C#CCC(C)(C(=O)N1CCC(C(=O)NC)C1)NC(c1cc(CO)c(C)o1)=O 14753,c1(C(=O)NC(CC=C)CNC(=O)CNC(c2cccs2)=O)cc([N+](=O)[O-])oc1C 14754,c1(OC)ccc2c(C)c(C(=O)NC(c3ccc(-c4ccncc4)cc3)C)[nH]c2c1 14755,O=C(C1CCCn2cnnc21)N1CC2CC2(CNC(C2(n3cnnn3)CC2)=O)C1 14756,CC(C)(C)C(CNC(c1ccc2nccn2c1)=O)C(=O)NC1(CO)CC(F)(F)C1 14757,CC(CCCC(=O)NCC1(C#N)CCC1)NC(c1ccc(F)c(O)c1)=O 14758,Cc1nccc(C(=O)NC2(C(=O)NCc3ccc(Cl)cc3)CCN(C)C2)n1 14759,C=CCCCC(=O)NC1(CNC(=O)CCN2CCCC(C(N)=O)C2)CCOC1 14760,Cc1ccc(C)c(CC(=O)NCCCCCNC(c2nccc(Cl)c2F)=O)c1 14761,N1(c2nnc(CCC)s2)CCCC(C2CC2NC(=O)CCNC(=O)CC(C)C)C1 14762,Cc1ccc(CN2CCC(O)(C(=O)NCCC(C)CO)CC2)c(F)c1F 14763,Cc1ccc(NC(=O)NNC(=O)NC(O)(Cn2cnnc2O)C(F)(F)F)cc1C 14764,C=CCC(C)(CC)C(=O)NCCC1(O)CCCN(C(c2ccc(OC)nc2)=O)C1 14765,c1(NC(C=C)C)nc(N2CCc3nocc3C2)nc2c1ncn2C(C)C 14766,c1(OCC(=O)NC2CC(C)(NC(CC(C)CF)=O)C2)cccc([N+](=O)[O-])c1 14767,CC(CNC(c1cc(CCNC(=O)CC2CC(=O)C2)on1)=O)C(C)(C)C 14768,C1(C(=O)NCC2(CC(=O)NC(C(C)C)C)CC2)COC(=O)N1C 14769,CSC1=C(C(=O)NCC2CC3(CO2)CN(C(=O)C(C)(O)CC(C)C)C3)CCCC1 14770,c1(CC(=O)NC2CC(NC(=O)CCn3ccnn3)CC2O)c(O)ncnc1O 14771,c1(C(=O)NC2CCC(NC(c3ccncn3)=O)C2)cccc2nscc12 14772,N1(C(C(C(C)C)SC)=O)CCN(C(=O)CCn2ccnc2)C(CF)C1 14773,N1(C(COC)=O)CCOC2CCN(C(c3cccc(C4(F)CC4(F)F)c3)=O)CC12 14774,C(=O)(CCC(=O)NCC1(NC(C2SCC=C2C)=O)CCCCC1)OC 14775,c1(C(C)=O)ccc(C(=O)N(C)CC2CCCCN2C(C2CC(C)N(C)C2)=O)cc1 14776,CCCCN=C(NCC(c1cc(Cl)cc(Cl)c1)O)NCC1(C)CC2CC2C1 14777,c1(C(N(CCCN(C(C(C)OC(C)(C)C)=O)C)C)=O)cc2n(c1)CCCC2 14778,c1(OCC(=O)NCC(C)(C)NC(C(=Cc2cnc[nH]2)C)=O)ccc(F)cc1 14779,n1(CC(=O)NC2CCC2NC(=O)CC2(CO)CCCCC2)nc(O)ccc1=O 14780,c1(OC)cn(C)c(C(=O)NC2CCCC2CNC(=O)CCCCC2CC2)cc1=O 14781,N1(C(c2cc(C)nnc2)=O)CCN(C(=O)C(C)CC(F)F)CC1CC(F)(F)F 14782,C1(C(=O)NCC2CCN(C(=O)C(c3cccc(C)c3)C)C2)(CC)CCCCC1 14783,N1(C(c2ccc(C)cc2N)=O)CCCC(O)(CNC(c2cnncc2C)=O)CC1 14784,C1(C(N(CC(CC)NC(C2(F)CCOC2)=O)CC)=O)C2CCC1(C)C2(C)C 14785,c1(C(=O)NCCC(C)N(C(CCCC(=O)OC)=O)C)cccc2c1CCO2 14786,CC1=C(C(=O)N(CCCNC(=O)C(F)n2ccnc2)C(C)C)C(=O)OC1(C)C 14787,C1(SC(F)F)CCCCN1CC1CCCN1 14788,C1(C(=O)NCc2cc(C(=O)NCC(COCC)O)ncc2)C2C3CCC(C3)C12 14789,N1(C(C=CCOC)=O)CC(NC(=O)CC(C)C(C)(C)CC)C2(CCOCC2)C1 14790,C1(F)(CNC(c2cc(CC)no2)=O)CCCN(C(C2CCCCCCC2)=O)CC1 14791,C(CC(C)(C)C(F)(F)F)c1ccc(NC(C)(C)CN2CC(C)(C#N)C2)cc1 14792,c1(C(C)NC(=O)NC(C2CC(=C3CCC3)C2)C)cc(Br)ncc1F 14793,CCCCCC(=O)NC1CC1CNC(=O)CN(c1ccc(Br)cn1)C 14794,O=C1CC(CCCN2CC3CC2C2CC32)C12CCC2 14795,C1(NC(CCC=C)=O)CCN(C(=O)Cc2ccc(C(N)=O)nc2)CC1C(=O)OC 14796,Cc1ccc(F)cc1C(=O)NC1C2CC3C(C2)C13C(=O)NC1CN2CCC1CC2 14797,C1(CNC(C2N(C(c3c(C(C)C)noc3)=O)C(C)C2)=O)C(C)(C)C1(F)F 14798,N1(C(Cc2onc(C)n2)=O)CCC2CN(Cc3cccc4sccc34)CC12 14799,N1(C(C2CCCO2)=O)CCC2(CCN(C(C3CC4C=CC3CC4)=O)C2)C1 14800,C1(C(=O)NCCNC(CN(CCC)C)=O)CCCC(C)(C)C1 14801,C(CCN=c1[nH]c(=N)[nH]c(=NC(C)c2csc(C3CC3)n2)[nH]1)(C(C)C)OCC 14802,c1(C(=O)NC2CN(C(Cn3c(C)csc3=O)=O)CC2C)cnc2ccc(F)cn12 14803,N1(C(c2ccc(OCC#N)cc2)C(=O)NC(CC)(C)C)CCOC2(CCCCC2)C1 14804,N1(C(c2c(CC)oc(C)c2)=O)CCC(NC(=O)C(F)C2CCOC2)C12CCCC2 14805,C1(CN(C(=O)CC(C)(C)O)C)CC(F)CN1c1nnc(CO)s1 14806,C1(C(=O)NCC(C)NC(c2ccn(CCC(F)(F)F)n2)=O)CS(=O)(=O)CCO1 14807,C1(NC(c2cc(C3(C)CC3)on2)=O)CN(C(C2CC(C)CC(C)C2)=O)CC2CC12 14808,c1(-c2c(CN(C)C(C3CNCCC3(F)F)=O)csc2)cc(F)c(F)c(F)c1 14809,C1(S(C)(=O)=O)(C(N2CCCC(CN=c3nc(CC)[nH]s3)C2)=O)CCCC1 14810,C12(C(N3CCC(N(C)C(C4CC=CCC4)=O)C3)=O)CC(C#N)(C1)C2 14811,c1(OC)nccc(C(=O)NC2COCC2C(=O)N(C(C)(C)C(=O)OC)C)n1 14812,C1(C(N2CCC(N(C(Cc3c(C)non3)=O)C)C2)=O)CCCC(=O)N1C 14813,CC1CCN(S(=O)(=O)CC(=O)N(CCCN(C)C(C2CC2C(F)(F)F)=O)C)CC1 14814,C(C)(CCN=c1[nH]c(Cl)nc(CC)c1Cl)NC(C(CC)CCOC)=O 14815,c1(NC(CC(C)OC)=O)cccc(CNC(=O)C(=O)NC2CC2C(C)C)c1 14816,Cc1cccc(CS(=O)(=O)N(C)CCOCCN(C(=O)C#CC(C)C)C)c1 14817,C(=O)(C(C)CN(C)C(C1CCC1C)=O)N1CC(CSC)C1 14818,c1(NC2CCN(C(C(C(C)(C)C)NC(C)=O)=O)CC2)nc(C)c([N+](=O)[O-])cc1Cl 14819,N1(C(C#CC(C)(C)C)=O)CC23CCCCC2(C1)CN(C(=O)CCOCCCOC)C3 14820,C1(CNC(CCC)=O)CC2(CCOCC2)CN1C(c1cc2cc(Br)sc2[nH]1)=O 14821,C(CC(=O)N(C1CN(C)C1)C)(C(F)(F)F)NC(C(CC(C)C)O)=O 14822,C1(CCOC)(NC(c2ccsc2Cl)=O)CCN(C(C2OCCC2C)=O)C1 14823,N1(C(C=C(CC)CC)=O)CCC2(CC1)CN(C(c1cnc3n1CCC3)=O)C2 14824,C1(CNC(CCOCCC)=O)CN(C(c2c(N)cc(C)cc2F)=O)CC(C)(C)O1 14825,N1(C(CCCN(CCC)CCC)=O)CC(CNC(=O)CCC(C)(C)F)CCC1C 14826,C1(C(=O)NC2CC(c3ccccc3)(NC(C=CC=CCC)=O)C2)C2CCCOC12 14827,C(=O)(C1=CC2(CCN(C(c3csc(=N)[nH]3)=O)C2)C1)N(C)CCC1CCOCC1 14828,c1(C(=O)NC2C(F)CCN(C(CC(C)(C)C#N)=O)C2)cc(Cl)ccc1[N+](=O)[O-] 14829,c1(C(=O)NCCNC(=O)C(F)CC2CCC2)c(F)ccc2nc[nH]c12 14830,c1(CC)nn(C)c(CC)c1C(=O)NC1CN(C(=O)CC2CC3CC3C2)CC1C 14831,C1(NC(CC(C=C)C)=O)CN(C(=O)CC23CCCN2CCC3)CCC1F 14832,c1(OC)ccc(C(N2CC(CNC(C3CCSC3)=O)C2)=O)c(OC)c1 14833,c1(C(=O)NC2CCC(NC(C(CC=C)(C)C)=O)C2)cccc2nccn12 14834,Cc1cc(C(=O)NC(CC2CCOCC2)C(N2C(C)CC2(C)C)=O)sc1C 14835,Cc1c(CC(N2CC(NC(c3cccnc3S)=O)CC2C)=O)sc2ccccc12 14836,c1(OC)ccc(Br)c(C(N2C3CCC2C(C(=O)NC24CC(F)(C2)C4)C3)=O)c1 14837,c1(NC)cnncc1C(=O)NCC(C)NC(c1cncn1-c1ccc(Cl)cc1)=O 14838,C1(CC(=O)NC23CC2CN(C(=O)C(C)(C2CC2)OC)C3)(OC)CCCCC1 14839,C(c1cccc(F)c1)=CC(=O)N(CCCNC(C1(C)CC2CC2C1)=O)C 14840,c1(C(=O)NC(C(C)C)CNC(=O)C=CCF)cc2cc(Cl)cnc2[nH]1 14841,CC1CCC(C)(C)N1C(c1cnc(CNC(C2CC23CCCC3)=O)nc1)=O 14842,N1(C(CNC(CCCCC)=O)=O)CC(NC(=O)Cc2ccc(C)nc2)C2CC2C1 14843,Cc1ncn(C)c1NC(C1CC(O)CN1c1ncc(OC(F)F)cn1)=O 14844,N1(C(C(CCC)C)=O)CC(NC(c2cnc(N(C)C)c(Cl)c2)=O)CC2(CCC2)C1 14845,CC1(C)CC=C(c2ccc(NC(C3(O)CC3)=O)cc2F)CC1 14846,CCC(CC)C(C)C(=O)NCC(=O)N(C1CC(O)C1(C)C)C 14847,c1(C(CC(N2CCC(C)C2C)=O)NC(C)=O)ccccc1C.c12nonc1C2 14848,c1(C(=O)NC(C)CCN(C(=O)CCC2CCCCO2)C)ccnc2ccsc12 14849,C=C(C)C1OCCC1C(=O)NCCCN(C(=O)COCCCF)C(C)C 14850,c1(C(N(CC(C)NC(C2CSCCS2)=O)CC)=O)cnn(CCN(C)C)c1C 14851,CC(C)(CCC(=O)N1CC(NC(C2CCC(CN(C)C)O2)=O)C2(CC2)C1)[N+](=O)[O-] 14852,Cc1ccnc(O)c1C(=O)N(C)CC1CCN(C(=O)CCc2cnn(C)c2)C1 14853,c1(C(=O)NCC(CNC(c2c(CC)scc2)=O)O)ccc2c(c1)C(=O)NCC2 14854,C(=O)(CC1OCCc2sccc21)N1CCC(CNC(C2OCCO2)=O)C1 14855,CC1OCCC1N=c1[nH]c(N2CCC(C)(C)C(CO)C2)nc2ccccc12 14856,C1(NC(=O)CC2CSCCS2)CCCC(CNC(c2cc(F)c[nH]2)=O)C1 14857,c1(C2N(C(c3cc(C4CC4)no3)C(=O)NCCOC)CCC2)cccc(Cl)c1 14858,c1(CC(N2CCC(CCN(C(C3(C(F)(F)F)CC3)=O)C3CC3)C2)=O)ccncc1Cl 14859,Cc1cnc(NC(C(C)C)c2cccs2)c(S(=O)(=O)NCCCCS(C)=O)c1 14860,c1(OC)ccncc1C(N1CC(O)(C(F)C(=O)NCc2nccnc2C)C1)=O 14861,c1(OC)ccc(C(N2CCN(C(=O)C(C(C)(C)C)OC)CC2CCO)=O)nc1Cl 14862,C1(C(N(CCC(N2CCC(C(C)(C)O)C2)=O)C)=O)CC2(CC2)CN1C 14863,c1(OC)cnc2ccccc2c1C(N1CC(CC(=O)O)OC(C)(C)C1)=O 14864,CC1(C(=O)NCC2(O)CN(C(c3ns[nH]c3=O)=O)C2)Cc2ccccc2NC1=O 14865,c1(OCC(C)C)ccc([N+](=O)[O-])cc1C(=O)NCC1CCCN1C(=O)CC1CC1 14866,O(C1CCCc2ccccc21)CC(=O)NC1(C#N)CCCCC1 14867,C1(C(N2CC(O)(CCNC(C3CC(SC)C3)=O)C2)=O)CCOC(=O)CC1 14868,CC#CCCC(=O)NCC1CC2CC2N1C(c1cnn(C2CCCC2)c1CC)=O 14869,CCC(C)C(O)C(=O)NCCCCCN(C(=O)C(C)SC(C)C)C 14870,CCC(C)C(=O)C(=O)N(CCCNC(=O)C(N1CCCCC1)C)C 14871,C1(NC(C2(CC=C)CC=CC2)=O)CC2CC1CN(C(=O)C(C)(C)C(C)(C)C)C2 14872,c1(C(N2CC(C)C(NC(=O)CC3(C)CC3)C2)=O)ncnc2c1c(Br)cn2C 14873,C1(NC(c2c(Cl)cc(C)s2)=O)CCOC12CCN(C(=O)C=Cc1ccsc1)CC2 14874,C1(CNC(C(C)=C2CCC2)=O)CCCCN(C(=O)CC(C)N(C)C)C1 14875,C(=O)(CCCCCC#N)N1CCC(NC(C(C)(O)c2ccccc2)=O)C(O)C1 14876,C1(C(=O)NC2C3CN(C(c4c(C)n(C)nn4)=O)C2C3)CC12CCS(=O)(=O)CC2 14877,Cc1cccc(CNC(c2c[nH]nc2CCNC(=O)Cn2cc(C)cn2)=O)n1 14878,c1(C(=O)NCCC(=O)NC(C#C)CC)c[nH]nc1[N+](=O)[O-] 14879,Cc1ccc(CN2CCC(C)C2CNC(=O)C=CC(C)(C)C)cc1C#N 14880,c1(C(N(C2CCNCC2(C)C)c2cc(CC(C)C)ncn2)=O)cc(Br)ncc1Cl 14881,c1(SC)nc(N2CCOCC2CNC(=O)Cc2cc(C)ccc2C)cc(C)n1 14882,C(N=c1[nH]c(N2CCCN3CCCC3C2)nc2c1SCC2)C1CCC(C)(C)CO1 14883,C1(NC(CCC(C)O)=O)CC2CCCC(C1)N2C(=O)Cn1cnc(=N)[nH]1 14884,c1(C(=O)NCC2(O)CN(C(CCCCSC)=O)C2)ccc2nn(C)cc2c1 14885,C1(CC(=O)NC2CN(c3cc(CC)ncn3)C(C)C2)CCC(C)(C)CC1 14886,c1(C2(C(N(C)CCNC(=O)CCC3CC3(C)C)=O)CC2)cccnc1Cl 14887,C(=O)(CCCC#Cc1ccccc1)NC1C(C)N(C(=O)C2=COCCO2)CCC1 14888,c1(C(N(CC(C)NC(c2c(CC)nn(C)c2)=O)C)=O)ccc(COC)c(F)c1 14889,CC(CC(N)=O)C(=O)NCC1=CCN(C(=O)C(C(C)(C)C)C2CCCCC2)CC1 14890,C#CC1(NC(=O)C(C)(C)CCNC(c2n[nH]c(=N)[nH]2)=O)CCC(C)CC1 14891,c1(C(C)=O)cc(C(N2CCOCC2CCNC(=O)C=C2CCC(C)C2)=O)oc1C 14892,C(=O)(C(C(C)C)C1CC1)NCC1(O)CC(C(=O)NCC(=O)N(C2CCC2)CC)C1 14893,C1(CC)CCN(C(c2ccc(I)cc2)C(=O)NCC(F)F)C1C 14894,Cc1ccc(COCC(CN2CCCC(C)C2)NC(=O)OC(C)(C)C)cn1 14895,C(=O)(C(COC)CC(C)C)N1CCC(C#C)(C(=O)NCC2CCN(C3CC3)C2)C1 14896,C1(OC)CN(C(=O)C(=O)NCCNc2ccc3c(c2)CCO3)C2(CCC2)C1 14897,Cc1ccc(C(N2CC(C(C)NC(=O)CCCn3cccn3)C2)=O)c(N)c1Br 14898,N1(C(CC(C)SC)=O)CC=C(CNC(=O)C(c2ccc(F)cc2)(C)F)CC1 14899,C1(NC(CNC(CNC(C2C(C)OCCO2)=O)=O)=O)CC2(C1)CC(O)C2 14900,N1(C(C2(SC)CCC2)=O)CCC(C(N2CC(C(C)O)C2)=O)CC1(C)C 14901,O=C(C1CCCc2cncn21)NCC1(F)CCCN(C(=O)Cc2c[nH]nc2O)C1 14902,S(=O)(=O)(c1ccc(F)c(CCNC(=O)OC(C)(C)C)c1)NC(C)CO 14903,C(=O)(CC1OCc2ncccc21)NCC1C(C)(C)CCCN1C(=O)C1=CCCC1 14904,N1(C(c2c(C)nn(C)c2)=O)C(C(N2CCOC(C(C)C)C2)=O)CCC12CC2 14905,N1(C(C(Cc2ccoc2)NC(C2=NOC(C)C2)=O)=O)CCc2nocc2C1 14906,C1(OC)CC(CNC(=O)CCc2cnoc2)(NC(c2cnsc2C)=O)C1 14907,CC1CC(CNC(=O)CCc2cc[nH]n2)CN1C(=O)Cc1cccc(Br)c1 14908,N1(C(c2cc(C)[nH]n2)=O)C2CCC1C(C)C(NC(c1cn(C)cn1)=O)C2 14909,c1(CCc2n(CCCSCC)nnn2)cccc2nn(C)cc12 14910,c1(CC(=O)N(C)CC2OCCN(C(C(C=C)(C)O)=O)C2)cc(F)c(C)cc1F 14911,Cc1c(NC(c2cc(I)cs2)c2nnnn2C2(C)CC2)cccc1Cl 14912,C1(NC(=O)NCCc2ccc(F)c(Cl)c2)CCOC2(CCS(=O)(=O)C2)C1 14913,C1(NC(c2cccc(O)c2F)=O)CN(C(c2ccoc2)=O)CCC1C(F)(F)F 14914,C(=O)(C#CC1CCC1)NC1(C)CC(NC(=O)CCC2CC2(F)F)C1 14915,C(=O)(C1=C(Cl)CCCC1)N(CC(=O)NC(c1cnnn1C)C)C(C)C 14916,N1(c2nnc(C(C(C)(C)C)O)n2CCCN2CCOCC2)CCOC2(CCC2)C1 14917,c1(C(=O)NC2CCCC(NC(C(CCC)(C)C)=O)C2)ccc2nccc(C)c2c1 14918,c1(C(=O)NCC(C)N(C(C23COCC2C3)=O)CC)cc(F)cnc1O 14919,C(C(F)CNC(=O)COC1CC(NS(=O)(=O)CC)C1)NC(COCCOCC)=O 14920,C1(C2(O)CN(C(=O)COCCOCCO)C2)(CNC(C(CC)(C)F)=O)CC1 14921,CCCCC(C(=O)N1CC=CCC1C(=O)N(C)Cc1cccc(F)c1)N(C)C 14922,c1(C(N2CC(N(C(C3C(=C)C3)=O)C)C(O)C2)=O)ccc2[nH]c(=N)sc2c1 14923,Cc1ccc(=N)[nH]c1C(N1CCCC(CCNC(c2nc(Br)c[nH]2)=O)C1)=O 14924,CC(CS(C)(=O)=O)C(=O)N1CC2(CC(NC(=O)Cn3ncn(C)c3=O)CO2)C1 14925,N1(C(c2n(CC)ncc2)=O)CCC(CCC(=O)NC(C)C(C)CC)CC1 14926,N1(C(C(C)Br)=O)CCCn2nc(C(N3CCC(O)C(F)C3)=O)cc2C1 14927,CC(CC(=O)NC1C=CCN(C(c2sccc2CN(C)C)=O)C1)CC(C)(C)C 14928,C1(NC(CN(C)C(N)=O)=O)CCC(NC(c2ccc(NC(N)=O)s2)=O)CC1 14929,C1(c2nnnn2C2(C)CC2)(NCCC(C=C)(C)C)CCOC(CC(=O)OC)C1 14930,CC1CC(CCNC(=O)C=CC2CCCN2C)CCN1C(=O)CCNC(N)=O 14931,c1(CCC)cc(C(=O)N(C2CCCN(C(C3(F)CCCC3)=O)C2)CC)c(C)o1 14932,c1(OC)cc(C(=O)N(C2CCCC(N(C(=O)C3=C(C)OCC3)C)C2)C)c(Cl)cn1 14933,c1(C(=O)OC)cc(C#N)cnc1NCC1CCCN(C(=O)CCc2cccs2)C1 14934,N1(C(CC(CC)C)=O)CCCC2C1CCN2C(c1scnc1-c1ccccc1)=O 14935,CC(C)(F)CCC(=O)N1CCC(CCCCCNC(=O)Cc2csc(=N)[nH]2)CC1 14936,Cc1ccc(C(=O)N(C)CC2(CNC(c3csc(C)c3)=O)CC2)cc1 14937,S(=O)(=O)(c1cccc(F)c1)NCCNC(c1cc(CC)oc1C)=O 14938,NC(=O)CS(=O)(=O)c1ccc(C(=O)NCCN(CCO)CCO)cc1 14939,C(=O)(CS(=O)(=O)C(C)C)NCCCN1CCN(c2c(OC)ncnc2Cl)CC1 14940,C1(CC(N)=O)CN(C(c2ccc(Cl)cc2OCC(F)(F)F)=O)CC12CCC2 14941,N1(C(CNC(CNC(C(CCSC)O)=O)=O)=O)CCCC2C(O)CC12 14942,c1(SCC(=O)N(CC(C)NC(C23CCC(CO2)C3)=O)C)ccc(N(C)C)cc1 14943,N1(C(COCC(C)(C)C)=O)CCCCC(CNC(C2(CCF)CC2)=O)C1 14944,C(C(CNC(C1CCCO1)=O)C(F)(F)F)NC(Cn1c(C)ncc1)=O 14945,N1(C(CCOCC#C)=O)CCCC1(C)CNC(c1ccc(Cl)cn1)=O 14946,C(=O)(C1=CC2CCCC12)N1C(CCNC(CC2CC(=O)OC2)=O)CSCC1 14947,C1(CNC(C(C)(F)F)=O)CN(C(c2cnc(Br)c(N)n2)=O)CC12CC2 14948,Cc1ccc([N+](=O)[O-])c(NC(C23CC2CN(C(c2cc(Cl)ccc2I)=O)C3)=O)n1 14949,c1(C(=O)NCC2CC(NC(C(C3CCOCC3)OC)=O)C2)nc(Cl)c(=O)[nH]c1N 14950,C(=O)(C1=CC2CCCC12)NCCOCCNC(c1c(C)c(O)ccc1)=O 14951,C1(C(=O)NCCOCCN(C)C)CC2(CCC2)CN1C(c1cn(C)nn1)=O 14952,Cn1ncc(NC(=O)CCC(N)=O)c1-c1cn(CC2CCCO2)nn1 14953,CN1CC2CCN(C(c3ccc(CNC(c4c[nH]ccc4=O)=O)s3)=O)C2C1 14954,c1(CCC(=O)NCCNC(CCc2c[nH]c(=N)[nH]2)=O)ccc(C2CC2)cc1 14955,c1(CN(C(C2C(CC)CCO2)=O)C)cccc(CNC(=O)CN2CC=CC2)c1 14956,C1(C(C)=O)CCC(c2nc(-c3ccc(C(F)F)cc3)nn2C2CCSC2)CC1 14957,c1(C(=O)NCC(CC)NC(C2CC(C3CCC3)C2)=O)c(F)ccc(OC)c1N 14958,c1(N2CC3(C(C(=O)NC(CCCC)CO)C3)C2)nc(C)nc2ccccc12 14959,C1(CC(=O)NCC2(CN(C(CSCC(C)C)=O)C)CC2)CC2(CCC2)CO1 14960,Cc1ccc2ncc(NC(N3CC(OCc4ccc(Cl)nc4)C3)=O)c(=O)n2c1 14961,c1(NCC2(CC)CCCCCC2)cc(=NCC2(F)C3CCCCC23)[nH]c(C)n1 14962,CCCCCC(O)C(=O)NCCC(C)(C)NC(=O)CC1(n2cncn2)CC1 14963,C#Cc1ccc(C(=O)NC2CC3(C(N4CCCC(CC)(CO)C4)=O)COC2C3)cc1 14964,C1(C)(OC)CCCN(C(=O)C(C)(C)CCCNC(C2CC(C)(C)CCO2)=O)CC1 14965,C(=O)(CCc1ccco1)C(C(C)NCCC)=O.C(CN=[N+]=[N-])NC 14966,c1(C(N2CCCCC(N(C(CCCC(C)C)=O)C)C2)=O)nccc2n[nH]cc12 14967,c1(C(=O)NCCC2CN(C(C3(C)CC(C)OCC3)=O)C2)cnc2c(ccn2C)c1 14968,C1(CNC(c2ccc(CC)c(CC)c2)=O)CC2(CCC2)CN1C(=O)CC(C)(F)F 14969,CCCC(O)CC(=O)NCC1C2CCC(C2)N1C(c1cnn(CC(F)(F)F)n1)=O 14970,c1(CC(CNC2(CCC)CNC2)C)ccccc1C(F)(F)F 14971,c1(C(=O)NCC(C)CNC(C2(C)CC(F)C2)=O)cccc2c1nc(O)n2C 14972,N1(Cc2ccc(OC)c(Br)c2)CC2CCC1CN2C(c1cocn1)=O 14973,O=[N+]([O-])c1cnn(-c2ccccc2)c1.c1(N)cnc(C2CCOCC2)nc1.C1=[SH]CC1 14974,C1(N(C(c2c(CCC)n(CC)nn2)=O)C)CCN(C(c2cc(Cl)c[nH]2)=O)CC1C 14975,C=CCCCC(=O)N1CC(O)(C2CCCN2C(=O)C=CCCC=C(C)C)C1 14976,c1(OC)ccc(Cl)c(CN2CCCCC2CNC(=O)CC2CCC2)c1 14977,Cc1nc(C)c(C(N2CC(O)(CNC(c3scnc3C3CC3)=O)C2)=O)s1 14978,N1(C(C(C(C)C)=O)=O)CCC2(CCCN2C(=O)CC2NC(=O)NC2=O)C1 14979,c1(CC)cnccc1C(=O)NCC1CN(C(c2csc(=NC)[nH]2)=O)C2CC12 14980,N1(CC)CCOCC1CC(=O)NC1CC(N(C)C(c2cccc(C(C)C)n2)=O)C1 14981,CN1CCN(C)CC(C(N2CC(C3CN(C(c4cccc(O)n4)=O)C3)C2)=O)C1 14982,C1(CSCC)CCN(C(c2ccc(C(F)(F)F)n2C)=O)CC1 14983,CC1CCCN(C(c2ccc(F)c(F)c2)=O)C1CNC(C1CC(F)(CO)C1)=O 14984,N1(C(CC2C(CNC(C=CC)=O)C2)=O)CC(C2=NOC(C)C2)C1 14985,N1(C(C2(C(C)C)CCN(C(c3cccc(OC)n3)=O)C2)=O)CCC2(CC1)N=N2 14986,C1(C(=O)NC(C)CCN(C)C)OCCC1CNC(=O)CC1CC1 14987,c1(C(=O)NC(CC)CNC(=O)CCC2CCOCC2)cc(C)nc(Cl)c1 14988,c1(C(N(CC(O)CO)C(C)C)=O)cccc(CNC(=O)CC2CC(=O)NC2=O)n1 14989,C1(C(N(CCCNC(=O)CCCN2CCCC2)C)=O)CCc2nncn2C1 14990,C(CCC(N)=O)(C(=O)NC1CCN(C(=O)COCC(C)(C)C)CC1O)NC(C)=O 14991,N1(C(=O)NC(c2c(N(C)C)cccc2F)C)CCOC(C)(CN(C)C)C1 14992,C1(NC(C2C(OCC)C2)=O)CN(C(=O)CCn2cc(Br)cn2)CC2(CC2)C1 14993,N1(C(c2ccc(C#C)nc2)=O)CC(NC(=O)C(O)CN(C)C)CC2(CC2)C1 14994,C1(C)(C(N(CC(C)O)CCNC(=O)C(=O)NCC2CC2)=O)CCN(C)C1=O 14995,c1(C(C)CNC(=O)C(C)c2ncco2)ccncc1 14996,N1(C(C(C(CC)C)O)=O)CC2CCCC1C2CNC(=O)C1=CCOCC1 14997,C(=O)(C1=CCCC(C)(C)C1)NC(c1cccc(Cl)c1)CNC(c1cc(C)ns1)=O 14998,N1(C(c2cccc(OC)n2)=O)CC(C(=O)NC(c2ccc(F)cc2)C)CC(F)C1 14999,C1(CN(C(=O)C=Cc2cc[nH]n2)C)CCCN(C(C2CCOC(=O)N2)=O)C1 15000,c1(C(=O)NC(CC)CNC(c2ccnnc2O)=O)cc(O)ccc1[N+](=O)[O-] 15001,C12(C(=O)NC3(C)C(C)CCC3)CC(CN(C(c3cccc(O)c3)=O)C1)C2 15002,c1(OC(C)C)ccc(F)c(C(=O)Nc2cncc(-c3cccc(C#N)c3)c2)c1F 15003,C(CN=c1cc(C)[nH]c(=NCC23CCC(CO)(CC2)CO3)[nH]1)=CCCC 15004,c1(C(=O)NC2(C)CCCN(C(C3CCC(O)C3)=O)C2)cncc2c1CCC2 15005,Cn1cnnc1C1C(=O)N1.C(CCCF)NC1(CC(=O)OC(C)(C)C)CC1 15006,Cc1cnc(-c2noc(C(C3(C)CC3)F)n2)nc1 15007,c1(NC(C2C(C)CCCC2)=O)ccc(CN=c2[nH]nc(C(F)F)o2)cc1F 15008,Cc1nn(C(C)(C)C)c(C)c1C(N1CC=CC(NC(C2(F)CC=CCC2)=O)C1)=O 15009,Cc1cc(F)ccc1NC(=O)C(c1cccc(C(N)=O)c1)SC(F)F.c1ccsc1 15010,C1(C(=O)NC2C(c3cn(CCCCCC)nn3)CCC2)CN(C)CC(C)O1 15011,C1(C(=O)NCC2CCN(C(c3ccnnc3O)=O)C2)CC2(C1)CC1(CCC1)C2 15012,Cc1cccc2cc(C(N3CC4(C3)CN(C(=O)C3CC3)CCO4)=O)nn12 15013,C1(CNC(CC(=O)N(C)C)=O)CN(C(=O)C(O)c2ccsc2)CC12CC2 15014,C1(C(C)C)(C(=O)N(C)Cc2cnc[nH]2)CCN(C(=O)COC(C)(C)C)C1 15015,C1(NC(C2(F)C(C)OCC2)=O)CC2(CCN(C(=O)C=Cc3ccccc3)C2)C1 15016,C1(NC(C=C(C)C(F)F)=O)CCC(N(C(=O)C(c2cnn(C)c2)C)C)CC1 15017,C(=O)(C1=NNC(C(F)(F)F)C1)N1CC(C)C(NC(=O)CCC(C)(C)F)C1 15018,c1(OC)ccc(NC(=O)C(c2cc(C)ccn2)N2CCC(F)(COC)C2)cc1 15019,C1(C)(CNC(CCOCCOCC)=O)CCN(C(c2cc3occc3[nH]2)=O)CC1 15020,C=CC1CN(C(=O)CC#N)CC1NC(C1CCCCN1C(c1ccncc1)=O)=O 15021,c1(CCC)n[nH]cc1C(=O)NC(C1CCOC1)CNC(c1cnns1)=O 15022,N1(C(Cc2n(C)c(S)nn2)=O)CC(NC(C2C3(CC3)C23CC3)=O)C2(CCC2)C1 15023,c1(C(=O)NCCCN(C(=O)C(C)C2CC2)CC)cc(C)ccc1C1CC1.N(C)(C)C 15024,C1(C(N2CCN(CCC#C)CC2)=O)CC2(CCN(C(C3CC3(F)Cl)=O)C2)C1 15025,N1(C(C(CC(=C)C)C)=O)CCC(C2CC2NC(C2(O)CCC(C)(C)CC2)=O)CC1 15026,C1(C)(C(N2CCC3C(NC(C(C)=CC)=O)C32)=O)CC(c2ccccc2)=NO1 15027,N1(c2nc(N(C)Cc3ncc(CC)s3)nc(C)c2)CCCc2ccccc2CC1 15028,C1(CC)(NC(C2CCC(=O)C(C)C2)=O)CCN(C(C2CCC(=O)N2CC)=O)CC1 15029,c1(CC)ccccc1OCCC(=O)NCC1CCN1C(=O)Cc1ccnnc1O 15030,c1(C(N2C(CNC(c3cc(CF)on3)=O)CC(OC)C2)=O)csc2cccnc12 15031,c1(C(=O)NCC(CO)NC(CS(=O)(=O)NC)=O)c[nH]ccc1=Nc1cnn(C)c1 15032,N1(C(C(CC)COC)=O)CCC2CC2(C(=O)NCC(C)(C)C#N)CC1 15033,c1(C(=O)NCCCCCNC(CCC(=C)Br)=O)cc2c[nH]nc2s1 15034,C1(CNC(=O)C=Cc2cccnc2)CC(F)(F)CN1C(c1cc(Cl)cnc1O)=O 15035,c1(C(=O)NCC2N(C(C=CC(=O)OCCCC)=O)CC2)noc2c1CCCC2 15036,Cc1nn(CC(N2CCC(CO)C(NC(=O)CCOCC(F)F)C2)=O)c(C)c1Cl 15037,N1(C2CCN(C(C(CSC)OC)=O)C2)CCN(C(=O)CC2CCOCC2)CC1 15038,c1(C(N2C(CCCNC(C3CCC(C)C3)=O)CCC2)=O)cc2c(o1)CCCC2 15039,c1(C(N(C(CNC(C(C)NS(C)(=O)=O)=O)C2CC2)C)=O)sc(F)cc1Cl 15040,S(=O)(=O)(CCC(=O)NCC(C1CCOC1)NC(=O)C(F)(F)c1cscn1)NC 15041,CC1(C)CCCC2(CN(C(C3COCCO3)=O)C2)O1 15042,C(=O)(C(C)CC(F)(F)F)NCC1N(C(c2n(CC)ncc2)=O)CC(OC)C1 15043,C(C(C)CN=c1c(C#N)c[nH]c2cccc(I)c12)c1ccc(OC)c([N+](=O)[O-])c1 15044,c1(C(=O)NC23CC(C(=O)NCC4CCC(C)CO4)(C2)C3)coc2ccccc12 15045,CN1CCCC(C(c2scc(CC(=O)NC(c3cccs3)=O)n2)=O)C1=O 15046,c1(OC)cc(N)c(C(=O)NC(C2CCCCC2)CNC(=O)COC(F)F)c(F)c1 15047,C(CO)(C(=O)NCC1C=CC(NC(C2CCC(C(N)=O)O2)=O)C1)NC(N)=O 15048,c1(CNC(=O)NC2(c3cccnc3)CCC2)ccc(CN2CCOCC2)cc1 15049,C1(CC(N2CC(C)(NC(=O)CCC(=O)N3CCOCC3)C2)=O)CCOC(C)(C)C1 15050,C(=O)(C1CCCc2nc[nH]c21)NC1(C)CN(C(=O)CC2CSC2)C1 15051,c1(C(=O)NC2C(C)CCN(C(C3CCS(=O)(=O)C3)=O)C2)cnc2cc[nH]c2c1 15052,C1(CNC(c2ccc3ncccn23)=O)CCCC(F)(F)CC1 15053,CC#CCCC(=O)NC1CN(C(c2cnc(-c3ccc(Cl)s3)s2)=O)CC1OC 15054,C1(CC)=NC(C)(C(=O)NCCCC(C)(C)NC(C2CCC(=O)N2C)=O)C(C)=N1 15055,c1(C(=O)NCC(CC(C)C)NC(c2ccc(CO)c(F)c2)=O)ccc(N)c(Cl)n1 15056,C1(C(=O)O)CN(CCC(F)(F)F)C2(CCC2)CO1 15057,C1(C(N2CCN(C(CC(C)(C)O)=O)C(C(F)F)C2)=O)CC2CCC(C1)S2(=O)=O 15058,c1(C(N2C(CNC(=O)COC(F)(F)F)CCCC2)=O)cnc2sccc2c1 15059,c1(C(=O)NC2COCCN(C(c3cnc(SC)s3)=O)C2)ccc2c(c1)SCCN2 15060,c1(C(N2CCOCC2)C(=O)NCCCNC(=O)C(F)F)ccccc1 15061,C1(C(=O)NC(CC)CNC(=O)C(F)(F)COC)Cc2cccc(F)c2O1 15062,C(N=c1[nH]cnc(Cl)c1C1CC1)C1C(C)CN(C(=O)Cc2cc(CO)on2)CC1 15063,CCCC(C)(C)C(=O)N1CC(CNC(=O)CCc2nnc(C)n2C)C(O)C1 15064,N1(C(c2nn(C)c(Cl)c2Cl)=O)CCN(C(C2CCNC2=O)=O)CC12CC2 15065,C(C)(C)(C(C)(C)CO)NC(CCC1CCCN(C(C2(CC(=O)OC)CC2)=O)C1)=O 15066,c1(CC)nc2c(C)csc2c(=NCC2CCCN2C(=O)C(C)NS(=O)(=O)CC)[nH]1 15067,N12CCCCCC1OC(CC1CC(C(=O)OC)C1)C2=O.C(C)(C)(C)OC(C)=O 15068,C1(NC(=O)C=CC2CC2)CCCCN(C(C2CCS(=O)(=O)C2)=O)C1 15069,C1(C(=O)NC2CC(CNC(CCCNC(C(C)(C)C)=O)=O)C2)C(Cl)(Cl)C12CC2 15070,N1(C(C2N(C(C(CC)NC(=O)OC(C)(C)C)=O)C(CO)C2)=O)CC(F)CC1CO 15071,CC(CS(C)(=O)=O)C(=O)NCC1(F)CCN(C(c2ccc3ncnn3n2)=O)CC1 15072,C1(NC(CSCC=C)=O)COC2(CCCN(C(c3ccc(N(C)C)cc3)=O)C2)C1 15073,C1(C(=O)NC2CCN(C(C)C)C2)CCN(C(=O)Cc2ccn(C)c2)C1(C)C 15074,S(=O)(=O)(c1c(Cl)cc(Br)cc1Cl)N1C2CN(C(c3c(F)cncc3F)=O)CC21 15075,N=c1[nH]nc(Cl)cc1C(=O)NCC1(CO)CCN(C(=O)CCc2cnc[nH]2)CC1 15076,C1(CN(C(CCCOCC)=O)C)CN(C(=O)CC2(O)CCCOC2)CCO1 15077,N1(C(C(C)=CC)=O)CCN(CCCNC(=O)C(C)C(C)O)CC1 15078,c1(C(=O)NCC(c2ccccc2)NC(C(CSC)OC)=O)ccc(N)c(Cl)c1 15079,N1(C(=O)OC(C)(C)C)CCC(C)(C)C(C(=O)NCCc2nc(C3CC3)no2)C1 15080,C(=O)(C1=C(Cl)CCOC1)N1CCC2(C(C(N(C(C(C)C)C)C3CC3)=O)C2)C1 15081,C1(C(=O)NC(CC(=O)NC)C)(NC(C2C(C(=O)OC)C2(C)C)=O)CCCC1C 15082,CC1CCC(NC(=O)CCOCC(F)F)CN1C(=O)Cc1ccc(O)c(O)c1 15083,c1(C(=O)NCC2OCCN(c3c(C(N)=O)cnc(Cl)n3)C2)cnc2nccn2c1 15084,C12(OC)CCC(C(=O)NC3(C)CN(C(=O)C(F)(F)C(F)(F)F)C3)(CC1)CC2 15085,N1(C(C2C(C)OCCC2)=O)CC2(CC2)CC1CNC(=O)C1=NNC(C(F)(F)F)C1 15086,c1(C(C(=O)NCCCSC)N(C(CF)CF)C)cncc(Br)c1C 15087,N1(C(c2ccc(C#C)o2)=O)CC2CC(NC(=O)C(C)(C)c3ccc(Cl)s3)CC1C2 15088,N1(C(CCCC(=C)C)=O)CCOC2(C1)CN(C(C1CC(=O)N(CCOC)C1)=O)C2 15089,C1(N(C)C(c2ccc(F)o2)=O)CCCN(C(=O)CC(c2cccc(F)c2)O)C1 15090,N1(C(c2c(CC)noc2)=O)CC2(CNC(c3ccn(C)n3)=O)CC(F)(C1)C2 15091,C1(CCNC(C=C(CC)C)=O)(NC(=O)COC(F)F)CCC1 15092,C1(C(N(C(C)CO)Cc2ccccc2)=O)CN(C(C2CCC=CO2)=O)CCO1 15093,N1(C(C(CC)C)=O)C2CCC1CC(F)(CNC(=O)C=CC(F)(F)F)C2 15094,N1(C(C2COCCN(C(C3CN(C(C)C)C3)=O)C2)=O)CCC12CCCOCC2 15095,C(C1=CCN(C(=O)CC2C=CCC2)CC1)NC(C1(C)CC(C#N)C1)=O 15096,N1(C(=O)NCc2ccc(NC(=O)NC)cc2)CCSC(C)CC1 15097,C1(CC=C)(C(=O)NCc2n[nH]c(C)n2)CCCN1C(=O)CCc1cn[nH]c1 15098,CC1(C)COCC(CS(=O)(=O)Sc2ccsc2)O1.C12(CC1)CNC2 15099,c1(C(C(=O)NCCOCC)N(CC(F)(F)Cl)C)cc(NC(C)=O)cn1C 15100,N1(C(CC2C(C)C(=O)CC2)=O)C2CC1CN(C(c1ccc(C(F)F)o1)=O)C2 15101,c1(C(=O)OCc2nn(C)c(Cl)c2)nc(Cl)c(=O)[nH]c1N 15102,C=C=Cn1ccccc1=O.C1(=O)CCC(C)(C)N1C(=O)CC(C)CN(C)C 15103,CS(=O)(=O)c1ccccc1-c1ccc2c(C(=O)N=c3cc(CO)[nH][nH]3)nsc2c1 15104,N1(C(CSCC)=O)CC(F)(F)CC1CCNC(=O)Cc1ccccc1OC 15105,C1(C)(C(=O)NCC(C2CC2)NC(C2(C(=O)OC)C=CCC2)=O)C(C)(C)C1(C)C 15106,N1(C(C2C(C(C)C)CCC2)=O)C2CCC1C(F)C(NC(c1cc(Cl)cs1)=O)C2 15107,c1(SC)ccccc1C(=O)NC1CC1NC(=O)C(C)(C)CO 15108,C1(NC(c2ccncn2)=O)CCN(C(C2CC(CF)C2)=O)CC1CO 15109,c1(C(N2CCCC(C(=O)OCC)C2)=O)cc2ccc(-c3cccc(F)n3)nc2[nH]1 15110,C(=O)(C(C)(C)CC(C)(C)C)NC1(CC)CN(C(c2cc(OC)c(F)c(F)c2)=O)C1 15111,C1(CNC(C(C)NC(COC)=O)=O)CC2CC2N1C(c1ccc(C(C)=O)o1)=O 15112,c1(C(=O)NCCN(CCCN(C)C)C(c2cnn(C)c2)=O)cc(Cl)ns1 15113,c1(Cn2cc(CS(CC)(=O)=O)nn2)ccccc1CNC(=O)CC12CCCC1C2 15114,Cc1cc(C(N2CC(O)(CNC(=O)CCc3nc(C(C)C)no3)C2)=O)c(O)c(C)c1 15115,C1(C(=O)Oc2ccc(CO)cn2)CCC2(CC1)CN(C(=O)OC(C)(C)C)CCO2 15116,c1(C(=O)NCC2(COC)CCCN2C(C2CC2(C)C)=O)cncc(N=[N+]=[N-])c1 15117,c1(N2CCC(C)C(F)(F)C2)nc2cc[nH]c2c(=NCC(C)(C)c2ccccc2)[nH]1 15118,C1(N(C)C)CCC(c2ccccc2)(NC(=O)NCC2(S(C)=O)CC2)CC1 15119,c1(N2CC3C(C)C3C2)nc2ccccc2nc1N(C)Cc1ccc(S(C)=O)cc1 15120,C1(NC(CNC(C)=O)=O)CCN(CCNC(=O)CNC(=O)CC(C)(C)C)CC1 15121,C#Cc1cnn(C)c1C(=O)NC1CCCC1CC(N1CCCC1CCCO)=O 15122,CCC(C(=O)N1CC(NC(=O)CCC2CCCO2)C1)N1CCCC1=O 15123,CC(O)C(C(=O)NCCCCCCC1CC1)NC(c1ccc(O)cc1)=O 15124,c1(CN(C2CC3(CN(C(C)C)C3)C2)C)cc(Cl)c2cnn(C)c2n1 15125,c1(C(N2CC(C3N(C(C4(COC)CCOC4)=O)CCC3)(O)C2)=O)cnn(C)c1C 15126,C1(CC(=O)N(CC(C(C)C)C)C)CC(NC(=O)C=CC(=O)NC2CC2)C1(C)C 15127,N1(C(C2ON=C(C)C2)=O)CCC(C(C)(C)CNC(=O)C=CC2CCCN2C)CC1 15128,C1(NC(C2(CC)CC2(F)F)=O)C2CN(C(C)=O)CC12 15129,C1(COC)(CNC(=O)C(CSC)OC)CN(C(=O)CC2(C(F)(F)F)CCC2)C1.CF 15130,CC1(C)CN(C(c2csc(S(N)(=O)=O)c2)=O)C(CNC(=O)C(C)(C)C(F)F)CO1 15131,c1(SCC(=O)NC2CC(NC(C3COCCC3(F)F)=O)C2)ccc(F)c(F)c1 15132,S(=O)(=O)(c1cccnc1N(C)CC1CCCS(=O)(=O)C1)NCCN(C(C)C)C 15133,Cc1ccc(C(=O)NCCCC2CCCCN2C(=O)C(N)=O)c2ccccc12 15134,C(=O)(C(c1ccccc1)=CC(C)(C)C)NCCN(C(C(C=C)(C)O)=O)C1CC1 15135,N1(CC)CCN(CC(N2CCCC(CNC(c3cccc(C4CC4)c3)=O)C2)=O)CC1 15136,CC(C)CC(O)C(C)C(=O)N1CC(F)(F)CC1C(=O)NC1CCC12CCCC2 15137,N1(C(C(CCC)O)=O)CC(C2CCCN(C(c3cnc4cccnc4c3)=O)C2)C1 15138,C1(NC(C2(SCC)CC2)=O)CCC(F)(CNC)C1.c12cc(c[nH]1)CC(=O)C2=O.C(C)(C)C 15139,C1(F)(CNC(c2c(C)snc2)=O)CCCN(C(c2cnnn2C2CC2)=O)C1 15140,CCCCC(C(=O)NC(C)CC(C)C(F)F)NC(c1ccc(O)cc1)=O 15141,CC1CN(C(C2CN(C(c3ccc(C#N)o3)=O)CC2(C)C)=O)CCS1=O 15142,C1(NC(c2c(CC)ccs2)=O)CCN(C(=O)CP(C)(C)=O)CC1CC 15143,c1(C(=O)NC(C)CC(C)NC(=O)C(C)(C)N2CCCC2)csc(=NC2CC2)[nH]1 15144,Cc1ccccc1Oc1ccc(C(N2CCC(N(C(=O)CC#N)C)CC2)=O)cc1 15145,c1(CC)ncc(C(=O)NCc2ocnc2C(=O)N(C)CC2(O)CCOC2)cn1 15146,CC1CN(C(=O)C=Cc2ccco2)CC(CCNC(=O)CCc2cncs2)O1 15147,c1(CC)nc(C(N2CC(NC(=O)CC(C)OC)C(C)C2)=O)c2ccccn12 15148,C1(NC(c2ccc(Cl)cn2)=O)CCCC(C(=O)NCC(Cc2ccco2)CO)C1 15149,c1(C(C(C)NC2CC(C)(C(=O)OC)C2)C)ccc(C(=O)OC(C)(C)C)cc1 15150,c1(NC(C2(F)CN(S(C3(CC=C)CC3)(=O)=O)C2)=O)cc(O)c2ccccc2n1 15151,C1(N(C(=O)CCC2CCCCC2)C)CCC(NC(C2CCNC2=O)=O)CC1 15152,Cc1ncc(CNC(=O)C(CN(C)C)NC(=O)Cc2cnnn2C)s1 15153,C(C)(C)(C(=O)NC1CN(C(c2cn(Cc3ccccc3)nn2)=O)C1)SC 15154,C1(NC(C(CCCOC)C)=O)CCCCN(C(c2cccc(N)c2F)=O)CC1 15155,Cc1cccc(C(N2CCCC(C)C2CNC(c2c[nH]ccc2=O)=O)=O)c1O 15156,c1(NC(c2scc(C(=O)Nc3ccc(I)c(Cl)n3)n2)=O)cccc2[nH]ncc12 15157,N1(C(c2cc(C)ncc2C)=O)CCCC(O)(CNC(=O)CCSCC(N)=O)CC1 15158,N1(C(Cn2c(=O)sc(C)c2C)=O)CC2ON=C(CNC(c3ccn(C)n3)=O)C2C1 15159,N1(C(c2c(C)nco2)=O)CCC2(CC1)CC2C(=O)N(C1CC1(C)C)C 15160,N1(C(c2c(C)cns2)C(=O)NCc2ccco2)CCCC(c2cccnc2)C1 15161,N1(C(C=CCC)=O)CCC(=CCNC(C2CC=CC(O)C2)=O)CC1 15162,C1(OC)CN(C(=O)C(C)=CC2CC2)CC1NC(c1ccc(F)s1)=O 15163,c1(CCCC(=O)NCCN(C)C(c2ccc(F)c(N)c2)=O)c[nH]c2ccccc12 15164,N1(C(C2(C)N(C(c3c(C)cno3)=O)CC2)=O)CC2CC(C1)c1ccccc12 15165,Cc1cc(C(=O)NC2CCN(C(C3(C)CC3)=O)CC2C)c(C)n1-c1cnn(C)c1 15166,C1(C(N(C2CCN(C(C(C)OC3CCCCCC3)=O)C2)C)=O)CCCCS1(=O)=O 15167,C12(NC(=O)CCCc3cccnc3)CC(C1)N(C(c1cc[nH]c1)=O)C2 15168,C1(CNC(CSCC=C)=O)CC2COCC2N1C(C1(CC=C)CCOCC1)=O 15169,C(C)(C(=O)NNS(=O)(=O)c1ccccc1N)OCC.C1CCCCCN1 15170,C(CCC(CO)NC(c1cc(C2CC2)no1)=O)NC(=O)CCCF 15171,c1(OC)cc(OC)[nH]c(=NCC2(C)CCN(C(=O)C=C3CCSCC3)C2)n1 15172,Cc1cccc(O)c1C(=O)NC1CC(CCC(=O)NCc2cn(C3CC3)cn2)C1 15173,N1(C(C(CC)OC2CCCC2)=O)CCCC(CC#N)C1 15174,c1(OC)cnc(Cl)[nH]c1=NC1CCC(C(N2CC3C=CC2C3)=O)CC1 15175,C1(C(=O)NC(CSC)(C)C(=O)N2CCOC(C(C)C)C2)CC2(CC(=O)C2)C1 15176,C(C(CC(C)C)C(=O)Nc1cnn(C)c1C(F)(F)F)OC 15177,C1(CNC(c2cc(CC)no2)=O)CC12CCN(C(C1(O)CC1(C)C)=O)CC2 15178,CCCCCS(=O)(=O)NC(=O)CCS(=O)(=O)c1ccccc1 15179,Cc1c(C(=O)NC2(CO)CCN(C(C3(CF)CCOCC3)=O)C2)cnn1C1CC1 15180,N(C1C(=O)Nc2cccc(Cl)c21)C(CCn1cc(-c2ccc(C)cn2)nn1)=O 15181,N1(C(c2ncn(C)n2)=O)CC2CC2C1CNC(c1cncc(O)c1)=O 15182,c1(NC(NOCCS(C)(=O)=O)=O)ccc(Cl)c(C(=O)NCc2ccco2)c1 15183,N1(C(c2c(Cl)cn(CC)n2)C(=O)NCC(F)F)C(C)C2CCCCC2C1C 15184,CC1(C(N2CC3C(NC(=O)C=CC4CCOCC4)C3C2)=O)CCCCNC1=O 15185,c1(OC)ccc(Cl)c(C)c1C(N1CCC2(NC(c3cc(CO)[nH]n3)=O)CC2C1)=O 15186,CCCC(O)CC(=O)NC(C)(C)CN(C(=O)C(c1ccc(Br)cc1)CC)C 15187,c1(C(=O)NC2CC(NC(C(CC=C)C)=O)CC2O)ncc(F)c(OC)n1 15188,c1(C(=O)NC(CC)CN(C(C2CCCSS2)=O)CC)ccc2ccccc2c1 15189,c1(C(=O)NC2CC(NC(=O)CC3COCCO3)C2)c(Br)ccc2cccnc12 15190,Cc1ccc(-c2cc(CN(CCCNC(=O)C(CO)NC(N)=O)C)on2)cc1 15191,c1(SC(C(N2CCC(N(C(C3(C=C)CCC3)=O)CC)C2)=O)C)ccc(C#N)cc1 15192,C(=O)(C=CS(C)=O)NC(C1(O)CN(C(=O)C(F)(F)c2cscn2)C1)C 15193,CC1(C)CCCc2c1n[nH]c2C(N1CC(NC(c2occc2F)=O)C1)=O 15194,c1(SCC(=O)NC2(C)CC(C(=O)NCC(=O)OCC)C2)cccc(F)c1 15195,N1(C(C(C)CC2CCC2)=O)CCC(CO)(CNC(c2c[nH]cc2C2CC2)=O)CC1 15196,C1(NC(C2(C)CCOCC2)c2n(C3(C)CC3)nnn2)CC2CCC(C1)S2 15197,Nc1cc(C(N2CCCC3(NC(C4CC=CCO4)=O)CC3C2)=O)cc(F)c1O 15198,C1(c2cccnc2)(C(=O)NCC(CNC(C(F)=CCC)=O)F)CCCC1 15199,C1(NC(C2(CC#C)CCCC2)=O)CCC(C)N(C(c2ccc(Cl)cc2N)=O)C1 15200,c1(CNC(C2CSCCN2C(c2cc(F)c[nH]2)=O)=O)ccccc1F 15201,c1(C(N2CC(COC)(CNC(=O)CC=CC(C)(C)C)C2)=O)ccc2cc[nH]c2c1 15202,C1(C(N(C2CCCN(C(C(=O)NC(C)C)=O)C2)C)=O)CC2COCC2C1 15203,C1(CC(C(=O)C=CC(=O)NC2CC2)=O)CCCCCO1.CCCCNC 15204,CC(c1cnn(C)c1)=CC(=O)NC1(CNC(C2CCNC(=O)C2)=O)CCOC1 15205,C#CCCC(O)C(=O)N1CCN(C(=O)COCCCC)CC1C(F)F 15206,c1(C(=O)NC2CC(C)(NC(C(CC)NC(N)=O)=O)C2)cnn(C)c1Br 15207,C1(C(=O)N(C2CC2)CC2CCCCO2)CCCN(C(=O)CNc2sccc2Cl)C1 15208,C1(CNC(C=C(C)Cl)=O)CC2CCC1N2C(=O)Cc1cccc(F)c1 15209,N1(C(COCCC#C)=O)CC(C2CCCCN(C(c3cc(Cl)ccc3F)=O)C2)C1 15210,N1(C(CN(C)C)=O)C(CNC(=O)C=Cc2ccccc2)CC2CC12 15211,N1(C(CC(=C)C)=O)CCN(CCNC(=O)CC(F)(F)Cl)C(c2ccccc2)C1 15212,CC1(CNC(C2(CF)COC2)=O)CCN(C(C2OCCC2c2ccccc2)=O)C1 15213,C(=O)(NNC(=O)CNC1CCC(CC(=O)OC)CC1)n1cc(COC)nn1 15214,C(CCN=c1ncc(F)c[nH]1)N(C(C1CC1CO)=O)Cc1ccccc1 15215,Cn1cccc1C(=O)NC1(CCNC(C2CCN(c3ccncc3)C2)=O)CCC1 15216,C(C(C)(C)C(=O)N1CC(CCNC(c2cc(-c3ccncc3)on2)=O)C1)OC 15217,N1(C(C)=O)CCC(F)(c2cn(C3(C(N4CCNC(=O)C4C)=O)CC3)nn2)CC1 15218,C1(C)(C(N(C)CC2(O)CCN(C(c3cncs3)=O)C2)=O)CCCCNC1=O 15219,CCCCC(CN=c1cc(C(C)(C)C)nc[nH]1)NC(=O)CC1CCOC1 15220,C=CC(C)(C)C(=O)NCC1CCN(C(=O)CC2(OCC)CC2)CC1 15221,N1(CCNC(C)=O)CCC(CC(=O)NC(CNC(=O)CC2CCCC2)CO)C1 15222,C1(C(C)C)CCOC1C(=O)NCCOCCN(C)C(c1nnn(C)n1)=O 15223,C1(NC(C(CC)(C)C)=O)CCC2CCN(C(=O)CCc3ccccc3[N+](=O)[O-])C12 15224,c1(N2CC=CC(NC(c3nn(CC)nc3C)=O)C2)ncc([N+](=O)[O-])cc1CO 15225,C1(CC(=O)N(C(c2ccncc2)C)CCO)CCN(C(c2sccc2Cl)=O)C1 15226,C(=O)(C(CNC(c1cc(C)[nH]n1)=O)C(C)(C)C)N1CCC(C)(COC)C1 15227,C1(NC(CSCCCC)=O)(CC)CCN(C(=O)C(c2cccnc2)C)CC1 15228,c1(C(N(CC(C)(C)NC(C2CN(c3nncs3)C2)=O)C)=O)c(Br)noc1C 15229,C1(CC(=O)NC(C)CCNC(=O)C(CO)NC(N)=O)Cc2ccccc2NC1=O 15230,C1(OC)CN(C)C(C)(C(=O)NC2CC3CN(C(c4ccsc4C(F)F)=O)CC23)C1 15231,CC(O)(CC(=O)N1CC(O)CC1Cn1cc(-c2cc(C(F)F)no2)nn1)C1CC1 15232,c1(SCC(N2CCN(C(C34CCCC3C4)=O)CC2)=O)nc2ccccc2[nH]1 15233,c1(C(=O)NCC2N(C(C(CC(C)C)O)=O)CC=C2)ccc(Br)c2cn[nH]c12 15234,c1(CNC(C2N(C(c3c(OC)csc3)=O)C3C(C2)C3)=O)ccc(F)nc1C 15235,N1(C(CC=C=C)=O)CCC2(CCCCN(C(c3cnn(C)c3F)=O)C2)C1 15236,c1(C(=O)NC2CCC(CNC(CC(=C)Br)=O)C2)nnc(O)cc1O 15237,c1(C(N2CCCC(N(C(c3ccns3)=O)CC)C2)=O)c(OC)cccc1O 15238,c1(C2(C(=O)OC)CCC2)cccc(C(=O)Nc2cccc(-c3ccncc3)c2)c1 15239,c1(C(=O)NC2CCCC(NC(CC=CC)=O)CC2)cnn2c1CC(F)(F)C2 15240,c1(CSC)nc(-c2cn(C)cn2)n(-c2cnnn2C)n1 15241,C1(NC(c2n(C)cnc2-c2ccccc2)=O)=CC2=NC=CC=C1S2(=O)=O 15242,C1(C(=O)NCCCN(CC(F)(F)F)C)CCC2(CC1)NC(=O)N(C)C2=O 15243,CCCC(C)(C)C(=O)NC1CC(CCNC(=O)C(F)OC)C1 15244,Cc1cc(C(=O)NC(C)CCN(C)C(c2cc(C(C)C)no2)=O)n(C2CC2)n1 15245,C(=O)(C(O)CC(C)(C)C)NC(C(C)C)(C)CNC(=O)C1=CC(C)(C)C1 15246,c12cccnc1C(=O)CCc1cn-2nn1.CC(C(=O)O)OC1CCCC1 15247,N1(C(C2C(OC)CC2)=O)Cc2occ(C(=O)NCC34CCCCC3C4)c2C1 15248,C12(O)CN(C1)C(=O)C2.c1(CCC(N2CC(CC)C2)=O)nc(O)n[nH]1 15249,C(=O)(C1=NOC2(CCC2)C1)N(CC(CO)(CO)NC(Cc1c(C)con1)=O)C 15250,N1(C(C2(OCC)CCC2)=O)CC2(CCN(Cc3ccc(C)cc3)CC2)C1 15251,Cc1cnc(C(=O)N(C)CC2CC(F)CN2C(C2CC2F)=O)c(C)c1 15252,Cc1cc(C)c(C=CC(=O)NCC2CC(NC(C3CCOC3=O)=O)C2)cc1C 15253,Nc1nc(C(N2CCC(NC(=O)CC3(CO)CC3)C(O)C2)=O)ccc1[N+](=O)[O-] 15254,C(=O)(CC(C)CC(C)C)N1CCC(C(N2CC(O)(CC)C2)=O)(CCOC)CC1 15255,C(=O)(C#CC1CCOC1)NCCC(CNC(c1c(C)n(C)nn1)=O)O 15256,c1(OC(C)C(=O)NCC2(O)CC(NC(C3OCCO3)=O)C2)ccc(F)nc1 15257,c1(C(=O)NCC2N(C(c3scc(COC)c3)=O)CC(F)C2)cccc2c1CCC2 15258,C(=O)CCCCCN=[N+]=[N-].CN(C)CCOCCOC(C)=O 15259,C12(NC(c3cc(OCC)n[nH]3)=O)CCC(CC1NC(=O)CC13CCC(CC1)C3)C2 15260,c1(C(=O)NC(C(C)(C)C)CNC(C2CCCCO2)=O)cnc2[nH]ccc2n1 15261,Cc1ccc2oc(C(=O)NC3CC4CCC(C3C)N4C(=O)CCC(F)F)cc2n1 15262,c1(OC)ccc(CN2CC(F)(C(=O)NCCC3CCCN(C)C3)C2)c(OC)c1 15263,C1(NC(=O)CN2CCCCC2)CC2CCCC(C1)N2C(c1ccnc(Cl)c1Cl)=O 15264,CC1(C)CN(C(c2cnc(Br)s2)C(=O)NC2CC(F)(F)C2)CCS1=O 15265,C(=O)(C1=NOC(C(=O)NC2CCCN(C(=O)CC(C)(C)O)C2)C1)OC(C)(C)C 15266,C1(O)(C(C(=O)OCC)(F)F)CN(N2CCC3(COC(C)C3)C2)C1 15267,N1(C(C)CCc2nccs2)C(=O)NC(c2ccsc2)C1=O 15268,C1(O)(C(C)NC(=O)CNc2cnn(C)c2)CCN(C(C2CCOC2C2CC2)=O)C1 15269,CCC(CN(C)C)CC(=O)NCC1CC1CNC(c1csnc1C)=O 15270,N1(C(C(CNC(CC2CCCN(C)C2)=O)N(C)C)=O)CC23CCC2(COC3)C1 15271,C1(NC(C(C)C)=O)CCCCC1CNC(=O)C(O)COCc1ccccc1 15272,CC1(C)CC(NC(c2c[nH]ccc2=N)=O)CN(C(C2CC(C)(C)OC2(C)C)=O)C1 15273,c1(C(=O)NCC(CO)NC(c2csc(CO)n2)=O)cc(C(F)F)ccc1Cl 15274,CCCC(CNC(=O)CC1CCC(C)(C)O1)C(=O)NCC1OCCC1(C)C 15275,c1(C(N2CCC(C(CNC(C3C4CCCC34)=O)F)CC2)=O)cccc2cncn12 15276,C1(NC(=O)CSCCC(F)(F)F)(CO)CCCN(C(c2csc3nccn23)=O)C1 15277,C1(NC(CS(CC)=O)=O)CC2CC1CN(C(c1c(C)ccc(Cl)c1F)=O)C2 15278,CC1CC(C(=O)NC2CCCC(NC(=O)C(C)(C)c3nncn3C)C2)=NO1 15279,C1(C(CC(=O)OC)NCC(c2ccncc2)OC)CCC(F)(F)CC1 15280,c1(C(N(CCCNC(C2(C)CC(C)C2)=O)C2CC2)=O)n[nH]c2cc(Cl)ccc12 15281,C(=O)(CC(C)(O)C(F)(F)F)NC(C1CCCN1C(=O)C=Cc1cccc(O)c1)C 15282,C(=O)(C(S(C)(=O)=O)C1CC1)NC(C)CC1CN(C(C2(CCO)CC2)=O)CCO1 15283,C1(C2CN(C(C3C(Cl)(Cl)C34CC4)=O)C2)(NC(C(=O)NCCOCCCC)=O)CC1 15284,Cc1noc2nc(C(=O)NC(C)CCCCNC(c3cnc(Cl)s3)=O)ccc12 15285,CC1CN(C(=O)CCC(=O)C2CC2)CCC1NC(=O)C(C1CCCCCC1)(C)C 15286,N(C(=NCc1ccc(C#N)cn1)N1CCC2=C(CCCC2)C1)C1C(C)C1 15287,C(CC(=O)NC1(c2noc(C)n2)CC1)(C(F)F)NC(c1cc(OC)no1)=O 15288,C1(CC)C(NC(c2cn(CCC(C)C)nn2)=O)CCCN1C(=O)C=C(C)C 15289,O=C1CN(C(C2CN(C(=O)CC3CCCSC3)CC2F)=O)CCN1 15290,N1(C(CN2CCN(C)CC2)=O)CC2(CC(NC(=O)C(O)CF)CO2)C1 15291,C12(NC(CC3(C#N)CC3)=O)CC(C(=O)NC34CSCC3C4)(C1)C2 15292,C1(C(N2CC(c3c(C)cccn3)C2)=O)CN(C(c2ncn(C)c2C)=O)CCN1C 15293,c1(N(CC(c2cccc(I)c2)O)C)ccc(C#N)nn1 15294,c1(C(=O)NCC2(O)COC2)ccc2nc(-c3cccc4ccncc34)cn2c1 15295,c1(C(=O)NCCC(C(C)C)NC(c2c(CC)nn[nH]2)=O)cncc(Cl)c1C 15296,c1(C(N2CCCC(C)(C(N3CC(O)(C(C)C)C3)=O)C2)=O)cnc2cc(Cl)ccn12 15297,CCC(C(=O)N1CC(O)CC1CNC(C1(c2ccccc2)CCC1)=O)C(C)C 15298,c1(OC)c(Br)ccc(CN2CC(C)CC2C(N2CC3C(CO)C3C2)=O)c1F 15299,C(=O)(C(C(C)CC(C)(C)C)N1CC2OCCN(C(C)=O)C2C1)NC 15300,N1(C(CC(CN(C)C)O)=O)CC23CCCC2(C1)CN(C(=O)Cc1csc(=N)[nH]1)C3 15301,c1(CC)c(C(N2CCOC(CC(=O)NC3CCC(O)C3)C2)=O)cnn1C 15302,c1(CC(=O)N(C(C)CNC(=O)CC2OCCOC2(C)C)C)coc2ccccc12 15303,C1(NC(c2cc(C)[nH]c2C)=O)CC2CCC1C(NC(=O)CSc1ccccc1)C2 15304,CC(CNC(=O)COCc1cnoc1-c1ccoc1)(CO)NC(c1cccs1)=O 15305,c1(CCC(=O)NC2CCCC2CNC(=O)COC2COC2)ccc(C(F)F)cc1 15306,C(C1=CCN(C(=O)C(C)n2ccnc2)CC1)NC(C(C1CC(F)(F)C1)OCC)=O 15307,c1(OC)ccc(Cl)cc1C(=O)NC1CN(C(C2CC(C(C)=O)C2(C)C)=O)CC1(C)C 15308,S(=O)(=O)(c1nc(N2CCC(O)C(C)(C)C2)ccc1Br)N1CC2N(C)CC(C2)C1 15309,C1(CNC(c2c(C)nn(C)n2)=O)CN(C(=O)Cc2ccccc2)C2CCN1C2 15310,c1(C(=O)NCCN(C(c2c(CC)cncc2)=O)CC)n[nH]c2c1CC1CC21 15311,N1(C(C(C2(O)CN(C(CSC(C)C)=O)C2)F)=O)CCCC12CCOC2=O 15312,CC1(NC(=O)CC2CCC3CC23)CCCN(C(c2ccccc2C(F)F)=O)C1 15313,c1(C(N(CC(C)NC(=O)C(C)(C)N2CCCCC2)CC)=O)c[nH]cc(C)c1=O 15314,C(=O)(CS(=O)(=O)C1CC1)N1C(C2CCN(C(c3c(OC)cccc3)=O)C2)CCCC1 15315,c1(CC)cccc(CNC(C2CCCCN2C(C2(C)CC=CC2)=O)=O)c1 15316,C1(OC)C(OC)CN(C(c2ccon2)=O)C1CNC(C1(C)CC2CC2C1)=O 15317,c1(C(N2CC(CNC(CC(CC)C3CCC3)=O)OCC2)=O)ccc(S(C)(=O)=O)s1 15318,c1(C(=O)NCC2C3N(C(c4ncn(C)n4)=O)C(CC3)C2)cn2cccc(Cl)c2n1 15319,c1(C(=O)NCCC(C)NCC2(C)CCC(=O)C2)ccnc2c1cnn2C 15320,C1(N(CC#C)C(c2cc(CCO)on2)=O)CCN(C(=O)COC2CCC2)CC1 15321,C(=O)(C1(Cl)C(=O)N(CC2CCCCC2)c2ccccc21)N1CCC(C(C)=O)CC1 15322,C1(NC(C2CCCO2)=O)CN(C(C2CC(=C3CCC3)C2)=O)CC1CO 15323,c1(C(N2C(CNC(C3ON=C(CC)C3)=O)CC2)=O)cc[nH]c2nccc1-2 15324,CON(CC1CCCc2ccccc21)C(=O)CC(C)(C)C(C)c1ccccc1 15325,C1(NC(C2C(C)CCO2)=O)CCSC12CN(C(C1CCCCC1N=[N+]=[N-])=O)C2 15326,C1(C(C)NC(C(C2CCCC2)NC(C)=O)=O)CCN(C(C2(O)CCOC2)=O)C1 15327,c1(OC)cc(O)ncc1C(=O)NCCCC1CCN(C(=O)COC(F)(F)F)CC1 15328,CC(CC(=O)NCC(C)(C1CCC1)NC(=O)C(F)C(C)(F)F)C(F)F 15329,C1(CCC)CN(C(c2cn(C)nc2C2CCC2)=O)CCN1C(=O)CCF 15330,c1(SC)ncc(C(=O)NCCC2CCN(C(c3cnn(C)c3N)=O)C2)c(O)n1 15331,Cc1cc(O)nc(C)c1C(N1CC2(CO)CC1(CNC(=O)C#CC(C)(C)C)C2)=O 15332,C1(CC)CN(C(C2CC(F)C(=O)N2)=O)CCN1C(=O)CC(=O)NC1CC1 15333,c1(CC)cc(F)ccc1C(=O)NC(C1CCCCC1)CNC(=O)C(C)(O)C(C)C 15334,C1(C(=O)NC2CC(N(C)C(c3cc[nH]c3)=O)C2)Cc2ccccc2O1 15335,N1(C(CC(COC)(C)O)=O)CC2C3CCC(C2C1)N(C(=O)CCS(C)=O)C3 15336,N1(C(C=C(C)C(F)F)=O)CCCCC1c1n[nH]cc1C(=O)N(CC(N)=O)C 15337,C1(C(N2CCC(F)(CNC(=O)C(Cl)=CCl)C2)=O)Cc2ccccc2O1 15338,S(=O)(=O)(C1CCCN(C(C2CC2(c2ccc(C#N)cc2)C(=O)O)=O)C1)NC 15339,c12ncnc3c1ncn3N2.N1(C(CN(C)CC)=O)CCC(CCO)C1 15340,N(C(=NCCC(C)(C)O)NC1CC1C1CC1C)C(C)C1CC1 15341,Cc1ccc(C(=O)NC2CCN(C3CC3)C2)cc1Cl 15342,C(=O)(CS(=O)(=O)CC)NC1(C2N(C(c3cn(CCC)nc3C)=O)CCCC2)CC1 15343,N1(C(CN(CCOC)C)=O)C(CNC(c2nc(Cl)ccc2F)=O)CC2COCC12 15344,c1(C(=O)NCC2C(NC(c3cn(CC=C)nn3)=O)C2)cc(OC)cc(Br)c1 15345,c1(N2CCC(=C)C2)nc(=Nc2cccnc2C)[nH]c2c1ncn2C 15346,C=C(C(=O)N1CCC(Oc2ccccc2)C1)C1CCN(C(=O)OC(C)(C)C)CC1 15347,N1(C(CSc2nc(C)[nH]n2)=O)CCN(C(=O)CC(O)C2CCCC2)C2CCC12 15348,N1(C(C)=O)CCCCCC1C(=O)NCc1ccc(F)cn1.N12CCCC1C2=O 15349,c1(C(=O)NC(CNC(C(C(C)C)C)=O)CO)cc(N)cc2ccccc12 15350,c1(C(=O)NCCC(C)NC(C2CC23CC(O)C3)=O)cnc(C(F)F)nc1 15351,C#CCCN=C(NCCC(C)(C)CC=C)N1CCC(C2CC2)C1 15352,C#CCCCC(=O)N1CC(NC(C2(CC)CC2(F)F)=O)C(O)C1 15353,N1(C(C2(C)CC=CC2)=O)CCCC(CCNC(c2ncsc2C2CC2)=O)CC1 15354,N1(C(c2ccc(CC)s2)=O)CCC(C(=O)NCCCN2CCCC2C)CC1 15355,c1(C(N2CC(O)(CNC(CC3(C)CC3)=O)C2)=O)ccncc1Br 15356,C(C)(CN(C(c1ccc(C2CC2)o1)=O)CCO)(C(C)C)NC(c1cn(CC)nc1)=O 15357,c1(OC)ccc(NC(c2sccc2Cl)=O)c(OC(F)F)c1 15358,Cc1cccn2c(C(N3CCCC(NC(c4cccn4C)=O)CCC3)=O)cnc12 15359,C(=O)(CC(C)(C)CNC(C1CC=CCC1)=O)NCC1CCCC(C)O1 15360,N1(C(c2c(C)cn(C(C)C)c2)=O)CCN(C)C(CNC(c2n[nH]c(C)c2C)=O)C1 15361,C1(CNC(C(C(C)C)SC)=O)CN(C(=O)CC(C)(C)C)CC1(C)C 15362,C1(C)(C(=O)NC2C(NC(C(CO)OC)=O)CCCC2)CCCCCC1 15363,c1(OC)ccc(N2CCC(C(c3ccccc3Cl)OC)CC2)nn1 15364,C1(C(=O)NCC=CCNC(c2c(C(C)C)n(C3CC3)nc2)=O)CN(C)C(=O)CCO1 15365,C1(NC(C=CCN(C(=O)CC2CCSCC2)C)=O)C=CCCCC1 15366,C#CCC(C)(C(=O)N1CC(CO)CC1CO)NC(c1ccc(F)s1)=O 15367,C1(C)(C(=O)NCC(CNC(C(CC)C2CCC(=O)N2)=O)O)CC(C)(C)C1 15368,C(CCC(C)(C)C(=O)N1CCCC1C(N1CC(O)(CCO)C1)=O)OC 15369,N1(C(c2n(C(C)C)ccn2)=O)CC2C(CNC(=O)Cc3cn[nH]c3)C2C1 15370,c1(COC)cccc(CN(C2CCN(CCC(=O)O)C2)C2CC2)c1 15371,c1(C(=O)NC(C)C(=O)NC2C3CN(C(=O)C4=CCCC4C)CC23)ccc(Cl)c(Cl)c1 15372,C1(CC)CN(C(=O)CC(C)(F)F)CCC1NC(c1cccc(C2CC2(F)F)c1)=O 15373,c1(C(=O)NC2C(C)CN(C(=O)CSc3nc[nH]n3)C2)nc(Cl)ccc1F 15374,c1(C(=O)NC2(C)CN(C(c3c(C)ccc(OC)c3)=O)C2)cccc2nc(O)oc12 15375,c1(C(=O)NC2CCN(C(c3c(CC)nccn3)=O)C2)c(Br)sc(C)c1C 15376,n1(CC)ccc(C(=O)NCC2(C(N3CC(CO)CC3C)=O)CC(C)(C)C2)c1C 15377,c1(N2CC(NC(C3CC4(CCC4)CO3)=O)CC(C)(C)C2)nc2cccc(F)c2s1 15378,C1(CNC(C(CNC(c2ccnc(O)c2)=O)OC)=O)CC2(CC2)C(=O)O1 15379,Cc1cc(C(C)(C)C(=O)NCC2(C)CCN(C(C3CCO3)=O)C2)ccc1F 15380,N1(C(C2(C)CC=C(C)CC2)=O)CC2CC1CCC2NC(=O)C(C)C1CCCC1 15381,Cc1ccc(C(=O)NCC2CC2NC(C23CC(F)(C2)C3)=O)cc1C#N 15382,n1(C(CC)C)nnnc1C(C(C)(C)OC(C)C)NCCCCCO 15383,C1(C(=O)NCc2cc(OC)no2)CCC2(CN(Cc3ccc(C#N)cc3Cl)C2)O1 15384,N1(C(C)=O)CCN(C(=O)NCC2COCOC2)C(C)C1 15385,N1(C(C=C(CCC)C)=O)CCCC2CN(C(=O)CCCOCCOCC)CCC12 15386,c1(CNC(C(=Cc2ccco2)C)=O)nnn(C)c1C(N1CCC(C)(CO)C1)=O 15387,C=CCC(C)(CNC(C1CCCC1CNC(c1coc(C(C)OC)n1)=O)=O)CO 15388,N1(C(C)C(=O)Nc2ccsc2)CCN(C(=O)CCCCc2cnn[nH]2)CC1 15389,C1(NC(C2CS(=O)(=O)C2)=O)C2CC3CN(C(=O)COc4ccc(O)cc4)C1C3C2 15390,CC1(C(N2CCC(NC(c3cccn4ccnc34)=O)C2)=O)CCCC(F)(F)C1 15391,C12(NC(=O)CC3CCCC3O)CCC(CN(C(=O)COc3cccnc3)C1)C2 15392,C12(NC(C(C)OC3CCCC3)=O)CC(C1)N(C(C1CCCCS1)=O)C2 15393,c1(C(=O)Nc2ccnc(C(C)(C)C)n2)cn(CCO)c(=O)nc1O 15394,C1(C)(CC)CCN(CC2CC3C=CC2CC3)CC1 15395,C1(C#N)(C(=O)NC(CC(C)NC(C(C)OC)=O)C)CC1(C)C 15396,C#CCC(C)(CC)C(=O)NC(C1CN(C(C2(C)CNC(=O)C2)=O)C1)C 15397,N1(C(c2cnc(C)s2)=O)CCC(C)C(NC(C2CC(n3cnnc3)C2)=O)C1 15398,N1(C(C(F)=C(C)C)=O)CCC(C)C1C(=O)NCC(F)Cl 15399,C(C(=O)NC1CC(C)(NC(c2ccon2)=O)C1)(C(C)C)n1ncc(C)c1 15400,C1(C(=O)NCCOCCOC)CCOC1NC(=O)CCN(C(C)=O)C1CC1 15401,O=C(CC(CNC(C1CCC2CC12)=O)C1CCC1)NCC1(Cl)CC1(F)F 15402,C1(CNC(=O)COCC2CCOC2)CC(F)(F)CN1C(=O)CC12COCC(C1)C2 15403,c1(CC(=O)N(CCNC(=O)C(C2CCC(=O)N2)C)CC)cn2cccc(C)c2n1 15404,C(=O)(C(C(C)C)NC(=O)C(C)C)NCCN(C(C(C)OCC)=O)CC 15405,c1(OC)ccnc(NCC(=O)N(CC(O)CNC(c2ccnc(CO)c2)=O)C)n1 15406,Nc1c(C(=O)NCC(O)CNC(C2(Cc3ccccc3)CC2)=O)cccc1Cl 15407,Cc1cncc(C(=O)NCCC(C)CCNC(c2coc(CC3CC3)n2)=O)n1 15408,c1(CNC(CC2(N(C(C(C3CC3)SC)=O)C)CC2)=O)ccc(Cl)o1 15409,Cn1nc(C(=O)NC2CCOCC2C(=O)NCCc2ncnn2C)cc1F 15410,N1(C(C)=O)CCOC2(CCN(C(=O)C(c3cccc(Br)c3)O)C2)C1 15411,c1(CC)nc(C(=O)NCC(C2CCC2)NC(C2(C(F)F)CC2)=O)co1 15412,N1(C(CCOC(N(C)C)=O)=O)CCn2c(cnc2C2CCC2)C1 15413,C(CC(=C)C)(C(=O)N1CCCC2(C1)N=N2)NC(COCCC=C)=O 15414,c1(CC(N2CC(CCn3cc(CC(C)(C)C)nn3)C2)=O)c[nH]ccc1=O 15415,c1(C2C(C(=O)NC3(CCNC(c4n[nH]cc4Br)=O)CC3)CC2)ccccc1 15416,c1(CC2N(C(c3c(-c4c(C)csc4)cncn3)=O)CCC2)ccc2cc[nH]c2n1 15417,CC(C)(C)C(CCO)NC(C1(CCNC(=O)C2=COCCC2)CC1)=O 15418,Cc1ccc(CCCCC(=O)NCCCC(C)NC(C2COCCN2C)=O)cc1 15419,C1(CNC(CCCOCC)=O)CC2CCC1N(C(C1(C)CCCS1(=O)=O)=O)C2 15420,C1(NC(c2c(C)ocn2)=O)CN(C(c2cc(Cl)cn2C)=O)CC1C 15421,c1(C(=O)NC2CN(C(C3N(C)CCOC3)=O)CC2F)cccc2nn[nH]c12 15422,C(=O)(CCO)N(CCC)CCSC.C1(CC(C)C)(OCCOCCN(C)C)CCC1 15423,c1(OC)cccc(OC)c1CC(=O)NC1CCSC1C 15424,c1(C(N(C2CC(NC(CCCCCC)=O)C2)C)=O)cn(CC)c2ccccc12 15425,C1(CC(=O)NC2CCN(C(CCCC)=O)C2CC)NC(=O)CN(C)C1=O 15426,CC(C)CC(CNC(c1cnn2ccccc12)=O)C(=O)NC1COCCC1(F)F 15427,c1(C(C)NC(C2(c3ccno3)CC2)=O)ccc2c(c1)CN(C(=O)C1=CCSC1)C2 15428,C12(C(=O)N(C3CC4C(NC(Cc5n[nH]c(=N)s5)=O)C4C3)C3CC3)CC=CC(C1)OC2 15429,N1(C(c2nc(CC)oc2C)=O)CCC(C)(C)C(NC(c2cc(C)nc(O)n2)=O)C1 15430,C1(NC(c2n[nH]cc2I)=O)C2CN(C(c3cccc(O)c3)=O)CC12 15431,c1(C(=O)NC(CC)CNC(C2CCCC2(C)C)=O)cccc2c[nH]nc12 15432,c1(C(=O)NCC=CC(=O)NC(CN(CCCC)C)C)cccc(C)c1N 15433,N1(C(C(C)C2CCC2)=O)CC(NC(=O)CC2(O)CCCC2)CC(C)(C)C1 15434,Cc1cccnc1CNC(=O)C(O)C(C)C 15435,N1(C(CSCC)=O)CCC(CNC(C2CCC23CCC3)=O)C12CCC2 15436,C1(CC)(CC)SCCNC1C(=O)NCc1ccc(N2CCCCC2C)cc1C 15437,Cc1nc(C(N2CCC(C3CCCCN3C(c3cn[nH]c3)=O)C2)=O)c(C)s1 15438,C12(C(=O)NCC3C(C)(C)C(NC(c4cc(Cl)no4)=O)C3)CC=CC(C1)OC2 15439,O=C1CC(CC(=O)NCC2(NC(C3CC3OCc3ccccc3)=O)CCC2)CN1 15440,CCCCC(CN(C)C(c1cc(CNC(C2(C#N)CC2(C)C)=O)ccn1)=O)CC 15441,Cc1cc2c(cc1C)OC(C(=O)NC1CCCC1NC(=O)C(N)=O)C2 15442,n1(CC(=O)NC2CCCN(C(=O)C(=O)NC3CC3)C2)nc2ccccn2c1=O 15443,c1(CC(CC)C)nc(C2CCC2(F)F)n(-c2cccc(Br)c2)n1 15444,Cc1cc(C(N2CCCC2Cn2cc(-n3cnnc3)nn2)=O)c(-n2cccc2)s1 15445,C1(NC(C(CC)(C)C)=O)CN(C(c2ncsc2Br)=O)CCC1F 15446,c1(C(=O)NC2(CC)CCOC2)nc(C)ccc1F 15447,CC1(C)CN(CC(=O)NC2COCC2CNC(=O)C(F)CC2CC2)C1.C(C)(C)(C)O 15448,CS(=O)c1ccccc1CC(N1CCCN(C(=O)Cc2ccsc2)CC1)=O 15449,C(=O)(CCCC(=O)NC(C(N1CCOCC(CO)C1)=O)C1CCC1)OC 15450,C1(C(=O)NC2C(NC(c3occ(C)c3)=O)COC2)CC2CCCC(C1)C2 15451,N1(C(=O)C(Cl)(Cl)Cl)CCC2(CC1)CN(S(=O)(=O)Cc1ccccc1Br)C2 15452,C1(F)(CNC(CC2N(CC)CCOC2)=O)CCN(C(=O)CN(C)S(N)(=O)=O)CC1 15453,c1(C(=O)NCC(C(C)C)NC(=O)C(c2ccc(Cl)s2)=O)ccnc(O)c1 15454,C(=O)(C(CC)CCOC)NC(C(CO)NC(C(C=C)(C)C)=O)C 15455,Cc1ccc(C(=O)NC2CN(C(C3C4CCC(F)(F)C34)=O)C(C)(C)C2)c(N)c1F 15456,c1(Cc2cccc(C(=O)NC(C)CCNC(=O)CO)c2)ccc2[nH]ccc2n1 15457,C(=O)(C1CCC(=O)c2cccn21)NC1(CNC(CC(C)P(C)(C)=O)=O)CCCC1 15458,c1(C(C)C(=O)N(c2cccc(Br)n2)CC2CCCO2)ccc(Cl)nc1 15459,c1(OC)ccc(C(=O)NC2CC(NC(=O)C(F)C(C)C)C(O)C2)cc1Cl 15460,N1(C(c2cn(CCC=C)nn2)=O)CC(NC(=O)C=Cc2cc[nH]n2)C(CCC)C1 15461,c1(OCC(C)C)ccccc1C(=O)N(C)CC1(NC(C2CCOCC2)=O)CC1 15462,C1(CNC(C2C(C(N)=O)C2)=O)CCC2(CCC2)CN1C(C1(C(F)(F)F)CC1)=O 15463,c1(C(=O)NC(C2CN(C(=O)C(C)(F)C(F)(F)F)CCO2)C)cc2n(c1)CCCC2 15464,N1(C(CP(C)(=O)OC)=O)CCC2CCN(C(=O)OC(C)(C)C)C2C1 15465,N1(C(C(C)Cc2ccc(Cl)cc2)=O)CCN(C(=O)Cc2ccno2)CC12CC2 15466,C1(O)(CCC)CN(C(C2(CNC(=O)C(C)CC3CCCC3)CCC2)=O)C1 15467,c1(C(=O)NCC(C2(O)CN(C(C=CSC)=O)C2)(C)C)ccnc(O)c1 15468,C1(C(=O)NC(CC)CN(C(C2CC2(C)C)=O)CC)CCc2nc(C)ncc2C1 15469,Cc1nnc(NC2CC(F)(CNC(=O)Cn3ccc(O)nc3=O)C2)nc1C 15470,c1(SC)ccc(O)c(C(=O)NCC2(O)CCCN(C(C3CC3C)=O)C2)c1 15471,C(CCN=C(NCC1CCSC1(C)C)N1CCN(CC2CCCO2)CC1)OC 15472,N1(C(c2ccc(CC)cc2)C(=O)NCCCOC)CCC(F)(F)C(C)C1 15473,CN=c1[nH]cc(C(N2CC(OCCNC(C3CC(C(F)(F)F)C3)=O)C2)=O)o1 15474,CCCCCCCCCC(C)CC(c1nnnn1C(C)C)NCCC1(C)COC1 15475,CN1CCC(O)(CC(N2CC(C)(NC(c3ccc(Cl)o3)=O)C2)=O)CC1 15476,Cc1cc(C(F)F)n2nc(C(N3CC4CC(C3)C4O)=O)cc2n1 15477,c1(-n2c(C3C(=C)CC3)nc(CC3CCC3)n2)ccccc1S(C)(=O)=O 15478,CCCC(C(=O)NC(CN(C(c1ccn2cccc2c1)=O)CC)CC)C(C)C 15479,c1(C(=O)OC)cc(CN(C)C(C2CCN(c3cnn(C)c3)C2=O)=O)oc1C 15480,CC1CN(CC(=O)N(C)CCC2CCCCC2)CCN1C(C1CCCCN1C)=O 15481,Cc1cnc(C)c(C(=O)NCC2CCCN2C(=O)C(C2CCCCCC2)C)c1 15482,c1(C(=O)NCCn2cc(C(N(CC(C)O)CC)=O)nn2)cc(C)n(C)c1 15483,C(=O)(C(CN=[N+]=[N-])NC(=O)C(O)C1CCC1)N(C)Cc1ccccc1 15484,C(CCOCCO)(C(=O)NCC1(Cl)CC1(F)F)NC(C(N1CCNC1=O)C)=O 15485,N1(C(COCC(=C)C)=O)CC(C2(NC(c3ccc(-c4cscn4)cc3)=O)CC2)C1 15486,N1(C(C=CCOC)=O)CCC(C(C)NC(c2cccc(-n3cnnn3)c2)=O)CC1 15487,Cc1c(F)ccc(C(=O)NCC2CCN(C(C3(C)CC3(F)F)=O)CC2O)c1F 15488,C(=O)(C(O)CC(F)(F)F)N1C(C(C)NC(c2cc3n(c2)CCC3)=O)CCCC1 15489,c1(C(=O)NCC2(COC)CN(C(=O)C(O)C(F)(F)F)C2)ccc2oc(C)nc2c1 15490,N1(C(C2C(NC(c3cn(C(C)(C)C)nc3)=O)CCC2)=O)CCC(O)C(F)C1 15491,c1(C(=O)NC2CN(C(Cc3ccc(C)c(C)c3)=O)C(C)C2)cc(O)cc(C#N)c1 15492,C#CC12CCC(C(N3C4CCCC3CN(C(=O)C(C)OCC)C4)=O)(CC1)CC2 15493,c1(OC)ccc(C)cc1C(=O)N(CCCNC(c1nnn2c1CCC2)=O)C 15494,C1(NC(CCOc2c(CC)cccc2)=O)CC(F)CN(C(=O)C(F)C2CCC2)C1 15495,S(=O)(=O)(c1cc(NC(C2CCNC(=O)C2)=O)ccc1O)NC 15496,c1(CC)sc(C(=O)NCC#CCNC(=O)Cc2ccc(Cl)cn2)cc1C 15497,N1(C(CCCC(=O)OCC)=O)CC2CC3CC2C1C3NC(c1coc(C)c1)=O 15498,c1(C(N(CCCCNC(C2(Cl)CC2(C)C)=O)C)=O)ccn2c1CCCC2 15499,C(CC(C)(C)NC(c1cc(CNC(=O)C(C2CCC2)OC)cs1)=O)OC 15500,c1(N2CC3N(C(C4N(N=O)CCC4)=O)CC(C3)C2)ncnc2c1ncn2C1CC1 15501,Cn1nc(C(N2CC=CC(NC(C3CN4CCC3CC4)=O)C2)=O)c2c1CCOC2 15502,c1(C(=O)NC(C2CCN(C(C3(COC)COC3)=O)CC2)C)ccccc1CC#N 15503,C1(CCNC(CCC2CCC(C)O2)=O)(Nc2nnnn2C)CCOCC1 15504,N1(C(CCC)=O)CCN(C(=O)C(c2cnn(C)c2)C)C(c2cccc(F)c2)C1 15505,C(N=c1[nH]c(=NCCn2cccn2)[nH]c2c1CCC2)c1ccc(OC)c(C)n1 15506,c1(C(N2C(C(=O)O)(CC)CC(OC)C2)=O)cc2scc(Cl)c2[nH]1 15507,N1(C(C=C)=O)CC2(CC2)CC1CNC(c1cc(COC)ccc1F)=O 15508,CC(CNC(=O)CC(C)(C)O)C(F)C(=O)N(C)Cc1cccnc1O 15509,C1(C(=O)NCC(CCNC(c2ccc(CO)o2)=O)O)CN2CCCN1CC2 15510,C1(C(=O)NCC(C(C)O)(C)C)CC2CC1CC2NC(=O)C=C1CCCCC1 15511,c1(C(=O)NCC(CN(C(=O)Cn2ncn(C)c2=O)C)O)ccccc1C1(C)CC1 15512,N1(Cc2ccc(N(C)C)nc2)CCOc2ccc(C(N3CCOCC3)=O)cc21 15513,c1(C(=O)NC(CC)CNC(=O)CC2(O)CCCC2)ccc(Cl)cc1O 15514,C12(C(N3CCN(Cc4cncc(OC)c4)CC3)=O)C3C4C1C1C2C3C41C 15515,Cc1oc(C)c(C(=O)NCc2cc[nH]c2C(=O)NCCOCC2CC2)c1C 15516,C(=O)(C1CCc2cccc(Cl)c21)N1CCC(NC(c2ccccc2F)=O)C(F)C1 15517,C1(CC)(COC(=O)CCCONC(C2(C)CC3CC3C2)=O)CCCCO1 15518,N1(C(C2CN(c3ncc(OC)cn3)CC(F)C2)=O)CC2COCC(C1)C(=O)N2 15519,C1(C)(C(=O)NCCCNC(CC(C)Cc2cccc(F)c2)=O)CCC(=O)NC1 15520,N1(C(Cc2cc(C)on2)=O)CC=CC(NC(=O)C(C)(C)CN2CCN(C)CC2)C1 15521,C1(NC(=O)CC2C=CCC2)CC(F)(CNC(c2cc(C(F)(F)F)cs2)=O)C1 15522,C(=O)(C1=CCC2(COC2)OC1)NC(CC)CN(C)C(c1nc(Cl)cs1)=O 15523,C(=O)(CCCC(=O)NC1CN(C(=O)C(O)Cc2cccc(Cl)c2)CC1O)NCC 15524,CC(C)(C(=O)NC1CCC2CCN(C(=O)CC3(CO)CC3)C1C2)S(=O)(=O)C1CC1 15525,C(c1ccccc1Cl)=CC(=O)NCCC1CCCN(C(C(C)(C)OC(C)=O)=O)C1 15526,c1(C(=O)NCC2(O)CN(C(CC3CCCC(OC)C3)=O)C2)ccc2nsnc2c1 15527,CC1(C)CCC(C)(NC(=O)CC(CNC(c2cccnc2O)=O)C2CCC2)C1 15528,C1(NC(=O)NC(CC=C(C)C)Cc2ccccc2)CC2CCC(C1)N2C 15529,CC1CCC=C1C(=O)NCC=CCC(=O)NOC1CCCC1 15530,C(=O)(CCC(=O)N(C)C(C)C)NC(C)CN(C(=O)CCCn1ccnn1)C 15531,N1(C(c2ccc(C#C)cn2)=O)CCC2(CC(C(N3CCC4(CC3)CC4)=O)C2)C1 15532,C(c1ccncn1)=CC(=O)NCc1cc(C(=O)NC(C)CO)on1 15533,C(C(=O)NC1CCN(C(C2(F)CC=CC2)=O)C1)(C(C)C)OC 15534,c1(-c2ccc(CNC(C)(C)C(F)(F)F)cc2)ccc2oc(O)nc2c1 15535,C(=O)(C(C)(O)C(C)(O)C(=O)OC)NC1(c2ccc(CC)cc2)CCCC1 15536,c1(C(=O)NCC2CN(C(CCC)=O)C3C(O2)COC3)cc2cccnc2cc1F 15537,Cc1ccc(C(=O)NC2(C(=O)NC3(C)CCSCC3)CCSC2)nc1O 15538,n1(CC)cnc(C(=O)NC2CCCC2NC(=O)C(n2ccnc2C)C)n1 15539,C#Cc1cc(C(N2CCC(C3(NC(c4ncn(C)n4)=O)CC3)C2)=O)ccc1Cl 15540,C(CCN(C(=O)C(C)n1ccnc1)C)(C(C)(C)C)NC(CCOC(C)C)=O 15541,C(=O)(C(F)(F)CNC(C1CC(CNC(=O)CCN(C)CCO)C1)=O)OC 15542,N1(C(C2(C(C)NC(c3ccc(O)nn3)=O)CC2)=O)CCCN(C)CC1 15543,c1(COC)cc(CNC(c2ccoc2CNC(C2(C(C)C)CC2)=O)=O)no1 15544,c1(C(=O)NC2C(CNC(=O)CSC(F)(F)F)CCCC2)ccc2nccn2n1 15545,CC1(CNC(=O)CCC2CCCC2)CCCN(C(=O)Cc2ccnc(O)c2)C1 15546,C12C(CC1O)NC(=O)C2.C(=O)(C(C)(C)n1ccnn1)NC(c1cn[nH]c1)C 15547,N1(CC(CNC(c2ccccn2)=O)O)CCCC(c2ccc(Cl)nc2)C1 15548,CC1(O)CCCN(C(C2(NC(=O)CSc3cn[nH]c3)CCOCC2)=O)C1 15549,C#Cc1ccc(C(=O)NCC(=O)NC(CO)(C(F)(F)F)c2ccc[nH]2)cc1Br 15550,c1(NC2CC(C(=O)OC)CN(C(=O)NCCO)C2)cc(Br)c(OC)cc1C 15551,c1(-c2cccc(-c3c(C)cccc3)c2)ccncc1S(=O)(=O)NC(CO)C(C)C 15552,N1(C(C(C=CCCC)O)=O)CCN(CCCNC(=O)C(C#N)CC)CC1 15553,c1(C(=O)NCCCC(=O)NCCO)ccc(CNC(C2C3COCC23)=O)cn1 15554,C1(NC(c2nccc(CO)n2)(c2nnnn2CCCF)C)CCC2(CCC2)CC1 15555,CC1(C)CCN(C(=O)C2=CCCSC2)C1CC(N1CCOCC1)=O 15556,C12(CNC(=O)NC(c3ccc(OC)cc3)C(CC)O)COC(CF)(C1)C2 15557,C1(NC(C2(OCC)CCCC2)=O)CN(C(c2cnn(CCF)c2)=O)C2CC12 15558,CCCC(C(O)C(=O)N1CCCC(C(C)(C)C)C1)NC(C1CCOC1C1CC1)=O 15559,N1(C(C2CC(NC(=O)Cn3ccnn3)C23CCC3)=O)CCC(F)(F)C(F)C1 15560,c1(CC(=O)NC2(C)CN(C(C34CCCCC3C4)=O)C2)cc2ccccc2o1 15561,O=C(C1=CCCOC1)NCCC1CC(NC(n2ccc(NC3CC34CCC4)c2)=O)C1 15562,CCC(C)CC(CO)NC(=O)CSCCNC(c1ccncc1CC)=O 15563,C(=O)(C(CC1CCCO1)C(F)(F)F)CCSCC(=O)Nc1c(C)nn(C)c1C 15564,CC(N)(C(=O)N(CC(c1cccnc1)O)CCO)C(F)(F)F 15565,Cc1cc(C(N2CC(NC(C3CC4(CNC(=O)N4)C3)=O)C(C)C2)=O)c(C)cc1Cl 15566,c1(C(=O)NC2C(CNC(C(CCC)F)=O)CCCC2)c(C)cccc1C 15567,N1(C(c2cn(CC(C)=O)nc2)=O)CC2CN(C(c3ccnc(C)n3)=O)CC12 15568,CC(C)C(C#N)C(=O)NC1(C(=O)NCCC2CC=CC2)CSC1 15569,C1(NC(C2CCN(CCC#C)CC2)=O)CC2CCC(C1)N2C(c1n[nH]cc1F)=O 15570,c1(C(=O)NCCCCNC(CSCCOC)=O)ccc(F)c(Cl)c1 15571,N1(C(CSCC(N)=O)=O)CCC2C(C1)CN2C(=O)C(=Cc1c[nH]cn1)F 15572,Cn1cc(C(c2nnnn2C(C)(C)C)Nc2cccc(CO)c2)c(OC(F)F)n1 15573,Cc1cnc(C(=O)NCC2CN(Cc3ccc(C(F)F)cc3)CCCO2)cc1C 15574,C1(C(=O)NCc2cccc(C)n2)(COC)C=CCN1C(c1sccc1CO)=O 15575,c1(N2CCC(CCNC(=O)C(c3ccc(F)cc3)F)C2)ncnc(O)c1Br 15576,C12(C(=O)NCCOCCOCCNC(c3c(C)noc3C)=O)CCCC(F)(C1)C2 15577,CC1OC(=O)NC1C(=O)NCC(C)(C)CCNC(=O)Cn1ccnn1 15578,C=CC(C)C(C)C(=O)N(CC(C)(C)CNC(=O)CC1(C(=O)OC)CCCC1)C 15579,C=C(F)C1(CC(=O)NC2CCCC(NC(C3(CO)CCCO3)=O)C2)CCC1 15580,N1(C(C2CCCC(C)C2)=O)CC2(CNC(c3coc(N(C)C)n3)=O)CCC1CC2 15581,C1(CC)CN(C(c2cc(-c3ccco3)on2)=O)CCO1 15582,c1(OC)ccc(CCC(=O)NC2(CNC(=O)COc3ccsn3)CCC2)cc1 15583,O(N1C(=O)c2ccccc2C1=O)CC(=O)N(C1CCOC(C)C1)CC 15584,N1(C(C(C2CC2)OC)=O)CC(F)(F)CC1C(=O)NC(C)CN1CCCCC1 15585,c1(C(=O)NC(CC(C)NC(CCOC)=O)C)ccc(C(C)=O)c(F)c1 15586,C#Cc1cncc(NC(C2C(CC)CCN2C(=O)C(C)C=C=C)=O)c1 15587,C1(CNC(CCSCC)=O)CCC2(CN(C(c3cc(N)c(N)cc3F)=O)C2)O1 15588,S(=O)(=O)(c1ccc(C(F)(F)F)c(C#N)c1)N(C1(C)CCOC1)C 15589,c1(NC(C2C(NC(C3(COCC)CC3)=O)C2)=O)c(O)cccc1C#N 15590,C1(C)(C(=O)NCC(C)N(C(c2c[nH]nc2C2CC2)=O)CC)CCC(C)C1 15591,C1(CC(=O)NCC23CC(NC(C(c4cccs4)SC)=O)(C2)C3)CC(O)C12CCC2 15592,c1(C(=O)NC2CC(CNC(C(C3CCOC3)OCC)=O)C2)scc2c1OCCO2 15593,C1(C(N(C)CC2COCCO2)=O)CN(C(=O)CN2CCC(F)CC2)CCN1C 15594,c1(C(=O)NCC(CC)(C)NC(=O)C=Cc2cocn2)noc2c1CCCC2 15595,N1(C(C2(CC(C)C)COC2)=O)CCCC(C2CC2NC(=O)Cc2nncn2C)C1 15596,CCC(C)(C)C(O)C(=O)NCC1CC(C)CN(C(=O)COCCN(C)C)C1 15597,c1(C(=O)NC23C(NC(C4(C(C)=O)CC4)=O)CC(CC2)C3)ccc2nc(C)sc2c1 15598,c12ccc(cc1)CN(C)C(=O)C2.C1(NC(C2(OCC)CC2)=O)CNC(=O)N1 15599,N1(C(c2n(CC)ncn2)=O)CCCC(N(C)C(c2cc(=O)cc(Cl)[nH]2)=O)CC1 15600,C1(C(=O)NC2C(C)CCC2C)CC2(CC(NC(=O)Cc3cn[nH]c3)C2)C1 15601,CCCC(C)(C)NC(=O)NC(C(=O)N(C)C)c1ccco1 15602,C#CCCCC(=O)NCC1C=CC(NC(c2ncsc2-c2ccccn2)=O)C1 15603,CCCC(F)C(=O)NCc1cccc(CNC(=O)C(F)CC)c1 15604,c1(C(=O)NCC(CCOC)NC(=O)C#CC(C)C)noc2c1CC(C)CC2 15605,CC1CCCC(O)(C(=O)NCCCCN(C(=O)COc2cnc(Cl)cn2)C)CC1 15606,Cc1nccnc1C(N1CCC2CC12C(=O)Nc1cnc(F)nc1)=O 15607,C(=O)(CCCCC(C)(C)OC)N1C(C(C)(C)NC(CCC=CCC=C)=O)CCC1 15608,Cc1cc(C(=O)NCCC(C)(C)NC(=O)C(=O)N(C)C)nn1CC(F)(F)F 15609,CC1CC(CNC(=O)CN2CCCC2)CN(C(C2CCSC2)=O)C1 15610,c1(N2CCN(CC(=O)Nc3ncn(C)n3)C(=O)C2)ccnc2cc(Br)nn12 15611,CCCC(CCCNC(=O)CCC(C)OC)NC(c1cc(F)ccc1N)=O 15612,c1(C(N2C(CNC(C(CNC(C)=O)(C)C)=O)COCC2)=O)n[nH]c2c1CCCCC2 15613,C1(CC(=O)NCCCC(C)NC(c2c(C)nsc2C)=O)CCCNC(=O)C1 15614,C1(C(=O)NCC2CCCCN2C(c2ccc(F)c(Cl)c2)=O)CC2(CCC2)CCO1 15615,O=S(=O)(c1c[nH]c2cc(Cl)ccc12)N1CC(O)(c2cccnc2)C1 15616,C=C(C)CCC(C)(c1nnnn1Cc1ccco1)NC(CCC)CCCC 15617,N1(C(C2CCC(=O)N2)=O)CC2CCC1C(C(N1CCCCC1CCO)=O)C2 15618,Cn1cc(C#N)cc1C(N1CC(NC(=O)CCNC(=O)C=CCl)C(C)(C)C1)=O 15619,C1(NC(C2(CC=C)CN(C(=O)CC3CCC(=O)CC3)C2)=O)CCC(N=[N+]=[N-])CC1 15620,N1(C(c2nccc(C)c2)=O)CC(CNC(=O)CCc2cnc(C)o2)CC1(C)C 15621,CC1CCCCCC1NC1CCN(C(=O)Nc2cccc(N(C)C)c2)C1 15622,c1(-c2ccc(C(=O)Nc3c(C)n[nH]c3)nc2C)ccc(F)c2ccoc12 15623,C1(CC=C)(NC(=O)CN2CCCCC2C)CCN(C(c2cnn(CCF)c2)=O)C1 15624,C=C1CCN(C(=O)C(C)NC=O)C(C(=O)NC(c2ccc(C)cn2)C)C1 15625,N1(C(C(C2CC2)OC)=O)CCC2(C)CN(C(=O)C(O)C(C)(C)C)CC12 15626,CCCCC(C(=O)NCC(C)(C)C#CC(=O)NC1CC(CCF)C1)C(C)C 15627,C1(CC(=O)NCCC(CC2CCC2)C(N2CCCC2C2CC2O)=O)COCCO1 15628,C1(NC(CCNC(=O)NC)=O)CCCC2CN(C(=O)C(C(C)C)OC)CC12 15629,C(=O)(C(O)CCC(F)(F)F)N1CCN(C(c2c(CC)nns2)=O)C2C1C2 15630,CC(C)C(C(=O)NCC1(C(=O)NC2CCOC2(C)C)CCCO1)NC=O 15631,c1(OC)cc(C(=O)NC(C)CCCCNC(C2CCC3(CC3)C2)=O)cc(OC)n1 15632,C#CCC(C(=O)NC(CO)CC=CC)NC(c1cnc(CC)nc1)=O 15633,c1(N(C)CC2CCCN(CCc3ccccc3)C2)nccc(C(F)F)c1F 15634,C#Cc1ccc(C(N2CCC(O)(CCNC(C3(C4CCCCO4)CC3)=O)C2)=O)o1 15635,C=C(F)C1(CC(=O)N(CC(C)NC(=O)CCCC(=O)OCC)C)CCOCC1 15636,n1(CC(=O)NC2CC(N(C(C)=O)C)C2)cc(C(F)(F)F)cn1 15637,C=CCC(CC(=O)N1CCC(C(=O)N(C)C)C1)NC(=O)Cn1nc(C)oc1=O 15638,C1(CNC(C(C)(C)OC(C)=O)=O)CN(C(=O)CN2CCS(=O)(=O)CC2)CCCO1 15639,c1(C(N2C(C(=O)Nc3ccc(F)cc3Cl)CC3(CC3)C2)=O)c(Cl)cc(F)cc1Cl 15640,c1(CN2C(C(=O)NC(CCC)C)CC3(CC3)C2)c(F)cc(Br)cc1Br 15641,C1(C)(C(=O)NC(C(CO)NC(c2cc(CSC)c(C)s2)=O)C)CCC(=O)N(C)C1 15642,CC(C)C(CCO)N=c1ccnc(NC2CNC(=O)C2)[nH]1 15643,C1(C(C)NC(C2(C(=O)NC)CCC2)=O)CCN(C(=O)C(C)O)CC1 15644,C(CCCCC(=O)N1CCC(C(=O)Nc2cccc(Cl)c2O)C(O)C1)OCC 15645,C1(C(N(CC(C)(C)NC(CCC(=O)N(CC)CC)=O)CC)=O)CC12CCCOC2 15646,N1(C(c2c(SC)csc2)=O)CC(NC(=O)Cc2cc(=O)n(CC(C)C)[nH]2)C(O)C1 15647,c1(OC)cc(=NC(=O)C(F)C2CN(C(C3CC(C(C)C)C3)=O)C2)[nH]n1C 15648,N1(C(C(CC)CN(C)C)=O)CCCC12CCN(C(c1cnc(O)n(C)c1=O)=O)C2 15649,c1(C(C)=O)ccc(NCC2CCN(C(C3CCOCC3(C)C)=O)C2)c([N+](=O)[O-])c1 15650,CC(CNC(=O)C1=NNC(=O)C1)C(F)C(=O)NCCCc1cnn[nH]1 15651,C(=O)(C(CCCCCN)C(C)(C)C)NC1CC2(CC(C(=O)OC)C2)OCC1 15652,C1(COC)CC(OC)CN1Cc1cccc(C2CC2)c1 15653,N1(C(C2C3(CCC3)C23CCC3)C(=O)NCSc2ccccc2)CCC(F)(F)C(O)C1 15654,c1(C(=O)NC2C(C(=O)NCCC)COCC2)cc2cnccc2[nH]1 15655,C(=O)(CCC1=CCCCC1)NC1(C(=O)NCCC(C(C)C)O)CCC1 15656,C(CC(F)F)(C(=O)NC1C(O)CC1O)N(C)C(C1CCC1)=O 15657,CCC(CNC(C1CC(=O)CN1C(=O)CSCCC(C)C)=O)(CC)CO 15658,C1(C)(C(N(CC(CNC(C(C=C)O)=O)(C)C)C)=O)CCC2CC2C1 15659,C12(CC(=O)NCC(F)CO)CCC1CN(C(c1cc(CO)on1)=O)C2 15660,Cc1cc(=NCc2csc(C)c2C)[nH]c(=NCc2ccnc(O)c2)[nH]1 15661,Cc1ccc(C(=O)NC2COCC2NC(c2snnc2C(C)C)=O)c(Cl)c1 15662,c1(NC(N2CC(C(C)NC(CNC(CCC)=O)=O)OCC2)=O)cccc2c[nH]nc12 15663,Cc1ncsc1C=CC(=O)N(CCC(C)NC(=O)CS(=O)(=O)NC1CC1)C 15664,C1(CCN(C(c2c(CC)occ2)=O)C)CCN(C(c2ccsc2C(F)F)=O)CC1 15665,c1(N(CCC)C)ccc2cc(S(=O)(=O)NCC3(F)CCC3)ccc2n1 15666,C1(COC)(CNC(=O)CCC2C(=O)NN=C2C)CCCN1C(C1CC(Cl)(Cl)C1)=O 15667,C1(OC)CC(CNC(=O)C=C(C)C)N(C(=O)CCCc2cccs2)C1 15668,c1(CN2C(CNC(c3c(OCC)nccc3)=O)CCC2)c(F)ccc(F)c1O 15669,C1(NC(C2(OC)CC2)=O)C2CN(C(C3CCCN3Cc3ccccc3)=O)CC12 15670,c1(OC)c[nH]c(C(=O)NC(C)CCCCNC(=O)C(F)n2cccn2)cc1=O 15671,N1(C(=O)CCN(C(=O)CC2CC(F)(F)C2)C2CC2)CCOc2ccccc21 15672,N1(C(Cc2nc(C)sc2)=O)CC(NC(c2ccsc2Br)=O)C2CC2C1 15673,C1(CC(=O)NCC(C23CCC(CC2)C3)NC(C2CC(F)C2)=O)CC2C=CC1CC2 15674,C1(NC(=O)CCc2ccc[nH]2)CCC(NC(C2(C(F)(F)F)CCC2)=O)C1 15675,N1(C(CC2(CC)CCOCC2)=O)CC2CC(NC(c3cnoc3C)=O)CC2C1 15676,Cc1ccc2ncc(C(N3CCC4CCN(C(C5(F)CC5)=O)CC4C3)=O)cc2c1 15677,c1(C(N2CCCC(NC(c3cncc(CC)c3)=O)C2)=O)c(C)cc(F)cc1Br 15678,CC1CN(C(C23CCN(C(C45CCC(C4)C5)=O)CCC2C3)=O)c2ccccc21 15679,N1(C(C(C2(O)CN(C(c3cccnc3O)=O)C2)F)=O)CC2C(C1)C2(F)F 15680,N1(C(C2(C)CC(F)C2)=O)CC(C)CN(C(c2ccc(C3CC3)cn2)=O)C(C)C1 15681,N12C(CCC1c1ccccc1)C2=O.C1(SC(C)(C)C)CC(C(=O)OC)CO1 15682,C#CCC(O)C(=O)NC(C(=O)NC1CC(CC(N)=O)C1)C1CCOC1 15683,C1(NC(C(F)=CC)=O)CC2CCC1CN(C(c1cc(C(F)(F)F)ccc1C)=O)C2 15684,c1(C(=O)NC2C(C)(CNC(C3C(=C)C3)=O)CCC2)c(S(C)(=O)=O)cnn1C 15685,CS(=O)(=O)CC(=O)NC(C(=O)N1CC(CC(F)F)C1)C1CC1 15686,CC(CCCCCO)NC(c1c(Br)ncn1C)c1nnnn1Cc1cccs1 15687,c1(CC(N2CC(CN(C(C3C(OCC)CC3)=O)C)C2)=O)cnn(CC)c1 15688,Cc1cnccc1C(=O)NC(CNC(=O)C(C)NC(c1cccs1)=O)C1CCC1 15689,Cc1cnccc1C(C)C(=O)NCC(C)(C)CN(C)C(c1[nH]nnc1C1CC1)=O 15690,C1(NC(c2cncc(CC)c2)=O)CN(C(C2COC(=O)N2)=O)CC1S(C)(=O)=O 15691,N1(C(CCCn2cc(C(C3CCCC3)OC)nn2)=O)CCn2nccc2C1CO 15692,CN1CC=C(CC(=O)NC2(C3CN(C(C4CCS4(=O)=O)=O)C3)CC2)CC1 15693,C(=O)(CCCCC(=O)OC)NCC1CCC(N(C(C(CCOC)OC)=O)C)CC1 15694,CCCCC(COC)NC(C1(CF)CCN(C(=O)C=CC(F)(F)F)C1)=O 15695,C1(C(=O)NCc2cn(CC#C)nc2)COCCN(C(=O)Cc2scnc2C)C1 15696,c1(C(=O)NCC2N(C(=O)C3=CCCS3)CCC(C)C2)cnc2ccoc2c1 15697,C1(C(=O)NC2(C(=O)OC)CC2)CCCC1CNC(C1CCOC1C(C)C)=O 15698,N1(C(C(C)C(C)(F)F)=O)CCOC2(CCCN(C(=O)Cc3csc(S)n3)C2)C1 15699,N1(C(C2(OC)CCCOC2)=O)CCC=C(CNC(=O)C(C)C(C)C)C1 15700,C1(CNC(c2cc(CNC(CCCC)=O)on2)=O)CCCCCC1 15701,C12CN(C(C3CCS3(=O)=O)=O)CCC1CNC2=O.c1(CC)c[nH]nc1[N+](=O)[O-] 15702,Cc1nnc2n1CCCC2C(=O)NC1CN(C(=O)C(c2ccnn2C)C)C1 15703,c1(C(=O)NC2C3CN(C(c4cnc(C)nc4)=O)C(C3)C2)ccc2c(c1)CCC=C2 15704,c1(C(=O)NCC(CNC(=O)CO)OC)cnn(-c2ccccc2Cl)c1C(F)(F)F 15705,C(=O)(C(C)(C)C)NCC(n1cc(C2CCCC2O)nn1)C.C(=O)COCC 15706,Cc1cc(CNC(=O)CC2CN(C(C3OC4CCC3C4)=O)CC23CC3)cnc1C 15707,Cc1cn(C)c(C(c2nnnn2CCN2CCOCC2)Nc2cscc2C)n1 15708,C(=O)(CCC(CF)CF)N1CC2C(NC(c3n[nH]c(C)c3Br)=O)(CC2)C1 15709,c1(CCC)nc(C)c(C(=O)NCCNc2ncc(C(=O)OC)cn2)s1 15710,c1(CC(=O)NC2C(CC(C)(C)C)CN(C(C3CCCS3)=O)C2)ccc(Cl)cc1F 15711,c1(CC(=O)NCC(CNC(=O)CC(C)F)OC)ccc2cnccc2c1 15712,C(CCN=c1[nH]c(=NCC(C)C2CCC2)[nH]c2c(F)cccc12)N(CCOC)C 15713,C(CCCC1CC1)NC(C1(N(C(CC2(COC)CC2)=O)C)CC1)=O 15714,CC1CC(CO)CN(C(=O)C(N2CCN(C(=O)CC3CCCC3(F)F)CC2)=O)C1 15715,c1(C(=O)NCC2(F)CCC(NC(CCC(C)OCC)=O)C2)cnc(C)nc1CC 15716,N1(C(CCC2C(C)(C)C2)=O)CC2CCCC2(COC(C2(CC(=O)N(C)C)CC2)=O)C1 15717,c1(CC(=O)NC(C(C)NC(=O)C=Cc2cnc[nH]2)C)ccc([N+](=O)[O-])cc1 15718,C12(C(=O)NC(c3ccn(C)n3)C)CCCC1CCN2C(C1CCCCC1O)=O 15719,C1(C(=O)NCC(C)N(C(c2cn[nH]c2)=O)CC)COCCC1(F)F 15720,c1(C(N(C(C)CNC(c2c[nH]c(C#N)c2)=O)C)=O)ccc([N+](=O)[O-])s1 15721,C(=O)(C(O)C(F)F)N1CCC(N(C(COCCOCC)=O)CC)C1 15722,c1(C(=O)NC2C(CNC(c3ccn(CC)n3)=O)CC2)cc(Cl)cc2c1NCCC2 15723,N1(C(C2(CNC(CN(C(COC)=O)C)=O)CCCCC2)=O)CC(F)(F)CCC1C 15724,C1(C(N(CC(C(C)C)C)C)=O)CSCCN1C(=O)CC=C(Cl)Cl 15725,N1(C(c2c(C)cco2)=O)CC2(CC(NC(=O)C(F)C3CCC3)CO2)C1 15726,C1(C(N2C(C)(CNC(CSCCC)=O)CCC2)=O)COCC(C)(C)O1 15727,c1(C(=O)NC(C(CC)CC)C)n[nH]c2c1CN(C(C1(F)CC=CCC1)=O)C2 15728,N1(C(c2cnc(CNC(C3(C)CCCC3)=O)nc2)=O)CC2CCCC(O)C2C1 15729,Cc1cnc(Br)cc1NC(C1(F)CCN(C(=O)CCc2cccc(C#N)c2)C1)=O 15730,N1(C(C2(SCC)CC2)=O)CC(NC(=O)C=C(C)c2ccsc2)C(O)C1 15731,C12(NC(N3CCCCC(C(=O)O)C3)=O)CCCN(CC1)S2(=O)=O 15732,C1(NC(C(CCOC)C)=O)CC2CCC(C1C)N2C(c1cc(CN(C)C)on1)=O 15733,C1(O)(CNC(c2nn(C)c(F)c2)=O)CCN(C(=O)CC2CCCC(=O)N2)CC1 15734,N1(C(CCC(=C)Cl)=O)CC(NC(C2(c3ccncc3)CC2)=O)CCC1C 15735,c1(NC(COC)C)[nH]c(=NCC2OCCc3ccccc32)nc2c1cnn2C 15736,c1(OC)cccnc1C(=O)NCC1(CCNC(=O)CC(C)CF)CC1 15737,N1(S(C2CC(OC)C2)(=O)=O)c2ccccc2C(C)(C)C1C 15738,C(C(C)(C)NC(=O)CCc1ncco1)N(C(=O)CNC(=O)NC1CC1)C 15739,N1(C(C(C=C)CC)=O)CCOC(C(=O)NC2COC3(CCC3)C2)CC1 15740,N1(C(C2C(CCC)C2)=O)CCC2(C(=O)NCC(N3CCOCC3)C)CCCC12 15741,c1(C(=O)NC2(CNC(C3CC(C)(CC)C3)=O)CCOC2)cncc2c1CCC2 15742,c1(C)cccc(Cl)c1C.n1(CCSC)nnnc1C(C1CC1)NCCOCCO 15743,CC1CCCC1(C(=O)N(CC(N)=O)C)NC(=O)Cc1cncnc1O 15744,CCC(CC)(CCNC(C1(F)CCOC1)=O)NC(c1ccc(C)c(Cl)c1)=O 15745,C1(C(=O)NC(C2CCCO2)(C)C)COCCN1C(=O)C=CC1CCOCC1 15746,Cc1[nH]nc2c1CCC(C(N1CCC(C)(CNC(c3cccc(N)c3)=O)C1)=O)C2 15747,Cc1cc(F)c(F)cc1C(=O)NC1CN(C(c2ccc(F)c(O)c2)=O)CC1F 15748,Cc1cc[nH]c1C(=O)NCCCNC(C1CC(Cc2ccnn2C)C1)=O 15749,C1(CNC(C(=O)NCC)=O)CCN(C(=O)C(C)Cc2ccccc2)CCC1(F)F 15750,CCCCCCCCC(=O)NCC(C)(CC(C)C)NC(=O)CC1CC1(Cl)Cl 15751,N1(C(C(CC)C2CC2)=O)CCN(C(=O)C(c2cccc(OC)n2)(F)F)CC(O)C1 15752,c1(C(=O)NCC(CO)NC(=O)C(C2CCCC2)C2CCC2)ccc2c[nH]nc2c1 15753,C1(C(=O)NC2C(NC(CC)=O)CC2)CCN(S(=O)(=O)NC)CC1 15754,c1(C(N2CCCCC(NC(c3ncn(C)n3)=O)C2)=O)ccc(Br)cc1C#N 15755,c1(C(N2CC(CC=C)(NC(C3(F)CCOC3)=O)C2)=O)ccc(C)c(C)n1 15756,c1(C(=O)NCC2(NC(c3c(C#C)c[nH]n3)=O)CCCCC2)cc(C)ccc1O 15757,CCC(CC(=O)NC(C)(C)CNC(=O)CCCNC(c1ccccc1)=O)C(F)F 15758,Nc1cnc(C(F)(F)F)cc1C(N1CCC(F)(CNC(C2CC(F)C2)=O)C1)=O 15759,S(=O)(=O)(c1cncc(Br)c1)N(CC)Cc1cccc(C2CC2)c1F 15760,C1(O)(C(C)NC(c2cn(C3CCC3)nn2)=O)CCN(C(C2(F)CCC2)=O)C1 15761,C1(C(=O)NCC(C)C#N)CC(N=[N+]=[N-])CN1C(=O)CC(C)(C)C#N 15762,c1(C(=O)NC(CO)C(O)C2CCCCC2)cnn2ncccc12 15763,c1(OC)cc(CCC(=O)NC23CC(NC(=O)CC4CCCO4)(C2)C3)ccc1O 15764,c1(OCC)cccc(C(=O)NC2CCC(CCNC(C3(OC)CC3)=O)C2)c1 15765,CC(C)C(C)C(C)CC(=O)N1CC2(CC2)CC1CNC(c1coc2c1COC2)=O 15766,C12(NC(c3ccc(C)cc3C)=O)CCC(CN(C(=O)CCC3CC3)C1)C2 15767,C1(CC(=O)NCCCOCCN(C(C(C)NC(N)=O)=O)C)CCCCCC1(F)F 15768,C1(C2C(N(CC(F)(F)F)N(C3CCCOC3)C=O)C2)CCC2CC2C1 15769,C(=O)(C1CCCc2ncnn21)NC(C(C)(C)NC(c1c[nH]c(=NCC)s1)=O)C 15770,N1(CCC)CC(C(=O)NCCC2(C)CCN(C(c3cncnc3C)=O)C2)CC1=O 15771,CC(C)CC(C)(O)C(=O)NCC12CCC(CC1)N(C(C1CCCC1C(C)C)=O)C2 15772,C(CC(F)=C(F)F)NC(C12CC(NC(=O)C=Cc3cc[nH]c3)(C1)C2)=O 15773,c1(C(=O)NCCC(C(C)C)C)cccc2c(Cl)cccc12 15774,c1(NC2CC(C)N(C3CC3)C2)ncccc1[N+](=O)[O-] 15775,C1(CC=C)(NC(C2CC(OC)C2)=O)CCCN(C(c2cnccc2C)=O)C1 15776,N1(C(c2ccn(CCC)n2)=O)CC2CN(C(=O)Cc3cc(O)nnc3O)CCC12 15777,N1(C(C(C)NC=O)=O)CCCCC1C1(C(=O)NCC2(F)CCOCC2)CC1 15778,c1(NC(N2CCN3CC(F)(F)CC3C2)=O)cc2c(cc1Br)OCCO2 15779,Cc1ccc(C(C)CC(=O)NC23CC(NC(c4cncc(N)n4)=O)(C2)C3)cc1 15780,C1(CC(=O)N(CC(C)NC(C2(C(C)(C)C)CCCC2)=O)C)CCCC2(CC2)C1 15781,C1(C(=O)NCC2(NC(C3CC(CC)C3)=O)CCOC2)CC2CC1CC2O 15782,c1(CC2C3CN(C(=O)NCc4cnco4)CC32)c[nH]c2cc(F)c(F)cc12 15783,c1(C(C)(C)C)ccc(C(=O)NC2CC2CNC(=O)C=Cc2cncs2)nc1 15784,c1(C(=O)NCC(C)CNC(c2ccccc2Cl)=O)ncc(C(F)(F)F)cc1O 15785,c1(C(N(C2C(C)CCNCC2)C23CC(CO)(C2)C3)=O)ccc([N+](=O)[O-])cc1I 15786,c1(NC(C2C3CN(C(C(C)Cc4ccccn4)=O)C2C3)=O)cc(Cl)nnc1Cl 15787,C1(CC(=O)NC(C(C)C)(C)CNC(C23CCCC2C3)=O)CCCCCCC1 15788,C(=O)(C1=CNS(=O)(=O)N=C1C)NC1CN(C(C2CCN(C(CC)=O)C2)=O)CC1C 15789,c1(C(=O)OCC)ccc([N+](=O)[O-])[nH]1.C1(n2c(CC)ncc2)CCCN(CC=O)C1 15790,N1(C(C2OCC(C)C2)=O)CCOCC(CNC(=O)CC2NC(=O)NC2=O)C1 15791,C(=O)(C1=CNC2=NCCC2=C1)N1CC(O)(CNC(=O)CC2CCCCCO2)C1 15792,C1(N(C(=NC)Nc2ccc(C#N)cn2)C)CC2CN(C(=O)OC(C)(C)C)CC2C1 15793,CC(c1ccccc1)=CC(=O)NCC1CN(C(C2(C(F)(F)F)CC2)=O)CCN1C 15794,c1(CC)cnc(CNC(=O)C(c2cnn(C)c2)NC(c2cc(C)c[nH]2)=O)[nH]1 15795,CC(C)CC(C(=O)NCC(C)(C)CCNC(=O)CC1CCCN1C)C(C)C 15796,C1(CC(=O)NCC=CCNC(C2CC3OC(=O)OC3C2)=O)CCc2sccc2C1=O 15797,C(CCS(=O)(=O)c1ccccc1)NC(=NCCC=C)NC1CCSC1 15798,c1(C(N(C2CC(NC(CN(CC)CC)=O)C2)C)=O)cnn2c1CCCC2 15799,N1(C(C(C)=CC)=O)CCC(NC(=O)CC(O)c2ccccc2)C1(C)C 15800,c1(C(N2CCC(NC(C(CCOC)C)=O)(CO)CC2)=O)cc([N+](=O)[O-])ccc1C 15801,N1(C(=O)CC2(C3CC3)CC2)CC2ON=C(CNC(C3(CO)CC(F)(F)C3)=O)C2C1 15802,c1(OC)ncnc(OC)c1C(=O)NCCOC1CCN(C(=O)C(O)P(C)(C)=O)C1 15803,n1(CC)nc(C2CC2)cc1C(=O)NC1CN(C(=O)COC(C)=O)CC1OC 15804,C1(S(N)(=O)=O)(C(=O)NCCNC(C(c2ccc(Cl)cc2)(C)N(C)C)=O)CCCC1 15805,C1(C(=O)NC2CN(C(c3n[nH]c(C)c3O)=O)CC23CC3)CCc2cn(C)nc2C1 15806,CC1(Cc2ccncc2)CCCN1C(=O)CSCc1cn(Cc2cscn2)nn1 15807,C=CCC(C(=O)NCCCOC1CCCCCC1)C(C)C 15808,c1(C(=O)NC2(C)CC(NC(c3cnc(C4CC4)s3)=O)C2)ccc(C(=O)CF)cc1 15809,C(=O)(C1COc2ccc(F)cc21)N1CCC(NC(C2(C(F)(F)F)CC(=C)C2)=O)C1 15810,c1(N2CCC(C(N3CC(CCC)(C(=O)O)C(O)CC3)=O)C2)cnn2cnnc2c1 15811,c1(OCC)ccc2nc(C(=O)OCC)sc2c1.C12(OC(C)=O)CC(C1)N2 15812,c1(CN(CC=C)C)ccc(C(=O)N(C)CC2CN(C(=O)C(F)CC)C2)cc1 15813,c1(C(N2CC3CC2CO3)=O)cc2n(n1)CCCN(Cc1cc(F)c(Cl)c(F)c1)C2 15814,N1(C(C2CC(=O)C2)=O)CCC(C2(CNC(C3CCCSS3)=O)CCOCC2)CC1 15815,c1(C(N2CCN(Cc3cc(OC)ncc3Cl)CC2CO)=O)cc(F)c(O)c(F)c1 15816,C=C(C)C1OCCC1C(=O)NCCC1(NC(c2cc(O)nc(O)c2)=O)CCC1 15817,c1(OC)ccc(OC)c(CCC(=O)NCC(C2CC2)N(C(=O)CC=C(C)C)C)c1 15818,c1(OC)cccc(C(=O)NCC2(F)CC(NC(c3c[nH]nc3C(F)(F)F)=O)C2)c1 15819,CC(C)C(CNC(c1cn(CC2CC(=O)C2)nn1)=O)NC(C1CC12CCC2)=O 15820,c1(C(N2C(CCNC(C3CCCSS3)=O)CCCC2)=O)ccc2ncsc2c1 15821,C1(C(N(Cc2cccc(C)c2)Cc2ccc(N)c(F)c2)=O)CCS(=O)(=O)N1C 15822,N(C(=NCCc1ccccn1)N1CCC2(CCOC2)C1)CC1CCN(CCOC)C1 15823,N1(CC(=O)NCC(CC)(C)NC(=O)C#CC(=O)N(C)C)CCC(CO)CC1 15824,C1(NC(c2c(OCC)cccc2)=O)CCN(C(=O)CCC2CC2(F)F)C(C)C1 15825,c1(C(N2CCC(CNC(C(=O)NCC)=O)CC2)=O)c[nH]c(=N)cc1C 15826,C(=O)(CC(C)CC(C)(C)C)NCC(CCC)C(=O)N(C)CC1CCSC1 15827,C12(CNC(C=Cc3n(C)ccc3)=O)CCCC1CCN2C(=O)C=C1CCSCC1 15828,CC(CN=c1nc(N2CCc3ncncc3C2)c2c([nH]1)COC2)c1nccs1 15829,c1(OC)cc(C)cnc1C(N1CC(CNC(c2cc(C)co2)=O)C(C)(C)C1)=O 15830,C1(NC(C(CSC)O)=O)C2CCN(C(=O)CCSc3nnnn3C)C12 15831,CCC(C(=O)N1CCCC1CC(=O)NC(C1CC1)C1CC1)NC(N)=O 15832,C(c1ccoc1)=C(C)NC(=O)CC1CCN1C(=O)COCC1CCOC1 15833,N1(C(CN2C(C)CC2)=O)CC2CC1CCC2NC(c1ccc(F)c(C2CC2)c1)=O 15834,Cc1cccc(OCCC(N2CC(NC(=O)Cc3occc3C)C(C)C2)=O)c1C 15835,c1(C(=O)NC2C(NC(C(CC)N(C)C)=O)CCOC2)cccc2[nH]cc(C#N)c12 15836,C1(C(N(CCNC(C)=O)C)=O)CC2CC1CC2NC(c1cncc(O)c1)=O 15837,Cc1ncc(-c2cn(CCOc3sccc3-n3ccnn3)nn2)o1 15838,N1(C(C2CCC(=O)O2)=O)CCCCC1CNC(C1CCC(O)CC1)=O 15839,c1(C(=O)NC(CC(C)C)C(=O)N2CCC(N3CC=CC3)C2)ccn2ccccc12 15840,C#CCCCC(C)C(=O)N1C(CNC(=O)Cn2ccccc2=O)CC2CCCC12 15841,C(=O)(C(C)CNC(C1CCSCC1)=O)NC(c1ncco1)C 15842,C1(C)(C(=O)NCC2CN(C(C3C(CC(C)C)C3)=O)C2)CCC1 15843,C=CCC(C)(C)C(=O)N1CCN(C(C2CC23CC(OCC)C3)=O)C(CF)C1 15844,N1(C(C(COCC)N=[N+]=[N-])=O)CCc2ccc(C(=O)NC(CSC)CC)nc2C1 15845,N1(Cc2ccc(C#N)cc2)CCC2CN(C(=O)CCc3ccc(F)cc3)CC2C1 15846,c1(N(CC(=C)C)C(C2CC(O)CN2C(=O)CN(C)C)=O)ccc(C)c(C)c1 15847,N1(c2nc(OC)cc(OC)n2)CCC2(CCC(NC(=O)CC(O)C(C)C)CC2)C1 15848,CC1CC2CCC(C1)N2C(=O)CC1C(NC(=O)C(C#N)C(C)C)CC1O 15849,C=C(C)CN=c1[nH]c(=NCc2ccc(OC(C)C)cc2)c2[nH]ccc2[nH]1 15850,N1(c2n(CC=C)c(CCC3CCCCC3)nn2)CCCC2CN(C)CCC12 15851,c1(CC(N2CCN(C(c3cc(N)c(F)cc3)=O)CC2)=O)cnc2c(=O)[nH]ccn12 15852,CCCCCCC(=O)N1CCCC(CN(C)C(C2CCCNC2=O)=O)C1 15853,Cc1ccc(C)c(C(=O)NC2C=CC(CC(N3CCC4CC34C)=O)C2)n1 15854,N1(C(CC(CC)OC)=O)CCc2nc[nH]c2C12CCN(C(=O)C=CI)C2 15855,c1(C(=O)NC2C(CNC(COC)=O)C2)cc2ccccc2nc1C(F)F 15856,N1(C(C2C(n3nc(C)c(-c4ccc(CO)cc4)c3)C2)=O)CCC2(CCCC2)CC1 15857,c1(C(N2CC3C(C(N(C(C)CC(N)=O)C)=O)(C3)C2)=O)c(O)cccc1F 15858,C1(N(C)C)(CNC(C2OCCC2NC(C2C=CCC2)=O)=O)CCOCC1 15859,C1(C(=O)NCCN2CCC(C)(C)C2)CCC(C)(C)N(C(=O)C=C2CC2)C1 15860,C1(C(=O)NCC2CC(F)(F)CO2)CCN(C(=O)COCC(F)F)C12CC2 15861,C1(NC(C2CN(C(C=C(CCN(C)C)Cl)=O)CC2CO)=O)CC2CCCCN2C1 15862,C1(NC(CCCc2[nH]c(=N)sc2)=O)CN(C(c2cccc(=O)o2)=O)CC2CC12 15863,c1(OCC)cc(C(=O)NC(C)CC2CN(C(=O)CSC)C2)[nH]n1 15864,C(=O)(CC(O)CCCCC)NC(C(=O)NC1(C=C)CCCC1)CCSC 15865,N1(C(C2CCC(CNC(C(COC)C)=O)C2)=O)CC2(C1)CN(C)C2 15866,c1(OC)ccccc1C1(OCC(N2CC(n3c(O)nnc3O)C2)=O)CCC1 15867,C1(C(N2CCC(CNC(CCN(c3ccncc3)C)=O)C2)=O)CCC2(CC2)C1 15868,CC(C)CC(CNC(C1(C)CCCCO1)=O)C(=O)NCc1ccc(O)nc1 15869,C(C1CC1)(C1CC1)=CC(=O)NC1CC(NC(C2CSCC2c2ccccc2)=O)C1 15870,C(=O)(CS(=O)(=O)C(C)(C)C)NCC1N(C(CC2(C=C)CCOCC2)=O)CCCC1 15871,N1(C(C2(CC=C)CCOCC2)=O)CC2CCC1CC2NC(=O)C=C(Cl)Cl 15872,c1(N2C(CN(C(C(C(COC)C)C)=O)C)CCC2)ncc2c(Br)cccc2n1 15873,C(=O)(C(C)C(F)(F)F)N(C(C)C)CCN(C(=O)C(O)Cc1ccc(Cl)cc1)C 15874,C(=O)(C(F)(CNC(=O)CCc1cnco1)C(C)C)NC(c1cccs1)CC 15875,c1(C(=O)NCCC2CCN(C(C(C)OCCOC)=O)CC2)nccc2n[nH]cc12 15876,C(CCCC(=O)NCC1CCC(NC(=O)CC2CCCN2C)CC1)N(C(C)C)C 15877,C1(c2cccc(F)c2)(NC(CCOCCC)=O)CCN(C(=O)C=NOC)C1 15878,C(c1cccc(O)c1)=CC(=O)NCC1CN(C(c2cccc(C)n2)=O)CC1C 15879,C1(NC(c2c(CC)nc(C)o2)=O)CCC12CN(C(c1cccc(F)c1OC)=O)C2 15880,O=C1CCC(CC(N2CCC(O)(C(F)F)C2)=O)CN1 15881,N1(C(c2noc(CC)c2C)=O)CC(C)CN(C(=O)C2=NNC(C(F)(F)F)C2)C(C)C1 15882,C1(C(=O)NCC2(NC(=O)Cc3ccccc3Cl)CCC2)CCC(F)(F)CC1 15883,c1(C(N2CCC(CNC(C(CCC)OC)=O)C23CC3)=O)cc2ccncc2[nH]1 15884,N1(C(C2(NC(=O)CC3CC(O)C3(C)C)C(C)(C)C2)=O)CC(O)C(O)C1CO 15885,C1(C(=O)OC(CC(=O)OCC)CC#N)CC2(CCCCC2)C1 15886,C#CCC(C)(CC)C(=O)N1CCCC1CNC(C1CC12CC(F)(F)C2)=O 15887,C(CCCCC(=O)NC1(C2CCCCN2C(=O)C(C)n2cccn2)CC1)OCC 15888,Cc1cnccc1CN(C)C(c1cc(C2CC2)nn1C(C)(C)C)=O 15889,C1(NC(=O)C=Cc2cn[nH]c2)CC2CC1N(C(=O)CC1(c3ccc(F)cc3)CC1)C2 15890,C1(NC(C)=O)CCC(C(=O)NC2CCCC2NC(C2(CC(C)C)COC2)=O)CC1 15891,N1(c2n(CC)c(C(c3ccc(Cl)cc3)CC)nn2)CCCc2ccccc2C1 15892,C1(C2(O)CN(C(C3(Cl)CC3(F)F)=O)C2)(CNC(C(F)=C(C)C)=O)CC1 15893,c1(NC(C)=O)cccc(C(N2CC=CC2CNC(c2c(C)[nH]c(C)c2C)=O)=O)c1C 15894,C(C)(CCCCN=c1nc2c(cnn2C)c(NCC(C(C)C)C(C)C)[nH]1)OC 15895,Cc1csc2ncnc(N3CCCCC(CNC(=O)CCc4cc[nH]n4)C3)c12 15896,c1(CCOC)n[nH]c(=NCCCN(C)C(C2CCCC2OC)=O)s1.c1cccc(Cl)c1 15897,c1(-c2cc(C(=O)OC)sc2)ccc2c(c1)CCN(c1cc3ncnn3cn1)C2 15898,c1(N2CC(CN(C)C(c3cn(CC4CC4)nn3)=O)OCC2)ncnc(Cl)c1C#N 15899,O=C(C1=NOC(CC2(O)COC2)C1)NCC1CCCN1C(=O)CCOCC(F)F 15900,c1(CC(N2CC(CCNC(C)=O)C2)=O)c(N)nc(C)nc1O 15901,C(C(C)CC(F)(F)F)NC(CCCN(C(C(C)C)=O)CCCO)=O 15902,Cc1csc2ncc(C(=O)NC3CCCN(C(C4CC5(C4)CC(O)C5)=O)C3)n12 15903,N1(C(C2CC(F)(F)C2)=O)CC2CC(C1)N(C(c1csc(-c3nc[nH]n3)n1)=O)C2 15904,C1(n2cc(CCNC(C3(C)C(C)C3)=O)nn2)CCCC=C1Br 15905,C1(NC(C(=O)Oc2ccccc2)C)CCN(C(c2ncccn2)=O)C(C2CC2)C1 15906,c1(C(=O)NCC2(CNC(C=Cc3cc(C)no3)=O)CC2)ccccc1S(C)(=O)=O 15907,C1(NC(c2n(CC)ncc2)=O)CC2CCC(C1)N2C(c1nonc1N)=O 15908,N1(C(C(=C(C)c2ccco2)C)=O)CCCC(NC(=O)C(C)(C)Cc2cnn[nH]2)C1 15909,Cc1cc(=NC(=O)C=C2CC3C2CCN3N(C(=O)C(C)C)C(C)(C)C)[nH]o1 15910,N1(C(C=CC)=O)CCC(C2CC2)C1C(=O)N(C1CC(CO)C1)C 15911,Cc1cc(C(N2CCOC(C(C)NC(=O)CN=S(C)(C)=O)C2)=O)cnc1C(F)F 15912,Cc1cc(C(=O)N(C(C(=O)NCC2(C)NC(=O)NC2=O)C2CC2)C)nc(O)n1 15913,C1(C2CCN(C(C=C(C)C3CC3)=O)C2)CCCCN1C(=O)CC1CCCOC1 15914,CC1CC(C)N(C(=O)CC2CC2)CCN1C(=O)Cc1nc2cc(Cl)ccc2s1 15915,c1(CNCc2cc(C)cc(F)c2)ccc2c(c1)CCC2NC(=O)OC(C)(C)C 15916,c1(C(N2CC3CCN(C(COCCC#C)=O)C3C2)=O)cnc2c(c1)CCOC2 15917,C1(NC(c2c(CC)cno2)=O)CN(C(=O)Cc2cscn2)CCC1O 15918,C12(C(N3C(CNC(c4nccc(C(C)(F)F)c4)=O)CC3)=O)CCC(CC1)OC2 15919,C1(NC(c2cc(F)c[nH]2)=O)CC2CC1N(C(c1cnc(O)cc1O)=O)C2 15920,n1(CCCC)nc(CC2CCCCC2)nc1-c1nc(-c2ccccc2)n(C)n1 15921,C1(NC(c2c(CC)nc(=N)[nH]c2)=O)CCN(C(=O)CC2COCC2O)CC1(C)C 15922,Cc1csnc1C(=O)NC(Cc1ccoc1)C(=O)NC(C)CCC1CC1 15923,c1(NC(C2N(C(Cc3cccc(OC)n3)=O)CCOC2)=O)ccc2cnoc2c1 15924,C(=O)(C(F)CCCC)NC(C1CCN(C(CCC=CC)=O)CC1)CO 15925,C1(NC(C(n2ccc(C)n2)(C)C)=O)CN(C(c2cnc(O)c(C)c2)=O)CCC1O 15926,c1(C(=O)Nc2c(CC)nnn2C)ccc(C(=O)OC)c(Cl)c1 15927,Cn1ncc2c1CC(C(N1CCC(CCNC(c3cnc(O)o3)=O)CC1)=O)CC2 15928,c1(C(N(C2COCC2C(N)=O)CCNC(C2(CC#C)CCC2)=O)=O)cc(C)c[nH]1 15929,C1(CNC(=O)NCc2cnc(Br)s2)CC(O)CN1C(=O)C(Cl)(Cl)Cl 15930,C(N=c1[nH]c(N2CCC(CCF)C2)nc2c1CCC2)C1(C)CC1.NC 15931,c1(NC(C2(C)CCCN2C(=O)Nc2ccccn2)=O)nc(Cl)c(Br)cc1[N+](=O)[O-] 15932,N1(C(C2C(C#N)CC2)=O)CCC(C(=O)NCC2CC23CC3(F)F)(CO)CC1 15933,N1(C(CCc2c(OC)ccc(F)c2)=O)CCCC2(NC(=O)C(=O)N(C)C)CCCC12 15934,c1(CC(C)(O)C(N2CCCC3NCC[SH]23)=O)ccc([N+](=O)[O-])cc1 15935,C(C(O)C(=O)NC1CC(CNC(C2(CCN3CCOCC3)CC2)=O)C1)OC 15936,Cc1ccc(SC(C)C(=O)NC2CCC(NC(C3CCC(CO)CC3)=O)C2)cc1 15937,C12(NC(C(C)N(C)C(c3c[nH]c(C#N)c3)=O)=O)CC1COC21CCC1 15938,N1(C(c2c(CCC)occ2)=O)CCC(C2CCN(C(=O)CCCCO)C2)C1 15939,C(=O)(C(CCC)S(N)(=O)=O)NC1(C)CC(NC(CCC#CC)=O)C1 15940,C1(F)(C(=O)NCC(CNC(C2(CC3CCC3)CC2)=O)CO)CCCOC1 15941,Cc1ccc(C(=O)NC2CCC(C)(NC(=O)C#CC(C)C)CC2)c(C)c1 15942,Cc1nc(CC(C)C)c(C(N2CCC2CNC(c2cccc(CO)n2)=O)=O)s1 15943,C=CCC(C)(C(=O)N1CC(O)(C(C)NC(=O)C(O)C2CCC2)C1)N(C)C 15944,N1(C(C(CC)SC2CNC2)=O)CCC2(CC1)CN(Cc1cccc(C)c1)CCO2 15945,C1(NC(=O)C=NOC2CCCCO2)COC2(C1)CN(C(c1nc(Cl)ccc1F)=O)C2 15946,c1(NC(c2c(CCC)[nH]cc2)=O)ccc(NC(C2CC2[N+](=O)[O-])=O)c(C)c1 15947,N1(CC(=O)NC(CNC(=O)C=CSc2nc[nH]n2)C2C(CO)C2)CCCOC1=O 15948,c1(C(N(CCCN(c2nc(COC)nc(O)c2)C)C)=O)ccc(F)c(C#N)c1 15949,Cc1cc(C(=O)NC2CC(NC(C3CCCN(CC(C)C)C3)=O)C2)ncc1C#N 15950,C1(C2(O)CN(C(=O)C=C3CCCCC3)C2)(CNC(C2(CC=C)COC2)=O)CC1 15951,c1(C(=O)NC(CC)CNC(C2(CF)CC2)=O)ccc2c(n1)NC(=O)CO2 15952,c1(C(=O)NC2CN(C(=O)CC3CCC(F)(F)C3)C2)cnc2cccnc2c1 15953,c1(N2CCC(CNC(CC(CC)OC)=O)C(C)C2)ncnc2n[nH]c(C)c12 15954,C#CCC(C)(C(=O)NC1(CC)CCOC1)NC(c1nc(C)ccc1C)=O 15955,N1(C(c2cn(CCCOC)nc2)=O)CCC(C)C(CNC(C23CC(CO2)C3)=O)C1 15956,C1(NC(CCCCN(C)C)=O)CCCC12CN(C(C1CN3CCCC1C3)=O)C2 15957,CON1CCC(C(=O)N(C)CC2(O)CCN(C(=O)C(CC3CC3)SC)C2)CC1 15958,c1(C(=O)NCCc2nc(CC)sc2)cccc(Oc2ccc(Cl)cc2)c1 15959,C1(C(=O)NC(c2ccco2)COC)CN(C(=O)Cn2nc(C)nc2C)CC1C 15960,C1(N(C)C(c2ccc(-n3cnnc3)cc2)=O)CN(C(=O)C(C)(F)F)CCC1O 15961,c1(C(=O)NCC(CC)NC(=O)CC2CCC(C)(C)CC2)csc2cncn12 15962,CCCCCCC(C(=O)OC)N1CCN(C(=O)C(CCC)C(C)C)CC1 15963,CC(CC(=O)NC1(C2CCN(c3nc(Cl)ncc3C3CC3)C2)CC1)C(F)(F)F 15964,CC1(F)CN(C(c2n[nH]cc2Cl)=O)CCN(C(C2COC(=O)C2)=O)C1 15965,CN1CCCCC1C(=O)NC(CNC(c1ccc(OC2CC2)cc1)=O)CO 15966,C1(C(=O)NC2(CF)CCN(C(C3C(OC)(OC)CC3)=O)C2)CC2(CCCC2)CO1 15967,N1(C(C2C(C)C2)=O)CC(NC(=O)C(=O)N(C)C)C2(CCOCC2)C1 15968,Cc1cc2c(C(N3CC4CC(NC(C5CCC(C)CC5)=O)C3C4)=O)nccn2n1 15969,C(CC1=CCCCC1)NC(c1c[nH]nc1-c1ccc(Cl)cc1)(c1nnnn1C)C 15970,C1(C)(NC(C(C(C)(C)O)NC(c2ncc(F)cc2F)=O)=O)CCCC(C)(C)C1 15971,C1(C(N(C2CCCC(NC(=O)COCCCF)C2)C)=O)Cc2cccnc2C1 15972,C12(C(=O)NCC(C(=O)OC)Cc3ccccc3OC)CCCC(C1)C(=O)NC2 15973,C1(NC(=O)NC2CN(C(CCC)C)C(=O)C2)CCOCC1(C)C 15974,Cc1nc2cc(F)ccc2cc1C(=O)NC(C)CNC(c1ccnn1C)=O 15975,S(=O)(=O)(c1ccc(NCCCC2CC2(Cl)Cl)cc1Br)NCc1cncc(OC)n1 15976,c1(C(N2C(C(C)(C)C)CCOCC2)C(=O)NCC2CC2)c[nH]c2ccc(Cl)cc12 15977,C1(N2C(C3(N(c4cc(CC)ncn4)C4CCC4)CC3)CCC2)CCC(=O)NC1=O 15978,CC1(C)CC(C(=O)NC(c2cscn2)CO)CN(C(c2cnc(=N)[nH]c2)=O)C1 15979,C1(NC(CCOCCOC)=O)C(C)(C)C(NC(c2cc(F)n[nH]2)=O)C1(C)C 15980,N1(C(C2N(C)C(=O)NC2)=O)CC2(CC2)CC1CNC(=O)CCC(F)(F)F 15981,C(C#CC(F)(F)F)NC(C1CCCN1C(=O)CNC(=O)NC1CCCC1)=O 15982,N1(C(C2CCC(C)C2)=O)CCC2(CCN(C(C3(O)CCOCC3)=O)CC2)C1 15983,C1(C(=O)OCC)CC(NC(=O)NCc2ccnn2CC(F)F)CCO1 15984,Cn1c(C(=O)NC2CCOC(C(N3CCC(NC(=O)NC)CC3)=O)C2)cnc1S 15985,Cc1cc(F)cc2[nH]c(C(=O)NCC34CC3CN(C(=O)C3=CCCS3)C4)cc12 15986,C(=O)(C1=CCN(C(C2CC(=O)N(OC)C2)=O)C1)NC(CC)CCCO 15987,c1(C(=O)NC(C(=O)NC(C#C)Cc2ccco2)C2CC2)cc([N+](=O)[O-])c[nH]1 15988,C1(C(=O)NCC(C)CN(C(=O)C(F)CC2CCCCC2)C)CCC2(CC1)CC2 15989,c1(CCC(=O)NCCOCCN(C(C(c2cncnc2)C)=O)C)n[nH]cc1Br 15990,c1(C(=O)NCCC2CC(NC(CC=C)=O)C2)cn(-c2ncccn2)cn1 15991,S(=O)(=O)(c1ccccc1)NCC(N1C(C(CNC(C(C)SC)=O)(C)C)CCC1)=O 15992,C1(C(=O)NC2C(NC(Cc3nc(C)c(C)o3)=O)CC2)C2CCC3C(C2)CC13 15993,C(=O)(C(CC(C)C)N(C)C(C1CNC(=O)N1)=O)N(C(CC)C1CC1)C 15994,N1(C(CC(C=C)(C)O)=O)CC2CCC(C1)C(NC(c1cnc(OC)c(C)n1)=O)C2 15995,C1(C)(CCCC(=O)NCC2(CNC(C3(C)CCC3)=O)CC2)NC(=O)NC1=O 15996,N=c1nc2c(c[nH]1)CCN(N1CCC(c3nc4ccccc4s3)CC1)C2 15997,N1(C(C(c2ccc(F)cc2F)(C)C)=O)CCCCCC(NC(C2CC2(F)F)=O)C1 15998,C1(C(=O)NCC=CC(=O)NC2(CC=C)CCCC2)CC12CCOC2 15999,CC(O)C(C)C(=O)N1CCCC1CN(N1CCCCC1)C.CCO 16000,C1(NC(C=CC(C)(C)C)=O)CCNCC1c1cccc(F)c1 16001,C(=O)(CC(C)(O)C(F)(F)F)NCC(C)NC(CCC(=C)Cl)=O 16002,C1(OC)CC(CNC(=O)CCC=C(C)C)N(C(=O)CC(C)n2ccnc2)C1 16003,C1(NC(C(C=C)(C)CC)=O)CCN(C(c2ccc(OCOC)cc2)=O)CC1(C)C 16004,N1(C(c2cc(C)nc(C)n2)C(=O)NC(CC)C)CCc2ccc(F)c(Br)c2C1 16005,N1(C(C23COCC2CN(Cc2cccnc2)C3)=O)CCC(C2CCOCC2)C1 16006,N1(C(c2cnc(C(C)=O)s2)=O)CCCC(C)(NC(C2C(F)(F)C23CCC3)=O)C1 16007,c1(CN(C(CCc2c(C)cccc2)=O)C)ccc(S(=O)(=O)C(F)(F)F)cc1 16008,c1(CC(=O)NC2CC2NC(=O)C=CC2CCOC2)cc(C2CC2)no1 16009,N1(C(c2c(CC)c(C)ccc2)=O)CCCC12CCN(C(C1CCC(F)(F)C1)=O)C2 16010,c1(C(N2CCC(C)(NC(c3cnn(C)c3F)=O)C2)=O)ccc2ncncc2c1 16011,n1(CC)ccc(=NC(=O)C(=O)NC2CC23CCOCC3)[nH]1 16012,N=c1c(C(=O)Nc2cccc(N(C(=O)CCF)C3CCC3)c2)c[nH]cc1Br 16013,c1(C(CCC(=O)N2CC(NC(C(CCCC)C)=O)C2)=O)ccc2c(c1)CCCC2 16014,C(CC(C(=O)Nc1cn(C)nc1Cl)NC(c1ccnn1CC)=O)=CC 16015,CCCC(C)(O)C(=O)NCC1CCCC1C(=O)NC1CN(C)CCC1O 16016,c1(C(=O)NCC2(COC)CCN(C(C3CCC3C)=O)C2)cc2ccccn2n1 16017,S(=O)(=O)(c1cccc(NC(=O)NCc2cc(=O)cc[nH]2)c1)N1C(C)CCCC1 16018,C(=O)(CS(N)(=O)=O)NC1C(CNC(C(CC2CCC2)OC)=O)CCC1 16019,c1(C(N2CC(C)CC(NC(CC3(OC)CC3)=O)C2)=O)cc2n(n1)CCCO2 16020,C1(NC(c2nc(-c3ccccc3F)no2)=O)(CO)CCCOC1 16021,C1(C(=O)N(C)CCNC(c2ccn(C(C)C)n2)=O)(CC)CCOC1 16022,CN1CC(C(=O)NC2CC(F)(CNC(=O)Cn3cnc(=N)[nH]3)C2)C(C(F)(F)F)C1 16023,C12(C(=O)NCC3N(C(C4CC(OC)C4)=O)CC3)CCC(O)C1CC2 16024,C1(CN(C(=O)CC2CCOC2)C)CN(C(=O)CCc2ccc[nH]2)CC12CC2 16025,CC1CCC(c2nnnn2C2(C)CC2)(NCCCc2ccccc2Br)C1 16026,C(c1cccc(F)c1)=CC(=O)NCC(C)(F)CNC(=O)CC12CCCC1C2 16027,C1(c2cccc(OC)c2)CCN(Cc2nnnn2CC(F)(F)F)C1(C)C 16028,CC(C)(C)C(C(=O)N1CCC(O)CC1C1CC1)Oc1ccccc1F 16029,N1(C(CC(CC)OC)=O)CC(C)(C)C(NC(c2cnc(Cl)s2)=O)C(C)(C)C1 16030,Cc1cccc(C(=O)NCCCCCNC(C2(C3CCCCO3)CC2)=O)c1O 16031,N(C(=NCc1c(Br)cncc1Br)N1CC(O)C(C)(C)C1)C(CC)C 16032,C1(C(N)=O)CCCN(CCCCO)C1=O.c1(NC)ccc(OC(F)(F)F)cc1 16033,C1(CN(C(CN(CCC#C)C)=O)C)CCCN1C(=O)C(C)NC1(CO)CCCC1 16034,C(=O)(C(C)CC(F)F)N(C1CCN(C(c2ccc(C(C)C)s2)=O)CC1)CC#C 16035,N1(C(CCc2n(C)ccn2)=O)CCC2(CC2C(=O)NCC2CC3C=CC2O3)C1 16036,Cc1cc(C(=O)NC(C2(C(=O)NCC3C4CCCCC34)CC2)C)sc1C 16037,CC1CC(NC(=O)C(C)C(=O)OC(C)(C)C)CCN1C(=O)CN1CCS(=O)CC1 16038,c1(C(=O)NC(CC(C)NC(C(CN(CC)CC)F)=O)C)cc(S(N)(=O)=O)sc1C 16039,N1(C(C(CC=C)CNC(=O)C(CC)CCCC)=O)CC2(CCN(C)CC2)C1 16040,C(CCC(=O)NCCC(C)NC(=O)CN(C(=O)C(C)C)C)=CCC=C 16041,C1(NC(C(C)(C)n2cc(Cn3cncn3)nn2)=O)CC2CCCN2C1 16042,CC(C)C(C(=O)NC(C)CCN(C)C)NC(C1(CO)CC(C)(C)C1)=O 16043,CC1C(NC(c2c[nH]nc2C(F)F)=O)CCCN1C(=O)Cc1cnccc1Cl 16044,c1(C(=O)NCC2CCN(C(C3CCCS3)=O)CC2)cccc2ncccc12 16045,C1(CNC(=O)Cc2cnn(-c3ccccc3)n2)C2CN(C(c3ccsn3)=O)CC12 16046,[N-]=[N+]=NC1CN(C(c2cc(C#N)cs2)=O)CC1NC(=O)CCN1CCNC(=O)C1 16047,N1(CC)CCC(S(=O)(=O)Nc2cnc(N3CCC(C(N)=O)CC3)nc2)C1 16048,C1(CNC(CS(CC)(=O)=O)=O)CN(C(=O)CC2(COC)CC2)C2COCC2O1 16049,C=CCCN=C(NCCC(c1ncc(C)s1)C)NC1CCS(=O)(=O)C1 16050,c1(OC)ccc(C(N2CC(C)(NC(C3CC3c3cnc(C)nc3O)=O)C2)=O)c(Cl)c1 16051,N1(C(CCS(C)(=O)=O)=O)CCC2(CC1)CC(NC(C1CCCO1)=O)CO2 16052,c1(CC)nc(C(C(=O)NCC(C)C)N(C)Cc2csc(C(F)(F)F)n2)cs1 16053,CN1CCN(C(=O)C2=NOC(CNC(=O)CN3CC(C)(C)C3)C2)CCC1=O 16054,C(=O)(C1CCc2ccccc21)NCC(C)N(C)C(c1ccc(CO)cn1)=O 16055,CN1CC(O)CC1C(=O)NCCNC(=O)CCCc1ccsc1 16056,CC1(C)CCC(CNC(C2CCCC2CNC(c2ccc(F)cn2)=O)=O)CC1 16057,C=C=CC(C)C(=O)N(CC=C)Cc1c[nH]nc1C(=O)N(C1CCCC1)C1CC1 16058,Cc1cc(CC(N2CC(C(=O)NC(=O)CCCN(C)C)C2)=O)c(C)s1.C1C=CC1 16059,c1(CC)cccc(C(=O)NC2CCC(N(C)C(c3cc(OC)nn3C)=O)C2)c1 16060,c1(C(=O)NCC(CNC(c2c(C)n(C3CC3)nc2)=O)C)cc(S(N)(=O)=O)cn1C 16061,c1(C(=O)NC2CCCC(N(C(C=CC=CCC)=O)C)C2)c(F)cc(OC)cc1Cl 16062,C1(NC(CCSCCC)=O)CC(O)CN(C(c2cnc(CC)s2)=O)C1 16063,C(=O)(C1CCc2c(Cl)cccc21)NC1CCN(CC2(NC(C(C=C)O)=O)CC2)CC1 16064,C(=O)(CC(=O)NC1CCC1NC(c1nnc(C(C)C)s1)=O)OC 16065,c1(C(N2C(C)CCC(NC(c3ccc(C(N)=O)o3)=O)C2)=O)ncn2ccccc12 16066,C1(NC(C2(CC#C)CC=CCC2)=O)CC2CCC(C1C)N2C(=O)Cc1cscn1 16067,C1(C(N2CC(OC(=O)NC)C2)=O)CN(C(=O)C(C)(C)OC)CC1F 16068,C12(C(=O)NCCC3CCCC(C)C3)CC(CCO1)N(C(C1CCC1C#N)=O)C2 16069,CC(CC(N)=O)C(=O)N1CC(CNC(c2ccnn2C(C)(C)C)=O)C2(CC2)C1 16070,c1(CC)nc(C(=O)NCC2(CN(CCC(C3CC3OC)=O)C)CC2)co1 16071,c1(C(=O)NC(C(=O)NCC(O)CC2CCCC2)C2CCCO2)ncoc1C1CC1 16072,Cc1cccc(F)c1CC(=O)NC1CC(NC(C2C3CCC(F)(F)C23)=O)C(O)C1 16073,N1(C(C=C2CCN(C)CC2)=O)CCC(NC(C23CCN(CC2)C3)=O)CC(C)(C)C1 16074,CC1=C(C(=O)NC2CCN(C(=O)C=C(C3CC3)C3CC3)C(C3CC3)C2)CCC1 16075,C1(F)(CNC(C2C(=O)NCC2)=O)CCN(C(c2cccc(OC(F)(F)F)c2)=O)C1 16076,C1(NC(c2nncc(CCC)c2)=O)CCN(C(c2cc(OC)ns2)=O)CC1C 16077,c1(NC(C)=O)cccc(-n2nc(C3CC34CC4)nc2-c2coc(C)n2)c1 16078,CCCCS(=O)(=O)NC(C)C(=O)NC1CC(CNC(=O)C(C)(C)NC(C)=O)C1 16079,CC1=C(C(=O)N(C)CCOCCNC(=O)CCc2cncc(Br)c2)CCC1 16080,N1(C(CCCC)=O)CCC2(CCC2)C(CNC(c2cnc(C)nc2C2CC2)=O)C1 16081,CC1(C(=O)NCC(O)CCNC(c2ccc(C3CCC3)cc2)=O)CCC(=O)NC1 16082,c1(CCC)cc(C(N2CC(NC(C3(C(N)=O)CCC3)=O)C(O)C2)=O)ccn1 16083,O=C(CCCc1cccs1)NCC(O)CCNC(C1(F)CCC1)=O 16084,c1(CC(N2C(CNC(=O)C=CCF)CCC(C)C2)=O)csc2ccccc12 16085,C1(NC(C2CCC(C)C2)=O)CCOC2(CCN(C(C3(O)CCSC3)=O)CC2)C1 16086,c1(C(N2C3CC(CNC(c4nc(C)oc4)=O)C2CC3)=O)cccc2sncc12 16087,C1(NC(CCCCC#C)=O)CN(C(c2cc(F)c(N)cc2F)=O)C2CCCCC12 16088,C12(C(=O)N)CC1COC21CCC1.c1(CC2(NC(CN(C)C)=O)CC2)cccs1 16089,Cc1cc(C(=O)NC2(c3nc4ccccc4[nH]c3=O)CCC2)n2nc(C)cc2n1 16090,C(=O)(C(F)(F)C(C)O)NCC(C1CCCCC1)NC(C(CCC)O)=O 16091,C1(NC(c2cc(C)cc(C)c2)=O)CN(C(C2CC2C(N)=O)=O)C2CCCC12 16092,CS(=O)(=O)C1CC(C(=O)NC23CC2CN(C(=O)C(C#N)C2CC2)C3)C1 16093,CCCCCCCC(=O)N1CCC(NC(=O)C(C)(C)COC)CC1C 16094,c1(CNC(C2C(C)CN(C(=O)C(C3CC3)C3CC3)CC2)=O)ccc2c(c1)CCC2 16095,C1(NC(C(C)c2ccsc2)=O)CCC12CN(C(c1ccc(CO)cc1)=O)C2 16096,C(CC1CC1)(C(=O)NOCCn1ccnc1)NC(C1CC2CCC1O2)=O 16097,C(=O)(C(CC)(CC)OC)NCCc1cc(C(N2C(C)(CCC)CC2)=O)no1 16098,N1(C(=O)OC(C)(C)C)CCC(O)(C(N2CCC(OC)C2)=O)C1.C(=O)(CC(F)(F)Cl)N 16099,N1(C(C=CCOCCOC)=O)CC2CC(O)C1C2NC(C1CC(n2ccnn2)C1)=O 16100,C(=O)(C1=NNC(=O)CC1)NCC1CC(NC(C(C(C)(C)C)N(C)C)=O)C1 16101,c1(C(=O)NCC2(C(=O)NCc3ncc(C)nc3)CC2)cccc(O)c1C 16102,CC(C)CCC(=O)C(=O)N1CCC(C(=O)N(C)CC2CCCC2O)CC1(C)C 16103,c1(C(N2CC(NC(COCCC#C)=O)C(C)(C)CC2)=O)cc(S(N)(=O)=O)c(C)s1 16104,C1(NC(c2nc(COC)[nH]n2)=O)CCN(C(C2CCC3CC3C2)=O)C(C)C1 16105,Cc1ccc(C(F)(F)C(=O)NC(C2CCCN(C(=O)CSCC(N)=O)C2)C)cc1 16106,c1(C(=O)NC(CNC(CSCCN(C)C)=O)CO)cc(N)c(Cl)c(O)n1 16107,CCC(CC)CCC(=O)NC(C1CCN(C(=O)Cn2cnc(C(F)(F)F)c2)C1)(C)C 16108,C1(C(=O)NC2CN(C(C=CCOC)=O)C2)(OC)CCCC(C)C1 16109,C1(CNC(C(CC)N(C)C)=O)CN(C)CCN1C(C1C(c2ccccc2)C1C)=O 16110,C1(CC)CCN(C(=O)CONC(=O)CC2OCCCO2)CC1O 16111,CCCCCCCCNC(=O)C(=O)NC(C)CNC(=O)CC1CC(SC)C1 16112,c1(C(=O)NC(c2cn(C)nc2)C(F)(F)F)nc2c(o1)CCSC2 16113,C1(C(=O)NCC=CCNC(=O)CC2CCCC2(F)F)CCn2ccnc2C1 16114,c1(C(COC)NC(=O)C(c2ccnn2C)O)ccccc1F 16115,C1(NC(C(C(C)C)SCC)=O)CC2CCC(C1)N2C(c1ccc(C(C)(C)C)[nH]1)=O 16116,N1(C(C=C(COC)C)=O)CCC(C)CC1C(=O)NC(COC)C(C)C 16117,C(C1CCc2ncnn21)N(C1CCN(C(CC(=C)C)=O)C1)C 16118,C12(NC(c3c(OC)nn(C)c3)=O)CCOC(CNC(=O)CCOC(C)=O)(C1)C2 16119,Cc1ccc(C(=O)NC(C)C(CO)NC(C2CC(S(C)(=O)=O)C2)=O)cc1C 16120,C1(C(CC)O)CCCN1C(=O)C#CCNC(c1ccoc1Cl)=O 16121,c1(C(C)NC(C(C)N(C(=O)COC2CCCC2)CC)=O)ccc(C)cn1 16122,Cn1ccc2c(C(N3CCN(C4CCCCC4O)CC3)=O)cccc12 16123,C1(CC)CN(C(C2(F)CCOC2)=O)CCN1C(=O)CCCCc1ccc(Cl)cc1 16124,n1(CC)cc(CNC(=NCCSC2CC2)NCCSC(C)C)ccc1=O 16125,C1(NC(=O)C(C2CC2)C2CC2)CN(C(C2CC(=O)N(C3CN(C)C3)C2)=O)CC1F 16126,C12(C(=O)NC3CC4(C(C(N(C)Cc5c(C)n[nH]c5)=O)C4)C3)CC(C)(CCO1)C2 16127,N1(C(Cn2c(C)ccc2C)=O)CCN(C(=O)COC2CC2)C(C2CCCC2)C1 16128,c1(OC)cc(C(N2CC(NC(=O)CC3CC(F)C3)C(C)(C)C2)=O)nnc1C1CC1 16129,C(=O)(C(C)(C)C(=O)NCC1(O)CCN(C(=O)CC2CC(C)(C)CO2)C1)NC 16130,C(c1ccc(F)cc1)=CC(=O)NCC1CC(NC(c2cccnc2O)=O)C1 16131,C12(CC(=O)NCCN(C(CCCCOC)=O)CC(C)O)CCCN1CCC2 16132,C(CC(C(C)C)NC(=O)C(C)(F)CC1CCCC1)N(C(CCN(CCC)C)=O)C 16133,c1(C(=O)NC(C2CCN(C(Cc3ncc(CC)[nH]3)=O)C2)C)cc(F)cc(F)c1N 16134,CS(=O)CCC(=O)NCCN(C(=O)COCC1(F)CC1)Cc1ccc(Cl)nc1 16135,CC(C)CC(O)CC(=O)N1CCC(N(C(=O)CC(C)C2CCCC2)C)C1 16136,C(=O)(CCS(N)(=O)=O)NCC1N(C(c2cccc(C(C)C)c2)=O)CC=C1 16137,c1(NC(C(C2CN(C(c3cc(CCC)[nH]n3)=O)C2)O)=O)ccc(C)c(C)c1 16138,c1(C(=O)NC(C)CNC(c2cnsc2)=O)cccc(-c2nc(=O)o[nH]2)c1 16139,C1(CC#C)(C(N2CCC(N(C(=O)CC3CCCN3C(=O)OC)C)C2)=O)CCCCC1 16140,CC1CC(C(=O)N2CCC2CNC(c2cncc(-c3cccc(F)c3)c2)=O)=NO1 16141,CC(C)(C)C(C(=O)NCCc1nc[nH]n1)NC(c1ccnnc1)=O 16142,c1(CC(N2C(CN(C(c3cnc(C)s3)=O)C)CCC2)=O)ccc2[nH]ccc2c1 16143,CC1CCCN1CC(=O)NCC1CCC1C(N1CCC(N2CCC2)C1)=O 16144,n1(CC(=O)NCC(CNC(CC(n2ccc(C)n2)C)=O)O)cc2ccccc2n1 16145,C#CCCC(O)C(=O)Nc1cccc(NC(=O)C(c2ccc(F)cc2)OC)c1 16146,n1(CCC)nc(C)cc1C(=O)N(C(C)CN(C(=O)C(C)CC)C)C 16147,N1(C(CSCC)=O)CCC2(CCN(C(c3ccc(OC)nc3)=O)C2)C1 16148,Cn1cc(C(=O)NCC2(C)CCCC2NC(C2CCOCC2)=O)c2ccccc12 16149,c1(COC)ccc(NC(C2(CCNC(=O)CC3COC(=O)N3)CC2)=O)cc1 16150,c1(C(=O)NC(CC)(CNC(=O)C(C)(O)CC)CC)ccc2nc(N(C)C)oc2c1 16151,CC1(C)CN(C(=O)CC2OCCC2(C)C)CC1C(=O)N(c1ccc(O)nc1)CCO 16152,C1(NC(c2c(C)nc(CO)s2)=O)CCCC12CN(C(C1CN(CC(C)C)C1)=O)C2 16153,C#CCC(C(=O)N1CCCC1(CC=C)C(N1CC(F)C(F)C1)=O)C1CC1 16154,c1(C(N2CCOC(CCO)C2)C(=O)NC(C(=O)OC)C)ccncc1Cl 16155,C1(CNC(CN2C(C)CC2)=O)CCC2(CCN(C(c3cccc(N)n3)=O)CC2)O1 16156,CC(C)CC(C(=O)N1CC(N2CCOC2=O)C1)NC(c1ccc(F)cc1F)=O 16157,c1(NCC(CNC(C2CC(C)(C)C2)=O)F)ncnc2cccc([N+](=O)[O-])c12 16158,CC(C(=O)NCC1=CCN(C(=O)C(c2ccccc2Cl)(F)F)CC1)C(C)(C)C 16159,C1(C(N(CCNC(CCOC(CC(C)C)C)=O)CC2CC2)=O)CCCCCC1 16160,c1(C(=O)NC(CNC(=O)CC2(O)CCOC2)C2CC2)cccn2ccnc12 16161,N1(CC)CCCCC1C(N1CC(C(=O)NC2CCS(=O)CC2)C(F)C1)=O 16162,CC(O)C(=O)N1CC(C(=O)NCC2(CO)COC2)C1 16163,c1(C(N2CCCC(C(C)NC(Cc3c(C)scc3)=O)C2)=O)cc2ncccc2[nH]1 16164,n1(CCCOC)nnnc1C(c1ccc(C(N)=O)o1)NC(COC)CCOC 16165,C(=O)(CC(C)C(=O)N(CC(=O)NCC1CC(C)C1)C1CC1)OC 16166,c1(-c2cc(CN(C)C(C34COC(CF)(C3)C4)=O)on2)ccc(Cl)cc1Cl 16167,N(C(=NCCC(C)C)N1CCc2ocnc2C1)CC(c1c(C)noc1C)C 16168,C1(C)(C(=O)NC(CCCNC(c2c(CC)n(C)nn2)=O)C)CC2(C1)CC2(F)F 16169,c1(CNC(c2c(OC)ccs2)=O)ccc(NC(=O)C(C)OCC2CCCO2)cc1 16170,c1(C(=O)NCC23OCC(NC(C4C(C=C)CC4)=O)(C2)C3)cc([N+](=O)[O-])ccc1Cl 16171,C(=O)(CC1OCCc2ccccc21)NC12CCCN(c3c(OC)cncn3)CC1C2 16172,N1(C(CN(C)C(C2CCC(C3CC3)C2)=O)=O)CCCCCCCC1 16173,C1(C(=O)NCCCN(C(C(C)NC(COC)=O)=O)C)COCC(C)(C)O1 16174,C1(NC(C2CC3(CCCO3)C2)=O)CN(C(c2cncc(F)c2)=O)C2(CCCC2)C1 16175,C(=O)(C#CC1CCCOC1)N1CCOCC(C)(CNC(C=CCCC)=O)C1 16176,N1(C(C2CC(=C)C2)=O)CC2C3CCC(C2C1)N(C(=O)COc1ccc(Cl)cc1)C3 16177,N1(C(C(C(CC)C)NC(C)=O)=O)CCC2(CCC2)C(NC(C2CCC(=O)N2)=O)C1 16178,C1(NC(CNC(=O)NC)=O)COCCC1NC(c1scc(C)c1Br)=O 16179,n1(-c2ccc(C(=O)OCC)cc2)c(C)cc(CN(CC(F)F)C(C)COC)c1C 16180,C(=O)(C1=NOC(C)(C)C1)N1C(C(C)C)(C(=O)NCCC2CCCN2C)CCC1 16181,N1(C(=O)C=Cc2ccco2)CC2(CNC(=O)CC3(O)CCCCC3)CCC1C2 16182,C(=O)(C1=NNC(=O)CC1)N1CCN(C(c2c(C)nn(C)c2C)=O)C(C2CC2)C1 16183,N1(C(c2c(CC)ccs2)=O)CC2CCC2(CCNC(=O)CCCOC)C1 16184,c1(C(=O)NC2CCCN(C(=O)C=Cc3cnccn3)C2)cccc2nc(Cl)sc12 16185,c1(C(CC(=O)N(CC(C)N(C(CCNC(C)=O)=O)C)C)C)ccc(F)c(F)c1 16186,C1(C2CCCN(C(c3c(C4CCC4)cnn3C)=O)C2)(NC(CC(C)C)=O)CC1 16187,N1(C(c2nscc2Br)C(=O)NCCC2(C)CC2)CCC(=O)N(C)CC1 16188,Cc1noc(C)c1CC(C)C(N1CCN(CCNC(C2(CCO)CC2)=O)CC1)=O 16189,N1(C(C2C(C)(C)OC(=O)C2)=O)CC2(C1)CN(C(c1cnsn1)=O)CCO2 16190,O=c1nc(O)c(C2CC(NCCc3nc4c(s3)CCCC4)C2)cn1C1CC1 16191,CC1CCN(C(c2cc(C3CC3)ccn2)=O)C1CNC(=O)C=Cc1cc[nH]c1 16192,CCC(CC)CCC(=O)N1CCN(C(=O)CC(O)CC(C)C)CCC1C 16193,C1(N(C(c2ccc(C)cc2)C(=O)NCCC#N)CCC)CCN(C)C1(C)C 16194,C(=O)(C1CCc2nccn21)NC(C(=O)NC1(CC)CCCC1)CC1CC1 16195,C1(C)C(=O)NN2CCN(CC2)c2cccc(c2)S1.S(=O)(=O)(c1cn(C)nc1C)NC 16196,N1(C(C(CCC)F)=O)CCN(C(=O)Cn2cc(C3CC3)cn2)CC1C1CCC1 16197,Cc1cnc(C(=O)NC2CCC(N(C)C(c3c(N)cnn3C)=O)CC2)c(C)c1 16198,C1(NC(CCc2n(C)c(S)nn2)=O)CCN(C(=O)C2=CCOC2)C12CC2 16199,N1(C(C(C)c2ccsc2)=O)CCCOC(CNC(=O)CC(O)C2CCCC2)C1 16200,C1(NC(CCCN(CCC)CCC)=O)CCN(C(=O)CCC(=O)OC)C1CC 16201,C=CCC(C)(C)C(=O)N1CCCC(F)(C(=O)NCc2nnc(O)o2)C1 16202,N1(C(c2noc(C(C)(C)C)n2)C)CC2C(C(=O)NCc3cccc(Cl)c3)C2C1 16203,C1(CN(C(C(c2ccc(CC)s2)=O)=O)C)CCCCN1C(=O)CCSC 16204,C1(C(N2C(CC)CC(C)C2)=O)CCC2(CC2)N1C(C1CC1C#N)=O 16205,c1(CC)ccc(C(=O)NCCCC2CCCN2C(=O)C(F)C2CCOC2)cc1Cl 16206,C12(OC)CCC3(C1)N(C2)C(=O)NOC(C)C(=O)N3.C(C)(C)(C)NC(C)=O 16207,C1(C)(CNC(C=C=C(C)C)=O)CN(C(=O)CC2CCC(=O)N2C)CCO1 16208,N1(C(C(C=C)O)=O)CC(NC(=O)CC2CCCCCC2)CC2(CCC2)C1 16209,c1(CCC)cccc(OC(=O)Cc2csc(Cl)c2)c1 16210,N1(C(C(CN(C)C)O)=O)CCC2C(CCCN2C(C2CCCCN2C)=O)C1 16211,C1(CC)CCC(NC(=O)CC2(N(C)C(C3CCCN3C3CC3)=O)CC2)C1 16212,N1(C(CC2(C)CCOC2)=O)CCC2(CC1)CC2C(N1CC2CC2C2CC12)=O 16213,C12(CNC(C3C(C)(C)C3)=O)CCC(C1)N(C(=O)CCCN1CCCC1)C2 16214,Cc1ncc(C(N2CC=C(CNC(C3CCC4C3C4(F)F)=O)CC2)=O)cc1C#N 16215,c1(NCC(C)CNC(=O)C#CC2(C)CCCO2)cccc(CO)c1[N+](=O)[O-] 16216,N1(CC(=O)N(C(=O)C(F)F)NC(C)C)CCN(CCc2cccs2)CC1 16217,c1(COC(C(=O)NCC(C)CN(C)C)C)ccccc1 16218,C1(NC(C#CC(C)C)=O)CN(C(=O)C(C2CCOCC2)=O)CC12CCOCC2 16219,C(CC(C)C(=O)N1CC(C)(NC(=O)C(C)NC(=O)OC2CCCC2)C1)OC 16220,C=CC1(C(=O)N(C)Cc2ccccc2F)CCN(C(c2ccsn2)=O)C1 16221,N(C1CCCc2occc21)C(C(CC(C)C)NC(C1CCC(=O)O1)=O)=O 16222,c1(OC)cc(CCC(=O)NC(C)CCNC(=O)CC(C)OC)ccc1F 16223,Cc1cc(C)n(C(C)C(=O)NC2CC(NC(C3CCC(F)(F)C3)=O)C2)n1 16224,c1(C(N2CCN(C(c3n(C=C)nnc3)=O)C(CCO)C2)=O)cc(F)cc(N)c1F 16225,N1(C(c2cc(C)no2)=O)CCN(C(=O)CN2CC(=O)NC2=O)C(C(F)F)C1 16226,Cc1ccc(C)c(C(N2CC(C(F)(F)F)OC(CNC(=O)C(F)(F)CO)C2)=O)n1 16227,Cc1cc(N2CCC3NC(=O)CCC3C2)nc(=NCC(F)(F)Br)[nH]1 16228,c1(C(N2C(C)CC(CNC(c3ccncc3F)=O)C2)=O)cc2c(O)cccc2[nH]1 16229,c1(OC)cc(O)c(C(=O)NCC(C)N(C)C(C2CC(OC(C)C)C2)=O)cc1OC 16230,N1(C(CC2CCN(C(C(C)=CC=C)=O)C2)=O)CCC(C)(C)C(CO)C1 16231,c1(COCC(=O)NCC=C(C(=O)OCC)C)ccc(F)nc1 16232,C12(NC(c3cc(C)nc(O)c3)=O)CCCC1N(C(=O)CCCCC(F)F)CCC2 16233,c1(CC)cccc(C(=O)NCC2(C(C)NC(c3cnc(C)s3)=O)CC2)c1 16234,C1(NC(C=CC(=O)OC)=O)CC2CN(C(=O)C=CC(=O)NC3CC3)CCN2C1=O 16235,CC1CCN(C(c2cn(C)nc2C(C)(F)F)=O)CCN1C(C1CNC(=O)C1)=O 16236,CC1CC(CNC(c2cn(C3CC3)nn2)=O)CN1C(c1cn(C)c(O)n1)=O 16237,Cc1nn(C(C)(C)C)cc1C(=O)NC1CCCCC1CNC(c1cocn1)=O 16238,N1(C(C2(C)CCOCC2)=O)CCC(F)(CNC(=O)Cc2ccc(Cl)c(F)c2)CC1 16239,c1(C(=O)NC2CCN(C(C3N(C(=O)OCC)CSC3)=O)C2)c[nH]nc1[N+](=O)[O-] 16240,c1(C(N(CCC(C)NC(C2CC(OC)C(OC)C2)=O)C)=O)c(F)cc(F)cc1F 16241,C1(NC(C(C)c2cccs2)=O)CN(Cc2ccccc2CCBr)CC1C#N 16242,c1(C(=O)NCC(CNC(c2cc(F)cc(F)c2)=O)CO)cnc2cc[nH]c2c1 16243,N1(C(=O)NC(c2ccncc2)CC=C)CCCc2cc(Br)cc(F)c21 16244,C1(CC=C)CCN(C(=O)C(=O)NCc2ccc(Nc3ccc(Br)cc3)cc2)C1C 16245,C#Cc1ccc(C(=O)NCC2CCN2C(c2nocc2CC)=O)o1 16246,c1(C(=O)NCC2(NC(c3cnc(CC(C)C)[nH]3)=O)CCCC2)cc(O)cc(=O)o1 16247,C1(C(=O)NCCN(C(=O)CC(C)(C)c2ccccc2)CCC)CC(O)C1(C)C 16248,CC1(C)CCN(C(=O)CSCC(F)F)CC1C(N1CCCC1C1CCOC1)=O 16249,CCCCCC(C(=O)N(C(C)CNC(=O)CCCc1ccccc1)C)C(C)C 16250,N1(C(C2CN(C(C(CCC)=CCC)=O)CC(C)C2)=O)CCC(=O)N(C)CC1 16251,C(C(CC(C)C)C(=O)N1CC2=C(C1)CN(C(=O)CC1CC13CC3)C2)OC 16252,c1(C(=O)NC)cc(=NC(=O)C2(Sc3ncccc3C)CC2)[nH][nH]1 16253,c1(C(=O)NC23CC(CNC(CCOC)=O)(C2)OC3C)snc2ccccc12 16254,C1(NC(c2c(C)ncnc2)=O)CC2CC1N(C(c1ccc(F)cc1Br)=O)C2 16255,c1(CNC(C(C)N(CCC)C(C2CC2(C)C(F)F)=O)=O)cccc(F)c1C 16256,C=Cc1cccc(-c2cn(CC(N3CCCC3c3ccccc3SC)=O)nn2)c1 16257,C1(CC)CN(C(C2COC2)=O)CC1NC(c1ncccc1Br)=O 16258,c1(N2C3CCC2CC3)nc(SC)nc(Cl)c1C.c1(CC(=O)OC)ccc(F)cn1 16259,C1(CC(N2CC(C(CNC(CCN(C)CC)=O)O)C2)=O)CCCC1O 16260,C(=O)(C(C)CC(F)(F)F)N(C1CN(C(c2cc(C)cc(N)c2)=O)CC1(C)C)C 16261,CCS(=O)CC(=O)N1CC(CNC(c2ccnn2C2CCCCC2)=O)C(C)C1 16262,N(C)(C1CCCCC1)Cc1cn(C(C(=O)NC(CC)CN(C)C)(C)C)nn1 16263,N1(C(CCN(C)CC)=O)CCC2CCN(C(=O)CCNS(C)(=O)=O)CC12 16264,c1(NC(C2N(C(CC3CC(OC)C3)=O)C(C)C2)=O)ccc(Cl)cc1C 16265,c1(NC(C2CC(Nc3ncc(C4CC4)cn3)C2)=O)cnc(Br)c(Cl)n1 16266,C1(C(=O)NCC2CC(NC(c3cnn(C)c3C3CC3)=O)C2)CCC2C1C2(F)F 16267,C(CCC(=O)NNC(=O)c1ccc(F)cc1Br)OC 16268,c1(CC(N2CC(NC(C(CC)O)=O)C(CO)C2)=O)cnc(OC)cc1OC 16269,c1(NC(C2CCN(C(C3(F)CCCCC3)=O)C2)C)ncnc2sccc12 16270,Cn1nncc1CC(=O)NC1(C(=O)NCCSCCO)CCSC1 16271,N1(C(C(CSC)O)=O)CC=CC(C(=O)N(C)CCOCCO)C1 16272,c1(C(C2(O)CN(C(=O)C(O)C3CC3)C2)C)cccc2[nH]cc(CC(=O)OC)c12 16273,C1(C(=O)NCC(C)(C)NC(CCc2c(C)nccc2)=O)CCc2ncncc2C1 16274,C1(NC(c2c(C)cc(Br)o2)=O)CN(C(C2CC2F)=O)CC1S(C)(=O)=O 16275,C1(CNC(c2nc(N3CCCC3)ccc2Cl)=O)CCC(c2ccccc2)=NO1 16276,C1(C2CN(C(C3CC3Cl)=O)C2)(NC(c2ccc(COC(C)C)cc2)=O)CC1 16277,c1(C(=O)NC(CNC(=O)Cc2cnccc2Cl)CO)cc(Cl)c([N+](=O)[O-])[nH]1 16278,N1(C(C(C)(C)OC(C)C)=O)CCN(C(=O)CC(C)Sc2ccccc2)C(CO)C1 16279,C1(C(=O)NC(CNC(C(C)OCC=C)=O)C2CC2)CCC(C)(O)CC1 16280,CCCCC(O)C(C)C(=O)NCCC1CC(NC(=O)CCc2nc(CC)no2)C1 16281,N1(CC(=O)N(CCCNC(=O)C(C2CCCO2)C2CC2)C)CCNC(=O)C1 16282,C1(C(=O)OC)CC12CCN(c1nnc(CCC3CC3)n1Cc1ccccc1)CC2 16283,N1(C(c2c(CC)c(C)sc2)=O)CCC2(CC1)CC2NC(C1COCCO1)=O 16284,c1(C(=O)NC(CC)(C)CNC(c2ccnn2C)=O)nc(C)n2ccccc12 16285,C(C(C)CN=c1cc(NCCn2ccnc2C)nc(C(C)C)[nH]1)OC 16286,c1(C(=O)NCC2(O)CC(CNC(CSCC)=O)C2)cc(N)cc(C(F)(F)F)c1O 16287,Cc1cnc(C(N2CCC(C(C)(C)NC(c3cnc(N)c(Cl)c3)=O)C2)=O)cc1Cl 16288,C1(C2CC2)(NC(C=CC(C)(C)C)=O)CCN(C(c2ccc(C(=O)OC)cc2)=O)C1 16289,c1(C(=O)NCC2(F)CCN(C(CC(C)N(C)C)=O)C2)cnc2[nH]nc(O)c2c1 16290,N1(C(c2c(OC)cncc2)=O)CC2=C(C1)CN(C(=O)C(c1cnccn1)C)C2 16291,O=C(CC(C(F)(F)F)NC(C1CCC2(CC2)C1)=O)NCc1ccco1 16292,C1(C(=O)NCCc2csnn2)CC(F)CN1C(=O)CC1CC=CC1 16293,C(=O)(CCC(=O)NC1CCCCC1CNC(=O)C(=O)NCC1CC1)NCCC 16294,c1(C(N2C(CCC(=O)NCC(CNC(N)=O)O)CCC2)=O)ccc2c(c1)CC2 16295,C1(OC)CCCN(Cc2ccccc2)C1C.N12CC(CC1C)OC(=O)C2=O 16296,C1(CNC(CCSCCCC)=O)CC(C)CN(C(=O)C(F)C2CCOC2)C1 16297,CC1=C(C(=O)NC2CCCC(NC(c3c(N)sc(C)c3C)=O)CC2)CCCC1 16298,C1(C(=O)NC2C(C)N(C(=O)CC3CC4CC4C3)CC2)Cc2ccccc2NC1=O 16299,C1(C(=O)NC(CCNC(c2ccc(C(C)=O)c(F)c2)=O)C)CC2(C1)CC1(CC1)C2 16300,C1(NC(c2nn(CC(F)(F)F)cc2Cl)=O)C2CN(C(=O)C3=CCSC3)CC12 16301,c1(NC(C2CCN(C(C3C(=C)C3)=O)C(CC)C2)=O)cccc2cnccc12 16302,c1(OCC(N2C(C(C)(C)NC(C(CC)(C)C)=O)CCC2)=O)ccc(F)cc1F 16303,C(CS(=O)(=O)N=S(C)(C)=O)N(C(c1cccc(Br)c1)CN)C 16304,C1(C)(CNC(C2C(C)C2)=O)CN(C(c2ccc(CO)c(Cl)c2)=O)C(C)(C)C1 16305,C1(C(N(C(CC)CC)C)=O)CC2(CCN(C(=O)CCC3CCCCO3)C2)C1 16306,C(C)(CNC(=O)C(C)(C)CF)(C(C)C)NC(CC(n1ccc(C)n1)C)=O 16307,C(=O)(C(F)C(C)(F)F)N1CC(C(=O)NC2CCC3(CC3)C2)(SC)C1 16308,c1(OC)ccc(C)c(C(N2CCCCC2Cn2ccnn2)=O)n1 16309,Cc1[nH]nc(Br)c1C(=O)NC(C)CC(C)NC(=O)CSC1CC1 16310,CC(=O)CCCCC(=O)N1CCC(NC(C2(CN(C)C)CC2)=O)CC(O)C1 16311,C1(C(N2C(C)COCC2)=O)CC12CCN(C(c1cc(Br)cs1)=O)CC2 16312,S(=O)(=O)(c1cccc(C(N2CC(=O)NCC2C)=O)c1)NCC(C)O 16313,c1(C(N2C(CNC(C3CC4CC4C3)=O)CC(C)(C)C2)=O)cc2ccnc(Cl)c2[nH]1 16314,c1(OC)ccc(C2=CCN(C(=O)CC3CC3C)CC2)cc1 16315,c1(OCCOCC)ccccc1C=CC(=O)OC(C)Cc1ccccn1 16316,C1(CNC(C(C)(C)C)=O)Cc2ccccc2CN1C(C1CC(S(C)(=O)=O)C1)=O 16317,C1(C(=O)NCC(CNC(COC(CC)(C)C)=O)(C)OC)OC(C)(C)OC1(C)C 16318,N1(CC(=O)NCCCNC(c2c(C)onc2)=O)CCC(O)CC1 16319,Cc1cc2ccc(C(=O)NCC3CN(C(c4cocc4C)=O)C3)cn2c1 16320,C=C=C(C)CC(=O)NC1(CN(C)C(C2CCN2C2CCCC2)=O)CC1 16321,N1(C(CC2C(C)C2)=O)CC2=C(C1)CN(C(=O)CSc1c[nH]nc1Br)C2 16322,C(=O)(C(F)(F)C(O)C(C)C)N1CC2(C(NC(c3cccc(C)c3F)=O)CCC2)C1 16323,c1(C(N2CCN(C(C)C(=O)NCC(F)(F)F)CC2)=O)nccn2nccc12 16324,c1(C(N(CCN(C(=O)CC23CCCC2C3)C(C)C)C)=O)cccc(C(=O)N(C)C)c1 16325,Cc1c(Cl)ccc(C(N2CCOC(C)(CNC(=O)C(C)OCC(C)C)C2)=O)c1O 16326,c1(C(=O)NCC2(C)CCCN2C(=O)C#CC2CCCO2)cccc2c1OCCC2 16327,N1(c2c(C#N)cncc2)CCC2C(CCCN2C(=O)CC2(O)CCOC2)C1 16328,C1(OC)CCCCC1(c1nnnn1C1CCCCC1)NCc1ccc(C)cc1F 16329,C1(NC(CC(C)SC)=O)CC2(CCN(C(c3cc(N)nc(Cl)c3)=O)CC2)C1 16330,C1(O)(CCNC(Cc2ccc(OC)cc2)=O)CCN(C(=O)Cc2cnns2)CC1 16331,c1(OCCC)ccnc(N2CCC(NC(=O)C(C3CCC3)OCC)C2)n1 16332,N1(CC(=O)NCC2N(C(Cc3nc(C)[nH]n3)=O)CC=C2)CCCCS1(=O)=O 16333,N1(C(COCCC)=O)CC2COCCC2(NC(c2cc3sccc3[nH]2)=O)C1 16334,C(=O)(NN1CCCC(C(=O)N(N2CC3CC3C2)C)C1)c1cnc(C)[nH]1 16335,n1(CC)cc(Cl)c(C(N2CC(CNC(=O)CC(C)(F)F)CC2C)=O)n1 16336,C1(C(N2C3(CNC(C4(CN(C)C)CC4)=O)CC(C2)C3)=O)CC12CCC(=O)CC2 16337,C1(C(C)C(=O)NCC(F)Br)CCN(C(C2CC(=O)C2)=O)C1 16338,C(CCCCS(=O)(=O)CCCCCO)NC(c1ccc(N2CCCC2)cc1)C 16339,N1(C(=O)CCc2ccsc2)CC2(CO)CC1(C(=O)NCCc1ccon1)C2 16340,N1(C(c2cnn(CC)c2C)=O)CCC(N(C(=O)Cn2cccn2)C)C(C)C1 16341,N1(C(Cc2cc(OC)n[nH]2)=O)CC2(CCN(C(C3CC(CC(F)(F)F)C3)=O)C2)C1 16342,C1(C(N(C2CCN(CC(COC)O)C2)C)=O)CCN(C(c2ccncc2)=O)CC1 16343,Cc1cc(Cl)ncc1CC(=O)NC1CC(C)(NC(c2nc(Cl)oc2C)=O)C1 16344,C=C(C)CC(C)C(=O)N1CC2CC2(CNC(=O)CCC=Cc2ccccc2)C1 16345,c1(C(N2C(CN(C(c3nc(Cl)oc3C)=O)CC)CCC2)=O)cnn2ccsc12 16346,N1(C(CCC2N(C)CCCC2)=O)CCN(C(=O)CCC(N)=O)C(CC2CC2)C1 16347,c1(OC)ccc2cc(C(=O)NC3CC3NC(=O)C(C)(C)CC(C)(C)C)n(C)c2c1 16348,N1(C(C2(F)C(C)C2)=O)CCC(NC(=O)COc2cccnc2Cl)CC1 16349,Clc1ccc2ccc(=NCCc3noc(-c4ccccn4)n3)[nH]c2n1 16350,C1(NC(C2CC3CCCC23)=O)CCCNC12CC2 16351,c1(NCc2ccc(-c3ccc(C(C)(C)S(C)(=O)=O)s3)cn2)cc(Cl)nc2ncnn12 16352,c1(NCC(c2ccco2)OC)ccc(S(=O)(=O)NCC(C)(C)OC)cc1Cl 16353,c1(-c2cn(CCNC(C3C(CC)OCC3)=O)nn2)ccc(Cl)cc1Cl 16354,c1(C(=O)NCCOCCNC(C2(C)CNC(=O)C2)=O)cc(Cl)cc(F)c1F 16355,N1(C(CC)=O)CCC(C)C(NC(c2cc(C(=O)NCC#N)cc(C(C)C)c2)=O)C1 16356,c1(C(C)C)ncc(C(=O)NC2CC(CNC(c3cn(CCO)nn3)=O)C2)s1 16357,C1(CNC(=O)OC(C)(C)C)CN(C(=O)Cc2cn[nH]c2)CC1O 16358,C1(NC(C2(SC)CC(O)C2)=O)CN(C(=O)CSc2cccc(Cl)c2)CC1(C)C 16359,C(N=c1[nH]cnc2c(Br)nn(C)c12)C1CN(C(C=NOC)=O)C(C)C1 16360,c1(CC)cc(C(=O)NCC2CCC2NC(C2(C#N)CCC=CC2)=O)cc(F)c1 16361,N1(C(c2cc(OCC)n[nH]2)=O)CC(C(=O)NC2CC(CN(C)C)C2)C(C)C1 16362,CCCCCCCCC(F)C(=O)NC(C)CNC(c1cnc2ccnn2c1N)=O 16363,c1(CC)ccc(C(=O)NCC2CC(F)(F)CN2C(=O)CN2CCOC2=O)c(F)c1 16364,C12(CNC(C=CSC)=O)CCC(CC1)N(C(c1cc[nH]c1)=O)C2 16365,c1(C(=O)NC2(COC)CCN(C(C(CCC)OC)=O)C2)cncc2ccsc12 16366,c1(C(=O)NCC(CC=C)NC(=O)CCc2cncs2)n[nH]c2c1CC(C)OC2C 16367,c1(OC(C(=O)N(C(CNC(C2(C(=O)NC)CC2)=O)C2CC2)C)C)cccc(C)c1 16368,C(=O)(CC(C)CNC(c1ccccc1C1CC1)=O)NCC(=C)Cl 16369,c1(-c2cn(CCCC(=O)NCC(CC)NC(N)=O)nn2)cc2ccccc2o1 16370,c1(NC(c2ccc(NC(C3N(C(C)=O)CC(O)C3)=O)o2)=O)c(C)ccnc1C#N 16371,c1(C(N2CC(CNC(C(CC)CO)=O)C(C)CC2)=O)cn2cnnc2cn1 16372,C1(NC(=O)CN2CC(C(F)(F)F)CCC2=O)CCCCN(C(C2CCC2)=O)CC1 16373,C1(C(=O)NC2(CC=C)CCC2)C2CCC(C2)N1C(=O)Nc1cc(NC)ccc1Cl 16374,c1(-c2n(C(C=C)C)nc(-c3cnn(C)c3)n2)nc2ccccc2cc1Cl 16375,c1(OC)ccnc(OC)c1C(=O)NCC1(NC(C2COC(=O)N2C)=O)CCOC1 16376,Cc1ccc(F)cc1N(C)C(C1C2CN(Cc3cncnc3)CC12)=O 16377,C1(N(C(=O)CC2CCCCC2)C)CC2CC1N(C(c1c[nH]cc1C(F)(F)F)=O)C2 16378,C1(CC#C)(C(=O)N(C(C)CNC(=O)Cc2ccnn2C(C)C)C)CCCCO1 16379,N1(C(CNC(CN(C)C)=O)=O)CC(NC(C23CCCC2C3(F)F)=O)C(C)(C)C1 16380,c1(C(=O)NC2CCC(NS(=O)(=O)CC3CCC3)CC2)ccc(C(F)(F)F)c(Cl)c1 16381,C(N=c1[nH]c(=NCCC(F)(F)Cl)[nH]c2c1SCC2)c1nc(CC)[nH]n1 16382,c1(SC)ncc(C(=O)NCCC2(O)CN(C(c3csc(F)c3)=O)C2)n1C 16383,c1(C(N2CCC(NC(CC(CCC)O)=O)CC(O)C2)=O)cnc2c(cnn2C)c1 16384,C#CCCCCC(=O)N1CCN(C(=O)CNC(C2CCCCC2OC)=O)CC1 16385,N1(C(c2n(CCC)nc(C)c2)=O)CCCCC(CNC(=O)CC2CC(SC)C2)C1 16386,N1(C(c2cc(N3CCOCC3)ncn2)=O)CCC(C2CC2(F)F)C1 16387,CCC(F)(F)C(=O)NCc1ccccc1N1CCN(C(C2(C#N)CC2C)=O)CC1 16388,c1(C(=O)NCC(O)CCNC(C2CCCCCCC2)=O)cncc2c1CCCC2 16389,C1(N(C(C=C(C)C(F)F)=O)C)CCC2CN(C(=O)Cc3ccsc3C)CC12 16390,N1(C(CCCC(C)(C)NC(C2CC2(F)Cl)=O)=O)CCCC2(CCOC2)C1 16391,C1(CNC(C(CCOC)(C)C)=O)CC2COCC2N1C(=O)Cn1ncn(C)c1=O 16392,N#Cc1ncn(CC(=O)NCC2CCC(NC(=O)Cc3ccn(C(F)F)n3)C2)n1 16393,C(CNC(=O)Cc1cccc(C2CC2)c1)(CC(C)C)NC(Cc1c(C)con1)=O 16394,c1(C(=O)NCC=CCNC(C(F)OC)=O)cc(F)cc2cccnc12 16395,N1(C(CC2(NC(C)=O)CC2)=O)CCCN(C(C2CCS(=O)(=O)N2)=O)C(CO)C1 16396,C(C(=O)N(CC=C)OC)C1(CNC(=O)CC2=CCCCC2)CC(=C)C1 16397,c1(C(N2C(C)CCC(NC(c3c(CC)cns3)=O)C2)=O)ccc2cnncc2c1 16398,c1(C(=O)NC2CC(CCNC(c3cncc(C#C)c3)=O)C2)cc(S(C)(=O)=O)cs1 16399,N1(C(c2cn(CC=C)nn2)=O)CCC2(CCC2)C(CNC(=O)Cn2cnnc2)C1 16400,C(=O)(C#CC(C)(C)CNC(c1c[nH]c(C)c1)=O)NC1CCCN(CC)C1 16401,C(=O)(C(C)CC(C)C(C)=O)N1C(C)(CC(=O)NCC=CCSC)CC1 16402,Cc1cc(-c2cn(CC3(C(=O)Nc4c[nH]c(Br)c4)CC3)nn2)ccc1F 16403,C1(C(N2CCC(N(C(=O)CCSCC)CCC)C2)=O)CC(F)CN1C 16404,C(=O)(CCCC(=O)NCC1CN(C(c2cocn2)=O)CCC1C)NCC 16405,C1(CNC(c2c(C)nn(C)c2Cl)=O)CN(C(C2CCC(=O)N2C)=O)CCC1(F)F 16406,C1(CCC(=O)NC(C)(CNC(c2cccs2)=O)C2CC2)CCCCO1 16407,c1(NC(CCC(C)NC(=O)C(C)(C)N2CCCC2)=O)cn(C)c(=O)nc1O 16408,Cc1cc(F)c(C(N2CCN(C(=O)CC(C)(C)C)CC2C(C)C)=O)cc1F 16409,N1(C(CC2CC(C)(C)OC2)=O)CCC2CN(C(c3ccncc3)=O)CC2C1 16410,n1(CC(=O)NC2CN(C(C(=O)NCC)=O)C3C2C3)nc(C)ccc1=O 16411,N1(CCN2CCC(CC=C)CC2)Cc2ccccc2C(C(=O)OC)C1 16412,Cc1cc(CC(=O)NC2(CF)CCN(C(C3CCS(=O)(=O)CC3)=O)C2)cc(F)c1 16413,c1(SC)ccc(C(=O)NCC2CC2CNC(c2nn(C)cc2Cl)=O)cc1 16414,Cc1cc(C)c(C(=O)NC2CC(NC(=O)C(O)CC(F)(F)F)C2)c(O)n1 16415,C(C(=O)NOC)(C(C)C)N(C(C=NOC)=O)C 16416,CC(C(CO)NC(=O)CCOCc1ccccc1)NC(=O)CNC(C1CCC1)=O 16417,C1(C)(CNC(CCc2c(C)ncs2)=O)COCCN(C(=O)C(C)C(F)F)C1 16418,N1(C(CC2(C)CC2)=O)CC2CCC2(NC(=O)CCc2ccc[nH]2)C1 16419,CC1CCN(C(=O)CC23CCCC2C3)C1CNC(c1[nH]nnc1C1CC1)=O 16420,c1(C(N)=O)nc(OC2CS(=O)(=O)CC2C(=O)O)cc(SC2CC2)n1 16421,Cc1ncc(C(N2CC3(CCN(C(=O)C(C)(C)C)C3)C2)=O)c(Br)c1Cl 16422,C(=O)(C#CC1CCOCC1)N(C)CC1CCCN1C(c1cc(F)cnc1Cl)=O 16423,C12(C(N3CCC(CN(C)CC)C3)=O)CC(CO)(CN1C(=O)CCOC(C)C)C2 16424,c1(C(N2CC(CN(C(=O)C(N)=O)C)OCC2)=O)cn2ccsc2n1 16425,C1(NC(C(CC2CN(C(C3CCN(CCOC)C3)=O)C2)F)=O)C(C)CCC1C 16426,Cc1ccc2nc(C(=O)NC34CC(C3)N(C(=O)CN3CCOC3=O)C4)ccc2c1 16427,C1(OC)CCCC(C(=O)NCC23CC2CN(C(=O)C(CCSC)OC)C3)C1 16428,CC1CN(C(c2cc(Cl)c(F)cc2Cl)=O)CC(C)N(C(c2ncccc2N)=O)C1 16429,c1(CC(=O)NCC2C(NC(C(C)OC)=O)CC2)cc(C)nn1C 16430,C#CCC(O)C(=O)NCC1C=CC(NC(c2cc(Nc3ccccc3)cs2)=O)C1 16431,N1(C(c2c(OCC)cccn2)=O)CC2CC(NC(=O)C(=O)N(C)C)C2C1 16432,C(=O)(NNc1cc(F)ccc1C(F)(F)F)c1c(Cl)ccc(NC(CC(C)C)=O)c1 16433,C1(NC(c2cc(-n3ccnc3)ccn2)=O)CN(C(=O)C(F)(F)Cl)CC1(F)F 16434,c1(OCC=C)ccc(S(N)(=O)=O)cc1C(N1CCC1CNC(=O)C(O)C1CC1)=O 16435,c1(CN(C(C(CSC)C)=O)CCNC(=O)CNC(=O)C(C)(C)C)cccc(Cl)c1 16436,C=C1CON(C(=O)COC2CCN(C(=O)C(O)C(C(C)C)OC)C2)C1 16437,c1(SCCC)ccc(-c2ccc(C3(C(=O)NC4CC(O)C4)CC3)cc2)cc1 16438,Cc1ccc(C(O)CNC(C2(CO)CCCO2)c2nn[nH]n2)cc1 16439,C1(NCC(Cc2ccncc2)C2CCC2)CC2CCCOC12 16440,c1(C(=O)NC2C3CN(C(c4n(CC)ccc4)=O)C2CC3)nc(C)c(N)cc1C 16441,C(CC(C(=O)N1CCC(C)(CN(C)C)C1)NC(=O)COC)=CC 16442,C1(NC(c2ccc(CSC)cc2)=O)CC2CN(C(C3(C)CCCC3)=O)CC12 16443,C1(CNC(COC(CC)CC)=O)CCCN(C(c2nnsc2C)=O)CC1 16444,N1(C(C)C)CCC(C(=O)NCC2CCCN2C(C2CCCC3CC23)=O)CC1 16445,Cc1ccc(I)cc1CN1CCS(=O)CC1c1cnn(C)c1 16446,N1(C(=O)C2=CCC2)CCCC2(C1)CN(C(C1C3C4CCC(C4)C13)=O)CCO2 16447,c1(C(N(C(C)C(=O)NCc2cc(O)cc(F)c2)CCC)=O)cnn2cccc2c1 16448,Cn1c(C(=O)NCCCCC(CO)NC(c2cnc[nH]2)=O)c2n(c1=O)CCCC2 16449,CCCC(C)CC(C)(c1nnnn1C(C)C)Nc1ccc(C(=O)N(C)C)c(C)c1 16450,C12(NC(CCCCC(N)=O)=O)CN(C(=O)CCN3CCCC3)CC1CS(=O)(=O)C2 16451,CC(CC(=O)NCC1CN(C(c2cc(C(n3cccn3)C3CC3)on2)=O)C1)C(F)F 16452,CC1CCN(C(=O)CCc2nncs2)CC1NC(C1CCN(C(=O)N(C)C)CC1)=O 16453,CCCC(CC)CC(=O)N1CC(CO)(NC(=O)CNC(=O)Nc2ccccc2)C1 16454,N1(C(c2[nH]nc(OC)c2Cl)=O)CCC2(NC(=O)Cc3cscn3)CCCCCC12 16455,c1(C(N2CC(CC)N(C(c3cc(Cl)n(C)n3)=O)CC2)=O)cc2ccc(C)cc2[nH]1 16456,C(=O)(C(C)P(C)(C)=O)NC1C(N(C(c2cncc(C(=O)OC)c2)=O)C)CCCC1 16457,Cc1cc(Cl)c(C(=O)N(CC(C)(C)NC(c2onc(C)c2C)=O)C)s1 16458,CCCC(CNC(=O)C(C)SC(C)(C)C)CCO 16459,S(=O)(=O)(c1ccc(NC2CCCC3(CCOC3)C2)c(Cl)c1)N1CCN(CC)CC1 16460,c1(OC)ccc(C(N2CCCC(C)(CNC(C3(N(C)C)CCC3)=O)C2)=O)cc1Cl 16461,CC1CC(C(N2CCCC2CNC(c2occc2C2CC2)=O)=O)CC(C)C1 16462,c1(CNC(C2CC2Cl)=O)cccc2c1CN(C(c1ccn3nnnc3c1)=O)C2 16463,c1(CC(=O)NN2CCC(C)C2)ccc2nc(O)[nH]c2c1.C12CC(C1)C(=O)N2 16464,N1(C(c2ccc(C(C)F)cc2)=O)CCCC(C)(CNC(=O)CN(C)C2CC2)C1 16465,Cc1nc(C)c(F)c(=NCCN(C(=O)C(C)(O)C(C)c2ccccc2)C)[nH]1 16466,CC(CC(C)(C)C)NC(=O)C(c1cccs1)NC(=O)CC1NC(=O)NC1=O 16467,C(=O)(CCCCCn1cc(C(c2ccccc2OC)(C)C)nn1)NCCC(=C)C 16468,c1(OC)ccnc(CC(=O)N(CC(C)(C)CNC(C2CC2c2ccco2)=O)C)n1 16469,N1(C(C(C)(C)C#N)=O)CCN(C(c2ccc(F)nc2F)=O)C(CCO)C1 16470,C=C1CCN(C(=O)CSCCC)C(C(=O)N(CCn2ccnn2)C2CC2)C1 16471,C1(CN2C(CC(=O)NCC(O)C(F)(F)F)COCC2)CCC(F)(F)CC1 16472,N1(C(C(C(C)C)C)=O)CC(CNC(c2cc3ccccc3o2)=O)OC(C)(C)C1 16473,N1(C(CC(C=C)CCC)=O)CCC2(CCC2NC(=O)C=CCOCCOC)CC1 16474,C1(C(=O)N=c2nc[nH]s2)Cc2cc(O)ccc2CN1C(c1ccc(F)c(O)c1)=O 16475,c1(CC(C=C)O)cn(CCCC(=O)N2CC(CS(C)=O)C2)nn1 16476,C1(CNC(c2c(C)scn2)=O)CC2CCC1N2C(C1(C)CC(F)C1)=O 16477,CC(CC1CC1)C(=O)N(CC(C)(C)NC(=O)C(C)n1ccnc1)C 16478,C1(C(=O)N2CCC(COC)C2)(CCC)CCOc2ccccc21 16479,CS(C)(=O)=NC(=O)C(=O)NC1CC(c2ccccc2)(NC(=O)COC(F)(F)F)C1 16480,C1(CNC(C(COC)OC)=O)CN(C(=O)CC2CN(C(C)=O)C2)CCN1C 16481,O=C1NCC2(CCN(C(C3CCOCC3NC(=O)C(O)Cn3cncn3)=O)C2)N1 16482,C(=O)(CC(C)NC(=O)CC1(C)OCCO1)NC(CC#C)C 16483,N1(C(CS(C(C)C)(=O)=O)=O)Cc2nccn2CC(NC(=O)C=C2CCC(C)C2)C1 16484,C(c1cccc(CO)c1)=CC(=O)N(C1CCN(Cc2nccc(C)c2)C1)C 16485,c1(OC)ccc(C(=O)N(C(C)CNC(c2ncc(N)nc2C)=O)C)c(Cl)c1 16486,Cc1cc(CCC(=O)NC(C)(CNC(=O)CCCF)CO)n[nH]1 16487,CCC(CC(=O)N1CCC1CNC(c1ccc(CSCC)o1)=O)c1ccccc1 16488,N1(C(c2c(C)noc2C)=O)CC2(C1)SCCC2NC(=O)C(O)C1CCCC1 16489,CC(Cc1cccs1)N=c1ccnc(N2CCOCC(C)(F)C2)[nH]1 16490,c1(OC)cc(Br)cnc1C(=O)NCCC1(NC(c2cnn(C)c2)=O)CCC1 16491,c1(C(=O)NCC(C)N(C(=O)C=Cc2cc[nH]c2)C)cc2cc(Cl)cc(Cl)c2[nH]1 16492,c1(CCC(=O)NCC(CNC(c2ccn(CC)c2C)=O)CO)ccc(C)cc1C 16493,C1(NC(CCN(C)C(c2cccnc2O)=O)=O)CCOC12CCOC2 16494,N1(C(c2ccc(-n3ccnc3)nn2)=O)CC(NC(C23CC2C3)=O)CC2(CC2)C1 16495,CC(=O)CCCC(=O)NC(C)(CNC(c1nccc(Cl)c1Cl)=O)C1CC1 16496,n1(CCNC(C(C)C2(O)CCC2)=O)ccc(C(=O)NC2(C(F)(F)F)CC2)c1 16497,CC1CN(C(C)CCc2ccccc2)CC1NC(=O)CN1CCCNC1=O 16498,CCCCCCN(CCNC(C12CC(F)C1C2)=O)C(c1cccnn1)=O 16499,C(=O)(CCCCCCn1cc(-c2cncc(F)c2)nn1)NC(C(CC)C)CO 16500,C(C)(C)(CCN=c1[nH]cnc(C)c1Br)NC(C(c1cccc(C)c1)C)=O 16501,CC(C)(C(=O)N1CC=CC(C(=O)NCC(CO)C(C)(C)C)C1)C(F)(F)F 16502,C#CCN(OC)C(=O)C1(CF)CCN(C(c2cn(C)c(C)n2)=O)C1 16503,C1(CNC(CC2CC(CC)C2)=O)CN(C(=O)CSC2CC2)CC1C(F)(F)F 16504,CC(CCC(F)(F)F)NC(=O)CC(C)(C)NC(=O)CC1CCCC1O 16505,C(=O)(C1=CCCCCC1)NCc1ocnc1CNC(=O)CC1NC(=O)NC1=O 16506,c1(C(C)C(=O)NCC2(O)CN(C(=O)CSCc3cc(Cl)no3)C2)ccc(F)cc1 16507,Cn1cc(CC(=O)NCCCN(C(c2cn(C)cn2)=O)CC2CCCC2)c(Cl)n1 16508,CCC(CC(F)F)C(=O)N1CCC(CN(C(=O)C(C)c2ccco2)C)C1 16509,c1(NCC2(OC)CCN(C(C(C)OC)=O)CC2)nc(C)nc2scc(C)c12 16510,C(C(=O)NNC(=O)c1ccc(Br)cc1)C12CCCCC1C2.c12ccccc1SC2=O 16511,C1(NC(CS(C)(=O)=O)=O)CC(NC(=O)Cn2cnc(C#N)n2)C12CCC2 16512,C(=O)(CC1=CCCCC1)N1CC2C(Nc3ccc(OCC)c(O)c3)(CC2)C1 16513,c1(C(N2C3C(NC(=O)C=CC(F)(F)F)C(CC3)C2)=O)sc2ccccc2c1CO 16514,Nc1nc(C(N2CCC3(NC(=O)COC(F)F)CC3C2)=O)ccc1O 16515,C1(C(=O)OC)CCC(NC(=O)C(N2CCOCC2C(=O)N(C)C)=O)CC1 16516,c1(C(N2CCC(N(C(C=CC=CCC)=O)CC)C2)=O)csc(=NC2CC2)[nH]1 16517,N1(C(c2cn(CC=C)nn2)=O)CCC(NC(=O)Cc2cccc(C)c2)C(CC)C1 16518,C(C1=CCN(C(=O)OC(C)(C)C)C1)Sc1occ(NC(C)=O)n1 16519,CCC(C)(C)C(=O)N1CCC(N(CCO)C(C2CCC(C)(C)O2)=O)C1 16520,c1(C(=O)NCC23N(C(COCC)=O)CCC2CC3)cc(Cl)c(OC)c(Cl)c1 16521,C1(C2CCCN(C(=O)CN3CC4CC4C3)C2)(NC(C2(OC)CCOC2)=O)CC1 16522,CN1CCCC2(CCN(C(CC3CCC4CC34)C(=O)NC(C)(C)C)C2)C1 16523,N1(C(Cc2c(OC)nccc2)=O)CCN(C(C2CC2C(F)F)=O)C(CCO)C1 16524,N1(C(C2CC3(CCCCC3)C2)=O)CCn2ncc(C(N3CCC(O)C3)=O)c2C1 16525,N1(C(c2ccn(CC)n2)=O)CCC(C)C(NC(=O)CCCCN(C)C)C1 16526,c1(C(N2CC(N(C(C3C(C)OCC3)=O)C)C2)=O)ccccc1Cl 16527,N1(C(CCSCCC)=O)CCOC(CN(C(=O)CN2CC(C)(OC)C2)C)C1 16528,Cc1ccc(C(N2CCC(F)(C(=O)NCCCC(O)CO)CC2)=O)nc1C 16529,C1(C(C)C)CN(C(C2CCOC2C(C)C)=O)CC1C(=O)N(C)Cc1cccs1 16530,CCC(C)(CNC(=O)COC1CC(NC(=O)CC2CCCCO2)C1)CC 16531,C1(O)(C(=O)NC2CC(NC(Cc3ccn(CC)n3)=O)C2)CCCC(C)(C)CC1 16532,Cc1ocnc1C(N1CSCC1C(N1CCC1c1ccccc1)=O)=O 16533,N1(C(C)=O)CCCC1CC(N1CC(O)(CCNC(=O)C(C)(C)c2ccno2)C1)=O 16534,C(=O)(C1=NOC(C)C1C)NCC1(NC(c2cc(F)cc(Cl)c2N)=O)CC(OC)C1 16535,CN1CC(N=c2nc3sccc3c(NCC(=O)NC3CC3)[nH]2)CC12CCC2 16536,c1(NC(=O)NC2CCCC(O)C2)nc2ccc(F)cc2s1 16537,CCC(C#N)(CC)C(=O)NC1CCCC(NC(=O)CCNC(=O)CC(C)C)C1 16538,CC(C)(CC(F)C(=O)NCCC1CCCC12CC2)NC(C1CC2CC2C1)=O 16539,c1(C(N2CC(NC(C3(CO)CC3)=O)CC(O)C2)=O)ccc2ncccc2n1 16540,c1(C(=O)NCC2CCCC(O)C2)cn2c(n1)CCC2.C12(CCCCC1)CCC(=O)N2 16541,C(=O)(CCCN=[N+]=[N-])N(CCOCCCN(C(C1(OC)CCCC1)=O)C)C 16542,C1(CNC(c2coc3c2CSC3)=O)CN(C(=O)CO)C2CCN1C2 16543,c1(C(N2CC(c3n(C)cnn3)OCC2)=O)ccc(OC(F)F)c(F)c1 16544,c1(C(=O)NCC2C(OCC(=O)NCCOC(C)=O)COC2)ccnc(O)c1 16545,C1(C(=O)NCCN(C(=O)C(C)OC2CCCC2)C(C)C)CCC2C(C1)C2(F)F 16546,C1(NC(c2c(C)cc(CO)o2)=O)CN(C(C2(C)CCCCO2)=O)CC1(C)C 16547,C1(NC(C2(C(=O)OC)CC2)=O)CC2CCC1CC2NC(c1cc(Cl)ncc1OC)=O 16548,N1(C(C(CC)=O)=O)CCC2CC(C(N3CCC(F)(CO)CC3)=O)C2C1 16549,c1(OC)cc(C(N2CCC(OCCNC(=O)C(C)c3ccco3)C2)=O)oc(=O)c1 16550,N1(C(C=CC(C)(C)C)=O)CC2(C1)SCCC2NC(=O)COC1COC1 16551,C1(N(C(C=CC(CC)=CC)=O)C)CN(C(=O)Cn2ncc(Cl)c2C)CC1(C)C 16552,Cc1nnccc1C(=O)N(C)CC1CCN(C(c2ccc(C(C)(C)C)cn2)=O)C1 16553,N1(C(C2C(=C)C2)=O)CCC2CN(C(=O)CCCc3nncn3C)CC12 16554,C1(C(=O)NCCC2(C)CCCO2)(NC(C2CC2C(F)F)=O)CCCCC1 16555,Cc1nn(C)c(N)c1C(N1CCOC(CC(N2CC(C)C2(C)C)=O)C1)=O 16556,CC1(C)C(C(=O)NCC2CN(C(=O)C(C)(C)c3sccc3Cl)CCO2)C1(C)C 16557,NC(CC(=O)N1CCCCC1Cc1ccccc1F)C(=O)O 16558,c1(OC)c(Br)cc(CNC(C)CC2CCC2)cc1Br 16559,Cc1cnc2n1CCC(NC1CCS(=O)(=O)CC1)C2 16560,c1(OC)ccc(C(=O)N(CC(C)(C)CNC(=O)Cn2nnc(=N)[nH]2)C)c(F)n1 16561,S(=O)(=O)(c1ccc(C)cc1F)NCC(=O)N(CCN(C(=O)C(C#N)C(C)C)CC)CC 16562,N1(c2cc(C)nc(Cl)n2)CC2CCC1C1CN(C(=O)C=CC(=O)NC3CC3)CC21 16563,C(C(C)(O)CC(=O)NCC1(NC(c2nc(C)n(C)c2C)=O)CCC1)OC 16564,c1(CC)[nH]nc(C(=O)NC(CNC(c2ccnc(C(C)C)n2)=O)C(C)(C)C)c1Cl 16565,c1(C(=O)NC2CC(NC(c3c(C)ccc(F)c3)=O)C(O)C2)cccc2c1NCC2 16566,O=C1CN(C(=O)Cn2ncnn2)C2CCN(C(C3CC=CCC3)=O)CC2N1 16567,C(=O)(CCC(C)NC(C1CC(O)C(F)C1)=O)NC1(C(=O)OC)CC(C)C1 16568,c1(C(N2CC(C)C(NC(=O)C#CC3CCC3)C2)=O)cc2c(F)ccc(F)c2[nH]1 16569,c1(C(=O)NCC(C(C)(C)C)NC(c2cnc(S)[nH]2)=O)cc(O)ccc1Br 16570,C1(C(N2C(C(=O)NCC3(SCC)CC3)CC(O)C2)=O)CCCCN1N=O 16571,N1(C(=O)Cc2cocn2)CC2CN(C(C3CC4C=CC3C43CC3)=O)CC2C1 16572,C(=O)(C(CC(C)C)C(C)C)NCC(CC=C)C(=O)NC1(CN(C)CCOCC)CC1 16573,N1(C(C2(CC=C)CCOCC2)=O)CC(NC(c2cccc(F)c2C)=O)C(C)(C)C1 16574,C(=O)(C1=NOC(C)C1)NCC(C(C)C)NC(C=CC(C)C)=O 16575,NS(=O)(=O)c1cccc(NC(C2CC2NC(c2cc(O)cc(Br)c2)=O)=O)c1 16576,C(=O)(C1=CCC2CCC1N2C(=O)C(C#N)C(C)(C)C)NCC=CC=CC 16577,C1(OCC)CC2(C1)CC2C(=O)NC1CCC(NC(C2CCCS2)=O)CC1 16578,C1(C(=O)NC2(C(=O)NCc3ncc(C)cn3)CCN(C)C2)CC2(CCC2O)C1 16579,N1(C(C(CC(CC)C)C)=O)CCc2ccc(C(=O)NCC(C3CC3)OC)nc2C1 16580,CN=c1[nH]c(C(N2CC(C(C)NC(C3CCN(CC(F)F)CC3)=O)C2)=O)cs1 16581,c1(OC)ccc(C(C(=O)O)NC(C2CCCCC2(F)F)=O)cc1Cl 16582,C(=O)(C(CNC(c1cc(C(N)=O)[nH]n1)=O)OC)NCC(=C)Cl 16583,C1(O)(C(CNC(C(C)N(C)C)=O)C)CCN(C(=O)Cc2sccc2Cl)C1 16584,N1(C(C=C(C)C(C)(C)C)=O)CCCC(NC(=O)C=C2CCCC2)C(F)C1 16585,Cc1ncccc1C(=O)NC1CC(O)(CNC(C2CC3(CSC3)C2)=O)C1 16586,C(=O)(C(C)CCCOC)N1CCC(C(C)NC(C(C)OCCCC)=O)CC1 16587,c1(SCC(=O)NC(C2CCN(C(C(CC)F)=O)C2)=O)ccc(Br)cc1C 16588,c1(C(N2CC(NC(C3CN(OC)C(=O)C3)=O)C(C)C2)=O)nccn2cc(C)nc12 16589,C1(NC(=O)COCC2CCCO2)CC(F)CN(C(=O)Cc2cc(F)cc(F)c2)C1 16590,N1(C(CC2CCC(C)CO2)=O)CCC2CN(C(c3ccc([N+](=O)[O-])[nH]3)=O)CC12 16591,S(=O)(=O)(c1ccc(=NCCc2cnoc2)[nH]c1)N(C)CC12CCC(CC1)OC2 16592,Cc1c(NCCCCN2CCC2)nc[nH]c1=NCCNC(N1CCOCC1)=O 16593,N1(C(C(=C(C)C2CC2)F)=O)CCCCC(CNC(c2cc(CO)n(C)n2)=O)C1 16594,c1(C(=O)NC2C3CN(C(c4ccc(NC)c(F)c4)=O)C2C3)cc2n(n1)CCCO2 16595,N1(CC(COC)O)CCC(N(C(=O)CC2CCN(c3ccccc3)C2)C)CC1 16596,C1(C(N2C(CNC(=O)Cc3cccs3)(COCCO)CCC2)=O)CCOC(=O)CC1 16597,C#CC1CCN(C(=O)C(CNC(=O)CCCOCC=C)N(C)C)CC1 16598,c1(C(=O)NCC2COCCN2C(C2CCS(=O)(=O)N2)=O)cc2nc[nH]c2cn1 16599,N1(C(C2CCN(C(C3(CO)CCC3)=O)C2)=O)CCCC2(CCC2)C1 16600,C1(CC)C(C(=O)NCCNC(C)=O)CCN1C(=O)CC(=O)NC 16601,CC1(C)CC(NC(c2ccc(C3CC3)cn2)=O)CN(C(c2cccnc2S)=O)C1 16602,N1(C(C(CC=C)CNC(C2C3(CC3)C23CC3)=O)=O)CCc2ccc(F)cc21 16603,N1(C(=O)Cc2ccc(Cl)cc2Br)CC(c2ccccc2)Oc2ccccc21 16604,c1(C(=O)NCC2(COC)CN(C(C3CCNC3=O)=O)C2)noc2ccc(Cl)cc12 16605,N1(C(c2c(C)oc(CNC(=O)Cc3cc[nH]n3)n2)=O)CCc2nc(O)[nH]c2C1 16606,S(=O)(=O)(c1cc(Cl)sc1Cl)N(C(C(=O)OC)C)CC1CC1 16607,c1(CNC(C2C(NC(c3cncc(OCC)n3)=O)C2)=O)cc(C)sc1OC.C 16608,CC1CN(C(c2cccc(C#N)n2)=O)CCC1NC(c1cc(=O)cc[nH]1)=O 16609,C1(OC)CCC2(C(=O)NCCC(C)(C)NC(c3cccc(OC)n3)=O)CCC12 16610,C(C(C)(C(=O)N1CC(C)(N(C)C)C1)NC(c1ccc(C)nc1)=O)SC 16611,c1(NC(C2(CC)CCCC2)=O)cccc(CNC(c2ccoc2Br)=O)c1 16612,C1(NC(CSCCC)=O)CCCN(C(c2c[nH]cc2C(C)(C)C)=O)CC1 16613,C1(C2(O)CCN(C(C3CC3(C)Br)=O)CC2)(NC(C=C(C)c2ccco2)=O)CC1 16614,C1(C)(CC)CN(CCCOC(C)=O)CCO1.c1(CN(CCCC2CC2)C)ccccc1 16615,Cc1ccc(Cl)c(C(=O)NCC23CC(NC(=O)Cc4cnn(C)c4)(CO2)C3)c1 16616,n1(C(C)(C)C)cc(Cl)c(=NC(=O)NCC(F)(F)F)[nH]1 16617,N1(C(C=CC(CC)=CC)=O)CCOCC(C)(CNC(c2cnncc2C)=O)C1 16618,Cc1c(C(=O)NCC(C2CC2)N(C)C(c2cc(-c3ccco3)no2)=O)nnn1C 16619,N1(Cc2ccc(OCC#N)cc2)CCSC2CCCCC12.c12ccc(cc1)OC2 16620,c1(CC(=O)NC2CCC(C)N(C(=O)CCCF)C2)cccc2ccsc12 16621,C1(CC(=O)OC)(NC(C2CN(Cc3ccc(C)o3)CCS2)=O)CCCCC1 16622,C1(NC(c2cc(C)c(C)o2)=O)C2CC3C(C2)C13C(=O)N(C)CC1CCCS1 16623,c1(C(N2C3CC(CNC(C(CC#C)N(C)C)=O)C2CC3)=O)ccn2ccccc12 16624,C1(CNCCC2C(C)CCO2)CCOCC1CC(F)(F)F 16625,c1(CC(=O)NCC(C2CC2)NC(C(C2CCC2)OCC)=O)sc(O)nc1O 16626,C12CCN(CC1)C(=O)N2.C=CC1(CC(=O)NCCNC(C2CCCC2)=O)CCC1 16627,N1(C(CC2C(C)CCN(C(C(C)(C)OC)=O)C2)=O)CCCc2ccccc21 16628,C1(N(C)C)CCCN(CC(=O)NCCNC(=O)Cc2ccc(CO)cc2)C1 16629,CCCCN=C(NCc1ncc(C)cn1)NCC1(CCC)CC1 16630,CC1OCCOC1C(=O)NC(C)(C)CC(=O)N1CCC(C(F)F)C1 16631,c1(C(=O)NCC2CCN(C(=O)Cc3cn[nH]c3)C2)cc2n(n1)CCO2 16632,C1(NC(c2nc(C(C)C)sc2)=O)CCN(C(=O)C(C)CF)C1C(C)(C)C 16633,C1(C(N2CCOCC(CNC(CC(C)C)=O)C2)=O)CCCN2CCCCC12 16634,CCCCCC(C(=O)N1CCC(NC(c2ccn(COC)n2)=O)C1)C(C)C 16635,C1(C(=O)NCC2(NC(C(CC)F)=O)CCCC2)CCCCN1S(C)(=O)=O 16636,N1(C(c2ncc(CC)cn2)=O)CCC(C2CC2)C1C(=O)N(C1CC2CCC1O2)C 16637,CC(C)(F)CC(=O)NCC1COC(CNC(c2ncsc2Br)=O)C1 16638,C(=O)(C1=NN(CC)C(=O)CC1)N1C(CCC)CN(C(c2ccnc(S)c2)=O)CC1 16639,CS(=O)CCC(O)C(=O)NC12CC(NC(=O)C=Cc3cccs3)(C1)C2 16640,CCCCCC(O)C(C)C(=O)N1CC(CNC(C2Cc3nccn3C2)=O)C(O)C1 16641,c1(CC(C)NC(=O)C(Cn2cncn2)NC(c2cncs2)=O)ccccn1 16642,C=CC1CN(C(C2(N(C)C)CCCC2)=O)CC1NC(=O)CC(C)C1CCCCC1 16643,N1(C(C2CC(C(C)C)C2)=O)CCCC(CO)(CNC(=O)C(C2CCCCC2)F)C1 16644,c1(NC(=O)NC(c2ccccc2)C2CCCCC2)nccc(-c2ccncc2)n1 16645,C1(NC(C(CNC(C2C3COCC23)=O)N(C)C)=O)CCC(O)C(O)C1 16646,C1(CNC(CC=C)=O)CCCCC1NC(c1cnn(C2CC2(F)F)c1)=O 16647,Cc1oc(C)c(C(=O)NC2CCCC(NC(=O)CC3CC(=O)C3)C2)c1C 16648,C1(C(N2C(C)(CNC(=O)C=CBr)CCC2)=O)CCCC12CCC2 16649,C1(CNC(CC(C=C)c2ccccc2)=O)CN(C(=O)C(F)(F)CC)CCCO1 16650,N1(C(C(C)c2cncs2)=O)CCCCC1CCCNC(c1ccco1)=O 16651,C1(C(=O)NC(C(N2CC(C(N)=O)OCC2)=O)c2ccco2)CC2CCCC2C1 16652,Cc1cc(=NC(C)CCNC(C2(F)CCC2)=O)c([N+](=O)[O-])c(C)[nH]1 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16721,c1(OC)cc(C(=O)NC(Cc2cnn(C)c2O)C(=O)N2CC(C(C)C)C2)n(C)n1 16722,C1(OC)C2CC3CN(C(c4sncc4Br)C(=O)NC4CCOC4)C1C3C2 16723,C1(N(C(CC(=O)NC)=O)C)CN(C(=O)C(C)C=Cc2ccccc2)CC1O 16724,c1(CCC(N2C(C3(NC(C(CSC)C)=O)CC3)CCC2)=O)csc2ccccc12 16725,C(=O)(C(CCC)NC(=O)C(C)(C)O)NCc1cn(CC#C)nc1 16726,Cc1cc(F)cc(C(=O)N(CC(C)NC(c2nc(C)n(C)c2C)=O)C)c1N 16727,CC(C)(C#N)CCCC(=O)NC1CC(NC(C2(C)CC2F)=O)C1 16728,n1(CC(=C)C)nnnc1C(c1nc(C(F)(F)F)cs1)NCC1(C)CCCC1 16729,CCC(C)CCC(=O)N(CCC(C)NC(c1cnn(CCN(C)C)c1)=O)C 16730,c1(NC)ccc(C(N2CC3CC(NC(c4cc(C)c(C)o4)=O)C2C3)=O)cc1F 16731,N1(C(C(C)O)=O)CCN(C(=O)C=C(CC)CC)CC(CO)C1.CCCC 16732,c1(CNC(C2CCC3(CCC3)CC2)=O)nc2cccnc2[nH]1 16733,C12(C(=O)NCCOCCNC(C3CCS(=O)(=O)N3)=O)CCN(CC1)CC2 16734,c1(C(N2C3CC(CNC(C(COC)COC)=O)(OC3)C2)=O)nccn2nccc12 16735,c1(NC(C(C)OC(C(CCSC)OC)=O)=O)ccc(CN)cc1F 16736,C1(NC(c2c(OC)cccn2)=O)CCCC12CCN(C(=O)Nc1ccccn1)C2 16737,c1(C(N2CC3C(C(=O)NC4CCCCC4(F)F)C3C2)=O)cc(F)cc(F)c1F 16738,Cc1cnc(C(N2CC(C(=O)NC3(C)CCCC3C)C(C(C)C)C2)=O)cn1 16739,C1(C(N2CCCC(NC(=O)CCc3ccncc3)CC2)=O)CCC2(CCC2)CO1 16740,N1(NC(C2CCC(CCO)CC2)=O)CCC(O)C(CCN2CCC(F)CC2)C1 16741,N1(C(C(=O)Nc2cc(C)sc2C)=O)CCSCC1(C)C 16742,c1(CCC(=O)N(CCN(C(=O)CCN2CCOCC2)CC)CC)cncn1C 16743,CCCCC(O)CC(=O)N1CCC(C(=O)N(C)Cc2cccc(C)n2)C(C)C1 16744,C1(C(=O)NCC2CN(c3nccc(-n4ccnc4)n3)CCO2)C2C3CCC(C3)C12 16745,c1(C(=O)NCC2C(NC(C3CC(C)(C)C3)=O)CCC2)c[nH]c(=O)cn1 16746,C1(NC(C(CC2CC2)OC)=O)CN(C(=O)CCCn2cccn2)CC2CCCC12 16747,c1(C(N(CCCOCCNC(C2C(C=C)C2)=O)C)=O)ccc(C)nc1N 16748,c1(CCC(=O)NC2CCC(NC(CN(CCOC)C)=O)C2)cc(F)cc(F)c1 16749,C1(NC(c2c(SCC)nccn2)=O)COC2CN(C(c3cc(OC)cs3)=O)CC12 16750,C(=O)(C(CCOCCO)NC(=O)CCC1(C)N=N1)N(CC(COCC)O)C 16751,C(C1CCCN1C(=O)COCCC)=CC(N1C(C#C)CC1)=O 16752,c1(C(=O)NC2C=CCN(C(CC(CCC)O)=O)C2)cc(O)nc2cnccc12 16753,C(C1=NOC2CN(C(C3(C)CCCC3)=O)CC12)NC(C1(COC)CC1)=O 16754,c1(CNC2CC(NS(CC)(=O)=O)C2)c(Br)cncc1Br 16755,C1(NC(c2c(C)ccn2C)=O)COC2(CNC(=O)CSc3n[nH]c(C)n3)CC1C2 16756,C1(C(=O)NCC2C=CCN2C(c2cnc(C3CC3)s2)=O)C(Cl)(Cl)C12CC2 16757,c1(OC)cncc(NC(C2(O)CCN(C(=O)C(C)(C)OC(C)=O)C2)=O)c1 16758,N1(C(CCC(=O)N(C)C)=O)CCCC12CCN(C(=O)CCC(F)(F)C(F)F)C2 16759,S(=O)(=O)(c1cnn(C)c1)N1CCC(CC(=O)NC(C#C)C)C1 16760,C1(NC(C(C=C)(C)CC)=O)CC2(CCN(C(C3(C#N)CCCC3)=O)CC2)C1 16761,N1(C(C(CNC(c2cnn(C=C)c2N)=O)CC2CC2)=O)CCC2(COC(=O)N2)C1 16762,CC1=C(c2ccccc2)CN(C(c2ncncc2Cl)=O)CC1 16763,CN1CCC(C(=O)NC2(C(=O)Nc3ccccc3O)CC2(C)C)CC1=O 16764,n1(C(C)C)cc(C(=O)NC2(C)CN(C(=O)CN3CCCC3C)C2)c(O)nc1=O 16765,c1(C(C)NC(=O)NCCC2CCCC2(C)C)cc(Cl)cc2c1OCC2 16766,CC1CC2(CC(NC(c3ccnc(OCc4ccccc4)c3)=O)C2)C1 16767,C1(NC(=O)NC2(c3cc(C(F)(F)F)[nH]n3)CC2)CN2CCC1C2 16768,Cc1nc2cccc(C(N3CC(CNC(c4ccc(=N)[nH]c4)=O)CC3C)=O)c2[nH]1 16769,N1(C(=O)Cc2nc(Cl)cs2)CCN(Cc2ccc(Br)c(F)c2)C2CC12 16770,N1(C(c2snnc2C)C(=O)NC(C(=O)OC)C)CCC(CC(=O)N(C)CC)CC1 16771,c1(C(=O)NC2CC(NC(C(COC(C)C)(C)C)=O)C2)ncn2c1CCC2 16772,C1(CC(=O)NCC(C2CCCN2C(=O)CN2CSCC2=O)(C)C)CCCCO1 16773,c1(NC(C2N(Cc3cnn(C)c3Cl)C3CCC2C3)=O)cccc(Br)c1[N+](=O)[O-] 16774,C1(C(N2CCN(C(c3n[nH]c(C)c3F)=O)CC2)=O)CCC2CCCCN12 16775,N1(C(COCCCC)=O)CC2CCN(C(C3(CCCF)CC3)=O)CCC2C1 16776,N1(C(C(C)NC(c2ccoc2)=O)=O)CC(NC(=O)C(O)P(C)(C)=O)CC(F)C1 16777,c1(CC(N2CC(C)C(CNC(C3C4CC5C(C4=O)C35)=O)C2)=O)ccc(F)cc1Cl 16778,N1(c2nnc(C(C)CO)n2C)CCCC2(CN(CCO)CCO2)C1 16779,N1(C(C(C)CN(C)C)=O)CC2CC(NC(=O)CCC3CCC3)CC1C2 16780,N1(Cc2nnc(C(C)(C)C)o2)CCC2(CCN(C(c3c(F)cccc3Cl)=O)C2)C1 16781,N1(C(c2nc(OC)c(C)s2)=O)CCN(C(C2(C3CC3)CC2)=O)CC(CO)C1 16782,C(=O)(C(CO)C(C)(C)C)NC(C(=O)N(CC(C(=O)OC)C)C)C 16783,N1(C(c2c(CC)oc(C)c2)=O)CCCC(C)(C)C1CNC(=O)COCC(C)(C)C 16784,C=CC(C)(C)CC(=O)NC1CCCO1.C12(C)CCC(CC1)N(C(=O)CC)C2 16785,C(CNC(C1(S(C)(=O)=O)CCC1)=O)(C(C)C(C)C)NC(c1nc(CC)oc1)=O 16786,c1(CC(=O)NC2CC(CNC(c3cc(F)cs3)=O)C2)nnc(O)s1 16787,C1(Nc2c(OCCOC)cc(C(N)=O)cc2)CCc2nnc(C(F)F)n2C1 16788,C1(CNC(C=CSC)=O)CCCCC1Nc1ncc(I)cn1 16789,C1(NC(C2C(OC)CCC2)=O)CCN(Cc2ncc(C)o2)CC(C)(C)C1 16790,N1(C(C=CC)=O)CC2CN(N(C(=O)OC(C)(C)C)Cc3c(Br)ccnc3Br)C2C1 16791,C1(C(=O)NC2(CNC(c3c(C)[nH]cc3)=O)CCOCC2)CC12CCOCC2 16792,c1(OC)cc(C(=O)NC23CC2CN(C(C24CCC(OC)C2C4)=O)C3)cc(Cl)n1 16793,c1(CC)ccc(C(=O)N(C)CCNC(c2ccccc2CS(C)(=O)=O)=O)cn1 16794,c1(C(c2nnnn2CCSC)Nc2cnn(CCC)c2C)cc(Br)cc(F)c1O 16795,c1(C(=O)NC2CC(O)CN(C(c3ccnc(Cl)c3O)=O)C2)cnc2nccn2c1 16796,N(C(=NCCCC(C)(C)C)NC1CCC1)CC1C(C)COCC1 16797,C1(NC(=O)C=Cc2cccs2)CC2(CCN(C(=O)Cc3ccsc3)C2)C1 16798,C1(NC(c2cnn[nH]2)=O)CCN(C(c2nnc(O)cc2O)=O)C(C2CC2)C1 16799,C1(C(N(CCCNC(CCOC)=O)CCO)=O)CCCCN(C)C1=O 16800,c1(C(N2CCN(C(c3c(SC)ccs3)=O)C(CO)C2)=O)cccn2nncc12 16801,C(CCCCC(=O)NCC=C(C)C)NC1(n2cc(-c3cn(CC)nc3)nn2)CC1 16802,O=C(C1Cc2ccc(Cl)cc21)N1CCOCC1c1ncn[nH]1 16803,C(=O)(C1=NOC2(CCNC2)C1)N1CC(C)N(C(=O)Cc2ccc(F)cc2)CC1 16804,C1(C(=O)NCC2N(C(C(c3cccc(Cl)c3)CC)=O)CC2)CCc2cncn2C1 16805,N1(C(c2ccn(CC)n2)=O)CC2CN(Cc3ccc(C)cc3C)C2C1 16806,N1(C(CCCC)=O)CCN(C(=O)C(CC)CC)C(c2cc(F)cc(F)c2)C1 16807,C1(CC(NOCCCC)=O)CCN(C(c2ncoc2C2CC2)=O)CC1 16808,C(=O)(CC(F)(F)Cl)NCCOC1CCN(C(C2CC(CC(C)(C)C)C2)=O)C1 16809,CC1CC(C(=O)NC(C)CCNC(=O)C(C)(F)F)CC(C)C1 16810,CC(CC(=O)NC1C(C)(C)CN(C(=O)C2=CCCSC2)CC1(C)C)CC(C)(C)C 16811,Cc1ccc(CNC(C2(C(=O)O)CCCCO2)=O)cc1C1CC1 16812,CN1CCOC(C(=O)NCCC(O)CNC(c2cnc(N(C)C)nc2)=O)C1 16813,C#CC1(C(N2CC(COCC)C2)=O)CN(C(=O)Cn2cccc2)C1 16814,C(=O)(CCC(=O)N1CCOC(CNC(=O)CN2CCCC2=O)C1)OC 16815,c12c(C)sc(C)c1NC(=O)Cn1cc-2nn1.C1(C)(C(=O)OC)CCC1(C)C(=O)O 16816,N1(C(c2ccc(OC)cn2)=O)CCC(N2CCC(CCCO)CC2)C2(CC2)C1 16817,N1(C(=O)Cc2nc[nH]n2)CCC(C2CCCN(C(c3cc(CO)ccn3)=O)C2)C1 16818,N1(C(c2cnns2)=O)CC2CCCC2(Nc2cc(C(F)F)ncn2)C1 16819,c1(C(CC)=O)ccc(C(=O)NC2CC(NC(=O)C(C(C)C)n3cncn3)C2)cc1 16820,C=Cc1cnn(C)c1C(=O)NCC(C)N(C(=O)C(C)NC(=O)C(C)(C)C)C 16821,c1(C(=O)NCCNC(C2(n3cnnn3)CCOCC2)=O)cc2n(n1)CC(F)C2 16822,CC1CCN(C(=O)CCN2CCN(C)CC2)CCN1C(C1CC2(CCC2)CO1)=O 16823,CC(F)(C(=O)NC(CNC(=O)CSCC(=O)NC1CCCCC1)C1CC1)C(F)(F)F 16824,c1(C(=O)NCC(c2cccc(C)c2)NC(c2cnns2)=O)ncc(Cl)cc1F 16825,c1(C(=O)NC(CC(C)NC(=O)C=C(Cl)Cl)C)nccc2c1[nH]c1ccccc21 16826,C12CCN(CC1)CC(=O)N2CCO.C1(C(N2CC(C(N)=O)C2)=O)CCS(=O)(=O)C1 16827,N(C1c2ccccc2C2CC1C2)C(C1CCOc2ccccc2O1)=O 16828,C(=O)(C1=CS(=O)CCC1)NCCN(CCC)C(c1cn(C(F)F)c(C)n1)=O 16829,N1(C(c2nccc(C)n2)=O)CC(N(C)C(c2oc(C)cc2C)=O)C2(CC2)C1 16830,c1(OC)cc(C(=O)NCC(O)CN(C(=O)C=C2CCOCC2)C)c(OC)cc1Cl 16831,Cc1ccc(N)c(C(N2CCC(C(C)NC(C3C(C)C3C)=O)C2)=O)c1 16832,c1(C(N2CCN(C(=O)Cc3cccs3)CC2)=O)cn2ccc(Cl)cc2n1 16833,N1(C(c2cc(C)n(Cc3ccccc3)c2C)=O)CCc2cc(C(=O)O)ccc21 16834,C1(C)(CC)C=C(C(=O)N2CC(C)(C(=O)NC3CN(C(C)C)CC3C)C2)C1 16835,C1(C(=O)NCC(CC(C)C)NC(=O)COC(C)C)CCC2C(C1)C2(F)F 16836,c1(OC)cc(C(N2CCCCC2C2CCN(C(=O)CC(C)=C(C)C)C2)=O)ncn1 16837,Cc1cc(C(F)(F)F)ccc1S(=O)(=O)NCC1CCc2cc(F)ccc21 16838,N1(C(CCC)=O)CCCC1(C)C(=O)NCCN(C1CCCC1)C(C)=O 16839,C1(COC)(NC(=O)CCNC(N)=O)CCN(C(=O)CC2CCNC2=O)C1 16840,C(=O)(C1CCCc2nn[nH]c21)NCC(C)(C)NC(C(c1ccc(F)cc1)C)=O 16841,c1(C(N2CC(NC(c3cnc(C)[nH]3)=O)C(F)C2)=O)c(F)cc(C(F)(F)F)cc1F 16842,C1(C(=O)NCC(c2ccc(F)cc2)NC2CC2)CC2CC2N1C(c1cnc(Cl)s1)=O 16843,c1(C(=O)NCC2N(C(c3nc(NC(C)=O)sc3)=O)CC2)cc2c(s1)CCOC2 16844,C(=O)(C(F)CC(C)(C)NC(=O)C(C)=C1CC1)N1CC(OC(=O)NC)C1 16845,c1(CCC(=O)NC2CN(C(C(CSC)O)=O)CC2C(F)F)ccc2c(c1)CCO2 16846,N1(C(c2ncc(C(=O)OC)nc2)=O)CC2CCN(C(=O)C(C3CCC3)OC)C2C1 16847,O(NC(=O)C(C)(C1CC1)N(C)C(c1ccc(SC)o1)=O)CCCOC 16848,c1(COC)nc(NCc2csc(Br)n2)cc(N2CCC(Cc3ccn(C)n3)C2)n1 16849,N1(C(C(C2CC2)OCC)=O)CCN(C(c2c([N+](=O)[O-])cnn2C)=O)CC(C)(F)C1 16850,CC1CC(O)CCN(C(C2CC(CNC(=O)C(O)CC(F)(F)F)C2)=O)C1 16851,c1(C(N2CC(C#C)(CO)C2)=O)nn(C)c2c1CCC2 16852,C(=O)(CCCN(C)C(=N)NCCNC(=O)C(O)(c1ncnn1C)C1CC1)OCC 16853,S(=O)(=O)(c1ccc(N2CCC(O)C(F)C2)c(C#N)c1)NC(c1cccs1)(C)C 16854,c1(OCC)ccc(C(N2CC(CO)(NC(c3ccc(F)o3)=O)C2)=O)c(F)c1F 16855,N1(C(c2n(CC)cnn2)=O)CC(NC(c2nc(Cl)cs2)=O)CC(C)C1 16856,C(=O)(CCCCCO)NC12CC(C(N3CCCC3c3ccc(Br)cc3)=O)(C1)C2 16857,C1(N(C)C)CCCN(C(C2CC23CC(NC(c2ccc(Cl)cn2)=O)C3)=O)C1 16858,C(=O)(C(O)C(C)(C)C)N1C(C(=O)NC(C2(CC(F)F)CCC2)C)CCC1 16859,CC1CCC(O)C(NC(=O)C(C(C)(C)C)NC(=O)C=CC2CC2)C1 16860,CC1CCc2nc(C(=O)NC3CCCC3NC(=O)CC3CC=CC3)cn2C1 16861,CC1(C)C(C(=O)NC2(CNC(C3CC3c3ccccn3)=O)CCOC2)C1(C)C 16862,c1(C(=O)Nc2c(C#N)scc2)ccc(F)c2c1CCC2 16863,c1(C(N)=O)cncc(NC(=O)C(C2CCC2)NC(=O)Cc2cn(C)cn2)c1 16864,c1(CN(C(c2cscc2Br)=O)C2CC2)cccc(F)c1 16865,CCC(CCCC(=O)OCC)NC1CN(C)CC(F)(F)C1 16866,c1(CC)ccc(OCCC(=O)NCC2CCN2C(=O)CC(CC)C2CCC2)cc1 16867,c1(NC(CC(CC)NC(C2CCC(=C)CC2)=O)=O)cccc2ccccc12 16868,C1(C(N2CC(SC)C2)=O)CCN(C(C2C3CCCC23)=O)C(C)C1 16869,c1(NC(N2CCCC(c3noc(C(F)F)n3)C2)=O)cc(F)nc(F)c1 16870,c1(CN2CC(C(N3CC4C(C3)C4(F)F)=O)NCC2)c(Cl)ccnc1Br 16871,C1(C(=O)NCCC=C=C)CN(C(=O)Cc2ccccn2)CCN1C 16872,C(=O)(C(CC(C)C)OC)NC(C(N1C(CC)(CC)CC1)=O)CC1CC1 16873,N1(C(C(CCCC)O)=O)CCc2[nH]nc(C(=O)Nc3cc(Cl)nc(Cl)c3Cl)c2C1 16874,C1(OCC(C)C)CN(C(=O)NCCC(C)SCC)C1.C(C)(C)(C)O 16875,c1(C(=O)NC2CCC(NC(c3nocc3C3CC3)=O)C2)cc2ccc(F)cc2o1 16876,Cc1[nH]nc2c(C(N3CC4(CNC(=O)Cc5cc[nH]n5)CCC3C4)=O)cccc12 16877,c1(-n2cc(C(C)N(C)C(c3nn(C)nc3Br)=O)nn2)cc(F)cc(F)c1 16878,n1(CC(=O)NC(C2CCCC2)CNC(=O)C2=CCC2)nc2n(c1=O)CCCCC2 16879,C(C)(C(C)(C)C(=O)NC1COC(C(C)C)C1)NC(c1cccc(CC)n1)=O 16880,N1(C(CCC=CCC=C)=O)CC2CC(C)N(Cc3ncc[nH]c3=O)C2C1 16881,c1(OCC=C)ccccc1C(=O)NCC(=C)CCNC(=O)Cc1sc(C)nc1C 16882,C#CC1(OCC(=O)NCC(=O)NCCc2noc(CC)n2)COC1 16883,n1(CCC)cc(C(=O)NC2C3CC2N(C(=O)Cn2nnnc2C(C)C)C3)c(C)n1 16884,C1(C)(CNC(C2C(CCC)C2)=O)CCN(C(C2(CCC)CCC2)=O)C1 16885,N1(C(C2CCCN(C(CCC(=O)NCC)=O)C2)=O)CCCCCC(N(C)C)C1 16886,N1(C(CC(=C)C)=O)CCC2(CC1)CC(NC(=O)Cc1cnn(C)c1)CO2 16887,C#CCC(CC(F)F)C(=O)NCC(C)CCNC(=O)COCCNC(C(=O)OC)=O 16888,Cc1oc(C(N)=O)cc1S(=O)(=O)N(C)CNCc1cn(C2CCC3CC3C2)nn1 16889,C123COC(C1)(C2)C(=O)NCC=CCNC3=O.c1(COC)ccc(C)nc1 16890,C(=O)(C(C)C(O)CC(C)C)N1C2(C(=O)NCCn3c(CC)ncc3)CC(C1)C2 16891,C1(C(C(=O)NCCC(=O)N(C)C)NC(C(=O)NCCOC)=O)CC=CCC1 16892,c1(NC(C2C3CCC(C3)N2Cc2ccc(Br)cc2O)=O)ccc2nc(O)[nH]c2c1 16893,C1(C(=O)NCC2CN(C(C(C)(C)c3nccs3)=O)C2)CCCC2C1C2(F)F 16894,C(=O)(CCC(=O)N1CCN(C2CCC2)CC1)NCC(CC)CC 16895,N1(C(c2c(C)nn[nH]2)=O)CCC(C(=O)NC2C(O)CC2O)=C(F)C1 16896,c1(C(N(CCOC)CCF)=O)conc1C(C)NC(=O)C(C)N(C)C 16897,C=CCC(C)(N)C(=O)NC1CC(C)CCC1C 16898,c1(C(=O)NC2C(CNC(C(CC)NC(N)=O)=O)CC2)cccc2c1OCC2 16899,c1(C(N2CC(CN(C(CN(C3CC3)CC)=O)C)C2)=O)cnn(CC)n1 16900,CC1(C)CCC(C)(C(=O)NC2CC(O)CN(C(=O)Cn3cnccc3=O)C2)CC1 16901,C1(NC(C(N2CCCC(NC)CC2)=O)=O)CCC(F)(F)CC1F 16902,C1(OC)CCCC(C(=O)NCC(C2CC2)N(C(=O)C(C)=C2CCCC2)C)C1 16903,N1(C(c2nc(COC)sc2)=O)CCCC(C(C)(O)CNC(=O)CCF)C1 16904,C1(NC(C2CCCC(C)(C)CC2)=O)CCC2(CCN(C(=O)C3=CCCS3)CC2)C1 16905,C1(OC)CN2CCCC2(C(=O)NCC(C)(C)NC(=O)Cc2ccc(O)cc2Cl)C1 16906,C12(C(=O)NC(CC)CN(C)C(C3CC(C)(C)C3)=O)CC1COC2(C)C 16907,C1(CNC(Cn2c(C(C)C)ncc2)=O)CC2CCCCC2N1C(=O)CC(C)O 16908,C1(F)(C(N2CCN(CC3CN(C(C4CCC(C)O4)=O)C3)CC2)=O)CC2(CCC2)C1 16909,C1(CNC(C(C)(C)OC)=O)CCC2(CCC2)C1NC(c1ccc(C)cn1)=O 16910,c1(C(=O)NC2CC(CNC(c3c(COC)noc3)=O)C2)ccc(C(N)=O)c(Cl)c1 16911,c1(OC)cccc(C2=NOC(C(=O)NC3CCCC(C4CC4)C3)C2)c1 16912,c1(NC(CCNC(CCCOCC=C)=O)C(C)C)ncc(C)c(S(C)(=O)=O)n1 16913,C(=O)(NNc1cc(Br)ccn1)NCc1cc(C)c(C(N2CCC(C)CC2)=O)cc1 16914,C1(COC)(CNC(=O)CSC2CC2)CCCN1C(N1CCC(C)C1)=O 16915,CC1(CO)CCN(C(C2(NC(C3(C)CC=CCC3)=O)CSC2)=O)C1 16916,CC(O)CC(C)(C)CNC(c1cc(C2CC2)on1)c1nnnn1CCCF 16917,CC(C(=O)NCC1CCC(NC(C2C=CC=CC=C2)=O)CC1)C(F)F 16918,N1(C(C(C(C)C)SC)=O)CC2CCCC(NC(c3cn(CCCF)nn3)=O)(C2)C1 16919,C(=O)(CC=C(Cl)Cl)N(C1CCN(C(=O)COCC=Cc2ccccc2)C1)C 16920,c1(C(=O)NCC#CCNC(C2C(C)(C)COCC2)=O)c(N)cc(F)cc1Cl 16921,C12(NC(c3cnccn3)=O)CCOCC1CN(C(c1ccc(Cl)c(Cl)c1O)=O)C2 16922,N1(C(CN(CC(C)(C)C)C)=O)CCN(C(C2CC3C=CC2O3)=O)C(C2CC2)C1 16923,N1(C(C2CCC(C)O2)=O)CCC2(NC(c3ccnc(F)c3)=O)CCCCCC12 16924,Cc1cc(C(N2CCCC(CC(N3CC(CO)CC3CO)=O)CC2)=O)nc(O)c1 16925,C1(CNC(=O)CCc2cncnc2)CC(F)CN1C(C1OCCCO1)=O 16926,c1(NC(C(=O)NC2C3CC(N)CC2C3)=O)ccc2c(c1)CCC(=O)N2CC(F)F 16927,c1(CC)onc(C)c1CNC(=O)CCN(CCO)C(C12CCCCC1C2)=O 16928,C1(OCCCC)CC(OC(c2scc(C)c2I)=O)C1(C)C 16929,N1(C(c2sc(CC)c(C)c2)=O)CCCC(C2(NC(c3cnsn3)=O)CC2)C1 16930,C(c1cccc(C#N)c1)=CC(N1CCN(C(C(CC)N(CC)CC)=O)C2C1C2)=O 16931,c1(CC)ccc(NC(=O)CN(CCCOC)CCCO)cc1 16932,C(=O)(C1=NN2CCCN=C2N1)N1CCN(C(C=CC)=O)CC1CC(F)(F)F 16933,c1(C(=O)NCCCNC(CC2(OC)CC2)=O)cc(=O)n(-c2ccccc2)[nH]1 16934,c1(C(N2CC(C(=O)NC3CCN(C)C3=O)(COC)C2)=O)ccccc1C(C)C 16935,C(=O)(C(F)CC(CC)CC)NC(CC#C)(C)C(N1CCC2(C=CCO2)C1)=O 16936,C1(NC(C(CCC)(C)C)=O)CCC2CC1CN2C(c1ccc(F)cc1OC)=O 16937,c1(OCC)cc(CN2CCCC(C)(C(F)F)C2)ccc1OC 16938,c1(CC(=O)NCC2C(C)CCN2C(c2cnc(Cl)nc2)=O)cccc(F)c1Cl 16939,O=C(CC(C(F)F)n1ccnc1)NCCCNC(=O)C=Cc1nc[nH]n1 16940,c1(CCC)cc(C(=O)NC(C)(C)CNC(=O)C=C(CC)CC)ccc1Cl 16941,c1(C(=O)NCC2C(NC(c3c(CC)nccc3)=O)C2)cc2nc[nH]c2cn1 16942,c1(C(=O)NC2CCN(C(C(COC)C)=O)CC2F)nc2ccccn2c1F 16943,CS(=O)(=O)c1ccc(Cl)cc1NC(=O)C(=O)NCC(F)C1CCC1 16944,C1(NC(CC(=C)C)=O)CCC2CN(C(C3CCN(CC4CC4)CC3)=O)CC2C1 16945,C1(C)(C(N(C2(C(=O)NCC(C(C)O)O)CCC2)C2CC2)=O)CCN(C)CC1 16946,C1(NC(CCN(C(C(C)O)=O)CCCO)=O)CCNC1=O 16947,C1(C(=O)NCCC2COCCN2C(C2CCSCC2)=O)Cc2ccccc2O1 16948,Cc1c(C(=O)N(C2CCN(C(C34CC(C(C)C)(CO3)C4)=O)C2)C)cccc1Cl 16949,N1(C(c2nn(CC)c(C3CC3)c2)=O)CC2CCC(Nc3ncncc3I)CC2C1 16950,c1(C(=O)NC(CC)CN(C(=O)COCC(C)C)C)cc(C)nn1C1CC1 16951,c1(C(=O)NC2C(NC(C3(C#C)CC3)=O)CCC2)c(C)cc[nH]c1=N 16952,c1(C(N2CCC(C(CNC(C(C)SC)=O)C)CC2)=O)ncc(Cl)cc1F 16953,C1(CCC=C)(C(=O)NC(C)CC2CCOC2=O)CN(C(c2csc(O)n2)=O)C1 16954,c1(C(=O)NC2C(N(C(CC(C)C3CC3)=O)C)CCCC2)ncc2cc(Cl)ccn12 16955,Nc1c(C(=O)NCC2CN(C(=O)CCSCC(N)=O)CCO2)cnc2ccnn12 16956,C(=O)(C#CC(C)(C)CNC(=O)Cc1cn(C)cn1)NC(C(=O)OC)CCF 16957,c1(C(N2CC(NC(C3CC(OC)C3)=O)C2)=O)cnoc1C1CC1 16958,C(=O)(C(C)(C)C(C)NC(=O)COc1cc(C)on1)NCCCOCC#C 16959,c1(C(=O)NCCNC(N2CCCC2c2ccncc2)=O)ccccc1Cl 16960,N1(Cc2cc(CC)cc(C)c2)CCn2cccc2C12CCNC2 16961,C(N=c1[nH]c(C(F)F)ccc1OC)C1(c2c(OCC)cccc2)CCC1 16962,C1(CN(C)C(c2csc(O)n2)=O)COCCN1C(c1cc(C2CCCC2)[nH]n1)=O 16963,N1(CC)C(=O)CCC1C(=O)NCC=CCNC(=O)Cc1ccc(CSCCCOC)cc1 16964,C1(NC(=O)Cc2ccc(Cl)cc2Cl)CC2CC(C1)N(C(=O)C(O)C1CC1)C2 16965,c1(C(=O)NCC2N(C(CNC=O)=O)C3CCC2C3)cc2c(F)cc(Cl)cc2[nH]1 16966,C1(CNC(C2C(C)CC(=O)N2)=O)CCN(C(c2cc3sccc3s2)=O)CC1C 16967,c1(C(N2C(C(=O)Nc3cc(Cl)cnc3Cl)CC(C)C2)=O)ccc(F)c([N+](=O)[O-])c1 16968,C#CCCCCCC(=O)N1CCCC1c1cn(CCCCCCC=C)nn1.CC#N 16969,c1(NC)ccc(F)cc1C(N1CCCCC1CNC(=O)CC1(C)CCCO1)=O 16970,c1(C(N(C)CC2CCCC(NC(CN(C(C)C)C)=O)C2)=O)ccc(CO)c(F)c1 16971,N1(C(c2c(C)[nH]nc2CO)=O)CC2(C1)CN(C(C1COCCN1C=O)=O)C2 16972,C(=O)(CC1=NN(C)C(=O)C1)NC(C(C)NC(CCCNC(COC)=O)=O)(C)C 16973,C1(C(N(CCN(C(c2n[nH]cc2Cl)=O)CC)CC)=O)CCC2(CCOCC2)CO1 16974,c1(OCC(=O)N(CC(O)CNC(C23CCCC2C3)=O)CC)ccc(C(C)O)cc1 16975,C1(C(NOCC=C)=O)CC2(CCN1C(=O)CC(C)C(C)(C)C)CC2 16976,c1(NCC2(NC(C3CCNC3=O)=O)C(C)CCCC2)ncc2c(n1)CCOC2 16977,c1(C(N2C(C)CC(CNC(c3ccsn3)=O)C2)=O)sc2nccnc2c1N 16978,CC(C)(C)C(C)(C)C(=O)N1CCOC(C(N2Cc3c[nH]nc3C2)=O)C1 16979,N1(C(C2CC(SC)C2)=O)CC(C)CCC1CNC(c1[nH]cnc1C)=O 16980,C1(NC(c2cc(C)cc(C)n2)=O)CC2CCC(C1)N2C(=O)CCCc1cnn[nH]1 16981,C(CC1CC1)(C(=O)NC1COCC1NC(=O)C=CSC)OC 16982,c1(C(N2CC(NC(=O)C(C)(F)F)CC(C)C2)=O)cc2c(Br)cccc2c(=O)o1 16983,c1(NC(C(C)(C2CCC2)NC(=O)C(C2CCOCC2)F)=O)ccc(F)cc1 16984,C1(NC(=O)C=CC2CC2)CCC1C(=O)NCc1cnc[nH]1 16985,c1(OCCC(=O)NCC2COCCN2C(c2cccc(F)n2)=O)cccc(F)c1 16986,Cc1ccc(S(=O)(=O)N(C2CCNCC23CC3)Cc2ccsc2)cc1[N+](=O)[O-] 16987,c1(C(CC(=O)N2CCC(CC(F)F)C2)O)ccc(OC(F)(F)F)cc1 16988,C1(CNC(=O)C=CC=C(Cl)Cl)CCCC2(CN(C(=O)CCC(F)(F)F)C2)O1 16989,C1(C(=O)NC(C2CN(C(CC3CC(C)C3)=O)C2)C)NC(=O)OC1C 16990,C(=O)(CC(C)CC(C)C)NC1C(CC(=O)NC(CCCCC)C)CCC1 16991,C(=O)(C(CCC1CCC1)NC(=O)NCc1cnsc1)NC 16992,Cc1ncccc1CC(N1CCC(N(C(=O)CN(CC(C)(C)C)C)C)CC1)=O 16993,c1(C(CNC(c2cncn2C)=O)NC(C2C(C)OCC2)=O)ccc(F)cc1 16994,C1(C)(NC(COC(CNC(CC2CC(=C)C2)=O)(C)C)=O)CCOCC1 16995,C12(C(=O)OC)CCCC1(C(=O)N(CCNC(C1C3CC4C(C3)C14)=O)C1CC1)C2 16996,C12(C(N(CC(N3CC(C(=O)NC)C3)=O)CC(C)C)=O)CC1CNC2=O 16997,Cc1coc(C2CC2)c1C(=O)NCCOC(C)(C)CNC(c1cnc(C)n1C)=O 16998,c1(C(N2CCC(NC(CS(C)(=O)=O)=O)C2)=O)c(Cl)ccc(F)c1F 16999,C1(SC)CC(C(=O)NCCN(C(=O)Cc2ccsc2)C(C)C)C1 17000,c1(C(=O)NCC2N(C(C3COC(=O)O3)=O)CCC2)cn(C(F)F)nc1C(F)F 17001,C1(NC(COCCN(C)C)=O)CCCC12CCN(C(c1ccc([N+](=O)[O-])o1)=O)C2 17002,C1(CN(CC(=O)NC(c2ccccc2)CC)C)(OC)CCOCC1 17003,C1(OC)CN(C(c2ccc(C3CC3)o2)=O)C(C)(CNC(c2cnn[nH]2)=O)C1 17004,CC(C)C(N=[N+]=[N-])C(=O)N1C(C(=O)NCCOC2(C)CCC2)CCC12CC2 17005,C(=O)(C#CC1(C)COC1)N1C(C2(C(N3C(C)C(=O)NCC3)=O)CC2)CCC1 17006,c1(C(=O)NC(C(C)C)C(=O)NCC2CC(C)(C)CCO2)cncc(C#N)c1 17007,C1(CCNC(COC)=O)CN(C(c2cc(C(F)F)n(C)n2)=O)CC1C 17008,CCCC(O)CC(=O)NCC(CNC(c1ccc(CCC(F)(F)F)cc1)=O)CO 17009,Cc1nc(=N)[nH]cc1C(N1CCOCC(CNC(=O)Cc2ccc(F)cc2)C1)=O 17010,C#CCC(C)(C(=O)Nc1ccc(CC)c(F)c1)NC(C1CCN(CC)CC1)=O 17011,N1(C(=O)C=Cc2ccsc2)CC2CN(c3ncncc3F)CC2C1 17012,c1(OC)cccc(C)c1NC(=O)CCCCCNC(C1NC(=O)OC1C)=O 17013,N1(C(Cc2ccn(CC)n2)=O)CCN(C(c2cc(C)ccc2O)=O)C2CCC12 17014,N1(C(c2c(C)ocn2)=O)CCC2(CC1)COC(CNC(C1(C(N)=O)CCC1)=O)C2 17015,c1(C(=O)NC(C(C)NC(=O)Cn2cnnn2)C)cncc(Br)c1 17016,CC1N(C(C2(C)CCN(C(C3CC(C)(C)CO3)=O)CC2)=O)CCC1(C)C 17017,N1(C(=O)CN2CCOCC2)CCN(C(c2ccncc2Cl)=O)C2CC12 17018,C1(C(N(CCC(C(C)(C)C)NC(C(CCC)O)=O)C)=O)CN2CCN1CC2C 17019,N1(C(c2ccc(C)s2)=O)CC(C)CCC1C(N1CCCC(O)(CO)C1)=O 17020,C(=O)(CCC(=O)NC(C)(C)CC(=O)N1CCCCC1C(C)CO)NCCC 17021,C12(C(N(C)CC3CCCN3C(C3CC4CCC3C4)=O)=O)CC3CC(CC(C3)C1)C2 17022,N1(C(C)=O)CCC2OC(=O)OC2C1.C12(CN(CC)C1)n1cc(nn1)COC2=O 17023,c1(C(N(C(C)CNC(c2n[nH]c(=N)[nH]2)=O)C)=O)cncc2ccccc12 17024,c1(OC)cc(C(=O)NCC2CC2NC(C2(C)CC=CC2)=O)on1 17025,C1(CC)CCN(C(C23CCC(NC(C4CCCCC4)=O)(CC2)C3)=O)CCO1 17026,N1(C(c2c(CC)con2)=O)CCC(NC(C2(Br)CC23CCC3)=O)CC1C 17027,c1(OCC)cc(C)c(NC(C2CC(O)CN2c2ncncc2I)=O)cc1Br 17028,c1(C(N2CC(O)(CC)C2)=O)nc2nc(C(=O)O)ccn2n1 17029,C(=O)(C(C)(C)C(=O)N1CCC(N(CCO)C(C2CCCC(C)(C)C2)=O)CC1)NC 17030,c1(C(N2C(C)CC(CNC(c3cncc(F)c3)=O)CC2)=O)nn(C)c2c1CCC2 17031,C1(C(=O)NC2CC(N(C(c3ccnc(C)n3)=O)C)C2)CCCCC12OCCO2 17032,N1(C(c2n(CC)nnc2)=O)CCN(C)CC1C(=O)NCC1CC2CCCC2C1 17033,C(c1ccc(Cl)c(Cl)c1)=CC(N1CC2C(NC(=O)CC3CCCC3(F)F)(C2)C1)=O 17034,C1(C(=O)NC2(C(N(C)Cc3cc(C)no3)=O)CC(O)C2)CC(C)CCO1 17035,C=CC(C)CC(=O)NCCn1cc(CNC(c2cncs2)=O)nn1 17036,C1(C(=O)NC2CC(CCNC(c3cccc(C(F)F)c3)=O)C2)CC2CCCC2C1 17037,c1(CNC(c2cccc(Cl)c2)CO)cc(Cl)cc2c1CCC2 17038,N1(C(C(CC=C)C)=O)CCN(C(C2CCN(CC)CC2)=O)CC1C 17039,N1(C(CC)=O)CC(N=c2nc3scnc3c(NCc3ccc(C(F)(F)F)s3)[nH]2)C1 17040,C1(C(N2CC(CN(C)C)C2)=O)CN(C(c2cn(C)cn2)=O)CCC1O 17041,CC(C(=O)N1CCOCC(CNC(=O)C(C)(C)CO)C1)C(F)(F)C(F)F 17042,c1(C(=O)NCC(C)C(=O)NC2CC2)cc(=O)n(C)cn1 17043,c1(C(N2CC3(CCN(C(C(CC(=C)C)C)=O)C3)C2)=O)cc([N+](=O)[O-])c(C)cc1C 17044,C1(CC)CCCC(C(=O)OC)C1.N12CCC1C(=O)N1CC(C1)C2=O 17045,C(=O)(C(C(C)(C)C)NC(=O)CCc1ccc(C)nc1)NCc1cn(CC=C)nn1 17046,C(=O)(C(C)CC(C)(C)C)NC1(c2nnc(C3C(C)OCC3)o2)CCC1 17047,N1(C(C(CC)CC)=O)CCN(C(=O)CSc2ccncc2)C(CO)C1 17048,C1(c2onc(-c3n(C=C)ccn3)n2)CCCSC1 17049,C(=O)(C(F)(F)CCn1cccn1)NC(CCNC(C(C(C)C)N(C)C)=O)C 17050,N1(C(C(CCC)F)=O)CCN(C(c2cc(Cl)nn2C)=O)C(CCO)C1 17051,c1(C(N2CC(C)(NC(=O)CN3CCOCC3)C2)=O)ccnc(C(C)(C)O)c1 17052,C1(NC(C2C(=C)C2)=O)CC2(C1)CC(NC(=O)C(C)Sc1ccccc1)C2 17053,c1(N2C(C)CC(CNC(C3(C)C(CC)CCC3)=O)C2)ccc(C#N)nn1 17054,c1(C(=O)NCCC(CCNC(C2CC(=C)C2)=O)C)cc(Br)ccc1OC(C)C 17055,N1(C(c2cc(C(C)=O)c(C)o2)=O)CCN(C(c2cscc2C)=O)CC1CF 17056,c1(CC(=O)NC2CC2C(=O)Nc2ccc(OC(F)(F)F)nc2)c(F)cccc1Cl 17057,c1(C(=O)Nc2n(C)nc(-c3ccc(Cl)cc3)n2)cc(Cl)ccc1Cl 17058,C#CCC(O)C(=O)N(C)CC1CN(C(=O)CC2CCCCC2)CCO1 17059,Cn1nc2c(c1C(N1CCC(NC(C3CCCOCC3)=O)C(F)C1)=O)COCC2 17060,C1(NC(c2c(OC)cc(C)cn2)=O)CCC2(CCN(C(=O)CC3(SC)CC3)C2)C1 17061,S(=O)(=O)(c1cnc(NC2CC3CCCC3C2)c(Cl)c1)NCCCCC 17062,C1(C(=O)NCC(C)NC(=O)C(C)(C)n2cc(Cl)cn2)(OC)CCCCC1 17063,N1(C(C(C)C(C)(C)C)=O)CC2CC(O)C1C2NC(=O)C=CC1(C)COC1 17064,C(=O)(N=c1cc(Cl)nc(C)[nH]1)c1c(OC)nc(-c2ccc(C)nc2)cc1 17065,N1(C(c2c(O)nc(CC)c(C)c2)=O)CCC2(CCCN(C(=O)C3=CCC3)C2)C1 17066,C1(C2CN(C(c3scnc3Cl)=O)C2)(NC(c2cccc(N)n2)=O)CC1 17067,C12CCCCN1C2=O.c1(CCC(=O)Nc2coc(CC3CC3)n2)cnccn1 17068,N1(C(C2CC2(C)C(F)F)=O)CC(C(C)=O)C2(CC2)C1.C1(CC)(CN(C)C)CC1 17069,C1(NC(C2CCC2(F)F)=O)CC2CC1CN(C(c1cccn3nccc13)=O)C2 17070,Cc1nc(NC2CCCN(C(=O)Cn3nnnc3C(C)C)C2)cc(Cl)n1 17071,c1(C(=O)NCCCN(C(c2c[nH]c(C#N)c2)=O)CC)ccc2c(c1)COC2 17072,c1(CN2CC(CNC(c3cc(C)c(C)s3)=O)C2)ccc(F)cc1F 17073,C(=O)(C1=C(Cl)CCC1)NC1C(NC(c2ccn(C(CC)CC)n2)=O)CC1 17074,CC(C)C(CCNC(=O)OC(C)(C)C)C(=O)N(C)CCNC(=O)C1=CCCSC1 17075,c1(NC2C(CC)(CC)C(OC)C2)ncnc2ncn(-c3ccccc3)c12 17076,C(=O)(CC(F)(F)F)CC(=O)N(c1cccc(-c2noc(C(F)(F)F)n2)c1)C1CC1 17077,CC1=C(C(=O)N2CCC(F)C(NC(c3cnc(C)o3)=O)C2)S(=O)(=O)CCO1 17078,N1(C(=O)Cc2cccnc2Cl)CCC2(CCC2N2CCCC(F)C2)CC1 17079,C1(CC)CCN(C(C2CC(=O)N(C)C2)=O)C(C(=O)N(CC)Cc2cccs2)C1 17080,Cc1cc(F)ccc1NC(=O)C(C)CN(C)Cc1cn(C)nc1I 17081,C=CCCCCC(=O)NC1CN(C(C2CCCCN2N=O)=O)C(CC)(CC)C1 17082,c1(C(=O)NCC(CC)(C)NC(c2cc(Br)co2)=O)cncc(OC)c1 17083,Cn1cnc(C=CC(=O)NCCC2CSCCN2C(=O)CCC(N)=O)c1 17084,N1(C(c2ccc(C)c(C#N)c2)=O)CC2(CCN(C(c3ccc(Cl)nc3)=O)CC2)C1 17085,Cc1ccc(SCCC(=O)N(C)CC2(NC(=O)CCc3csc(C)n3)CC2)cc1 17086,c1(C(=O)NCCN(C(C2(CC)CCNC2=O)=O)C2CC2)nccc2ccn(C)c12 17087,N1(C(c2scc(CC)c2)C(=O)NCC2CCCO2)CCN(C)C(=O)C1C 17088,C#CCC(C)C(=O)NC(CNC(c1cnc(COC(C)(C)C)s1)=O)CC(C)C 17089,c1(CC(N2CCCC(CNC(C3C(C(=O)OCC)C3)=O)C2)=O)ncc(F)cc1F 17090,C1(CNC(CC2C(C)OCC2)=O)CCN(C(=O)CC2CC3(CCO2)CC3)CC1O 17091,C(=O)(CC(CN(C)C)CC(C)C)NC(C1(O)CN(c2cc(OCC)ncn2)C1)C 17092,C1(NC(=O)CCCCCn2cc(C3CCOC3)nn2)CCNCC12CCC2 17093,C1(CNC(=O)Cc2cccs2)CCC1C(N1CCC1C(N)=O)=O 17094,C1(CC)CN(C(=O)CC2CCC2(C)C)CCN1C(=O)CN1CCCCS1(=O)=O 17095,c1(C(N2CCCC(NC(C3C(C)C3)=O)C2)=O)cc(S(N)(=O)=O)cc(Cl)c1Cl 17096,C1(C(N2CCC(OC3CC3)C2)=O)COCCN(C(C2(O)CCCCCC2)=O)C1 17097,N1(C(C(C)CN(C)C(C2(CO)CCCC2)=O)=O)CCC(N=[N+]=[N-])C1 17098,C(=O)(CCOC(C1CCCC1)=O)NC(COC(C)C)C.OCC 17099,c1(CC(N2CCC(COC)(NC(=O)CCC(C)SC)C2)=O)ccc(C)c(F)c1F 17100,c1(OCC(=O)NCC2(CNC(c3[nH]c(=NC)sc3)=O)CCC2)ccc(F)cc1Cl 17101,CC(C)(C)CC(C(=O)NCc1cccnn1)NC(=O)CCCC#N 17102,CCCC(C(=O)NC(c1nc[nH]n1)C1CC1)NC(=O)C(CCC)NC(N)=O 17103,Cc1oc2ccccc2c1C(N1CCCC(C(C)NC(C2SCCS2)=O)C1)=O 17104,N1(C(C(C)=C2CCCC2)=O)CCC(C)(C)C1C(=O)N(CCCCCO)C 17105,c1(NC(C2C(CC)C2)=O)ccc(NC(C2CN(CC(F)(F)F)C2)=O)c(C)c1 17106,c1(OC)ccc(F)c(CC(=O)NC(C)CCNC(=O)C(F)CC2CCCCC2)c1 17107,C(c1cccc(F)c1F)=CC(=O)NC1C(NC(C(CC)N(C)C)=O)CCC1 17108,c1(C(CC)CNCc2cn(C3CC3)nn2)ccc(Cl)cc1 17109,N1(C(c2cc(OC)c(F)c(F)c2)C(=O)NC(C)C)CCS(=O)(=O)C2COCCC12 17110,C1(CC(=O)NCC2CN(C(c3nc(COC)sc3)=O)C2)CCCCC1C 17111,c1(CN(CC(=O)NCC2C=CCN2C(=O)CCc2cnoc2)C)ccccc1Cl 17112,c1(C(C)(C)NC(=O)NCC23CC(CO2)C3)ccc(O)cc1F 17113,CCCCCCC(C)C(=O)N1CCC(O)(CCNC(c2csc3nccn23)=O)C1 17114,c1(NCCc2c(C)nc[nH]2)cc(N(C)Cc2cccc(F)c2)ncn1 17115,c1(OC)cccc(OC)c1C(=O)N(C)CCN(C)C(C1CC1(F)Br)=O 17116,N1(C(C2=CCCCC2C)=O)CC=C(CC(=O)NCCC2OCCC2C)CC1 17117,C1(CNC(C2CN(C)C(=O)C2)=O)CN(C(c2cccc(C3CC3)c2)=O)CCCO1 17118,c1(C(=O)NCC(CC)NC(c2ncccn2)C2CC2)cc(C2CC2)sn1 17119,N1(C(C(C)CC(F)(F)F)=O)CC(CNC(=O)CS(C)(=O)=O)CC12CCOCC2 17120,CC1(C)CC(NC(C2CCCN2CC(F)(F)F)=O)CN1C(c1cncs1)=O 17121,C1(C(N2CC(c3nc(C)on3)C2)=O)CCC=CC1NC(c1cc(C)sn1)=O 17122,C=C(C)CCCC(=O)NCCC(O)C(=O)N(CCCN(C)C)CCC 17123,Cc1ccc(C(F)(F)C(=O)NC2CCC(NC(C3CCNC3=O)=O)C2)cc1 17124,c1(COC)cccnc1OC.C12CC(C1(C)C)CNC2=O.C1(=O)CC2(CC2)N1 17125,CC(CCS(=O)(=O)c1ccc(Cl)c(Cl)c1)NC(=O)CC1CCN(C2CC2)C1 17126,CC1CN(c2nnco2)CC1NC(=O)Cc1cccc(C(N)=O)c1 17127,Cc1cc(C(=O)NCC(C)N(C)C(C2CCN(C)C2=O)=O)cnc1C(F)F 17128,Cc1nn(C)c(=O)c(C(=O)NCC2CN(C(=O)C3=CCCS3)C(C)(C)C2)c1C 17129,C#Cc1ccc(C(=O)N(C(CNC(c2cnn(C(C)C)n2)=O)CC)C)c(C)c1 17130,C1(NC(=O)C2=CCCCCC2)CCN(C(c2cc(C3CC3)no2)=O)CCC1(F)F 17131,CC1CCN(C(C2CCCC(O)C2)=O)C1CNC(=O)CC(O)C1CCCC1 17132,C1(CNC(CS(CC)=O)=O)CCC2(CN(C(=O)Cc3ncc(C)o3)C2)O1 17133,C1(c2c[nH]nn2)CCc2cc(N)ccc2O1.CCC1Cc2ccccc2NC1=O.OC 17134,Cc1sc(C(=O)NC2CC(CNC(C3CC4CCC4C3)=O)C2)cc1[N+](=O)[O-] 17135,C1(NC(CC(C)(C)N(C(CCCC=C)=O)C)=O)CCOC12CCOC2 17136,c1(C(N2C(CC(N3CC(CC)C(F)C3)=O)CCC2)=O)cc(O)nc(C)n1 17137,C1(C(=O)OC)COCC2(CCN(C3CN(S(C)(=O)=O)CCC34CCC4)C2)O1 17138,c1(C(=O)NC(C)(C)CCNC(c2cc(C3CC3)ccn2)=O)cc(Cl)cnc1O 17139,c1(OC)cccc(Cl)c1C(N1CC(NC(C2CC23CCC3)=O)CC(F)C1)=O 17140,c1(OC)nc(N2CCC(F)(C(=O)Nc3cccc(-c4nnco4)c3)C2)ncc1Br 17141,C1(OC)CN(C(=O)NCc2ccc(C)c(OC)c2)CCC1NC(=O)OC(C)(C)C 17142,CCC(C(=O)NCC1(O)CCCN(C(C2CC(F)(CO)C2)=O)C1)C(C)(F)F 17143,CC1CC(NC(c2cc(-c3ccco3)nn2C)=O)CN1C(c1cnc(O)s1)=O 17144,CC(C)(C)C(CNC(=O)CC(=O)C(C)(C)C)C(=O)NCC(C)(O)CO 17145,C1(NC(=O)Cn2cc(Cl)cn2)CN(C(C2CC(CF)C2)=O)CC2(CC2)C1 17146,CC(C)CC(CNC(c1ccn(C(F)F)n1)=O)C(=O)N(CCC(=O)NC1CC1)C 17147,C(c1c(C)noc1C)=CC(N1C(C(C)NC(C=C(C)c2cccs2)=O)CCC1)=O 17148,c1(OCC)cc(N2CCC(N(C)C(C3CCCC4CC34)=O)CC2)ccc1[N+](=O)[O-] 17149,CCCCCC(O)CC(=O)N1CCN(C)C(C(=O)NCc2nnc(C)n2C)C1 17150,CC(C)CC(C(=O)N(CC(C)CNC(=O)CCC1CC1)C)N(C)C 17151,c1(C(N2CC(NC(C(C)=C(C)C)=O)C3(C2)CC3)=O)nc2cccnn2c1Br 17152,N1(C2CN(CCNCC)C2)CCN(C(=O)C(COC)COC)CC1 17153,c1(C(=O)NCC2CCCC(NC(C(CSC)C)=O)C2)c(C)ccc(N)c1C 17154,C1(CNC(CCOC(C)C)=O)CN(C(c2cc(OC(F)F)ccn2)=O)CC1(C)C 17155,C1(NC(c2ccc(Cl)s2)=O)CN(C(C2CC(C3CC3)=NO2)=O)C2CCCC12 17156,C1(F)(CNC(=O)COC2CCCC2)CC(NC(c2occc2C2CC2)=O)C1 17157,C(=O)(CC(CC)CC)NC(CSCC)C(=O)NC(CO)C1CC1 17158,CCC(CC)CC(F)C(=O)NC1(C(N2CCCN(C)CC2)=O)CC1 17159,c1(C(N2C(C(N(C)CCC3CCCC3)=O)C=CC2)=O)ccncc1F 17160,C1(NC(c2cn(CC(C)(C)CNC(C3CCSCC3)=O)nn2)=O)CC(F)C(=O)N1 17161,N1(CCCCNC(=O)NC(c2sccc2C)CC)CCC(NC(C)=O)CC1 17162,c1(OCC(N2C(C)CSCC2)=O)c(Cl)cc(Cl)cc1Cl 17163,C#CCCCCCCC(=O)NCc1ccc(C(=O)NC2(C3CC3)CCOC2)n1C 17164,N1(C(C(C)OC2CCCC2)=O)CC2CCCC(NC(=O)C=C(Cl)Cl)(C2)C1 17165,c1(C(=O)NCC(CC=C)NC(=O)CCC(N)=O)cccc2occc12 17166,c1(C(=O)NC(C)(C)CNC(=O)CC2CCOCC2)coc(S(N)(=O)=O)c1 17167,C(C(C)(C)CCNC(c1ccnc(O)c1)=O)NC(c1cn(CC=C)nc1)=O 17168,C(=O)(C(F)(F)C1=CCOCC1)NC1CC(NC(Cc2n(C)ncc2Cl)=O)C1 17169,C(c1cn(CC(=O)Nc2ccccc2)cn1)=CC(=O)OC(C)C(=O)N(C)C 17170,S(=O)(=O)(c1cccnc1N1CC2(CC(C)CO2)C1)NCC(c1ccsc1)N(C)C 17171,C1(C(N2C(C)CN(C(=O)CC#N)C(C)C2)=O)=CC=CC=CC=C2N(C=C1)C2=O 17172,N1(C(C(CC)SC)=O)CC2CCCC(CNC(C3(C4CCCCC4)CC3)=O)C2C1 17173,CN1CCN(C(c2cc(CF)on2)=O)C(CNC(c2cnn(CC(F)F)c2)=O)C1 17174,c1(NC(C2C3CN(C(CCCN(C)C)=O)CC32)=O)ccc2ncnn2c1 17175,c1(C(=O)NCC(C)(O)CNC(=O)CSC(F)F)ccccc1O 17176,c1(C(C(=O)NC(C)C)N(C)Cc2nc(CO)n[nH]2)cc(C#N)cs1 17177,N1(c2cc(C)nc(CO)n2)CCC(C2CC2)C1CNC(=O)CCc1nccn1C 17178,c1(OC)ccccc1C(O)C(=O)NC1CCC1CNC(c1ccc(Cl)cn1)=O 17179,C12(C(=O)NCC(C)(CO)NC(c3cc(OC)cc(Cl)c3)=O)CC=CCN1CCC2 17180,c1(C(N(C(CNC(CC2ON=C(C)C2)=O)C)C)=O)cc2ccoc2cc1F 17181,N1(C(C2(COC)CCCO2)=O)CCCC(NC(=O)CCNC(=O)OC)C1 17182,N1(C(N)=O)CC2=C(C1)CN(C(=O)C1=CCCCO1)C2.c1(N(CC=O)C)cnn(C)c1 17183,C(C)(C)(CC(=O)NCc1ncccc1C(N1CCCC1)=O)OC 17184,c1(C(=O)NC(C(C)NC(=O)C=CS(C)=O)C)cccc2nc(C(F)F)[nH]c12 17185,n1(C(C)C)cnc(C(=O)NCCC2CCCN2C(c2csc(C(F)F)n2)=O)n1 17186,C(=O)(CCCC(=O)NC1CCCCC1CNC(C12COC(C1)C(O)C2)=O)OCC 17187,C1(NC(c2c(OC)scc2)=O)CCN(C(=O)CCn2cc(Cl)cn2)CC1F 17188,S(=O)(=O)(c1cccc(F)c1)N1C(C(N(C)Cc2ccccc2F)=O)CSCC1 17189,N1(C(CCCN(C)C)=O)CCCC(NC(c2ccnc(OC3CCOC3)c2)=O)C1 17190,n1(CCOC)ncc(C(=O)NCC(C)CNC(C2C3CCN2CC3)=O)c1C 17191,C1(COC)CN(C(=O)CC2(C)CC(F)(F)C2)CCN1C(C1CC(C)(C)CO1)=O 17192,S(=O)(=O)(c1ccc(F)c(F)c1)N1C2CCN(C(c3cc(Cl)ccn3)=O)C2CC1 17193,N1(C(=O)Cc2cnn(C(F)F)c2)CCC2C(CCCN2C(C2COCCO2)=O)C1 17194,c1(CNC(C2C(NC(CC(C=C)C)=O)C2(C)C)=O)cnc(F)c(C)c1 17195,c1(NC(C)=O)cccc(C(=O)NC2CCCN(C(=O)C(C)(C)C3CC3)C2)c1C 17196,C1(C(N2CCC(COCC)C2)=O)CCC(CNC(c2ncn(C)c2C)=O)CC1 17197,c1(SC)ccccc1CC(C1CC(CO)C1)N(C)C.C(C)(CO)(c1nn[nH]n1)N 17198,Cn1nc(O)cc1C(N1CC(O)CC1CNC(c1ccoc1C(F)(F)F)=O)=O 17199,C(N=c1cc(NCCOc2cccc(Cl)c2)nc(C)[nH]1)c1ccc(OCC)cc1 17200,c1(CC(=O)NC(C2(O)CN(C(Cn3nc(C)oc3=O)=O)C2)C)c(Cl)cccc1Cl 17201,CC(C)CC(O)C(C)C(=O)N1C(C(=O)N(C)CC2(C)CCCO2)CC2CC12 17202,N1(C(CC2CCCC(C#N)C2)=O)CCC=C(C(=O)Nc2cnn3cccc3c2)C1 17203,Cc1c(Cl)c(C(N2CCOCC(NC(=O)CCCC(F)F)C2)=O)nn1C 17204,C(C)(C)(CC(F)C(=O)N1CC2CC2C2CC12)NC(C1C(C(=O)OC)C1)=O 17205,CCCC(C)(C)CC(=O)NC1COC2(C1)CN(C(c1n[nH]c(C(C)(C)C)n1)=O)C2 17206,N1(C(c2nc(C)c(C)[nH]2)=O)CCC(C2CCNC2)C1 17207,C1(C(N(C(C)CNC(=O)C2=CCCCC2)C)=O)CCCC2(CCC2)C1 17208,N1(C(CCCOCC=C)=O)CC=CC(C(=O)NC(c2scnc2C)C)C1 17209,CC1CC(NC(=O)C(c2ccccn2)O)CN1C(c1cc(C(N)=O)cs1)=O 17210,c1(C2(O)CN(C(c3cc(C(=O)OC)on3)=O)C2)ccc(-c2nn[nH]n2)cc1 17211,C1(CCC)CN(C(=O)CCS(=O)(=O)NC)CCN1C(c1ccc(O)cc1)=O 17212,c1(N2CCCC(CCC(C)C)C2)nc(NCc2cc(Cl)n(C)n2)c2ncsc2n1 17213,Cc1ncccc1CC(=O)NC(C(=O)NC1CC1c1cncs1)c1ccco1 17214,N1(C(c2cnc(C)nc2)=O)CC2CCN(C(C3CCC(N(C)C)CC3)=O)CC2C1 17215,C(C(=O)NCC(C)(C)CCNC(c1ccc(C(C)(F)F)cc1)=O)(C(C)C)OC 17216,c1(OC)ccc(S(C)(=O)=O)cc1C(N1CCC(NCc2nc(Br)cs2)C1)=O 17217,CC(C(=O)N(CC(=O)N(CCCc1cn[nH]c1)C1CC1)CC1CC1)NC=O 17218,CCCC(C)(CC)C(=O)NC1CCN(C(c2cnc[nH]2)=O)CC1(C)C 17219,c1(C(N2CC3C(C(=O)OC(C)(C)C)C3C2)C(=O)NC)ccc(C#N)cn1 17220,c1(C(C)C(=O)NCC2CC(F)(CNC(C3CC3F)=O)C2)ccc(F)cc1F 17221,CC(C)(O)C(C(=O)NCc1ccsc1)NC(=O)COCCCF 17222,N#Cc1cccc(-c2cscc2C2CC2)c1 17223,c1(C(=O)NCC(C#C)C(C)C)ccc2c(c1)C(=O)N(C)C2=O 17224,N1(CCOCC=C)CCN(C2CCN(C(C3CC34CC4)=O)C2)CC1 17225,N1(C(=O)COCCF)CC2CCN(C(c3cnc4c(c3)COC4)=O)C2C1 17226,c1(CC)ccc(F)c(C(N2CCC(NC(c3ccnc(Cl)c3N)=O)C(C)C2)=O)c1 17227,C1(COC)(NC(=O)C(O)C(C)C)CCN(C(=O)COC2CCOCC2)C1 17228,C(C)(C(C(=O)NCCCC1CC(C)C1)C(C)C)NC(C(C)=C(CC)C)=O 17229,C(=O)(C(F)(CNC(=O)C=C=C(C)C)C(C)C)NCC(COCC)O 17230,c1(C(N2CCC(O)C2C)C(=O)NCC=C)ccc(C)c2c1CCC2 17231,N=c1cc(C(N2CCN(CCC(N3CCNCC3)=O)CC2)=O)cc[nH]1 17232,Nc1cc(C(N2CCC2CNC(C2(CC3CC3)CCCO2)=O)=O)cc(O)c1 17233,C1(C)(CNC(C(CC)COC)=O)CCC(NC(c2csc(C3CC3)n2)=O)CC1 17234,c1(C(=O)NCC(CCCC)NC(c2cccs2)=O)n[nH]c2c1COCC2 17235,C(=O)(CCS(C)(=O)=O)N1CC(OCC)C(CNC(c2cc(N)ccn2)=O)C1 17236,c1(CC)nc(N2CC(NC(c3cc(=O)c(OC)c[nH]3)=O)C(C)(C)C2)cc(C#N)n1 17237,c1(C(=O)OCC(CC)F)cnc2sc(C)nc2c1 17238,C=CCCCC(C(=O)NCC(C)Cc1ccc(OC)cc1)N(C1CC(F)(F)C1)C 17239,N1(C(C2C(NC(c3ccncc3Cl)=O)CCC2)=O)CCc2c(cccc2[N+](=O)[O-])C1 17240,c1(CC)[nH]nc(-c2nc(CCOC)nn2C2CCC(C)C2)c1Br 17241,C(CC(F)F)(C(=O)N1CC(C)(O)C1)NC(c1scc(C(C)=O)c1)=O 17242,C1(c2ncc(C(=O)OCC)s2)CCCN(C(c2nc(Cl)c(CC)[nH]2)=O)C1 17243,C#Cc1ccnc(C(N2CCC(N(C)C(c3cccc(N)c3F)=O)C2)=O)c1 17244,N1(C(C2(NC(=O)CC3CCCSC3)CCSC2)=O)CCc2cncnc2C1 17245,C(=O)(C(C)CCCC(C)C)N1C(C(=O)NC(CCC)C2CC2)(COC)C=CC1 17246,CN1CC(=O)N(CC(=O)NC2CC(CO)N(C(c3nccc(Cl)c3F)=O)C2)C1=O 17247,C(=O)(CC(CC(N)=O)CC(C)C)NC(CN(C(c1c(C)nco1)=O)C)(C)C 17248,C(=O)(CCCCCC(C)C)NC(CCCCNC(C(C)=CC)=O)C 17249,N1(C(C(=C(C)C2CC2)F)=O)CC(CNC(=O)CN2CCS(=O)CC2)C(C)(C)C1 17250,C(=O)(C1=C(c2ccccc2)SCCO1)NC1CN(C(CC(C)(C)C#N)=O)C2C1C2 17251,c1(C(N2CC(NC(COCC(=C)C)=O)C(N=[N+]=[N-])C2)=O)cn2cccc(C)c2n1 17252,CC1CC(C(=O)N2CCN(C(=O)CNC(c3cccnc3)=O)CC2CCO)=NO1 17253,c1(C(C)C)ccc(F)c(C(=O)NCC2C(F)(F)C23CC3)c1 17254,N(C(=NCC(C(C)C)C(C)C)NCc1cc(C)on1)C(CC)CC 17255,C1(O)(COC)CCN(C(c2cn(-c3ccc(C)cc3)nn2)=O)CC1 17256,Cc1ccc(C)c(C(=O)NCC2CC(NC(=O)C=Cc3cccs3)C23CCC3)n1 17257,c1(OC)ccc(SCCC(=O)NC2CCC(CN(C(=O)CCC(C)=O)CC)C2)cc1 17258,C(=O)(C(C(C)C1CCOCC1)N1CCC(C)(O)C1)NCCC(C)C.C(CC)S 17259,Cc1nc(C2CC2)nc(C)c1C(=O)NCC1(C)CCN(C(=O)CC2(CO)CC2)C1 17260,CCCCCC(C)(CC)C(=O)NC1CCC(NC(=O)CCc2ccn(C)c2)CC1 17261,C12(C(N(CCCCNC(C3CC(=O)CS3)=O)C)=O)CC3CC(CC1C3)C2 17262,C(C)(C)(CC(F)C(=O)Nc1ccc(Cl)c(O)c1)NC(c1cc(C)nnc1)=O 17263,Cn1c(O)nc2ccc(C(=O)NCCC3CCC(NC(=O)CNC=O)C3)cc12 17264,C=Cc1cnn(C)c1C(=O)NCC(CCCC)NC(c1scnc1CC)=O 17265,c1(CC)cnn2ccc(C(=O)NC(C)CCCNC(=O)CN(C)CC)nc12 17266,C1(NC(c2coc(C(=O)NC(C3CCCCC3)CO)c2)=O)(CO)CC(CO)C1 17267,C1(NC(CCCCC)=O)C(CNC(=O)C(C2CC2)C2CC2)CCC12CCC2 17268,C(CCN(C)C(C1CC2(C1)CC(F)C2)=O)(C(C)(C)C)NC(CC(=O)OCC)=O 17269,c1(CC(C(=O)NC)NC(c2cc(F)c(C)cc2N)=O)c[nH]c2ccccc12 17270,CC1=C(Br)CCN(C(C2CCC(c3nc(C)no3)CC2)=O)C1 17271,CC(C)(CCC(=O)N1CC2(CSC2)C1)NC(c1cc[nH]c(=N)n1)=O 17272,C1(=CC(=O)NCC(C2CCC2)NC(=O)Cc2cnc[nH]2)CN2CCC1CC2 17273,Cc1sc(=O)n(CCC(N2CC(N(C(=O)CCCCCF)C)C(F)C2)=O)c1C 17274,c1(C(N(CC)Cc2ncccn2)=O)ccc(CNC(c2oc(C)cc2C)=O)nc1 17275,N1(C(C2CC(C)S(=O)(=O)CC2)=O)CCC(NC(C2(F)CCCC2)=O)C12CCCC2 17276,c1(C(=O)NCC(CNC(C(C)OC)=O)O)nc2ccccc2n1-c1ccccn1 17277,CCC(CC)CC(F)C(=O)N1CCCC1C(C)(C)CNC(c1n[nH]cc1C)=O 17278,CC(C)C(C(=O)NC(C1CCCC1)CNC(=O)C(c1ccccc1)F)NC(N)=O 17279,c1(N2CCC(c3onc(C)n3)C2)nc(C2CCOC2)nn1C(C1CCOCC1)C 17280,CCC(C)C(C(=O)NCC1(CNC(=O)C(C2CC(F)(F)C2)O)CC12CCC2)OC 17281,N1(C(CC2CC(C)(C)OC2)=O)CC2CCC(C1)N2C(c1cncc(O)c1Cl)=O 17282,C1(CNC(C(CC)(C)CO)=O)N(C(c2nc(C)ccc2F)=O)CCCC1(C)C 17283,CC(F)(F)C(C)(C)CC(=O)N1CCCCCC(S(C)(=O)=O)C1.c12cncc(c1)N2 17284,C=C1CC(C)(NC(C2CCN2C(C2(OCC)CCSC2)=O)=O)C1 17285,C1(C)(C(=O)NCc2cccc(NC(CCCCCOC)=O)c2)CC(C)OC(C)C1 17286,CC(C)C(O)C(=O)N1CC=CC1(C)C(=O)N(C)CCC1CN(C)C1 17287,C(=O)(C(C#N)C(C)(C)C)N1CC(OCCC(=O)NCc2ccc(C)cc2F)C1 17288,C12(CCNC(C(CC)(F)F)=O)CCC1CN(C(c1cncc(C)n1)=O)C2 17289,C1(C2CC2)(CNC(=O)CCc2cnoc2)CCN(C(c2cccnn2)=O)C1 17290,CC(C)(C)CCCC(=O)N1CCCC(CNC(C2COC(=O)C2)=O)C1 17291,CCC(CNC(=O)C(c1ccccc1)Sc1ccccc1)(CCOC)C(=O)O 17292,c1(CNC(c2c(CNC(CCCOCC=C)=O)noc2)=O)cccnc1F 17293,C(=O)(C(CCOCC)NC(C1CC2(CC2)C1)=O)N(CCCN(C)C)CCC 17294,C1(CNC(=O)CC2(O)CCOCC2)CCC2(CN(C(=O)C(O)C3CC3)C2)O1 17295,C1(CNC(CC2CC(OC)C2)=O)CCC(NC(c2cccc(C(F)F)c2)=O)CC1 17296,N1(C(c2cn(CC)nc2)=O)CCCC2C(CCCN2C(c2n[nH]c(C)c2Cl)=O)C1 17297,c1(C(N(CCNC(=O)C(c2sccc2C)=O)CC)=O)ccc(F)c(F)c1F 17298,C(=O)(C1=NN(C)C(=O)CC1)NCC(CCOC)NC(c1c(C)cccc1Cl)=O 17299,c1(N(CC(CN(C)C(C2(F)CCCCC2)=O)O)C)nc2c(cc1C#N)CCOC2 17300,Cc1cc(C(N2CC(NC(C3C(C)(C)C3(C)C)=O)CCC2C)=O)cc(Br)c1C 17301,n1(C(C)C)ncc(C(=O)NC(CNC(=O)Cn2cccn2)C(C)C)c1F 17302,C1(C(=O)NCC2(C3CC3)CCC2)(OC)CCN(C(=O)Cc2ccoc2C)C1 17303,C(=O)(C1=CC2CCC(C1)C2)N1CC2C(CN(c3ccccc3)C(C)C)(CC2)C1 17304,N1(C(C2CC(OC)CN2C(=O)CC2CCN(C)CC2)=O)CCC2(CNC(=O)O2)C1 17305,c1(C(=O)NCC(=C)CCNC(=O)CC2CCCN2C(C)C)cnc(OC)cc1C 17306,C1(OC(C)=O)CCC=CCCC1.C12N(CC1(C)C)C(=O)c1cn(nn1)CCNC2=O 17307,c1(CC(N2CCC(N(C(=O)C=CCO)CCC)C2)=O)cnccc1Cl 17308,c1(CC2(O)CC(NC(=O)NC(C)Cn3cncn3)C2)cc(OC(F)F)n(C)n1 17309,c1(C(CC(=O)OCC)NC(C2(C(C)N)CCC2)=O)ccc(C2CC2)cc1 17310,N1(C(C(C)Cc2cccnc2)=O)CCCN(C(C2(NC(N)=O)CCC2)=O)CC1 17311,C=Cc1cncc(C(N2CCC3CC23C(=O)NCCc2cc(C)no2)=O)c1 17312,C1(CNC(COCC)=O)CCN(c2ccnc(NC3CCCCC3C)n2)CC1 17313,C(=O)(CC(C)(C)COC)NC1(CC=C)CCN(C(c2cc(Br)nn2C)=O)C1 17314,c1(C(N2CCCC(N(C(=O)CCN3CCOCC3)C)C2)=O)ccc2c(n1)COCC2 17315,C1(C(=O)OC)CC2CCN1C(=O)C(C)C(=O)N2.c1(CC)cccc(C)c1 17316,C1(NC(C2(CC)CCCCO2)=O)CCN(C(c2cnc(CC3CC3)s2)=O)C(C)C1 17317,c1(C(N)=O)cc2c(cc1NCC1CC3(C1)CC3F)CCC2 17318,C1(NC(C(CSC)(C)C)=O)CN(C(c2cc(Cl)c(Br)[nH]2)=O)CCC1C 17319,C1(CC(=O)NC(C=C)(C)CC)CCN(C(C)=O)C1(C)C 17320,N1(C(CCOCCOCC)=O)CCC(C(C)CNC(C2(C)CC=CCO2)=O)CC1 17321,C1(Nc2ccc(C(C)C)nc2)CP(C)(=O)CC1O 17322,N1(C(CCC)=O)CC(NC(c2ccc(Br)c(C)c2F)=O)C2(CCC2)C1 17323,c1(C(=O)NCc2c(C(=O)NCCc3ocnc3CO)c[nH]n2)c(Cl)cccc1Cl 17324,N1(C(Cn2nc(C)oc2=O)=O)CCC(NC(C2(CO)CCCO2)=O)C(O)C1 17325,c1(N(C)CC2CCN(C(c3cc(Br)co3)=O)C2)ccc([N+](=O)[O-])cn1 17326,CC(C)(C)CC(C)(C)C(=O)NCC(F)CNC(c1nccnc1N)=O 17327,c1(C(=O)NC(CNC(c2nc(C)[nH]n2)=O)C)coc(=O)c2ccccc12 17328,c1(C(=O)NCC2CCC(NC(C3CC(N4CC(O)C4)C3)=O)C2)sc(F)cc1Cl 17329,c1(COC)cc(C(N2CCC(CNC(c3cc(C(N)=O)cs3)=O)CC2)=O)c(C)o1 17330,c1(OC)cc(Br)ccc1C(=O)CN(C1CCCCC1NC(=O)OC(C)(C)C)C 17331,C1(NC(c2n(CC(=C)C)nnn2)c2ccno2)CC2CCC(C1)O2 17332,n1(CC=C)cc(C(=O)NC2(C)CC(C(N3CCC3(C)C(=O)NC)=O)C2)cn1 17333,N1(C(c2cccc(-c3cn[nH]c3)c2)C(=O)NCC=C)CCC(C)C(C)(C)C1 17334,c1(C(N2CC(N(C(=O)C3=NOCC3)C)C(F)C2)=O)ccc(O)nc1Cl 17335,C1(CNC(=O)C(C2CCCCC2)O)CN(C(c2cc(C3CC3)[nH]n2)=O)CCCO1 17336,C1(NC(c2nc(CC)oc2)=O)(COC)CCN(C(c2ccc(CC3CC3)s2)=O)C1 17337,CCCCCCCC(=O)N1CC(NC(c2cc(F)ccc2C)=O)C(O)C1 17338,c1(CC)cccnc1C(=O)NC(CC)C(=O)N(C1CCCOC1)CC 17339,c1(NC(=O)NC(CCCNC(C(=O)OC(C)(C)C)=O)(C)C)cnn2c1CCC2 17340,Cc1sc(Cl)c(C(=O)NCCOCCCNC(=O)CCC2CCN(C)CC2)c1C 17341,CC#CCCCC(=O)N1CCCC1CCCNC(=O)COc1cccc(C)c1 17342,N1(C(C(COCC)C)=O)CCC2C1CCCN2C(c1cccc2ccnn12)=O 17343,C1(C(=O)NCC2CN(C(=O)Cc3ccsc3Cl)C2)COCCC1(F)F 17344,CC(C)CS(=O)(=O)CCC(=O)NCC1CCC(C)CN1C(c1cc(Cl)cn1C)=O 17345,C1(C(N(C)Cc2c(C)cco2)=O)CC(NC(=O)Cc2cncn2C)C1(C)C 17346,N1(C(C23CC(=O)C2CCC3)=O)CCc2ccc(Cl)nc21 17347,c1(OC)ccc(C(=O)N(C2CN(C(=O)CN3CC4CC4C3)CC2O)C)cc1OC 17348,CC1CCCC(N(C(c2csc(C3CC3)n2)C(=O)NCC2CCCO2)C)CC1 17349,N1(Cc2c(C(=O)OCC)ccs2)CCN(C(=O)C(O)CC(C)C)C2CC12 17350,C1(NC(CCn2ncn(C)c2=O)=O)CC(NC(C2(S(C)(=O)=O)CC2)=O)C12CCC2 17351,N1(C(CCC2CCN(C(c3ccc(=N)[nH]c3)=O)CC2)=O)CCC2=C(CCCC2)C1 17352,C#CCCCCC(=O)NC1CC1C(=O)NN1CCN(c2cccc(C#N)c2)CC1 17353,c1(C(N2CCN(C3CN(C(C4ON=C(C)C4)=O)C3)CC2)=O)ccc(O)nc1C 17354,C1(C(=O)NC(C(C)NC(c2cc3occc3s2)=O)(C)C)CCc2nncn2C1 17355,c1(C(N(CCNC(c2c(CC)nc[nH]2)=O)CCOCCO)=O)cc(O)ccc1N 17356,C=CCC(C)(C)CC(=O)NC1CN(C(c2cnc(CC)s2)=O)CCC1CO 17357,c1(C(N2CCC(NC(c3ccc(Cl)s3)=O)C(O)C2)=O)c(F)cc(F)cc1Cl 17358,N(C1CCc2c(Br)cccc21)CCCn1c(C(C(CC)CC)N)nnn1.OC 17359,CCCC(CCC)C(=O)NCCC(C)NC(C1CCS1(=O)=O)=O 17360,C1(C(N2CCC(OCCNC(c3ccc(SC)cc3)=O)C2)=O)CCCCN1N=O 17361,c1(C(N(CC(=O)C2(N(C3CC3)C3CC3)CC2)CCOC)=O)cc(C(N)=O)co1.OC 17362,C=C(C)CCCNC(=O)COC(C)(C)CNC(C1(CCCC)CC1)=O 17363,O=C(C1=C(F)CN(C(C2(F)CCOC2)=O)CC1)NCc1nn[nH]n1 17364,C1(NC(C(CC)=CC)=O)CCC2CCN(C(=O)CCc3nc(C)no3)C1C2 17365,N1(C(CNC=O)=O)CCOCC1CNC(=O)COC1CCOC1 17366,O=C1COc2ccc(C(=O)NC34CC3CN(C(c3cnc(Cl)s3)=O)C4)cc2N1 17367,c1(C(=O)NCC(C)(C)NC(=O)Cc2ccc3c(c2)CCC3)cc(Cl)c([N+](=O)[O-])[nH]1 17368,N1(C(CCS(C)=O)=O)CCC(NC(=O)Cc2ccc(F)c(Cl)c2)C12CC2 17369,c1(C(N(CC(CNC(Cc2scc(C)n2)=O)C)C)=O)cccc(C2CC2)n1 17370,CCCC(O)(CCC)CC(=O)N1CCCC(C2(NC(C3(N(C)C)CC3)=O)CC2)C1 17371,C(c1cnn(C)c1C)=CC(N1CC=CC(NC(c2ccc(NC)cc2)=O)C1)=O 17372,c1(C(=O)NCC2C(CNC(c3ccc(SC)s3)=O)C2)cnnc2ccccc12 17373,c1(CC(N2CC(n3cc(CNC(c4cnn(C)n4)=O)nn3)C2)=O)cccc(F)c1 17374,C(=O)(C1CCCc2nncn21)N(CCN(C(=O)C=Cc1ccco1)C)C 17375,S(=O)(=O)(c1ccc(C(N2CCC(C)(CNC(c3ccoc3)=O)C2)=O)cc1)NCC 17376,c1(C(=O)NCC(CC=C)NC(c2nn(C)nc2Br)=O)cnc(C)n1C 17377,N1(C(c2cc(CCC)on2)=O)CCCC(CC(=O)NC2CC3CCC2O3)C1 17378,Cc1oc(S(C)(=O)=O)cc1C(=O)NCCOC1CCN(C(C2(C)CCC2)=O)CC1 17379,c1(C(N2CC3C(C(=O)NCc4c(C)noc4C)C3C2)=O)cc(O)nc(Cl)c1 17380,C1(NC(C(C)(C)OC)=O)C2CN(C(C3CCCC3C(C)C)=O)CC12 17381,C1(C)(NC(c2ncn(C(C)C)n2)=O)CCN(C(c2cc3n(n2)CCO3)=O)CC1 17382,c1(C(=O)NC2C=CCN(C(CCN(C)CC)=O)C2)c(C)[nH]c2ccc(F)cc12 17383,N1(C(c2scc(C)c2Br)=O)CCCN(C(=O)C(C)CF)CC1 17384,S(=O)(=O)(c1csc(C(N2CC(CNC(=O)C(C)(C)F)C3CC23)=O)c1)NC 17385,c1(C(N(CC(C)NC(c2c(C(C)C)con2)=O)C)=O)cn(C)nc1C(F)F 17386,c1(C(N2CC3C(CNC(c4n(CC)cnn4)=O)(C3)C2)=O)ccc2c(n1)CCCC2 17387,CC(O)CC(=O)NC(Cc1cc[nH]n1)C(=O)N1CC(O)(c2cc[nH]n2)C1 17388,CN1C(=O)Cc2ccc(-c3cccc(CN4CCC(CC#N)CC4)c3)cc21 17389,N#Cc1cc(N2CCC(NC(=O)CSc3n[nH]c(O)n3)C2)nc(C2CC2)n1 17390,C1(NC(c2c(CC)occ2C)=O)CN(C(c2ocnc2C2CC2)=O)CCC1F 17391,CC1CCCN(C(c2cnsc2)=O)C1CNC(C1OCCN(C)C1=O)=O 17392,C1(C(N(CC(C2CC2)OC)C)=O)CN(C(c2cn(C)cc2C)=O)CC1(F)F 17393,c1(N(CCNC(CC2C(OC)COCC2)=O)C2CC2)ncn(C)c(=O)c1Br 17394,c1(C(=O)NCC2CC(NC(CCCCN(C)C)=O)C(O)C2)ccc(O)c(F)c1F 17395,C=CCCCCC(=O)N1CC(C)C(C)(C(=O)NC2CCC(N(C)C)C2)C1 17396,c1(C(=O)NC(CC)(C)CNC(c2sncc2C)=O)cc(Cl)ccc1Cl 17397,CC1(C)CC(NC(C2CC2c2ccc(Cl)cc2)=O)CN1C(c1ccc(F)cn1)=O 17398,C(CCCC(=O)NC(C)(C)C(=O)N1CCC1C(C)C)OC 17399,C1(NC(Cc2cc(CC)no2)=O)CC2CCC1C1CN(C(C3CC=CC3)=O)CC21 17400,C1(C(=O)NCC(C2CC2)NC(c2c(C)cc(C)nc2)=O)CCc2nnc(O)n2C1 17401,c1(C(N2CCN(C(C3CC3c3ccccc3)=O)C3C2C3)=O)cn2ncccc2n1 17402,N(C1CC(F)(F)c2ccccc21)C(=O)C(N1CCc2ccc(F)cc21)=O 17403,Cc1nc2cc(C(=O)NCC3(F)CCN(C(c4cnc[nH]c4=N)=O)C3)[nH]c2s1 17404,C(C1CCOC1)=CC(=O)NCC1C=CC(NC(=O)Cn2nccn2)C1 17405,C1(CC(N2CCC(COC)(NC(=O)C3=CCCS3)CC2)=O)CC(C)CC(C)(C)C1 17406,c1(CNC(C(C)N(C)C(C2CCC2C#N)=O)=O)cc(C2CC2)no1 17407,c1(C(=O)NC2CC(C(N(CCCC(C)O)C)=O)C23CCC3)cccc2[nH]ncc12 17408,Cc1cccc(CNC(C2CCCN2C(=O)C=CC2CCOCC2)=O)c1 17409,CCC(CC)C(C)C(=O)N1CCN(C(=O)CC(F)(F)CC)C(c2ccccc2)C1 17410,c1(C(=O)NCC(C)CNC(=O)CCN(C)CCO)ncnc(O)c1Cl 17411,CC1CCC(CCC(=O)N(C(Cc2ccco2)CO)CCN)O1 17412,c1(CN2CCCC(CN(C)C(c3cccnc3S)=O)C2)cccc2ncccc12 17413,C(=O)(CCCC(C)(C)C(=O)OCC)NC(C(C)NC(CSCCC)=O)C(C)C 17414,Cc1ccc(CNC(C2C3CC3CN2C(=O)CCC2CC2C)=O)nn1 17415,N1(C(C(C=C)CC)=O)CC2(C1)CN(C(=O)CCn1ccc(C)n1)CC2CO 17416,c1(C(=O)NC2CCCC(NC(c3c(N)cncc3)=O)CC2)nnn2c1CCCC2 17417,c1(C(N2CC(NC(CS(=O)(=O)NC)=O)C(F)CC2)=O)ccc2c(c1)OCCCO2 17418,N1(c2ncc(C#C)cn2)CCN(C(c2cc(F)c(Cl)cc2F)=O)C(C#N)C1 17419,Cc1cc(C(N2CCC(NC(=O)Cc3sc(C)cc3C)C2)=O)c([N+](=O)[O-])c(O)n1 17420,C1(NC(C2(CCCC)CC2)=O)CC2(C(=O)NCC3CC(=O)N(C)C3)COC1C2 17421,c1(C(N(C2CN(C(=O)CN3CCNC(=O)C3)CC2O)C)=O)cc2occc2n1C 17422,C(C(=O)N(CCCCN(C(=O)C(O)C(F)F)C)C)(C(C)C)NC(CC(C)C)=O 17423,N1(C(CCC=C(C)C)=O)CC2CCN(C(c3scc(C)c3Cl)=O)C2C1 17424,Cn1cnc2c(C(N3CCOC(CNC(=O)CC4(C)CCCO4)C3)=O)ccnc12 17425,Cc1cc(C(N2CC(C)C(C)(CNC(=O)CN(C)C3CC3)C2)=O)nnc1C 17426,CCCCCC(CC)C(=O)NC1CCC1CNC(c1cnnc(C)c1)=O 17427,C(c1ccc(F)c(F)c1)=C(C)COC(=O)Cc1ccc(F)cc1C#N 17428,c1(CC)nn(C)cc1C(=O)NC(C)(C)C(C)NC(=O)CCc1cn(C)nc1C 17429,Cc1cc(C)c(S(=O)(=O)N2CCC(O)(C(=O)NCC(CO)C(C)C)CC2)c(C)c1 17430,O=C1Cc2ccc(CNC(C3CC3c3ccc(Cl)c(Cl)c3)=O)cc2N1 17431,N1(C(CC2(NC(c3cc(C(C)C)on3)=O)CC2)=O)CCCC(CNC(N)=O)C1 17432,C1(C)(C(=O)NCC(C2CCCN2C(c2sccc2Cl)=O)(C)C)CCCOC1 17433,C1(C(N(CC(NOCC#C)=O)C(C)C)=O)CC12CCCC2 17434,C(=O)(C(C)(C)CC(F)F)NC(C)CC(C)NC(C1CCN1C(C)(C)C)=O 17435,CCC(C(=O)N1CCC(CCNC(C2CCC(N(C)C)CC2)=O)C1)C(C)C 17436,Cc1sc(O)nc1C(N1CC(C(N)=O)(CNC(=O)Cn2cnnc2)C1)=O 17437,CC1OCC2(CCN(C(C3CC3C(=O)Nc3ncc(Br)cc3Cl)=O)CC2)C1N 17438,CC1C(C)CCN1C(c1c[nH]nc1CCNC(=O)CCC(=O)N(C)C)=O 17439,N1(C(C2(NC(c3cn(CC)nc3C)=O)CC2C)=O)CCN(C)C(CO)C1 17440,c1(NC(C2CCN2C2CC2)=O)ccccc1NCCc1cscn1 17441,C(CCNC(C1CCCN1C(N)=O)=O)(C(=O)NCC(O)(COC)CO)OC 17442,CC1CN(C(C2CS(=O)C2)=O)CCC1NC(=O)CC(C)(O)C1CC1 17443,CC(C)(C)CCCCC(=O)NC1CN(C(=O)Cc2ccno2)CC(C)(C)C1 17444,C(C)(CCC(=O)NCC1CCCC1C(=O)NC(C1(O)CCC1)(C)C)OC 17445,c1(C(=O)NCC2CC(NC(C(C3CCC3)OC)=O)C2)cc(Cl)c(F)cc1Cl 17446,C1(NC(c2sc(CC)c(C)c2)=O)CN(C(C2(CCOC)CCC2)=O)CC1(C)C 17447,CC1CC(C(=O)N(C(=O)CC(F)(F)F)CC=C)CN1c1nnnn1-c1ccccc1 17448,c1(CC)ccc(C(=O)NCC2CCCN(c3nccnc3F)CC2)cc1CC 17449,C1(C(=O)NCCC2N(C(CCC(=O)NC(N)=O)=O)CCSC2)CCCC(F)(F)CC1 17450,N1(C(C=CCC)=O)CCC(NC(c2cc(C(C)=O)c[nH]2)=O)CC1 17451,C12(C(N3CCC(NC(c4[nH]cc(C)c4)=O)C3)=O)CCCC(C)(C1)OC2 17452,c1(C(=O)NC(COCC#C)C)cncc(OC2CCC2)c1.C(=O)(CCO)CN 17453,C1(CNC(c2cc(C)ns2)=O)CC(F)(F)CN1C(c1ccc(N)c(Cl)n1)=O 17454,N1(C(c2n(CC)ccc2)=O)CC(NC(c2cc(-c3ccccc3)co2)=O)C(C)C1 17455,N1(C(c2ncn(CC)c2)=O)CCCC2CN(C(c3cc(O)ncn3)=O)CCC12 17456,N1(C(CSS(C)(=O)=O)=O)C2CCC1CC(NC(c1cc(Cl)no1)=O)C2 17457,c1(NC(CCC(C)NC(=O)CC2CC(N(C)C)C2)=O)cccn2ncnc12 17458,CC1(C)CCC=C1C(=O)NCC1CC(NC(C2CN(c3nncs3)C2)=O)C1 17459,CN=c1cc(C(=O)NCC(c2cn(C(C)C)nn2)(C)C)c(Br)c[nH]1 17460,C1(CNC(C(C)OCCN(C)C)=O)CN(C(=O)C(c2ccn(C)c2)C)CCN1C 17461,C(c1ccc([N+](=O)[O-])cc1)=CC(=O)NCCNC(c1cc(F)c(OC)c(F)c1)=O 17462,c1(CN2CCC(N(C(c3cccc(CC)n3)=O)C)C2)ccc2c(c1)OCCO2 17463,C1(CNC(C2(NC(=O)OC)CCCC2)=O)CCC(NC(C2CC2C(C)C)=O)CC1 17464,C=CCCC(O)CN(C)C(C1CC(F)CN1C(=O)C=C1CCCCC1)=O 17465,C1(NC(c2c(C)[nH]nc2C(F)F)=O)CC2CC1N(C(=O)COC1CC=CC1)C2 17466,c1(CC)ncc(Br)cc1C(N1CCC1CNC(C1(N2CCCC2)CCC1)=O)=O 17467,c1(C(N(CC(F)F)C)=O)c(NC(c2nccc3ccccc23)=O)sc2c1CCCC2 17468,c1(CC(=O)NC(CNC(CNC(C2C(C)C2)=O)=O)C2CC2)cccc([N+](=O)[O-])c1 17469,N1(C(C2C(OC)CCC2)=O)CCC(C)C1C(=O)N(C1CN(C)C1)C 17470,CC1(C(=O)NCCCNC(=O)Cc2ccc(Cl)cn2)CS(=O)(=O)C1 17471,Cc1ccc(CC(=O)NC(C)(C)CCNC(C2(C)CC2F)=O)o1 17472,C12(CN3CCN(CC(N4CCCC4)=O)C(C)C3)COCC(C3CC3)(C1)C2 17473,CC1CCC(c2cn(-c3cnn(C)c3)nn2)N(C(=O)Cc2cccc(F)c2)C1 17474,c1(C(N2CC(CC)N(C(c3cccc(=O)o3)=O)CC2)=O)ccc2c(c1)COCC2 17475,N1(C(Cc2cc(C)on2)=O)CCOC2CN(C(=O)C(C)(O)C(F)(F)F)CC12 17476,C12(NC(=O)CCC3CC3(F)F)CCCN(C(=O)COc3ccccc3O)CC1C2 17477,N1(C(C(CO)NC(N)=O)=O)CCCC(CNC(C2(S(N)(=O)=O)CC2)=O)CC1 17478,C1(NC(C(CCC)NC(N)=O)=O)CCN(C(=O)CS(=O)(=O)CC)CCC1CO 17479,C(=O)(C1=CSCCO1)N1CC(CNC(C2CN3CCC2CC3)=O)C2C1C2 17480,c1(CC(N2CCC(N(C(=O)C(F)C(C)C)CCC)C2)=O)cc(F)cc([N+](=O)[O-])c1 17481,c1(C(=O)NCCCCCNC(C2(C)CC2(Cl)Cl)=O)cc2c(nn1)CCC2 17482,Cc1cc(F)c(C(=O)NCC(C)(C2CCC2)NC(c2cscn2)C2CC2)c(Cl)c1 17483,CC1CCN(C(c2c[nH]c(=N)s2)=O)CCC1N(C1CS(=O)(=O)C1)C 17484,c1(OC)ccc(-c2noc(C3CCCC3N)n2)c(Cl)c1 17485,N1(C(C2C(=O)NCC2)=O)CCC2CC1CN(C(c1ccc3c[nH]nc3c1)=O)C2 17486,c1(C(=O)NC2CN(C(c3c(C)c[nH]n3)=O)CC2F)noc2cc(Cl)ccc12 17487,Cn1cc(SCCc2cn(CC3COC3)nn2)cn1 17488,N1(C(C(C(C)NC(CSCCOC)=O)(C)C)=O)CC2CCCC(O)C2C1 17489,CC1(CC(=O)NCC(C2CC2)NC(=O)C(F)=C2CCC2)CC1(F)Cl 17490,N1(C(CCc2nnc(C(C)C)o2)=O)CCN(C(=O)C=CCF)CC12CCC2 17491,c1(C(N2CC3C(C(=O)Nc4cncc(N(C)C)c4)C3C2)=O)ccnc([N+](=O)[O-])c1 17492,N1(C(C(C)C2CCOC2)=O)C(C(=O)NCCNC(=O)CO)CCC1C 17493,c1(OCC)cccc(C(=O)N(c2cc(N(C)CC3CCNCC3)ncn2)CC)c1 17494,CC1(CNC(C2(F)CC=CCC2)=O)COCCN(C(c2ccc(Cl)c(O)c2)=O)C1 17495,c1(CC(=O)NC(CSC)(C)C(=O)N2C3CCC2CC3)cccc(C#N)c1 17496,C#CCC(CC#C)C(=O)NCC(C)NC(=O)CCc1cccc(OCC)c1 17497,c1(C(N2CCN(CC(N3CCCC(C)(O)C3)=O)CC2)=O)ccc([N+](=O)[O-])cc1Br 17498,c1(NC(C(CSCC)C)=O)cccc(-c2nncn2C)c1 17499,C1(NC(c2c(SC)n(C)nc2)=O)CN(C(=O)CN2CCCCC2)CC(C)(C)C1 17500,N1(C(=O)C=Cc2cscn2)CCCN(C(=O)CC2CCC3(CCC3)O2)CCC1 17501,N1(C(c2cc(C(C)(F)F)on2)=O)CC2CCN(C(C3(c4cc[nH]n4)CC3)=O)C2C1 17502,C12(NC(c3cc(C(F)(F)F)ccn3)=O)CCC1CN(C(C1CCCCC1O)=O)C2 17503,c1(OC2CC(NC(=O)NC3C(NC(=O)OC(C)(C)C)CC3)C2)ccccc1Cl 17504,C(=O)(C#CC1CCOCC1)NCC(CCC)C(=O)NCC(CCC)OCC 17505,c1(OC)cc(OC)c2ccnc(C(C)Sc3cccnc3C)c2c1 17506,c1(C(C)C)ccc(C(=O)NCCn2cc(-c3cccs3)nn2)cc1F 17507,c1(C(N(CCNC(=O)C(C)NC(=O)NC)CC)=O)ncc(CSC)s1 17508,c1(C(=O)NCC(CCCC)NC(=O)CCCCOC)ccnc2[nH]cnc12 17509,c1(C(C)=O)ccc(C(=O)NC(C)(C)CNC(=O)C(C)OCc2ccccc2)nc1 17510,C1(C(N(C(C)C(=O)NCC(C(C)(C)C)OC)CC)=O)CCN(C)C(=O)C1 17511,c1(C(=O)OC)ccnc(N(CCCNC(c2occc2Br)=O)CC2CCCC2)n1 17512,C(CC(C)CCNC(c1nocc1Br)=O)NC(C(C)NC(c1ccoc1)=O)=O 17513,C12(CNC(CCSC)=O)CCC(C1)N(C(c1cccc(-c3ccc[nH]3)c1)=O)C2 17514,N1(C(C(CC=CCC)C)=O)CC(C(=O)N(CC(F)Cl)C)CC12CCC2 17515,C1(C)(C(=O)NCC(C)CN(C)C(c2cnn(C(F)(F)F)c2)=O)CCNC1 17516,C1(C(N2CCCC(CCC(=O)NC3(C)CCC3)C2)=O)CC2CCCC2C1 17517,C1(NC(C(CCCCC)O)=O)CCN(C(=O)C(C)(O)C2CC2)CC12CCC2 17518,c1(C(C(=O)NC2CC(NC(c3c(CC)occ3)=O)C2)(F)F)ccc(Br)cn1 17519,c1(C(N2CCCC2c2ccsc2)C(=O)NCC)ccc(C(=O)OC)cc1 17520,C(=O)(C(C)(C)C(=O)NCCC(COC(c1cc(Cl)ncc1OC)=O)OC)OC 17521,CC1(C)CCCC(C(=O)NC2CN(c3nc(Cl)ncc3C(F)(F)F)CC2(C)C)C1 17522,N(C(=NCCc1ncccc1C)NCc1nn(C)cc1Br)C(COC)C 17523,N1(C(C(C)n2ccnn2)=O)CCN2CCN(C(=O)C(C)n3ccnc3)CC2C1 17524,N1(C(C(C)=C2CCCC2)=O)C2CCCC1CN(C(C1CC3CCC1O3)=O)C2 17525,CCC(CC)C(C)C(=O)N(CC(=O)NC1(COC)CC(C)(C)C1)CCOC 17526,c1(CC)occc1C(=O)N(CCCN(C(=O)CC#N)C)C 17527,c1(C(=O)NC2C(CC)CN(C(=O)CCNC(N)=O)CC2)cc(C)cc(C)c1N 17528,C12(NC(C(C)(Cl)Cl)=O)CN(C(c3ccc(=O)oc3)=O)CC1CS(=O)(=O)C2 17529,CC1CCCN(C(c2cnn(C(F)(F)F)c2)=O)C1CNC(c1ccsn1)=O 17530,c1(NCC(CCC)N(C)C)ncccc1S(=O)(=O)NCc1cc(F)cc(F)c1 17531,C1(CNC(=O)COCC2CCOC2)CC2CCC(C1)N2C(=O)C=Cc1cnc[nH]1 17532,c1(C(=O)NCC(C2CCN(C(CC(C)SC)=O)CC2)(C)O)c(O)cccc1F 17533,CCCCC(F)C(=O)NC1CC(OCC(N2CCC(C(F)(F)F)C2)=O)C1 17534,c1(SC)cccc(C(=O)NC2CCC(CCNC(=O)CC3(NC(C)=O)CC3)C2)n1 17535,CCC(CC(=O)N(CC(=O)NC(C)Cn1cnnc1)C1CC1)CC(C)C 17536,C1(F)(CNC(C=CCCC)=O)CCN(C(=O)CN(C)CCOC)C1 17537,C(=O)(C(O)CC(C)(C)C)NCC1(F)CCN(C(C(CC)C#N)=O)CC1 17538,C(=O)(C1=C(Cl)CCC(C)C1)NCC1(CNC(C(C)S(N)(=O)=O)=O)CCC1 17539,C1(CC(=O)NCCCc2n(C)c(S)nn2)CC2(CCCCN2C(N)=O)C1 17540,N1(C(C(CC)(C)O)=O)CCCC(N(C(=O)Cc2cc(Cl)cc(Cl)c2)CCO)CC1 17541,Cc1ccc(CSc2ccc(C(=O)NC3(C4CCCCO4)CC3)o2)cc1 17542,c1(C(C)(C)C)cc(C(c2nnnn2C2(C)CC2)NCC(CO)C2CC2)on1 17543,CN1CCOCC1CC(=O)NC1CCC1NC(C1CC(n2ccnn2)C1)=O 17544,c1(C(N2C(CNC(C(C=C)(C)CC)=O)CC(F)C2)=O)cc(S(=O)(=O)NC)oc1C 17545,C(C(=O)NOCC1CCS(=O)(=O)C1)(c1ccccc1)NC(C1C(CC(C)(C)C)C1)=O 17546,C=CCC(C(=O)NCCC1(SC)CN(C(=O)C(C2CCCCC2)O)C1)NC(C)=O 17547,N1(C(C(=O)NCCCSCC)C2CC2CC)CC(N2CCOCC2)C(C)C1 17548,N1(C(c2nn(CC)c(C)c2)=O)CCC2(CCCN2C(=O)C(O)C2CC2)CC1 17549,Cc1nn2cc[nH]c(=O)c2c1C(=O)NCCC(O)CNC(=O)C(C)C(C)(C)C 17550,C1(C)(C(=O)NC2CCN(C(COCC#C)=O)C2C2CC2)CCS(=O)(=O)CC1 17551,c1(NC2CC(CC)C2)ccc(S(=O)(=O)Nc2ccc(F)cc2C)cc1F 17552,N1(C(c2cnc(CCC)s2)C(=O)NCC2CC2)CC(C(=O)OC)CC(CC)C1 17553,CC(C)CC(C)(C)CNC1(c2nnnn2C2CC2)CCCC1N(C)C 17554,C1(C(N(C(CC(=O)NC)C)C)=O)COCCN(CC2CCCO2)C1 17555,C1(NC(C(C)NS(C)(=O)=O)=O)CN(C(C2C3CCCC23)=O)C2(CCOCC2)C1 17556,c1(NC(C2COCCN2C(C2CC(O)C2)=O)=O)c(F)c(F)nc(F)c1F 17557,c1(OC)cc(C)[nH]c(=NCC2CN(C(c3cccc4c3COC4)=O)CCO2)n1 17558,C1(C)(CNC(c2n(CCCC)nnn2)c2ccnn2C(C)C)CCC(=O)N1 17559,CC1(C)C(NC(C2CC23CCOCC3)=O)CCN1C(c1ccnc(F)c1N)=O 17560,c1(C(=O)NC2CCN(C(c3c(C)c(F)ccc3N)=O)C2)c(F)cccc1[N+](=O)[O-] 17561,CS(C)(=O)=NCC(=O)NC1CCOCC1NC(=O)C=Cc1ccccn1 17562,C#CCC(CC#C)C(=O)NCC12CC1CN(C(C1(COC)CCCC1)=O)C2 17563,C12(NC(CCS(C)=O)=O)CCOCC1CN(C(c1cccc3oncc13)=O)C2 17564,C1(NC(C2N(C(c3c(CC)cc[nH]3)=O)CSC2)=O)CC2(CCOC2)C1 17565,c1(CC(N2CCC(CCNC(CCC=C=C)=O)C2)=O)ccc2[nH]ccc2c1 17566,N1(C(=O)CCCC2CCCO2)CCC(CO)(CNC(=O)CN2CCC(O)CC2)C1 17567,c1(C(=O)NC2C(CNC(c3c(CC)[nH]cc3)=O)CCCC2)nn(C)c(N)c1C 17568,Cc1nc(-c2cccs2)sc1C(=O)NCC1CC1CNC(c1csc(F)c1)=O 17569,Cc1ccc(-c2ccnn2C)cc1NC(N1CCC(c2ncc(Br)cn2)C1)=O 17570,N1(C(CCCOC(C)=O)=O)CC2CCC2(CNC(=O)CN2CCS(=O)(=O)CC2)C1 17571,C1(NC(C2C(CC(=O)OC)CC2)=O)CCCN(c2ncc[nH]c2=O)C1 17572,N1(C(c2cc(C)c(Br)c(Cl)n2)C(=O)NCCSC)CCC12CCN(C)CC2 17573,c1(C(=O)NC(CN(C(=O)C2=CCCC2(C)C)C)(C)C)cc(F)cc(N)c1F 17574,C(=O)(CCS(C)(=O)=O)NCC(CC)(CC)NC(C1CC2C=CC1O2)=O 17575,Cc1cc(Cl)ccc1C(N1CC(CNC(=O)CSCc2cccs2)C1)=O 17576,C1(C(N2C(C)C(C(F)(F)F)OCC2)=O)CC2CC1CN(Cc1ccccc1)C2 17577,C1(NC(Cn2c(C)nnn2)=O)CN(C(=O)C(C)O)CCC1c1ccccc1 17578,Cn1cc2c(n1)CCC(C(N1CCC(NC(=O)C=Cc3ccc(Cl)cc3)C1)=O)C2 17579,Nc1ncc(C(=O)NCC2CN(C(=O)Cn3cnnn3)CC2C(F)(F)F)cc1Cl 17580,C1(C(=O)N(CCCN(C)C(C2CC2C(F)F)=O)C)(OC(C)=O)CC1 17581,N1(S(Cc2nc(C(C(C)C)c3ncn[nH]3)on2)(=O)=O)CCCCCC1C(=O)NO 17582,CC1CN(C(c2coc(C3CCC3)n2)=O)CCN1C(c1cc(Cl)c[nH]1)=O 17583,c1(NC2CN(C(c3cc(C)cc(C)c3)=O)CC(F)C2)ncnc2occc12 17584,CC(C)C(C)CC(=O)NC(CN(C)C)C(=O)N1CC(c2cncnc2)C1 17585,CC(C)(C)C(CNC(C1CC2CCC1CC2)=O)C(=O)N1CCC(CCO)CC1 17586,C1(CNC(c2ccc(C=C)cc2)=O)CN(C(=O)CO)C2(CCC2)C1 17587,C(=O)(C1=CCC(C)CC1)NCC(CC)(CC)NC(=O)Cn1nnc(=N)[nH]1 17588,C1(C(N2C(Cn3cc(C(C)OC)nn3)CCCC2)=O)Cc2cccc(C)c2O1 17589,N1(C(CCCCCC)=O)CC(C)CN(C(=O)CCC=CC(C)C)CC1C 17590,c1(C(=O)NC(CNC(C2N(C(C)C)CCCC2)=O)C2CC2)ccc(N)c(O)c1 17591,c1(C(N(CC(C)N(C)C(C2CCC(=O)N2)=O)C)=O)coc2c(F)c(Cl)ccc12 17592,CC1CCOC(C(=O)NCCCN(C(=O)Cc2cccs2)C2CC2)C1 17593,c1(C(=O)NC2C(CNC(C3C(CC)CCO3)=O)CCC2)ccc(C2CC2)cc1C 17594,CC1(C)C(C)(C(=O)NC2CN(C(c3sccc3C(F)F)=O)CCC2CO)C1(C)C 17595,c1(-c2n(CCCC=C)ccn2)ccc(C2CC2c2ccc(-c3nn[nH]n3)cc2)cc1 17596,C1(C(N2CCC2CNC(C23CCN(CC2)C3)=O)=O)CC12CCCOC2 17597,N1(C(=O)Nc2c(CC)cccc2)CC2CC1CN2C(=O)OC(C)(C)C 17598,C1(C(N2CCC(CCNC(c3ccccc3Cl)=O)C2)=O)CCC2(CC1)CC2(F)F 17599,N1(C(Cc2cc(OC)no2)=O)CC(CNC(=O)C(C)(F)C(C)(C)F)CC(C)(C)C1 17600,N1(C(CCCC#N)=O)CC2CC(C1)C2NC(=O)COCC(F)F 17601,CC1CCN(C(C2C3CCCC23)=O)CC1N(C)C.C12CC(C1)OCC(=O)N2 17602,N1(C(=O)CCc2ccsc2)CCC(CNC(C2(F)CCOC2)=O)C1 17603,C1(NC(C2CC(n3cnnc3)C2)=O)(CO)CCN(C(=O)CC2CC2)C1 17604,C1(C(=O)NC2(C)CC(NC(c3ccc(C(=O)OC)cc3)=O)C2)CC2(CCO1)CC2 17605,C1(NC(c2n(CC)cc(Cl)c2)=O)CCC(C)N(C(=O)C(=Cc2cccnc2)C)C1 17606,c1(CC)nc(C)oc1C(=O)NC(CO)C(=O)NCC1CCCSC1 17607,C(=O)(C1=CC2CCCC12)NCC=CCNC(c1cc(C)c(Cl)s1)=O 17608,N1(C(CC#N)=O)CCC2C(C(=O)NC3CCCCCC3F)C2C1 17609,N1(C(N2CCC(C)CC2)=O)CCc2c1ccc(F)c2F 17610,C1(CC(=O)NCCc2n(C)c(=O)on2)CN(C(=O)C2=COCC2)CC12CC2 17611,c1(C(NOCC(c2ccccc2)C)=O)cc(O)c(F)cn1 17612,C1(CNC(c2n(CC)ncc2Br)=O)CC2CCC1N(C(=O)C=CCOC)C2 17613,C=CCCCCCCCC(=O)N1CC2(C1)CN(C(c1cnccc1Cl)=O)CCO2 17614,C(CS(=O)(=O)CC(=O)NCc1ccc(C(=O)NCC(CO)C2CC2)nc1)OC 17615,C(=O)(C(O)C(F)(F)F)N(C(CC(N1CCC(C)(C(=O)NC)C1)=O)C)C 17616,C=CC(CC)CC(=O)NCCOC1CCN(C(=O)C(Cc2cnc[nH]2)N(C)C)C1 17617,C1(C2CCCN(C(=O)C3=C(Cl)CCC3)C2)(NC(C2(C)ON=C(C)C2)=O)CC1 17618,c1(CC)ccc(OCC(=O)NC2CCN(C(C3(C)COCCO3)=O)C2)cc1 17619,c1(C(=O)NC(CC)CNC(C2C(c3n[nH]c(C)n3)C2(C)C)=O)n[nH]cc1[N+](=O)[O-] 17620,C1(CNC(C(N2CCOCC2)C)=O)CCC(NC(c2ccnn2CC(F)F)=O)C1 17621,c1(C(N(C)CCNC(C2CC3C(C2)C3(F)F)=O)=O)cc(=O)c2ccncc2o1 17622,c1(OC)cc(C(=O)N(c2ccccn2)CC)c(NC(c2nccnc2Cl)=O)cn1 17623,C(C)(CO)(C(=O)NCCCN(C(c1cnc(N)cn1)=O)C1CC1)OC 17624,C(C)(CCC(=O)NC(C)CC(C)NC(=O)CCC1CCCC1)SC 17625,N1(Cc2ccc(C(=O)NCc3ccc(CC)cc3)cc2)CCC(C#N)(OC)C1 17626,C(CC(=O)NC1CCCC1NC(c1c(C)nn(C)c1Cl)=O)(C1=CCCC1)OCC 17627,Cc1nc2ccc(C(N3CC(N(C)C(C4CC4(C)C)=O)C4(CC4)C3)=O)cc2s1 17628,c1(SC)cc(C(=O)N(C2CCC(NC(c3cnc(C)n3C)=O)CC2)C)n(C)n1 17629,C(=O)(C(C)C(O)C(C)C)N1CCC2C(C(=O)NCC(CSC)OC)C2C1 17630,N1(C(CNS(N)(=O)=O)=O)CC2CCCN(C(c3cc4n(n3)CC(F)C4)=O)C2C1 17631,Cc1ccc(O)c(NC(c2cc(CNC(C3(COC)CCOC3)=O)cs2)=O)c1 17632,C1(C(=O)O)CN(C(c2cc[nH]n2)=O)CC12CN(C(c1cnc(Cl)cc1I)=O)C2 17633,N1(C(CCOCCN(C)C(C2CC(C)(C)CO2)=O)=O)CCC2(CCCCC2)C1 17634,CC1(F)CCC(C(=O)NC2CCC(NC(C3CC(O)C3)=O)CC2)CC1 17635,Cc1cc(CNC(=O)CC2CC(NC(C3CCOC3C3CC3)=O)C2)nn1C 17636,CC(C)P(=O)(CC(=O)NCC(O)CN(C)C(c1ccoc1C1CC1)=O)C(C)C 17637,c1(C(C(=O)NCCC2(O)CN(C(C(C)SC(C)C)=O)C2)C)ccccc1Cl 17638,c1(-c2sc(CCOC)c(C)c2)ccnc(OC)c1SC 17639,C1(NC(C(C=C)c2ccccc2)=O)CCN(C(c2n[nH]c(CC)n2)=O)C(C)C1 17640,Cc1cc(C)n(C2CCCN(c3nnnn3CCS(N)(=O)=O)C2)n1 17641,Cc1cc(=O)oc(C)c1C(=O)NC1CCN(C(=O)C(C)Cc2ccc(O)cc2)C1 17642,N1(C(c2cnn(CC)c2C)=O)CCCCC(CNC(C2(F)CCOC2C)=O)C1 17643,c1(-n2cc(C(C)NC)nn2)ccccc1C(=O)NC(C)Cc1noc(C)n1 17644,CN=C(NCc1csc(CC2CCCC2)n1)N1CCC(C)C1C 17645,n1(CC(=O)NCC(C(C)C)NC(c2cncc(OC)n2)=O)cc2ncccc2n1 17646,C=Cc1cc(C(=O)NCC2(O)CCN(C(=O)CC3CCCN(C)C3)C2)cc(F)c1 17647,C12(C(N(C3CCN(C(=O)CN4CCCC4C)CC3)CC)=O)CCC(F)(CC1)C2 17648,CCC(CC(=O)N1CCC(CO)(CNC(=O)CNS(=O)(=O)CCOC)C1)SC 17649,C(CC)(CC)(CCNC(C1C=CCCC1)=O)NC(c1c(NC)cncc1)=O 17650,N1(C(c2c(C)cc(Cl)cc2)=O)CC2CN(C(C34CCCC3C4(F)F)=O)CC2C1 17651,N1(C(C2C(C(=O)OC)C2)=O)Cc2ccccc2CC1C(N1C(C)CCC1C)=O 17652,c1(CNC(c2n[nH]cc2F)=O)cccc(F)c1.O=C1CN(C2CC2)CCN1 17653,CC12CC(NC(c3cncnc3)=O)(C1)C1(CN(C(=O)CCC3CC3(F)F)C1)O2 17654,c1(-c2cc(C(=O)NCc3cc(Br)ccc3O)c(F)nc2)ccc(F)c2[nH]ncc12 17655,O=C1CC(N=c2nc3scnc3c(NCC3CCCC(O)C3)[nH]2)CN1C1CC1 17656,C(C1c2ccsc2CCN1C(=O)CC(C)CC)NC(CN(CCC#C)C)=O 17657,c1(OC)cncc(C(N2CC(NC(=O)COC3(C)CCOCC3)CC2C)=O)n1 17658,N(C)(C1CCc2c(Cl)cccc21)C(c1c(C)[nH]c2cc(Cl)ccc21)=O 17659,N1(C(C(C)C)=O)CCC(C2CC2)(CNC(c2coc(O)n2)=O)C1 17660,c1(OC(C)C)cccnc1C(N1CC2CC2(CNC(C2CC2C)=O)C1)=O 17661,c1(C(=O)NCC(C2(O)CCN(C(=O)CNC(N)=O)C2)C)cc2c(cn1)OCCO2 17662,Cc1ccc(O)c(C(=O)NCc2cc(C(=O)NOC(c3c(C)noc3C)C)n[nH]2)c1 17663,C12(C(=O)NCC3CC(OC)CN3C(=O)CN(C)C)CCC(C1)C(C)(C)O2 17664,N1(C2CC(OC(C)C)C2)CCCC(C2CCCCN2C(c2cc(F)n(C)n2)=O)C1 17665,c1(C(=O)NCC2(F)CCC(NC(Cc3nc(C)sc3)=O)C2)c(Cl)ccc(O)c1N 17666,C=CC1(C(=O)NCCOCCN(C)C)CCN(C(=O)CC2CCCN2C)C1 17667,c1(C(N2CC(COC)(NC(=O)C(C)C3CCCC3)C2)=O)cc(C)c(OC)c(C)c1 17668,C1(C(N2CC(C(C(N3CCC(C(=O)OC)C3C)=O)OC)C2)=O)CCC(=O)N(C)C1 17669,c1(C(=O)NCCCC(C)NC(=O)C(F)C2CC2)ccc(C(F)F)c(F)c1 17670,C1(NC(CC(C)SC)=O)CC2(CCN(C(=O)CC3CCCC(C)C3)C2)C1 17671,N1(C(c2c(C(C)C)c[nH]n2)=O)CCC(F)(F)C(NC(=O)C2CC2)C1 17672,C1(OC)CCC2(C(N3CC(CCNC(C4CC(N(C)C)C4)=O)C3)=O)CC12 17673,c1(C(=O)NCC2(NC(C(CC)C(C)O)=O)CCOCC2)nccc2cc[nH]c12 17674,c1(C(=O)NCC(C(C)C)NC(C2CC3CCC2O3)=O)ccc2ncnn2c1 17675,Cc1coc(C)c1C=CC(=O)N(C(C)CCNC(=O)CC(C)(C)CN(C)C)C 17676,C1(C(c2n(CC(=C)C)nnn2)(C)NC2CC3(C2)CC3(F)F)CCCCC1(F)F 17677,C1(NC(CC2(C)CC2)=O)CC2COCC(C1)C2NC(c1cnn(CCO)c1)=O 17678,C(=O)(C1=CC2CCC=CCCC12)N1CCC(NC(CS(=O)(=O)NC)=O)C(C)C1 17679,C(c1ccccc1F)=CCC(=O)NCC(CC)(C)NC(c1cnc(O)n1C)=O 17680,CC(C(=O)N1CC(O)CC1CC(N1CC(C(=O)N(C)C)C1)=O)S(C)(=O)=O 17681,C1(NC(CC(=O)NCC#C)=O)CC2CCC(C1)N2C(C12CCC(F)(CC1)CC2)=O 17682,c1(C(N2CCN(C(Cc3nc(C)[nH]n3)=O)C(CO)C2)=O)c(C)[nH]c2ccccc12 17683,C(c1ccc(C(F)(F)F)cc1)=CC(=O)NC1(C)CCN(C(c2ccsn2)=O)C1 17684,C12(C(=O)NC3C(CC)CN(C(=O)CCCC(C)C)CC3)CCC(CC1)C(C)(C)O2 17685,c1(NC(=O)CO)ccc(C)cc1C(=O)NC1CC(OC)C1.C(CCOC)OCC 17686,C12(NC(=O)CCSC(F)(F)F)CCC1CN(C(=O)C=CC1CCOC1)C2 17687,CC1=C(C(=O)NCCC2CCN(C(=O)CCCc3ccncc3)C2)CCO1 17688,C(=O)(C(F)(F)CCn1cccn1)N(CCCn1cc(C(CC)O)nn1)C1CC1 17689,C(c1ccc(O)cc1)=C(C)C(=O)NOCc1cc(-c2cccnc2O)ccc1OC 17690,CC1(C)CN(C(=O)CC2OCCCO2)CCC1C(=O)NCCC(O)C(F)(F)F 17691,C1(CC)CN(C(C2CCNC2=O)=O)CCN1C(c1cnc(OC)nc1C(F)F)=O 17692,C1(O)(C(C)NC(c2c(C)scn2)=O)CCN(C(c2ccnc(F)c2)=O)C1 17693,Cc1noc(C)c1C(C)C(N1CC(C(N)=O)(N(C)C)C1)=O 17694,C(=O)(CCCC(C)(C)C#N)N1CC(NC(C(C2CCCN(C(N)=O)C2)C)=O)C(C)C1 17695,C1(C(=O)NCC(C2CC2)NC(c2ccc[nH]2)=O)CCCN(c2cc(O)ncn2)C1 17696,c1(C(=O)NCC2CN(C(CCOCCOC)=O)C2)ccc(N)c(C)c1Cl 17697,c1(CC2(C#CC(=O)NCC3C(CC)CCCC3)CC2)c(OC)nc(C)nc1Cl 17698,c1(OC)c[nH]nc1C(=O)N(C(CNC(=O)CN1CCCC1C)C1CC1)C 17699,Cc1cn(C)cc1C(=O)NC1C=CC(C(=O)NCCOCCC2CC2)C1 17700,C1(c2noc(C(F)(F)F)n2)CN(C(=O)OCC(C)(C)C)CC1C1(NC(CC)=O)CC1 17701,CC(C)(C)CC(=O)NCC(=O)NC1CC(CNC(=O)CSc2ccc(F)cc2)C1 17702,N1(C(COCC=C)=O)CC2(CCC2CNC(=O)C(=O)NOC)C1 17703,c1(C(N(C(c2ccccn2)C)C)=O)c[nH]n(C)c1=O 17704,CC(C(C)(C)NC1COCC1C(N1CCCCC1)=O)NC(=O)OC(C)(C)C 17705,Cc1nc(N2CCCC3(CCN(C(C4CC5CC5C4)=O)C3)C2)c2cnn(C)c2n1 17706,Cc1nc(C2CCOC2CN(C(=O)Nc2cnn(C(C)C)c2)C(C)C)n[nH]1 17707,N1(C(c2ccc(C(C)C)cc2)=O)CCC2(NC(c3cn(C)ccc3=O)=O)CC2C1 17708,c1(COC)cc(=NC(C)CC(C)NC(=O)C(C)NC(C)=O)[nH]c(C)n1 17709,C1(C)(C(N2CC(O)(CN(C(=O)Cc3n[nH]c(=N)s3)C)C2)=O)Cc2ccccc2C1 17710,N(C1COc2ccccc21)C(C1N(Cc2cc(OCC)c(O)c(Br)c2)CCC1)=O 17711,N1(C(CNC(=O)OC)=O)CC2C(CNC(=O)C(c3ccc(F)cc3)N(C)C)C2C1 17712,C1(C(=O)NCC(C(C)C)O)C2CN(C(=O)CC3CCOC3=O)CC12 17713,C1(CC(=O)NCc2cc(C)ns2)CN(C(=O)CCc2cncs2)CCO1 17714,C(=O)(C(C)(C)C(=O)N(C)CC1CCCN1C(=O)CCc1csc(C)n1)NC 17715,C(=O)(C(F)(CNC(=O)C1=CCN(C)C1)C(C)C)N(C)Cc1cccc(C)n1 17716,N1(C(C2CC(=O)NCC2)=O)CC(NC(=O)CCc2cnc[nH]2)C(F)(F)C1 17717,CCCC(C)(C)C(=O)N(CC(=O)O)CCC1CC1 17718,c1(COC)cc(F)c(C(=O)NCC(C)CNC(=O)CSC(F)(F)F)c(F)c1 17719,C(=O)(C1=C(Cl)CCCC1)NC1C(N2CCN(C(C(C(C)C)C)=O)CC2)COC1 17720,CC(CC1(C)OCCO1)CN=c1[nH]c2c(c(=NCn3ccnn3)[nH]1)SCC2 17721,C12(C(N(C3CCN(C(=O)C(O)c4ccsc4)CC3)C)=O)CCCC1CC(=O)CC2 17722,C1(CNC(C2(C(=O)NC)CCC2)=O)C2CCC(C2)N1C(c1ccc(C(N)=O)[nH]1)=O 17723,N1(C(C2C(C)C2(F)F)=O)CCN(C(c2cscc2C(F)F)=O)CC(C)(C)C1 17724,C1(C(=O)NCCOCCC(=O)NCC(C)(O)CC)CCCC2(CC2)C1 17725,CC1CC(N(C(=O)C(=O)N(C)Cc2ccc(Cl)cc2F)C)CC(C)O1 17726,Cc1ccc(C(=O)NCCC2CCN(C(C3CCOC3=O)=O)C2)c2ncccc12 17727,N1(C(c2c(C)cc[nH]2)=O)CCOC2CN(C(C3CC34CCCCCC4)=O)CC12 17728,N1(C(C(=O)NCCCCCCCC)=O)CCc2sc(C(=O)N(C)C)nc2C1 17729,CC1CN(C(C2CCCC(CF)C2)=O)C(C)CN1C(=O)CC1CSCCO1 17730,C1(C(=O)NCCCCCC=C)CCN(C(=O)C(C)(C)C(F)F)CC1C 17731,c1(C(=O)NC2CC2C(=O)Nc2ccc(Cl)c(Cl)c2F)ccc2cnccc2c1 17732,CCCCC(C)C(=O)N1CC(CNC(=O)CCOCC)C(O)C1 17733,Cc1c[nH]c(C#N)nc1=NCCN(C)C(C1COc2ccc(F)cc2C1)=O 17734,C1(NC(C(C)NC(N)=O)=O)CCN(C(=O)CCCc2csc(=N)[nH]2)C12CC2 17735,c1(OCC)ccc(Cl)cc1-c1nc(Cc2cc(F)ccc2Br)no1 17736,N#CC1CN(C(C2CCCN2C(C2CC(OC3CC3)C2)=O)=O)CC12CCC2 17737,c1(C(N(CCCCCC)CCNC(=O)Cc2ccco2)=O)ccc(OC)cc1C 17738,CC(C)C(O)CC(=O)N(C1CCN(C(C23CSCC2C3)=O)CC1)C 17739,C1(CC(=O)NCC(CC)C)CN(C(c2c(C#N)cnn2C)=O)CC12CC2 17740,c1(C(c2n(CC)nnn2)NC(C2CCC2)C2CC2)ccc(OC)cc1[N+](=O)[O-] 17741,C1(NC(C=C(C)C(C)C)=O)CCCCC1CNC(c1ccno1)=O 17742,C1(C(=O)NC(CNC(c2ccc(C(F)(F)F)s2)=O)C2CC2)CCCCS1 17743,n1(CC)nnc2c1CCC(C(=O)NCC1CCN(C(C3COC(=O)N3)=O)CC1)C2 17744,c1(C(=O)NC2(CCNC(C3C(C(=O)OC)C3)=O)CC2)cccc2c1NC(=O)CO2 17745,C(=O)(C(CC=C)CC(C)C)NCC1C2CN(C(COc3ccc(C#C)cc3)=O)CC21 17746,c1(C(N2C(C(=O)NCC(C)CC3CC3)C=CC2)=O)cc(F)ccc1O 17747,C1(NC(c2ccc3occc3c2)=O)CN(C(C2CC2CF)=O)CC2(CCC2)C1 17748,n1(CC)cc(-c2ccc(CC(=O)N(CC)Cc3ccncc3)nc2C)ccc1=O 17749,c1(C(N2CCC(NC(C3(OC)CCCC3)=O)C(O)C2)=O)ccc(P(C)(C)=O)cn1 17750,c1(C(=O)NCCCOCCC(=O)NCC2(SCC)CC2)ccc(C)cc1C 17751,C(=O)(CCS(=O)(=O)Nc1ccccc1)N1CCCC(NCc2c(C)ccs2)C1 17752,O(NC(=O)C(C)(C)C1CCCN1C(=O)CCNC(=O)NC)CC#C 17753,C1(NC(C=Cc2nc(C)sc2)=O)CC(CNC(=O)CC2(O)CCC2)C12CCC2 17754,c1(C(=O)Nc2c(C(C)(C)C)ncs2)cnc(C2CCNCC2)nc1 17755,N1(C(c2cn(CCC)nn2)C(=O)NC2CCCC2)C2CCC1CN(C)CC2 17756,C1(CC(=O)Nc2ccc(Br)nc2)COCCN1Cc1ccc(-c2ccccc2)s1 17757,CCCCC(C)(F)C(=O)N1CC(NC(C23CC(C)(C2)OC3(C)C)=O)C(O)C1 17758,C(=O)(C(CNC(=O)C1=CC2(CCOC2)C1)CC(C)C)Nc1c(COC)cccc1 17759,c1(C2(N)CC2)ccnc2ccccc12.n1(CC(=O)C=O)cc(C(F)(F)F)cn1 17760,C12(C(=O)NC)CCCCC1CN(C(c1c(C(=O)OC)cccc1[N+](=O)[O-])=O)C2 17761,N1(C(=O)OC)CC2(C1)CN(C)CC2c1cc[nH]c(=NCC2CCC(C(N)=O)O2)n1 17762,N1(C(CSCC)=O)Cc2ccccc2CC1CNC(c1cc(Cl)ccc1OC)=O 17763,NC(=O)CCCC(=O)N1CCC(C2OCCCC2Nc2ncc(O)cn2)CC1 17764,CC1CC2(C(=O)N(C)CC3(NC(c4cc(-c5ccns5)on4)=O)CC3)CC12 17765,CCC(C)CCCCC(=O)NC(CCOC)C(=O)N(C1CN(C)C1)C 17766,CN1CCN(c2ccc(C(N3CC(NS(=O)(=O)CC4CC4)C(O)C3)=O)cc2)CC1 17767,c1(C(N2CC(C(=O)NC3C(C)(C)COC3=O)C(O)CC2)=O)[nH]nc([N+](=O)[O-])c1Br 17768,c1(C(N2C(CN(C)C(C3NC(=O)NC3=O)=O)CCC2)=O)ccc(C(F)F)cc1F 17769,N1(C(c2c(C)c[nH]n2)=O)CCCC(NC(=O)Cc2ccsc2Cl)C1C 17770,c1(C(N2C(C3(NC(C(CCSC)O)=O)CC3)CCCC2)=O)cc([N+](=O)[O-])c[nH]1 17771,CN1CCC(NCCOCCN(C(=O)C(c2ccc(Br)cc2)(C)O)C)CC1 17772,C1(C(=O)NCCOCCCC#C)CCN(C(C2CC(C)CCO2)=O)C1(C)C 17773,C1(CNc2c(C)c(N(CCC(N)=O)C)ncn2)CCC2(C1)CC2(F)F 17774,C1(C2CC2)(CNC(c2c(CCC)n[nH]c2)=O)CCN(C(=O)CC(C)(F)F)C1 17775,C(=O)(CCCC(c1ccccc1)NC(=O)Cc1cocn1)OC 17776,C(=O)(CCCC(=O)NCC)NC1(CC=C)CCN(C(C2CNC(=O)C2)=O)C1 17777,C1(F)(CNC(c2cccc(SC)c2)=O)CCN(C(=O)C(F)=CC2CC2)CC1 17778,c1(C(=O)NCC(CNC(Cn2c(C)nnn2)=O)(C)C)cccc(OC2CCC2)c1 17779,c1(NC(CN2CCCC(C)C2)=O)ccc2nn[nH]c2c1 17780,C(=O)(CCCNC(C)=O)N(C1CCN(C(=O)CC(=O)N2CCOCC2)C1)CCC 17781,C1(F)(CNC(=O)CSC(F)(F)F)CC2CCC(C1)N2C(=O)CC1CS(=O)(=O)C1 17782,Cn1cnc(NC(C23CC(C(=O)NCc4ccn(-c5ccccc5)n4)(C2)C3)=O)c1 17783,c1(C(=O)NC2C(CNC(C(COC)(F)F)=O)CCCC2)cnc2c(c1)CCC2 17784,c1(C(=O)NC2C=CCCC2)cccnc1CNC(C1CS(=O)(=O)C1)=O 17785,C1(C)(CCCC(=O)NCc2ccc(C(=O)NCc3cc(C)sc3)o2)NC(=O)NC1=O 17786,S(=O)(=O)(c1cnc(C(C)(C)C)[nH]1)N(C1C(CCC)C1)C 17787,NS(=O)(=O)c1ccsc1C(N1CCC(CO)C(NC(c2cn[nH]c2)=O)C1)=O 17788,c1(C(N2CCC(CCC(C)O)CC2)C(=O)NC2CC2)ccc2c(c1)CCCO2 17789,c1(C(N2CCC(N3CCN(C(CCSC)=O)CC3)C2)=O)c(C)cc(O)nc1C 17790,N1(C(CCC(C)N(C)C)=O)CCC=C(C(=O)N2CCC(C)(C#N)CC2)C1 17791,Cc1ccc(C(C)C(=O)NCCOCCCNC(C2CC(Cl)(Cl)C2)=O)o1 17792,c1(OCC)ccc(SCC(N2CC(NC(=O)CCc3cn(C)cn3)C2)=O)cc1 17793,C1(C(=O)OC)(C)CCCS1(=O)=O.c1(-c2cn(CC)nn2)cn(C)nc1C(=O)O 17794,c1(C(=O)NCC2C(C(N3CC(CC)SCC3)=O)OCC2)ccc2cc[nH]c2n1 17795,C1(NC(CC2(C(=O)OC)CC2)=O)CCCCN(C(C2CC(F)C2)=O)C1 17796,N1(C(CCCOC(C(C)C)=O)=O)CCCC(C(=O)Nc2cccc(O)c2)C1 17797,c1(CN2CCCN(c3ncnc(C)c3Br)CC2)oc2ccccc2c1C 17798,C1(C(N(C)CC2CCC2)=O)CCCC1CNC(C1CS(=O)(=O)C1)=O 17799,C1(C)(C(=O)NC2(C)CN(C(=O)CC(C)(O)c3ccccc3)C2)CCCCNC1=O 17800,CC(C#N)C(=O)N(CC(O)CN(C(=O)CN(CCc1ccccc1)C(C)=O)C)C 17801,C1(CCOC)(C(=O)N(CCCO)C)CCN(C(=O)CN(C)C2CC2)C1 17802,C#CCCCC(C)C(=O)NCc1ccc(C(N2CCCC(C)(C)C2C)=O)cn1 17803,N1(C(C(CC)(C)C)=O)CCN(C(C2CCCC23CCC3)=O)C(C)C1 17804,c1(C(=O)NC2(C)CC(NC(C3N(C(C)=O)CC(O)C3)=O)C2)cc(O)cc(C#N)c1 17805,Cn1cnc(C=CC(=O)NCC(=O)NC2CC(O)C(F)C2)c1 17806,n1(CC)cc2ccc(C(N3CC4CCOC4(CNC(=O)CSC)C3)=O)cc2n1 17807,c1(C(=O)NC2CCCC(NC(CC3C(C)(C)C3)=O)C2)c[nH]cc(F)c1=O 17808,c1(-n2c(CC(CCC)C)nc(CCC)n2)nc2ccccc2n1C 17809,Clc1ccc(-c2cc(-c3nc(C4CCCC4)nn3C34CC(C3)C4)n[nH]2)cc1Cl 17810,c1(CNC(C2(C)C=CCC2)=O)cccc(NC(=O)CC2CCSC2)c1 17811,C1(C)(C(=O)NC(C)Cn2ccnc2)CCN1C(=O)COC1CCCCC1 17812,C1(NC(C(C)NC(=O)NC)=O)CN(C(c2cc(C)co2)=O)Cc2nccn2C1 17813,C1(c2cn(CCOCC)nn2)CN(C(=O)Cc2csc(C)c2C)CC1C 17814,c1(CNC(CC(C)NC(CCCOC)=O)=O)cc(F)ccc1C 17815,N1(C(c2ccc(OC)cc2)=O)CCN(C(c2cc(OC)no2)=O)C(CF)C1 17816,c1(OC)cc(C(N2CCC(NC(=O)C=CC(C)(C)C)C(C(C)C)C2)=O)ccc1C 17817,c1(C(N2C(C)CN(C(=O)C(N3CCOCC3)C)CC2)=O)cn2cnnc2cn1 17818,C1(CCNC(c2[nH]cc(C)c2C)=O)CCN(C(=O)C(C)n2ccnc2)CC1(F)F 17819,N1(C(=O)CC=Cc2ccccc2)CCC(F)(C(N2CCC(CO)C2)=O)CC1 17820,C(c1cccs1)=CC(=O)N(CC(CC)NC(=O)CC1CCOC1)C 17821,c1(C(=O)NCC2N(C(C(C=C)OC)=O)CC(F)C2)cc(C)c(C#N)c(C)c1 17822,C=CCC(C(=O)NC(C=C)CO)NC(=O)C=CC1CCCN1C 17823,C1(CNC(CSCC=C)=O)CN(C(C2COCOC2)=O)CCC1C 17824,CN1CCCC12CCN(C(=O)C(=O)Nc1ccc(C(F)(F)F)cn1)CC2 17825,C=C(C)C(C)(C)C(=O)NC1CCCC1NC(C1CCC(C#N)C1)=O 17826,CC1CC(NC(=O)Nc2nccc(-n3cccn3)n2)CCN1C 17827,N#CC1(C(=O)O)CC(Nc2ccc(C(CF)OCc3ccccc3)cc2)C1 17828,N1(C(COCCCCC)=O)CCC(CC)C1CNC(=O)Cn1cnc(C#N)n1 17829,C1(C(=O)NC2(CNC(c3ccc([N+](=O)[O-])s3)=O)CCOC2)Cc2nccnc2C1 17830,c1(NC(=O)C(C)(CO)CO)ccc(C(F)(F)F)cc1O.C12(CC)CN(C1)C2=O 17831,C1(NC(c2c(CC)c[nH]n2)=O)CN(C(=O)CC2CCCC2(F)F)C2CCCCC12 17832,c1(CC)cc(F)ccc1C(N1CCCC1C(N1CCC(C)C(C(=O)OC)C1)=O)=O 17833,C(=O)(C1CCc2c[nH]nc21)NC1CCC(C(N(c2cccc(O)c2)C)=O)CC1 17834,C1(C(N2CC(n3cc(C(C)O)nn3)C2)=O)CCC(S(C)(=O)=O)C1 17835,CCC(CCOC)NC(C1CC(NC(=O)C(F)OC(F)(F)F)C1)=O 17836,Cc1nc(Br)oc1C(=O)N(C(C)CNC(c1cc(C(C)(C)C)n[nH]1)=O)C 17837,c1(CC=CC(=O)N(C(CNC(C=CC(CC)=CC)=O)C)C)ccccn1 17838,C1(C(=O)NC2C(NC(Cc3ccc(OC)cc3C)=O)C2)OCCOC12CCC2 17839,N1(C(c2n(C(C)C)ccn2)=O)C2CCCC1CN(C(C1CCCS1)=O)C2 17840,CC1C(NC(C2(N(C)C)CC2)=O)CCN1C(=O)CC(F)(F)F 17841,N1(C(CC(CC)OC)=O)CCC(C2(O)CN(C(C3(CC)CCC(=O)N3)=O)C2)CC1 17842,N1(C(c2ccc(C)nc2C)=O)CCC2C(CCN2Cc2cc(Br)cc(Cl)c2O)C1 17843,CCC(C)CC(=O)C(=O)N1CCOC(C(=O)NCC2(C)C=CCCC2)C1 17844,N1(C(c2c(F)cccc2F)=O)CCCC2(C1)CN(Cc1cncnc1)CCO2 17845,Cc1csc(C(=O)NC(C2CCCC2)CNC(=O)C(F)F)c1Cl 17846,c1(C(=O)NC(CC=C)CNC(=O)Cc2csc(=N)[nH]2)nn(C)c(Cl)c1Cl 17847,C1(C(N(CCN(CC=C)C)CC)=O)C=CCN(C(=O)C(C)(O)C2CCC2)C1 17848,C1(C)(C(=O)OC)CCN(C(C2CCC2NC(=O)CC(C2CC2)C2CC2)=O)C1 17849,C1(NC(c2ccc(Cl)nc2Cl)=O)CCN(c2ncncc2I)CC1F 17850,O=C1NC2CCC1CN(C(=O)CC1C3CCC(C3)N1C(C1CCS1(=O)=O)=O)C2 17851,C1(O)(C(=O)NC2C(NC(=O)CCc3cccnc3F)CC2)CCCCCC1 17852,N1(C(c2c(CC)non2)=O)CCC(CNC(C2(C#N)CC3CC3C2)=O)C(C)C1 17853,C1(CNC(CN(C)C)=O)(CO)CN(C(=O)COCCNC)C1.c1(O)cccnc1 17854,c1(C(N2CCCC(c3ncc[nH]3)C2)=O)cccc(-n2cnnn2)c1 17855,c1(C(=O)NCCC(=O)OC)cnc2c(c1)CCN(Cc1cc(Cl)c(Cl)cc1F)C2 17856,c1(C(=O)NC2CN(C(C(CSC)(C)C)=O)CC23CC3)ccn2ccnc2n1 17857,c1(OC)ccc2c(c1)CCC2C(=O)NC(c1ccccc1C)CF 17858,C#Cc1ccc(F)cc1C(=O)NCCC(C)(C)NC(c1cn(C(F)F)c(C)n1)=O 17859,N1(C(CC)=O)CCCC(C(=O)NC(CNC(c2ocnc2C(F)F)=O)C2CC2)C1 17860,N(C1CC2(CC2)Oc2c(F)cccc21)C(C1(F)CC=CCC1)=O 17861,C12(CNC(CCC=C)=O)CC1CN(C(c1cc(C(=O)OC)sn1)=O)C2 17862,c1(SC(C)C)cccc(C(=O)Nc2ccc(C(=O)N(C)C)nc2)c1.C(C=O)N 17863,Cc1cc(C)c(C(N2CCC(NC(c3cn(C(C)(C)C)nc3Br)=O)C2)=O)cn1 17864,CCCCCC(=O)N1CCC(CNC(=O)COc2ccc(F)cc2)(COC)C1 17865,N1(c2nnc(CCC)o2)CCCC(C(N2CCC(C(=O)O)CC2)=O)CC1 17866,C1(NC(Cc2ccc(C(C)=O)s2)=O)CN(C(c2ccccc2)=O)CC1C 17867,CC#CCCCC(=O)NCC1(F)CC(NC(=O)Cc2noc(C)c2C#N)C1 17868,N1(C(C2C(C(C)C)C2)=O)CCC(C)(CCNC(c2cc(Cl)n(C)n2)=O)C1 17869,C1(NC(C2(C(C)=O)CC2)=O)CCC(C)(C)CC1CNC(=O)C(C)(C)c1ccns1 17870,C1(CC(=O)NC)CN(C(c2cc(C(N)=O)[nH]n2)=O)CCN1C(=O)C(C)C(C)O 17871,N1(C(CC(CC#C)NC(C2CC(=O)C23CCC3)=O)=O)CC2(C1)OC(=O)NC2C 17872,C1(CC)CCCN(C(=O)C(n2ccnc2C)C)C1C(=O)NC1COCC(C)(C)C1 17873,Cc1cc(C(N2CCC3(C2)CN(C(=O)C(C)C(F)(F)F)C3)=O)c(Br)c(C)c1 17874,c1(NC(C2N(C(CCc3ccc(C)cn3)=O)CC2)=O)ncc([N+](=O)[O-])cc1I 17875,c1(C(=O)NC(C(C)NC(C2CCOCC2(C)C)=O)CO)cc2cc(Cl)cnc2[nH]1 17876,c1(Cn2cc(COC)nn2)cc2cc(C)cc(C)c2[nH]1 17877,CC1CN(C)C(C)CN1C(C1CC12CN(C(=O)C=Cc1ccc(F)cc1)C2)=O 17878,c1(C(=O)NCCC(CNC(C2N(C)CC(O)CC2)=O)O)cc2ccncc2o1 17879,Cc1ccc(C(=O)NCCCC(O)C(=O)N(c2csnc2C)C)c(O)c1 17880,c1(C(=O)NC2CCC(C)(CNC(C3C(C)=CCS3)=O)C2)cc(C)nc2onc(C)c12 17881,c1(C(=O)NC2C(C(=O)NOC3CN4CCC3C4)COCC2)ncnc(O)c1F 17882,c1(C(N(CCC)CCNC(c2c[nH]cc2Br)=O)=O)ccc(CF)cc1 17883,C1(CC(=O)NCC2C(NC(COCC(C)C)=O)C2)CC(OC(C)(C)C)C1 17884,c1(OC(C)C)ccc(CC(=O)NCC2(CSC)CC2(F)F)cc1.C12(CC1)C(=O)N2 17885,c1(C(=O)NCC2N(C(c3cncc(C#C)c3)=O)CC2)[nH]cc2c1CCCC2 17886,c1(C(N2C(CN(CCCC3CCOC3)C)CCCC2)=O)cc2sccc2[nH]1 17887,N1(C(C2C(C(C)(C)C)CC2)=O)CCC(O)(Cn2cc(C3(CO)CC3)nn2)C1 17888,C1(C)(C(N(CC(C)(C)NC(C(c2ccc(Cl)s2)C)=O)C)=O)CC2CC2C1 17889,CCCC(C(=O)OC)N1CC2C(C(=O)NCCCOC)C2C1 17890,c1(CC(=O)NC2C(SC)CN(C(c3cnc(O)o3)=O)C2)ccc2c(c1)NC(=O)C2 17891,N1(C(CCSC)=O)CCN(C(C2(CO)CCC2)=O)CC1c1ccccc1Cl 17892,c1(OC)nc(Cl)ccc1C(=O)NC(C)CC1CN(C(=O)C(c2ccc(Cl)s2)C)C1 17893,c1(N2CCC(CC)CC2)[nH]c(=NC(CCO)CC(C)(C)C)nc2c1ncn2CC 17894,C1(O)(C(C(=O)N(CC=C)C2CC2)NC(=O)CC2(N(C)C)CCC2)CCCCC1 17895,C#CCC(C(=O)NC(c1cccc(Cl)c1)CNC(=O)CSc1nncn1C)C1CC1 17896,c1(N(C(CNC(C(C(C)C)OC)=O)C)C)cc2nnc(-c3ccccc3)n2cn1 17897,C(=O)(C1Cc2c(Cl)cccc21)N1CC(C(C)NC(c2ccc([N+](=O)[O-])n2C)=O)C1 17898,c1(NC(C=CC2N(C(CN3CCC(OC)C3)=O)CCC2)=O)ccc(Cl)nc1C 17899,N1(C(C(C=C)(C)C)=O)CC(NC(c2cc(C(C)C)on2)=O)CC2(CCC2)C1 17900,N1(C(c2n(CC)ncc2)=O)CCOC(C)(CNC(c2nn(C)nc2Br)=O)C1 17901,C1(CNC(=O)NC(C)COC(F)(F)F)Cc2ccc(F)cc2C1 17902,C12(C(N3CCC4(NC(=O)C=Cc5ccco5)C(C3)C4)=O)CCC(F)(CC1)CC2 17903,Cc1ccc(-n2cc3c(n2)C(=O)N3)cc1.C(CCC(=O)O)NC(=O)C(C)C 17904,N1(C(C2N(N=O)CCC2)=O)CC(F)(F)CC1CNC(=O)C=CC=C(Cl)Cl 17905,C1(C(=O)NCC=CCC(N2CCC(C)C2)=O)C2C3CCC(C3)C12 17906,Cc1ccc(Cl)c(C(=O)NCC2CCCCN2C(=O)Cc2cc(C)ccc2C)c1 17907,c1(CC(=O)N(C(CNC(C=C(CC)C)=O)C)CC)ccc(NC(N)=O)cc1 17908,c1(CC(N2CCC(NC(c3c(CC)c[nH]c3)=O)(CF)C2)=O)cc2ccccc2o1 17909,c1(C(=O)NCC2N(C(C(C=C)OC)=O)CC(OC)C2)c[nH]c(=NCC)s1 17910,N1(C(C(CC)SC)=O)C(C(N2CCC(C(=O)OC)C2(C)C)=O)CCC12CC2 17911,Cc1ccncc1-c1cn(CC(N2CCCC(COc3ccccc3)C2)=O)nn1 17912,Cn1c(C(N2CCCC3C(=O)NCC23)=O)c(Cl)c2ccccc12 17913,N1(C(CC(=C)C)=O)CC2CC(NC(c3cc(OC)cs3)=O)C(C2)C1 17914,N1(C(C(C)=C2CCCC2)=O)CC(NC(=O)Cc2sc(S)nc2C)C2CC12 17915,c1(C(=O)NCCCCCNC(c2cncc(N)n2)=O)ccc(S(N)(=O)=O)cc1Cl 17916,c1(CC)cc(C(=O)NCCNC(=O)COCc2cccc(C)c2)nn1C 17917,C1(C(=O)NC(c2cnc(C)s2)C)CCC(C)(C)N(C(=O)CC2=CCCCC2)C1 17918,c1(C(=O)NCC(C)CNC(C2(CCF)CC2)=O)ncnn1C1CCOCC1 17919,N1(C(C=Cc2nc(C)sc2)=O)CCCCC1C1CCCN1C(=O)C(O)C1CCC1 17920,n1(C(C)C)cc(C(=O)N(C)CCN(C)C(c2cc(F)n[nH]2)=O)c(Br)n1 17921,C(=O)C(C)(C)C(=O)c1ccccc1.C=CCCOCCN(C(=O)CN(C)C)CC 17922,c1(C(=O)NCC(C)NC(c2n(C(C)C)ccc2)=O)cc(Cl)ccc1F 17923,C1(O)(CNC(C2C(COC)CC2)=O)CCN(C(C2C=CCS2)=O)CC1 17924,c1(C(N(CC(C)NC(c2cn(C3CCC3O)nn2)=O)C)=O)cc2ccsc2s1 17925,C1(C#N)(C(=O)O)CC2CCC1CC2NCc1cnns1 17926,C1(C(=O)NC2(C(COC)O)CC2)CC2CC1CN(C(=O)Cn1ccnc1C)C2 17927,CC(C(=O)NCC1CCN(C(=O)Cc2cncs2)CC1CO)C(F)(F)C(F)F 17928,c1(C(=O)NCC(CO)NC(c2cnc(O)c(F)c2)=O)cc2cn[nH]c2cn1 17929,C1(NC(C2N(CC#C)CCC2)=O)CC2(CCCN(C(=O)C(F)C(C)(C)O)C2)C1 17930,C=C1CC(C(F)(F)F)(C(=O)Nc2cc(C(=O)NCCC(C)O)[nH]n2)C1 17931,c1(C(N2CCC(OCC(=O)NCCCCN=[N+]=[N-])C2)=O)ccc(O)cc1F 17932,CNS(=O)(=O)NCC(=O)NCCOCCNC(=O)Cc1conc1C 17933,C1(C(N2CCCC2)CC)CCCN(c2cccc(C(N)=O)n2)C1 17934,N1(C(CC(C2CCC2)NC(=O)OC(C)(C)C)=O)CC(O)CC1(C)CO 17935,Cn1cccc(-c2cncc(C(=O)Nc3ccc(CO)c(F)c3)n2)c1=O 17936,C1(O)(C(C)NC(C2CN(C)C(=O)N2)=O)CCN(C(c2scnc2C(F)F)=O)CC1 17937,n1(CC(=O)Nc2nc(C3CCCC3)cs2)cc(Br)c(O)nc1=O 17938,C(c1ccc(F)cc1)=C(C)C(N1CCC(C)(NC(=O)CN2CCCCS2(=O)=O)C1)=O 17939,c1(-c2cn(CC(CN)OC)nn2)ccc(C(F)(F)F)cc1Cl 17940,C(=O)(C(C)CC(F)F)NC(CN(C(c1ccc(C(C)C)cn1)=O)CC)C 17941,N(C(=NCCCN1CC(C)(C)OC1=O)N1CCN(C2CC2)C(=O)C1)C(C=C)C 17942,c1(C(N)=O)ccc(C(=O)NCc2cn(CCNC(N)=O)nn2)cc1 17943,C=CC(C)(C)CC(=O)N1CCC(CO)(NC(=O)C(CC2CCCCC2)CCC)C1 17944,Cc1ccn(C)c1C(N1CC(O)(CN(C(=O)CCc2ccnc(Cl)c2)C)C1)=O 17945,C(=O)(C1=CCC2CCC1N2C(=O)C(Cl)Cl)NC(c1ccco1)C 17946,c1(OC)cc(Br)ccc1C(c1nnnn1Cc1cccc(OC)c1)NCC(N)=O 17947,c1(OC)cc(CC(=O)NCC2CCCN2C(=O)Cc2cc(C)[nH]n2)c(F)cc1O 17948,C1(NC(CCCC#C)=O)CCCC12CN(C(c1cccnc1OCCOC)=O)C2 17949,C1(NC(CCOCC#C)=O)CC2(C1)CC2NC(c1cnn(CCN(C)C)c1)=O 17950,C1(CNC2CC(CNC(C3(OC)CCC3)=O)C2)CCCC1C 17951,c1(C(=O)NCC2C(NC(CC(C=C)C)=O)CCCC2)ccc(C(F)(F)F)c(N)c1 17952,C1(NC(CCC2(C)CC2(F)F)=O)CN(C(=O)Cc2cccc(O)c2)CC1F 17953,c1(-c2scc(C)n2)ccc(C(=O)N(C2CN(C(C3(C)CCCN3C)=O)C2)C)cc1 17954,c1(C(N2CCC(NC(CCC(CC)C)=O)(COC)C2)=O)cnc2ccccn12 17955,N1(C(=O)C=CC2CC2)CCC(C2CC(NC(C34CCC(CC3)CC4)=O)C2)C1 17956,c1(C(=O)NCC(c2ccc(C)cc2)NC(C2(C3CC3)CC2)=O)cnc2n1CCS2 17957,CC1CN(C(c2cn(CCNC(=O)C(C)(Cl)Cl)cn2)=O)CC1(C)CO 17958,C(=O)(CCCC(F)(F)CO)N1CCC(N(C(c2c[nH]cc(C)c2=O)=O)CCO)CC1 17959,N1(C(c2ccc(Br)cn2)=O)CCC(F)C(NCc2cc(O)cc(F)c2)C1 17960,N1(C(C2C(C)CCO2)=O)CCC(F)(C(N2CC(C3CCCO3)C2)=O)C1 17961,N1(C(C(C)=C2CC2)=O)CCC(O)C(NC(c2cc3n(c2)CCC3)=O)C1 17962,CC1CC(C(=O)NC(C)CNC(=O)C=Cc2ccc(=O)n(CCO)c2)CC(=O)N1 17963,N1(C(CC2CC(=C)C2)=O)CC(NC(c2cncc(C3CCCCC3)c2)=O)C(C)C1 17964,C1(C(C)NC(=O)Cc2cnc[nH]2)CCCCN1C(c1ccc(C2CCC2)cc1)=O 17965,c1(C(N(C2CC3CC3C2)C2(C)CC2)=O)ccccc1Cn1cncn1 17966,CC1(C)C(CC(=O)NCc2nc(C3CC3)cs2)CCN1C(=O)CC1(C#N)CC1 17967,C1(C(=O)NC2C(NC(c3ccc(C)o3)=O)CCC2)CCCN(C(=O)C(C)(C)C)C1 17968,C1(C(N2CC(C#N)C2)=O)CC(OC)CCN1C(C1CC2CCC(C1)C2)=O 17969,c1(SCCN(C)C(C2(F)CCN(C(=O)OC(C)(C)C)C2)=O)ccc(Cl)c([N+](=O)[O-])c1 17970,N1(C(CC2CC(CC)C2)=O)CC(C)N(C(=O)CN2CSCCSC2)CC1C 17971,c1(-c2cncc(OC)c2)ccc(CN2CCCC2(C)CO)c(C)c1 17972,C(=O)(C1(C)CCn2c(C)nnc21)N1CC(NC(c2ncc(C)cn2)=O)C(O)CC1 17973,c1(C(=O)NC2CCCC3CN(C(CCSC)=O)CC32)cccc(S(N)(=O)=O)c1C 17974,N1(C(c2ccc(C#C)c(Cl)c2)=O)CC(NC(C)=O)C2(CCOCC2)C1 17975,c1(NC(C2(C)CCN(C(C(C)(C)CCl)=O)CC2)=O)c(F)cccc1C#N 17976,Cc1cccc(C(O)C(=O)NC(C)CN(C(=O)CC2CC3C=CC2CC3)C)c1F 17977,C1(NC(c2ccc(N(C)C)cn2)=O)CC2CCC1C(NC(=O)C1=CCCOC1)C2 17978,C1(C(N2C(C(N(C3CCCC3(F)F)C)=O)COCC2)=O)CC(=O)NC(=O)C1 17979,c1(C(N2C(CNC(c3ccn(C)c3)=O)CCCCC2)=O)c[nH]c2cc(O)ccc12 17980,N1(C(c2c(CC)nco2)=O)CCC2(C1)CN(C(=O)C(C)NS(=O)(=O)CC)C2 17981,N1(C(c2cc(CC)oc2C)=O)CC(C)N(C(c2cn(C)c(C)cc2=O)=O)CC1C 17982,CCC1=NOC(C(=O)N(C)CC2(NC(c3cnc(CC(C)(C)C)s3)=O)CC2)C1 17983,c1(CNC(CCC(C)NC(C2CCCCCN2C)=O)=O)cccc(C#N)n1 17984,C(=O)(CC1c2ccccc2CCN1S(C)(=O)=O)NCC1N(C(CC=C)=O)CC1 17985,N1(C(C2CCC(CC)CC2)=O)C(CNC(c2cc(Cl)on2)=O)CC2COCC12 17986,N1(C(c2ccc(C)cc2)=O)CC2(CC(NC(c3cnc(N)c(Br)c3)=O)C2)C1 17987,C1(C(=O)OCC)CCN(C(=O)CCP(C)(C)=O)CC1(F)F 17988,N1(C(Cc2ccc(C#C)cc2)=O)CCC2(CC1)CN(C(C1CCCS1)=O)C2C(C)C 17989,N1(C(C(COC)C)=O)CCOC2(CCN(C(C3CC(=O)C3)=O)C2)C1 17990,c1(C(=O)NCCN(C)C(c2cc(C3CC3)ncn2)=O)cccc(C2(F)COC2)c1 17991,CCCC(CCC)CC(=O)NCC1CN(C(c2cnn(CC)c2)=O)CCC1C 17992,n1(CC(=O)N(C(C)CNC(c2nn(C)cc2C(=O)O)=O)C)cnc([N+](=O)[O-])n1 17993,N1(C(C=NOC)=O)CC(NC(=O)CSc2cccc(F)c2)CC2(CCC2)C1 17994,CC1CCCn2cc(C(=O)NCC3CC3NC(C3CN(S(N)(=O)=O)C3)=O)nc21 17995,CCC(O)(C(=O)NCCCCC(C)NC(c1nc(C)cs1)=O)c1ccccc1 17996,N#CC1C2CCC1CN(C(C13CC(CCO1)N(C(=O)C=CC1CCOC1)C3)=O)C2 17997,CN1CC(NC(=O)CCC2CC(NC(C3(C)CCC(=O)N3)=O)C2)C(C)(C)C1 17998,C1(C(N2CCCC(CN(C(=O)CC(C)(C)C)CC)C2)=O)CC12CCOCC2 17999,Cc1cc(Cl)cc(NC(C2CC(F)CN2Cc2ccc(C)c(F)c2)=O)c1O 18000,N1(C(C(C)OC(C)(C)C)=O)CCCN(C(=O)COC2CCCCC2)CC1 18001,c1(C(N(CCCN(C(c2c(C)ccnc2)=O)C)C)=O)c(C)nc(O)nc1S 18002,n1(CC)nc(C(=O)NC2(C3CCCN3C(=O)CCCOCCOC)CC2)c(Br)n1 18003,c1(CC(N2C(CNC(C3(C#N)CCCO3)=O)CC2)=O)cc(F)ccc1Cl 18004,CC(C)CC(O)Cc1cn(CCCC(=O)NCC2CCCN2N=O)nn1 18005,N1(CC)CCN(C(=O)CCC(=O)C(C)(C)C)C(=O)C12CCCC2 18006,N1(C(C(C)OC(C)(C)C)=O)CC2(CNC(=O)Cc3cncnc3O)CC1CCO2 18007,c1(CC(=O)NCCC2(O)CN(C(c3c(C)coc3C)=O)C2)cccc(Cl)c1Cl 18008,C1(CCNC(CCC)=O)CSCCN1C(=O)CCNc1ccccc1C(N)=O 18009,C1(NC(c2conc2C2CCC2)=O)CCCN(C(C2CC=CCC2)=O)C1 18010,c1(C(N2CC(CNC(C3CC(C(C)C)OCC3)=O)C2)=O)cc2nc[nH]c2cn1 18011,C(c1ccc(C)c(C)c1)=CC(=O)NC(CCOC)CNC(=O)C(O)CC1CC1 18012,c1(C(N(CC(C)N(C(C(CCC)CC)=O)C)C)=O)ccc2c(c1)CN(C)CC2 18013,C=CCC(C(=O)NCC1(CN(C)C(C2CCC3CC3CC2)=O)CC1)C(C)C 18014,C(=O)(C(C)(F)C(F)(F)F)NCC(C(C)C)(C)NC(C1CCN(C(N)=O)CC1)=O 18015,Cc1cc(Cl)cc(CNCC2OCCN(C)C2c2ccccc2)c1O 18016,C(C(CC(=O)NC(CNC(c1occc1C)=O)CO)CC(C)C)NC(C)=O 18017,C1(NC(C(C2CCC2)OC)=O)CCCCN(C(=O)CSc2ccccc2Cl)C1 18018,C=C(Cl)CC(C(=O)N1CCC1CO)NC(c1nnn(C)c1C)=O 18019,C(=O)(C(C)(C)C(=O)NC1CCCN(C(c2cscc2Br)=O)CC1)NC 18020,C1(NC(c2c(CC)oc(C)c2)=O)CN(C(c2cocn2)=O)CC12CC2 18021,C(=O)(C1=CCSC1)NCCC(CNC(CC(C)C)=O)O 18022,N1(C(CCN(c2ccncc2)C)=O)CCC2CC1CN2C(c1csc(Cl)c1)=O 18023,C1(CNC(c2c(C)nco2)=O)C(C2CC2)CCN1C(=O)CC1CC12CC2 18024,N1(C(C23CC(C)(C2)OC3(C)C)=O)CCC2CC(NC(c3cscn3)=O)CCC2C1 18025,C1(CN(C(=O)C(N2C(=O)CCC2=O)C)CC)CCN(C(C2CC23CCC3)=O)CC1 18026,C1(NC(CCC#CC)=O)CCSC12CN(C(=O)CCOc1cccc(C)c1)C2 18027,C=CC12CCN(CC1)CC1(C)CN(C1)C2=O.C1(C(=O)OC)CC1C1CCC1 18028,CC1(C)CC(SC(=O)NOCC(C2CCOC2)O)C1 18029,C1(C(=O)NCC2N(C(COc3cn(C)nc3)=O)CCC2)C2CCC(F)C12 18030,N1(CC(N2C(C)CC(NC(c3cc(CN(C)C)on3)=O)C2)=O)CCc2ccccc21 18031,C12(NC(c3n(C)ccc3)=O)CN(C(C3CCOCC3)=O)CC1CS(=O)(=O)C2 18032,N1(C(c2ccc(OCC)cc2)=O)CCCC(F)(CNC(=O)CC2CC3(CC3)C2)C1 18033,Cc1ccc(NC(C23CC(C(=O)NCC4(O)CCC4)(C2)C3)=O)cc1C(F)F 18034,CCCCCCCC(=O)NCC(C)(O)CNC(C1CNC(=O)CC1(C)C)=O 18035,c1(C(=O)NC(C(=O)NC(c2cc[nH]n2)C)CC2CC2)cccc(F)c1N 18036,c1(C(=O)NCC2C(C)CCCN2C(C2(N(C)C)CCC2)=O)cccc2ccnn12 18037,Cc1oc2ccccc2c1C(N1CC(NC(C2CCCCN2C)=O)CC1(C)C)=O 18038,C1(NC(=O)Cc2cncnc2)CN(C(=O)CCF)CCC1c1ccc(F)cc1 18039,c1(CCC(=O)N(CC(C)O)CCNC(C(C)NC(C)=O)=O)ccc(Br)nc1 18040,C1(C(=O)Nc2cccc(C(F)F)n2)CC(O)CCN1C(c1cccc(Cl)c1Cl)=O 18041,Cc1ccc(OCC(=O)NCCOCCNC(C2CNC(=O)CC2C)=O)c(C)c1 18042,CC1CN(C(=O)C=CI)CC2(CCN(C(c3cc(O)nc(O)c3)=O)C2)O1 18043,C(=O)(CC(C)C(F)F)N1C(C(=O)NCCc2c(C)cncc2)C2CC2C1 18044,Cc1ccc(Cc2nc(-c3ccc(Br)cn3)nn2CC(N)=O)c(C)c1 18045,C1(NC(CC(=C)I)=O)CC(C)CN(C(c2ccc(C)nc2)=O)C1 18046,c1(-c2cn(C3CCN(C(C4CCCO4)=O)C3)nn2)ccc(Cl)c(Cl)c1 18047,CC(C)(C)CCC(F)C(=O)NC1CC(NC(c2cn3ccnc3cn2)=O)CC1O 18048,C1(N(C)C(=O)NCCc2nc(-c3ccccc3)no2)CCCCC1C(F)(F)F 18049,C1(CC(=O)OCC)CN(C(=O)C(C)c2cc[nH]n2)CC12CC2.C(CCO)N(CC)CC.CCO.N 18050,CCC(C)(CO)C(=O)NCC(F)CNC(=O)CCN1CCOC1=O 18051,N1(C(COC(CC)(C)C)=O)CC(NC(=O)CC23CCCC2C3)C2CCCC2C1 18052,C1(C(=O)NCC(CC(=C)C)N)CCC2(CCCC2)C1 18053,C1(O)(C(=O)NC2CCC(NC(C3=NOC(C)C3)=O)CC2)CCCC(C)(C)CC1 18054,Cc1cc(C)c(CN2CCC(=CC(=O)NCc3cnc(N(C)C)nc3)CC2)c(C)c1 18055,C1(CNC(C2(CC#C)CC=CCC2)=O)N(C(=O)Cc2cnsc2)CCC1(C)C 18056,C1(C(C)(C)C)CCC(n2nc(C3CCC(C(C)(C)C)CC3)nc2CCCF)CC1 18057,c1(C(N(C)CC2N(C(COCCC#C)=O)CC(F)C2)=O)cc2c(C)cccn2c1 18058,c1(C(C)=O)csc(C(=O)NCC2(O)CN(C(C3CC3(C)C)=O)C2)c1 18059,N1(C(CC(C)OC)=O)CC(NC(=O)CNC(=O)CN(C)C)C2CCCC12 18060,N1(C(C(=O)NC(C)C)=O)CC(NC(=O)C(c2ccccc2Cl)O)CC12CCC2 18061,C1(NC(CCC)=O)CC(F)(F)CC1NC(c1ccc(SCC(C)C)o1)=O 18062,c1(N(C)CC2CCCN2C(=O)CC2NC(=O)NC2=O)cc(C(F)F)nc(Cl)n1 18063,c1(C(=O)NCC2CCCC2NC(C2(CF)COC2)=O)cc(Cl)cnn1 18064,C1(NC(Cn2c(C)cnc2)=O)CN(C(C2CN(S(C)(=O)=O)C2)=O)CC1C 18065,S(=O)(=O)(c1ccc(F)cc1)NCCC(=O)N(c1ccccc1)CC(C)C 18066,c1(NC(C2C(CC)N(C(c3cc(O)nc(O)n3)=O)CC2)=O)cc(C)cnc1C 18067,c1(C(=O)NC(CNC(CC(C=C)C)=O)CCOC)cc2cccnc2o1 18068,C1(NC(COCC(N2CCCC2)C)=O)CC2CC1N(C(c1cnnc(O)c1)=O)C2 18069,c1(NC(c2ccc(C(=O)NC34CC(C5CC5)(C3)C4)cc2Cl)=O)cccc(Br)c1Cl 18070,C(=O)(C(C)(C)C(C)NC(C1CCNC1=O)=O)NC1(C#C)CCOC1 18071,C(=O)(CC(C(F)F)NC(=O)CC1CCSC1)NCCCCC 18072,C(=O)(C1=CCCCO1)N1CC(NC(c2c(C)oc(-c3cccs3)n2)=O)C2C1C2 18073,CC1(C)CC(C(O)CNC(=O)CNC(c2cccs2)=O)C1 18074,C1(C(=O)NCCCC(C)NC(COCCCC)=O)CN(C(C)C)CCO1 18075,Cc1nc2c(Cl)cccc2cc1C(N1CCCN(C(=O)CC2CCC2)CCC1)=O 18076,c1(C(N2CC(O)(CCNC(c3c(CC)ocn3)=O)C2)=O)c(C)cc(Cl)nc1N 18077,C1(NC(CC2(NC(c3nccc(CC)c3)=O)CCCCC2)=O)CCCCC1(C)O 18078,C1(NC(C2CCCC2)=O)CCOC12CCN(C(C1COC3COCC13)=O)CC2 18079,c1(C(=O)NCC(CNC(C(C=C)O)=O)CO)ccc2c(c1)OCCC2 18080,C1(CNC(C2CCN(C3CC3)CC2)=O)CC2(CC2)CN1C(=O)C1=NOCC1 18081,N1(C(C2CC(=O)NC2)=O)CCOCC(F)(CNC(C2CC2c2ccsc2)=O)C1 18082,c1(C(=O)NC(C(C)NC(CCN(C(CCC)C)C)=O)C)cc(C)nc(O)n1 18083,c1(OCC)ccc(C(=O)NC2CCC2NC(=O)CSc2nncn2C2CC2)cn1 18084,N1(C(C(=O)Nc2c(C)noc2C2CC2)=O)CCC2(CCOC2=O)C1 18085,CON1CCC(CC(=O)NC23CCC(C2)N(C(c2cc(Cl)ccn2)=O)C3)CC1 18086,N1(C(c2cccc(C(C)C)n2)C(=O)NC(CC)C)CC(OC)CC(O)C1 18087,C(=O)(C1CCC(=O)c2cccn21)N1CCN(C(C2C(C)C2C)=O)C(CO)C1 18088,N1(C(C(=O)N(CCOC)C(C)C)=O)CCCCCC(NC(C2CC23CC3)=O)C1 18089,N(C(=NCCCP(C)(C)=O)NCCSC)CC(c1cc(OC)cc(OC)c1)(C)C 18090,C1(CNC(C2(OC)CCSCC2)=O)C2CCCC1N(C(c1nc(=O)n(C)[nH]1)=O)C2 18091,CN1CCC(C2(C(=O)OCC(C)(C)CC(F)(F)F)CC2)CC1 18092,CC1CCC(CNC(=O)Cc2ccno2)CN1C(c1cccc(C(F)F)c1F)=O 18093,N1(C(C(Cc2cc[nH]n2)NC(C2CN(C)C(=O)C2)=O)=O)CCN(C)C2(CCC2)C1 18094,c1(CC(=O)NCCN(C(=O)C2=CCOC2)CCOC)ccc(C#N)cc1F 18095,CCC(C(C)CN(C)C)NC(=O)C(Cc1cc[nH]n1)NC(=O)CCc1ccco1 18096,c1(C(=O)N(c2ncncc2I)CC2(F)CNC2)ccc(Cl)c(F)c1 18097,C(=O)(C(O)P(C)(C)=O)N1CCCC(NC(CS(N2CCC(C)CC2)(=O)=O)=O)C1 18098,c1(OC)c(C(=O)NC(C)CCCCNC(c2c(C)ncn2C)=O)cc(F)cc1F 18099,CC1(C)CC(NC(C2(C(N)=O)CC2)=O)Cc2ccsc21 18100,C1(CNC(C(CC)N(C)C(c2cn(C3CC3)cn2)=O)=O)CCCN(CC)C1 18101,N1(C(C2CC(C(C)C)C2)=O)CCCC(C)(CNC(C2(C)CCCCO2)=O)C1 18102,c1(SCCNC(N2C(c3scc(C(=O)OCC)n3)CCC2)=O)cccc(Cl)c1C 18103,c1(C(N2CC(NC(c3c(NC)nccc3)=O)C2)=O)ccc(-n2ccnc2)cc1C 18104,N1(C(CCc2nc(C)sc2)=O)CC2(CNC(C3CCS3(=O)=O)=O)CC1CO2 18105,O=C(C1=Cc2cc(Cl)ccc2OC1)NC1C2CC1N(C(=O)COC(F)(F)F)C2 18106,CC(C)C(C(=O)NC(C1(C)CN(C(=O)C(=O)NCC2CC2)C(C)(C)C1)C)C(C)C 18107,C(=O)(C(C)CC(F)F)N1CCC(N(C(=O)C=CC2CCCN2C)CC#C)CC1 18108,C1(C(=O)NCCc2cc(C(=O)NC(C)CC3CCCCC3)no2)C2CCC(=O)C12 18109,N1(C(CC=C=C)=O)CCC2(CCCN(C(=O)C(C3CCOCC3)F)C2)CC1 18110,C(C(C)(O)C(C)CC)NC(CC1CCC(NC(C2(CCC)CC(=O)C2)=O)CC1)=O 18111,Cc1ncsc1C(=O)N(CC(O)CNC(=O)C=CCCc1ccccc1)C(C)C 18112,C1(C(C)N)CCN(C(=O)C(=O)N(Cc2ccccc2)CC2CCOCC2)C1 18113,c1(C(N2CC(CCCCNC(CCC=C)=O)C2)=O)nnn(COCC)c1N 18114,c1(C(=O)NC(CC(C)NC(CNC(=O)NC)=O)C)cc(C(C)C)ccc1F 18115,CN1C2CC(O)C1CC(CO)(N)C2.c1(C)cnn(CC(F)(F)F)n1 18116,N1(C(COCC(=C)C)=O)CC=CCC1C(=O)NC1CC(C)OC1=O 18117,C(=O)(CC(O)C(C)CC)NC1(CC=C)CCN(C(C2(Cl)CC2)=O)CC1 18118,C(=O)(CC(CNC(=O)C(C(C)C)NC(=O)NC)c1ccc(Cl)cc1)OC 18119,n1(CC)nncc1C(N1CCC(NC(=O)CCCn2cccn2)C1)=O 18120,c1(C(N2CCC(NC(CCc3cnn(C)n3)=O)C2)=O)c(C2CCC2)cnn1C 18121,C1(S(C)(=O)=O)(CNC(c2c(SC)cc(Br)cc2)c2nnnn2C(C)C)CCCC1 18122,OCCCCCN=C(NCC1CCCCO1)N1CCC(c2ccncn2)CC1 18123,N(C(=NCCC)NN(C1C(c2cccc(OC)c2)C1)C1CC1)CC1CCCO1 18124,c1(CC)ccc(NC(=O)Cn2nc(C(F)(F)F)cc2C)nc1 18125,c1(CC)nc(C(=O)N(CC(N2C(CO)CC2C)=O)CC2CC2)co1 18126,N1(C(c2c(COC)cco2)=O)CC2CC1CN2C(c1cc(C(C)C)on1)=O 18127,CC1CN(C(C2CCCC2CNC(C2CC(O)CN2C)=O)=O)CCS1 18128,Cc1nc(Cl)ccc1CC(N1CC(OC2CCN(C(=O)C(C)C3CC3)CC2)C1)=O 18129,c1(C(=O)NCC(CN(C(C2CN(C)C(=O)N2)=O)CC)(C)C)cc2[nH]ccc2s1 18130,C1(CNC(c2c(C)coc2C)=O)CC(C)(C)CCC1NC(=O)CC1CCOCC1 18131,c1(C(=O)NCC2CCC(C)CN2C(=O)C2=COCCO2)cccc([N+](=O)[O-])c1O 18132,C1(NC(C(CC)(C)C)=O)CC2CN(C(=O)C=Cc3ccn(C)c3)CC2C1 18133,C1(NC(c2ccc(CC)[nH]2)=O)CCCC(CNC(c2cn(C3CC3)nn2)=O)C1 18134,N1(C(CSCCOC)=O)CC=C(C(=O)NC2(CO)CCOC2)C1 18135,C(C(C)(C)CN(C)C(c1ccc(CSCC(C)C)o1)=O)NC(CCSC)=O 18136,C1(C(=O)NC2CC(N(C(c3ncn(CC)c3)=O)C)C2)CC(C(C)C)=NO1 18137,c1(C(=O)NCc2ccnc(-n3cccn3)c2)cc(F)c2c(c1)OCCO2 18138,O=S(=O)(c1[nH]c(=NCC(O)c2ccncc2)ccc1Br)NC1CC2(CCC2)C1O 18139,N1(C(C(C(C)C)(C)C)=O)CC2CCOCC2(NC(=O)COc2ccc(Cl)nc2)C1 18140,C(=O)(CCCC(C)(C)C)N(C1CCN(CCC2CCCCO2)CC1)CCC 18141,C1(NC(c2ccc(OCCCOC)cc2)C)CCCC(C)(C)C1 18142,c1(C(=O)NC(CCC)CNC(c2cnc(C3CC3)s2)=O)cncc(Cl)c1 18143,C1(NC(C=C2CCC(C)CC2)=O)CCC(C)(CNC(=O)Cc2[nH]cnc2C)CC1 18144,N1(C(c2nccc(C(F)F)n2)=O)CCCCC2(CCN(C(C3CC3(Cl)Cl)=O)C2)C1 18145,c1(C(N2CCC(NC(C(C)OC3CCOC3)=O)(CF)C2)=O)nnn2c1CCCC2 18146,CCC(C)(CCC(C)C)C(=O)N1CC(NC(=O)CCc2cnn(C)n2)C2(CC2)C1 18147,c1(C(=O)NC(C(C)C)C(C)NC(=O)COC2(C)CCC2)cnc(O)nc1O 18148,C1(CC(=O)NCC(CSC)CC(=O)O)CCC2(CCN(C(=O)OC(C)(C)C)C2)C1 18149,N1(C(CCCCCNC(=O)C=Cc2ccc[nH]2)=O)CCCC2CCCC12 18150,CC1(C)CC(C(=O)NC2CC2NC(c2cnc(-c3cccs3)s2)=O)=NO1 18151,c1(C(=O)NC(CC)CN(C(=O)C(C)Sc2nncn2C)C)c(C)nc2sccn12 18152,c1(OC)ccc(CC(N2CCC(NC(C3(O)CCSCC3)=O)C(O)C2)=O)cc1Cl 18153,N1(C(c2cc(CNC(COCCCCC)=O)[nH]n2)=O)CCCC(C)C1CO 18154,O=C(NOCCc1ccccc1)C(=O)NC1(C(=O)O)CCOCC1 18155,CCCC(CC)CCC(=O)N1CCC(CCCNC(C2CCS2(=O)=O)=O)CC1 18156,CN1CC2CN(C(C3CCCN(C(c4cc(Br)c[nH]4)=O)C3)=O)CC2C1 18157,C1(NC(=O)C(=Cc2c[nH]cn2)F)CCCN(C(C2CC3(C2)CC3F)=O)C1 18158,c1(N2C3(CN(C(c4c(OC)ccs4)=O)C3)CCC2)ccnc(S(=O)(=O)C(C)C)n1 18159,Cc1cc(C(=O)OCc2cnoc2C2CC2)ccc1Br 18160,C1(c2nc(C(F)(F)F)no2)(CC=C)CCN(C(n2cnnn2)=O)CC1 18161,N1(C(Cc2nnc(C)o2)=O)CCC(CNC(=O)Cc2cnsc2)C12CCC2 18162,N1(C(c2cc(F)cc(Br)c2F)=O)CCN(Cc2csc([N+](=O)[O-])c2)CC12CC2 18163,C1(NC(c2[nH]cc3c2CCCC3)=O)COC2(C1)CN(C(=O)CO)C2 18164,N1(C(c2n(C)c(O)nc2)=O)CC(NC(C2CC2c2ccc(Cl)s2)=O)CCC(O)C1 18165,CCC(CCCC(=O)NOCc1ccccc1)NC(C1CC2(CC2)C1)=O 18166,Cc1csc2ncc(C(=O)NCC3CCCN(C(C4CNC(=O)C4)=O)C3)c(=O)n12 18167,C1(NC(C2C(C)(C(F)F)C2)=O)CCCCC1CNC(=O)Cc1ccon1 18168,c1(CCC(N2CC3(CN(Cc4cnc(C)[nH]4)C3)C2)=O)c[nH]c2ccc(F)cc12 18169,C(CC(=O)NC1(C)CCCC1(C)C)(C(C)OC)NC(CC=CCCCCC)=O 18170,c1(CC)oc(C)cc1C(=O)OCc1ccnn1C(F)(F)F 18171,N1(C(CN(S(CC)(=O)=O)C)=O)CCC2(CC1)CC2CNC(=O)CC(C)CN(C)C 18172,CC1C(=O)N(C)CCN1C(c1nc(-c2ccccc2)n(-c2ccc(Cl)cc2)n1)=O 18173,N1(C(CN2C(C)CCCC2)=O)CCC(C(N2CC(O)C(O)C2)=O)C(C)(C)C1 18174,N#Cc1cc(C(=O)NCC2CCN2C(=O)C(O)CC(N)=O)n2c1CCCC2 18175,C=C(C)CCC(=O)NCCOCCNC(=O)CCCOC1CCCCC1 18176,c1(C(N2CC(C)N(C(=O)CC3CCC4CC4C3)CC2)=O)cc2ncccc2[nH]1 18177,C1(C(=O)NCC(C)(C)NC(Cc2c(C)noc2)=O)CCS(=O)(=O)C1 18178,C1(NC(C(=O)OC)=O)CCC(CCC(=O)NCCOCCN)C1.N1(C(C)=O)CCCC1 18179,C1(CCOC)CN(C(C2CCCN2C)=O)CCN1C(=O)CP(C)(C)=O 18180,N1(C(CCSC)=O)CC2(CCC(NC(C34CCCCC3C4(F)F)=O)CC2)C1 18181,C1(C2CCN(C(c3ccc(Cl)cc3Cl)=O)C2)(NC(c2cc3ccsc3[nH]2)=O)CC1 18182,c1(CC)cc(F)ccc1CC(N1CCC(NC(=O)COC(C)CC)C1(C)C)=O 18183,N1(C(CC=CCCCCC)=O)CCN(C(=O)CN=S(C)(C)=O)CC(C)C1 18184,C(=O)(NNC(=O)C(C)(C)CCCCNC(c1cccnc1)=O)c1c(C)ccs1 18185,n1(CCNC(C(C)C2CCCC2)=O)cc(C(=O)NC2(C)CSC2)cn1 18186,CC1(C)C(C)(C)C1(F)CNC(=O)CNc1cnc(Cl)c(Cl)c1 18187,C1(NC(CC(C)(C)C2CCCCC2)=O)CCN(C(=O)CCCC#N)CC1O 18188,N1(c2ncnc(C)c2Br)CCC(F)(F)C(C(=O)NC2CCCC(O)C2)C1 18189,c1(OC)ccccc1C(=O)C(=O)NC1CC(C)N(C(=O)CCc2cnc[nH]2)C1 18190,C1(C(N(CC(C)(C)NC(=O)CC(F)(F)Cl)C)=O)CCCC1S(C)(=O)=O 18191,c1(CCC(=O)NC2C(NS(CC)(=O)=O)C2)ccc(O)nc1 18192,c1(NC(C2N(C(c3c(C)cnnc3)=O)CC=C2)=O)ncc(Br)c(C)c1[N+](=O)[O-] 18193,N1(C(C(=O)NCc2c(Cl)cccc2Cl)=O)CCC2(CC(=O)NC2=O)C1 18194,c1(CC(=O)NC2C=CCN(C(C(C)Oc3ccccn3)=O)C2)c(Cl)cccc1Cl 18195,N1(C(CC=CC)=O)CCN(C(c2cncc(S(C)(=O)=O)c2)=O)C2CCCCC2C1 18196,C1(C(=O)NCC2C(CNC(Cc3c(C)cnn3C)=O)C2)CC2CC(=O)C1C2 18197,C1(C(N(CC)CC2CCCN2C(=O)CC#N)=O)Cc2cccc(F)c2O1 18198,N1(C(C(C)(C)O)=O)CCC(C(=O)N2CCn3ccnc32)=C(F)C1 18199,C1(CC)CCN(C(=O)CC2CN(C(c3cc(C)[nH]n3)=O)C2)C1CNC(C)=O 18200,c1(CC(=O)NC(CC)CNC(C2(C)C=CCC2)=O)ccc(OC)cc1Br 18201,C1(=O)CC(C)C(=O)N(C)C2(CC2)CC(=O)O1.C(C(CC)n1cccn1)NCC 18202,Cc1cc(Br)cnc1C(c1nnnn1C1COC1)NCCC1CCC(C)(C)C1 18203,CCC(CN(C)C(c1cnsn1)=O)NC(C1CCCO1)=O 18204,S(=O)(=O)(CC(=O)NC1COCC1NC(=O)CSCC1CCCO1)N(CC)CC 18205,Cc1ncc(C=CC(=O)NCC2CCN(C(C3(O)CCOC3)=O)C2)c(O)n1 18206,c1(C(=O)NCC(C2CCOC2)NC(Cc2nc(C)[nH]n2)=O)nc(O)c(C)s1 18207,N1(C(c2cn(C3CCN(C)C3)nn2)=O)CCCC(CN(C(=O)CC(F)F)C)C1 18208,N1(C(C(N2C(=O)CCC2=O)C)=O)CCC2(CC1)CC(NC(=O)CC(C)(C)C1CC1)C2 18209,c1(C(C)C)ncc(Br)c(C(=O)NC2C3CN(C(=O)Cc4[nH]cnc4C)CC23)n1 18210,Cc1cccc2c(C(N3CC(C)CCC3CNC(=O)CC(F)F)=O)nccc12 18211,C=CC1(C(=O)NC2(C(=O)OC)CC2)CCN(C(C2CC=CC2)=O)CC1 18212,C=CCC(CO)NC(=O)COCCNC(C1CC12CC2)=O 18213,C1(NC(C(C)Oc2cccnc2)=O)CC(C)N(C(=O)CCC2CC2(F)F)C1 18214,c1(OC)cnccc1C(N1CCC(NC(C2(C)COCCO2)=O)C1C)=O 18215,c1(C(N)=O)cccc(OCC(N2CC=CC(NC(c3ccc[n+]([O-])c3)=O)C2)=O)c1 18216,c1(OCC)cc(C(N2CCC(CNC(=O)C3=CCC(C)CC3)C2)=O)cc(Cl)c1O 18217,C1(NC(c2cc(C)c(O)nc2)=O)CC2CCC(C1)N2C(C1(n2cccn2)CC1)=O 18218,CCCCCC(CC)C(=O)N1CCC(COC)(CNC(=O)CCC2CC2)CC1 18219,N1(C(c2cc(C)[nH]n2)=O)CC2CN(C(=O)Cc3ccc(C(F)(F)F)nc3)CCC12 18220,C(=O)(CC(C(C)OC)NC(c1ccc(O)cc1F)=O)NCCCCCC=C 18221,c1(CN2CC3C(C(=O)NCc4ccc(F)cn4)C3C2)cccc(O)c1F 18222,C1(C(=O)NCC2N(C(c3c(C)cc(C)s3)=O)CCC2)CCC(=O)CC1(C)C 18223,N1(C(C2C(C)OCC2)=O)CCC(NC(=O)CSc2cnn(C)c2)C12CCC2 18224,c1(C(N2CCC(NC(c3c(C)noc3)=O)C(O)C2)=O)cc2c(cc1O)OCCO2 18225,c1(OCC)ncc(C(=O)NC2CC(CNC(c3ncn(C)n3)=O)C(O)C2)cn1 18226,Cc1cc(C(C)C(=O)NC2CCCN(C(C3(C)COC3)=O)C2)cc(F)c1 18227,C(=O)(C(C)P(C)(C)=O)NC(C)CCNC(=O)Cc1c[nH]ccc1=O 18228,CC1CCN(C(c2scnc2C2CC2)=O)CC1CNC(c1cc(Cl)c[nH]1)=O 18229,C(CCCCCN=[N+]=[N-])N(CCOc1ncccn1)C 18230,C(=O)(CCC(F)(F)C(F)F)OCC1C2N(C(=O)OC(C)(C)C)CC(CC2)C1 18231,Cc1ncc(C(N2CCC23CN(C(c2cn4ccnc4s2)=O)C3)=O)c(C)n1 18232,C1(N2C3(CCC3)C2=O)CCCCC12CC2.Cc1nc(CC(=O)NCCO)cs1 18233,N1(C(c2c(CC)ncs2)=O)CCOC2CCN(C(=O)C(C)c3ccsc3)CC12 18234,c1(C(=O)NCC(C)(CNC(=O)CCOC2COC2)OC)csc(C)c1C 18235,c1(CCC(=O)N(CC(O)CNC(=O)CN2CSCC2=O)C)cc(F)cc(F)c1 18236,c1(C(CC)=O)cc(C(N2CCC(CCNC(C3CC4CC3C4)=O)C2)=O)ccc1F 18237,c1(OCC(C)O)ccccc1NC(=O)NCC1CCCC(C(F)(F)F)C1 18238,n1(C2CN(CC(C)C)C2)cc(COC2CN(C(c3cc(CO)c[nH]3)=O)C2)nn1 18239,C1(O)(CC)CCCN(C(c2ccc(CNC(=O)CC3(C#N)CCC3)o2)=O)C1 18240,C1(C(=O)C2CC2)CCN(C)CC1.CCC(C)OCC(=O)N(CCNC1CC1CF)C 18241,C1(NC(CCSCCC)=O)COC2(CCN(C(=O)CN3CCOCC3)C2)C1 18242,Cc1ccc(C(=O)NC2CC3CN(C(C4(F)CCCC4)=O)CC23)c(C(C)C)n1 18243,C(=O)(CCCCCC#N)N1C(C)(C)CC(NC(C2CC23CCC3)=O)C1 18244,c1(C(=O)NCCCCC2CN(c3c(C)cnc(C)n3)C2)cc(C)c(C)cc1Cl 18245,c1(C(N2C(CCNC(C3CCC(=C)CC3)=O)CCC2)=O)ccc2nc(S)oc2c1 18246,N1(C(CSC)=O)CCN(C(c2ccccc2Oc2cccnc2)=O)C(C(C)C)C1 18247,c1(C(=O)NC(C(C)NC(C2(CC)COC2)=O)C)cccc(P(C)(C)=O)c1 18248,C1(C(=O)NC(CC=C)CO)CN(Cc2ccccc2C(=O)O)CCS1 18249,c1(C(=O)NCCOCCCNC(C2(C)CC2(F)F)=O)cc2ccncc2s1 18250,N1(C(CCOc2cn(C)nc2)=O)CCN(C(c2cnn(C)c2)=O)CC12CCC2 18251,N1(C(C2(CC)CC2(F)F)=O)CCC(C2(NC(C3CCCCCC3)=O)CC2)C1 18252,c1(C(N2CC3C(NC(=O)C4=CCCC4)C3C2)=O)ccc2c(c1)C(=O)NCCO2 18253,N1(C(=O)Cc2ccccc2)CC2(CC2C(=O)Nc2ccc(N3CCCC3)nc2)C1 18254,C1(C(N2CC(C(=O)NC)OCC2)=O)CN(c2ccncc2)CCO1 18255,N1(C2CN(CC(=O)N(C(c3nnnn3C(C)C)C)C)C2)CC(C(=O)N(C)C)CC1=O 18256,c1(C(=O)NC(C2CCN(C(=O)C(CC)(CC)OC)CC2)CC)cncc(F)c1C 18257,C1(CN(C(c2c(OC)csc2)=O)C)COCCN1C(=O)CCCc1n[nH]c(=N)s1 18258,N1(CCN(CCCC)CCCC)CCCC(C)(C#N)C1.C(=O)CC 18259,S(=O)(=O)(c1cccc(Br)c1)N1CC2(CCN(C(C(CC)(C)C)=O)C2)C1 18260,c1(NC(C(C2CCN(C(c3c(C)nncc3)=O)C2)F)=O)cc(CO)cc(F)c1 18261,CCC(O)C(C)(C)C(=O)NOCC(N1CC2CCC2(C(=O)OC)C1)=O 18262,C1(CC)CNC(=O)CN1C(C1CC=CCN1C(=O)C(C)NC(C)(C)CC)=O 18263,N1(C(C2C(C)OC(=O)N2)=O)CC2CN(C(c3cnc(O)o3)=O)CC2(C(F)(F)F)C1 18264,c1(C(N(C2CCN(C(C3CCC3(F)F)=O)C2)CCC)=O)ccnn1CC 18265,CCC(C)(C)C(O)C(=O)NCCCN(C)C(C1CC1c1ccoc1C)=O 18266,c1(C(C)C)nocc1C(=O)NC1CCN(Cc2nnn(C)n2)C1 18267,C(=O)(C(CCCCSC)N(C)CCOCc1ccccc1C)NC 18268,C1(O)(C(=O)NCCC2(C(=O)OC)CCCC2)CCNCC1 18269,C1(C(=O)OCC2CC2)CCC(C)N1C(c1ncn(C(C)C)n1)=O.C(C)(C)(C)O 18270,Cc1nn(C)c(Cl)c1C=CC(N1CC(CNC(=O)Cn2ccc(O)nc2=O)C1)=O 18271,N1(C(C2(NC(c3n[nH]c(O)n3)=O)CSC2)=O)CC2(C1)NC(=O)NC2=O 18272,c1(OC)cccc(CC2CCCN2C(C2CC(Cl)(Cl)C2)=O)c1.C1(=O)CCN1C 18273,C1(C(=O)NCCN(C(=O)CCCc2nccs2)CCC)CCCC(N(C)C)C1 18274,CC(CCc1ccccc1)CC(=O)N(C1CN(C(=O)CCCF)CC12CC2)C 18275,c1(CN(C(c2nocc2CC)C(=O)NCCSC)C(C)C)ccccc1F 18276,c1(C(=O)NC2CC(NC(C3(CC=C)CCOCC3)=O)C2)ccc2nc(C)sc2c1 18277,C1(CC(=O)NCCCCNC(C2CC(CC(=O)OC)C2)=O)CCCC(=O)N1 18278,C1(NC(c2c(SC)ccs2)=O)CCC2CN(C(c3nccnc3N)=O)CC2C1 18279,c1(NC(c2ccc(CCNC(CCCC=C)=O)cc2)=O)ccc2nnsc2c1 18280,CC(C)CC(C)CC(=O)NC1CCCC1NC(c1cscc1-c1ccccc1)=O 18281,N#Cc1cc(F)ccc1C(=O)NCC1CN(C(c2cc(Cl)cc(Cl)c2Cl)=O)C1 18282,CC1C(C)N(C)CCN1C(=O)CC1COCCN1C(c1c[nH]nc1Cl)=O 18283,Cc1c(C(N2CC(=O)CC2C(=O)NC(CC2CC2)C2CC2)=O)nnn1C 18284,N1(C(C(C(C)C)c2cccnc2)=O)CCN(C(c2cn(C)cn2)=O)C(C)C1 18285,C(=O)(CC(O)CC(C)(C)C)NCC1N(C(c2nc(OCC)sn2)=O)CC=C1 18286,N1(C(=O)NCC2(OC)CC2)CCC(O)C(C(=O)NCCC(C)OC)C1 18287,c1(C(=O)NC2CC(C)(NC(=O)CC3CC34CC4)C2)csc2c1CCCC2 18288,Cc1nc(NCC(C)C(C)(F)F)cc(=NCc2c[nH]nc2C2CC2)[nH]1 18289,c1(OC)nc(C)ccc1C(=O)NC1CN(C(c2cnc(O)cc2O)=O)CC12CC2 18290,C(CCC(C)(C)C(=O)NCC(C)(C(=O)OC)OC)NC(c1ncc(CC)cn1)=O 18291,c1(C(N(C2CCCN(C(=O)Cc3cnns3)C2)C)=O)cnc2c(c1)NCC2 18292,C(C1CN(C(C2CC2c2ccco2)=O)CC1C(=O)NC1CC(C)C1)=CC 18293,N1(C(CC(C)SC)=O)CC(C)(C)CC1CNC(=O)CC1CCS(=O)(=O)C1 18294,N1(C(c2c(C)nco2)=O)CC(C)(C)OCC1CNC(C1(C)CC2CCC1O2)=O 18295,C1(C)(CC(NOCCOC)=O)CCCN1C(c1nnn(CC)c1C)=O 18296,CC1CN(C(=O)CSCC(N)=O)CC1NC(=O)CCc1cn(C)nn1 18297,CC(CO)C(C)N=c1[nH]c2cc(Cl)c(S(=O)(=O)NCCC3(C)CCCC3)cc2s1 18298,C1(C(C2CCOC2)NC(CSS(C)(=O)=O)=O)CCCN1C(=O)CC1CC=CC1 18299,C(=O)(CC(COC)COC)NC(C(=O)N(CCCCCCC)C)c1cccs1 18300,c1(C(N(C(C)CNC(c2sccc2C)=O)CC)=O)cc(F)ccc1OC 18301,C(=O)(C#CC1CCCC1)N(CCCNC(c1c(C)cnn1C(C)C)=O)CCO 18302,CC1(C(=O)NC2CCCCC2NC(c2cc(N)cc(O)n2)=O)CCC(=O)NC1 18303,N1(CC)CCCC(C(=O)NC2CC(NC(c3cn(C)cc3C)=O)C(O)C2)C1 18304,N1(C(C(CSC)O)=O)CCOC(CNC(c2cc(C)co2)=O)C1 18305,C(=O)(CS(=O)(=O)CC(C)C)NCC1(F)CN(C(c2cnc(C)[nH]2)=O)C1 18306,CC(C)(CC(=O)NC1CCCN(C(c2nccc3c[nH]nc23)=O)C1)CC(F)(F)F 18307,CCC(C(=O)NC12CC(CNC(c3c(C)cc[nH]c3=N)=O)(C1)C2)C(C)(F)F 18308,CC(CCNC(=O)CC1CCCO1)N(C(=O)C=CCO)C 18309,CCC(CC)(CO)C(=O)N1CCC(O)C(NC(=O)C=CC2CCCN2C)C1 18310,CC(C)CC(O)C(C)C(=O)N1CC(C(=O)NCC2(C)CC=CCC2)C(C=CC)C1 18311,N1(CCNC(CC(C=C)C)=O)CCN(C(=O)CN(C2CCSC2)C)CC12CCC2 18312,Cc1nn2ncccc2c1C(=O)NCC1CCCCN1C(c1ccncc1Cl)=O 18313,CC(C)(C)CC(C)(C)C(=O)NC1CCN(C(=O)CC2CCCC3(CCC3)O2)C1 18314,CN1CC(C)(C(N2CCC(CO)(CNC(C3CC4(CCCO4)C3)=O)C2)=O)CC1=O 18315,c1(C(C(=O)NCCC2(O)CN(C(C(C)SCC)=O)C2)C)ccc(F)c(F)c1 18316,c1(N2CCN(C(C(=O)NCC=C)COc3ccccc3)CC2)ccccc1C#N 18317,c1(CNC(C2(F)CCN(C(C=Cc3cn(C)nc3)=O)C2)=O)nnc2n1CCC2 18318,C=CCC(C)(C)CC(=O)N1CCC(C)C(CNC(=O)C(CC)C(=O)OCC)C1 18319,c1(C(N(CCNC(=O)C(C2(O)CCCCC2)(F)F)CC)=O)cnc2nccn2c1 18320,N1(C(CC2CC(OC)C2)=O)CCN(CCN(C)C(C2CCCS2(=O)=O)=O)CC1 18321,C(CCN=c1cc[nH]cc1S(=O)(=O)NC1CCCc2c1cnn2C)SC 18322,c1(C(=O)NC(C)C(C)(C)NC(C2CC2C)=O)cc(=O)c2cc(Cl)ccc2o1 18323,c1(C(=O)NCC2N(C(CNS(C)(=O)=O)=O)CC(F)C2)c(OC(F)F)cccc1F 18324,c1(OCCOC)cc(OC(C23CN(C(=O)OC(C)(C)C)C(C)(C2)C3)=O)ccc1O 18325,c1(C(=O)NCC(C)NC(c2snc(O)c2Cl)=O)ccc(C2COC2)cc1 18326,C1(NC(CN(C(=O)CCCF)CCC)=O)CCCC1(C)CO 18327,n1(CC)ccc(C(=O)NC(CNC(=O)C(C)n2cnnn2)CO)n1 18328,C1(NC(=O)OCC)CN(C(=O)C(C2CCCCC2)NC(N)=O)C2(CCOCC2)C1 18329,c1(OC)cccc2cc(CCNC(=O)NCc3ccc(C#N)c(OC)c3)oc12 18330,c1(C(=O)NC(C(C)NC(=O)CCC2CC2)(C)C)cc2ccccc2n1C 18331,CCCCCC(C)CC(=O)NC(C(=O)NCC1(CN=[N+]=[N-])CC1)C(C)(C)C 18332,C(=O)(CC(C)CC(C)(C)C)NCC1(F)CCCN(C(CCN(CC)CC)=O)C1 18333,Cc1cc(C(=O)NC(CNC(C2(C)CCC(=O)NC2)=O)CO)ccc1Br 18334,c1(C(C)C)cccc(C2CC2)c1.c1(C2c3nnnn3NC2)cnc(Cl)n1C.C1(CC)CC1 18335,CCC(C)(C)C(O)C(=O)N1CC(F)CC1CN(C(=O)CC1CC1)C 18336,CC1CN(C(C2CC(O)CN2C(c2ccc(CO)s2)=O)=O)CCC1N(C)C 18337,CC1CCCN(C(=NCCS(=O)Cc2ccccc2)NCC(C)(C)C)C1 18338,N1(C(COc2c(OCC)cccc2)=O)CCC(C)(C(=O)N(C)CCl)C1 18339,c1(C(=O)NC2(CO)CN(C(CC(C)O)=O)C2)ccc2[nH]c(=O)cnc2c1 18340,c1(C(=O)NCC23C(CN(C(Cn4c(C)csc4=O)=O)C2)C3)cccn2cncc12 18341,C(=O)(CCCCCNC(N)=O)NC(C)CN(C(=O)Cn1cc(C(C)O)nn1)C 18342,Cc1cncc(CC(=O)NC23COC(CNC(c4cc(CO)c(C)o4)=O)(C2)C3)c1 18343,Cn1c(C(N2CC3CCN(C(c4cncc(O)c4)=O)C3C2)=O)cc2sccc12 18344,C1(NC(C2(C)CNC(=O)C2)=O)CCCCN(C(C2CC2(F)F)=O)C1 18345,c1(C(N2CCC(OCCNC(C3CC(CC)C3)=O)C2)=O)cncc2cnccc12 18346,C1(N(CCC)C(C2CC=CCC2)=O)CCN(C(C2CC2c2ccncc2)=O)CC1 18347,N1(C(c2cn(CCCC)nn2)=O)CC2CC1C2NC(c1scnc1C(C)(C)C)=O 18348,Cc1cc(CCCNC(=O)C(C)Sc2ccccn2)oc1C(=O)O 18349,c1(C(N(CCN(C(CC(CC)OC)=O)C)C)=O)[nH]cc2c1CCS2(=O)=O 18350,Cc1cccc(C(=O)NCCC2(O)CN(C(=O)CCOc3cccnc3)C2)c1 18351,C1(NC(C2CCC(C)(C)O2)=O)CN(C(=O)C=Cc2cc[nH]n2)Cc2nccn2C1 18352,N(C1CCC(NC(c2ccnc(-n3cccn3)c2)=O)c2ccccc21)C(=O)CO 18353,c1(C2C(C)C2)ccc(CCC(=O)NCCCCN(C)C(c2coc(Cl)c2)=O)o1 18354,C(CC(=O)NCc1ccc(Cl)cn1)(C(F)(F)F)NC(c1n(C)ccc1)=O 18355,c1(C(C(=O)NCC2(C(N3CC(CN(CC)CC)C3)=O)CC2)(C)C)cccc(C#N)c1 18356,c1(C2(NC(C3CCOC3)CC)CCC2)c(F)cccc1F 18357,c1(C(N2CC(C)C(NC(=O)CCOC3CCC3)C2)=O)cc(F)ccc1Br 18358,CC1CC(N(C)C)(NS(=O)(=O)CC2=CCCCC2)CC(C)(C)C1 18359,C(c1ccncc1C)=CC(=O)NCCc1c(CNC(C=CC(CC)C)=O)nco1 18360,CC1(C)C2COC1(C(=O)NCC(C)(C1CC1)NC(c1cc(Cl)c(Cl)s1)=O)C2 18361,C1(CNC(c2cnn(C(C)C)n2)=O)C2CN(C(=O)C(C3CCCCC3)F)CC12 18362,C12(CNC(c3cnc(C4CCCCC4)s3)=O)CC(CO1)N(C(=O)C1CC1)C2 18363,C1(CNC(C2N(C(CC3N(C)CC=CC3)=O)CCC=C2)=O)CC(C(N)=O)=NO1 18364,c1(C(=O)OCC(=O)NC2C(C3C(C)C3)C2)cnn2cc(C#N)cnc12 18365,CC(C)(CNC(=O)Cn1cc(Cl)cn1)C(=O)N1CC2C=CC2C1 18366,c1(CC(=O)NC2CC(F)CN(C(c3c[nH]ccc3=O)=O)C2)cccc2sccc12 18367,CC(C)C(C(=O)NC12CC1CN(C(C1(N(C)C)CCCC1)=O)C2)C1CCC1 18368,c1(NCCCC(N(C(=O)NC)C2CC2)OC)nc2ccccc2c(Cl)c1Br 18369,c1(-c2onc(C3N(C)CCNC3)n2)ccnc2[nH]ccc12 18370,c1(C(N(CCCCCNC(=O)CCCCNC(N)=O)C)=O)ccnc2c1CCO2 18371,C(=O)(C(C)(C)C(F)F)N(c1cn(CC(O)(C(F)(F)F)c2ccc(Cl)cc2)nn1)C 18372,C1(NC(CCC2CC(C)C2)=O)CCCC1NC(c1ccc(Cl)s1)=O 18373,N(C1COc2ccc(F)cc21)CCO.n1(CCCOC)nnnc1C(C)CCOC 18374,C1(C#N)(C(=O)NCC(CNC(=O)C(C(C)C)N(CCO)C2CC2)OC)CC1(C)C 18375,N1(C(C(C(C)SC)O)=O)CCOC2(C1)CN(C(c1cc3c(C)nn(C)c3s1)=O)C2 18376,C1(NC(C2(C(=O)OCC)CCCC2)=O)CC(C)N(C(=O)CCN2CCOCC2)C1 18377,CP(C)(=O)c1cccc(C(=O)NCC2CCC2NC(C2CC3CCC3C2)=O)c1 18378,c1(OC)cc(C(=O)Nc2cccnc2O)ccc1I 18379,Cc1nc2nccc(C(N3CC(N(C(=O)CC4CC(F)(F)C4)C)C3)=O)n2n1 18380,C1(C(N2C(CCNC(C(COC)O)=O)CCC2)=O)CN2CCN1CC2C 18381,N1(C(C=C(CCC)C)=O)CC(C2CC2)(C(=O)NC(C)CCc2cn[nH]c2)C1 18382,c1(C(=O)NC(CCN(C(C=C(C)Cl)=O)C)C(C)(C)C)sc2cncn2c1C 18383,C=CC1(CC(=O)NC2CCCC(O)C2)CN(C(c2cocc2CC)=O)C1 18384,S(=O)(=O)(c1c(OC)cccc1O)N.C(CCC)N(CC#C)CC 18385,C12(C(N3CC(C)(NC(CC(CC)C4CC4)=O)C3)=O)CCCC(C1)OC2 18386,n1(CC(=O)N(C2CN(C(C=C(C)C(F)F)=O)CC2F)C)cc(S(N)(=O)=O)cn1 18387,c1(C(N2CCN(C(C(C)OC)=O)CC2CCO)=O)cc(C)cc2c1OCC2 18388,N1(C(CC2(C)CN(C(c3ccc4n[nH]cc4c3)=O)C2)=O)CCCCC(C)(F)C1 18389,N1(C(CCCC2C(C)C2)=O)CC(CNC(=O)C2=CSCCO2)OC2(CCC2)C1 18390,c1(CC(=O)NC2CC(CC3CC3)C2)ccc(CNC(C(=O)Nc2nccs2)=O)cc1 18391,C1(C(N2CC(CC)C2)=O)(CNC(=O)COc2ccsn2)CC12CCC2 18392,N#Cc1cnc(C(=O)NCC2C=CC(NC(=O)CC3(O)CCCCC3)C2)c(Cl)c1 18393,CC(O)C(C)C(=O)N1CCN(C(=O)C(CSCc2ccccc2)N(C)C)CC1 18394,C1(NC(=O)CCn2cncn2)CCC(CNC(c2cc(-c3cccs3)[nH]n2)=O)C1 18395,N1(C(CC(C)C(F)(F)F)=O)C(C)CC2CN(C(=O)Cc3c(Cl)cnn3C)CC12 18396,n1(CC)cnc2c(C(N3CCCC(NC(C4(F)CC4C)=O)C3)=O)cccc12 18397,c1(C(N2CC(C)C(NC(=O)C=CC3(C)CCOCC3)C2)=O)cc2cnn(C)c2s1 18398,C(C(C)(C)C(=O)N1CCN(C(=O)CCOC2CC2)CC1)SC.C1C(=O)N1 18399,c1(C(N2C(CNC(C3CC4C=CC3O4)=O)COCC2)=O)cc(Cl)ccc1Cl 18400,c1(C(N2CC(NC(CN(c3ccccc3)C)=O)C3C2C3)=O)cc2occc2s1 18401,C12(C(=O)NC3C(NC(c4cncc(Cl)c4Cl)=O)CCC3)CCCN(CCC1)C2 18402,c1(C(=O)NC2CCC(NC(C(CC)(C)C#N)=O)C2)cnn2c(Br)cccc12 18403,C1(CC)C(C)CCN1C(c1cccc(CNC(=O)CNC(=O)CN(C)C)n1)=O 18404,c1(-c2c(C)cccc2)nc(=NC(C)(C)CCNC(=O)C=CCN2CCOCC2)s[nH]1 18405,c1(N2CC(CNC(C(CCC)NC(N)=O)=O)OCC2)ncc2c(ncn2C)n1 18406,C(C1=NOC2CC12)(c1nnnn1C1CC(F)(F)C1)NCC(C(C)C)(C)C 18407,C(=O)(CCCCCCSC)N1C(CNC(C(C=C)(C)CC)=O)CC2CC21 18408,c1(C(N2C(CC)CN(C(=O)C(C)NC(=O)NC)CC2)=O)nc2n(c1Cl)CCCC2 18409,C(c1nc2ccccc2o1)=CC(=O)NCC(C)CNC(=O)Cc1ccnc(O)c1 18410,CCC(CCCC(=O)N1CCCOCC1C)NC(C1CC(C)CCO1)=O 18411,c1(CC(=O)NC2CC(F)(CNC(=O)Cc3ccccc3O)C2)cc(F)ccc1Cl 18412,N(C1CCc2ccccc2-n2ccnc21)C(C(C)NC(c1ccc(Cl)cc1)=O)=O 18413,N1(Cc2ccc(C#C)s2)CCCN(C(c2nc(C)c(CC)s2)=O)C(C)C1 18414,c1(C(C(=O)NCCCC2N(C(C3CN(CC(C)C)C3)=O)CC2)O)cnccc1C 18415,c1(COC)nc(C)cc(=NCC2CN(C(c3cnc(C)nc3SC)=O)CC2C)[nH]1 18416,N1(C(C(C)OCC2CC2)=O)CCCC(C)(CNC(c2ncccc2F)=O)C1 18417,Cc1coc(C=CC(=O)NCC(CC(C)C)NC(c2coc(Br)c2)=O)n1 18418,C(=O)(C1=CCN(C)C1)N(CCC(C(C)C)NC(=O)CC1CCC(C)(C)C1)C 18419,Cc1nccn1CC(=O)N(CCN(C)C(c1ncoc1C1CCC1)=O)C(C)C 18420,c1(NC(C(CC)N(C)C(C2CC2(C)C(F)F)=O)=O)cc(C)cc(O)c1 18421,CON1CC(C(=O)NC(C2(C(N3CCC(OCC(C)C)C3)=O)CC2)C)CC1=O 18422,C1(NC(C2C(CC(C)C)C2)=O)CCCC(CC(=O)NCc2cc(O)ncn2)C1 18423,C(=O)(C(COC)C(F)(F)F)N1CCC(C2(NC(C(C)OCC#C)=O)CC2)C1 18424,Cc1cc(=NCCN2CCC(C)CC2)[nH]c(NC2CCCC(F)C2)n1 18425,CCC(C)CC(C)C(=O)N(CCNC(c1ccc(C)nc1OC)=O)CCOC 18426,C(=O)(CCCC(O)c1ccccc1)NC(C1CCCN1C(C1CCCO1)=O)C 18427,N1(C(C2C(C)(CC)C2)=O)CCCCC12CC(NC(=O)Cn1ccnc1C)C2 18428,N1(C(c2cn(C)c(=O)cn2)=O)CCN(C(C2(F)CC2(Cl)Cl)=O)CC12CCC2 18429,N1(C(c2scc(OC)c2)=O)CC2(NC(c3ccc(F)cc3O)=O)CCCC2(F)C1 18430,C=C(C)CC(C(=O)NCc1ncc(C)s1)NC(C1CCCN1CC)=O 18431,C1(C(=O)NC2C(C#C)CCC2)CNC(=O)CN1C(=O)COC1CCC1 18432,Cc1ccc(C(N2CC(C)CCCC2C)=O)cc1S(=O)(=O)NCCC(=O)O 18433,N(C1CCCc2c(F)cccc21)C(C(=O)NCCCC=C)=O 18434,C#CC1CN(C(C2CN(C(c3ns[nH]c3=O)=O)CC2(C)C)=O)CCN1C 18435,C1(CC)CC(C(=O)NC2(CNC(c3ccc(Cl)nc3C)=O)CC2)CCC1=O 18436,c1(C(=O)NCC(CC=C)NC(=O)C(c2cnn(C)c2)O)nc(Cl)sc1C(C)C 18437,C1(NC(C=C2CCC(C)CC2)=O)CCN(C(c2cc(Cl)cn2C)=O)C12CC2 18438,c1(C(N(C)CCN(C)C(C2CC(C(F)(F)F)C2)=O)=O)ccoc1I 18439,N1(C(C(C(C)(C)C)=O)=O)CC(CNC(C2CC(F)(CO)C2)=O)CC12CCC2 18440,N1(C(c2cc(OC)ncc2)=O)C2CCC1CN(C(C1CC1c1ccnn1C)=O)C2 18441,c1(OC)nccc(NCC2(CNC(C3CCCCC3)C(=O)OCC3CC3)CC2)n1 18442,CC(C)C(C(=O)NCCC1CN(C(c2cccn2C)=O)CCO1)c1ccn(C)n1 18443,N1(C(C(C)=C2CC2)=O)CCC2(C1)CN(C(c1ccc(F)c(O)c1F)=O)C2 18444,N1(C(CC2(C)CC2(F)Cl)=O)CC(C2(NC(=O)CSS(C)(=O)=O)CC2)C1 18445,n1(CC)nc(CN2CC3CC2(C)C3)c2c1CCOC2 18446,C1(NC(C2(CCOC)CC2)=O)CN(C(c2cncn(C)c2=O)=O)C2CCCCC12 18447,C=CC(CCC)CC(=O)N1C2CCC1CC(CNC(=O)C(C)(C)n1cccn1)C2 18448,Cc1nn(C)cc1CCC(=O)NCCC(C)NC(c1[nH]ncc1C#N)=O 18449,c1(C(N2CC(N(C(c3c(C)cn(C)c3)=O)C)C(F)C2)=O)ccc2nonc2c1 18450,c1(C2CC(NC(C(N3CC(OC)C(OC)C3)=O)=O)C2)ccc2c(n1)NCCC2 18451,C1(C)(C(=O)NCCOCCCNC(C(C2CCOC2)OC)=O)CC2(CCC2)C1 18452,C(=O)(C1=CC2CCC1C2)N(CC(C)NC(c1cnn(CCOC)c1C)=O)CC 18453,C1(CNC(C(C)(C)SC(F)(F)F)=O)CN(C(c2cnns2)=O)CCO1 18454,C(CCC(C(=O)NCC1(O)CCSC1)NC(=O)CC(C)C)OC 18455,N1(c2nnc(CC)s2)CCC(NC(=O)CNC(c2cscn2)=O)C(C)C1 18456,N1(C(c2c(CC)onc2)=O)CC(C(=O)NCC2CC(C)(C)C2)C2(CC2)C1 18457,N(C1c2ccccc2CC1NC(=O)C1CCCc2ccnn21)C(CCC(C)C)=O 18458,c1(CN2CCC(C(C#C)C)C2)cnc(OC)cc1C.c1(C)ccccc1 18459,C(CCN=C(NCc1cncc(O)c1)NC1CCOCC1F)OC(C)C 18460,C#Cc1ccc(C(N2CCCC2CN(C(=O)C(F)CC)CC)=O)c(OC)c1 18461,C(=O)(CCC(F)(F)CN=[N+]=[N-])NCCC1N(c2nnc(CCC)s2)CCC1 18462,N1(C(C=CCOC(C)(C)C)=O)CCCC2CCN(C(=O)C3=C(Cl)CCC3)CC12 18463,Cc1cnc(C)c(C(=O)NCC2CC2CNC(c2n[nH]cc2C(C)C)=O)c1 18464,c1(C(=O)NC2CC(C)N(C(=O)CCC(C)(C)O)C2)ccc(C#N)c(Cl)c1 18465,C1(C(=O)NCC(C(C)C)NC(C2(CC#C)CC2)=O)CC2(C1)CC(C#N)C2 18466,c1(C(C)C)ccc(C(N)CC(=O)N(c2ccc(Cl)cn2)C2CC2)cc1 18467,c1(OC)cccc(C(N2CCC(N(C)C(C3C(C)(C)C3(F)F)=O)C2)=O)c1[N+](=O)[O-] 18468,C1(=O)N(OC)C(C)C(=O)NC2CCCCC12.C(=O)(C1=NN(C)C(=O)CC1)OC 18469,N1(C(C2CC(OC)C2)=O)CC(CNC(=O)CSCc2ncc[nH]2)C(C(F)(F)F)C1 18470,C(C1CCCCCC1)=CC(=O)NC1(CCNC(C2(C)CCCOC2)=O)CCCC1 18471,C1(C(C)(C)C)CCN(C(=O)C(=O)NCC(C2CCCC2)=O)C(C(N)=O)C1 18472,c1(NCC2(CC)CCCC2)[nH]c(=NCCC2CCCS2)nc2c1ncn2CC 18473,N1(C2(c3nc(C)oc3)CC2)CCN(c2ccc(C)c(C)c2)CC1C.c1nnnn1C 18474,C(=O)(C(C)C1=CCCC1)NC(CCCNC(C=CC=CC)=O)c1ccccc1 18475,C1(C(=O)OC)CCC(C(=O)NC(CNC(c2nc(C)no2)=O)CC)S1 18476,c1(CC)cc(C(=O)NCCCC(C)NC(C23CCC(OC)C2C3)=O)n(C)c1 18477,N1(C(C(CCCC)C)=O)Cc2n[nH]cc2C1C(=O)NCCc1nnc(C)s1 18478,CN1CCC(C)(C(=O)NCC(O)CCNC(=O)C(CN(C)C)N(C)C)CC1 18479,c1(CN2CC(NC(=O)CCN3CCCC3)CC(F)(F)C2)ccc2c(c1)OCCO2 18480,N1(C(CC=C=C)=O)CCOC2CN(C(c3[nH]c(=N)ccc3C)=O)CC12 18481,N1(C(C2(CC#C)CC2)=O)CCc2nc(O)cc(C(=O)NC3CCN(C)C3C)c2C1 18482,C12(C(N(C3CN(C(=O)COC4(C(F)(F)F)COC4)C3)C)=O)CC(F)(C1)C2 18483,c1(C2OCCN(C(C34CCC(OC)C3CC4)=O)C2)ccc(F)cc1C#N 18484,c1(OCC)cccc(C=CC(=O)NC2CCCN(C(C3(C)CNC(=O)C3)=O)C2)c1 18485,CC1(C)CCN(C(=O)CCC(F)F)CC1CNC(=O)CN1CCC(CO)CC1 18486,CC1CCCN(C(=O)CC(F)(F)c2ccccc2)C1CNC(=O)C(O)C1CC1 18487,S(=O)(=O)(c1c[nH]ccc1=NCC1CCCOCC1)NCc1c(Cl)cn(C)n1 18488,N1(C(C2N(Cc3cc(OC)cc(F)c3)CCNC2)=O)Cc2ccc(O)cc2C1 18489,c1(OC)ccc(F)cc1C(=O)NCCC(C)(C)NC(C1CC12CC(C)(C)C2)=O 18490,C1(C(N2CCC(c3ccon3)C2)=O)COC2(C1)CN(C(c1cccnc1O)=O)C2 18491,C#Cc1ccnc(C(=O)N(CCCOCCNC(=O)C(C(C)CC)OC(C)=O)C)c1 18492,C(CC(=O)N1CC(C)(CCO)C1)(C(C)OC)NC(C(C)OCCOC)=O 18493,C1(NC(c2cc[nH]n2)=O)CN(C(c2cscn2)=O)C2(CCC2)C1 18494,C1(C(=O)NCC2OCCN(C(C3(n4cncn4)CC3)=O)C2)CCCCNC1=O 18495,c1(OC)cc(C(N2CC=CC(NC(=O)C(c3cncnc3)C)C2)=O)cc(N)c1O 18496,C(=O)(N=c1[nH]nc(Cl)c(C)c1C)NCc1c(F)ccc(OC)c1 18497,N1(C(C2C(NC(C(C)N(C(C)=O)C)=O)CC=CC2)=O)CCOC(C)C1C 18498,C1(C(=O)NC(C)C=CC(=O)NCCN2CCC2)OCCCC1(C)C 18499,S(=O)(=O)(c1ccc(S(=O)(=O)NC2CC2)cc1)N1C(C#N)C2(CC1)CCC2 18500,C1(CCC)(NC(=O)C=C(C)C(C)C)CCCN(C(=O)C(C)CC(F)F)C1 18501,c1(C(=O)NC2CN(C(Cc3ccc(C)o3)=O)CC2(C)C)cc(Cl)cc2c1CCC2 18502,Cc1cc2c(cc(C(N3CC4CCN(C(=O)C(F)F)C4C3)=O)n2CC2CC2)s1 18503,C1(NC(c2c(C#C)cn(C)n2)=O)CCN(C(=O)C(C)OCCOCC)CC1(C)C 18504,C12(NC(CC3CN(C(C(CC#C)O)=O)CC34CC4)=O)CCC(C1)C(O)C2O 18505,c1(C(=O)NC2CC(F)(CNC(Cc3n(C)ccn3)=O)C2)cc2cccc(F)c2o1 18506,N1(C(C2C(OC(C)=O)C2)=O)CCCC1C(=O)NC(C)CC(N)=O 18507,C1(O)(CNC(Cc2c(C)cccc2)=O)CCCN(C(c2c(C)noc2C)=O)CC1 18508,c1(SC)cc(C(N2CCC2CNC(=O)C2CC2)=O)nn1C 18509,C(=O)(CCC(=O)N1CC2C(CNC(c3cnccn3)=O)C2C1)NCCC 18510,C1(C(N2C(C)(CC(=O)NC3(CO)CCOCC3)CC2)=O)(CC)CCOCC1 18511,C1(C(N2CCOCC2)=O)CN(Cc2ccnc(Br)c2)CC(F)(F)C1 18512,c1(CC(=O)N(C(C)CCNC(c2c[nH]c(=N)s2)=O)C)cccc2ncccc12 18513,Cc1cccc(C(=O)NC2CCN(CCNC(c3cc(C)n(C)c3)=O)CC2)c1N 18514,Cc1ncn(C)c1C(N1CC(n2cc(CNC(c3csc(=N)[nH]3)=O)nn2)C1)=O 18515,c1(C(=O)NC2CCC(CC(=O)NCCC=C=C)CC2)cc2occc2[nH]1 18516,C1(NC(Cc2c(C)cco2)=O)CCCCCN(C(c2ccc3cnnn3c2)=O)C1 18517,N1(C(C=C(C)C(C)(C)C)=O)CCCCCCC1C(N1CC2CCOC2C1)=O 18518,CC(C(=O)NC1CCN(C(=O)C(c2cc(F)ccc2F)=O)C1)C1=CCCC1 18519,Cc1oc(S(C)(=O)=O)cc1C(=O)NCC1CC(O)CN1C(C1CC12CCCC2)=O 18520,N1(c2cc(N(CCC(C)O)C)nc(C(F)(F)F)n2)CCC(CO)C(C)(C)C1 18521,N1(c2nnc(CC)o2)CCC2(CC1)CN(C(=O)C=CSC)CC(C)O2 18522,c1(N2CCN(C(C(c3ccc(F)cc3)OCC)=O)CC2)ncc([N+](=O)[O-])cc1F 18523,N1(C(C2=CC(C)(CC)C2)=O)CC2CCCC2(NC(c2ccn(C)c2)=O)C1 18524,N1(C(C2CC(C)SCC2)=O)CCC2(C1)CN(C(=O)Cn1cccc1)CCO2 18525,n1(CC)cc(C(N2CC(C(O)C(=O)NC3CC(C(C)C)C3)C2)=O)nn1 18526,C1(NC(c2ccc(C)nn2)=O)CN(C(C2CC2C(C)O)=O)CCC12CCC2 18527,N1(C(C(C(C)C)n2cnnn2)=O)CC2(CCC2CNC(=O)C(=O)N2CCCC2)C1 18528,N1(C(C(CCF)NC(C2CCC(C)(O)CC2)=O)=O)CC(C2CC2(F)F)C1 18529,c1(C(=O)NCCCCNC(C(C)OCOC)=O)cnn(CCCN2CCCC2)c1 18530,C1(NC(c2ccc(C)o2)=O)CCCCC12CCN(C(c1cncc(F)n1)=O)C2 18531,C1(C(N2CC(CC(C)NC(CCNS(CC)(=O)=O)=O)C2)=O)CCCN1C 18532,Nc1ccc(C(N2CC3(CC3)CC2CNC(=O)C(F)=CCCF)=O)c(Cl)c1 18533,c1(CC(=O)NC2C(COCC(=O)NC3CC(F)(F)C3)CC2)ccc(C(F)F)cc1 18534,c1(C(=O)OC)cccnc1-n1ccnn1.CCC(C)C(=O)N(C)CCN(C)C 18535,c1(NC(C2(F)CCN(C(C(CC)O)=O)C2)=O)ccc2c(c1)OCCO2 18536,CONC(=O)C(C)(C)CCNC(c1ccc(C(C)C)o1)=O 18537,c1(C(=O)NCCC(C)CCNC(=O)CS(C)(=O)=O)cc(C(F)F)cc(F)c1 18538,C1(NC(CCC(C)OC)=O)C(C)CCN(C(=O)COCCN(C)C)C1C 18539,C1(NC(CN2CCN(C(=O)C(C)(C)C)CC2)=O)CCCC(CC2CCN(C)C2)C1 18540,C(=O)(C1=CCS(=O)(=O)C1)N1CCC(O)(C(C)CNC(c2cc(O)nc(Cl)c2)=O)C1 18541,CS(=O)C1CCCC(OC(=O)CCOCOC(C2CCCO2)=O)C1 18542,c1(C(=O)NCC2CC(NC(=O)Cn3ccnn3)C(O)C2)coc2ccc(F)cc12 18543,Cn1c(C(=O)NCC(O)CNC(c2ccc(Cl)o2)=O)cc2c1CCOC2 18544,N1(C(C(CO)N(C)C)=O)CCC2(CCC(NC(c3ccc4n[nH]cc4c3)=O)C2)C1 18545,C1(CNc2c(N3CCC(C#C)(O)CC3)cccc2)CC2(CO1)CC(F)(F)C2 18546,c1(CC)cc(C)c(C(N2CCN(c3cccs3)CC2)C(=O)NCCOC)cn1 18547,c1(-c2cn(CCOCCNC(CCn3ccc(C)n3)=O)nn2)cn(C)nc1C 18548,c1(CNC(CNC(=O)NC)=O)ncc(C(=O)OCCC)o1.C1(CN)C=NNC1=O 18549,CC1CC(C(=O)N(C2CCCC2O)C)N1C(=O)CCN(C)C 18550,c1(CNC(C(C(C)C)C)=O)n[nH]c2c1CN(C(=O)CSc1n[nH]c(O)n1)CC2 18551,C1(CSc2cccc(NC(NNC(=O)C3C(C)CCO3)=O)c2)CCn2ccnc2C1 18552,N1(C(C(CC)NC(C)=O)=O)CCN(Cc2cc3ccccc3s2)CC12CC2 18553,c1(C(=O)NCCN(C(C2CC(CCC)C2)=O)C)occ(C)c1C 18554,N12CC(O)(C1)CNC2=O.C1(c2nnnn2CC2CCOC2)(CC2CC2)CCSC1 18555,N1(C(C(CNC(C(CC2CC2)OC)=O)C)=O)CCc2ccc(C#N)cc21 18556,c1(C(=O)NCC2CCN(C(C3(CCCC)CC3)=O)CC2O)cccc2c1CCN2 18557,c1(C(N2CCC(C)(C(N(C(C)CO)CC)=O)C2)=O)cnc2cc[nH]c2c1 18558,c1(C(=O)NC2C(NC(C3(C#N)CCCC3)=O)COCC2)ccc2c(c1)CCO2 18559,N1(C(c2c(C)cc(C)[nH]2)=O)CCC(CNC(c2c[nH]nc2C2CCC2)=O)C(C)C1 18560,C(c1ccc(Cl)c([N+](=O)[O-])c1)=CC(=O)NCC1N(C(c2nc(C)sc2)=O)CC1 18561,c1(CNC(C2(C)CC(C)C2)=O)cc(C(=O)NC2CCN(C)C2=O)n(C)n1 18562,C1(C(=O)NC(c2onc(C)n2)C)CN(C(=O)CCCN2CCCC2)CC1C(C)C 18563,C(=O)(C1=CCOCC1)N1C(C2(NC(COC3CN(C(C)=O)C3)=O)CC2)CCC1 18564,N1(C(=O)NCc2cncn2-c2cccc(Br)c2)CCCN(CCO)CC1 18565,c1(SC)nn(C)cc1C(N1CCCC1(C)CNC(=O)Cn1cc(CSC)nn1)=O 18566,N1(C2CCN(c3ccc(C)cc3Cl)CC2)CCN(CCO)C(C)(C)C1 18567,N1(C(CN(C)C(c2cnn(C)n2)=O)=O)CCN(C(C2CCC(=O)NC2)=O)CC1 18568,c1(OC)ccnc(NNC(=O)c2ccc(S(=O)(=O)NCc3ccco3)s2)n1 18569,C1(NC(c2cc(OC)no2)=O)CC2CCC1CC2NC(C1CCCC1(C)C)=O 18570,C=C(C)C(C)(O)C(=O)N1CCCC(C)(NC(c2cnc(S)n2C)=O)C1 18571,Cc1ccc(Br)c(N)c1C(=O)NC1CCN(C(=O)C(N)=O)C1 18572,CCC(C)C(C(=O)NCC1CC2(CC2)CO1)NC(=O)Cn1cnnc1O 18573,N1(C(CN(CCOC)C)=O)C2CCC1CC(NC(C1(C)CCC(O)CC1)=O)C2 18574,Cc1cc(CC(N2CCC(C(=O)NCC3C(CO)C3(F)F)C2C)=O)n(C)n1 18575,CC1CC(CCNC(c2c[nH]ccc2=O)=O)CCN1C(C1CN(C2CCC2)C1)=O 18576,c1(C(=O)NC2CC(C)(NC(C(CC=C)OC)=O)C2)ccc2nccnc2n1 18577,C1(C(=O)NC(C)CCCNC(c2cc(C(C)(C)C)ccn2)=O)COC2(CCC2)C1 18578,CC1CCC(Cl)=C(C(=O)N2CC(NC(=O)C(C)(F)F)C(C)C2)C1 18579,c1(CC)ccc(C)cc1C(N1CCCC1C(C)NC(c1[nH]nnc1C)=O)=O 18580,C1(C(=O)NCC2(C(N(CCN(C)CCO)C)=O)CC(C)(C)C2)CC(=O)NC(=O)C1 18581,C1(NC(=O)C(O)C(F)F)CN(C(=O)Cc2ccc3nonc3c2)C2(CCC2)C1 18582,C1(N(C(c2cccn2C(C)C)=O)CC)CCCN(C(c2ccc(CO)cc2)=O)C1 18583,c1(C(=O)NC2C(NC(c3ccc(C4OCCO4)cc3)=O)COC2)ncc(F)cn1 18584,Cc1cc(C(=O)NC(C2(CNC(c3sc(Cl)cc3Cl)=O)CC2)C)c(C)[nH]1 18585,c1(C(N2CC(C(=O)NCc3nn[nH]c3C(F)(F)F)C2)C)ccccc1F 18586,C1(N(C(=O)Nc2ccc(C)cc2C)CC)CCC(F)(F)CC1 18587,c1(NC(N2C(C3C(=O)CCCC3)CCC2)=O)cc(F)ccc1Br 18588,C1(F)(C(=O)NCCC2(CNC(C3CC=CCC3)=O)CC2)CC1(Cl)Cl 18589,C(=O)(C1CCCc2ncnn21)N1CCC(CC(=O)Nc2cnc(C)c(F)c2)C1 18590,C(=O)(CC(C)O)NCC(C)=CC(=O)NCc1nn[nH]n1 18591,c1(C(=O)NC(CC)CNC(c2ccc(C(C)C)cc2C)=O)c(C)nc(C)nc1C 18592,Cc1nccc(C(=O)NCC2(CNC(c3cnsc3C)=O)CCCCC2)c1N 18593,c1(C(=O)NC2C(NC(C(C)C#N)=O)C2)c(F)ccc(F)c1Cl 18594,c1(CCNC(=O)CCC2CCCN2C(=O)CC2CCC3CC23)cccnc1F 18595,N1(C(CC(C=C)(C)C)=O)CC2CN(c3ncc(C(=O)OC)cc3Cl)CC2C1 18596,c1(C(N(C(C)CNC(c2ccoc2C)=O)CC)=O)cc(Cl)n(C)n1 18597,N1(C(c2c(OC)csc2)=O)CCOCC1C(=O)Nc1cncc(C(F)(F)F)c1 18598,C1(CC(N2C(CNC(C(C)n3cccc3)=O)CCC2)=O)SC(=N)NC1=O 18599,C(CCC(C(=O)NC(C)(C)C(C)(C)CO)NC(=O)C(C)SC(C)C)OC 18600,C1(C(=O)NCCC2(C)CC2(F)F)(OC)CCN(C(c2nc(C)sc2C)=O)C1 18601,c1(C(C)NC(C2C(NC(c3ncc(C)s3)=O)C2)=O)ccc(F)c(F)c1 18602,C(CC(F)(F)F)SCC(=O)NC(C)CN(C(=O)C(F)n1cccn1)C 18603,c1(C(=O)NCC23CC(NC(C(c4ccccc4)OCC)=O)(C2)C3)cnn(C)c1F 18604,C1(C(N(C2CCCN(C(=O)CC3=NNC(=O)C3)C2)C)=O)CCCC12CCOCC2 18605,C1(NC(C(C)n2cncn2)=O)CCCC1NC(c1cnn(CCF)c1)=O 18606,C1(CNC(c2cc(C)[nH]n2)=O)CC2CC2N1C(=O)CC(F)(F)Cl 18607,C(CC(=O)NOCC1CC1)(C(F)(F)F)NC(C(CCC)=CCC)=O 18608,N1(C(CCCSC(C)(C)C)=O)CC2CC1C2CNC(C1C=CCCC1)=O 18609,c1(C(=O)NC(C2N(C(CCC=CC)=O)CCC2)C)nc(O)sc1C 18610,C(=O)(C(C)CC(N)=O)NC(CC=C)C(=O)NCC(=O)N(C)O 18611,C1(CN(C(C(CC)SC)=O)CC)CCN(C(c2c[nH]cc2Br)=O)CC1 18612,NS(=O)(=O)c1sccc1C(=O)N(CCNC(C1COCCO1)=O)C1CC1 18613,c1(C(=O)NCCCC(CCC)NC(=O)CNS(N)(=O)=O)cc(F)cc2nc[nH]c12 18614,C1(CC(N2C(CC(=O)NCC(COC)C)CC2)=O)CSCCO1 18615,c1(C(=O)NCC2OCCN(C(C(C(C)OC)O)=O)C2)ccc2c(n1)NCCO2 18616,c1(C(c2n(CCC)nnn2)NC(C(N)=O)C2CC2)ccc(C(F)F)cc1 18617,c1(NCCC=C=C)cc(=NCC2(OCCO)CCCCC2)[nH]cn1 18618,c1(C(N(CC(=O)NCCC(C=C)C)C2CC2)C)ccccc1C 18619,N1(C(Cc2cn(CC)nc2)=O)CCOC2(C1)CN(C(C1CC3CC3C1)=O)C2 18620,C1(CN(C(C(C=CCCC)O)=O)C)CN(C(=O)C=CCCCCC)CCO1 18621,c1(C(=O)NC2CCN(C(c3cn(CCC)nc3)=O)C(C)C2)ccc(C)c(C)c1N 18622,CC1CCC(CNC(c2cc(CNC(c3cc(C4CC4)[nH]n3)=O)cs2)=O)N1C 18623,C1(CNC(C(C)(C)OCC)=O)CCC(CN(C(=O)CCc2cn[nH]c2)C)CC1 18624,c1(CNC(CCN(C(=O)Cc2ccc[nH]2)CC#C)=O)cc(C)cnc1O 18625,N1(C(C(Br)=C(C)C)=O)CCCCC1CCNC(=O)C(n1ccc(C)n1)C 18626,N1(C(c2cc(OC)nn2C)=O)CC(C)N(C(c2cc(C)n(C)c2)=O)CC1C 18627,Cn1c(C(c2nnnn2C2COC2)NCCCc2ccccc2)ccc1Cl 18628,N1(C(c2c(C)nc(Br)s2)=O)CC2CCC(C1)N2C(c1ccc2c(c1)OCO2)=O 18629,c1(NC(C23CC(NC(=O)Cc4cncnc4)(C2)C3)=O)cc(N2CCCC2)ncn1 18630,C1(NC(C(CC#C)(C)C)=O)CC(C2CCN(C(c3c(N)sc(C)c3C)=O)C2)C1 18631,c1(NC(C2(F)CN(C(c3cc(Br)ccc3Cl)=O)C2)=O)cnc2ccc(F)cn12 18632,c1(C)cccc(Br)c1.n1(CC)nnnc1C(c1ccn(C2CC2)n1)NCCOC(=N)O 18633,N1(C(CSCCNC(c2cccn(C)c2=O)=O)=O)CC2(CC=CC2)C1 18634,N1(CC(=O)N(CCNC(C2CC2(F)Cl)=O)C2CC2)CCCCS1(=O)=O 18635,N1(C(c2scnc2C2CC2)=O)CC2CCC(C1)N2C(C1CCCC1O)=O 18636,C(=O)(C(F)(CNC(C1(CF)CCOCC1)=O)C(C)C)NC(C#C)CC(C)(C)C 18637,C1(C#N)(COC)CCCN(C(=O)CC(C)C(=O)NCC(=O)Nc2ccccc2)C1 18638,C1(NC(C2(C#C)CCC2)=O)CCN(C(c2cc(C(C)=O)c[nH]2)=O)CC1F 18639,C(=O)(CCCC(=O)N1CCCN(C(=O)CNC(=O)CCCCO)CC1)OC 18640,c1(C(=O)NC(C)C2CC2)cc2c(s1)CCN(C(=O)CN1CCCCC1=O)C2 18641,CC(O)C(C)(C)C(=O)NCC#CCNC(C1CC(O)CN1C(=O)OC(C)(C)C)=O 18642,C1(Cc2c(F)ccc(OC)c2)CCN(C(=O)CC(C)c2ccccc2)CCC1CO 18643,N1(C(CC2(CC)CCC2)=O)CC(C(=O)Nc2ccc(OC(C)C)nc2)CC(C)C1 18644,C1(C(=O)NC(Cn2cc(-c3c(C)nn(C)c3C)nn2)C)Cc2cncn2C(=O)N1 18645,c1(OC)cccc(NC(C2(C)CCN2C(c2cccnc2O)=O)=O)c1 18646,C1(NC(CCC#C)=O)COC2(CNC(c3cc(Cl)sc3Cl)=O)CC1C2 18647,C1(NC(C2CN(S(CC)(=O)=O)C2)=O)CC(F)CN(C(c2csc(C(F)F)n2)=O)C1 18648,C1(NC(c2n(CC)ccc2)=O)C2COCC1CN(C(c1ncc(F)cc1C)=O)C2 18649,Cc1ccc(Cl)c(C(=O)NCCN(CC(C)O)C(=O)CN2CCC2C)c1 18650,C1(CC(C)NC(=O)CC2(C)CC2(F)Cl)CCN(C(C2(O)CCCCC2)=O)CC1 18651,c1(OC)ccc(N)c(C(N2CCC(NC(C3CC3(C)C)=O)C2(C)C)=O)c1 18652,c1(C(=O)OC2CCS(=O)(=O)CC2)cc(Br)cc2c1CCN2 18653,c1(C(=O)NC(C(C)C)CNC(=O)COCP(C)(C)=O)ccc(F)c(Cl)c1N 18654,CN1CC(F)CC1C(=O)NCC1CCC(C(=O)NCC2(O)CCCC2)O1 18655,CC1(C)OCCCC1C(=O)NCC1CN(Cc2ccccc2)CCCO1 18656,N1(C(CSC)=O)CC(NC(=O)Cn2nc(C)c3cccnc23)C2CCCCC12 18657,c1(C(C(=O)N(C2CN(C(=O)CC3CCCC(O)C3)C2)C)(C)C)cccc(C#N)c1 18658,C1(NC(C(C(C)(C)O)F)=O)CC(C2CCN(C(=O)CCc3nc(=N)[nH][nH]3)CC2)C1 18659,C12(CC(=O)N(C3CCCC3)CCNC(C(C)O)=O)CC3CC(C1)CC(O)(C3)C2 18660,c1(NC2CCC2)ccc(C(=O)NC2C(NC(C(C3CC3)OCC)=O)CC2)nc1 18661,CN1CC(C)(C(N2CC(N(C)C(c3cc(C4CC4)ns3)=O)C3(CC3)C2)=O)CC1=O 18662,C(=O)(C(CC(C)(C)C)NC(=O)OC(C)(C)C)Nc1ccc(C(C)O)cc1 18663,C(C(C)C(=O)NC(C)CNC(c1cnc(-c2ccoc2)s1)=O)OC 18664,c1(CC)cccc(C)c1C(N1CCCC(O)(CCNC(=O)CC2CC2(Cl)Cl)C1)=O 18665,CC(CC(=O)NCC1(C(=O)NCC2CC2CO)CC=CC1)C1CC1 18666,C1(NC(c2cn(CC3CC3)nn2)=O)CCCN(C(c2ccc(Cl)nc2)=O)CC1 18667,Cc1cc(C#N)nc(N2CCC(CNC(=O)CCc3ccc(O)nc3)C(C)C2)n1 18668,c1(C(=O)NCC(c2ccccc2Cl)N(CC)CC)ccc2c(c1)CC(=O)N2 18669,c1(CC)cc(C(N2CCC2CNC(C2(F)C(C)(C)C2(C)C)=O)=O)cn(C)c1=O 18670,c1(C(N2C(CC(=O)Nc3ccc(C)c(F)c3)COCC2)=O)c(O)cc(O)cc1O 18671,Cc1cc(-c2ccnc(NC(c3ccccc3N(C)C(C)C)=O)c2)ccc1F 18672,N1(C(Cc2c(C)cccc2)=O)C2CCCC1CN(C(C1CCN(C)C1)=O)C2 18673,n1(CC)cc(Cl)cc1C(N1CC(CCNC(c2ccc(C#N)[nH]2)=O)C1)=O 18674,N1(C(C2(CC)CCC2)=O)CC2(CCN(Cc3nnc(C(C)C)s3)C2)C1 18675,C1(C(=O)NCCCc2c(C)n[nH]c2)CCN(C(c2[nH]nnc2C(F)F)=O)CC1O 18676,C1(C)(C(=O)NCC2(NC(C3CCCN(C)C3)=O)CC2)Cc2ccccc2C(=O)O1 18677,c1(C(N(CC(C)N(C(=O)C=Cc2cccnc2)C)C)=O)ccc(=N)[nH]c1 18678,C1(=CC(CC)C)CCN(CCC#N)CC1.C12CCC(CC1)C(=O)N2C1CC1 18679,C(=O)(NNc1ccc(F)nn1)C1CN(C)C(=O)CC1 18680,N1(CC)CCC(C(N2CCC(N(C(=O)CNC(c3ccncc3)=O)CC)C2)=O)C1 18681,C1(NC(COCCC=C)=O)CC2(CCN(C(=O)C=Cc3cnccn3)C2)C1 18682,CCC(C)(CCNC(=O)CCCn1ccnc1)NC(=O)C(C)n1ccnc1 18683,c1(C(N(C(C)CNC(=O)CC(c2ccc(Cl)cc2)O)CC)=O)ncccc1Cl 18684,c1(OCC)ccc(F)c(F)c1-c1cncc(C(N2CCC(OC)C2)=O)n1 18685,C1(CNC(C2CCS(=O)(=O)CC2)=O)CC2CCC(C1)N2C(C1CCOC1)=O 18686,C1(OC)CN(C)C(C)(C(N2CCCCC(CNC(C3(O)CCCCC3)=O)C2)=O)C1 18687,C1(CNC(c2c(C)n(C3CC3)cc2)=O)CN(C(=O)CC(C)CN(C)C)CCCO1 18688,N1(C(C(COC)OC)=O)CC(NC(c2ccc(OC)c(Br)c2)=O)CC1(C)C 18689,Cc1cnccc1C(C)C(=O)N1CC(c2cn(CCN3CCC(F)(F)C3)nn2)C1 18690,C#CCC(C)(C)C(=O)N1CCC(C)C(NC(c2cncc(C(C)C)c2)=O)C1 18691,c1(C(N2C(C)CCC(NC(=O)CC3CCOC3)C2)=O)cccc2c1OCCCO2 18692,c1(OC)ccnc(C(=O)NC2CCCCC2NC(=O)C(O)CN2CCCC2)c1N 18693,C12(C(N3CCC(CN(C)C(C4CCCN4C)=O)CC3)=O)CC(C)(C1)OC21CCC1 18694,OC1COc2c(NCc3cc(Cl)sc3Cl)cnn2C1 18695,C#CCCCCCC(=O)N1CCC(N(C(c2cc(CO)[nH]n2)=O)CC)CC1 18696,c1(C(N(CCCNC(C2CCN(CC(C)C)C2)=O)C)=O)cc(Cl)cc2c1OCC2 18697,C#Cc1cccc(CC(=O)NC2CCOC2C(N2CCNC(=O)C2CCO)=O)c1 18698,C1(CNC(C2N(C)CCCC2)=O)CC2(CCC2)CN1C(=O)C(O)Cc1cnc[nH]1 18699,Cc1ccnc(CNC(=O)C(C2CC2)N(C(=O)C(C)C(C)C)C)n1 18700,C=C(Br)CCC(=O)N1CCCCC1CN(C(=O)Cn1nnc(C)n1)C 18701,c1(C(N(CC(=O)NC2(CC(=O)OC)CC2)C(C)C)=O)nnnn1C 18702,C=CCCCC(C)(C)C(=O)N1CCC(NC(c2ccc(C)c(Br)c2C)=O)CC1 18703,C=CCN=C(NCC(c1ccc(N2CCCC2)nc1)O)NCC(C)F 18704,N1(CC2(NC(CCOC)=O)CC2)CCN(C(C2OCCOC2C)=O)CC1 18705,c1(N(CC(CN(C)C)(C)C)C)nc(N2CCC(C)(C)C2)nc2c1cnn2C 18706,C(=O)(C(C)(C)CC(=O)OC)NCC(CC=C)C(=O)Nc1ccc(Cl)cc1 18707,n1(C(C#C)C2CCC2)cnc2c(N3CC(N(C)C(C)=O)C3)ncnc12 18708,c1(C(N2C(CNC(C(C)NS(C)(=O)=O)=O)CC2)=O)ccc(C2CC2)cc1F 18709,CC#CC1CCN(C(=O)C(C)=CCNC(C2CCN2C(C)(C)C)=O)C1 18710,C#Cc1ccc(C(=O)NCC2(NC(c3ccsc3COC)=O)CC2)cc1Cl 18711,c1(C(=O)NCCOCCNC(C(C)SCC)=O)ccc2cn(C)nc2c1 18712,c1(CC(=O)NC2CCN(C(c3cc4ccccc4s3)=O)C2)ccc2nc[nH]c2c1 18713,CC(C)CC(C)CC(C)C(=O)NC1(CNC(=O)CN2C(=O)CNC2=O)CCCC1 18714,C(=O)(N(CCC(=O)OC)OC)C12C(CN(C(c3n(C=C)nnc3)=O)C1)CCC2 18715,c1(C(N(CCCN(C)C(C2(O)CCOC2)=O)C)=O)cccc(O)c1F 18716,Cc1ccc2oc(C(=O)NC3CC(CNC(c4cc[n+]([O-])cc4)=O)C3)cc2n1 18717,c1(C(=O)NC(CNC(C2(SC)CCC2)=O)C2CC2)cnc([N+](=O)[O-])n1C 18718,C(C(CNC(C1(c2cc(C)no2)CC1)=O)C(F)(F)F)NC(C(COC)(F)F)=O 18719,C(=O)(C#CC1(C)CCCO1)N(C(C)CNC(=O)Cc1cnn(C)n1)C 18720,CC1=NC(C)(CNC(=O)CC2CCCN2C(=O)C(n2ccnc2C)C)CS1 18721,C1(O)(COC)CCN(C(=O)CCOCCCNC(c2occc2C2CC2)=O)C1 18722,N1(C(C(=O)NCc2cn(CCN(CCO)CC)nn2)C)CCN(C)CC1 18723,CC(C(=O)OC(C)(C)C)C(=O)N(C)CCN(C(=O)CCc1cncn1C)C(C)=O 18724,N1(C(C2(CC=C)COC2)=O)CCCC(CC)(NC(=O)Cn2ccc([N+](=O)[O-])n2)C1 18725,C1(C(=O)NC(C2N(C(C(CSC)O)=O)CCC2)C)CC2CCC1CC2 18726,N1(C(c2c(COC)ccs2)=O)CCCCC2(CCN(C(c3cnc[nH]3)=O)C2)C1 18727,N1(C(c2ncc(OC)cn2)=O)CCC(NC(c2cc(C)c[nH]2)=O)C(C)(C)C1 18728,c1(CCCC(=O)NCCCCN(C(C=CC(=O)N(C)C)=O)C)cc(F)ccc1F 18729,C1(C(N)=O)CNC(=O)CN1C(=O)COC1CCN(C(C2CC23CC3)=O)C1 18730,C1(OC)CC2(C1)CN(C(=O)C(CNC(c1ncccn1)=O)C(C)C)C2 18731,C1(NCCCN2CCC(C)CC2)Cc2nccnc2C1 18732,C1(SC)CC(CC(=O)NCCN(C(=O)C(C)C2CCCC2)CC(C)O)C1 18733,N1(C(Cc2ncn(C)c2)=O)CC(C(=O)NC(c2nc[nH]n2)C2CC2)C2(CC2)C1 18734,O=C(C(C(F)(F)F)C(F)(F)F)NC1C2CC1N(C(c1cc(C3CCC3)n[nH]1)=O)C2 18735,C(=O)(C1=CCC(C)CC1)NCC1OCCN(C(CCc2ccc(OC)cc2)=O)C1 18736,Nc1cccc(C2CN(C(C3CCOC(c4ccc(F)cc4)C3)=O)C2)c1 18737,C1(NC(CCC)=O)CCC12CN(C(=O)CCC(c1ccccc1)N(C)C)C2 18738,Cc1ncc(NC(C2CN(C(c3cncc(Cl)c3)=O)CCN2)=O)c(C)c1Br 18739,N1(C(c2c(OC)csc2)=O)CCOCC(NC(c2cc(F)cnc2Cl)=O)C1 18740,Nc1c(C(=O)NCC2CCCCN2C(=O)C(O)C2CCC2)ccnc1Br 18741,CC1=CCC(C(=O)NCC2CC2NC(c2ccc(NC3CC3)nc2)=O)CC1 18742,c1(CNC(C2CC(C)C2)=O)cc(O)nc(CNC(c2ccc(C(F)F)s2)=O)n1 18743,C(C(C)(C)C(=O)N1CCC(O)(C(F)F)C1)NC(c1ncn(C(C)C)n1)=O 18744,C1(C(=O)NCC2(COC)C=CCC2)Cc2ccccc2CN1C(=O)CNC=O 18745,Cc1cc(C#N)ccc1C(N1CCC2(CC2NC(C2CC3(CC(=O)C3)C2)=O)C1)=O 18746,CCCCCCCCC(C)CC(=O)NCc1ccc(OC)cc1 18747,C=C(C)CC(C(=O)OC)N(C)C(c1cc(C)nn1C1CCS(=O)(=O)C1)=O 18748,C1(CC)CCC(N(C(=O)CC2(OC(C)=O)CN(C(=O)C(C(C)C)OC)C2)C)CC1 18749,C(=O)(C(C)CCCC(C)=O)N1C(CNC(c2ccn(CC)n2)=O)CCC1 18750,N1(C(COC2CCC(C)CC2)=O)CCC(O)(c2cn(C3CCC3)nn2)CC1 18751,N#Cc1cc(NC(=O)NCC23CC(CCO2)C3)co1 18752,c1(OC)ncccc1C(C)NC(c1nnnn1C)C1CCC1 18753,c1(CCC(=O)NC(CC)CNC(=O)CN2CSCC2=O)cccc(F)c1Cl 18754,N1(C(C(c2cccnc2)C)=O)CCC2CC(CNC(=O)CCF)CCC2C1 18755,C1(CC(C)C)CC(C(=O)NCCCNC(c2cc(=O)cc[nH]2)=O)CC(=O)N1 18756,C1(C(N(CCCO)CC)=O)(CC)CN(C(=O)C(c2csc(C)n2)=O)C1 18757,N1(C(c2cc(OC)c(F)cc2)=O)C2CCCC1CC(NC(C1CC1C(C)O)=O)C2 18758,c1(CN2C(C(=O)OC)(CC)CCC2)cc2nccc(Cl)c2s1 18759,N1(C(=O)NC(Cc2cccc(C)c2)C2CC2)CCCC(O)(c2cnn[nH]2)C1 18760,C12(C(=O)NC(CC)CNC(=O)COCC3CCOC3)CSC(C1)C2 18761,c1(CC)nccnc1C(=O)NCC1CCN1C(=O)C(=CC1CCCC1)C 18762,C(=O)(C(CNC(=O)Cc1nocc1C)CC(C)C)NCC(CSC)OC 18763,CC1(C)CCCCC1C(=O)N(C1CC(C#N)C1)CC(=O)NCC(C)(C)CO 18764,N1(C(CCCNC(C)=O)=O)CC2(COC(CNC(=O)C(F)CC3CCC3)C2)C1 18765,S(=O)(=O)(c1ccc(C(=O)N(CC(F)(F)F)C2CCC2)cc1)N1CC(C)CC(C)C1 18766,c1(NCC(C)(C)NC(Cc2ccc(OC)cc2)=O)ccc(C#N)cc1[N+](=O)[O-] 18767,C1(NC(CCNS(CC)(=O)=O)=O)CC2CC1N(C(C1(O)CCOC1)=O)C2 18768,C12(NC(CCc3ccnc(C)n3)=O)CCCC1N(C(=O)COCC(F)F)CCC2 18769,Cc1cc(Cl)cc(C(=O)NCC2(NC(C3CC(O)C3)=O)CCCC2)c1C 18770,C=CC(CCC)CC(=O)N1CC(C(=O)NCC2CCOC(C)(C)C2)C(F)(F)C1 18771,c1(OC)cc(C)ccc1C(N1CCCC(CNC(c2cc(Cl)c[nH]2)=O)CC1)=O 18772,C1(CNC(c2cccc(CC)c2)=O)COCCN(C(=O)CCOCC2CCC2)C1 18773,c1(C(=O)NCC(O)CNC(C2CC2C2CCC2)=O)ccc2ccc(Br)cc2c1 18774,c1(C(=O)NCC(CCCC)NC(=O)C(C)CF)ccc2n[nH]c(C)c2c1 18775,N1(C(C(CC(C)C)ONC(C2COCC2C(N)=O)=O)=O)CCC2CCCC2C1 18776,c1(-c2cn(CCS(C)(=O)=O)nn2)cc(C#N)ccn1.C12CCC(CC1)CC(=O)N2 18777,C1(NC(CC2CCN(C(C(C)O)=O)CC2)=O)CCN(C)C12CCC2 18778,c1(NCC)ccc(C(N2CC(CCNC(=O)CCC3CNC(=O)N3)C2)=O)c(Cl)c1 18779,C1(C(N(C)CC2C(C)C2)=O)N(C(c2coc(N(C)C)n2)=O)CC12CCCC2 18780,CCC(CC(=O)N(C1CN(C(C2CC=CCO2)=O)CCC1O)C)C(C)C 18781,C(C)(N=c1[nH]c(N2CCC3(CCN(C)C3)C2)nc2ncn(C)c12)c1nc(C)sc1 18782,Cc1nnn(CC(=O)NC(C2CCCCC2)C(=O)NCCC(N)=O)n1 18783,c1(CC)cc(C(=O)NC(CC)CC(=O)NCC2COCC2(C)C)ccn1 18784,C1(F)(C(N2CCCC(N(C(=O)CC(C)(C)O)C)C2)=O)CCC(F)(F)CC1 18785,C1(CNC(CCSC)=O)CC2(CCN(C(c3cc(C(F)F)ccn3)=O)CC2)CO1 18786,C(=O)(CCCS(C)(=O)=O)N1CCN(C(C(C)NC(=O)NC)=O)C(C)C1 18787,c1(C(=O)NC(C2CCN(C(=O)CCc3ncc[nH]3)CC2)C)cc(Cl)cnc1O 18788,CCC(CCCC(=O)N(CC1CCC1)CC1CC1)NC(c1cc(C)cc(C)c1)=O 18789,c1(C(=O)OC)cnc(NC(C2CC23CN(Cc2ccc(F)c(Cl)c2)C3)=O)c(Cl)c1 18790,N1(C(N)=O)CCC(NC(=O)C(C2(O)CCC2)NC(C23CSCC2C3)=O)C1 18791,Cc1c(CC(=O)NCCCOCCNC(=O)C2=NNC(=O)C2)cccc1Br 18792,CCC(C)(C)C(=O)N1CCCC(C(=O)Nc2cccc(CNC(=O)C=CC)c2)C1 18793,N12CCCC(O)(C1)C1C(SC)CN(C1)C2=O.C(C)(C)(C)SN.C(C)C 18794,N1(C(c2ccoc2Cl)=O)CCC(N(c2ncnc(C(C)(C)C)n2)CC)CC1 18795,N1(C(c2cc(C)cc(C)n2)=O)CC(C)CN(C(C2CCCCN2C)=O)C(C)C1 18796,n1(CCC)cc(C(=O)N(CCCOCCNC(=O)CC2CCN(C)C2)C)cn1 18797,c1(CC(=O)NC2CC(C)N(C(c3cccn(O)c3=O)=O)C2)c(F)cccc1F 18798,N1(C(=O)C(c2ccc(F)c(F)c2F)O)CC2CCCC(O)C2C1 18799,O=C(C1=CCCOC1)NC(CO)C(=O)NCC1CCCCCC1 18800,CC1CCC(C)(C(=O)NCCNC(c2ccnc(Oc3ccccc3F)c2)=O)C1 18801,N1(C(C#C)C)CCN(C(=O)C(CCF)NC(c2cnncc2C)=O)CC1 18802,C(=O)(Nn1cccc1)C1C(C(=O)OC)C1 18803,c1(C(C(C)C(=O)NCC2CC2)=O)cc(CCP(C)(C)=O)[nH]n1.C12(CC1)CNC(=O)N2 18804,Cc1cccc(C(=O)NCCCCCC(=O)NC(c2cn(C)cn2)C)c1N 18805,N1(C(c2c(CNC(c3n(C=C)nnc3)=O)noc2)=O)CCC2C(CCN2C)C1 18806,N#Cc1cc(C(=O)NCCN2CCN(C(=O)C(O)C3CCC3)CC2)c[nH]1 18807,C1(C(=O)NCC(C)NC(C2(Cc3cnn[nH]3)CCC2)=O)CCSC(C)C1 18808,C1(F)(CNC(c2ccnc(O)c2)=O)COCCN(C(=O)C(O)c2cnc[nH]2)C1 18809,Cc1cc(C)c(C(=O)NC(Cc2ccoc2)C(=O)NCc2ccc(C#N)s2)s1 18810,C1(C(C)C)N(C(=O)Cn2nc(C3CC3)n(C)c2=O)CC12CCN(CC1CC1)CC2 18811,N1(C(CC(CCC)(C)C)=O)Cc2cccc(CNC(=O)C(COC)CC)c2C1 18812,N1(C(Cc2scc(C)c2)=O)CCC(CF)(NC(=O)C(C(C)C)n2cnnn2)C1 18813,C1(C(=O)NCC2C(Cn3cc(COCC4CC4)nn3)C2(F)F)CCCC1C1CC1 18814,c1(C(N)=O)ccc(C=CC(=O)NC2CCN(C(=O)CSC3CC3)C2C2CC2)o1 18815,C(=O)(C1=CCOCC1)NCC(C)OC.c12cccnc1C(=O)N1CCN(CC1)C2 18816,C(=O)(CC(C(F)F)C(C)(C)C)N1CCC(CCNC(C(CCC2(C)N=N2)O)=O)C1 18817,Cc1cc(Cl)cc(C(N2CCCC2CNC(c2ncnn2C)=O)=O)c1O 18818,Cc1cc(NC2CNC3(CCCC3)C2)c(C#N)cc1N1CCOCC1 18819,C1(C(=O)NCc2n(CC)ncn2)CC=CC(NC(=O)C(C(C)C)SC)C1 18820,C1(NC(CSCC)=O)CCCCC12CCN(c1nc(Cl)nc(C)c1Cl)C2 18821,c1(CCC(=O)NC2CN(C(=O)CCc3ccoc3)C2)cccc(F)c1 18822,c1(C(=O)NCC(CCOC)NC(=O)CN(C)C(N)=O)cnc2c(c1)nc(O)n2C 18823,c1(C(=O)OC)ccc(CC(C)C)nc1N1CC2CC(NC(=O)CC3CC3C)C2C1 18824,c1(C(=O)NCCCCC2CN(C(C3C(C)CC3)=O)C2)cc(Cl)ccn1 18825,N1(C(c2c(C(C)=O)cn(C)n2)=O)CC2CC(N(C(=O)CCC=C(C)C)C)C1C2 18826,c1(OC)ccc(-c2ccnc(C(N3CCC(F)(c4cn(CCO)nn4)C3)=O)n2)cc1 18827,c1(C(=O)NC(CC)CNC(c2csc(C)n2)=O)sc2ccccc2c1Cl 18828,c1(C(N(C(C)CNC(c2cccc(SC(F)(F)F)c2)=O)CC)=O)cc(C)n(C)c1 18829,CC1=NS(=O)(=O)NC=C1C(=O)N1CC(NC(=O)C2=CC(C)(C)C2)CCC1C 18830,c1(C(=O)NC(C(C)C)CCNC(C2(N(C)C)CC2)=O)nn(C)c(C(F)(F)F)c1Cl 18831,C1(C(=O)NCC2CCN(C(c3c(CC)c[nH]n3)=O)C2)C2CCCCC12 18832,c1(NCC2CC(O)C23CCC3)nccc(=NCCOCC(F)F)[nH]1 18833,C(=O)(CCCCCCCC1CC1)N1C(CNC(c2cn(C)c(=O)cc2)=O)CCC1 18834,c1(C(=O)OC(c2cccc(C#N)c2)C)ccnc(Cl)c1N 18835,c1(NC(C2CCN(C(c3cc(CC)[nH]n3)=O)CC2)=O)ccc2ccncc2c1 18836,N1(c2ncc(C(=O)OCC)s2)CCCC2(CC(NC(=O)C(C)c3ccco3)C2)C1 18837,C1(NC(CSC)=O)CC2CC(NC(c3ccc(C(N)=O)nc3)=O)CC12 18838,c1(C(=O)NCC2CC(SC)C2)c(CNC(=O)CCC2CCCC2)cnn1C 18839,C=CCCCC(=O)N(C1CCC(NC(C2(COC)C=CCC2)=O)CC1)C 18840,c1(C(N(CC(CC)NC(C(CC)C)=O)C)=O)nn2cccnc2c1Cl 18841,C(=O)(C(C)CC(F)F)NC(C(=O)NCC1(OCC)CCC1)Cc1ccoc1 18842,N1(C(C2C(OC)CCC2)=O)CCc2[nH]nc(CNC(=O)CC3(OC)CC3)c2C1 18843,C1(NC(=O)C=CC=C(Cl)Cl)CN(C(c2cnc3n2CCC3)=O)CC12CCC2 18844,Cc1csc2ncnc(N3CCC(C)(C)C(CNC(=O)C(C)S(N)(=O)=O)C3)c12 18845,C(=O)(CC(c1ccccc1)OCC)NC1CC(NC(C2(COC)COC2)=O)C1.OCC 18846,C1(C(=O)NCCNC(c2cc(F)cc(N)c2F)=O)(CC)CCC(F)(F)CC1 18847,N1(C(c2c(OC)cccn2)=O)CCC2(CC1)CC(CNC(C1CCCO1)=O)C2 18848,CCCC(C)CC(=O)NC(C)CN(C(c1ccncc1C1CC1)=O)CC 18849,c1(C(=O)NC2CC(CNC(c3c(OC)ccnc3)=O)C2)ccc2ncccc2n1 18850,CCN=c1cc(-c2nc(C(C)Oc3ccccc3)n(-c3cccnc3)n2)cc[nH]1 18851,c1(N(C)C)cccc2sc(C(=O)NC3Cc4ccccc4CO3)cc12 18852,Nc1nc2ncccc2cc1C(=O)NC1(CO)CCN(C(=O)CC2CCCC2)C1 18853,N1(c2nc(N3CCN(CCS(C)=O)CC3)cc(C)n2)CCc2oc(C)nc2C1 18854,Cc1nc2cccc(C(=O)NCC(C)(C)CCc3nn[nH]n3)c2[nH]1 18855,c1(C(N)=O)cccc(C(N2CCOCC2CC(=O)NCC(F)(F)F)=O)c1F 18856,N1(C(C(C2(O)CCCC2)OC(C)(C)C)=O)CCSC12CC(C(=O)O)C2 18857,S(=O)(=O)(c1ccc(N(C)CCN2CCOC2=O)c(Br)c1)N(C(C)CS(C)=O)C 18858,CC1CC(NC(=O)NNC(=O)c2cn(C)nn2)CCN1C 18859,S(=O)(=O)(CCC(F)(F)F)N(C(CC1(C)CN(CCCl)C1)=O)C(c1ccccc1)C#N 18860,N1(C(CC2C(CC)CC2)=O)CCN(CCSc2ccc(NC(C)=O)cc2)CC1 18861,c1(C(=O)NC2(CCNC(Cc3nc(C)sc3C)=O)CC2)cc(N)cnc1C 18862,C(CC(C(=O)N1CCC(NC(=O)CC2CCCC23CC3)C1)OC)OC 18863,C1(NCc2cnc(CCCC)[nH]2)CCN(C2CNC2)C1=O 18864,C(CC(=O)N1CCN(C(=O)CNC(=O)CC(C)F)CC1)(C(F)(F)F)OC 18865,Cc1nsc(NC2CC2)c1C(=O)NC1CCCCC1CNC(=O)OC(C)(C)C 18866,C(=O)(C1=NNC(=O)CC1)N1CCCC(C(=O)NCc2nccc(C)c2)C1 18867,c1(CC(=O)NCC(CC)(CC)NC(c2ccc(CO)nc2)=O)ccc(O)cc1Cl 18868,C1(O)(C(=O)NCC2CC(NC(COC(CC)C)=O)C2)CCCC1 18869,C(=O)(C1=CC2(CN(C(=O)CC3CCCC(O)C3)C2)OC1)NC(c1ccnn1C)C 18870,c1(NC(C2CC(O)(CC)C2)=O)ccccc1C(C1CC1)OC 18871,CC1(C)COc2ccc(C(=O)NCCC3(O)CN(C(=O)C4=CCCC4)C3)cc21 18872,N(C1CCCc2ccc(F)cc21)C(=O)NNC(=O)c1ccc(O)nn1 18873,C(=O)(C(C)CC(F)(F)F)NCC1(C(=O)NCCCNC(C(C)C)=O)CCCO1 18874,C1(NC(C2CCC(CC)CC2)=O)CC2CC(C1)N(C(=O)CCCCC(=O)NC)C2 18875,c1(OC)ccc(C(c2ccc(C)s2)NC(Cc2ccccc2)C2CC2)cc1Br 18876,c1(C(=O)NC23CC(C(=O)NC4CC(C)OC4=O)(C2)C3)cn(C)c(=O)cn1 18877,c1(C(=O)NC(C(C)NC(=O)CSCC(N)=O)C)ncc(F)c2ccccc12 18878,C1(CNC(C2CCCO2)=O)CCCN1c1ccncn1 18879,c1(OC)cc(CC(=O)NC2CCN(C(=O)COCCSC)C2C)ccc1O 18880,C(=O)(C#CC1(C)CCCO1)N(C1CCN(C(=O)C2=NOCC2)CC1)CC 18881,c1(NC(=O)COCCC)cc(CN(C(=O)C(F)CC2CC2)CCC)ccc1F 18882,N1(c2cc(NCc3cnc(C)o3)nc(C)n2)CCOC(C2CCCO2)C1 18883,c1(C(=O)NCC(C)CC(=O)NCC2CC3C=CC2CC3)ccc2n[nH]cc2c1 18884,N1(C(CNCCC=C)=O)CCc2ccccc2C1CCNC(=O)COCC1CC1 18885,c1(C(=O)NCc2c(CCNC(C(C)OCCC#C)=O)ocn2)cc(C)c(C)o1 18886,Cc1ccc(F)c(O)c1C(N1CC2CC(NC(C3CCCCC3)=O)CC2C1)=O 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18973,Cc1ccn(C)c(=O)c1NC(C1CC(C)N1C(=O)CCc1cnn[nH]1)=O 18974,C1(C(=O)NC(C(C)NC(=O)CSCC(N)=O)C)(CF)CCOCC1 18975,c1(OC)cc(C#N)ccc1NC(C1(C)CCN1C(c1cnc2[nH]ncc2c1)=O)=O 18976,CC(C)(O)CC(=O)NCCC1(C(=O)NCCCc2cccnc2)CCC1 18977,c1(C(=O)NCCC#C)cnc2ccc(-c3ccc([N+](=O)[O-])c(F)c3)cn12 18978,C1(NC(C=C(C)Cl)=O)CC(CNC(c2cc(-c3cnn(C)c3)no2)=O)C12CCC2 18979,C1(CC)(NC(=O)CC(C2CC2)NC(C2CC2[N+](=O)[O-])=O)CCOC1 18980,Cc1ccc(C)c(C2=NOC(C(=O)NCC#CCNC(C34CC(O)C3C4)=O)C2)c1 18981,c1(C(N(C)Cc2c(C)ccc(C)c2)=O)cccc([N+](=O)[O-])c1N1CCOCC1 18982,C1(=CC(=O)NC(CC(C)NC(=O)COC2(C)CCC2)C)CCC(C)(C)CC1 18983,c1(-c2nnc(CN(C(c3cccnc3)=O)CC)o2)ccc(C)cc1 18984,C1(C(C)C)(C(=O)NCC2(C)CCN(C)C2)CCCN1C(c1ccc(F)cn1)=O 18985,CC(C)CC(C(N)=O)NC(=O)CC(CNC(C1CC2CC(=O)C1O2)=O)C1CCC1 18986,C1(C(=O)NCC(O)C(C)(C)O)(NC(C(c2cncnc2)C)=O)CCN(C)C1 18987,Cc1cc(C(=O)NCC(C)(C(C)C)NC(c2ncn(C)n2)=O)n(C(C)C)n1 18988,C1(C(N(CCC(=O)N(CC(CC)C)C)C)=O)CCC2CC12 18989,C1(CCNC(CCCOC)=O)CN(C(c2ccc(C(F)F)cc2)=O)CC(C)O1 18990,C(=O)(C(F)(F)C(F)F)N(CCN(C)C(C1CC1c1ccc(F)cc1F)=O)C 18991,c1(C2(C(N(CCCNC(C(CC)C)=O)CC)=O)CCOCC2)ccc(Cl)cc1Cl 18992,C(CCCCCCC(=O)NC(CO)C(C)NC(c1nc(C)oc1C)=O)SC 18993,CCC(CC(=O)N1CC(C(N)=O)C1)NC(=O)Cc1ccc(C)cc1 18994,CCC(C)(C#N)C(=O)N(CCCCN(C)C(C1C(C)C1(F)F)=O)C 18995,N1(C(CCC(C(C)C)NC(=O)Cc2cc[nH]c2)=O)Cc2cccc(F)c2C1 18996,C1(NC(CCOC)=O)(CNC(=O)CSCc2cccc(Cl)c2)CCOCC1 18997,CCC(O)CC(=O)NCC(C)NC(C1(NC(C)=O)CCC1)=O 18998,c1(C(=O)NCC(CNC(C(C)NC(COC)=O)=O)F)ccc(=O)n(CCF)n1 18999,N1(C(COCCCCCC)=O)CC2(C1)CN(C(c1cc(O)cc(F)c1)=O)CCO2 19000,n1(CCNC(c2cc(CO)on2)=O)cc(C(=O)NC2CCOC2)nn1 19001,c1(CN2CCCC(CNC(C(c3cccc(C)c3)=O)=O)C2)cccc2nsnc12 19002,C(C(O)C(=O)NCCCC1CCCN1C(c1cc(-c2ccoc2)[nH]n1)=O)SC 19003,C1(CC(=O)NCC(N2CCOCC2)C)(OC)CN(C(=O)C=C2CCOCC2)C1 19004,c1(CC(=O)NC23CC2CN(C(C2CCOCC2)=O)C3)c(F)cccc1Cl 19005,c1(CC(C)C)ccc(NC(C2(F)CCN(C(C3CCO3)=O)C2)=O)cn1 19006,c1(C(N(CCN(C(C(F)=CCC)=O)C)C)=O)ccc(-c2nnnn2CC)cc1 19007,N1(C(CC2N(C(C3C(C)(C)OCC3)=O)CC(O)C2)=O)CCC2(CCC(O)C2)C1 19008,c1(C(C)C)cnc(O)c(C(N2CCC(C(C)NC(c3cncc(N)n3)=O)C2)=O)c1 19009,C1(C(N2CC(CNC(C(CC)(C)O)=O)(COC)C2)=O)CC(C)CC(=O)N1 19010,c1(C(=O)NCCC2CSCCN2C(=O)CC2CSCCS2)cccn2ncnc12 19011,Cn1cc(I)c(C(N2CCCC(C3(C)OCCO3)C2)C(=O)NCC(F)F)n1 19012,c1(C(=O)NC(C)CCNC(c2cc(O)n(C)n2)=O)cnn2cc[nH]c12 19013,CC1CN(C)CCC1NC(C1CC2(CCC2)CO1)=O.C12(CC1)N(C)C2=O 19014,c1(C(=O)NCCC2CCCN(C(=O)CC(F)(F)F)C2)ccn2ccsc12 19015,N1(C(c2c(C)nccc2)C(=O)NCCCC2CC2)CC(C)(C)c2ccc(Cl)cc21 19016,C1(NC(C)=O)CCCN(C(c2ccnc(N3CCOCC3)c2)=O)CC1F 19017,C1(NC(c2cccc(NC(C(=O)NC3CCC3)=O)c2)=O)CC2CCCN2C1 19018,c1(C(=O)NCC2CCCC(NC(C=CCOC)=O)C2)cc2oc(C)cc2[nH]1 19019,N1(C(CC2(C#N)CCC2)=O)CC(NC(=O)CCCC2CC2)C2(CCOCC2)C1 19020,CC(O)CCCC(=O)N1CCCC1C(C)(C)NC(c1cnccc1Cl)=O 19021,c1(N(C(=O)C(c2ccccc2)C)CC(Br)=C(C)C)ccc(F)cc1F 19022,C1(CCNC(C(CC)=CC)=O)CCN(C(c2cn(C)c(=O)n2C)=O)CC1(F)F 19023,CCCCC(=O)C(=O)N1CCN(CC(=O)NC2CC3CCCC3C2)CC1 19024,C(=O)(C(C)CC(F)F)NCC(C(=O)N(CCC#C)C)O 19025,N1(C(CCC(=O)NC)=O)CCOC2(C1)CN(C(c1onc(Br)c1C)=O)C2 19026,N1(C(C2C(=C)C2)=O)CCN(C(c2ccoc2CC(=O)OC)=O)CC1CC(=O)NC 19027,N1(C(c2cccc(SCC)c2)=O)CC2CCN(C(C34CC(CO3)C4)=O)C2C1 19028,N1(C(c2ccc(C)s2)=O)CCN(C)C(C2CC2)C1.C12CCOC1C(=O)N2 19029,C1(NC(C=Cc2nc(C)sc2)=O)CCC(O)CN(C(=O)C(C)(O)C2CCC2)C1 19030,c1(CC)cc(C(=O)NCC(C)CNC(=O)C(C(C)(C)C)n2ccnn2)ccc1Cl 19031,Cn1c(C(=O)NC2C3CC2N(C(=O)CCc2ccc(CO)cc2)C3)cccc1=O 19032,C1(NC(c2ccc(OCC)cc2)=O)CN(C(c2cncnc2C)=O)C(C)(C)C1 19033,C1(CNC(c2cccnc2C2CC2)=O)CCC(C(=O)NC2CCCC(O)C2)CC1 19034,N1(C(c2cc(C3CC3)nn2C)C(=O)NCC=C)CCOc2ccc(Br)cc2C1 19035,c1(C(C)C)ncsc1C(=O)NCC1CCN(C(=O)C(F)(F)Sc2cnn(C)c2)C1 19036,CCC(CC(=O)NC(C)(Cc1ccccc1)C(F)F)c1ccccc1 19037,N1(C(CN(C(=O)OC(C)(C)C)CCC(N2CC3CC3C2)=O)=O)CC=C(C(=O)O)CC1 19038,C(CCCCC(=O)NCC1CC=CCO1)N(C(C(C1CC1)OCC)=O)C 19039,N1(C(CNC(=O)CC(F)(F)F)=O)CCCCCCC1C(N1CCC(CF)C1)=O 19040,N1(C(CCSCC(C)C)=O)CCC(C)(NCC2CCC2CF)C1 19041,O=[N+]([O-])c1cc(NC2CC3CC3C2)cc(NCCN2CCSCC2)c1 19042,N1(C(C(C(=O)OC)C)=O)CCc2sccc2C1CNC(=O)CCCc1ncco1 19043,N1(C(CC2CCCC(=O)C2)=O)CC2CCC2(CC(N2CCC3CCCC23)=O)C1 19044,c1(C(N2CCC(N(C)C(C3CC(C)(C)CN3C)=O)CC2)=O)nccc2[nH]ccc12 19045,N1(C(c2c(C)cncc2)=O)CCN(C(=O)COc2cccc(O)c2)CC1C 19046,c1(OCC(=O)NCC(CC=C)NC(=O)CSc2cn[nH]c2)ccccc1OC 19047,c1(NC(C2N(C(CC3CCC(=O)NC3)=O)CC(O)C2)=O)nc(O)ccc1[N+](=O)[O-] 19048,Cc1nc(C(N2CCC(C)(NC(C3CC4C=CC3C4)=O)C2)=O)c2ccccn12 19049,N1(C(C2C(CC(C)C)C2)=O)CCCC12CCN(C(=O)Cn1nc(O)ccc1=O)CC2 19050,N1(C(C(n2cnc(C#N)n2)C)=O)CC(C)N(C(C2CC(Cl)(Cl)C2)=O)CC1C 19051,c1(C(N2CCC(NC(C3(C)C(CC)CCC3)=O)C(F)C2)=O)cc2ccccc2[nH]1 19052,C1(O)(C(C)NC(c2c(C)cc(C)s2)=O)CCN(C(=O)C(c2ccccc2)C)CC1 19053,c1(OC)ccc(C(F)F)cc1C(=O)NC1CC(O)CN(C(=O)CSC(F)(F)F)C1 19054,c1(C(N(CC#C)CCO)=O)ccc(OCCOC)cn1 19055,CCC(C)C(C(=O)N)N(C(=O)C(C)C1CCC1)CC.c1(CN2CCCC2)ccn(C)n1 19056,CC1CN(C(=O)NC2CCN(C)C2c2ccccc2)CCC1C.c1(C=O)ccc(Cl)cc1 19057,CC(C)C(CNC(=O)CCC(C)(C)F)C(=O)Nc1cn(C)nc1O 19058,C(CC(N=c1[nH]cnc2cnn(C)c12)C(C)C)N(C(c1n[nH]c(C)c1O)=O)C 19059,N1(S(CC(C)C)(=O)=O)CC2(CCN(Cc3ccccc3C(=O)O)C2)C1 19060,c1(C(=O)NCC2N(C(C=CC(C)(C)C)=O)CC(O)C2)cncc2ccccc12 19061,C1(C(N2CCN(C(C(C(=O)OCC)(C)C)=O)CC2C)=O)CCn2ncnc2C1 19062,N1(C(C(C)(F)F)=O)CCOC2(CCN(C(=O)C=Cc3c(F)ccc(Cl)c3F)C2)C1 19063,N1(C(c2cnccn2)C(=O)NCCCC)CCC(N(C)C)C(CC)C1 19064,c1(N2CC3C(N(C)C)C3C2)nc(=NCC2(C3CCC3)CC2)[nH]c2c1SCC2 19065,N1(C(CSCC#C)=O)CCC(C)(C(=O)NC(C)(C)CCOC)C1 19066,C(C(=O)NCC1CCCC1NC(c1ccc(CO)o1)=O)(C(C)C)n1ncc(C)c1 19067,c1(C(=O)NC(CC)CN(C(=O)C(O)C2CC2)C)cn(C(C)(C)C)cn1 19068,CN1CC(C)(C)CC1C(N1CC(C(=O)NCC2CCCCCCC2)CC1(C)C)=O 19069,N1(C(C(C)SC(C)C)=O)CC2(C(=O)NC3CC4(CCC4)C3)CCC1CC2 19070,c1(CC(=O)NCCCN(C(c2cc(Cl)cn2C)=O)CC)cccnc1C(F)(F)F 19071,N1(CC(=O)Nc2coc(C(F)F)n2)CCC(CNC(C2CCCC2(F)F)=O)CC1 19072,c1(CNC(c2cc(C(C)(C)C)on2)=O)c(F)cncc1F 19073,c1(NCC(CC(C)O)(C)C)cc(=NCC(c2ccsc2)N(C)C)[nH]cn1 19074,c1(CN(c2c[nH][nH]c2=NCc2nc(CO)cs2)C(C)(C)C)cc(Br)cnc1Cl 19075,C1(NC(=O)CN(CC(F)(F)F)CC(F)CNC(=O)CC2CCCC2)CCNC1=O 19076,CCC(C)(C)C(O)C(=O)NCC#CCNC(C1CCC2(CC1)CC2)=O 19077,N1(C(CC(CC)C2CCC2)=O)CC2CN(C(C3(Cl)CC3C(C)=O)=O)CC(C1)O2 19078,c1(C(CC)NC2C(c3ccccc3)C2C)ccc2c(c1)COC2 19079,N1(C(C(C)n2cccc2)=O)CC2CC1(C(=O)NC1CCOC1(C)C)C2 19080,C(=O)(C(C)CS(C)(=O)=O)NC1C(NC(c2ccc(-c3nc(C)[nH]n3)cc2)=O)C1 19081,C1(C(=O)NCC2CN(C(C(=O)N(C)C)=O)CC23CCC3)CCc2cnn(C)c2C1 19082,c1(C(N2CCC(CS(=O)(=O)NC)C2)C)cc(F)c(F)c(F)c1 19083,C(=O)(C1=CCCN(Cc2ccc(Cl)c(I)c2)C1)Nc1cc(C(=O)OC)cc(F)c1 19084,c1(N(CCC)Cc2cc[nH]c3nccc2-3)cccc2ccccc12 19085,C1(NC(CCNC=O)=O)CCN(C(=O)CCOC2CCC2)CC(O)C1 19086,c1(SC)cscc1NC(=O)C(=O)N(C(C)CO)Cc1ccncc1 19087,N1(C(C(C(C)C)C)=O)C2CCC1CN(C(c1cnnn1C1CCOCC1)=O)CC2 19088,N1(S(CCOC)(=O)=O)CCN(C(c2cc(C(F)(F)F)ccc2Br)=O)CC1C(C)C 19089,N1(C(c2c(Cl)cc(C)nc2)=O)CC2(CCC2)CC1CNC(=O)Cc1cnccn1 19090,C#Cc1ccc(CNC(C2CCCCN(C(C3CCC(CC)C3)=O)C2)=O)cc1 19091,c1(SCC)ccccc1C(=O)NCCCOCCN(C(=O)Cc1c[nH]nc1O)C 19092,N1(CC(=O)NCC(C(=O)NCC2(F)CC2(F)F)OC)CCNC(=O)C1 19093,c1(CCNCC(=O)NCCN(CCCCCC)C(C)=O)ncccc1F 19094,Cn1c(-c2ncccc2C(=O)Nc2ncc[nH]2)cc2ccccc12 19095,C1(C(=O)NC(C)Cc2nn[nH]n2)N(C(C2CC(N(C)C)C2)=O)CC12CCCC2 19096,C(=O)(CC(C)P(C)(C)=O)NCC(CNC(c1c(CC)c[nH]c1)=O)C(F)(F)F 19097,C(c1cc(Br)cs1)=CC(=O)NC1CCCN(C(C2CCNC2=O)=O)C1 19098,N(C1COc2ccc(Cl)cc21)C(C1C2CN(C(c3ncccn3)=O)CC21)=O 19099,Cc1ccc(F)c(C(=O)NC2COCC2NC(c2ncc(Br)cc2F)=O)c1 19100,C1(NCCc2cc(C)c(Cl)cc2)CC2CCCCCC2C1 19101,C(CCCCCCCO)=CC(N1C2(CN(C(=O)C3=CCCOC3)C2)CC1)=O 19102,C(=O)(CCS(=O)(=O)CC(C)C)NC1CC(N(C(COCCCOCC#C)=O)C)C1 19103,c1(CC)nc(C)c(C(=O)NCC2(CCNC(=O)C(C(C)C)NC=O)CC2)o1 19104,c1(COC)cc(C)[nH]c(=NCC(C)(C2CC2)NC(C2CC3C=CC2C3)=O)n1 19105,C1(C)(NC(Cc2c(CC)con2)=O)CCN(C(=O)CCC(F)F)CC1 19106,c1(C(N2CCC(N(C(c3cc(C)c(O)cc3)=O)C)C2)=O)ccc2nc(O)[nH]c2n1 19107,c1(OCCC(=O)NCC2CC(NC(C3N(C(C)C)CCC3)=O)C2)cccc(F)c1 19108,CCCC(C)(O)CC(=O)N1CC2(C1)CN(c1ccc([N+](=O)[O-])cc1)C2 19109,N1(C(c2nc(C)n(C)c2)=O)CCN(C(=O)CCC2CCCO2)C(C2CC2)C1 19110,N1(C(C2(CC)CCN(C(CSCC=C)=O)C2)=O)CCCC(N=[N+]=[N-])C1 19111,c1(C(N2C(CC(=O)NC)CN(C(=O)C(F)OC)CC2)=O)cc(C)c(C)cc1C 19112,CC1CCCN(CCNC(=O)CC2CCN(C(C3(C)CNC(=O)N3)=O)C2)C1 19113,N1(C(c2ccc(C(C)(C)C)[nH]2)=O)CC2CCCC2(Nc2ccnc3ncnn23)C1 19114,c1(NCCc2cc(Cl)no2)nc2ccccc2nc1N1CC2(CCC2)CC1CO 19115,c1(C(N2CCC(CNC(C(C=CC)O)=O)C(C)C2)=O)cc(C)cc(OC)c1O 19116,N1(C(CC=CC=C)=O)CC(CNC(=O)CC2CCC(=O)N2C)C2(CC2)C1 19117,O=C1CCC(F)(F)CC1N1CCC(c2ccc(CO)cc2)C1 19118,C12(C(N3CC(C(C)NC(C45CCN(CC4)CC5)=O)C3)=O)CCCCC1C2(F)F 19119,c1(C(N2CCCCC2C2CCC2)=O)ccnc2c1NCCO2 19120,CCC(c1cccc(Cl)c1)=CC(=O)NCCC(C)N(C)C(c1nc(=O)n(C)[nH]1)=O 19121,C12(CNC(c3cc(C)c(C)o3)=O)CCCCC1CN(C(c1ccc[n+]([O-])c1)=O)C2 19122,C#CCCCCCCC(=O)NCC1(O)CCN(C(=O)CCC2CCCCC2)CC1 19123,C(CCCCC(=O)NCC(c1ccccc1)NC(c1ccn(C)c(=O)c1)=O)OC 19124,N1(C(c2c(C)[nH]nc2C(F)(F)F)=O)CC2CCN(C(C3CC3F)=O)CC(C2)C1 19125,C1(COC)CCCCN(C(C2CC3(CC(NC(=O)C(O)C4CC4)C3)C2)=O)C1 19126,c1(NC(C2C=CCN2C(c2ccc(F)c(Cl)c2)=O)=O)cccc(F)c1Cl 19127,N1(C(Cc2cnc(C)s2)=O)CC2(CCC2NC(C2CCCC(=O)N2)=O)C1 19128,Cc1nc(CC(=O)NCC(O)CN(C(=O)C(C)(C)CN(C)C)C)c(C)s1 19129,c1(C(N2CC3C(CNC(c4c(OC)nsc4)=O)C3C2)=O)ccc(C(C)=O)nc1O 19130,c1(C(=O)NC2C(NC(Cc3ncc(C)s3)=O)C2)cncc(N)c1C 19131,n1(CC)nc(C(=O)NCC2COC(CNC(c3sncc3C)=O)C2)cc1O 19132,c1(CNC(=O)CC(C2CC2)NC(c2ccc(Cl)cc2)=O)cccc2[nH]ncc12 19133,N1(C(Cc2cc(C)c(Cl)cc2)=O)CCC2(CC1)CC2NC(c1cnn[nH]1)=O 19134,CC1(C)CCC(C)(NC(C2CCCCN2C(C2CCS2(=O)=O)=O)=O)CC1 19135,C1(CNC(C2N(CC)CCC2)=O)(NC(=O)CCC(F)F)CCC(C)(C)CC1 19136,N1(C(CSCC=C)=O)CC2CCC1CN2C(c1cc(CC(=O)OC)on1)=O 19137,C1(C2(O)CCOCC2)(C(N2CC(F)(CNC(c3c(CC)onc3)=O)C2)=O)CC1 19138,C1(C(=O)NCC(C)CNC(=O)CCCN2CCCC2)CC(C)OC(C)C1 19139,CCC(C)CCC(=O)NCCCCCC1CCN(C(=O)CNC(N)=O)CC1 19140,c1(C(N(CCCNC(=O)C(C)(c2ccccc2)OC)CC)=O)cnn(C)c1C#N 19141,C1(CCC)CCCC1CNC1(COC)CC(C)C1 19142,c1(OC)cc(C#N)ccc1C(=O)N(C)Cc1ccc(C)cn1 19143,C1(NC(C2(NC(C)=O)CCCC2)=O)CCCN(C(C2CC(=O)NC(=O)C2)=O)C1C 19144,Cc1n[nH]c(C)c1C(=O)NC(Cc1ccc(F)cc1)CC(=O)NCC1CCO1 19145,c1(C(N2CCC(NS(CCC)(=O)=O)C2)=O)cc(Cl)cnc1O 19146,c1(OC)ccc(CC(=O)NC2CC3(C2)CN(Cc2cc(Cl)cc(Br)c2)C3)c(F)c1 19147,c1(CC)[nH]nc(Cl)c1C(N1CCCC(CCNC(c2cc(F)cs2)=O)C1)=O 19148,Cc1ccc(F)c(C(N2CC3CC2C3NC(=O)C2=CCOC2)=O)c1 19149,C1(C)(NC(CCOC)=O)CCCN(C(C2OCCO2)=O)C1 19150,N1(C(C2CSCCN2C(=O)CN(CCO)CCO)=O)CCc2ccccc2C1 19151,c1(CC(=O)NC(C=CC(=O)NC(C)CF)(C)C)ccc(SC2CC2)cc1 19152,N1(C(CNC=O)=O)CC2OC(=O)N(C3CCN(C(=O)C=CC=C(Cl)Cl)CC3)C2C1 19153,Cc1c(NC(C2CC(C)CN2C(C2CCC(=O)N2)=O)=O)cc(Cl)cc1Br 19154,c1(C(=O)OC)nc(=NCC(C)NC(C2OC(C)CC2C)=O)c(F)c(Cl)[nH]1 19155,C1(CNC(COCCCC#C)=O)CCC(NC(C2CC2COCC)=O)CC1 19156,c1(C(=O)NCCCN(C(C2(C)CC(=C)C2)=O)C2CC2)ccnc(C2CC2)c1 19157,N1(C(c2ccc(C)n2C)=O)CCN(C(c2n[nH]cc2F)=O)C(CS(C)(=O)=O)C1 19158,C(C#Cc1ccc(C(F)(F)F)cc1)NC(C1C(C)(C)CC(=O)NC1)=O 19159,O=C(N=c1[nH]ccc2cc(Br)ccc12)C1CC2CC2N1Cc1ncccc1Cl 19160,C1(NC(C2N(C(C3=CCCC3C)=O)CC(C)CC2)=O)CCCCCCC1(C)C 19161,C(=O)(CCCC(F)F)NCC(C1CCCCN1C(=O)C1=NOCC1)(C)C 19162,c1(C(=O)NC(CC=C)CNC(=O)C(n2nccc2C)C)ccnc(N(C)C)c1 19163,N1(C(c2c(CC)ncs2)=O)CC2CC(C1)CN(C(=O)C(C)(C)CC)C2 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19181,CCC(C)(CC)C(=O)NC1CCN(C(c2sc(C)nc2C)=O)C(C)C1 19182,N1(C(CCCOCCC)=O)CCCCC1CN(C(=O)COCCCF)CC 19183,c1(C(N2CC3CC(CNC(C4(CC#C)CC4)=O)C3C2)=O)cc(OC)c(O)c(Cl)c1 19184,N1(C(c2c(CC)n(C)nn2)=O)CCC(C(=O)N2CC(CO)CC2C)=C(F)C1 19185,c1(C(=O)NC(C)CNC(=O)CC2CCCCC2)cn(C(F)F)nc1C(F)F 19186,N1(C(c2cccs2)=O)CCN(C(C2CCC3(CCC3)C2)=O)C(C(F)F)C1 19187,CC1CCC(C(=O)O)N1C(=O)NCCCC(C)(C)C 19188,Cc1c(C(=O)NC2CCC(NC(=O)CSCCC(C)C)CC2)cnn1CCC#N 19189,Cc1nc2c(C)cc(C(=O)N(C(CO)CC(C)C)C)cn2n1 19190,c1(C(N2CC(CN(C)C(c3cncnc3)=O)C2)=O)cccc(S(C)=O)c1 19191,C1(C(N(C(C)CNC(c2ccc(OC)cc2)=O)CC)=O)CC(F)(F)C1(C)C 19192,N1(C(c2c(CCC)[nH]cc2)=O)CCC2(CCC2)C(NC(=O)CCS(N)(=O)=O)C1 19193,CCC(CC1CCCC1)C(=O)N1CC(COC)(NC(=O)Cc2nonc2C)C1 19194,c1(CC(N2CC(CCNC(C(C(C)OC)O)=O)C2)=O)cn2ccccc2n1 19195,CC1CCC(CNC(=O)CC(C)(C)O)N(C(c2csc(C(F)F)c2)=O)C1 19196,C(=O)(CCCCCC#N)NCCC1CCCN(C(c2c(C)noc2C(F)F)=O)C1 19197,C(=O)(C1COc2ccccc21)N1CC(CN(C(C(C)OCC2CCCO2)=O)C)C1 19198,C1(CC(=O)NCCC(C)N(CCC)C)CCN(C(c2cscc2C)=O)C1 19199,c1(CNCc2ccc(F)nc2)c(F)cc(Cl)cc1Cl 19200,C1(C(F)F)(CNC(C(C)O)=O)CCN(C(=O)CCN(S(C)(=O)=O)C)C1 19201,N1(C(C)C)CCN(C(=O)C(CCF)NC(C2CCC(C(N)=O)C2)=O)CC1 19202,C(=O)(CC(C)(C)C)NC(C1CCN(C(c2cnc(C(C)C)[nH]2)=O)CC1)C 19203,[N-]=[N+]=NCCCCCC(=O)NCCC1CCN(C(=O)C=Cc2nccs2)C1 19204,C1(CNC(c2ccc(C(F)(F)F)s2)=O)CC2(CCC2=O)C1 19205,CCC(CC)(CO)NC(c1cncc(CNC(C2CCN(CC)CC2)=O)c1)=O 19206,CCCC(O)(CCC)CC(=O)NCC1(O)CN(C(c2ccc3nccn3n2)=O)C1 19207,N12CC(C3(CC3)C1)C(=O)N(C)CCC2=O.C(CC(C)C)OCCN(CC)CC 19208,C1(=O)C(CCC(C)C)N1.c1(C(=O)NCCN(C(C)=O)CC)ncn(C)n1 19209,C#CC1(C(=O)NCC(C)(F)C(C)C)CCN(C(=O)CNc2ncccn2)C1 19210,C1(N(c2ncc(Br)cn2)C(C2CCCS2)=O)CC2CCC(C1)N2 19211,C(=O)(C(F)C1=CCCCC1)N1CCC(O)(C(C)NC(C2C(CC)OCC2)=O)CC1 19212,c1(NC(c2cccnc2)CC)nc2ccccc2nc1NCC1CCC(C)CC1 19213,C1(=O)NNc2ccc(cc2)S(=O)(=O)CN1.c1(OCCC)ccccc1C(F)(F)F 19214,C(c1ccoc1)=CC(=O)NC(c1ccccc1)CNC(C=C(C)Cl)=O 19215,C1(NC(C(c2ccccc2Br)NC(C2CCC(=C)CC2)=O)=O)CCCC(C)(C)C1 19216,c1(C(=O)NCc2cc(C)c(C)nn2)coc2c1CN(C(=O)CC1CCOC1=O)C2 19217,C(=O)(CC(CNC(C1C=CCS1)=O)OC)NC1CCN(CC)C1 19218,C(CC1CC1)(C(=O)NCCS(=O)CC)NC(C=CC=CCC)=O 19219,C1CCCCCC(=O)N1.C1(C)(c2cn(CCCCSC(C)=O)nn2)CCOCC1 19220,C(C(C(C)C)NC(c1ocnc1CC)=O)NC(C1C(C(=O)NCC#C)C1)=O 19221,C1(=O)C(CC)N1.CCC(CSC)N(C(=O)CC1(N(C)C)CC1)C.C(C)(=O)N 19222,C=C(Br)CC(C)(C)C(=O)NC1CCCCN(C(c2cc(COC)on2)=O)C1 19223,c1(C(=O)NCCN(C(=O)Cc2cc[nH]n2)CC)cc(C(C)=O)cs1 19224,C(CCC1CCC1)(C(=O)NCCc1ccon1)NC(c1cc(CO)on1)=O 19225,c1(C(=O)NCC(C)(CO)NC(c2nc(Br)c[nH]2)=O)c(F)cc(F)cc1F 19226,C1(C2CC2)(NC(C(SC)SC)=O)CCN(C(=O)Cc2cc(C)ccc2F)C1 19227,c1(CC)nc(NCCc2nccs2)cc(=NC2CC3C=CCC(C3)C2)[nH]1 19228,CN1CC(NC(C2(C)CCCN(C(C3CN4CCN3CC4)=O)C2)=O)C2(CC2)C1=O 19229,CC1=C(C(=O)N2CC3=C(C2)CN(C(c2c(C)ncn2C)=O)C3)C(=O)OC1(C)C 19230,N1(C(CN(C2CC2)CC)=O)CC(F)(F)CC1CNC(c1cccc(C2CC2)c1)=O 19231,c1(C(=O)OC)cccc(CCCNC2CC(SC(C)C)C23CCC3)c1F 19232,C1(CNC(C2(C(C)(F)F)CC2)=O)(NC(C2CCCCS2(=O)=O)=O)CCCCCC1 19233,C#CC1(C(=O)N(C(C)CCCC)C)CCN(C(C2CCC(COC)C2)=O)CC1 19234,C1(NC(C(C)(C)CF)=O)CCN(C(=O)Cn2ccccc2=O)CCC1CO 19235,CC1CC(NC(=O)Cc2cc(C(F)(F)F)n[nH]2)CCN1C(=O)CC1CCC2CC12 19236,CCC(C(=O)OC)C(=O)N1CCN(C(=O)CCOCC(F)F)C(CC(F)(F)F)C1 19237,c1(C(=O)NC(C)(CNC(=O)C=CC(F)(F)F)C2CC2)csc(-c2ccco2)n1 19238,N1(C(C(COCC)C)=O)CCC2CN(C(=O)C=CC3CCCN3C)C2C1 19239,c1(C(=O)NC2(CC)CN(C(C3(NC(=O)OC)CC3)=O)C2)nccc(C)c1N 19240,CCCC(C)CCNC(=O)COCCNC(=O)CC1CCOC1(C)C 19241,Cn1cnc(CNC(=O)CC2CCN2C(C2CCCC2)=O)n1 19242,c1(C(N2CCCC2Cn2cc(COC(C3C(CC)C3)=O)nn2)=O)ccc(CO)cc1 19243,C(=O)(C(C(C)(C)C)NC(=O)C(O)Cn1cncn1)N1CC(S(C)=O)C1 19244,CCC(C)(CNC(C1(NC(=O)CC2CCCOC2)CC1)=O)CC 19245,c1(NC(Cc2nccc(CC)c2)=O)ccc2c(c1)CCC2N(C)C 19246,C12(C(N(C)Cc3nnc(O)o3)=O)CC(CO1)N(C(c1ccc(C3CC3)o1)=O)C2 19247,C1(C(=O)NCC(C(=O)NCc2cn(C(C)C)nc2)(C)C)CC12CCCCC2 19248,Cc1ccc(C(=O)NC2CC(N(C(=O)CC(C)C3CC3)C)C2)c(O)c1C 19249,C(=O)(C1=NOC(C)(CNc2cccc(OCC(=O)O)c2)C1)OC 19250,c1(NC)c(C(=O)NC2CC3(NC(=O)C#CC4(C)CC4)COC2C3)cccc1F 19251,c1(OCC)ccc(C(=O)OC(C)C(N)=O)cc1S(=O)(=O)NC 19252,Cc1nc(C2CC2)ccc1C(=O)NCC1CN(C(=O)C(F)C(F)(F)F)CCC1C 19253,C(CCSC)(CN=c1[nH]c(=NCc2csc3c(F)cccc23)[nH]c2cc[nH]c12)OC 19254,N1(C(COC(C)C)=O)CC2CN(C(=O)Cn3nc(Cl)ccc3=O)CC2C1 19255,c1(C(=O)NCCOCCNC(C(C)NS(CC)(=O)=O)=O)ccc(C(C)=O)cc1F 19256,C1(c2cn(CC3C(CC(N4CCCOCC4)=O)CCC3)nn2)CCCS(=O)(=O)C1 19257,C1(C(=O)NC2CN(C(c3ccc(C)cc3)=O)C(C)CC2)CC2(C1)CC1(CCC1)C2 19258,C(=O)(CCC(=O)NN(C)C)N1C(CNC(c2ncn(C(C)C)c2)=O)CC(O)C1 19259,N1(C(C2N(CC#C)CCC2)=O)CCOCC(NC(=O)C(C)N(C)C)C1 19260,C1(C)(C(=O)NCCSCC#C)C=CCN1C(=O)C(C)=C1CC1 19261,c1(C(=O)NC(C2CCOC2)CNC(c2c(C(C)=O)ccs2)=O)cc(F)ccc1N 19262,c1(-c2[nH]c(=NCc3ncc(C)c(O)c3)sc2)cccc(Cl)c1[N+](=O)[O-] 19263,C1(CNC(CC=CCC)=O)CN(C(C2C(C(=O)OC)C2(F)F)=O)CCN1C 19264,N1(C(c2c(C)cc(C)nc2)=O)C2COCC1CC(NC(C1(F)CC=CCC1)=O)C2 19265,c1(C(=O)NCC2N(C(C(C(C)C)C)=O)CCC2)ccn(C(=O)OC(C)(C)C)n1 19266,C1(NC(c2cnc(F)c(Cl)c2)=O)CCC2CCN(C(c3nocc3Cl)=O)C1C2 19267,Cc1ccc(Cl)c(C(=O)NC2CC(CNC(=O)Cc3nccn3C)C2)c1N 19268,C1(C(=O)NCC23CC(CN2C(c2sccc2Cl)=O)C3)(OC)CCS(=O)(=O)C1 19269,CC1CCc2sc(C(N3CC4CCCC3C4CNC(=O)C(C)C)=O)cc2C1 19270,C12(C(=O)NCCC(C)N(C(=O)C=CCOC(C)(C)C)C)C=CC(CC1)C2 19271,N1(C(C=CC(C)(C)NC(c2c(C)n(C)nn2)=O)=O)CCC(C)C2(CCC2)C1 19272,C1(C(C)NC(C(C)OCCCC)=O)CCCN(C(c2cccs2)=O)C1 19273,c1(C(N(C2CCCCC2)CCNC(C(C2CCOC2)OC)=O)=O)c(C)ccn1C 19274,C1(NC(c2ccnc(Cl)c2)=O)CCC2CN(C(C3CCC=CCCC3)=O)CC2C1 19275,C(CN=c1nc(C2CC2)[nH]s1)C1CC(NC(CC2N(C)CCC2)=O)C1 19276,c1(C(N(CCN(C(=O)Cc2ccc(F)cc2F)C)C)=O)ccc(F)c2[nH]ccc12 19277,N(C(=NCCc1cn(C)nc1C)NCC12CCCC(C)(C1)OC2)C(CC)C 19278,C1(CCC)CCC(NCC2CCC2C(F)F)CC1 19279,c1(OC)ccc2cc(C(=O)NCC3CN(C(=O)C(C)S(C)(=O)=O)CCO3)[nH]c2n1 19280,C1(NC(c2c(CC)nn(C)c2)=O)CC2CCC1CC2NC(c1sccc1SC)=O 19281,c1(NC2CC(C)C2)cc(N2CCOC(CNC(C)=O)C2)ncn1 19282,CC(C)C(C(C)NC(c1sccc1C1CC1)=O)NC(=O)CCc1ccc[nH]1 19283,C=CC1COCCN1C(=O)C(C)(C1CC1)N(C)C(C12CC(F)(C1)C2)=O 19284,c1(CC)n[nH]cc1C(c1nnnn1C1CC1)NC(C(C)NC(C)C)c1ccccc1 19285,N1(C(C2CCC(CC)CC2)=O)CCCC2(CCC2NC(=O)Cc2cnn(C)c2)C1 19286,CCCCCCCCC(=O)NCCN(CC(C)O)C(C1CC1c1ccoc1C)=O 19287,c1(-c2onc(COC(C)C)n2)ccc(OC(F)(F)F)c(Cl)c1 19288,N1(C(C(C)OCCC#C)=O)CC(NC(=O)C=C(C)C(C)C)CC(F)C1 19289,c1(CN2C(C(=O)Nc3ncn(C)c3)CC3CC32)cccc([N+](=O)[O-])c1F 19290,C1(CNC(Cc2c(C)scc2)=O)CCCC(CNC(=O)C(F)=CCCF)C1 19291,c1(C(=O)NCC(C)N(C(c2cncc(C)c2Cl)=O)CC)cc(F)cc([N+](=O)[O-])c1 19292,c1(CCC)cc(C(=O)N(CCC(=O)NC2CC(CC)C2)CC2CC2)no1 19293,N1(C(c2c(CNC(c3c(C)oc(Cl)n3)=O)ocn2)=O)CC2(C)COCC2(C)C1 19294,C1(NC(c2cc(C)c(C)o2)=O)CCC2CC1CN2C(c1coc(C(F)(F)F)c1)=O 19295,C1(O)(CNC(C(C)OCCN(C)C)=O)CCCN(C(c2ncccc2N)=O)CC1 19296,C(=O)(C(F)C(F)(F)F)NCC(C)N(C(c1c(NC(CC)=O)cccc1)=O)C 19297,C(=O)(NNc1cc(F)c(F)c(F)c1)c1n(CCN)ncn1 19298,CC1CCN(C(=O)CC2(N(C(=O)C3=CCC(C)CC3)C)CC2)CC1(C)C 19299,C12(C(N3CCC(CC#C)C3)=O)CC(C)(CN1C(C1NC(=O)CC1C)=O)C2 19300,N1(C(C2(C)C=CCC2)=O)CCN(C(C23CCC(CC2)OC3)=O)CC12CCC2 19301,S(=O)(=O)(c1cccc(=NCC2CC2Cl)[nH]1)N1CCN(CCC(=O)N(C)C)CC1 19302,CCC(CC)C(=O)N1CC(NC(C2(Cc3cccc(F)c3)CC2)=O)C(C)C1 19303,C(=O)(CCCC#N)NCC(CC)N(C(=O)C(N1CCCC1)C1CC1)C 19304,C(=O)(C(C)C(C)(F)F)NC1(C)CC(NC(c2c(C(C)C)n[nH]c2)=O)C1 19305,Cc1cc(C)c(C(=O)NCCOCCNC(=O)C(C)Cc2cnn(C)c2)c(Cl)n1 19306,CN1CCN(C(c2cccnc2)=O)CC1C(=O)N(C1CCCC1)C1CC1 19307,N1(C(CN(CCOC)C)=O)CC2CCC1C(NC(=O)C(C(C)(C)C)C1CCC1)C2 19308,Cc1ccccc1C1(C(=O)NCCC2CCCN2C(c2ccc(F)s2)=O)CCC1 19309,c1(C(=O)NCC2(N(C)C)CC2)ncc2ccccn12.C12(CC3(CC3)C1)C(=O)NC2 19310,Cc1noc(CCNC(C2CC(C)N2C(=O)CC2CCCC2)=O)n1 19311,C1(c2c(CC)c(C)no2)CCN(c2cc(NC3CC(C)N3CC)ncn2)CC1 19312,CS(=O)(=O)CCC(=O)N1CCC(C2OCCC2NC(=O)CO)CC1 19313,C1(NC(c2c(OCCC)cccc2)=O)CN(C(C2CSCCS2)=O)CCC1F 19314,C(=O)(C(C)CN(C(=O)C(Cc1cc[nH]n1)NC(=O)CCn1cc(C)cn1)C)NC 19315,C(=O)(C1=C(C)OCCS1)NC1CC2CN(C(c3nn(C(CC)C)c(C)c3)=O)C1C2 19316,C(=O)(C(F)CCC(C)C)NC12C(NC(C3N(C(CC)=O)CSC3)=O)CC(CC1)C2 19317,C12(C(=O)NC(CC)COCC3CC3)CC1CCN2C(C1CN(C2CCC2)C1)=O 19318,C1(C(=O)NCCC2(NC(c3c(OC)scc3)=O)CC2)CCCC(C(N)=O)C1 19319,N1(C(C#CC(=O)N(C)C)=O)CC=C(CCNC(C2(F)CCS(=O)(=O)C2)=O)CC1 19320,C(=O)(C1=CC(O)C(NC(c2cccc(CC)n2)=O)C1)NCC 19321,CCCC(CCCNC(=O)C=CBr)NC(=O)C(C1CC1)OCC 19322,CS(=O)c1cccc(C(N2CCN(C(=O)CCF)C3CCC23)=O)c1 19323,C(CC(C)(C)C)(C(=O)NCCOCCCNC(=O)CCCN(C)C)OC 19324,c1(C(=O)NCC(C)CNC(=O)CCc2cncs2)ccc2c(n1)NCC2 19325,C1(N(C(c2ccc(C3COC3)cc2)=O)CC)CCCN(C(c2cn[nH]c2)=O)CC1 19326,c1(CC)ncc(S(=O)(=O)Nc2c(C)[nH]c3cnccc23)n1-c1ccccc1 19327,c1(C(N(CCCNC(C(C2CCCC2)OCC)=O)C)=O)c(C)nn2ncccc12 19328,C1(NC(c2c(CCC)nns2)=O)CN(C(=O)C(C)S(N)(=O)=O)CC12CCC2 19329,N1(C(c2c(C)[nH]c(=N)s2)=O)CCC2(CC(NC(=O)COCC(C)(C)C)CO2)C1 19330,C1(CNC(C2CC3CCC2C3)=O)CCC2(CN(C(C3CC4CCC3CC4)=O)C2)O1 19331,c1(CC)nc(C)cc(=NC(=O)c2ccn3ncc(I)c3n2)[nH]1 19332,Cc1cc(C)c(CC(=O)NC2CC(N(C)C(c3ccc(C#N)[nH]3)=O)C2)s1 19333,c1(C(N2CC=C(CNC(C3CCOC3)=O)CC2)=O)ccc2nn[nH]c2c1 19334,C#CCCCCCCC(=O)NNC(=S)c1ccccc1NC 19335,c1(OC)cccc(C)c1C1(C(=O)NCCSc2cc(OC)ccc2O)CC1 19336,C#Cc1cn(C)nc1C(=O)NC(C)CC(=O)N(CC(N)=O)CC(N)=O 19337,c1(CC(=O)NCC(CNC(c2cc(C)c(C)o2)=O)F)ccc(F)c(Cl)c1F 19338,N1(C(C(C)(C)NC(=O)OC)=O)CC2CC(NC(c3ccnc(C)c3Cl)=O)C1C2 19339,Cc1nc2ccc(C(=O)NCC3CCCC3NC(=O)CC3CC3(Cl)Cl)cc2n1C 19340,N1(C(c2cnc(CCC)s2)=O)CCCC(CN(C(C)C(=O)NC)CCC)C1 19341,N1(C(CC(C)C(F)F)=O)CCC2CCN(C(c3cc(C(F)F)ccc3F)=O)CC12 19342,C1(C(N2CCN(CC)CC2)=O)CC12CCN(c1ncc(Br)c(C)n1)CC2 19343,CC(C)(C)CC(O)CC(=O)N1CC(CNC(=O)C=Cc2cscn2)C(C(F)F)C1 19344,C1(NC(=O)CCC2CC2(Cl)Cl)(CO)CCCN(C(C2CCCNS2(=O)=O)=O)C1 19345,C1(CC=C)(C(=O)NCCCC(=O)N(C)C)CCCN1NC(c1cncc(C)n1)=O 19346,N1(C(C2CC(CNC(=O)OC(C)(C)C)C2)=O)CC(O)CC1c1nc[nH]n1 19347,C1(NC(C(C)N2CCC2)=O)CCCC(NC(c2nnc(C(C)(C)C)s2)=O)C1 19348,N(C(C)S(=O)(=O)C(C)C)(C1CC1)Cc1c(C)cc(C)o1 19349,c1(OC)ccc(C)c(C(N2CC(NC(=O)C(C)CSC)C(C)(C)C2)=O)c1 19350,C1(NC(C(C)C2CC2)=O)CN(C(=O)CCc2cccc(Cl)c2)CCC12CCC2 19351,Cc1cc(N)cnc1-c1cn(CC2N(C(=O)Cc3[nH]cnc3C)CC2(C)C)nn1 19352,C(=O)(C1=NOC(C)C1C)N1CCC(NC(c2cc(C(C)C)on2)=O)(CO)C1 19353,Cc1cnc(C(N2CCC(NC(c3cc(F)c[nH]3)=O)C(CO)C2)=O)c(C)c1 19354,CC(CC(C)(C)C)C(F)C(=O)N1CCOC(CNC(c2n[nH]cc2[N+](=O)[O-])=O)C1 19355,CC1CCN(C(C2C=CCC2)=O)CC1CNC(c1cnccc1Cl)=O 19356,C(=O)(C(C)(C)C(C)C)N(CC(CNC(Cc1ncc(C)s1)=O)O)C 19357,C(CCCCCNC(C1CCCN1C)=O)NC(C=CCCC=C(C)C)=O 19358,C(=O)(CCCCC(=O)N1CCC(C)N(C(C2CCCN(C(N)=O)C2)=O)CC1)NC 19359,CC1CC(=O)NC(C(=O)NCC2(CNC(c3nocc3C3CC3)=O)CC2)C1 19360,N1(C(C(C)NC=O)=O)CCC2CN(C(c3cnc(O)nc3O)=O)CCC12 19361,N1(C(C(C(C)C)OC)=O)CC(CNC(c2cccc3nn[nH]c23)=O)CC12CCC2 19362,C12(C(N3CCC(CNC(C(C(C)C)O)=O)C3)=O)CC3CC(CC1C3)C2 19363,c1(C(N(CCN(C(CSCC)=O)C(C)C)C)=O)nc(C)ncc1Cl 19364,N1(C(c2c(C)noc2N)=O)CCCC(NC(=O)CC(O)C2CCCC2)CC1 19365,C12(C(=O)NC3CCN(C(C)C)C3=O)CC(CCO1)N(C(=O)Cc1ccco1)C2 19366,C(=O)(CC(=O)NC(C)CNC(=O)C(C)C1CCC1)NCC#C 19367,N1(C(C(C)NC(c2ccco2)=O)=O)CC2CCCC(NC(=O)C(C)(C)F)C2C1 19368,CC(C)CC(C)CC(=O)NC1C2CC1N(C(=O)C1=COCCO1)C2 19369,CC1CCCC(NC(N2CCN(CC(C)(C)O)CC2C)=O)C1C 19370,CC1CN(C(c2ncc[nH]c2=O)=O)CC(CCNC(c2cn(C)nc2Cl)=O)O1 19371,C12(C(=O)NC3C4CN(C(C5(NC(C)=O)CC5)=O)C3C4)CC=CC(C1)OC2 19372,N1(CC(=O)N(C(c2cn(Cc3nnc(C)o3)nn2)C)C)CCCC(C(C)O)C1 19373,C(=O)(CCC(=O)NN(C)C)N1C(C(N2C(C(C)C)C(C)(C)C2)=O)CC1C 19374,Cc1cc(NC(C2CC(O)CN2C(c2cnn(C)c2)=O)=O)cc([N+](=O)[O-])c1 19375,C1(CC(=O)NC(CNC(c2ccc(COCC)[nH]2)=O)CO)(OC)CCOCC1 19376,c1(C(N2CCCC(CNC(CSC(C)(C)C)=O)C2)=O)cccc2nonc12 19377,N1(C(C(c2ccc(OC)cc2)=O)=O)CCS(=O)(=O)CC1C(C)(C)C 19378,N1(C(C2CC=CC(NC(C(CC)(C)O)=O)C2)=O)CC=C(CO)CC1 19379,C(=O)(C(CC1CCC1)NC(=O)C(CO)OC)N(C(CC)C)C 19380,C1(C(=O)NCC2(C(=O)N(C)CCN3CCCC3)CC(=C)C2)CCCCCC1 19381,c1(C(=O)NCC2CCCC(NC(C(C)c3cccs3)=O)C2)ccc2nccn2n1 19382,C=CCC(C(=O)NCC1CC2CCC(C1)N2C(=O)C=NOC)C(C)(C)C 19383,C12(NC(CCC=C=C)=O)CCCC(CN(C(C3CCCN3C)=O)C1)C2 19384,C(C)(CNC(c1ccc(-c2nncn2C2CC2)cc1)=O)(C(C)C)NC(C)=O 19385,C#CCCC(O)C(=O)NCCNC(C1CCC(Cc2cccc(Cl)c2)C1)=O 19386,CC(C)(C(=O)NC(CNC(=O)CC1NC(=O)CNC1=O)CC(F)(F)F)C(F)(F)F 19387,CC1(C(=O)NCCc2n[nH]cc2C(=O)NCCC2CC(O)C2)CCCC1O 19388,N1(C(c2c(F)ccc(C)c2)=O)CCC2(CCCN2C(C2C(C(F)F)C2(C)C)=O)C1 19389,N1(C(Cc2ncc(C)o2)=O)CCC2(CCCC2NC(C2C=CC=CC=C2)=O)CC1 19390,CC(C)C(CC(=O)NCCCc1ccsc1)NC(c1c[nH]nc1C(F)F)=O 19391,C(C(C)(C)C(=O)NC1C2CN(C(C3CCCN3C(C)=O)=O)CC12)NC(C)=O 19392,c1(-c2cn(C3CC(C(=O)OC)C3)nn2)cc(F)c(F)c(F)c1 19393,C(C(=O)NCc1ccoc1C(=O)NC(C(O)CO)C1CC1)(C(C)(C)C)OC 19394,CCCC(C)C(=O)NC(C)(CNC(=O)Cc1nccc(OCC)n1)C1CC1 19395,C1(C(C)C)COCCN(C(c2sccc2CNC(=O)CC(F)(F)F)=O)C1 19396,N1(C(C2CCCN(C(CC)=O)C2)=O)CCCC2CN(CC3CCCCCC3)CC12 19397,C(=O)(C(F)CC(C)(C)NC(=O)CC(C)(C)CC)N1CCCC(C=C)C1 19398,C1(N(C(c2[nH]cnc2C)C(=O)NC(CC)(C)C)C)CCN(c2ncccn2)CC1 19399,c1(N2C(C)CN(C(c3cc(=O)cc(Cl)[nH]3)=O)CC2)ncc(C#N)cc1Br 19400,c1(C(=O)NCC(C)NC(c2c(F)ccc(F)c2O)=O)c(F)ccc2nc[nH]c12 19401,C1(CN(C(CCn2c(C)ncc2)=O)C)CN(C(=O)C(N)=O)CC12CC2 19402,c1(-n2c(C3C(C)(C)N3)nnn2)cccc([N+](=O)[O-])c1.C1(CSC)CC(C(N)=O)C1 19403,C(CCCCC(=O)N1CC(C)(OCC(N2CC3C(C)C3C2)=O)C1)=CC 19404,C1(C)(CNC(C(C2CCN(C(c3coc(C4CC4)n3)=O)C2)C)=O)CCCOC1 19405,Cc1cc(CC(N2CCC(F)C(NC(c3ccoc3Cl)=O)C2)=O)ccc1CO 19406,N1(C(c2c(C)ccs2)=O)CC2CCC(NC(c3ccc4n[nH]cc4c3)=O)(C2)C1 19407,C(=O)(CCCCCc1ccccc1)N1CCC(CC(=O)N(CCC(N)=O)CC)C1 19408,CC(C(=O)NCc1cn(C2CN(C(c3ncccc3Cl)=O)C2)nn1)C(C)(F)F 19409,C12CCN(C1)C2=O.C1(C2CCCO2)(C(N(CC(=O)NC)C)=O)CCCC1 19410,C(=O)(C(C#N)C(C)(C)C)N1C(CC)CN(C(c2c(C)c[nH]c2CC(N)=O)=O)CC1 19411,C1(CC(=O)N(CCCCO)CCCC)CCN(C(=O)C(C)CSC)CC1C1CC1 19412,CN1CC2CCN(C(=O)CC3CC3CNC(C3CS(=O)C3)=O)CC2C1 19413,c1(C(=O)NC2CC(C)N(C(c3ocnc3C3CC3)=O)CC2)ccc2c(c1)CCC2 19414,C(=O)(CS(=O)C(F)(F)F)NCC1C(N(C)C)CN(C(CC=CC=C)=O)C1 19415,CCCCCC(COC)C(C)NC(=S)NCCC(F)(F)F 19416,N1(C(C2N(C(C)(C)C)CC2)=O)CCCC2CN(C(=O)C3CC3)CC12 19417,N1(C(c2c(SC)cccc2)=O)CCCCC(NC(C23CC(C(F)F)(CO2)C3)=O)C1 19418,C1(CC(N2CCCC(CC=C)C2)=O)CN(C(C2(CCC)CC2)=O)CC12CC2 19419,C1(C(N2CCN(C(CN(CC#C)C(=O)OC(C)(C)C)=O)CC2)=O)COCCNC1=O 19420,c1(COCCN(C(CC)CC2CC2)C=O)cccc(F)c1Br 19421,c1(C(=O)NC(C(C(C)C)O)c2ccccc2)n[nH]c2c1CCCCC2 19422,N1(C(CCC=C)=O)CC(C2CN(C(=O)CCCOc3ccccc3C)C2)C1 19423,CCC(CC(=O)NC1(C(=O)NC2CCN(C(C)=O)C2)CC(F)C1)C1CCC1 19424,Cn1nc(C(N2CCCCC2CCC(=O)NCC(C)(F)C(C)(C)F)=O)ccc1=O 19425,c1(NC(CC)CNC(=O)C(C)(C)C2CCCCC2)nccc(OCC)n1 19426,C12(CNC(c3c(C(C)C)cccc3)=O)CCCC1CN(C(=O)C(C)N(C)C)C2 19427,c1(N(C)C)ncc(C(=O)NCC2CC(O)CN2C(c2ccc(O)nc2)=O)cc1Cl 19428,c1(C(=O)NCCN(C)C(C2CCCN2Cc2ccc(F)cc2)=O)csc(C#N)c1 19429,N1(C(=O)Cc2ccc(Br)cn2)CCN(C(=O)Cc2cc(Cl)sc2Cl)C(CO)C1 19430,C(=O)(C1=COCCO1)NCC(C)(C1CCC1)NC(c1cc(CN(C)C)on1)=O 19431,C(=O)(C1=C(Cl)CCOC1)NCC1N(C(CCCCCN(C)C)=O)CC(O)C1 19432,Cc1nc(C)n(O)c1C(=O)NC1CCCN(C(=O)C(C)(C)C(N)=O)C1 19433,N1(C(CC(C)n2ccnc2)=O)CCCC(CNC(C2(C3CCCO3)CC2)=O)C1 19434,C1(C(N2CCC(C(C)NC(=O)C(C)(C)F)CC2)=O)CC2(CCO1)CC2 19435,c1(OC)cc(C(=O)NC(c2nc(C(=O)N(C)C)cs2)=O)cnc1C(F)(F)F 19436,N1(C(C=CCN(C)C(c2ccc([N+](=O)[O-])o2)=O)=O)CCC2CCCCC2C1 19437,C1(C(N2CC(COC)(NC(=O)Cc3sc(O)nc3O)C2)=O)C2CCC1(C)C2(C)C 19438,Cc1ccc(C)c(COC(=O)CCCC(=O)C2CC2)c1 19439,Cc1cc(C(N)=O)cc(C(=O)N(C)CCN(C(C2CCCC2(F)F)=O)C(C)C)c1 19440,N1(C(CNC(c2n[nH]cc2CC2CC2)=O)=O)CCC2(CC1)CN(C(C1CC=CC1)=O)C2 19441,C=CCC(C)(C)C(=O)NC1CCC1NC(c1cccc(C(C)=O)c1)=O 19442,O=S(=O)(c1ccc(N2CCC3(C2)CC(F)(F)C3)c(Br)c1)NCC1=CCCCC1 19443,C=CCC(C)(CC)C(=O)N1CCC(C)(CC(=O)NCCc2cc[nH]n2)C1 19444,N1(C(c2nsnc2O)=O)CCC(F)(C(=O)NCCN2CCCC2=O)C1 19445,CC(O)(CNC(=O)C(C1CCC1)NC(c1cc(O)ccc1F)=O)C(F)(F)F 19446,N1(C(=O)Cc2ccc(Br)cc2)CCC2OCCN(C(C3CC(O)C3)=O)C2C1 19447,C1(C(=O)NCCc2cc(C(=O)NCC3CN(C(C)C)C3)no2)CCC(O)CN1C 19448,c1(OC)ncc(Cl)c(N2CCCC(NC(=O)CNC(=O)CC3CCCC3)C2C)n1 19449,N1(C(C(c2ccn(C)n2)C)=O)CC=CC(NC(=O)C(O)CCN(C)C)C1 19450,N1(C(c2c(C)nsc2)=O)CCC(C(C)NC(=O)CC2CCCO2)CC1 19451,Cn1nc(C(=O)NCC2CCCN2C(C2C(C)(C)C2(F)F)=O)c2c1CCCC2 19452,c1(C(N2CCC(OC)(CNC(=O)Cn3ncnn3)C2)=O)c(F)ccc(F)c1Cl 19453,C1(C(=O)NCCc2c(C(N(CCC(=O)NC)C)=O)c[nH]n2)OCCOC1C 19454,O=C(CC1CC2C=CC1C2)NOCC1CCOC1.C12(CC(F)C1)C(=O)N2 19455,C(C(C)(C)C(=O)NCC1CCC(CC)CC1)NC(CCSCCC)=O 19456,O=S(=O)(c1cnc(N2CCCC(F)C2)c(Cl)c1)NC1CCC1 19457,C1(CC=C)(NC(=O)CC(C)F)CCCN(C(c2cc(C(F)F)ccc2Cl)=O)C1 19458,CC(C(=O)NCC1(O)CCCN(C(c2ccn3c2CSCC3)=O)C1)C1=CCCC1 19459,CC(C(=O)N1CCCC1C(C)NC(C1(C)CCC(=O)N1)=O)S(N)(=O)=O 19460,Cc1cccc(F)c1C(=O)NC1CC(N(C)C(C2CC3COCC3C2)=O)C1 19461,N1(C(CSCC#C)=O)CCC(NC(=O)C(C(C)C)n2cnnn2)C1C1CC1 19462,C(=O)(CC(C)CNC(C1CCNC(=O)C1)=O)NC(COC)COC 19463,c1(C(=O)NC(CN(C(C2(C)CC2C(F)(F)F)=O)CC)C)ccc(C)cc1C 19464,C1(C(=O)NCC(=C)Br)CC2CC1CN(C(=O)CCC1OCCO1)C2 19465,N1(C(C=C(C)c2ccccc2)=O)CC(N=[N+]=[N-])CC1C(=O)NC(C)CCC1CC1 19466,N1(C(=O)CCc2cccs2)CCCN(C(C2CC3CC2CC3O)=O)CC1 19467,N1(C(C2(F)CCC(C)CC2)=O)CCOC2(C1)CN(C(=O)CCC1CC1(C)C)C2 19468,c1(OCC)ccc(C(=O)NCC2CN(C(c3ccnc(C)c3)=O)CC2C)cc1O 19469,C1(NC(c2n(CC)cc(Cl)c2)=O)CCCCN(C(=O)C=Cc2ccc(C)cn2)C1 19470,N1(C(c2c(OC)ccnc2)=O)CCN(Cc2ccccc2)CC12CCC2 19471,N1(C(C(CCSC)O)=O)CC(F)(F)CC1(C)CNC(=O)Cc1cnc(C)o1 19472,CC1(NC(=O)CNC(N)=O)CCN(C(C2CCCC(F)(F)C2)=O)CC1 19473,C1(C(=O)NC(C(=O)NCCC(=O)OC(C)C)Cc2cn[nH]c2)CCCCCCC1 19474,n1(CCC(=O)NC(CC(CC)=O)C(=O)O)ccc2ccc(F)cc12 19475,N1(C(CC2CCC(NC(CN=[N+]=[N-])=O)C2)=O)CC=CC(O)C1 19476,c1(COC)onc(O)c1C.C12CN(CC1C)C2.c1(NC)ccc(-c2ccco2)cc1 19477,C(C(O)C(=O)N(CC(C)NC(=O)C(CN(C)C)N(C)C)C)=CCCC 19478,c1(C(=O)NC2CCC(C(=O)NC3(C4CCCO4)CC3)CC2)nnc(O)nc1O 19479,c1(CCC)nc(C)c(C(=O)NCC2CC(NC(=O)C=Cc3cccs3)C2)s1 19480,CCC(CC)(CCNC(=O)CN1CCC(=O)CC1)NC(C1C(C)(C)C1(C)C)=O 19481,C(C)(CC(C)CC(C)C)(c1n(CCC)nnn1)NCc1ccc(CC(=O)OC)o1 19482,c1(OC)cc(C(=O)NCCC2CCN(C(c3ccc(Cl)cn3)=O)CC2)nc(C)c1 19483,C1(N(C(c2nc(C)sc2)=O)CC2CC2)CCN(C(=O)CC2(O)CCOC2)CC1 19484,Cc1nc(N2CCN(C(C34CCOC3CCOC4)=O)CC2C)c(Cl)cc1C#N 19485,C1(CNC(COCCCC)=O)CC2(CCN(C(c3cc(C4CC4)ns3)=O)CC2)C1 19486,N1(c2ncc(NC(C)=O)cn2)CC2CCC(C1)N(C(=O)CSc1nc[nH]n1)C2 19487,c1nc(C(=O)O)c(N)s1.c1(SC(c2cc(OC)no2)C(=O)OCC)ccc(F)cc1 19488,c1(CC(=O)NC2CN(C(C3CCC(CCNC4CC4)C3)=O)C2)csc(S)n1 19489,c1(C(=O)OC)ncc(C(=O)N(CC(C)NC(=O)C(C)c2cc[nH]n2)C)s1 19490,C1(C(=O)NCC(C)CNC(=O)CC2COC(=O)N2)CCC12CCC2 19491,N1(C(C(C)C2CCCO2)=O)CCC2CCN(C(c3ccc(O)nn3)=O)CC2C1 19492,c1(C(C)C)nnc(C=CC(=O)NC2CCCCC2NC(=O)CCn2cccn2)o1 19493,Cc1cccc(C)c1NC(=O)C(N1CCCC(c2nncs2)C1)c1cncs1 19494,C(c1cc(Cl)ccc1Cl)=CC(N1CC(CNC(C2(COC)CCC2)=O)C2C1C2)=O 19495,c1(OC)ccc(C(N2CC(NC(=O)CC(C)OC)C(F)C2)=O)c(F)c1 19496,C(C)(CC(=O)N1C2CCC1CC(NC(C1(CF)CC1)=O)C2)(C(F)(F)F)N(C)C 19497,C(=O)(C(F)CC(C)(C)NC(c1ccc(O)cn1)=O)N1CCN(C)CC1 19498,C(C(C(=O)NCC(CC)NC(=O)Cc1cncn1C)c1ccccc1)OCC=C 19499,S(=O)(=O)(c1cnn(C)c1)N1CC(C(N2CCC(CC#C)CC2)=O)C1 19500,S(=O)(=O)(c1ccc(NC2CCC2(C)C)c(F)c1)N(C)CCOC1CCCOC1 19501,c1(OC)ncc(C)cc1C(=O)NCC1CC(CNC(C2CCC(F)(F)C2)=O)C1 19502,N1(C(CCC#CC)=O)CCc2nc(CNC(c3cc4n(c3)CCCC4)=O)sc2C1 19503,C1(CNC(c2cc(C(F)F)cs2)=O)CCCN(C(c2conc2C2CCC2)=O)C1 19504,C1(C(C)OC(=O)CC(c2cccnc2)NC(=O)OC(C)(C)C)CC2(C1)CC(O)C2 19505,c1(CC)ccnc(C(N2CCN(C3CN(C(=O)C(F)CC4CC4)C3)CC2)=O)c1F 19506,N1(C(Cc2n(C)cnc2)=O)CCN(CC(C2CC2)NC(=O)CC2(O)CC2)CC1 19507,c1(C(=O)NCCN(C(C=CSC)=O)C)cccc2c1OCCN2 19508,C1(C2CCCN(C(=O)C3=CCCC3)C2)(NC(c2cc3cnccc3o2)=O)CC1 19509,c1(CC)nn(C)c(Cl)c1C(N1CCC(C)(CNC(C2CC23CCC3)=O)C1)=O 19510,c1(OC)ccn2ncc(NC(=O)NCCOCC(F)(F)C(F)F)c2c1 19511,C(C(=O)NCCC1(O)CN(C(c2ccnc(O)c2)=O)C1)(C(C)C)NC(C)=O 19512,C12(NC(COC(C)C)=O)CCC(NC(c3cc(Cl)ncn3)=O)(CC1)C2 19513,CCC(CC(=O)N1CC(O)(CN(C)C(c2cc(C(N)=O)ccn2)=O)C1)C1CC1 19514,c1(C(=O)NCC2CCCCN(C(C(C=C)O)=O)CC2)c(C)nn2c(C)cccc12 19515,N1(C(C2CCCN(c3c(C#C)nccn3)C2)=O)Cc2ccccc2C1C(=O)OC 19516,C(C)(C)(CCCC(=O)N1C2CCCC1COC2)NC(C(CC)COC)=O 19517,S(=O)(=O)(c1ccc2ccccc2c1)N1CC2N(C(=O)C(F)Cl)C(COC2)C1 19518,N1(C(C2C(C)(C)C(=O)C2)=O)CCC(C2CCN(C(C3CCC3)=O)CC2)C1 19519,C12(CC(=O)NCCCCCN(C(C3CC(SC)C3)=O)C)COCC(C1)C2 19520,C1(CNC(CC(CNC(=O)C(N2CCOC2=O)C)OC)=O)CCCCC1(C)C 19521,c1(C(N(C(CNC(C2(C)C(C(=O)OC)C2)=O)C)C)=O)cc(-c2ccncc2)on1 19522,C(=O)(C(C)CC(C)(F)F)NC1C(NC(C=CSC)=O)COC1 19523,C1(C(=O)NCCC(N)=O)C=CCN1C(=O)CCC1CCC(=O)C1 19524,Cc1cc(C(=O)NC2CCC2NC(=O)C=CBr)cc(Cl)c1Br 19525,c1(OC)ccc(C)c(C(=O)NCC2COCC2NC(=O)C(C)OCC2CC2)c1 19526,C12(C(=O)NCCCC3(NC(C4C(C)OCC4)=O)CC3)CC3CC1C2C3 19527,C1(C(=O)Nc2n[nH]c(-c3ccc(Cl)c(Cl)c3)n2)CCn2c(O)nnc2C1 19528,C1(NC(CNC(=O)OC)=O)CCCCN(C(=O)CC2CN(C)CC2O)C1 19529,C(=O)(C(CC(C)C)C(N)=O)N1CCCC(O)(c2cn(Cc3c(C)sc(Br)n3)nn2)C1 19530,C(=O)(C(F)(F)CO)NCC(C1CC1)NC(=O)C(F)=CCCF 19531,N1(CC)CCOCC1C(=O)N(CC(C)(C)CNC(C1(COC)CC1(F)F)=O)C 19532,N1(C(c2cc(CC)ncc2)=O)CC(C)(C)CC1CNC(C1CCCSC1)=O 19533,c1(C(C)C(=O)NCCCNC(=O)CC2NC(=O)NC2=O)ccc([N+](=O)[O-])cc1F 19534,N1(C(CS(=O)(=O)NCC)=O)CC2CC1CCC2NC(C1CC(OC)(OC)C1)=O 19535,C1(C(C(=O)OC)NC2CC(n3cncn3)C2)CC2CCC1C2 19536,C(=O)(C1SCCc2ccccc21)N1CC(CNC(C(=O)NCC)=O)C(C)C1 19537,c1(C(N2CCN(CCCNC(C3C(C)C3)=O)CC2)=O)cccc(F)c1Br 19538,Cc1ccoc1CNC(c1cnns1)=O 19539,C1(C)(CNC(C(C)C2CCCC2)=O)CCN(C(=O)CC2SC(=N)NC2=O)CC1 19540,N1(C(CC(CC)C)=O)CCCCC2(CCN(C(c3cccc(CSC)c3)=O)C2)C1 19541,c1(C(=O)NCC2CN(C(c3c(C)snc3)=O)CC2C)cc(Cl)cc(Cl)c1O 19542,Cc1ccc(C(=O)OC(C)(C)C)cc1C.C12CN(CC1O)C(=O)NCCC(=O)NC2 19543,C1(NC(C2=NNC(=O)C2)=O)CCCC2CN(C(C3CCCN3C3CC3)=O)CC12 19544,CC(C)CC(O)C(=O)NC(Cc1ccco1)C(=O)N(C)CC1(O)CCC1 19545,O=C(CCCCCCCO)NCC1CCCN1C(=O)Cc1cnc2[nH]ncc2c1 19546,C12(C(=O)NCCCCC)CCCC1CCN2C(c1ccc(CC)cn1)=O 19547,c1(NS(CC#N)(=O)=O)ccc(C2(Nc3nc(-c4ccccc4)no3)CC2)cc1 19548,C(=O)(CCC(CC)OC)NC1CCN(C(CCCC)=O)C1CC 19549,CCC(CC(F)F)C(=O)N1CCCCC1CNC(c1c(F)ccc(C)c1N)=O 19550,C1(CC)CN(c2ccccc2)CCN1C(c1cc(-c2ccccn2)[nH]n1)=O 19551,Cc1cc(CNC(c2nnnn2CCC2(C)CC2)C2CC23CC3)c2c(c1)CCC2 19552,C=CCC(CC)N=c1[nH]c(N2CCC(OCCO)C2)nc2ncn(C)c12 19553,C1(N(C(C(C=C)OC)=O)CCC)CCN(C(c2nnsc2SC)=O)CC1 19554,C(=O)(C(F)(F)C(O)C(C)C)NC(C1CN(C(CC2CCCC(OC)C2)=O)C1)C 19555,C1(CNC(CN(CCC#C)C)=O)CCOC1C(=O)N(C1CC(O)C1)C 19556,N1(C(=O)NC(c2nc(=O)[nH][nH]2)C)CCCC2(C=CCO2)CC1 19557,N1(C(CC(=C=C)C)=O)CCN(C(=O)C(C)Oc2ccc(Cl)c(Cl)c2)CC(O)C1 19558,c1(C(=O)NCC2CC(COC)CN2C(=O)C#CC2CC2)ccc(F)c(C2CC2)c1 19559,C1(C(N2CC(C)OCCC2)=O)CCCCCCN1C(=O)CCCCC#N 19560,C1(C(=O)OC)CCC2CN(C(=O)NC3CC(c4ccncc4)C3)CC12 19561,CC(C)C(Cc1ccccc1)C(=O)NCCC(C)N(C)C(c1cc(C#N)c[nH]1)=O 19562,c1(C(N2C(CNC(Cc3c(C)noc3)=O)CCC(C)C2)=O)cc(C#N)ccc1O 19563,C1(NC(c2c(CCC)n[nH]c2)=O)CN(C(C2C(C)(C)C2(C)C)=O)CCC1O 19564,CC1(CNC(=O)NC2CCN(C(=O)NC(C)(C)C)CC2)OCCc2sccc21 19565,N1(CC)CC(C(N2CC3CC2C3NC(c2nccnc2N)=O)=O)CCC1=O 19566,c1(N(CCC#C)CC#C)ccc(C(=O)CC)cc1I 19567,c1(C(=O)OCC)ccc(N(C2CCCN(C(c3cc(C(F)F)[nH]n3)=O)C2)C)nc1 19568,C1(C(=O)NC(C)CC(=O)O)CCCCC1C(N)=O 19569,C(=O)(CN1C(=O)CSc2ccccc21)N1CC(NC(C2C(C)CCC2)=O)(CO)C1 19570,c12cccc(c1)OCC21CC1.C1(NC(C=C)C2CCC2)CC(CO)C1 19571,N1(C(c2ccc(NC=O)cc2)=O)CC2C(CC(=O)Nc3c(C)cc[nH]3)C2C1 19572,O=C1CCC(C(N2CCN(C(=O)Cc3cn(C4CC4)cn3)C(CO)C2)=O)CCO1 19573,c1(SC(C)C)cc(N)nc(NCc2cn(C(C)C)nn2)n1 19574,c1(C(N(C(C)CNC(C2CCCNC2=O)=O)CC)=O)ccc(-n2ccnc2)nn1 19575,C#CC1CC2(CC2)CN1C(=O)CCC1CCCCN1C(=O)CCC(C)CC 19576,C1(N(C(=O)CC#N)CC)CCCN(C(=O)COCc2cc(C)[nH]n2)C1 19577,c1(NC(C(c2cccs2)NC(C(C)OCOC)=O)=O)cnc(F)nc1 19578,C1(CNC(C(C)C(F)F)=O)C(O)C(O)CN1C(=O)CC1(O)CCOCC1 19579,C1(NC(c2cc(-c3cccnc3)no2)=O)CCC(NC(C2CC2Br)=O)CC1 19580,N#Cc1ccc(C=CC(=O)NCCNC(=O)Cc2csc3ccccc23)cc1 19581,c1(OC)ccc(NC(C2CC3CC3N2C(c2cc(F)ncc2Br)=O)=O)c(F)c1 19582,CC1(F)CC2(CN(C(=O)CCC3CCN(C(=O)C(C)(C)N=[N+]=[N-])C3)C2)C1 19583,c1(C(=O)NCC(N(C(=O)C=CC2CCCC2)C)C2CC2)cc2cccn2c(O)n1 19584,N1(C(c2cc(C)sc2)=O)CCC(CNC(=O)CCOCC(C)C)CC1C 19585,N1(C(c2scc(C)c2C)=O)CCC2(CC2NC(C2CC(C(C)C)=NO2)=O)C1 19586,C1(NC(CCCCCSC)=O)CCN(C(=O)CC2C=CS(=O)(=O)C2)CCC1(F)F 19587,C1(CCNC(C23CC(C)(C2)C3)=O)CCCCN1C(=O)CC1(C)CCCO1 19588,CN1C(=O)CC(C(=O)Sc2ccccc2)C1SCC#N 19589,Cc1c(Br)cc(C(N2CC3CC3(C(=O)NCc3ccc[nH]3)C2)=O)cc1Br 19590,C(=O)(C(O)CC(N)=O)N1CC(NC(C23CC(OC)C2C3)=O)C(O)C1 19591,c1(NC2(CC(=O)NC(CC(C)C)CO)CCC2)ncnc2c(Br)csc12 19592,N#CC1(C(=O)NC2CC(NC(=O)CCF)C2)CCCC(=O)C1 19593,C1(NC(C2C(CCC)CCC2)=O)CC12CCC(NC(c1ccc(Cl)cn1)=O)CC2 19594,N#Cc1ccccc1-n1ccc(C(=O)OCCCc2cnoc2)n1 19595,N1(C(c2cnc(CC(C)C)s2)=O)CCN(C)C(CNC(=O)C(C)CN(C)C)C1 19596,CC1CN(C(C2(F)CCOC2)=O)CCC1C(N1CC2(CC2)C1)=O 19597,CCCCC(CC)CC(=O)N(C)CC1(NC(C2Oc3ccccc3C2C)=O)CC1 19598,C1(C)CCC1.C(C(=O)NCCC=C)N(C)C(=O)OC(C)(C)C.C12CC1CNC2=O 19599,c1(NC(C2CCCN(C(c3cc(CC)ncn3)=O)C2)=O)cccc(Cl)c1O 19600,C1(CC(=O)N(C2CCCN(C(C3C(Cl)(Cl)C34CC4)=O)C2)CC)COCCOC1 19601,C(=O)(C(CCN(C)C)NC(=O)C(C)OC)N(C(CC)C)CCO 19602,c1(C(N(C2CCN(C(=O)C=Cc3cccs3)C2)C)=O)cc(C(F)(F)F)ccn1 19603,N1(C(CC(=O)NC2CC2)=O)CC2CCC1C(CNC(c1cc(C(F)F)cs1)=O)C2 19604,C1(C)(CNC(c2n(C)ncc2)=O)CCCN1C(=O)CCc1ccc(CO)cc1 19605,Cc1ccnc(SCC(=O)NC2(C)CCN(c3nnco3)C2)n1 19606,c1(OC)sc(C(=O)NCC2(F)CN(C(=O)C(C)(Cl)Cl)C2)cc1Br 19607,C1(C(N(CC(CNC(C(C)=C(C)C)=O)(C)C)C)=O)CCCCC(F)(F)C1 19608,CC1C(NC(c2ccc(O)c(F)c2)=O)CCCN1C(c1coc(C(F)F)c1)=O 19609,c1(OC)cccc(F)c1C(=O)NC1CCN(C(C2CCC(F)CC2)=O)C1 19610,N1(C(C(c2cn(C)nc2)=O)=O)CCCC2(NC(=O)COC3CCCC3)CCCC12 19611,Cc1c(C(=O)NC23CC(NC(c4cc(O)ccc4F)=O)(C2)C3)cncc1Br 19612,C(C)(CCC1CC1(Cl)Cl)(c1nnnn1Cc1ccccc1)NC1CC(OC)C1 19613,c1(N2C(CNC(C3(C(=O)NC)CC3)=O)CC3COCC32)ncc2scc(Br)c2n1 19614,CC1CC(C(N2CCCC(CF)C2)=O)CCN1C(=O)CCc1cnccn1 19615,c1(CCC)ncc(C(=O)NCC2CCN(C(=O)C(C)c3ccsc3)C2)s1 19616,N1(c2nnc(C)c(C)n2)CC(C)(C)CCC1CNC(=O)C(C)Cc1cnn(C)c1 19617,C1(C(=O)NCCN(CCCF)C)CC(O)CCN1C(c1ccn(C(F)F)n1)=O 19618,C#CCC(CC(=O)NC1CCCC1)OCC=CC(N1CC(=CC)C1)=O 19619,C1(C(CNC(C2CCNCC2)(C)C)(C)O)CCCCC1 19620,c1(C(=O)NC2C3(CC(NC(C(CC=C)(F)F)=O)C3)C2)ccc2cnc(C)n2c1 19621,N1(C(C2(OC)CCSC2)=O)CCOC(CNC(=O)COc2cnn(C)c2)C1 19622,c1(C(CC)C)nc(C)cc(=NCC2(O)CN(C(=O)C(C(C)CC)OC)C2)[nH]1 19623,c1(C(N2CCC(OCc3ccccn3)CC2)=O)cnccc1Cl 19624,c1(CC(N2CC=C(CNC(C3(CC4CC4)CC3)=O)CC2)=O)ccc2[nH]ccc2c1 19625,CC(C)(C)C(O)C(=O)NCC1CC(NC(c2cccc(-c3cnco3)c2)=O)C1 19626,C(CC(C(=O)O)NC(=O)CCc1cncnc1)c1cn(C(COC)COC)nn1 19627,CCCCS(=O)(=O)CC(=O)N1CC2C(CN=c3[nH]ncs3)C2C1 19628,C1(NC(c2c(C)c[nH]n2)=O)CC2C1CCN2C(=O)C=C1CCCCC1(C)C 19629,N1(C(C=C(C)C2CC2)=O)CCSCC1C(=O)NC(C)C(N)=O 19630,c1(C2(C(NC(C(=O)NCCN(CC)CC)=Cc3cccs3)=O)CC2)ncccc1F 19631,C1(CNC(=O)OC(C)(C)C)(COC(C2C=CCCC2)=O)CC2(CC(F)C2)C1 19632,Cc1cc(C(N2CC(O)(CNC(=O)CC3(O)CCCN(C)C3)C2)=O)cc(C)c1F 19633,c1(-c2c(C(N(CC(=O)NC)Cc3ccccc3)=O)scc2)ccc(C)c(C)c1F 19634,CCC(CC)CCC(=O)NC1CN(C(c2cnn3cccc3c2)=O)CC1O 19635,c1(OC)ccc(CNC(=O)C(c2ccc(I)s2)N(CCF)C2CC2)cc1 19636,C1(CCC(=O)N(CC(O)CNC(c2csc(C3CC3)n2)=O)C)CCC(C(N)=O)O1 19637,C1(C(=O)NCC(C)(C)F)C2CC(O)C(C2)N1C(c1cccc2cc[nH]c12)=O 19638,C1(C)(NC(CN(C(C)C)C)=O)CCCCC1C(=O)NCC1CCNC(=O)C1 19639,CC1(CNC(C2(C)C=CCC2)=O)CCN(C(=O)C(c2csc(=N)[nH]2)=O)C1 19640,C(=O)(C1=CCOCC1)NC1CCC(NC(C2C(C#C)C2(C)C)=O)CC1 19641,CN1CC(C(=O)NCC2(NC(C3CC3c3cccs3)=O)CC2)NC1=O 19642,N1(C(C2(COC)CCCCC2)=O)CCN(C(=O)C(F)C(F)(F)F)C(C)C1 19643,C=CC(C)(C)CC(=O)NCC1(C)CCCN1C(=O)C=Cc1scnc1C 19644,CN(CCCC(=O)N1CCN(C(=O)C(C)(C)O)CC1c1ccnn1C)N=O 19645,c1(C(=O)NC2(C)CCN(C(C3(CCF)CC3)=O)C2)ccc(Br)cc1[N+](=O)[O-] 19646,c1(CNC(C2(CNC(CCc3onc(C)n3)=O)CC2)=O)cc(O)ccc1F 19647,c1(C(N(CCCCCNC(C(C)OCC2CC2)=O)C)=O)ccc(N(C)C)cn1 19648,N1(C(CCCC#CC)=O)CC(C(=O)NC(C)(CO)CCC)CC(C)(C)C1 19649,N1(C(CSC2C(=O)OCC2)=O)CCC2(C1)CN(C(c1c(Cl)nsc1Cl)=O)C2 19650,N1(C(CC2C(C(=O)OC)C2(C)C)=O)CCC(NC(c2nn(C)cc2C)=O)C(C)C1 19651,c1(C(N(CCOCCNC(C2C(OC)CC2)=O)C)=O)csc2nccn12 19652,c1(C(=O)NCC(C)NC(c2n(CC)nc(C)c2)=O)ccc(F)c(C)c1C#N 19653,N1(C(c2occ(C)c2)=O)CC(C)(C)CC1C(=O)NCc1ccc(Cl)o1 19654,CC1=NOC(C)(C(=O)NCC(CO)NC(C2CCN(C)C2=O)=O)C1 19655,c1(CC(=O)NC(CNC(C2CC(C#C)(O)C2)=O)C(C)C)noc(C)c1C#N 19656,C=CCC(CNC(C1CCOC1)=O)C(=O)NC1CCN2CCC1C2 19657,CCC(CC(=O)N1CCC(OCCNC(C2CCN2C(C)(C)C)=O)CC1)C(C)C 19658,N1(C(CN(C)C)=O)CC2C(NC(=O)CC(C)(C)C(C)(F)F)CS(=O)(=O)C2C1 19659,C1(NC(c2ccc(CNC(C(COC)COC)=O)cn2)=O)CN2CCC1(F)CC2 19660,Cn1nc(C(N2CCC(NC(C3CCN(CC(F)(F)F)C3)=O)C2)=O)cc1F 19661,C(=O)(C(F)C1=CCCCC1)NCc1ccc(CNC(C2C(=C)CC2)=O)c(F)c1 19662,C(=O)(CCC(F)(F)F)N1CCCC(C(=O)Nc2c(CC)nn(C)c2)C1 19663,c1(C(N(C)CC2(CNC(C3CC3Cl)=O)CC2)=O)ccc(CN2CCCC2)o1 19664,c1(C(=O)NC(C)(CNC(C2COCOC2)=O)C2CC2)c[nH]c2nccc-2c1 19665,N1(C(CC(C)(C)C)=O)CC2(CCCN(C(c3cccc4nscc34)=O)C2)C1 19666,C(=O)(C1=CNC2=NCCCN12)NCC1N(C(CC2C(OCC)COCC2)=O)CCC1 19667,c1(C(=O)NC2CN(C(c3cn(CC(C)O)c(=O)cc3)=O)C2)cc2ccccn2n1 19668,c1(C(=O)NCC(CC)N(C(=O)C(C)C(F)F)C)ccc(N)c(F)c1F 19669,c1(C(N(C2CCCCN(C(C=CC(=O)N(C)C)=O)C2)C)=O)ccnc2c1CCC2 19670,c1(C(=O)NCCC(C(=O)NCC(CC)C#N)(C)C)nccc2[nH]ccc12 19671,C1(NC(CC(=O)OCC)=O)CN(C(c2ccnn2CC)=O)CC12CCC2 19672,N1(C(c2c(CC)cccn2)=O)CCCC(C2CCCN(C(=O)CSC)C2)C1 19673,n1(CC)ccc(C(=O)N(CC(C)(C)NC(c2cc(C)c(Cl)s2)=O)C)cc1=O 19674,N1(C(c2scc(C)c2C)=O)CCN(C(C2CC(N(C)C)C2)=O)C(c2cn[nH]c2)C1 19675,N1(C(C(C)NC(N)=O)=O)Cc2nccnc2CC1C(=O)NC(C1CCOCC1)C 19676,C1(NC(COCCCOC)=O)CN(Cc2cc(C3CCCCC3)on2)CCC1C 19677,CC(N=c1ccc(C#N)n[nH]1)C1CN(C(c2ccc(CC3CC3)cc2)=O)CCO1 19678,C1(NC(CN(S(CC)(=O)=O)C)=O)CCCCC1NC(=O)C=Cc1ncco1 19679,Cc1ccccc1OCC(C)OC(=O)C(=O)NC1CC1(c1ccccc1)C 19680,c1(C(=O)NCC(CO)NC(C(C(C)C)OCC)=O)nc(C)c(C)nc1C 19681,CCC(C)(CNC(c1c[n+]([O-])c(C)cn1)=O)C(=O)N1CCCCC1C 19682,c1(C(=O)NCCCCNC(C2CC3CCC2C3)CC)cc2ccccc2o1 19683,N1(C(c2ccc(C)nc2C)=O)CC(NC(=O)CN2CC(=O)NC2=O)C(C2CC2)C1 19684,C1(C)(C(=O)NCCOCCN(C)C(c2cc(Br)cn2C)=O)CCCNC1=O 19685,N1(C(Cc2cn(CC)nn2)=O)CC(NC(=O)CNC=O)CC(F)(F)C1 19686,C(CC(O)C(=O)N(CCCNC(=O)CC1C=CCCC1)C)SC 19687,N1(C(C2C(OCC)C2)=O)CCC(NC(=O)C(N2CCCCCC2)C)C(C)C1 19688,C#Cc1cc(NC(=O)C(C)N(C(C2(C)CC2(C)C)=O)C2CC2)cc(F)c1 19689,c1(C(CNC(C(=O)NC2C(OC)CCC2)=O)OC)ccncc1F 19690,N1(C(C=C(CCC)C)=O)CCC2(C1)CN(C(C1(F)CC1C)=O)CCO2 19691,C12(CNC(C(CC)OC)=O)CN(C(=O)COCC(C)C)CC(F)(C1)C2 19692,c1(C(=O)NC(CCNC(c2nc(C)nn2C)=O)(C)C)nccc(N)c1Cl 19693,CC1CC(CNC(=O)C(=O)NCCc2cccs2)CC(C)C1.C1C(=O)N1 19694,c1(OC)cc(Br)c(C(=O)NCCN(C)C(c2nccc(C)c2N)=O)cc1OC 19695,N1(C(c2ccnc(NC3CC(=C)C3)n2)=O)CCC(C(=O)OC)C(O)C1 19696,c1(C(=O)NCC(CNC(c2nc(C(C)=O)sc2)=O)CO)nnc(C)cc1O 19697,Cc1noc(C)c1S(=O)(=O)N1CC2CN(S(=O)(=O)CCBr)C2C1 19698,c1(OC)cc(C(=O)NCC2CN(C(C3(OC)CC3)=O)C2)cc2cn(C)nc12 19699,c1(C(=O)OCc2onc(-c3c(C)cccc3)n2)c(C)ccc(F)c1[N+](=O)[O-] 19700,C(=O)(N=c1ccn(C2CC2)[nH]1)C1CC(OC)C1.C1(CC(=O)NC)(C(N(C)C)=O)CCC1 19701,c1(C(=O)NCCC2(O)CCCN(C(C3(N=[N+]=[N-])CC3)=O)C2)cccn2nccc12 19702,CCS(=O)(=O)CCCNC(N1CC(c2cc(C)ccc2C)OCC1C)=O 19703,N1(C(C2C(C(C)O)C2)=O)CC(C)CN(C(c2cccc(N)c2N)=O)C(C)C1 19704,N1(C(C(C=C)C)=O)CC(O)(C2(CNC(=O)COCc3cccc(C)c3)CC2)C1 19705,c1(N2CCC(C)(COC)C2)nc(=NC(C)COc2cccc(F)c2)[nH]c2ccsc12 19706,N1(C(c2c(CC)cno2)=O)CCC2C(C(=O)NCCCCC3CC3)C2C1 19707,c1(C(=O)NCC2CCN(C(C3ON=C(C)C3)=O)C23CC3)coc2ccc(C)cc12 19708,C1(N(C)C)CN(C(C2CC2(Cl)Cl)=O)CC1CNC(c1csc(O)n1)=O 19709,c1(C(N2C3CC(NC(CCC(C)(C)F)=O)CC2CC3)=O)cnnc2ccccc12 19710,c1(NC(C)=O)ccccc1SCC(N1CC(C)(NC(=O)CC2CCC(O)C2)C1)=O 19711,N=c1[nH]c(=NCC2(NC(=O)CC3CCC(O)C3)CCCC2)[nH]cc1[N+](=O)[O-] 19712,c1(C(N2C(C(=O)OC)(COC)CCC2)=O)ncn2c1CCNCC2 19713,CCC(Cc1ccccc1)CC(=O)N1CC(NC(=O)CCC(C)N(C)C)C1 19714,c1(CC)ccc(-c2ncn(C3CC(c4ccccc4)CCN3C)n2)c([N+](=O)[O-])c1 19715,N1(C(C(CC)(C)OC)=O)CCN(C)C(CNC(C2CN3CCC2CC3)=O)C1 19716,C12(C(N3C(CN(C(CCCC(C)C)=O)C)CCC3)=O)CC=CCN1CCC2 19717,C1(NC(c2ccnn2C2CC2)=O)COCCN(C(c2cncc(F)n2)=O)C1 19718,Cc1cc(CNC(C2CCS2(=O)=O)=O)oc1C(=O)NCC1(F)CC(CO)C1 19719,C(C1CN(C(=O)CC2(N(C)C)CCC2)CC1C(N1CCOCC1CSC)=O)=CC 19720,C1(NC(CC2CCN(C)C2=O)=O)CC2(C1)CC(NC(c1ccc(CO)cn1)=O)C2 19721,C1(C(N2CCN(C(c3c(CC)ncs3)=O)CC2COC)=O)CCc2nn[nH]c2C1 19722,C(C)(C(=O)NOC1CCOC1)(N(C(c1cccc(CC)n1)=O)C)C1CC1 19723,c1(SC)nccnc1C(=O)NCC(C)N(C)C(C1CCC1(F)F)=O 19724,C1(CNC(c2c(F)ccc(OC)c2)c2nnnn2C)CCOC2(CCC2)C1 19725,Cc1cc(F)cc(C(=O)NCC2CN(C(C34CCC3CC4)=O)CC2(C)C)c1N 19726,n1(CCC)c(C)cc(C=CC(=O)NC23CC(NC(=O)C(C)CC(N)=O)(C2)C3)c1C 19727,N1(C(c2c(C)nn[nH]2)=O)CCCCCCC1C(N1CCC(C)(CO)C1)=O 19728,Cc1cn(C)nc1C(=O)NC1(C)CN(C(C2CC(F)(F)C2)=O)C1 19729,C(=O)(C1=CCN(C(=O)CC(C)C2CC2)C1)N(C(CC(CC)C)C)C 19730,N1(C(C(C)NC(N)=O)=O)CCn2cc(C(N3CCC(OC(F)(F)F)C3)=O)nc2C1 19731,C1(C(=O)NC23CN(C(c4c(C)n(C)nn4)=O)C(CC2)C3)CNC(=O)CC12CCC2 19732,C#CCC(C)(CNC(=O)CC1CCCN1C(=O)C(C)C(C)(C)C)CO 19733,C(=O)(C1CCCc2nncn21)NCCNC(c1c(C(F)F)ccc(C)c1)=O 19734,N1(C(CSCc2ccc(C(C)C)cc2)=O)CC2CC1CCC2NC(C1(C)CC1)=O 19735,c1(C(=O)NC2CC(C)(NC(C(CC)CN(C)C)=O)C2)cc(O)cc(F)c1 19736,N1(C(C(C)=C2CCC2)=O)CCC(C)(NC(c2ccncc2C)=O)CC1 19737,C1(CNC(C=CC=CC)=O)CN(C(c2n[nH]cc2C2CCC2)=O)CCC12CCC2 19738,C1(OC)CCC2(C(N3CCC(C)C3CNC(C3C=C(C)CS3)=O)=O)CC12 19739,N#CC1(C(=O)NC2CC(CNC(C3(S(N)(=O)=O)CCC3)=O)C2)CC2CC2C1 19740,C=CC(C)(O)CC(=O)N(C(CC(F)F)C(=O)NCCCC(C)Cc1cn[nH]c1)C 19741,CCC(CC1CCCCC1)C(=O)NC1CCCCC1CNC(c1[nH]ccc1C)=O 19742,N1(C(C2CC(CC)C2)=O)CCCC(C)(CNC(=O)CS(=O)(=O)NC2CC2)C1 19743,CC(C)C(C)(C)C(=O)NCc1cc(C(=O)NC2CNC(=O)C2)n[nH]1 19744,C1(NC(C(C=C)O)=O)Cc2ccccc2C1NC(=O)CC1C(=O)ON=C1C 19745,C1(F)(CNC(c2cc(C)oc2C(F)(F)F)=O)CCN(C(=O)C(F)F)CC1 19746,C12(C(N(C3CC(=C)C3)C)=O)CC(NC(C3CC(C)(CC)C3)=O)(C1)C2 19747,Cc1cccc(C(=O)N(CC(C)N(C(=O)CCSc2ccccc2)C)C)c1C 19748,C=CC1(C(=O)NCCCCC2CCCN(C(=O)CC3CC34CC4)C2)CCCC1 19749,Cn1c(N(CCO)Cc2ccco2)ccc1C=O 19750,c1(C(=O)NC2CCC(NC(c3coc(O)n3)=O)CC2)ccc2c(c1)CCCC2=O 19751,C1(CC)CN(C(C23CC(F)(C2)C3)=O)CCC1NC(c1conc1C1CCCO1)=O 19752,C1(CNC(CCN(C(=O)CC2CCCC(O)C2)C)=O)OCCC1(C)C 19753,C(CCCCC(=O)N(C1CCN(C(c2cc(C)co2)=O)C1)C)OCC 19754,c1(C(N(CC(=O)Nc2ccc(SC)nc2)CC#C)=O)[nH]ccc(=O)c1C 19755,CC1(C)C=C(C(=O)NC(C)(CNC(C2(C(N3CCCC3)=O)CC2)=O)C2CCC2)C1 19756,C(=O)(CC(C)(C)C(F)F)NCCCCC(C)NC(C1CCS(=O)(=O)C1(C)C)=O 19757,c1(C(C)NC(=O)NCc2cccc(NC(=O)OC(C)(C)C)c2)cccc(Br)c1F 19758,c1(OC)ncc(C(N2CCC2COC2CCCC2)=O)cc1-c1cccc(CO)c1 19759,C1(NC(C(C)=CC2CC2)=O)CCC(C)N(C(=O)CCCn2ccccc2=O)C1 19760,C(=O)(CC(C)(C)NC(=O)C=CC1CCOC1)NC1C(CN(C)C)C1 19761,C1(C)(CNC(c2ccc(C(C)C)o2)=O)CN(C(=O)COC2(C)CCC2)CCO1 19762,n1(CC(=O)N(C2CCN(C(CC(=O)NCC(C)C)C)C2)C(C)C)ncn(C)c1=O 19763,N1(C(C2(CCC)CCC2)=O)CC2(CCC(CNC(=O)C(C)CC(C)(F)F)O2)C1 19764,Cc1cc(-n2cc(C(C(C)C)NC(=O)C(CO)NC(N)=O)nn2)cc(C)c1 19765,c1(OC(C)C)nccc(C(=O)NCC(CO)NC(C2(CO)CCC2)=O)c1F 19766,N1(C(c2ccc(CC)s2)=O)CCC(NC(c2c(C(F)F)nn(C)c2C)=O)C(C)C1 19767,C1(CCC(=O)Nc2cccc(CC)c2)CCCCN(C(c2cccnc2C)=O)C1 19768,C(CNC(=O)COCC1CCC1)(CC(F)(F)F)NC(C(c1c(C)cncc1)C)=O 19769,C1(NC(C2(F)C(C)OCC2)=O)CCCN(C(=O)CC2(CO)CCC2)C1C 19770,N1(C(CC(=C=C)C)=O)CC(CNC(=O)Cc2cnc[nH]2)CC(C)C1 19771,C1(NC(c2ccncc2Cl)=O)CC2CN(C(C3CCCSC3)=O)CC12 19772,C1(N(C)C(c2coc3c2COC3)=O)CCCC2CN(C(=O)CC3CC34CC4)CC12 19773,c1(C(=O)NCC2CC(CNC(C3COCC(C)O3)=O)C2)cc(=O)cc(Cl)[nH]1 19774,N1(C(c2cc(Br)ncc2Br)=O)CCC2CN(c3ncc(F)cn3)CC2C1 19775,c1(C(=O)NC(C(=O)NCCNC(=O)NC)CCOC)cccc2ccoc12 19776,C1(C(=O)NC2CCC3CC3CC2)CCOC2(CCN(c3cc(Cl)ncn3)CC2)C1 19777,C1(N(C(=O)C(O)C(C)(C)C)C(c2ccc(OC)nc2)C)CCCC12CCNCC2 19778,c1(C(=O)NC(COC)CC(C)(C)C)ccc2n1CCNC2 19779,N1(C(c2nc(CNC(C3N(C)CCOC3)=O)oc2)=O)CCC(O)C(O)C1 19780,C1(CC(=O)NC(CN(C(C23COCC(C2)C3)=O)CC)C)CC2CCC1C2 19781,Cc1cccc(F)c1CC(=O)Nc1nc(CNC(=O)Cc2cncn2C)cs1 19782,c1(C(=O)NCC(CC)NC(C2CNC(=O)N2C)=O)ccc2ccc(O)nc2n1 19783,CC1CCCN(C(c2cccnn2)=O)C1CCNC(c1cc(F)ccc1Br)=O 19784,N1(C(C(C)OCCCC)=O)CCCC(C)(CNC(C2(C)CCCO2)=O)C1 19785,N(C(=NCC=Cc1ccc(Br)cc1)NCc1ccnn1C)CC(=C)C 19786,c1(CC)nc(O)c(C(=O)NC2CCCCC2CNC(C2(C)CC=CC2)=O)cc1C 19787,N1(C(CC=CC)=O)CCN(C(=O)CSCCC)CC1CC 19788,C1(C(=O)NC2(C(C)O)CC2)CCCC(NC(C2COCC2(C)C)=O)C1 19789,N1(C(c2cc(I)c(F)cc2F)=O)CCC2C(CCN2Cc2cccc(Br)c2Cl)C1 19790,N1(C(Cn2c(C(C)C)nnn2)=O)CCC2CCC(C1)N2Cc1cc(C2CC2)on1 19791,C(C(C)C(F)C(=O)NCc1csc(C)c1C)NC(c1ncn(CC)c1)=O 19792,CC1C(C(=O)NC23CC(NC(C4OC(C)(C)OC4(C)C)=O)(C2)C3)C(O)C(=O)N1C 19793,c1(NC(C2CCCCN2C(c2ccnnc2O)=O)=O)cc(Cl)ccc1CO 19794,CCC1=C(C(=O)N2CC(NC(c3cnn4c3OCCC4)=O)C2)SCCO1 19795,c1(NC(C(COC(C)C)NC(CCC)=O)=O)nccc(C)n1.C1C(=O)N1 19796,C1(C(=O)NCC(C)(C)NC(c2cc(C(F)(F)F)no2)=O)C2CC2C2CC12 19797,C1(CC(=O)NC2C(OC)CCCC2)C2CCCC2N1C(c1nscc1C)=O 19798,N1(C(CCN(C(c2c[nH]c(=S)cn2)=O)CCO)=O)CCC2(C=CCO2)C1 19799,N1(C(c2ncc(C)cc2F)=O)CCC2C(CCCN2C(=O)CC(C)(F)F)C1 19800,C1(C(=O)NCCN(CCC)C(c2ccnn2CC(C)C)=O)CCCC1S(C)(=O)=O 19801,CCS(=O)CC(=O)NCC(c1ccc(F)cc1)NC(C1(OC)CC1)=O 19802,Cn1nc(C2CCC2)cc1C(=O)NCCCCCCNC(C12CCC1C2)=O 19803,C(=O)(CC(C)N(C)C)N(CC(C)N(C)C(c1sccc1Br)=O)C1CC1 19804,N1(C(C(C(CC)C)O)=O)CCCC2(C1)CN(C(=O)CN1CCP(C)(=O)CC1)C2 19805,CC1(C)CCOC(CNC(C2C(O)CCN2C(C2CN3CCN2CC3)=O)=O)C1 19806,c1(CC)cc(C(=O)N(CCCC(=O)NCCC(CC)CO)C)ccn1 19807,c1(-c2n(C)nc3c2CCCC3)nc(C2CCc3cc(Br)ccc32)no1 19808,c1(CCNC(c2cc(C)c(Br)s2)c2n(C(CC)C)nnn2)c(Cl)cccc1Cl 19809,N#CC1(C(N2CC(CNC(=O)CCCCCNC(N)=O)C2)=O)CC2CCC1CC2 19810,C(=O)(C(CC(N)=O)NC(=O)COC1CCCOC1)NCC(C=C)O 19811,C=CCCCC(=O)NCCC1(C(=O)NC2(C3CCC3)CC2)CCC1 19812,CC(C(C)(C)CO)NC(=O)C(C)(C1CC1)N(C(=O)COc1ccsn1)C 19813,c1(C(=O)NCC2(C(F)F)CCN(C(C(CC)OCC)=O)C2)c(Cl)ccc(C)c1O 19814,N1(C(C2CCC(C)CC2)=O)CCC(NC(c2cnn(C3CC3)c2)=O)CC(C)(C)C1 19815,c1(N(CCC)C)cc(S(=O)(=O)CN2CCCC2c2ccc(Cl)cc2)ccc1C#N 19816,N1(C(CCCC)=O)CCN(C2CCC(NC(C3(C)CCC(=O)N3)=O)CC2)CC1 19817,C1(NC(C(=Cc2ccccc2)CC)=O)CCCCN(C(=O)C(C)C2CC2)CC1 19818,N1(C(C(CC)OCC)=O)CCc2nc(CNC(c3cn(C)nc3C)=O)sc2C1 19819,C(N=c1ccnc(NC2CCCn3ncnc32)[nH]1)C1(CSC)CCC(F)(F)CC1 19820,C1(=O)C(CC)N1.C1(CN(C(=O)OC(C)(C)C)CC)CCCN1C(=O)C(C)(F)F 19821,C(CCCCCC(=O)NCCC1CCC(=O)N1)NC(C(=Cc1cn[nH]c1)C)=O 19822,C12(CNC(c3c(C)coc3)=O)CCCC1CCN2C(=O)C=CCF 19823,N1(C(Cc2cc(C)sc2)=O)CC2(CO)CC1(C(=O)NC1CC(O)CC1O)C2 19824,C(=O)(C(CNC(=O)C(N1CCNC1=O)C)N(C)C)N(CC(C)(C)OC)C 19825,C1(NC(=O)CCC(F)F)CN(C(c2nccc3[nH]ccc23)=O)CC1C1CC1 19826,c1(CNC(C2N(C(C)C)CCC2)=O)ccc(CNC(C2CC2(C)C)=O)cc1F 19827,N1(C(C2N(C)C(=O)CC2)=O)CCC(O)(C2CCN(C(=O)C3=CCC3)CC2)CC1 19828,N1(C(CSCCCC)=O)CCC2(CC1)CCN(C(C1CCC3CC3C1)=O)C2 19829,N1(C(C2(C(N)=O)CC2)=O)CC(NC(=O)CS(=O)(=O)CCO)C(C2CC2)C1 19830,c1(NC(N(CCC)CCNC(=O)OC(C)(C)C)=O)ccccc1C1(C)CC1 19831,c1(C(=O)NCCC(C)NC(c2nocc2Cl)=O)c[nH]c2ccc(Cl)cc2c1=O 19832,c1(C(=O)OC)ccc(N2CC(CCNC(=O)C(c3ccnn3C)C)(OC)C2)nc1 19833,c1(NC(C2CCCC2NC(c2cn(-c3ccccc3)nn2)=O)=O)c[nH]nc1Br 19834,c1(OC)ccncc1C(=O)NC(C)CCNC(C1(Oc2cccc(C)c2)CC1)=O 19835,Cc1ccncc1CC(=O)N(CCCNC(c1cnc(N2CCOCC2)s1)=O)C 19836,c1(C(=O)NC2C=CC(C(=O)NC(c3ncc[nH]3)CC)C2)ccnc(C)c1C 19837,Cc1cccc(-c2cncc(C(=O)NCC(O)CCNC(C3CCCS3)=O)c2)c1 19838,CCCC(O)CC(=O)NCCCCC(CO)NC(=O)CN1CCOCC1=O 19839,CC(C)(C)C1=NOC(C(N2CC3CC3(NC(c3ccns3)=O)C2)=O)C1 19840,C1(NC(C(CN(CC)CC)F)=O)C2CCCN(CC=C(C)C)C2C1(C)C 19841,c1(C(N2CC(O)(CCNC(C3C(C)(C(F)F)C3)=O)C2)=O)cccc([N+](=O)[O-])c1N 19842,Cc1cc(SC(C)C(=O)NC(C)CCNC(c2[nH]nnc2C)=O)cs1 19843,C1(CC)CN(C(c2cncn2C)=O)CCC1CNC(c1ccnn1C)=O 19844,C1(C(=O)NC(c2ccccc2F)CC)CC(F)CN(C(c2cc(O)ncn2)=O)C1 19845,N1(C(C(CC(C)C)(F)F)=O)CCCC2(C1)CN(C(c1ccnn(C)c1=O)=O)C2 19846,C(=O)(CS(=O)(=O)NCC1CCCO1)NCC(C)CNC(=O)C(O)C1CCCC1 19847,c1(C(N2C(C)CN(C(C3(C)CC=CCC3)=O)CC2)=O)cccn2ccnc12 19848,N1(CC)CC(C(=O)NC2CN(C(C3(F)CCCC3)=O)CC2C)CC1=O 19849,c1(C(=O)NCC2CC(NC(=O)C(F)(F)c3nccs3)C2)cc2c(Cl)cncc2s1 19850,c1(C(N(CCCNC(C(CCC)NC(C)=O)=O)CC)=O)c(Cl)ccc(Cl)c1O 19851,C12(CNC(C(C)(C)SC)=O)CCC(CN(C(C34CCC(C)(C3)OC4)=O)C1)C2 19852,C1(CNC(CN(CCC#C)C)=O)C(C2CC2)CCN1C(=O)C#CC1(C)CC1 19853,Cc1cccc(Cl)c1C(N1CC(CC(N2CCC(CF)CC2)=O)C1)=O 19854,c1(C(=O)NC2CCC(C)N(C(C3C4CC5C(C4)C35)=O)C2)ccc2nn[nH]c2c1O 19855,CC(C)CC(C(=O)NC1CCCCC1CO)ONC(=O)CC1(C)CCC1 19856,N1(C(C(=O)NCC=C)c2cccs2)CCc2ncncc2C1 19857,C1(C(=O)NCCCCC2CCCN(C(c3cnc(C)[nH]3)=O)C2)COC2(CCC2)C1 19858,c1(C(=O)OC)ccc(NC(C2CCCN(C(=O)CCCCC#N)C2)=O)cc1C 19859,c1(CC)ccc(C(F)(F)F)c(C(=O)NCCc2nc(C3CC3)n[nH]2)c1 19860,C(=O)(C(CC(C)C)N(C(=O)Cc1ccccc1C)C)N1CC(OC)(CO)C1 19861,c1(C(C)=O)ccc(C(=O)NCC2CC(C)N(C(=O)OC(C)(C)C)C2)cc1Cl 19862,Cc1ncc([N+](=O)[O-])n1CC(=O)NC1CC(C)(CNC(C2CC(C)CCO2)=O)C1 19863,C12(C)C3CCC(CC13)C2(F)F.C1(CC)CCC(c2cn(CCCC)nn2)CC1 19864,Cc1sc(O)nc1C(=O)N(C)CC1CCN(C(=O)COCC(F)F)C1 19865,c1(COC)c(F)cc(NC(c2ccccc2-n2ccc(C)n2)=O)cc1F 19866,C1(NC(CSCC#C)=O)CCCC(CNC(c2cc(SC)c(C)o2)=O)C1 19867,C1(CC)CCN(C(=O)CCN(CC)CC2CC2)C1.C1(C)(C)CNC(=O)CO1 19868,c1(CC(N2CC(O)(C(C)NC(C=C(C)C3CC3)=O)C2)=O)cc(F)ccc1F 19869,C1(CNC(c2ccc(F)cc2)=O)CCC2(CN(C(C3(CO)CCC3)=O)C2)O1 19870,C1(SC)CN(C(=O)CC(F)(F)F)CC1C(=O)NC1CC(N(C)C)C1 19871,O=C(C1=CCCC1)NCCCNC(C1(c2ccc(C(F)(F)F)cc2)CC1)=O 19872,c1(C(=O)NC(C2CN(C(C3(CC#C)CC3)=O)C2)C)ccn(CC)c(=O)c1 19873,c1(C(=O)NCC2CN(C(c3n(C(C)C)ccc3)=O)C2)cc2n(c1)CCC2 19874,c1(C(=O)NC2(C)CCN(C(=O)CC3CCCC(=O)C3)C2)onc2c1CCCC2 19875,N1(C(Cc2n(C)c(S)nn2)=O)CCCC(F)(CNC(=O)CC2CNC(=O)O2)C1 19876,Cc1ccn(CC(=O)NCCCOCCCNC(c2cccnc2)=O)c(=O)c1 19877,c1(C(N2C3C(NC(c4ccc(C)nn4)=O)C(C3)C2)=O)n[nH]cc1[N+](=O)[O-] 19878,C1(CNC(COC(CC)(C)C)=O)CC(O)CN1C(=O)C(CC1CCCCC1)OC 19879,N1(C(C(C)=CC)=O)CCCC2(CCCCC2NC(=O)CC(C)CCC=C(C)C)C1 19880,N1(C(COC)=O)CC(NC(c2nccc3c(F)cccc23)=O)C2(CCOCC2)C1 19881,c1(CN2C3C(C(=O)Nc4ccc(Cl)c(F)c4F)C(C3)C2)cncc2ccccc12 19882,S(=O)(=O)(CCCCCl)N1CC2C(C(N3CCC(CC#N)CC3)=O)(C2)C1 19883,C=CCCCCC(=O)NC(CO)C(C)NC(=O)COCc1ccnc(OC)c1 19884,N1(C(C2CCC2)=O)CC2C3CCC(C2C1)N(C(c1c(F)cc(F)cc1Cl)=O)C3 19885,CON1CCC(CN(C)Cc2ccc(O)cc2)CC1 19886,N1(C(c2c(CC)ocn2)=O)CCC(NC(C23CCC(C2)C3(C)C)=O)C(C(N)=O)C1 19887,c1(C(N2CC(NC(=O)C=CSc3nc[nH]n3)C(CO)CC2)=O)ccn2nccc2n1 19888,c1(NC(C=Cc2c(OC)ccc(OC)c2)=O)cccc2sc(C(F)(F)F)nc12 19889,c1(CC(=O)N(CCc2cn(CCC=C)nn2)C)ccc2c(c1)NC(=O)C2=O 19890,c1(C(=O)NCC2CC(OC)CN2C(=O)C(C)NC(C)(C)C)ccc2ccsc2c1 19891,CC1(C)CC(NC(=O)C(=Cc2ccccc2)C#N)CN(C(c2coc(Br)c2)=O)C1 19892,c1(CC)ccoc1C(=O)NCCCCNC(c1ccc(-c2ccco2)[nH]1)=O 19893,S(=O)(=O)(C=Cc1ccccc1)CC(=O)NCCC(N1CCC(F)(F)C(O)C1)=O 19894,N1(C(C(CSC)C)=O)CC(O)CC1CNC(c1nc(C2CC2)cs1)=O 19895,C12(C(=O)NCC3C(NC(CSCCOC)=O)CCCC3)CCN(CC1)S(=O)(=O)C2 19896,C1(CNC(COC)=O)C(C(C)NC(=O)C(C)Sc2ccccc2)C1(F)F 19897,N1(C(CC(CCC)O)=O)CC2(CCC2)CC1CNC(C1(NC(C)=O)CCCC1)=O 19898,c1(C(=O)NCC(CNC(CC2(OC)CCCCC2)=O)F)c(C)cc(F)cc1C 19899,N1(C(c2cccc(COC)n2)=O)CCC2CCN(C(c3ccoc3Cl)=O)CC12 19900,C1(NC(C2C(C(C)C)OCC2)=O)CC=C(C(=O)N(C(CC)C(=O)OC)C)C1 19901,CC(C(=O)NC1CC2(C1)CC(NC(c1cc(N(C)C)nc(Cl)c1)=O)C2)C(C)(F)F 19902,C1(C(=O)N(C2CC3CC3C2)C)(OC)CCN(C(=O)Cn2c(O)nnc2O)C1 19903,O=C(CCC(F)F)NCCCCNC(C1(CC2CCCC2)CCCC1)=O 19904,C(=O)(CCC(N)=O)N(CCC(=O)NCC(O)(CO)OC)C 19905,C1(C(=O)NC2C=CC(CNC(C3(C(F)F)CCCC3)=O)C2)(OC)CCSC1 19906,c1(OC)ccc(CC(=O)N(C)Cc2cc(Cl)ccc2C)c(Br)c1 19907,c1(OCC(=O)NC(C2CCOC2)CNC(CC(=C=C)C)=O)ccccc1C#N 19908,C(C1CCCC1)=C(C)C(=O)NC1C=CC(CC(=O)NCC2CC2Cl)C1 19909,C(=O)(C1=CCCCCC1)NC(C(N1CC[Si](C)(C)C1)=O)CC1CCOCC1 19910,c1(C(=O)NCC2CN(C(c3cnc(Cl)[nH]3)=O)CCCO2)ccc2c(c1)CCOC2 19911,Cc1cc(C)n(C(C)CC(=O)NC(C2CCCN2C(=O)CCC(=O)C2CC2)C)n1 19912,C(=O)(C(C)CC(=O)c1cccc(F)c1)NCCNC(C(N1CCNC1=O)C)=O 19913,C1(O)(C(N2C3C(NC(C4C(C=C)OCCC4)=O)CC(C3)C2)=O)CN2CCC1CC2 19914,c1(OC)cc(C(=O)NCCCN(C(=O)C(C)C(F)F)Cc2ccccc2)ncn1 19915,c1(C(N2CC(CNC(C3CC(OC(F)F)C3)=O)C3(CC3)C2)=O)cccc(F)c1Cl 19916,c1(C(N2CC3CC(NC(=O)C4=CCCOC4)CC3C2)=O)cc2nc(=O)ccn2[nH]1 19917,Cc1sc(=O)n(CC(N2CCCCC2CCNC(c2ccc(O)nn2)=O)=O)c1C 19918,C1(NC(c2c(C)cn(C)n2)=O)C2COCC1CN(C(=O)C=Cc1scnc1C)C2 19919,C(C)(C)(C(=O)NC(Cc1ccco1)C(=O)OC)N(CC)CC 19920,N1(C(CC=CCNC(C2(CCN=[N+]=[N-])CC2)=O)=O)CC2CCCCC2C1 19921,N1(C(C(CC)CC2CCCC2)=O)CCN(c2nc(C)cc(C)n2)C(C)C1 19922,O=C(C1=CC2(CCN(C(=O)C(F)n3ccnc3)C2)C1)NCC1(CC2CC2)CC1 19923,N1(C(=O)CC(F)F)CCN(C(c2ccc(C(F)(F)F)cn2)=O)C(CF)C1 19924,C(=O)(C(C)(C)C1=CCN(C(=O)CC=CCCCCC)C1)NCCCC=C 19925,N1(C(C(C2CC2)OC)=O)CCCC(N(C)C(c2cccc(F)c2SC)=O)CC1 19926,c1(C(=O)NCC(CC(C)C)NC(C(COC)(C)C)=O)cnn2cc(C)cnc12 19927,N1(C(c2scc(C(C)=O)c2)=O)CCCC(C)(NC(=O)CCN2CCCC2=O)C1 19928,CC(CC(F)(F)F)C(=O)NCC(C)(C)CCNC(c1cccc(NCCO)c1)=O 19929,c1(C(N(CCCCCNC(=O)CNC=O)C)=O)ccc2ocnc2n1 19930,C1(Nc2c(C(=O)OCCOCC3CCCC3)cccc2)CCc2c[nH]nc2C1 19931,N1(C(CCOCc2c(C)ncs2)=O)CC2CC(NC(=O)COCC(F)F)C1C2 19932,N1(C(C(F)=C(C)C)=O)CCN(C(C2CC2(Cl)Cl)=O)C(C(C)C)C1 19933,N1(C(CC(n2c(CC)ncc2)C)=O)CCCC2CN(C(=O)CC(C)OC)CC12 19934,Cc1nc(NCCc2csc(Br)c2)cc(=NC(C)c2nnc(O)o2)[nH]1 19935,C1(N(C)C(c2cncnc2)=O)CCCC2CN(C(=O)CC3(O)CCCC3)CC12 19936,c1(C(N2CC(SC)C(NC(=O)COC3CC=CC3)C2)=O)cc2oc(C)cc2[nH]1 19937,N12CCC(C3(CC3)NC1=O)C2.c1(OC(CC)(C)C)ccc(C#N)cc1C(F)(F)F 19938,c1(C(=O)NC(C)CC(C)NC(=O)C=CC(=O)NC2CC2)cccn2c(O)nnc12 19939,N1(C(c2c(CC)cno2)=O)CC(c2cccc(C(=O)NC)c2)C(SC)C1 19940,Cn1cc[nH]c(=NNC(=O)NCC2C(C(=O)O)C2(C)C)c1=O 19941,C12(C(=O)NC3CCN(C(=O)Cc4ccsc4)CC3)CCCCC1C2Br 19942,O=C1CCOCCN1CCNS(=O)(=O)CC1CCC1CSc1ccccc1 19943,C(CC(C)C(=O)NCC(CNC(=O)Cc1ccncc1Cl)CO)=CC 19944,C1(CCOC)(NC(c2ccc(Br)o2)=O)CCN(C(=O)Cc2ccco2)C1 19945,c1(CNc2scc(C(N3CCN(CCOC)CC3)=O)n2)cccc2ccn(C)c12 19946,n1(CC)cncc1CC(N1CC(c2ccccc2)(CO)C1)=O 19947,CC1(C)CC(NC(=O)Cc2ccc(Br)cn2)CN(C(C2COCCO2)=O)C1 19948,Cc1c(Cl)nc[nH]c1=NCC(O)CNC(C1CCCCC12CCC2)=O 19949,N1(C(COCCCC)=O)CC(NC(C2CCCN(C(C)C)C2)=O)C(C(F)F)C1 19950,C(=O)(CC1=CCN(C)CC1)NCC1(C(N2CC(C)C(F)C2)=O)CC(=C)C1 19951,c1(C(=O)NCCC2(COC)CC2)cc(C)n(C)c1.C12(CC1)C(=O)NC2 19952,c1(Nc2cccc(CN3CCC(OCC)CC3)c2)ccc2ncnn2c1 19953,O=C(CCC(F)(F)F)NCC1CC1NC(c1cnn[nH]1)=O 19954,c1(CNC(CC(C)CF)=O)nc(CNC(=O)C(C)c2ccco2)cc(O)n1 19955,C1(N(C(C2ON=C(CC)C2)=O)C)CCC2CN(C(c3cccc(F)c3N)=O)CC12 19956,C1(C(=O)NCC(C)(CNC(c2cc(C3CCOC3)[nH]n2)=O)OC)CC2(CCC2)C1 19957,N1(C(=O)C=CC=C(Cl)Cl)CCC(F)(CNC(C2CC(C(F)(F)F)C2)=O)CC1 19958,c1(C(N2CCC3(NC(=O)Cc4cscn4)C(C2)C3)=O)cc2c(O)ncnc2cn1 19959,C(C)(N=c1ccnc(Cl)[nH]1)C1CCN(C(CC(CCC)O)=O)CC1 19960,C1(C(N2CC(O)(CCNC(c3n(C)c(Cl)nc3)=O)C2)=O)CC1C1CCCC1 19961,C#CCC(CC(F)F)C(=O)NC1(C)CCCN(C(C2CCC=CCCC2)=O)C1 19962,C1(NC(c2ccn(C(C)C)n2)=O)CCC12CN(C(c1nc[nH]c1C(F)(F)F)=O)C2 19963,C(=O)(CN1C(=O)CCc2ccccc21)NC1C(C)CCN(C(C2(O)CCC2)=O)C1 19964,C(c1cccc(F)c1)=CC(=O)N(CCCN1CCCC(O)C1)CCC#N 19965,C1(N(C)C(c2ccc(NC=O)cc2)=O)CN(C(=O)COC(F)F)CC1(C)C 19966,N1(C(C(C(C)C)C)=O)CCC2(CC2NC(c2ncccc2F)=O)C1 19967,C1(C(N(CCN2CCC2)CCNC(=O)CSC)=O)CNC(=O)CC1C.CO 19968,C1(C(=O)NCCN(C)CCO)CC2CCC1N2C(=O)CCCOC(C)(C)C 19969,C1(NC(C=CS(C)(=O)=O)=O)CC2(CCCN(C(C3CC4CCC3C43CC3)=O)C2)C1 19970,N1(C(C(C)(C)CCF)=O)CCC2CN(C(C3CC(=O)OC3(C)C)=O)C2C1 19971,C1(NC(C23CC(C(C)(C)C)(C2)C3)=O)CCC2CN(C(c3cccc(N)c3)=O)CC12 19972,C(C(N=[N+]=[N-])C(=O)NCC(O)CNC(c1csc(C(C)C)n1)=O)OCC 19973,CC1(C)C(C)(C)C1(F)C(=O)NCCCNC(=O)Cc1cccc(N)c1 19974,C(=O)(CC(C)(C)COC)NCCOC(c1nc(C(CC)CC)cs1)=O 19975,c1(NC(N(CCCN=[N+]=[N-])C)=O)ccccc1C1CCC(=O)N1 19976,c1(C(=O)NCC2N(C(C3CC(OC)C3)=O)CC(O)C2)cccc2c1CNC2=O 19977,CC1(CNC(=O)CC2CCCO2)CN(C(c2ccsc2C(F)(F)F)=O)CCO1 19978,CN=c1[nH]c(=NCC(C)F)[nH]c(=NCCc2ccc3n[nH]cc3c2)[nH]1 19979,CC1(NC(=O)CC2(O)CCC2)CCC(NC(C2C=CCS2)=O)CC1 19980,c1(NCCN2C(CC(=O)OCC)CCCC2)ccc(C#N)cc1CC 19981,C1(NC(CS(N)(=O)=O)=O)CC(C2CCN(C(c3ccc4cnnn4c3)=O)CC2)C1 19982,C1(n2cc(C(C(OC)OCOC)C)nn2)CN(C(c2conc2C)=O)CC1C 19983,c1(C(=O)NC2C(CC)N(C(=O)CCS(C)(=O)=O)CC2)ccc2c(c1)OCO2 19984,N1(C(C2(CNC(C3CC3(Cl)Cl)=O)CCCCC2)=O)CCC(F)(F)C(O)C1 19985,c1(NC(C)=O)ccc(C(=O)NCCCN(C)C(c2ccc(CO)cn2)=O)cc1F 19986,C1(C(N2CCC(CO)C(O)CC2)=O)CC12CCN(C(C1(CO)CC1)=O)CC2 19987,N1(C(=O)NC)CCC(C(=O)NCC(C2CCCC2)NC(=O)CC2(C)CC2)C1 19988,O=C(C1=COCCO1)NCC1(NC(C2CC3C=CC2C3)=O)CCCCC1 19989,CC(=O)C(C)CC(C)C(=O)NC(C(=O)NCCSCCCO)C1(O)CCC1 19990,c1(C(N(CCCNC(c2c[nH]ccc2=O)=O)CC)=O)cc(OC)cc(C)c1 19991,C1(N(C)C)CC2(C1)CN(C(=O)CCOCCNC(c1cc(O)n(C)n1)=O)C2 19992,c1(-n2cc(C3C(C=C)C3)nn2)ccncc1Br 19993,c1(C(N(C2CCN(C(C(C(C)C)OC)=O)C2)C)=O)cc2nccn2c(O)n1 19994,C1(NC(CC(CC)C)=O)CCN(C(=O)CCN(CCCCOC)C)CC1F 19995,N1(C(N2CCOCC2)=O)CC2(CC(S(=O)(=O)N3CC(N4CC(O)C4)C3)C2)C1 19996,c1(C(=O)NC(COC)CNC(=O)C(C)(COC)OC(C)=O)cc2nc(C)sc2[nH]1 19997,N1(C(C2(C#N)CCC2)C(=O)NCC(F)F)CCN(Cc2ccc(F)cc2)CC1 19998,C(CCN=c1[nH]c(=NC2CCc3cccnc32)[nH]c2c1SCC2)=CC=C 19999,C(O)(C(=O)O)(C(F)(F)F)n1cc(-c2oc(C)c(C(N3CC4CC3C4)=O)n2)nn1 20000,N1(C(COC)=O)CC2CCC2(CNC(=O)C(C2CCCCCC2)O)C1 20001,C1(C)(CNC(COc2ccc(C)cc2)=O)CN(C(=O)CCCCCF)C(C)(C)C1 20002,c1(C(N2CC(CNC(C(C)n3cncn3)=O)N(C)CC2)=O)cnc2occc2c1 20003,C1(NC(c2cc(SC)oc2C)=O)CN(C(C2(C)CCCCO2)=O)CCC1O 20004,N1(CCNC(C2C(CC)OCC2)=O)CCCN(C(=O)CC#N)CC1 20005,N1(C(c2cnc(OC)s2)=O)CCCC1C1CCCN1C(=O)C=Cc1nc(C)co1 20006,C(CCC(C)(C)NC(c1sc(C(C)OC)nc1C)=O)NC(C(CC1CC1)OC)=O 20007,C1(C(N2CC(OCC(=O)NC)C2)=O)CCC(O)CN1C(C12CC(C#N)(C1)C2)=O 20008,n1(CC(=O)NC(c2cn(-c3ccsc3C(=O)O)nn2)C)cnnc1O 20009,C(=O)(CC(C(=C)C)OCC)NCC(C(N1CCC(C#C)C1)=O)C 20010,CC1CN(C(=O)Cc2ccon2)CC1(C)CNC(c1nn(C)cc1N)=O 20011,CC1=C(C)CC(C(=O)NCCC(C)(C)CNC(C2CC3CC3C2)=O)CC1 20012,C1(NC(C(C)C#N)=O)CN(C(c2ccc(CN3CCOCC3)s2)=O)CC12CC2 20013,c1(C(N2CCC3(C(CNC(CC=C=C)=O)C3)CC2)=O)coc2c(OC)cccc12 20014,CC(C)CC(C)(CNC(=O)COC1CCN(C)CC1)NC(c1cnccc1Cl)=O 20015,CCCCC(C(=O)NCC1CCCCN1C)NC(=O)CN(C(=O)COC)C 20016,CC(C)CC(CC(=O)O)NC(c1nnn(-c2cccc(F)c2)c1C(F)(F)F)=O 20017,c1(CC)nnc2cc(NCC3(CNC(C4CC(N(C)C)CCO4)=O)CC3)ncn12 20018,C(CCCC(=O)NCCOc1ncccn1)N(C(=O)C=Cc1ccsc1)C 20019,C1(NC(CC2C(C)(C)CCC2)=O)CN(C(c2cccc(N)c2O)=O)CCC1CO 20020,N1(C(C2N(C(C)=O)CCCC2)=O)CCC(C)C(NC(c2cnc(C(N)=O)s2)=O)C1 20021,c1(C(N2CCC(NC(CNC(=O)OC)=O)C(O)C2)=O)cc2c(C)[nH]nc2s1 20022,N1(C(C(c2cccc(F)c2)C)=O)CCN(C(=O)C(O)C2CCCC2)CC(C)(F)C1 20023,c1(N(CC(Cc2ccc(OC)cc2)C)C)ccnc2cc(O)ccc12 20024,c1(C(N2CC(NC(CC(C=C)C)=O)C(C)C2)=O)cc(Cl)ncc1O 20025,C1(C(N(C)CCC2CCN(C(C3CC3F)=O)CC2)=O)CC2CC(C1)CS(=O)(=O)C2 20026,O=C(C1CCCn2ncnc21)NCC1CN(C(=O)CSC(F)(F)F)CCO1 20027,c12ccc(cn1)CNC2=O.C(=O)(C=CC(=O)N(CCN)CC1CC1)OCC.SC 20028,N1(C(c2cccc(C)c2)=O)CCN(C(=O)CC2CCC(C(F)(F)F)O2)CC1CF 20029,CC(=O)C(C)CC(C)C(=O)N1CCN(C(=O)C#CC2CCC2)C(C(C)C)C1 20030,N1(C(C(C=C)(C)C)=O)CCC(C2CC2)(NC(=O)C(C)n2cccn2)C1 20031,C1(C)(NC(CC2(C=C)CC2)=O)CCN(C(c2cc(C)ccc2F)=O)CC1 20032,C1(CC(=O)NC(C(C)C)C)CN(C(=O)C(C)(C)CF)CCO1 20033,N1(C(C=CC)=O)CCC(C(=O)NCC2CSCCO2)C1C(C)C 20034,C(=O)(CCC(=O)N(C)C)N(C1CCN(C(CCCSC)=O)C1)CC1CCCC1 20035,Cn1cc(C(=O)NCCC2(NC(=O)C(O)C3CCC3)CC2)c(-c2cnccn2)n1 20036,C(=O)(CC(C(F)F)NC(=O)CC1CC(F)(F)C1)NCC1N(C)CCOC1 20037,C1(N(C(c2ccn(CCC)n2)=O)C)CCC(NC(=O)COCC2CCCC2)CC1 20038,C1(NC(C2(CCNC(c3c(C)coc3)=O)CC2)=O)CCCCC1N=[N+]=[N-] 20039,C1(=O)C(C(C)C)CN1.C1(OC)(CNC(=O)C(c2nc[nH]n2)N(C)C)CCOCC1 20040,c1(C(N2CCC(C(F)(F)F)(OC)C2)C(=O)NCC)ccc(OC)cc1Cl 20041,C1(n2c(-c3ccc(CN4CCCC4)o3)nc(C(C)C3CC3)n2)CCOC(C)(C)C1 20042,CC1CCCC(C(=O)NCCCOCCC(=O)NCc2ccn(C3CC3)n2)C1 20043,C(=O)(C1=CCCCCC1)NC(C)CCCCNC(=O)CNC(C1CCCCC1)=O 20044,c1(CSCC(=O)N(C)CC2CN(C(=O)C(C3CCCCC3)O)C2)ccccc1 20045,c1(C(=O)NC2C(CNC(c3cnn(C)c3Br)=O)C2)cc(F)cc(Cl)c1N 20046,C=C(C)CC(C(=O)NCC1CC(C)=NO1)NC(=O)C=C1CCOCC1 20047,N1(C(C(CCC)NC(N)=O)=O)CC2CC(NC(c3ccoc3Cl)=O)CC1C2 20048,CCCCCS(=O)(=O)CC(=O)NCC1CCN1C(C1CC12CC(OCC)C2)=O 20049,c1(C(C)=O)csc(C(=O)NC(C)(C)CNC(=O)COCC(c2ccccc2)C)c1 20050,Cc1ccc(-c2nc(Cn3nccn3)n(C3CC3)n2)cc1Br 20051,N1(C(C(CC2CCOCC2)NC(c2c(CC)n[nH]c2)=O)=O)CC(N(C)OC)C1 20052,C(=O)(CCC(F)(F)C(F)F)NC(C1CCOC1)CNC(c1c(C)cnnc1O)=O 20053,N1(C(C(COC)(C)OC)=O)CCC2(CC1)CN(C(c1cocc1C)=O)C2 20054,c1(C(N2CCSCC2)C)cn(CC2C=CCN2C(c2cc(C(=O)O)on2)=O)nn1 20055,N1(C(CC(C(C)C)O)=O)CCC(C2(O)CCN(C(=O)CN3CCCC3=O)C2)CC1 20056,c1(OC)c(C(=O)NC(CNC(=O)CCc2ccc(F)nc2)CO)ccnc1Cl 20057,c1(C(=O)NCC2CC(CNC(CSS(C)(=O)=O)=O)OC2)cc2ccnc(Cl)c2s1 20058,c1(C(N2CCC(CNC(C(CC)NC(N)=O)=O)C2)=O)cnc(C)c(CC(C)C)c1 20059,c1(CC(=O)N(c2cccc(OC)c2)CC#N)cccc2ccncc12 20060,C(c1ccc2c(c1)OCO2)=CC(=O)NC1COC2CCCC12 20061,C1(CNC(C2COC3(CCC3)C2)=O)CN(C(=O)C2=CCCSC2)CC12CCC2 20062,c1(C(N(C2CCCCN(C(=O)C(C)(F)C(C)(C)F)C2)C)=O)ccn2nncc2c1 20063,Cc1nnc2ccc(C(=O)NCCNC(C34CCCC3CC4)=O)cc2c1C 20064,CC1CC(CNC(=O)Cc2cscn2)CN1C(=O)CCN1CCCCC1 20065,CCCC(C)(O)CC(=O)N(C)CC=CC(N1C(C(=O)NC)CC1C)=O 20066,C1(N(C(=O)C(O)CC2CC2)CC)CCCN(C(c2oc(C)cc2C)=O)C1 20067,CCC(C)(C)CC(=O)N(C(CC(F)F)C(=O)N1CC(N(C)C)C(F)C1)C 20068,C(CC(=O)NCCN(C(=O)CC1(C)CCC1)C(C)C)OCCC 20069,CCC(COC)C(=O)NCC(C)(C)C(=O)N(CC(C)C(=O)OCC)C 20070,N1(C(C(C)OC2CCNCC2)=O)CC(C)(C)CC1(C)C 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20088,N1(C(C(c2cc(Cl)sc2Cl)C)=O)CCN(C(=O)C(C)(C)O)CC1C 20089,Cc1ccnc(C(N2CCCC2C2CCCC2)C(=O)NCC2CCOCC2)c1 20090,CC(C#N)CCC(=O)N1CCCC(NC(=O)CCCC2CCCC2)CC1 20091,C1(NC(c2n(C)nc(O)c2)=O)CS(=O)(=O)CC1NC(=O)CC1CCS(=O)(=O)CC1 20092,c1(CC(=O)NCC(C2CCOC2)NC(C2(CC=C)CC2)=O)csc(COC)n1 20093,C#CC1(CNC(C23CC2CN(C(=O)C(C)OCC(F)(F)F)C3)=O)CCCC1 20094,N1(C(c2n(C(C)C)ccc2)=O)CCCC(NC(=O)C(C)(C)c2cncnc2)CC1 20095,N#Cc1cnc(NC(C2CCCN2C(c2cc(F)cc(I)c2)=O)=O)c(Cl)c1 20096,c1(CC#N)ccccc1C(=O)NCC1CCN(C(=O)CC2CC3C=CC2C3)CC1 20097,C1(C(=O)NCCn2c(C)ncc2)COC2(C1)CN(C(=O)C(C)C(F)F)C2 20098,CC1(NC(C2CCC=CC2NC(c2cncc(C#N)c2)=O)=O)CCCC1(F)F 20099,c1(C(=O)NC2(C(N(CC)Cc3scnc3C)=O)CC(CO)C2)cc(CO)[nH]n1 20100,N1(C(C(C)NC(=O)C(C)(C)C)=O)CC2CCC(CNC(=O)CCC3(C)N=N3)(C2)C1 20101,N1(C(c2c(CCC)cccc2)=O)CCC(NC(=O)CCC(C)N(C)C)C(CO)C1 20102,C(=O)(N=c1ccc(C2CCOCC2)n[nH]1)c1c(Br)c(C)cc(OC)c1 20103,C1(C(=O)Nc2cnn(C3CC3)c2)CCC(C(=O)NCC2CC2Cl)CC1 20104,C1(F)(CNC(c2cc(CSCC)on2)=O)CCCN(C(c2nccnc2C)=O)C1 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20191,C1(C(N2CCCCC2c2nccs2)=O)CC2CCN(C3CCCNC3)CC12 20192,C1(NC(C(C)OC)=O)CCCCN(c2ncc(C(F)(F)F)cc2Cl)C1 20193,C(=O)(C1COc2ccc([N+](=O)[O-])cc21)NCC1CCN(C(CCOCC#C)=O)C1 20194,N1(C(=O)NC(c2cccnn2)CC)CCN(C2CCCN(C(C)=O)C2)CC1 20195,N1(CC(N2CC(CC(C)NC(c3cc(CC)oc3C)=O)C2)=O)C(C)CCCC1C 20196,N1(C(C2N(C)C(=O)CC2)=O)CC2(CCCC(CNC(C3CC(F)C(=O)N3)=O)O2)C1 20197,c1(CN2C(C)(C(=O)NC(CCC)CO)CC2)cc(Br)c(C)cc1F 20198,CCCC(C)CC(=O)N1CCC(O)C(NC(=O)COCCOCCO)C1 20199,C#CC1(O)CCCN(C(C2C3CN(C(=O)Cc4ccccc4F)CC23)=O)C1 20200,C1(COC)(CNC(C2CCN(C)C2C)=O)CCN(C(=O)C(C)CN2CCOCC2)C1 20201,c1(NC(C2C(CC)CCC2)=O)cccc2c1CCS2(=O)=O 20202,c1(SC)ncc(Cl)c(C(=O)NC2CN(C(=O)C=C(C)C)CCC2O)n1 20203,Cc1noc(C)c1-c1ccc(-c2nccn2C(C)CN2CCCC2)cc1 20204,C1(CN(C2(C(=O)NCCCC)CC2)C(C)=O)CCCC1 20205,C1(c2nnc(N3C(C)C(=O)NCC3)n2CCC#N)COC2(CCCCC2)C1 20206,c1(C(CC)O)nc(-c2csc(-c3csc(C)n3)c2)n(CC)n1 20207,S(=O)(=O)(c1ccc2c(c1)COC2)Cc1nc(C2CC(N)C(O)CC2)on1 20208,n1(CCOCC)c(N2CCN(C(C)=O)CC2)nnc1C1CC(O)CN1C 20209,c1(C(N2CCCC(Nc3cc(C)nc(C)n3)CC2)=O)ccc2sccc2c1 20210,C1(C(=O)NC2C(C(=O)NCCCn3ncc(C)c3)C2(C)C)CCCCCN1C 20211,C1(OC)CC(NC(=O)C(C)C)CN(C(C2CCCCN2Cc2ccccc2)=O)C1 20212,C#CC1(C(N2CCC(CNC(c3conc3COC)=O)CC2)=O)CCCC1 20213,N1(C(C2CCCC(C)C2)=O)C2CC(F)C(C2)C1C(=O)Nc1ccnn1C 20214,CC1(COC(C2CC2C#N)=O)CCc2ccccc21 20215,CCCCC(C(=O)NC12CC(C1)C2)NC(c1cncn1C)=O 20216,N1(C(C2(C(C)NC(C3C(C)CC(=O)CC3)=O)CC2)=O)CC2(CNC(=O)C2)C1 20217,N1(C(c2c(CC)cncc2)=O)CCC2C(CCN2C(=O)C=Cc2cscn2)C1 20218,C1(NC(CCC(C)(C)c2ccccc2)=O)CN(C(=O)CO)CC12CCOCC2 20219,C#CC1(O)CN(C(=O)C(C)CNC(C2CCOCC2)=O)C1 20220,c1(-c2n(C)cnc2)cnc2ncc(C(=O)Nc3cc4ccccc4cn3)n2c1 20221,C(=O)(C1=C(Cl)CCOC1)N(C)CC1CCCN(C(C2CCC3CC23)=O)C1 20222,Cn1ncc(C(=O)NC2CCCC(C(N3CCC(CO)C3)=O)CC2)c1C#N 20223,C(CC(CC)C(=O)N1CCC(O)(CNC(=O)COCc2ccnc(O)c2)C1)=CC 20224,c1(C(=O)NC2CCN(C(c3c(C)oc(Cl)n3)=O)CC2F)cncc(N=[N+]=[N-])c1 20225,N1(C(C2CCC(=O)OCC2)=O)CCC2(CC1)CCN(C(C1CC13CC(O)C3)=O)C2 20226,C(=O)(C#CC1CCCO1)N(C1CN(C(=O)Cc2ccc(F)cc2)CC12CC2)C 20227,c1(C(=O)NCCOCCN(C(CN2CCC(C)C2)=O)C)cc2cccc(O)c2[nH]1 20228,c1(C(N(C2CCN(C(C3(CC4CC4)CC3)=O)CC2)C(C)C)=O)cccc(C(N)=O)c1 20229,c1(CC(=O)NCCOc2ccc(Br)nc2)c(Cl)cncc1Cl 20230,C1(NC(c2nccc(C)c2)=O)COC2(CCN(C(=O)Cn3c(C)csc3=O)C2)C1 20231,C(=O)(C(C)(F)C(=O)NCC(C)NC(c1ccccc1C(C)(F)F)=O)OC 20232,Cc1nc(C)c(C(=O)NCC(C(C)(C)C)NC(=O)CN(S(C)(=O)=O)C)o1 20233,CC1CCc2nc(Cl)[nH]c(=NCC3CN(C(C4(C(N)=O)CC4)=O)CCO3)c2C1 20234,Cn1cc(Cl)cc1C(=O)NC(C1CCOCC1)C(N1CCCCC1CC(N)=O)=O 20235,CCC1=C(C(=O)NC23CCOCC2CN(C(=O)C(C)n2ccnn2)C3)SCCO1 20236,C1(NC(c2c(C)onc2)=O)CCN(C(=O)Cn2c(C)ccc2C)CC1C 20237,N1(C(c2c(NC(c3c(C)cnnc3)=O)ccs2)=O)Cc2ccccc2C(F)(F)C1 20238,CCC(O)(C(=O)NCC1(COC)CCN(C(=O)CC(=O)NC)C1)c1ccccc1 20239,C1(NC(C(CC)C)=O)CN(C(=O)Cc2ccc(CO)cc2)C2(CCCCC2)C1 20240,C(=O)(C#CC1CCOCC1)NC1(C(N2CCC(C)CC2C)=O)CSC1 20241,C(CC1=CCN(C(C2(C3CCOCC3)CC2)=O)CC1)NC(C(C)(C)C(N)=O)=O 20242,c1(C(Cc2ccccc2)NC(C(N2CC(S(C)=O)C2)=O)=O)ccccc1[N+](=O)[O-] 20243,c1(CC(=O)OC)occc1C(N1CCC(CN(C)C(c2csc(CO)n2)=O)C1)=O 20244,n1(CC)ncc(C(=O)NC(C)CNC(c2csc(-c3ncccc3F)n2)=O)c1C 20245,C1(CC)CN(C)c2ccccc2CN1C(c1ccc(C(n2cc(Br)cn2)=O)s1)=O 20246,C(=O)(C1CSc2ccccc21)N1CC(COC)(CNC(C2(C)COC2)=O)C1 20247,CN1CC=C(C(=O)OCCCOCc2ccccc2F)C1 20248,C1(NC(C2CC3(CCOC3)C2)=O)CC2(C1)CC(CN=c1[nH]nc(CO)s1)C2 20249,C(=O)(CC(F)(F)F)NCC(C)(CC)NC(c1ccn(C(CC)CC)n1)=O 20250,C1(OC)CN(C(c2ccccc2)=O)CC1NC(=O)NC(C1CCNCC1)CF 20251,n1(C(C)C)ncc(C(N2CCC2C(=O)NCC2(Cl)CC2(F)F)=O)n1 20252,Cc1cccc(CNC(=O)CC(C(C)C)NC(c2cncn2C(C)C)=O)c1C 20253,C12(NC(c3cccc(OCC)c3)=O)CCC(C1)N(C(c1sccc1CC#N)=O)C2 20254,c1(C(C)NC(C2C(OCC(=O)NC3CN(C(C)=O)C3)C2)=O)cccc(C)n1 20255,S(=O)(=O)(c1ccc(Cl)c(C(F)(F)F)c1)NC1CCC(NC(C2(F)CC2)=O)C1 20256,C1(COC)(CNC(=O)C(c2ccccc2)F)CCN(C(=O)CSCCC#N)CC1 20257,C1(CNC(c2csc(Cl)c2)=O)CCCCN(C(=O)CCCc2ccccc2)C1 20258,Cc1nc2c(NCc3ncccc3Nc3cc(OOC#N)ccc3F)cccn2n1 20259,Cc1ccccc1OCC(=O)NCCN(C1CC1)CC1(C)CC1 20260,N1(C(c2cccc(CC)n2)=O)CC(CNC(C2(n3cnnn3)CC2)=O)C2(CC2)C1 20261,C1(C(=O)NCC(C#C)OC)CC(C)(C)CCN1C(=O)CN1CC(C)(C)C1 20262,C(C(C)(C)CC(=O)NC1(C(=O)NCCC(O)C(=O)OC)CCCCC1)OC 20263,C(C(=O)NC(C)CC(N)=O)(C(C)OC)NC(CCCOCC)=O 20264,c1(C(N2CC(NS(C)(=O)=O)C2)=O)csc(Cl)n1 20265,C1(NC(c2cc(C(C)C)ncc2)=O)CN(C(C2CCCCO2)=O)CC1(F)F 20266,O=C(C1=CN=C2N=CNN2C1)OCC1CC(=O)N(c2ccccc2)C1 20267,CCC(CC(=O)NCC(CC(=O)Nc1ccc(C(C)C)nc1)C1CCC1)OC 20268,C1(C(N(C(C(C)C)CO)C)=O)C2CC3C(C2NC(c2cc(CO)on2)=O)C13 20269,c1(CN2CC(CC(=O)N(C(C(=O)OC)C)C3CC3)C2)ccc(C#N)cc1O 20270,c1(CC(=O)N(C(C)C)CCNC(C2(CCF)CC2)=O)ccco1 20271,c1(NCC(C)CO)nc(NC(CCC(F)(F)F)c2ccccc2)nc2sccc12 20272,c1(C(C)C)cc(=NC2CCCC(NC(=O)CC(O)C3CCCC3)C2)[nH]c(Cl)n1 20273,Cc1cc2n(n1)CCN(C(=O)CC1CN(C(=O)CSC(F)F)CCC1C)C2 20274,c1(C(=O)NCC(C)NC(C2(Cc3cccc(Cl)c3)CC2)=O)cnc2scnc2c1 20275,c1(C(=O)NCCNC(C2CC(=C)C2)=O)cc(Br)c(C)o1 20276,c1(C(c2n(CCC)nnn2)NCc2nc(C)n(C)n2)ccc2c(c1)OCC(=O)N2 20277,c1(C(=O)NC(CC)CN(C(=O)CSc2ccnn2C)CC)ccccc1C(C)C 20278,c1(C(N(CC(C)(C)NC(CCNC(=O)OCC)=O)C)=O)cc(C)c(Cl)cn1 20279,C(C(O)CS(C)(=O)=O)N(C=O)Cc1c(C)nn(Cc2ccccc2)c1 20280,CCCCC(C(=O)N1CC(c2cn(C(C)C)nc2C(F)(F)F)C1)c1nn[nH]n1 20281,Cc1cccc(C(N2CCC(F)CC2C(=O)NCCN2CCCC2)=O)c1O 20282,N(C1CCC(Nc2nc(Cl)ncc2Br)c2ccccc21)C(=O)CN1CCOCC1 20283,c1(OCC(=O)NCC2C(NC(c3sc(CC)c(C)c3)=O)CCC2)cccc(Cl)c1C 20284,Cc1nc[nH]c1CC(=O)N(C1CCC(NC(=O)Cc2cnc[nH]2)C1)C 20285,CON(CCO)C(=O)CC1CCN(C(c2c(C)cc(=O)n(C)c2C)=O)C1 20286,C1(CCCC)CNC(=O)CCCO1.n1(CC(=O)CC=C)cc(C2CC2)cn1 20287,C12(CNC(c3c(C)noc3)=O)CCCC1CN(C(c1cnc(N(C)C)o1)=O)C2 20288,C#CC1(C(=O)NC(CC)CCCCC)CCN(C(C2CN3CCC2C3)=O)CC1 20289,C1(NC(c2c(C)coc2C2CC2)=O)CC(F)CN(C(C2CCCOC2)=O)C1 20290,Cc1nc2nccc(N3CCCC3CNC(C3CC(F)(F)CCC3(C)C)=O)n2n1 20291,Cc1[nH]c(=N)sc1C(=O)NCC1CCC(CNC(c2cncc(F)n2)=O)CC1 20292,C1(NC(=O)C=Cc2ccc(Cl)cc2F)COC2(CCN(Cc3ccsc3)C2)C1 20293,C1(CNC(C2CCC(C)(CC)O2)=O)CN(C(=O)Cc2cc(COC)on2)CCN1C 20294,c1(C(=O)NC2C(CO)CCN(C(c3c(CC)ccs3)=O)C2)cc(S(C)(=O)=O)co1 20295,Cc1cccc2c1CC(C(=O)NC1CC(CNC(C3(C)CCC(=O)NC3)=O)C1)O2 20296,N1(C(CC(n2ccc(C)n2)C)=O)CCCCC12CC(NC(=O)CC(C)CF)C2 20297,CCC(CC)CC(=O)NC(CNC(=O)CC1CCCN1C)C(C)C 20298,N1(C(=O)OC(C)(C)C)CC2(C1)CC1(CC(C(=O)NCc3cccn3C)C1)C2 20299,N1(C(c2c(-c3c(C)c[nH]n3)cccc2)=O)CC2(C(=O)O)CC1(CF)C2 20300,CC1(CNC(C2CCCC(F)C2)=O)CCN(C(=O)CCCOc2cccnc2)C1 20301,Cc1cc(C(=O)NCC2CN(C(=O)CN3CCCS3(=O)=O)C2)ccc1Cl 20302,N1(C(c2n(C)ccc2)=O)CC2(CCCC(CNC(=O)C(F)CC3CC3)O2)C1 20303,C=CCCC(C(=O)NCC1(C)CCCO1)NC(c1ccccc1Cl)=O 20304,c1(COC)ccc(C(=O)NC2(CCNC(=O)CC3CCOC3C)CCCC2)cn1 20305,C1(CN)CCC(F)(F)C1.Cn1cc(C(C2CCC2)CC2CC(c3cccs3)(CO)C2)cn1 20306,CS(C)(=O)=NC(=O)C(=O)NC12CC(CNC(=O)CCc3cn[nH]c3)(C1)C2 20307,C1(CCNC(c2cnn(CC3CC3)c2)=O)CC(F)(F)CN1C(=O)Cc1ccno1 20308,N1(C(C(C)(F)F)=O)CC(NC(c2ccnc3ccsc23)=O)C2CCCCC12 20309,CCCCC(C(=O)NCC1CCC(CNC(C2CC2CC)=O)CC1)ON=C(C)C 20310,c1(C(=O)NCC(C)NC(C2CC(C(C)C)C2)=O)ccc2cc(O)ccc2c1 20311,C(C(C(C)C(C)C)NC(=O)Cc1ccc(C)cc1)NC(c1ccc(CCC)[nH]1)=O 20312,CC1(Cn2cc(CCN3CCSCC3)nn2)CCCCC1(F)F 20313,C#Cc1ccc(C(N2CCC(C(=O)NCC(O)COC)(CC)C2)=O)o1 20314,N1(C(c2cc(F)cc(Br)c2)C(=O)NC)CCC2CCCCC12 20315,c1(C(N(CCNC(C2(C)CC=C(C)CC2)=O)C)=O)cc(Cl)c(F)cc1Cl 20316,c1(-c2n(CC=C)c(N(CC(C)C)CC)nn2)ccc(S(C)(=O)=O)cc1 20317,C(=O)(C#Cc1ccccc1)NC1C(C(=O)NC2CCN(C(C)=O)CC2)CCC1 20318,c1(CC(=CC(=O)OC)C)ccccc1OC(C1C(OCC)C1)=O 20319,C1(NC(C(CSC)(C)NC(=O)Cn2cnnc2)=O)CCN(OC)CC1 20320,N1(C(CC(C)SC)=O)CCCC(C(=O)NCC2(n3ccnn3)CC2)C1 20321,N1(C(CN(C2CC2)CC)=O)CC2CC(C(=O)NCc3cnc(C)cc3C)(C2)C1 20322,CN=c1nc(N2CCC(C)(CO)C2)[nH]c(=NCC2(c3cnn(C)c3)CC2)[nH]1 20323,c1(C(N2CC(C)C(CCNC(=O)CCS(C)=O)C2)=O)cc(F)c(F)c(C#N)c1 20324,c1(C(C(C)C)NCC(Cc2ccc(OC)cc2)C)cc(Cl)cc(Cl)c1 20325,C1(CNC(C=CC(=O)OCC)=O)CC2CCC1N(C(=O)C(C)C1CCOC1)C2 20326,C(=O)(CC1=CCOCC1)NC1CCCC(CC(=O)NC(CCC)C(C)(C)C)C1 20327,n1(CC)cnc2c(N3CCC(CC(C)C)C3)nc(NC(C)(C)CF)nc12 20328,C1(NC(c2cc(COC)[nH]n2)=O)CCCCC1CNC(=O)Cc1ccns1 20329,CN1CC(CC(=O)NCCOCCN(C(=O)CC=C(Cl)Cl)C)C(O)C1 20330,c1(C(=O)NC(C(C)C)CNC(C2(C)C=CCC2)=O)cc(F)c2c(c1)CCC2 20331,N1(C(Cc2cc(C)nn2C)=O)CCCC(C)(C(=O)Nc2cccnc2C(C)C)C1 20332,C1(CCCC)CCCN1C(=O)C(C1CCC1)NC(=O)C=CCC1CCCC1 20333,c1(CC)cc(N2CCCC(NC(C3CCC(=O)N(C)C3)=O)C2C)nc(CC)n1 20334,CCC(CC(=O)N1CC(C2CC2C(=O)N(CC(C)C)C)C1)C(C)(C)C 20335,C1(NC(C(C)OCC)=O)CCCCN(C(C2(C)CCN(C)CC2)=O)CC1 20336,C(=O)(C1CCCc2nc[nH]c21)N1CCC(NC(=O)C=Cc2ccsc2)C12CC2 20337,Cc1nc(CO)ncc1NC(=O)C(C1(O)CN(C(C2(CO)CCC2)=O)C1)F 20338,CCCCCCCCCCCC(=O)N(CC(CC)NC(C1(OC)CCSC1)=O)C 20339,C1(NC(c2cc(SCC)ncc2)=O)C2CC(CN(C(c3cnn[nH]3)=O)C2)C1CO 20340,Cc1cccc2c(CC(=O)NC3COCC3NC(C3CC4(CCC4)C3)=O)c[nH]c12 20341,C1(CN=[N+]=[N-])CCCN1C(C1CCCN1C(=O)CC1OCCCO1)=O 20342,N1(C(C2(COC)CCCO2)=O)CC2CC2(CNC(c2cnc(C3CC3)cn2)=O)C1 20343,C(CC1=CCN(C(C2CC(=O)OC2(C)C)=O)CC1)NC(CC(C)CN(C)C)=O 20344,C1(CC(=O)NC(c2nc(C)cs2)CC)CN(Cc2ccc(C(=O)O)s2)CCO1 20345,Cc1cc(CCNC(C23CC2CCN3C(=O)CCc2ncccn2)=O)nn1C 20346,N1(C(C(CC)C#N)=O)CC2CCOC2(C(=O)OC)C1 20347,C1(C(C(=O)NC)(C)C)CCN(C(=NCc2cc(Cl)ccc2O)NC2CCC2)CC1 20348,CC1CCCN(C(c2c[nH]c(=O)cn2)=O)C1CNC(=O)CC1CCS(=O)(=O)C1 20349,Cc1ccc(C(F)(F)C(=O)NC2CCC(NC(C3CC(=O)N(O)C3)=O)CC2)cc1 20350,c1(C(=O)NCC2CN(C(=O)C(O)C3CCCC3)C2)cc(Br)c2occc2c1 20351,C=CCCCC(C(=O)N1CC(=O)N(C)C(=O)C1)NC(c1nc(C)ccc1C)=O 20352,O=C1NCCCCC1NC(c1ccc(I)cc1)c1nnnn1CCCF 20353,N1(C(C(CSC)O)=O)CCC(N=[N+]=[N-])(C(=O)N(C)Cc2ccoc2)C1 20354,Cc1cc(NCC2(F)CCCC2)ncc1S(=O)(=O)NC1CCC2C(CC1)C2(F)F 20355,O=C(CC1=CSC2=NCCN12)NCC1CCCCN(C(c2cnccc2Cl)=O)C1 20356,c1(OC)ccc(C(N2CC(O)(C(C)NC(=O)C(O)Cc3[nH]cnc3C)C2)=O)o1 20357,CCC(C(=O)N1CC2CC1(C(=O)N(C(C)C)CC1CCCO1)C2)C(F)(F)F 20358,c1(CC)occ(C)c1C(=O)NCC1CCCC(NC(C2(CC)CC2)=O)C1 20359,c1(C(N2CC(=C(CNC(=O)Cc3cnccn3)F)C2)=O)cn2cnnc2cn1 20360,CN1CCN(C(=O)Cc2n[nH]c(=N)s2)CC1CNC(C1CCCCC1CO)=O 20361,C(CC(=O)N1CCC(OC2CCC2)C1)(C(F)(F)F)NC(C(F)=CCC)=O 20362,C1(NC(c2c(C)n[nH]c2)=O)C2CCN(C(=O)C=CC(=O)NC3CC3)CC12 20363,Cc1ccnc(Oc2ccccc2NS(C)(=O)=O)c1Br 20364,Cc1cccc(CC(=O)NCCC2CCCCN2C(=O)Cc2cccnc2)c1 20365,c1(C(N(C(c2ccc(C)cc2)c2ccccn2)C)=O)ccc(F)c(C)c1Cl 20366,N1(C(C2(CC(C)C)CCC2)=O)CC2(CO)CC1(C(N1CC3C(C)C3C1)=O)C2 20367,CC1CN(C(=O)CC2(CO)CCCC2)CC(C)C1NC(c1cc(C2CC2)cs1)=O 20368,N1(C(CCCCC=CC)=O)CC2CCC(NC(c3ccn(CC(C)C)n3)=O)(C2)C1 20369,c1(C(=O)OC)no[nH]c1=NC(=O)c1nc(C(=O)Nc2csc(C)n2)cs1 20370,C1(C#N)(C(=O)NCC(CC)NC(=O)CCc2c(Cl)cncc2Cl)CCCOC1 20371,c1(C(N(C(C(COCC)n2cc(COC)nn2)=O)C)C)ncc(Br)cn1 20372,c1(C(N2CC3(OCC(NC(c4ccco4)=O)C3)C2)=O)c(F)ccc2occc12 20373,O=C(C#CC1CCCC1)N1CCN(C(c2cc[nH]c2C2CC2)=O)C(C2CC2)C1 20374,S(=O)(=O)(C1CC1)NCC(=O)NC(CN(C(=O)CC(C)C1CC1)CC)C 20375,C1(C(=O)NC2CCCC(C(N(CCCC(C)C)CCO)=O)C2)CC2(C1)CC(O)C2 20376,C1(C(N(CCCC(=O)NC)C)=O)C(C2CC2)CCN1C(C1CCCC1)=O 20377,C1(CNC(C(C)(C)F)=O)CC2(CCN(C(c3cnc(C#N)s3)=O)CC2)C1 20378,C1(C(=O)NC2CCN(C(C)=O)C2)CC(N=[N+]=[N-])CN1C(=O)Cc1cn[nH]c1 20379,C1(NC(C(C)(C)C)=O)CN(C(c2n[nH]c3ccc(Cl)cc23)=O)C2(CCOC2)C1 20380,c1(CC2CCN(C(c3cc(Cl)ccn3)C(=O)NCC(C)C)C2)ccc(F)c(F)c1 20381,N1(C(c2c(CC)nc[nH]2)=O)CCC2(C1)CN(C(=O)CCc1ccncn1)C2 20382,N#Cc1ccc(C(=O)NC2CC2CNC(C2CCS(=O)(=O)C2)=O)o1 20383,CC(CN(C)C)CCC(=O)NCC(O)CNC(C12CCC(CC1O)C2)=O 20384,c1(C(N(CC(CC)NC(c2nccc(OC)c2N)=O)CC)=O)cnn2c1CCC2 20385,C#CCCCC(C)C(=O)NCc1ccc(CNC(=O)C(C)(C)OC(F)(F)F)cc1 20386,c1(C(N2CC(OCCC(=O)NC(CCC)CC)C2)=O)cc2occc2[nH]1 20387,N1(C(CN2CC(C)C2)=O)CCOC2(CCN(C(=O)C3=CCCCCC3)C2)C1 20388,c1(C(=O)NCC(CC)NC(=O)C(c2cn(C)nc2C)C)cnc(O)cc1C 20389,C#Cc1ccc(C(=O)NC2CCCCN(C(c3scnc3CC)=O)C2)cn1 20390,c1(C(=O)Sc2ccccc2-c2cn(C3CCOC3)nn2)cc2cc[nH]c(=O)c2s1 20391,CC1C(NC(=O)C(C)NC(N)=O)CCCN1C(C1CC12CCCC2)=O 20392,C1(CCCC(=O)OC)CCN(C(C(=O)NCC2CCOC2)C(C)C2CC2)CC1 20393,c1(CC)ccc(C=CC(=O)NC2COCCC2NC(c2cc(Cl)c[nH]2)=O)cc1 20394,N(C1CCCc2cccc(F)c21)S(c1ccc(CC(C)C)o1)(=O)=O 20395,N1(CC(C)C)CC(C(N2CC(C)C2)=O)CC1=O 20396,N1(C(C(=O)NCCOC)=O)CCCC(C(=O)NCC23CC(C2)C(C)O3)C1 20397,c1(CN(C)C(C2CC3CC3N2C(c2ccc(F)cc2Cl)=O)=O)ccc(C#N)cc1 20398,C=CCC(C)(C)CC(=O)NCc1ccccc1CNC(C1NC(=O)CC1C)=O 20399,N1(C(C2C(=C)C2C(=O)OC)=O)CCC(C(N(CC(=O)OC)C)=O)C(O)C1 20400,O=C(N=c1nc(Cl)nc2[nH][nH]cc1-2)C1CN(C(=O)CCC2CCC2)CCO1 20401,C1(CC)CCCC1(C)C(=O)NC(C1CCN(Cc2ccsc2)CC1)C 20402,C12(NC(c3cccc4nonc34)=O)CCCN(C(C3CC(F)(F)C3)=O)CC1C2 20403,Cc1cc(C(N2CCC(CCNC(c3csc(Cl)n3)=O)CC2C)=O)nc(C)n1 20404,N1(C(CC2CC(C)(C)C2)=O)CC2(CC(NC(C3(C)CNC(=O)C3)=O)CO2)C1 20405,Cc1cc(F)c(CNC(=O)NCC(CO)C(O)C2CCCCC2)nc1Br 20406,c1(OC)cnc(Cl)nc1N1CCCOC(CNC(C2CC=CC2)=O)C1 20407,c1(C(=O)OC)[nH]c(C)c(C(=O)NCCOCCNC(=O)C(C)(C)C2CCC2)c1C 20408,Cc1ccc(N2CCOC2=O)cc1NC(c1cn(CC(C)N)nn1)=O 20409,C1(NC(C(C)C(F)F)=O)(CNC(c2nc(C3CC3)cs2)=O)Cc2ccccc2C1 20410,c1(-c2cn(CC=C)nc2)nc(C(=O)NCC2(c3ccccc3Cl)CC2)c(C)s1 20411,CC(C)C(C(=O)N(C)CCOCCN(C(=O)CC1CCCC(=O)C1)C)NC=O 20412,N1(C(C2(OC)CCN(C(c3scnc3C)=O)C2)=O)CC(C)(C2CCC2)C1 20413,C1(CNC(c2ccc(SC)s2)=O)CC(NC(=O)Cc2cncnc2)C12CCC2 20414,c1(C(c2nnnn2CCSC)NC2(COC)CCSCC2)ccc2occc2c1 20415,N1(C(c2c(=N)cc[nH]c2)=O)C2CCC1CN(C(=O)CC1CC(=O)NC1=O)C2 20416,c1(N)cccc(O)c1.c1(C(C)OC)nc(C(=O)OC(c2nn[nH]n2)CC2CC2)cs1 20417,N1(C(C=C(CCC)C)=O)CC(NC(c2ccc(O)cc2)=O)CC1(C)C 20418,C1(NC(C(C)c2cccs2)=O)CN(C(c2cncn2C2CC2)=O)CC1C1CC1 20419,c1(OC)ccc(-n2nnc(C(=O)Nc3cnn(C(C)C)n3)c2C)cc1 20420,c1(C(=O)NC2(C)CCCN(c3cnc(C#N)cn3)C2)cc2n(n1)CC1(CC1)C2 20421,c1(C(CN2CC(=O)N(Cc3ccc(OC)cc3C)C2=O)C)ccc2c(c1)CCC2 20422,C1(C(N(C2CCN(C(CNC(N)=O)=O)CC2)CCO)=O)CCCC2(CCOC2)O1 20423,CCCC(O)C(=O)N1CC(N(C(=O)C(CCO)N(C)C)C)C1 20424,C1(N(C(=O)CCCc2sccc2C)CC)CCCN(C(C2CCCCC2)=O)C1 20425,C#Cc1cccc(C(=O)NC2CC(O)CN(C(c3cc4scnc4[nH]3)=O)C2)c1 20426,C1(NC(C(COCC=C)C(C)(C)C)=O)CC2(CCCN(C(=O)C(CC)SC)C2)C1 20427,N1(C(c2n(CC)ccn2)=O)C2CCC1CC(C(=O)Nc1cnn(CC(N)=O)c1)C2 20428,c1(C(=O)NC(C(=O)NCCCOC=C)C2CCCO2)cnc(O)c(F)c1 20429,O=C1CC(C(=O)N2CCCOC(CNC(=O)CC3CCCS3(=O)=O)C2)=NN1 20430,C1(CC)CCN(C(=O)C(O)C(F)(F)F)C(C(=O)Nc2cccc(CCO)c2)C1 20431,c1(C(=O)NC2CC(NC(c3c(C)noc3C(F)F)=O)C2)ccc2c(c1)COCO2 20432,c1(C(=O)NCC(COC)N)cc(F)ccc1NC(=O)C(C)C 20433,c1(OCC(=O)NCC(C)CNC(c2ccon2)=O)ccc(C#N)cc1Cl 20434,C1(CC(=O)NCCC2CC(C(N3C(CCC#C)CCC3)=O)C2)CC(O)C1(C)C 20435,NS(=O)(=O)CCC(=O)NCCC1CCN(C(=O)CN2CCN(C3CC3)C2=O)CC1 20436,CCCC(CC(C)C)C(=O)NC1CCN(CCCNC(=O)C#CC(C)C)C1 20437,c1(C(N2CCCC2Cc2cccc(Cl)c2)C(=O)NC)ccccc1OC 20438,N1(S(C)(=O)=O)C2CCC1CC(CNC(=O)CCOC1CC1)C2.C(C(F)(F)F)S 20439,N1(C(C2(CNC(C(C)N3CCCC3)=O)CC=CC2)=O)CCCNC(=O)C1 20440,c1(OC)ccc(C(=O)NCC2(NC(=O)CC3CCC(=O)C3)CCCC2)cn1 20441,C=C=C(C)CC(=O)NCC(CC1CC1)C(=O)N1CCC1(C)C(C)C 20442,c1(C(N2CC(CNC(C3CC3C(F)F)=O)OCCC2)=O)scc2c1CCCC2 20443,c1(OC)cc(C)c(NC(=O)C(=O)NCCN2CCNC(=O)C2)cc1F 20444,N1(C(CC(C)F)=O)CCCCC12CN(C(=O)C(F)(F)c1csc(=N)[nH]1)C2 20445,C1(C(=O)NCC2(OC)CN(C(=O)CC3(O)CCCCC3)C2)CCCC(C)(C)O1 20446,C(=O)(C1=CCc2ccccc21)NC(C)CC(C)NC(c1sccc1S(N)(=O)=O)=O 20447,C1(NC(CSc2ccc(OC)cc2)=O)CCN(C(=O)CCCCCBr)CC1F 20448,c1(C(=O)NC2CC3CN(C(c4nc(N(C)C)oc4)=O)CC32)cncc2nc[nH]c12 20449,Nc1cc(C(=O)NCC2COCC2NC(C2(O)CCC2)=O)c(F)c(F)c1F 20450,C1(NC(C2(C)CCN(C)C2)=O)CC2CC(NC(c3occc3C3CC3)=O)C2C1 20451,c1(C(=O)NCC2(O)CCCN(C(C(C(C)O)(C)C)=O)C2)cccn2nccc12 20452,C(c1ccc2c(c1)OCO2)=CC(=O)NC1(CNC(C(CCCC)C)=O)CCOC1 20453,C1(OC)CC(CC(N2CC(N(C(=O)CCN3CCC(C)CC3)C)C2)=O)C1(C)C 20454,c1(N2C(=O)C(CCC(=O)NC)C(C)=N2)ccc(OC)c(F)c1C(=O)OC 20455,c1(C(=O)NCCC(CNC(CCC(=O)OCC)=O)O)ccc(OC)c(Cl)c1OC 20456,c1(OC)c(C(=O)NCCC2(O)CN(C(C3CCCC(F)C3)=O)C2)c(C)nn1C 20457,C12(C(=O)NCc3ccc(C)nc3O)CCC(CN(C(=O)C(F)CCC(C)C)C1)C2 20458,c1(C(N2CC=CC(NC(c3onc4ccccc34)=O)C2)=O)ccc([N+](=O)[O-])cn1 20459,c1(C(=O)NCC(C(C)C)NC(Cn2c(C)nnn2)=O)ccc(N=S(C)(C)=O)s1 20460,C(CNC(=O)C(=O)NC(=N)N)(CSC)OC 20461,C1(CC(=O)NCCOCCC#C)CCN(C(=O)Cc2cncnc2)C1(C)C 20462,C1(CNC(=O)C=Cc2cc[nH]c2)CC2CCC1N2C(C1(CO)CCOCC1)=O 20463,C(=O)(C(O)C(F)(F)F)N(CCNC(C1CCC(=C)CC1)=O)CC1CC1 20464,c1(C(N(C2CCN(C(CCCC#C)=O)CC2C)C)=O)ccc2cccnc2c1 20465,c1(C(=O)NCC2(O)CCCN(C(C3C(C)C3)=O)C2)cc2ncccc2o1 20466,Cc1c([N+](=O)[O-])c(C(=O)NC(C)Cn2cccn2)nn1C 20467,CCCC(C(O)C(=O)N1C(C)CC1(C)C)NC(c1sncc1C)=O 20468,C(C)(CO)(C(=O)NC1CCOC(C(=O)NCC(C)CC2CCCC2)C1)OC 20469,c1(N(C)C(=O)NC2CCCN2CC2(C3CC3)CCCO2)ccc(C#N)nc1 20470,CCCC(O)C(=O)N1CCC(OC2CN(C(C3COCCN3C)=O)C2)CC1 20471,C12(C(N3CC(N(CC(C)C)C)C3)=O)CC(CO)(CN1C(C1CCCSC1C)=O)C2 20472,C1(C(=O)NCC2CC(F)(CNC(=O)C(O)CSC)C2)(OC)CCOCC1 20473,c1(C(=O)NCCN(CCOC)C(c2c[nH]cc2Br)=O)scc(C)c1Cl 20474,CN1C(=O)CN(CC(=O)NCCCNC(=O)CCc2cc(Cl)no2)C1=O 20475,N1(C(C2(CC)CCOC2)=O)CC2CC2(CNC(C2CC(OC3CC3)C2)=O)C1.CO 20476,N1(C(C(C=C)O)=O)CC(CNC(c2cnn(C(CC)CC)c2C)=O)C(O)C1 20477,n1(CCCC(=O)NC2CC(F)(CNC(COCCCC#C)=O)C2)c(C)csc1=O 20478,N1(C(c2nnc(C(C)(C)C)s2)=O)CC2(CCN(C(=O)C=CI)CC2)C1 20479,C(CCSC)(C(=O)NCC(CO)NC(=O)C=Cc1scnc1C)OC 20480,n1(CCCC(=O)NCC2CCC2NC(=O)COCC2CC2)cnc2ccccc12 20481,Cc1c(NCc2cc(C(C)(C)C)n[nH]2)ncnc1N1CCCC(N2CCC2)C1 20482,N1(C(c2cnc(C)n2C)=O)CCC(n2cccn2)(C(N2CCSC2(C)C)=O)CC1 20483,CC1CC(C(N2CCC(CN(C(=O)Cc3cn(C)nn3)C)CC2)=O)CCO1 20484,C1(NC(C=CC)=O)CCN(C(=O)C(c2ccccc2Cl)(C)C)CC1F 20485,N1(C(C2CN(CC)C(=O)C2)=O)CCCC2(C1)CN(C(=O)CC1CC(C)C1)CCO2 20486,c1(C(N2CC(c3cnc4ccc(F)cn34)C2)=O)ccc(=O)n2c1CCC2 20487,C1(OC)C(NC(=O)CNC(=O)CN2CCC(C)CC2)CC1(C)C 20488,C(=O)(C1=CC2(CCOC2)C1)NCC(C1CC1)NC(c1nc(C(C)C)oc1)=O 20489,c1(C(C)(CCC)N(c2nnnn2C(C)(C)C)C(C)CCC2CC2)cn(C)nc1C1CC1 20490,C1(n2cc(CC(C=C)O)nn2)CN(C(c2cnccc2Cl)=O)CC1OC 20491,N1(C(C2(CC#C)CCC2)=O)CCC(NC(=O)CNS(N)(=O)=O)C2(CCC2)C1 20492,CC(C)CCCCC(=O)NC1CN(C(C2CC(c3cccc(F)c3)C2)=O)CC1O 20493,c1(C(=O)NC2(CN(C(CCn3c(C)ncc3)=O)C)CC2)cnn(C)c1C 20494,C1(C(N2C(CN(C(C3CC(=C)C3)=O)C)COCC2)=O)OCCCC1(C)C 20495,C=C=C(C)C(=O)N(C)C.C12CCCC1n1cc(nn1)C(C)N2 20496,C(C(=O)NCCC1CCCN(C(c2cn(C)nc2Cl)=O)C1)(C(F)(F)F)OC(C)=O 20497,C1(C)(CN(C(CC2OCC(C)(C)C2)=O)C2CC2)CCC(O)CC1.C12(CCC1)C(=O)N2 20498,N1(C(C(C)(O)CCc2ccccc2)=O)CCCC2(C1)CN(C(=O)C1=CCCS1)C2 20499,Cc1cc(F)ccc1N1CCCC(NC(N2CCNC(c3ccc(F)cc3)C2)=O)C1 20500,N1(C(C2CCCN(CCC)C2)=O)CCN(C(c2cnc[nH]2)=O)CC1C(F)F 20501,C1(NC(=O)CCSc2ccccc2)CCCC12CCN(C(=O)CCOC1CC1)C2 20502,CC1(C)CN(C(=O)C2=COCC2)CC1NC(C1C2CCCC12)=O 20503,N1(C(C(C)NC(=O)NC)=O)CCC2(CC1)CC(NC(=O)CC1(O)CC1)C2 20504,C=CCC(F)(F)C(=O)N1CCC(F)(C(=O)NCc2noc(COC)n2)CC1 20505,C(=O)(C(C)(F)C(F)(F)F)N1C(CNC(c2c(SC)cccc2F)=O)CCCC1 20506,Cc1ccc(C(N2CCCC2C(C)(C)C(N2CC3CCC(C2)O3)=O)=O)c(O)n1 20507,c1(CC23CCN(C2)C(=O)C(CC=Cc2ccncn2)NC3=O)ccc(Cl)cc1O 20508,CCC(CC(=O)NC(CCO)C(F)F)N(C)C(C1CC(C)(CC)C1)=O 20509,C1(CCNC(c2ccnc(O)c2)=O)CN(C(=O)COCC2(F)CC2)CCS1(=O)=O 20510,c1(C(=O)NC(C)C(C)NC(=O)C=Cc2nccs2)ccc(Br)cc1N 20511,C(=O)(C(O)CC(F)(F)F)NC(C(=O)N(CCOCC#C)C)CCSC 20512,c1(OCCC(=O)NCC(CO)NC(CC(C)N2CCCC2)=O)ccc(F)cc1 20513,C1(C(=O)NCC2C(CC(=O)N(C(CC)CC)CCO)C2)CNC(=O)O1 20514,c1(CCNC(C(CC2CC2)NC(C(COC)C)=O)=O)ccccc1F 20515,c1(C(N2CCC(N(C(C3CNC(=O)N3)=O)CC)C2)=O)cc2cccnn2c1 20516,C1(C(N(C2CCC(NC(C3(CO)CCCO3)=O)CC2)C)=O)C2CC3C(C2=O)C13 20517,C(C(C)(C)CS(=O)(=O)N1CC(CO)C(C)C1)OCC 20518,C1(NC(c2ccc(C)nc2O)=O)COC2(CCN(C(C3COC(=O)C3)=O)CC2)C1 20519,N1(C(C2OCCC(NC(C(C)(C3(C)CC3)OC)=O)C2)=O)CC2CC=CCC2C1 20520,c1(NC(C(C)OC(c2cccc(C#N)c2)=O)=O)ccc(C(F)(F)F)c(Cl)c1Cl 20521,CC1CN(C(C2(CF)CCC2)=O)CC1CCNC(c1csc(-c2ccsc2)n1)=O 20522,C(=O)(C#CC1CCC1)NC(CCNC(c1cnc(SC)n1C)=O)C 20523,C1(C(=O)NC2CN(C(C)=O)C2)CC12CCN(C(C13CCCC1C3)=O)CC2 20524,c1(OCC)ccc(C2(CNC(C3(OC)CCC3)=O)CC2)cc1.C12CCC1CNC2=O 20525,c1(C(=O)OC)cc(C)c(C(=O)NC(C)CNC(=O)C(C)(C)c2ccnn2C)o1 20526,CCC(C)CCCCC(=O)NCCC1CSCCN1C(=O)C1=CCC(C)CC1 20527,N1(C(c2sc3ccn(C)c3c2)=O)CCC2(CCN(C(c3cc(F)c[nH]3)=O)C2)C1 20528,C1(CNC(C(COC)OC)=O)CCC(N(C(=O)CN2CCCC2=O)C)CC1 20529,C1(C)(CC)CCCN(C(C2CCN(C(=O)C=NOC3CCCCO3)CC2)=O)C1 20530,CCCC(CCCNC(=O)C(O)C(C)(C)C)NC(c1cnc(C2CC2)[nH]1)=O 20531,C12(CC)CCC(C(=O)NC3CCN(C(c4sncc4C)=O)CC3F)(CO1)C2 20532,N1(C(C2C(CN(C)C)C2)=O)CCC(C)(NC(C2CC23CCOCC3)=O)CC1 20533,c1(CC(=O)NC2C3(NC(CCOC)=O)CCC(C2)C3)c(C)nc(O)nc1C 20534,C1(CNC(C2(C)ON=C(C)C2)=O)CC2(CO1)CN(c1cc(O)nc(O)n1)C2 20535,CC1CN(C(C2(NC(c3ccc(Cl)s3)=O)CCSC2)=O)CC(C)(C)O1 20536,c1(C(N(CC(CNC(C(C)OCC=C)=O)O)C)=O)sc(Cl)c(Cl)c1OC 20537,C1(NC(c2nc(C)oc2C)=O)CC(C)CN(C(=O)CC2(C)CCC2)C1 20538,S(=O)(=O)(c1ccc(C(N2CC(NC(C3(C)COCCO3)=O)C2)=O)cn1)NC 20539,C1(CNC(=O)C(C2CC2)C2CC2)CC2COCC2N1C(=O)CCCCCO 20540,C(=O)(CCC1=CCCCC1)NC1(CO)CCCN(C(CCN(CCC)C)=O)C1 20541,N1(C(=O)CN2CCCC2=O)CCCC2CN(c3cc4nncn4cn3)CC12 20542,C1(C(=O)NCCc2onc(C)n2)CC2CC1CC2NC(=O)C(C)CN(C)C 20543,C1(C(N2CC(C)(O)C2)=O)CCCCN1C(C1(C#N)CCCC1)=O 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20650,C#CCCCC(=O)NCC1(C(N2CCC(CCCC)C2)=O)CCCO1 20651,c1(CC(=O)NCC2(COC)CC(NC(C3(C#C)CC3)=O)C2)ccc(F)cc1 20652,C1(NC(C(c2cn(C)nc2)O)=O)CCCC12CCCO2 20653,Cn1nc([N+](=O)[O-])c(Cl)c1C(=O)NCC1C=CCN1C(=O)CCC1CCC(=O)N1 20654,c1(NC(C)=O)cc(C(N2CC(CO)(CNC(=O)C(C)C3CCC3)C2)=O)ccc1C 20655,c1(C(=O)NCC2C3CN(C(C4N(C)CCCC4)=O)C2C3)ccc2cnoc2c1 20656,C#CCCCCCC(=O)NC1CC(F)(F)CC1NC(=O)C(N1CCCCCC1)C 20657,CC1(C(N2CCN(C3CCCN(C(c4ccsc4)=O)C3)CC2)=O)CCCCCC1 20658,c1(SCC)cnc(O)c(C(=O)NCC(CNC(C2CN(C)CCO2)=O)CO)c1 20659,N1(C(c2ncc(F)cn2)=O)CC(F)(F)C1C1CC1.C12CC(CO1)C(=O)NC2 20660,C1(CC(=O)NC2C3(CC(OCC)C3)C2)CC2(C1)CN(C(C1CC3CC3C1)=O)C2 20661,c1(N(C2CC(=C)C2)CC)cc(NC(=O)COC2CCOC2)nc(COC)n1 20662,c1(C(N2C(CC(N3CCC(C)(O)C3)=O)CCC2)=O)ccc(Cl)cc1F 20663,C12(NC(C3CC(CNC(C4(C)C(C)C4)=O)OC3)=O)CCC(CC1)C2(C)C 20664,c1(NCc2nccc(CC)c2)[nH]c(=NC2CC(NC)C2)nc2c1ncn2C(C)C 20665,C(=O)(C(C#N)C(C)(C)C)N1CCC(NC(c2c(F)ccc(CC)c2)=O)C1C 20666,C(CCNC1CC1)(CN=c1cccc(S(=O)(=O)N(C)C2=NCCN2)[nH]1)OC.SC 20667,Cc1c(C(=O)NC2CC(N(C(=O)CCC3CCCC(O)C3)C)C2)nnn1C(C)C 20668,N1(C(C(C)S(N)(=O)=O)=O)CCCC(C2CN(C(C3(c4ccn(C)n4)CC3)=O)C2)C1 20669,C(=O)(CC(C)C(C)(C)NC(c1csnn1)=O)NCCn1c(C)ncc1 20670,N1(C(CN2C(=O)CSC2)=O)CCCOC(CNC(=O)CC2CCCOCC2)C1 20671,CC1OC2CCC1(C(=O)NC1CCCC(CC(=O)NCC3NC(=O)NC3=O)C1)C2 20672,CC(C)CC(=O)NCC1CC1CNC(=O)C(N1CCNC1=O)C 20673,C1(N(C(Cc2c(C)ocn2)=O)CCO)CCN(C(C2(c3ccco3)CC2)=O)CC1 20674,c1(C(C)=O)ccc2oc(NC(=O)C=Cc3cncc(F)c3)nc2c1 20675,N1(C(C)C)CCCC(NC(=O)C(C)N(C(=O)C(C)(C)CF)C2CC2)C1 20676,Cn1nc2n(c(=O)c1=O)CCN(C(c1cc(Cl)c(-c3nn[nH]n3)cn1)=O)C2 20677,N1(C(C(C(=O)OC)C)=O)CC2(CCC(C(=O)Nc3nc(-c4cccnc4)cs3)O2)C1 20678,CC(C)CC(C)C(=O)NCC=C1CCN(C(C2(C#N)CCC2)=O)CC1 20679,C1(NC(c2c(C)nc(CNC(=O)CCN=[N+]=[N-])o2)=O)CC(F)(F)C1(C)C 20680,N1(C(C(c2ccccc2F)OC)=O)CCC(CNC(=O)CCCC(N)=O)C1(C)C 20681,c1(CC)ncc(C(=O)NC2CC(CC(N3CCC3C(C)C)=O)C2)cn1 20682,N1(C(Cc2cc(C)n(CC)c2C)=O)CCCC2(NC(=O)C(C)CC)CC2C1 20683,N1(C(c2onc(CC)c2C)=O)CCC2(CCN(C(=O)COC3CCOCC3)C2)C1 20684,CC1CN(C(C2CC3(CCC3)C2)=O)CCC1NC(=O)C(C)(C)c1ccncc1 20685,N1(C(Cn2ccc(C)n2)=O)CCC(O)(C(C)NC(c2ccnc(O)c2)=O)C1 20686,c1(NCC(CCCC)NC(=O)CC(C)CN(C)C)cc(C)nc(OC)n1 20687,C(=O)(CCC(C)CC)NCC1(CN(C(C(CC#C)C)=O)C)CC1 20688,Cc1ccc(N(C(=O)CN(C)CCO)Cc2cccnc2)cc1F 20689,c1(CC(=O)NCC(C)NC(CC(C)(C)SC)=O)noc2ccc(Br)cc12 20690,C1(NC(CN(C)C)=O)CCCCC12CCN(C(=O)C(=O)N(C)C)C2 20691,Cn1cccc(C(=O)Nc2ncnc(Cl)c2F)c1=O 20692,CC(Cc1cnn(C)c1)C(=O)N(CCCCNC(=O)C(C)Cc1ccncc1)C 20693,C1(CC(=O)NC(CC)C(C)C)CN(C(c2c(C)noc2N)=O)CCO1 20694,C1(C(N2CC3N(C(CC4CC(=C)C4)=O)CC(C3)C2)=O)COc2ccc(F)cc2C1 20695,C#CCC(C)(CC)C(=O)N1C2CCC(C2)C1CC(=O)NCCC1CCCN(C)C1 20696,N1(C2C3CCCC3NC2=O)CC2C(CO)C2C1.C(C)(C)(C)OC(=O)NCCS.CS 20697,N1(C(c2c(CC)csc2)=O)CC2CCC1C(CNC(=O)C1=C(Cl)CCCC1)C2 20698,c1(C(N2CCCC(NC(CS(=O)(=O)NC)=O)C2)=O)c(C)c(C)nn(C)c1=O 20699,Cc1cc(C)c(NC(=O)Cn2cc(CN(C(C)C)C3CC3)nn2)cc1Cl 20700,N1(C(C(CCC)NC(C23CCC(C2)C3)=O)=O)CCOCCC1CC 20701,N1(C(c2cc(C)oc2)=O)CC2(CCCN(C(c3ccnc(Cl)c3N)=O)C2)C1 20702,C(=O)(C(C)CC(F)F)NCC(CC)NC(c1ccc(C2(CC)CC2)cc1)=O 20703,c1(C(N(C)CCNC(C2(n3cnnn3)CC2)=O)=O)cn(C2CC2)cn1 20704,c1(C(N2CC(CC)C(NC(=O)C3=CCCC3)CC2)=O)cnc2[nH]ccc2n1 20705,C1(CC)CN(C(c2ccsn2)=O)CCC1NC(c1nc(CC)sc1N)=O 20706,CC(C)CC(C(=O)N(C)CC1CCCC1NC(=O)Cc1cnns1)C(C)C 20707,C1(C(N2C(C(N(C)CC3C(C)C3)=O)CC2)=O)CCCCNC1=O 20708,CCC(C)C(C(=O)NC(C12CC(CO1)C2)C)N(C)C(c1sccc1CO)=O 20709,c1(C2CCC(NC(=NC)NCc3ccn(CC)n3)C2)ccc(F)c(F)c1 20710,C1(C(N(C)CC2N(C(C3CN(C(C)=O)C3)=O)CCOC2)=O)CCn2nncc2C1 20711,CCC(C)CCCC(=O)NCCC1(NC(c2cn(C3CCC3)nc2C)=O)CCC1 20712,c1(CCC(=O)NCC(C)NC(C(F)CCOC)=O)ccc(OCC#N)cc1 20713,C1(CCNC(c2nccc(CC)c2)=O)CCN(C(=O)Cc2ccccc2)C(C)C1 20714,N1(C(C2N(C)CCN(C(c3scc(C)c3)=O)C2)=O)CCN2C(=O)OCC2C1 20715,CCC(CC(=O)NC1CC(CO)N(C(=O)Cc2cccc(C)c2F)C1)C(C)C 20716,C1(C)(C(=O)NCc2cc(COC)on2)CCN(C(C2CC(=O)CS2)=O)C1 20717,C1(CC=C)(NC(=O)COCCCC)CCCN(C(C2CCC(F)C2)=O)C1 20718,C1(C(=O)NC(CCNC(C(COC)NC(C)=O)=O)(C)C)CCN(C2CC2)C1=O 20719,N1(C(=O)OC(C)(C)C)CCCC12CCNC2.c1(CN2CC2(C)C2CC2)ccccc1 20720,Cc1cc(F)ccc1CC(=O)NC1CCCC1NC(=O)CCC1OCCO1 20721,c12cc3ccccc3cc1C(=O)N2.c1(C(=O)NC2CN(C(C)=O)C2)ncn(C)n1 20722,C1(C(N2CCC(NC(CC3(CC(=O)OC)CC3)=O)C(C)C2)=O)CCC2CC1C2(C)C 20723,Cc1n[nH]c(C)c1C1CCCN1C(c1cccc(C(=O)O)c1)=O 20724,N1(C(c2ccc(C)nc2)=O)CCC2CN(C(=O)CN3CCCC3C)C2C1 20725,Cc1ccc(C=CC(=O)NC(C)CC(C)NC(=O)CCc2cccnc2C)nc1 20726,Cc1cc(C2(C(=O)NC3CC3CNC(c3cc(Cl)ccn3)=O)CCC2)cc(C)c1 20727,c1(C(=O)NCc2noc(C3CC3NC3CC3)n2)cc(C(F)(F)F)ccc1O 20728,C(=O)(C(C)CCC(C)(C)C)NC(CC)CC(=O)NCC1(C(=O)OC)CC1 20729,c1(OC)cccc(Cl)c1C(=O)NCCC1COCCN1C(c1cnn(C)c1Cl)=O 20730,CCC(C)(F)C(=O)N1CC2CC2(NC(c2ccc(F)cc2)=O)C1 20731,C1(C(=O)NCCC2(O)CCN(C(C=CCCC)=O)CC2)C2CCC(C2)C1(C)C 20732,N1(C(C(C(C)C)NC(N)=O)=O)CCC(C)C(NC(=O)CCC23CCC(CC2)C3)C1 20733,c1(C(N2CCC(n3cc(CC(=O)OC)nn3)CC2)CC)cc(C)nn1C 20734,C1(N(C(=O)NCCC(C)C(F)F)C)CCOC(C)(C)C1 20735,CCCCCC(=O)N(C)CCOCCCNC(=O)C(C1CCOCC1)OCC 20736,c1(C(N(C2CCN(C)CC2)CCCOC)=O)cccc(O)c1F 20737,C(CCC[Si](C)(C)C)N(C(Cn1cnnc1)C(=O)O)C 20738,C1(C(=O)NCCCCC2N(C(C3CCC4CC4C3)=O)CCC2)C2CC3C(C2=O)C13 20739,c1(OC)nccc(C(=O)NCC(O)CNC(=O)CC2CC3CCC2C3)n1 20740,CCCC(O)(CCC)CC(=O)N(CC(C)NC(C1CC1c1ccccc1)=O)CC 20741,c1(C(=O)NC2C(C)CCN(C(c3cccc(CC)c3)=O)C2)cnn2c1NCCC2 20742,c1(CNC(C2CN(C(C)=O)C2)=O)nc2c(s1)CCN(C(=O)CC1COC(=O)C1)C2 20743,c1(C(=O)NCC2C3CN(C(C(CC=CC)C)=O)CC32)ccc2c(c1)CC(C)(C)C2 20744,CP(C)(=O)c1ccc(NC(c2ccccc2)C(=O)O)o1.c12ccc(cc1)o2 20745,c1(CN2CCC(C(=O)Nc3c(OC)cccc3O)C2)c[nH]c2ncccc12 20746,C1(C(=O)NCC2(C(N3CC(C)(OCC)C3)=O)CCCC2)CCN(C)C1C 20747,C12(C(N(CC(C3CCC3)OC)C)=O)CCC(CC1)N(C(c1cn[nH]c1)=O)C2 20748,c1(CCC(=O)NCC(CC=C)NC(c2ccc(C)nc2)=O)ccccc1N=[N+]=[N-] 20749,c1(N(C(=O)NC(C)CCc2ccccc2C(F)(F)F)CC)ccc(C(F)(F)F)cc1 20750,n1(CC(=O)NCC(CC=C)NC(=O)CC2CC=CCC2)ncn2nccc2c1=O 20751,C1(C(=O)NCC2CCCCC2)(CNC(c2ccc[nH]2)=O)CC12CCC2 20752,N1(C(C(CC)c2cccnc2)=O)CCCN(C(=O)C=Cc2cnccn2)CC1C 20753,c1(C(N2CCN(C(COCC(=C)C)=O)C(CO)C2)=O)ccsc1S(C)(=O)=O 20754,CN1CC(NC(C2CCOCCN2C(c2cn(C3CC3)nn2)=O)=O)C(F)(F)C1 20755,CN=c1[nH]cc(C(N2CCOC(C3CCN(C(=O)C(CO)NC(N)=O)C3)C2)=O)o1 20756,c1(C(=O)NC2C(NC(C(C(C)(C)C)SC)=O)CCCCC2)nc2ncccn2n1 20757,c1(C(N(C)CC2(O)CN(C(CSC)=O)C2)=O)ccn(CC(F)(F)F)c(=O)c1 20758,C1(C(CNC(c2c(C)nsc2)=O)C)CCN(C(=O)C(C)C2(O)CCC2)CC1 20759,C(CCCCC(=O)NC(C)(CSC)C(=O)NCc1cccc(C)c1O)OC 20760,c1(OC)ccc(Cn2cc(Cn3ccnn3)nn2)cc1[N+](=O)[O-].N(CCO)CCO 20761,N1(C(C)=O)CCC(NC(C2CCCC(NC(=O)NC3CCCCC3)C2)=O)CC1 20762,C=C=CCCC(=O)NCCCN(C(=O)CC1(N(C)C)COC1)C 20763,c1(OC)nc(C)ccc1C(=O)NCC1(NC(=O)CCc2ccon2)CC1 20764,C#CC1CCCN(C(=O)C(C2CC2)NC(=O)CC2CCCN(C)C2)CC1 20765,C12(C(=O)NCCOCCC(N3C(CC(C)(C)C)CC3)=O)CCCCC1C2 20766,N1(C(C=CCNC(C2CCCC(CF)C2)=O)=O)CCC(O)(CO)CC1 20767,Cc1cc(Cl)c(C(=O)NCC2CC2NC(c2cc3occc3[nH]2)=O)cc1N 20768,N1(C(C(N2C(C(=O)NCC(C)C)CCC2)=O)=O)CCOC(C2(O)CC2)C1 20769,C(=O)(C(C(C)C)n1cnnc1)N(C1CC1)CC1N(C(C(COC)OC)=O)CCC1 20770,N1(C(C(=O)NC2C(NC(C3CCC(CC)CC3)=O)C2)CC)CCc2ccccc21 20771,N1(c2nc(C)cc(CC)n2)CC(C2CCCN(C(c3ccsc3OC)=O)C2)C1 20772,N1(C(C(C=C)(C)C)=O)Cc2ccccc2C(NC(c2cc(CC)cc(Cl)c2)=O)C1 20773,C1(NC(c2ccc(C)o2)=O)CC(O)CN(C(C2(C)C(C)(C)C2(C)C)=O)C1 20774,c1(CC)[nH]ccc1C(=O)NC(C1CC=CCC1)C(=O)N(CCCc1ccco1)C 20775,c1(CCC(=O)NCCC2(NC(C3CC(=C)C3)=O)CC2)cccc(F)c1 20776,N1(C(C2(COC)COC2)=O)CC(n2cc(COc3nccs3)nn2)C(O)C1 20777,c1(OC)ccc(SCC(=O)OCCNC(=O)CCn2cncn2)cc1 20778,CC1CCN(CC(O)CC(N2CC(C3CCCCCC3)C2)=O)CC1 20779,c1(CSC)nc(-c2nc(Cl)c(CO)[nH]2)n(C(C2CCCCC2)C)n1 20780,C1(NC(C(CC)NC)=O)COC2(CCN(C(c3cc(C)c4n[nH]cc4c3)=O)C2)C1 20781,N1(C(C(C)=C2CC2)=O)CCC(CO)(CNC(C2CCC2(F)F)=O)C1 20782,c1(C(=O)NCC(=C)CCNC(=O)CC(C)(C)O)ccc([N+](=O)[O-])cc1C 20783,Cn1cc(CN2CC(NC(=O)Cc3ccccc3-c3nn[nH]n3)C2)ccc1=O 20784,c1(C(N2CC(CNC(c3c(C)cns3)=O)C3(C2)CC3)=O)cc2c(C)cccc2o1 20785,C1(C(N(CCC(=O)N2CC(N3CCC3)C2)C(C)C)=O)C2CCC(=O)C12 20786,C(=O)(CCS(N)(=O)=O)N1C(CN(C(=O)CN2CCCNC2=O)CC)CCCC1 20787,C1(CCNC(C(C)OCC2CC2)=O)CCCN(C(=O)CN2CCS(=O)CC2)CC1 20788,c1(C(N2CC(N(C(CCC(CC)=O)=O)C)C3(C2)CC3)=O)ccc2nc(C)oc2c1 20789,C1(CNC(=O)Cc2cccs2)CN(C(=O)C(=O)NCC(F)F)CC12CCOCC2 20790,C1(C#N)(C(=O)NC2CC3CC(NC(CC(CC)CC)=O)CC32)CC12CCCC2 20791,C(=O)(CC(C)(C)C)NCc1c(C(=O)NCC(C)C2CC2)nco1 20792,C(C(C)(C)C)N(CC(=O)NCCCN(C(C1C(C(N2CCCC2)=O)C1)=O)C)C 20793,CC(C)C(C)CC(=O)N1CCCC1(C)C(=O)Nc1ccccc1O 20794,c1(C(C(=O)NC(c2cn(-c3cccc(COC)c3)nn2)C)O)c(C)cccc1C 20795,c1(C2(C(=O)NC(c3ccc(F)cc3I)C)CC2)cccc(C2=CC(=O)CCC2)c1 20796,c1(OCC)c(C(=O)NCCN(C)C(C2(C)CC(O)CN2C)=O)cccc1F 20797,c1(OC)cccnc1C(=O)NCC1COCC1NC(=O)C=Cc1ccc(C)o1 20798,c1(OC)ccc2c(c1)C(C(=O)NCC=CCNC(=O)CC1CCC(C)C1(C)C)CC2 20799,c1(C(=O)NC2(CNC(C(C3CC3)SC)=O)CC2)ccc(N)cc1Br 20800,c1(C(N2CCCC(CN(C(C(C(C)C)F)=O)C)C2)=O)cccc2nc(O)ccc12 20801,CP(C)(=O)c1cnn(CC(N2CCC2CNC(c2cc(O)ncn2)=O)=O)c1 20802,CN1CCC(CCN(C)C(c2conc2NC(=O)CCOC2COC2)=O)CC1 20803,C1(C(=O)OC)CCCC2(CCN(C(c3cc(Cl)c(F)cc3O)=O)C2)O1 20804,CC(F)(F)C(F)C(=O)N1CCC(C(=O)NCc2cccc(CO)n2)(CF)C1 20805,CCC(C)(CC(NC(=NCCF)NC1(C)CN(c2ccccc2F)C1)=O)C(N)=O 20806,c1(C(N(CCC#N)C)=O)ccc(CN2CCN(CCCC#N)CC2)cc1 20807,c1(C(N2CCCC(CNC(c3c(C)ccn3C)=O)C2)=O)ccc2[nH]ccc2n1 20808,c1(CC)noc(CC)c1CC(N1CC(CNC(C2(C)CC3CC3C2)=O)C(C)C1)=O 20809,C1(OC)CCC(CNC(=O)CCCN(C(=O)C(C)Cn2cccn2)C)C1 20810,C1(O)(C(C(=O)Nc2ncn(CC)c2)O)CCOCC1 20811,c1(CC)ccccc1C(=O)N(C(C)C(=O)NCC1CC(C)(C)CO1)C 20812,C1(C(N(C2CN(C(CCOC(C)C)=O)C2)C)=O)CNC(=O)CC1C 20813,c1(C(N(C2CCN(C(c3ccc(OC(C)C)cn3)=O)C2)C)=O)cc(Cl)ccc1N 20814,C1(NC(C(C=C)(C)C)=O)CCC(C)(C)CC1CNC(C1CC=CC1)=O 20815,C1(CNC(C(CC)O)=O)CN(C(c2cn(CCO)nn2)=O)CCCO1 20816,N1(C(C2CN(C(C)C)C2)=O)CCC(CCNC(C2CCSC2)=O)CC1 20817,c1(SC)ccc2c(c1)C(NC(=O)C(N1CCC3(CCNCC3)C1)=O)CCO2 20818,C(=O)(C(Cc1ccccc1)C1CC1)NCC(C)CN(C(=O)CC1COC(=O)C1)C 20819,c1(CC(N2CC(CC(C)NC(C3CC(=O)N3)=O)C2)=O)coc(C(F)F)n1 20820,C1(CN(C(=O)CC2(O)CCCCC2)CC)CCCCN1C(=O)C#CC1CC1 20821,c1(OCCC)cccc(OC2(C(=O)NC(C)CN(CC(=O)NC)C)CCOC2)c1 20822,CN1CCC(CNC(c2nncs2)=O)C1 20823,N1(C(c2cscc2C)C(=O)NCC=C)CCCCC(CO)C1 20824,Nc1c(C(=O)NCC(C2CCCC2)NC(=O)C(c2ccccc2)F)cccc1F 20825,CCC(C#N)C(=O)N1CCC(O)(C(C)NC(C2CCC(C)CC2)=O)C1 20826,N1(C(CN(C(=O)C(C2CC2)C2CC2)CC)=O)CCSCC1C 20827,N1(C(C(=O)NC(c2ccc(C#N)cc2)CF)=O)CC(S(=O)(=O)C2COC2)C1 20828,C1(CC)C(NC(c2ncccc2SC)=O)CCCN1C(=O)C1=CCCC1C 20829,C(C)(C(C(=O)NC1CCCC(CNC(c2sccc2SC)=O)C1)N(C)C)OC 20830,CC#CCCC(=O)NC(C1CCCN(C(C2CN(C)C2)=O)C1)C 20831,C1(NCc2c(OCC)cccc2[N+](=O)[O-])CCCCC(O)CNCC1 20832,C1(C(N(C(C)C)CCN(C(=O)CCCCc2cnn[nH]2)C)=O)CCCCN1N=O 20833,C(=O)(C1=CCC2(COC2)OC1)NCC1C(NC(c2c(C)nccn2)=O)CCC1 20834,C(=O)(C1CCc2cccnc21)N1CC(N(C)C(c2ccc(F)cc2C2CC2)=O)C1 20835,C12CCCCC1OCCN2.C1(N(C(=O)CCC2(C)CC2)CCC)CCCCCC1 20836,C1(CCNC(c2cnc(C(C)C)o2)=O)CSCCN1C(c1cccn1C)=O 20837,Cc1cc(C(=O)NCC=C2CCN(C(=O)CC(C)C3CCCO3)CC2)cc(C)n1 20838,Cc1ccc(C=CC(=O)NC(C2CCCN2C(=O)C(C)Cn2cccn2)C)cc1 20839,N1(CC2N(C(c3ccn(CC)n3)=O)CC2)CCc2c(ccc(C)c2Br)C1 20840,C12(C(N3CCCCC3C(C)NC(CN3CC(C)(OC)C3)=O)=O)CCC(CC1)CO2 20841,C(=O)(C(=O)CCc1cn(CC(N2CCC(CN3CCCC(O)C3)C2)=O)nn1)OC 20842,N1(C(c2ccc(C)[nH]2)=O)CC=CC(C(N2CCC(O)C2C(C)(C)C)=O)C1 20843,CC(CCC(=O)N(C)CCN(C)C(N)=O)NC(C1(Cl)CC1(F)F)=O 20844,N1(C(CC(C)(C)CO)=O)CCC2(CCC2)C(NC(c2ccccc2)=O)C1 20845,C1(C(N2CCC(COC)(NC(=O)CCCF)C2)=O)OC(C)(C)OC1(C)C 20846,c1(N2C3CN(C(c4ccc(F)cn4)=O)C(CC3)C2)c(Br)cncc1[N+](=O)[O-] 20847,C1(CNC(CCC=C)=O)CC2(CC2)CN1C(=O)C(C)Cc1cccc(Cl)c1 20848,c1(C(=O)NCC(C)N(CC)CC)oc(CNC(=O)C(CC2CC2)C2CC2)nc1C 20849,c1(C(=O)NC2C(C)N(C(=O)C=Cc3ccnn3C)CC2)ccc2c(c1)COC2 20850,c1(NC(C2CC(NC(C=CC=CC)=O)C2)=O)ccc(C(F)(F)F)nc1 20851,C1(OCC(=O)NCCN(CC(C)O)C(C2(CC)CC2)=O)CCCCC1C 20852,C1(NC(C2CCCC(C)(C)CC2)=O)CN(c2nncs2)C2(CCOCC2)C1 20853,c1(NC2C(C)CN(C(c3ccc4cnnn4c3)=O)C2)ccc([N+](=O)[O-])cc1Cl 20854,C1(N(C=O)Cc2ccc(OCC)c(OC)c2)CCOC2(CCSCC2)C1 20855,C(=O)(C#CC1CCOCC1)N1C(CNC(C(C)OCCN(C)C)=O)CC(O)C1 20856,CCCCCS(=O)(=O)CC(=O)NC(C)C(C)(C)NC(=O)C(C)CC(C)(F)F 20857,C1(C)(N(C)C)CCN(C(C2(CNC(=O)CC3(O)CCCCC3)CC23CCC3)=O)C1 20858,N1(C(C=C(C)C(F)F)=O)CCC(C(CO)NC(=O)Cc2cc(C)cs2)CC1 20859,N1(C(C(C2CCC(=O)N2)C)=O)CC(C)CN(C(C2CC(F)C2)=O)CC1C 20860,C1(NC(C2OCCC(C)C2)=O)CCC12CN(C(=O)Cc1cccc(C#N)c1)C2 20861,N1(C(CC2C(OC)CC2)=O)CCC2(CC2NC(=O)C(C)COC)C1 20862,CC(C)(O)C(F)C(=O)N1CCC(C(=O)NC2(C3CC3)CCC2)CC1 20863,c1(C(=O)NCC(CNC(c2ccnn2CC(C)C)=O)OC)ccc(N(C)C)cc1 20864,CC1(C)CN(C(=O)C(=O)C(C)(C)C)CC(CNC(C2CCCC2(F)F)=O)O1 20865,c1(N2CCN(C(c3ccccc3)CC)CC2)nc(C(=O)OC)ncc1F 20866,c1(C(=O)NCC(C2CCOC2)NC(c2scc(COC)c2)=O)ncccc1F 20867,C1(C(=O)NCC2C(F)(F)CCN(C(C(=O)N(C)C)=O)C2)CCCCN1S(N)(=O)=O 20868,C1(C(N(C(CC)CO)CC)=O)CC2(CC(NC(=O)C(C3CCCCC3)F)C2)C1 20869,c1(CNC(C2CCCN(C(=O)Cn3cccn3)C2)=O)nc2ccccc2n1C1CC1 20870,c1(CC)cccc(F)c1C(=O)NCC1(C)CCCN1C(c1n[nH]c(C)c1F)=O 20871,C(CSc1ccccc1)(C(=O)NCC1CC1CNC(=O)C(=O)N(C)C)SC 20872,c1(C(N2CC(CNC(c3scc(C)c3C)=O)C3(C2)CC3)=O)snc2ccccc12 20873,Cc1ccc(CC(=O)N(CC(C)NC(=O)C(O)CC2CCCC2)C)c(F)c1 20874,CC1(C)CN(C(=O)Cc2cccnc2Cl)C(CNC(C2(C)CC2C(F)F)=O)CO1 20875,c1(CC)cc(C)c(C(=O)N(C2CCC(NC(c3cn(C)[nH]c3=N)=O)C2)C)o1 20876,c1(C(N2CCC(CC(N3CC(C)C(=O)CC3)=O)CC2)=O)c(F)cccc1C#N 20877,CCCCCC(=O)N1CC(O)CC1C(=O)N(CC(C)(CO)CO)C 20878,c1(OC)ccc(N)c(C(N2CCC3(NC(=O)C(N)=O)CC3C2)=O)c1 20879,Cc1cc(F)cnc1-c1cn(C2CCN2C(c2n[nH]c(O)n2)=O)nn1 20880,C(=O)(CC(C)CC(C)C)NCc1cccc(NC(c2c(OC)n(C)nc2C)=O)c1 20881,c1(C(C(=O)NC)N(CC(=O)OC)C(C)C)cncn1CC 20882,c1(C(=O)NCC(CN(C(C2(OC)CCOC2)=O)C)(C)C)ccc(CF)cc1.C(N)=O 20883,C(c1ccccc1Br)=CC(=O)NCC1N(C(C(C)OCC#C)=O)CCCC1 20884,O=C1CC(C(=O)NCC2CCCN2C(C2(O)CCSCC2)=O)NC(=O)N1 20885,c1(C(N2CCC(C(C(N3CC(C)(CSC)C3)=O)F)C2)=O)cnc(C)cc1C 20886,C1(CC=C)(C(N2CCC(C(F)F)C2)=O)CCN(C(=O)COC2CCC2)C1 20887,N1(C(C2CCCN(C(=O)C(O)C3CCC3)C2)=O)CCOCCC1C1CC1 20888,Cc1c(Cl)ccc(C(=O)NC(C2CCN(C(c3ccc(=O)oc3)=O)CC2)C)c1N 20889,C1(NC(C(C)NC(C)=O)=O)CC(C)(C(=O)NCCc2cc(C)no2)C1 20890,c1(C(=O)NC(C(C(=O)NCCCN(CC(C)C)C)C)C)cc(F)ccc1F 20891,C1(CNC(Cn2c(C)ccc2C)=O)CC2(CC(NC(C3CCNC3=O)=O)C2)C1 20892,Cn1cc(C(=O)NC2CCCC(NC(=O)Cc3ccccc3)C2)c(O)nc1=O 20893,Cc1cc(C(=O)NC2CCC2CNC(=O)CNS(N)(=O)=O)cc(F)c1 20894,c1(CC(=O)NC(CNC(c2nc(C(C)=O)sc2)=O)C)ccc(C(F)F)cc1 20895,C1(NC(c2nccc(COC)c2)=O)CCCN(C(c2c(N)cccc2F)=O)CC1 20896,c1(C(N(CC(CC)NC(c2oc(C)nc2C(F)(F)F)=O)C)=O)cnc(O)cc1C 20897,c1(CC(=O)NCC2CC2CNC(=O)CCCCN2CCCC2)nnc2n1CCOC2 20898,c1(-n2ccc(C(N3CC(c4cn(CC(F)(F)F)nn4)C3)=O)n2)ccccc1C 20899,C(=O)(C(C)(C)C(C)O)NCC1CC(NC(c2ccc(C(C)=O)cc2)=O)C1 20900,C12(CNC(CCC#C)=O)CC(CN1C(=O)CC1CCCCC1)C2 20901,c1(-c2c(OC)cnc(OC)n2)c(C(F)(F)F)cccc1C1CCc2ccccc21 20902,c1(OC)ncc(C)cc1C(N1CC(NC(=O)C(N2CCOCC2)C)C(CO)C1)=O 20903,c1(CC(=O)NCCCNC(c2ccc(F)s2)=O)nsc2ccccc12 20904,c1(C(=O)NC(CC)CNC(C2CC2(F)F)=O)ncc(C)cc1C(F)(F)F 20905,N1(C(C(CC)CN(C)C)=O)CCC(C)(C)CC1C(=O)NCC1=CCCOC1 20906,c1(C(N(C2CCN(C(C34CC(C(F)F)(CO3)C4)=O)C2)C)=O)cnccc1Cl 20907,c1(C(=O)NCC2CC(NC(C(C)C(C)O)=O)C2)c(F)cc(F)cc1Br 20908,C1(C(N2CCN(C(=O)CNC(=O)C(C)OC)CC2)=O)(NC(C)=O)CCC(C)CC1 20909,C(=O)(CCCCC1CC1)NCCCN(C(C(C)N(C(C)=O)C)=O)C(C)C 20910,N1(C(CCC#C)=O)CC2CN(C(c3ccc(C#N)c(F)c3)=O)CCC2(CO)C1 20911,n12nc(ccc1=O)C1N(CCCSC1)C(=O)C2CCC.c1ccccc1.OC 20912,CC1(C(=O)NCC2CC(NC(c3ccnc(O)c3)=O)C2)CC2CC2C1 20913,C(C(C)(C)CNC(C12CCC1C2)=O)NC(C1(CC=C)CC1)=O 20914,C(c1ccccn1)=CC(=O)NC1(CC)CN(C(=O)C(C)=C2CC2)C1 20915,c1(C(N2CCCN(C(C(C(C)O)(F)F)=O)CC2)=O)nccc2[nH]ccc12 20916,C(=O)(C1=C(C)C(C)(C)OC1=O)NCC12OCC(NC(Cc3ccn(CC)n3)=O)(C1)C2 20917,n1(CC(=O)NC2C3CC(NC(C(C)=C4CCC4)=O)CC32)cccc(O)c1=O 20918,C1(NC(c2nc(SC)sc2)=O)CCN(C(=O)C(C)OCC(C)C)C12CC2 20919,c1(C(N2CCC(CCOC)(NC(=O)C(C(C)C)SC)C2)=O)cnc(Cl)c(F)c1N 20920,c1(CC)ccc(C(=O)NCC2OCCC2C(=O)NCCCOC2CCC2)cn1 20921,c1(NC(c2cn(CC)nc2C2CC2)=O)cccc([N+](=O)[O-])c1Cl 20922,C(CCCC(=O)NCC(C)N(C(=O)CCN1CCC(C)CC1)C)N(C(C)=O)C 20923,CC1CN2CCN1CC2C(N1CCN(C(c2cc(O)cc(N)c2)=O)C(C)C1)=O 20924,N1(C(c2n(C)cnc2)=O)CCC(NC(c2cn(-c3ccc(F)cc3)nn2)=O)CC1 20925,N1(C(CSc2c(C)n[nH]c2C)=O)CCN(C(c2cncn2C)=O)C(CF)C1 20926,C(N=c1nc(C#N)[nH]cc1Cl)C1CN(C(c2c(C(C)C)ocn2)=O)C1 20927,C(=O)(CCCCC(F)(F)F)N1CCC(CNC(C2CCN(CC)C2)=O)C(F)(F)C1 20928,c1(OC)cccc(Cl)c1CC(=O)NC(C)CCNC(c1ccnn1CC#N)=O 20929,N1(C(C(CC=C)(C)C)=O)C2CCC1CC(NC(=O)C=Cc1nc(C)c(C)[nH]1)C2 20930,C1(C(=O)NCC2CCCCC2O)COC2(C1)CN(C(C1CCC=CCCC1)=O)C2 20931,C(=O)(C(CC(F)F)N(C(=O)C(n1ccc(C)n1)C)C)N(CC#C)CC=C 20932,Cc1cccc([N+](=O)[O-])c1NC(C)CCNC(C1(CF)CCC1)=O 20933,c1(OC)c(C)ccc(C(=O)NCCC2CC(NC(c3cc(C)[nH]n3)=O)C2)c1F 20934,C=CC(C)(CCOC)C(=O)NCC1(CNC(=O)CCCC)CC12CCC2 20935,C(=O)(C(C)CCC(C)(C)C)N1CCCC(CC(=O)NC(c2cnc[nH]2)C)C1 20936,c1(NC(C2COC(CNC(c3ccc(NC(C)=O)s3)=O)C2)=O)ncc(F)cn1 20937,c1(CC(n2ccnc2C(=O)CN2CCC(C)(F)C2)C)c(Cl)cncc1Cl 20938,c1(NCC2(O)CCN(C(Cc3cccc(C)c3F)=O)CC2)cc2nncn2cn1 20939,Cc1ccc(CNC(c2ccc(-c3n[nH]c4c3CCC4)cc2)=O)c2ccccc12 20940,c1(N(C)C)ncc(C(N2CCCC(CNC(=O)C(F)CC3CCC3)C2)=O)cn1 20941,CC(C(=O)N1CCC(C)(CNC(=O)C(CCO)N(C)C)CC1)C(F)(F)C(F)F 20942,C(C(C(C)(C)C)NC(=O)CCC(F)F)NC(C1CCC(N(C)C)C1)=O 20943,N1(C(C(C(C(CC)C)O)C)=O)CCC2(CC1)CCN(C(C13CC(F)(C1)C3)=O)CC2 20944,C1(N(C)C)CCC(NC(=O)CCN2CCCC2)CC1 20945,N1(C(c2cnc(OCC)nc2)=O)CCN(C(c2nc(C)no2)=O)C2(CC2)C1 20946,c12ccc(cc1)NC(=O)CC2.C1(CCC)CC(C(C)(C)C)C1 20947,c1(OC)cc(C(N2CCC(F)(C(=O)Nc3cnc(C(C)(C)C)nc3)C2)=O)nn1C 20948,Cc1cc(C(=O)NC2CCC(CCNC(c3nonc3N)=O)C2)oc1Br 20949,C1(CCC(=O)OCC)CCN(C(c2csc(C3CCCNC3)n2)=O)CC1 20950,c1(CC(C)C(=O)NCC2CN(C(=O)CN(C)C)CC2O)ccc(Br)cc1F 20951,N1(C(CC(C)(C)C2CC2)=O)CCC2(CCCCN(C(C3CCCO3)=O)C2)C1 20952,C1(C(=O)NC2C(NC(C3(C)CC=CC3)=O)COC2)CCC2(CCOCC2)O1 20953,C1(C(=O)NCC2C(CNC(COCC=C)=O)C2)CCC(C(=O)OC)O1 20954,C1(C)(NC(C2C(C)C2C)=O)CCN(C(=O)CC2CCNC(=O)C2)CC1 20955,C1(NC(C2(CC)COC2)=O)CCC2CN(C(c3cc(C)cnc3C)=O)CC2C1 20956,c1(N(C(C)=O)C)ccccc1C(=O)NCC1CC1NC(=O)CCc1ccon1 20957,C=CCCN=C(NCCc1ncc(C)cn1)NC1CCN(CC2CCCC2)C1 20958,CCCCCCCCC(=O)N1CCN(C)C(CNC(C2C3CCC(F)(F)C23)=O)C1 20959,C1(C(N2CCC(N(C)C)C2)=O)CC2C=CC1N(C(=O)C(C)(C)C(=O)N(C)C)C2 20960,Cc1cc(Cl)c2ccc(C(N3CCC(C(C)NC(=O)CC(C)C)CC3)=O)cc2n1 20961,C(=O)(CCC1CCc2ccccc21)N1CCC(CNC(CCCCC)=O)C1 20962,C(=O)(C1CC(=O)c2ccccc21)N1CCC(NC(COCC)=O)C1 20963,c1(N2CCCC3(NC(Cc4cn(CC)nc4)=O)C(C2)C3)nc(O)c2c[nH]nc2n1 20964,C(=O)(CC(C1CCCC1)NC(=O)CCCn1cc(CC(C)(O)CC)nn1)OCC 20965,C=C(C)CCC(=O)N1CCC(N2CCN(c3ccc(C(=O)OC)s3)CC2)C1 20966,CCC(C(=O)NCC1CN(C(c2cnn(C(C)C)c2)=O)C(C)(C)C1)C(C)(F)F 20967,C(CC(C)C(F)(F)F)NC(c1n(CC(=C)C)nnn1)CCC1CCCO1 20968,C1(NC(=O)C=CCO)CN(C(c2[nH]ccc2C2CC2)=O)CC1CC1CC1 20969,c1(CCN(C)CCN(C(=O)CC2(CS(C)(=O)=O)CC2)C)ccccc1 20970,N1(C(C(C)(C)NS(C)(=O)=O)=O)CCC(NC(C2CCOC2)=O)C1C(C)(C)C 20971,N1(C(CCc2c(C)noc2)=O)CCC(C)(C)C1CNC(c1cc(F)cc(F)c1)=O 20972,c1(NCCCC(C)CO)ccncc1S(=O)(=O)NC1CCc2c(nnn2C)C1 20973,c1(C2C(C(N3CCC(N(C(C(CC)SC)=O)CC)CC3)=O)C2)cc(F)ccc1C 20974,n1(CC)ccc(C(=O)NC2(CC(=O)NOCC3CCCCC3)CCCCC2)c1C 20975,CC1(C)CCC(O)(C(=O)NCC(O)CNC(C2CCC=CO2)=O)CC1 20976,N1(C(Cc2c(C)ocn2)=O)CCC2(CC1)CC(C)N(C(=O)CCS(C)(=O)=O)C2 20977,c1(COC)ncc(C(=O)NC(C)(C)C(C)NC(C2C(C)C2C)=O)c(=N)[nH]1 20978,c1(C(=O)NC(CN(C(=O)Cc2nnc(O)s2)CC)C)nn(C)cc1S(C)(=O)=O 20979,c1(NC(C(C)NC(C)=O)=O)cn(CCCC2CCN(C(=O)CCC3CC3)C2)nn1 20980,C1(CNC(C2CC(C(C)(C)C)C2)=O)CCCCCN1C(C1CC12CC2)=O 20981,c1(C(=O)NCCC(C)N(C)C(C2CC(O)C2)=O)c[nH]c2cc(Br)ccc12 20982,c1(N(C)CC2CCCCN2C(=O)CCN2CCCS2(=O)=O)snc(Cl)c1C#N 20983,Cc1nncc(C(N2CC3CCC3(CCNC(c3cnsn3)=O)C2)=O)c1C 20984,c1(C(=O)NCC(CN(C(C2CCC3CC23)=O)CC)(C)C)cn2ccnc2s1 20985,C(C)(C)(CCC(=O)N1CCCC(NC(c2nn(C)nc2Br)=O)C1)OC 20986,C#CC1(O)CC(C(N2CCC(C)C2C)=O)C1.C1(CSCC)C(=O)N1C 20987,CCCCCC(C(=O)N(CCCN(C(=O)CN1CCCCC1C)C)C)C(C)C 20988,c1(C(C(N2CC(C)C(NC(=O)C3=CCCC3C)C2)=O)=O)ccc(F)cc1F 20989,c1(C(=O)OC)ccc(F)c(-c2cnc(C(F)F)s2)c1OC 20990,c1(CC(C(N2CC(CCO)(NC(Cc3nc(C)[nH]n3)=O)C2)=O)C)ccccc1C 20991,c1(CN(CC(=O)N(C)C)CCN(C)C)ccc(C2=CCCCC2)cn1 20992,C1(NC(c2c(CC)cno2)=O)CCC2(CC1)CN(c1nc(C3CC3)ns1)C2 20993,N1(C(C(C)SCCCC)=O)CC2(C1)CN(C(=O)C(CCC)OCC)CC(C)(C)O2 20994,c1(C2(C(N3CC(CNC(CC=CC)=O)C(N(C)C)C3)=O)CC2)ccc(Cl)cc1F 20995,C(CCOC)(C(=O)NCC(COC)OC)NC(C(C=C)OC)=O 20996,c1(N(C)C(C2CC(=O)NC2(C)C)=O)nc(C2CC2)nc(=N)[nH]1.C12(CC1)CN2 20997,C1(C(N2CCN(C(C3CCC(C)(C)O3)=O)CC2CCO)=O)CCc2ccnn2C1 20998,Cc1ccc2c(c1)c(CCNC(c1cc3c(Br)cnn3cn1)=O)cn2C 20999,C(=O)(C1CCc2ccccc21)NC1CC2(CN(C(C3=CCCN(CC)C3)=O)C2)C1 21000,C(CS(=O)(=O)CC(=O)NCC1CCCC1NC(=O)C=Cc1ccoc1)OC 21001,C1(C(=O)NCC#CC)C=CC(NC(=O)CC(=O)OCC)C1 21002,c1(NC(COC(C2C(CCOC)C2)=O)=O)cc(OC)cc(O)c1 21003,FC1CCCCCC1N=c1[nH]c(=NCC2CC3(CCOCC3)CO2)[nH]c2c1SCC2 21004,N1(C(CNC(C(C)NC(C)=O)=O)=O)CCC(C(=O)NC(CN(C)C)C(C)C)C1 21005,C1(OCc2cc(C)on2)C(C)CN(C(=O)C(=O)NCC(=O)N)CC1C.C(C)(C)(C)O 21006,C=CCN=C(NCc1cnn(CC)c1C)NCC(C(C)(C)C)OC 21007,N1(C(C(CC)C2CCOCC2)=O)CCC(NC(c2cnoc2C)=O)C1C(C)(C)C 21008,CC1Cc2cc(CC(N3CCCC(CNC(=O)C=C4CCC4)CC3)=O)ccc2O1 21009,C1(OC)CC2CCC(C1)N2C(=O)CNC(C1(C(N2CCCC2)=O)CCC1)=O 21010,Cc1nn(C)c(C(=O)NC2CC3(C2)CC3NC(=O)C(C)(C)C(=O)N(C)C)c1Br 21011,C1(NC(c2occ(C)c2)=O)CCCCC1NC(C1CCC(C(N)=O)O1)=O 21012,c1(C(=O)NCC2CN(C(CC=C(C)C)=O)C2)ccc2nc(C(F)(F)F)cn2c1 21013,C1(NC(C2CC(C(C)C)C2)=O)COC2(C1)CN(C(c1coc(C(N)=O)c1)=O)C2 21014,N1(C(C2N(C(C)=O)CC(O)C2)=O)CC2(CC(NC(c3cccc(F)c3O)=O)C2)C1 21015,CCCCC(CCCC)NC(C1CC(F)CCN1C(C1CCCC(=O)N1)=O)=O 21016,CC1(C)CCCC1C1CCN(C(N2CCCC3CC(O)CCC23)=O)C1 21017,C1(CNC(c2cc(OCC)no2)=O)CC(C(=O)NC2CCOC2=O)=NO1 21018,c1(CNC(C(C)c2ccsc2)=O)cc(Cl)cnc1O 21019,c1(OCC)ccc(C(=O)NC(C)(C)CNC(c2nccc(C(F)F)n2)=O)cn1 21020,C1(NC(=O)C(F)C2CCC2)CCCCN(C(c2cnc(C(F)F)cn2)=O)C1 21021,CC1(F)CC(N=c2[nH]c(N3C4C=CCC3CCC4)nc3c(F)cccc23)C1 21022,C(N=c1nc(N2CC(=O)NC3(COC3)C2)c2c([nH]1)CCCC2)C1C(C)CCNC1=O 21023,C1(C(=O)NC2CC(CC)OCC2)CCN(C(c2cn(C)nn2)=O)C12CC2 21024,c1(OC)nc(-c2ccc(-c3nccn3C(C)C)cc2)cc(C)n1 21025,CC1(C)NC(=O)CCC1NC(C1CNC(=O)CN1C(=O)CC1CSC1)=O 21026,c1(OC)cc(F)c(C(=O)NCCC(C)NC(=O)CC2C(=O)N(C)N=C2C)c(Cl)c1 21027,c1(CC)c(C(=O)NCCCN(C(=O)CC(C)(C)N(C)C)CC)nnn1C(CCC)C 21028,c1(NC(CC2C(CNC(C(C)(CO)OC)=O)C2)=O)cc(F)ccc1C 21029,C1(C2CCN(C(c3cc(CO)[nH]n3)=O)CC2)(NC(C(C)N2CCCC2)=O)CC1 21030,c1(OC)ccc(F)cc1NC(C1CC1C(=O)Nc1ccc(Br)c(F)c1)=O 21031,C#CCC(CC(=O)N1CC(n2cccn2)C1)NC(=O)CCNC(=O)COC 21032,c1(CN(C(Cn2c(C)cnc2)=O)C2CC2)ccccc1N(C)NS(C)(=O)=O 21033,c1(OCC)cccc(C(=O)NCCC2CCN(C(=O)Cc3conc3C)CC2)c1 21034,c1(C(=O)NC2(COC)CN(C(=O)Cc3ccsc3C)C2)cnc2c[nH]nc2c1 21035,CC(CC(=O)N1CC(C)(C)CC1CNC(C1CCc2ncnn2C1)=O)C(F)(F)F 21036,C1(NC(C2CC(O)CN2C(=O)CCN2CCC(F)C2)=O)CCCN(O)C1=O 21037,c1(C(N2CCC(F)(CNC(C3CCC3F)=O)CC2)=O)ccc2c(c1)CNC2=O 21038,N#Cc1ccc(C(N2CCCC(NC(=O)C=CC3CCOCC3)C2)=O)nc1 21039,N1(C(C=C(C)CNC(c2cn[nH]c2)=O)=O)CC(CCO)OCC1C 21040,C(CCCCCCCO)=CC(N1C(CCNC(CCCC#C)=O)CSCC1)=O 21041,N1(C(c2ccc(N(C)C)cc2)=O)CC(O)C(O)C1CNC(=O)CCCCCO 21042,C1(NC(CCOCCOC)=O)CN(C(c2ccc(F)c(C#N)c2)=O)CC2(CC2)C1 21043,CCC(C)CC(=O)NCCOCCNC(=O)CCCCN1CCCCC1 21044,C(=O)(CC(O)c1ccccc1)NC1C(NC(C(F)=CCC)=O)CC1 21045,CC1CCC(C(=O)N(CC(F)Cl)C)N(C(c2cncc(F)c2)=O)C1 21046,Cc1cc(NC(=O)CN2CCCC2)ccc1N1CCCC1=O 21047,C=CCC(C)(C)CCNC(C1CC(CCNC(=O)C(C)(C)C(=C)C)C1)=O 21048,N1(C(c2c(CCC)nns2)=O)CCN(C(c2ccc(C(C)F)cc2)=O)CC1CC 21049,C(=O)(C1CCCn2cncc21)NCC(CNC(c1sc(C)c(O)n1)=O)(C)C 21050,C(=O)(C(O)CC(C)C)N(CC)CC1CCCCN1C(c1csnc1C1CC1)=O 21051,S(=O)(=O)(c1cccc(=NCc2ccc(N3CC=CC3)cc2)[nH]1)N1C(C)CCC1 21052,C1(C(N2C(CO)CC(NC(Cn3ccc(C)n3)=O)C2)=O)CCOC(C)(C)C1 21053,N1(C(=O)NC(C)(C)C)CCN(C(N)=O)C(C2CC2)C1 21054,C(=O)(C(C)(C)C(=O)NCC1CC1CNC(=O)C1=CCCCO1)N(C)C 21055,C1(C(N2CCC(C(CNC(=O)CCc3cn[nH]c3)F)CC2)=O)CCC(F)(F)CC1 21056,c1(NCC(CC)NC(C2(CC#C)CCCC2)=O)cc(C)nc2cc(C)nn12 21057,n1(C(C)C)ncnc1CNC(=O)C=CC(c1cnn(C)c1)=O 21058,N1(C(CS(CC)=O)=O)CC2CC(NC(c3ccc(SC(C)C)cc3)=O)C1C2 21059,CC1=C(C(=O)N2CCCCCC2Cc2cn(CC3CCOCC3)nn2)CCC1 21060,CC(C)CCCC(=O)NC1(CF)CCN(C(c2coc3c2CSC3)=O)C1 21061,CC(C(=O)N1CC2CCC1C2NC(c1cc(N)c(F)cn1)=O)C(C)(F)F 21062,C(=O)(C(C)(CC)C(=O)NCCOC(CCCC(=O)OC(C)(C)C)C(C)C)OCC 21063,C1(NC(C2CC2c2cccc(F)c2)=O)C=CCN(C(=O)CNC(=O)C(F)(F)F)C1 21064,C(=O)(CCCCCCS(N)(=O)=O)N1CCCC(CNC(C(C(C)C)OCC)=O)C1 21065,C1(C(N2CC(OC)C(C(N3CCC(C)(N(C)C)C3)=O)C2)=O)CCC2(CC1)CC2 21066,c1(C(N(C2CCN(C(=O)CC=C(C)C)C2)CC)=O)n[nH]c2c1CCC2 21067,C#CCC(O)C(=O)N(C)CC1CCCCN1C(=O)CCSCc1ccc(C)cc1 21068,S(C(F)(F)F)CC(=O)N(C1CC(NC(=O)CSCC(F)F)C1)C 21069,c1(OC)c(CN=C(NCC(=O)NCC2CCOC2)NC2CCCC2)cccc1F 21070,N(C1CCc2ccccc21)C(C1CCC(NC(c2cc(C)c(N)cn2)=O)C1)=O 21071,C(CC(N)=O)(C(=O)NC1CC1NC(=O)CC1CC1)NC(CC(C)C)=O 21072,C1(O)(C(CNC(COCC(C)C)=O)C)CCN(C(=O)Cc2nc(=N)[nH][nH]2)C1 21073,c1(CC)ncccc1NC(=O)COC(c1[nH]c(C)nc1Cl)=O 21074,C1(CNC(c2c(C)cncc2)=O)CCCN(C(=O)Cc2cc[nH]c2)CC1 21075,C1(CCNC(C=COCC)=O)CN(C(=O)C(C)CNC(=O)OC(C)(C)C)CCO1 21076,c1(N(C2CC=CC2)C(N2CC(C#N)(CCF)C2)=O)nc2ccccc2s1 21077,N1(C(CCC2CCC(C)O2)=O)CC2CC(C(=O)NC(C)CF)(C2)C1 21078,c1(C(CC(=O)NCCCNC(c2cn(CCOC)nn2)=O)C)ccc(F)cc1F 21079,C1(C(N)=O)CN(C(c2csc(C(N)=O)n2)=O)CCC1NC(C1(C)CCC(=O)C1)=O 21080,c1(C(N2CCC(F)(C(=O)OC(C)(C)C)CC2)=O)cc2n(n1)CCCN2 21081,Cn1nc(C2CC2)cc1C(=O)NC(C1CCOC1)CNC(C1CC(O)C1)=O 21082,c1(C(C)NCC(COCC)C)cc(C(=O)OC)c2n1CCOC2 21083,N1(C(CCSCC)=O)CCC(C2CCC2)(CNC(c2cc(=O)n(C)o2)=O)CC1 21084,CC(C)C(C(=O)N1CCCCC1CNC(=O)C(C)CCN(C)C)n1cnnc1 21085,CN1CCCC(O)(CC(=O)NCCC2(O)CN(C(c3cc(Cl)ncc3O)=O)C2)C1 21086,c1(CC(=O)NCCCC2CN(C(c3c[nH]ccc3=O)=O)CCO2)ncncc1Cl 21087,Cc1ccc(F)cc1C(N1CC(C)(C(=O)NC(C)(C(N)=O)C(C)C)C1)=O 21088,CC(C)C(C(=O)NC1(CNC(=O)CSc2cccc(Cl)c2)CC1)c1ccn(C)n1 21089,CC(C)CC(O)C(=O)NC1CCN(C(=O)CN2CCN(C)CC2)C1C(C)(C)C 21090,C1(CNC(C2OCC(C)C2)=O)CC2COCC2N1C(c1c[nH]cc(F)c1=O)=O 21091,N1(C(C)=O)CCC(NC(=O)C(C(C)C)NC(C2CCCC2)=O)CC1 21092,C1(NC(C(C)NS(C)(=O)=O)=O)C=CCN(C(c2cc(-c3cccs3)on2)=O)C1 21093,N1(C(C(CC#C)O)=O)CCn2nc(CNC(C3(O)CCCC(C)(C)C3)=O)cc2C1 21094,C1(NC2CC(C(F)(F)F)(OC)C2)CNC2(CCC2)C1 21095,N1(C(C2CCN(C(C)=O)CC2)=O)CC(C)CN(C(c2cc(NOC)no2)=O)CC1C.CCN 21096,Cn1c(C(N2CCOC(CNC(c3csc(O)n3)=O)C2)=O)cc2c1CCOC2 21097,N1(C(C(C2CCC2)OCC)=O)CCC(C)(CCNC(c2c(Cl)nsc2Cl)=O)C1 21098,C1(NC(c2c(OC)nsc2)=O)CC(C(=O)NC2CCNC(=O)C2)C1(C)C 21099,C12(O)CCCN(C1)CC=CCC(=O)N(C)C2.C(C(C)C(=O)OC)SC 21100,c1(OC)ncc(C(=O)OCC(C2CCCCCC2)(C)O)cc1F 21101,CC1CCCCC1CN1CCC(NC(=O)CNC(=O)NC2CCOCC2)CC1 21102,CC1CCN(C(c2nnnn2C)c2cscn2)C(C(=O)OC(C)(C)C)C1 21103,c1(C(=O)NC2(CCNC(c3ncccc3Cl)=O)CC2)c(O)nnc2c1COCC2 21104,N1(C(C(C)NC(COC)=O)=O)CCC(O)(CCNC(=O)Cc2csnn2)C1 21105,C(CNC(c1ccc(NC(=O)CCCN(C)C(C)=O)o1)=O)(C(F)(F)F)OC 21106,Cc1sc(O)nc1C(=O)NCC12CC1CN(C(C13CCC(CC1)C3)=O)C2 21107,c1(C(C(=O)NCCCCN(C)C(C2CCCCS2)=O)(C)C)ccc(Cl)nc1 21108,CCCCCCCC(=O)NCC1(F)CCN(C(c2cnc(N(C)C)nc2)=O)CC1 21109,C(c1ccncn1)=CC(=O)NC1CC(NC(C2C3COCC23)=O)C1 21110,N1(C(CCC2CCN(C(=O)CCc3nncs3)CC2)=O)CC2CCCCC12 21111,c1(OCC)ncc(C(=O)NCCC(O)CNC(=O)CCC2CCCOC2)s1 21112,N1(C(C2C(NC(C(n3c(C)ccn3)C)=O)CCO2)=O)CCC(C(C)O)CC1 21113,CCS(=O)(=O)CC(=O)NCC(C)(C)CN(C)C(C1CC2CC(=O)C1C2)=O 21114,C1(C(=O)NC2(CO)CN(C(C3(COC)CC3(F)F)=O)C2)Cc2ccccc2S1 21115,c1(C(=O)NCc2ccsc2-n2cnnn2)ncsc1-c1ccccn1 21116,C(=O)(C1CCCc2scnc21)NC1C2N(C(c3ncc(C)cc3F)=O)C(CC2)C1 21117,C(=O)(CC(O)CC(C)C)N1CC(C(NOCC2CC(=C)C2)=O)C(F)(F)C1 21118,N1(C(c2cc(CC)no2)=O)CCCC(CCNC(C2CC23CC3)=O)C1 21119,CC1(C)NC(=O)OC12CCN(C(C1(O)CC(C)(C)C1)=O)CC2 21120,N1(C(c2cncc(C)c2C)=O)CCC2CN(C(=O)C(O)C3CC3)CC12 21121,c1(-c2c(C)ccc(C(F)(F)F)c2)ccc2[nH]c(C(N3CCNC(=O)C3)=O)cc2n1 21122,c1(C(=O)NC(CCNC(C=Cc2ccc(CC)o2)=O)C)ccn2cnnc2c1 21123,N1(C(CCc2ccc(C)o2)=O)CCOCC1CNC(c1ncoc1C(C)C)=O 21124,CCC(CC(=O)N1CCC(NC(=O)Cc2ccon2)C(O)C1)C(C)C 21125,C12(CNC(C(C)OCC)=O)CC(NC(=O)C=Cc3ccncn3)(CO1)C2 21126,N1(C(C2C(C(C)=O)C2)=O)CC(CNC(c2ccc(=O)n(CCO)c2)=O)CC(C)(C)C1 21127,C1(CC(=O)NCC2CC2c2ccc(Cl)cc2)CCN(C(C2(CO)CCC2)=O)CC1 21128,c1(C(N2CC(C)(CNC(c3cccc(OC)c3Br)=O)C2)=O)ccn2cnnc2c1 21129,c1(CC)ccc(C=CC(N2CCN(CCNC(C3CCCC3C)=O)CC2)=O)cc1 21130,N1(C(=O)CCCCC2CC2)CCCN(C(C2C3CCC23)=O)CC1 21131,C1(CNC(C2C(C)C2C)=O)CN(C(=O)COc2ccc(CO)cc2)C2(CCC2)C1 21132,c1(CC(N2CC(NC(CC(C(=O)OC)C)=O)C(C)(C)C2)=O)ccn2cncc2c1 21133,CN1CCOC2CN(C(=O)C3=CCN(C(C4CCOCC4(C)C)=O)C3)CC12 21134,C=CC1CCC1C(=O)N(C1CN(C(=O)C=CC(CC)=CC)C1)C 21135,c1(C(=O)NCCN(C(c2oc3ccccc3c2Cl)=O)CC)ccc2nncn2c1 21136,Cc1noc(C)c1CSCC(N1CC(NC(c2cc(C3CC3)no2)=O)C(C)C1)=O 21137,c1(C(C(=O)NC)N(CC(C)(C)S(C)(=O)=O)C)cccc2c1CCOC2 21138,c1(C(C(=O)NC2CCCC2)N(CC(COC)C)C)ccncc1F 21139,N1(C(C)C(=O)NC23CC(NC(=O)COCC(=O)OC(C)(C)C)(C2)C3)CCN(C)CC1 21140,c1(C(C)O)ccc(C(=O)NCC2CCCCN2C(=O)C(F)=CC2CC2)cc1 21141,C(=O)(CCCC(=O)NCC(CO)NC(c1cccc(C2CCC2)c1)=O)N(C)C 21142,N1(C(CCSC)=O)CC2CCC(CNC(=O)C(C)(C)c3ccno3)C2C1 21143,C1(CNC(c2cscn2)=O)CN(C(c2ccc(F)cc2F)=O)C2CCN1C2 21144,c1(C(=O)NCCC(C)NC(c2ccc(-c3ccccc3)[nH]2)=O)cc2sccc2s1 21145,C(C(=O)Nn1cccn1)C1C(C)CCC1.C12(CCCCC1)C(=O)N2 21146,C1(CCC)(NC(=O)Cc2ccc(OC)c(Cl)c2)CCN(C(=O)C2=COCC2)CC1 21147,c1(CC)n[nH]cc1CNC(=O)C=CC(C)(C)NC(=O)C(F)=C(C)C 21148,C1(O)(CN(C(=O)CC2CCCO2)C)CCN(C(C2CC3C=CC2C3)=O)CC1 21149,C(CC(C)C(F)(F)F)NC(C(C1(O)CN(C(C2(COC)CCCO2)=O)C1)F)=O 21150,C1(C(=O)NCCC(CCNC(C(C)=CC)=O)C)CC1C1(C)CCOCC1 21151,C(C(CC(C)C)C(=O)N(C)CC=CC(=O)NCC(C)(O)C1CCCC1)OC 21152,c1(C(=O)NC2CC3(C(NC(c4c(C)onc4)=O)C3)C2)cc2c(o1)CCCC2 21153,C1(NC(C(CNC(=O)OC)(C)C)=O)CCC2(CC1)CC2C#N 21154,C1(COC)(CNC(C2CCC2(C)C)=O)CCN(C(c2cc(Cl)nnc2O)=O)CC1 21155,C(CC(F)F)(C(=O)N=c1ccn(CCO)[nH]1)NC(C(COC(CC(C)C)=O)C)=O 21156,c1(C(NOC2CCC(N)C2)=O)cccc(Br)c1.C1(=O)CCCN1 21157,c1(C(N2CC3C(CNCc4ccc(C(=O)O)o4)(C3)C2)=O)cc(OC)c(O)c(Cl)c1 21158,C1(NC(c2nccc(OC)c2O)=O)CN(C(=O)CCCCF)C2(CCOCC2)C1 21159,C1(NC(C2C(NC(C(=O)N(C)C)=O)C2)=O)CCCC1C(C)(C)C 21160,c1(C(=O)NC2COCCN(C(C(COC)(C)C)=O)C2)ccc2ccccc2c1F 21161,Cc1ccnc(C(=O)NC2CCC(C(=O)NCC(c3ccccc3)O)C2)c1 21162,N1(C(C=Cc2ccc(C)s2)=O)C(C)CC2CN(C(=O)C(C)C(O)C(C)C)CC12 21163,C1(c2cccs2)(C(=O)NC2C(CNC(C(C=CC)O)=O)C2)CCCCC1 21164,c1(C(N2CCOCC2c2nc[nH]n2)C(=O)NCCC)ccc(C)c2c1CCC2 21165,N1(C(C(CC)OC)=O)CC2CCC(NC(c3cnoc3C)=O)CC2C1 21166,CS(=O)(=O)C1CN(C(C2CCOC2)=O)CC1NC(c1cn2cc[nH]c(=O)c2n1)=O 21167,N1(C(C(c2n(C)ncc2)CO)=O)CCC2(CCCO2)CC1 21168,C(=O)(CCC(C)(C)CNOC(C)(C)C)NC(CCOC)COC.OC 21169,c1(C(COC)NC(C2CC(O)(CO)C2)=O)ccc(F)cc1 21170,c1(SCC)cnccc1C(=O)NCCC(C(C)C)NC(=O)C=CC1CCCN1C 21171,Cc1cc(C)c(CC(=O)NC2C=CCN(C(c3n[nH]cc3C)=O)C2)c(C)c1 21172,C1(NC(C(COC)NC(=O)OC(C)(C)C)=O)C2CC1CN(C(=O)CC(C)C)C2 21173,N1(C(c2ccn(C)n2)=O)CC(CNC(=O)COc2ccccc2)C2CC12 21174,N1(C(C=C(CCC)C)=O)CCC(C)(C(=O)NC(c2cnn(C)c2)CO)C1 21175,CC12CC(NC(C3CCCS3)=O)(C1)C1(CCN(c3ncnc(Cl)c3CO)CC1)O2 21176,c1(C(=O)NCC2C(CC(=O)N(CC#C)C)C2)cnc(N)cn1 21177,N1(C(c2cccc(CC=C)c2)=O)CC(C)C(NC(=O)CNS(=O)(=O)NC)C(C)C1 21178,CCC(C)(CCCNC(C)CCC1CCC1)C1OCCO1 21179,C1(CC(=O)NCC(C2CCC2)NC(c2ccc[nH]2)=O)CC2(CCCC2)CO1 21180,N1(C(CCC)C(=O)NC(C)C(=O)OC(C)(C)C)CC(C)CCC12CC2 21181,C(=O)(C1CCCc2nnn(C)c21)NC(CNC(CCCCC)=O)CC(F)(F)F 21182,CCCCC(O)C(=O)N1CCC(CCNC(C2(C)CCCN2C)=O)C1 21183,C1(NC(CC(C)(C)c2cccs2)=O)CS(=O)(=O)CC1NC(=O)CCc1ccsc1 21184,C1(CC)CN(S(=O)(=O)CC2CC(C)(C)CO2)CC(C)S1=O 21185,N1(C(C(c2cn(C)nc2)NC(C2OCCCC2(C)C)=O)=O)CCc2ccsc2C1 21186,c1(C(=O)NC2CCN(C(C(CC)NC(N)=O)=O)C2(C)C)ccc2c(n1)CCCN2 21187,C12(C(=O)OC)CC(C1)C(N1CC(c3ccc(SC)cc3)C1)N2 21188,CCCC(CC(C)C)C(=O)NCCC1CN(C(=O)CC2CSC2)CCS1(=O)=O 21189,Cc1ccc2c(c1)CC(NC(c1ccc(F)c(F)c1)c1nnnn1C)C2 21190,C(=O)(CC(C)CC(F)(F)F)N(C1CCN(C(=O)C=C2CCC2)C1)CC#C 21191,N1(C(C2(C)CCCO2)=O)CCOC2CCN(C(=O)Cn3cnc([N+](=O)[O-])c3)CC12 21192,N1(C(c2c(COCC)nn[nH]2)=O)CC2CC1CN2C(C1CC1OC(C)(C)C)=O 21193,C(CC1=CCN(C(c2ccc(F)c(O)c2F)=O)CC1)NC(=O)Cn1cc(Cl)cn1 21194,C1(CC(=O)N(C(C)C(=O)NC2CC(=O)N(CC)C2)CCC)CCC(C)(C)C1 21195,N1(CC(=O)NCc2c(C)ccs2)CC(NC(=O)Cn2cc([N+](=O)[O-])cn2)CCC1C 21196,N1(C(C(CN(C)C)(C)C)=O)CC2(CCC(CNC(=O)CSCc3cscn3)O2)C1 21197,c1(C(N2C(C(C)NC(CCSCCCC)=O)CCC2)=O)cn(C)nc1OC 21198,C(CC(C)(C)C(=O)NCC1CC(F)CN1C(=O)CCCCCSC)SC 21199,c1(CC(=O)NCC(CC=C)NC(C2CC(O)C2(C)C)=O)ccc2cccnc2c1 21200,c1(C(N2CC(C)(NC(C3C(SC)CCC3)=O)C2)=O)nn(C)c(C(F)(F)F)c1Cl 21201,C1(NC(Nc2cccc(C(=O)OC)c2)=S)CCCN(c2ccccc2C)C1=O 21202,C1(NC(C(F)=C(C)C)=O)CN(C(=O)Cc2cccc(OCC(C)C)c2)CC1C 21203,n1(CC)cc(CC(=O)N(C(C)CN(C(=O)Cc2cnc(C)s2)C)C)cn1 21204,C(C)(C)(CC(=O)NC(CCNC(=O)C1CC1)=O)N(C(CCCOC(C)C)=O)C 21205,C(=O)(CC(C)(C)N(C)C(C1CCC=CCC1)=O)N(C)CC1CCCCO1 21206,c1(C(N(CCC(=O)NCCCNC(CC2C(C)C2)=O)C)=O)cnn2c1OCC2 21207,C1(C)(CNC(Cc2nc(CC)sc2)=O)CC(F)(F)CN1C(c1scnc1C)=O 21208,N1(C(CCSC)=O)CCC(C)C(CNC(c2nccc(Cl)c2C)=O)C1 21209,c1(C2(C(=O)NC(CC=C)C3CCC3)CCC2)ccc(F)cn1 21210,C1(OC)CC(CCNC(c2nc(C)sc2C)=O)N(C(C2CCSCC2)=O)C1 21211,C=CC1(NC(C23CC2CCN3C(c2sccc2F)=O)=O)CCCC1 21212,Cc1occc1CC(=O)NC1CCN(C(c2cn(C3CCCC3)nn2)=O)C1 21213,C#Cc1ccc(F)c(C(=O)N(CCCCCNC(C2CCC(C)(C)OC2)=O)C)c1 21214,c1(-c2c(-c3nccn3CCC(O)C(F)(F)F)cnc(C)n2)ccc(S(C)=O)cc1 21215,N1(C(C(C)Cc2ccccc2)=O)CC2CN(C(c3coc(O)n3)=O)CC2C1 21216,c1(C(N(C2CC(NC(c3ccc(Cl)cn3)=O)C2)C)=O)cnc2[nH]c(O)nc2c1 21217,c1(C(=O)NC(C(C)NC(C2CCCN2C=O)=O)CO)ccc(Cl)c(N)c1Cl 21218,c1(OC)ccc(CNC2CN(C(c3nccnc3Br)=O)CC23CC3)c(C#N)c1 21219,C(CCN(C)C)(C(=O)NCc1cn(C)cn1)NC(COCCC)=O 21220,C=CC1CN(C(=O)CC2C(=O)NN=C2C)CC1Nc1nccc(CO)n1 21221,C(C)(CCCC(=O)N1CC(n2cnnc2)C1)NC(c1[nH]cc(C)c1C)=O 21222,C(=O)(C(CC(F)F)NC(c1ccc[n+]([O-])c1)=O)NC(CCC)CCO 21223,CCC(C)C(O)C(C)C(=O)NC1C2CCC(C2)C1C(=O)NC1CCCC1(C)C 21224,C1(CNC(CCN(CCC)C)=O)C2CCCC1N(C(c1cccc(O)c1F)=O)C2 21225,C1(CN(C)C(C2(O)CC(C(=O)OCCOOC(C)(C)C)C2)=O)CC2(C1)CC(F)(F)C2 21226,c1(C(=O)NC2C3(CNC(CSCC=C)=O)CCC(C2)C3)cc2sccc2cn1 21227,c1(C(N2C3CCC(NC(=O)C=Cc4cc[nH]n4)(C3)C2)=O)ccc2[nH]ccc2c1F 21228,c1(C(N2CCCC(C(=O)NC(C)CC#N)C2)=O)ccc(Cl)nc1Cl 21229,C(c1ccc(C(F)(F)F)cc1)=CC(N1C(CNC(CCOCC#C)=O)CCC1)=O 21230,C#CCC(O)C(=O)NC(CCOCC)C(=O)NCCC1CCCCO1 21231,CC1(C)C(C)(NC(=O)C(F)CC2CN(C(=O)C(F)F)C2)C1(C)C 21232,C(C1Cc2ccccc21)NC(CCCCN(C(=O)C(C)(C)n1ccnn1)C)=O 21233,Cc1c(NC(=O)CC2CCN(C(=O)Cc3cccnc3)CC2)cnn1C1CC1 21234,c1(C(N2CCC(COC)(NC(c3cncs3)=O)C2)=O)c(C)oc2nc(Cl)ccc12 21235,C(=O)(CC1=CCCC1)NCC12C(CN(C(c3c(C)nsc3Br)=O)C1)C2 21236,C1(C)(C(=O)NC2CC3(CC(NC(CNC(C)=O)=O)C3)C2)CCc2ccccc2C1 21237,C1(CNC(c2c(C)nc(CO)o2)=O)C2CCC(C2)N1C(=O)CCn1cccn1 21238,C1(C(=O)N(CC(=O)N(C)C)C)(NC(C(CCOC)C)=O)CCC(C)(C)C1 21239,C1(NC(CC(C)OC)=O)CCC(C)N(C(=O)C(CO)c2ccccc2)C1 21240,c1(C(=O)NC2CCN(C(CCc3ccc(C)cc3C)=O)C2)ccc2sncc2c1 21241,C(O)(CC(=O)NCC1(CC2CC2)CC1)(C(F)(F)F)c1ncc(C)o1 21242,c1(-n2cc(C(=O)NC(CN3CCCC3)CO)nn2)cccc(Br)c1 21243,C1(C(N2C(C)(CNC(c3cccc(F)c3N)=O)CCC2)=O)CN(CP(C)(C)=O)C1 21244,N1(C(C2C(C)(C(F)F)C2)=O)CCCCCC(NC(=O)C2=CCCS2)C1 21245,CCCCC(C)CCC(=O)NCCCN(C(=O)CC#N)C1CCCC1 21246,c1(C(C(=O)N(CC(C)NC(CNC(CCCCC)=O)=O)C)=O)cc(F)cc(Cl)c1 21247,Cc1cncc(-c2cccc(C(=O)NC(c3cccc(F)c3)C)c2)n1 21248,N1(CC)CCCCC1C(=O)NCc1nnn(C)c1C(N1CC2(CC2)C1)=O 21249,CC1CN(c2nnc(-c3sccc3CO)n2Cc2ccc(F)cc2)CCS1 21250,CC(C)(O)C(F)C(=O)N1CCOC(CNC(C2CCCCO2)=O)C1 21251,C(=O)(CCOCCCNC(=O)Cc1ccsn1)NCC(=O)N(C)CC 21252,c1(OC)cccc(-c2cc(C(=O)NCC3(NCc4sccc4CO)CC3)on2)c1 21253,c1(C(=O)NCC2CC2C(=O)N(CC(O)CO)CCO)csnc1Cl 21254,C1(NC(=O)NC(C2CCO2)C)CCC(F)(F)CC1(C)C 21255,S(=O)(=O)(c1cnn(C)c1)NCC(=O)N(CCCNC(=O)CC1COCCN1C)C 21256,C1(C(N2C(C3(C(=O)NC4(C)CC(O)C4)CC3)CCC2)=O)CC2C(C1)C2(C)C 21257,CC1(C)OCc2c1n[nH]c2C(=O)NCC1CC(NC(=O)C(F)CC2CC2)C1 21258,c1(C(=O)NC2C(NC(COCCCCC)=O)CCC2)c2ccccc2nn1C 21259,c1(CN(C(=O)CC(C)(C)n2cc(C3CCCOC3)nn2)C)ccc(Cl)nc1 21260,CC(CNC(C1(c2cccnc2)CCC1)=O)(CO)NC(=O)C=CC1CCCC1 21261,c1(-c2nc(CC(C)CCO)on2)c(Cl)cccc1Cl.C1CCCCCN(C)C1=O 21262,C(=O)(C1CCOc2ccccc21)NCC(C1CCCN1C(C12CC(C1)C2)=O)(C)C 21263,C(CC(=O)NC(C)CCCCO)(C(C)C)NC(C1(OCC)CCCC1)=O 21264,c1(C(=O)NC2CN(C(CC3(OC)CCOCC3)=O)C(C)C2)ccnc(Cl)c1O 21265,C1(NC(C2(CNC(=O)CC3CCCC3)CCCO2)=O)CCCCCC1F 21266,c1(C(N2CC(C)OCC2C)=O)nc2ccccn2c1C1=CCOCC1 21267,c1(CNC(CSCC#C)=O)cc(C(=O)NCC2(C#N)CC2)no1 21268,c1(C(N2CCN(C(CCC(=C)Br)=O)CC2C)=O)cc(Cl)cc2nc(C)[nH]c12 21269,N1(C(c2cnn(CC)n2)=O)CC(C2CCCCN(C(=O)CC3CC4(CC4)C3)C2)C1 21270,S(=O)(=O)(c1[nH]c(=NC2CCCC(C(C)(C)C)C2)ccc1Br)NCCCOCC 21271,c1(C(=O)NCC2(CCNC(COC(C)C)=O)CC2)cncc2c(O)nccc12 21272,CCC(CC)CC(F)C(=O)NC(C12CCC(CC1)C2)CNC(=O)C(C)(C)O 21273,N1(C(CSCC)=O)CC2CCCCC2(NC(c2ccc(OC)cc2N)=O)C1 21274,C#CCC(O)C(=O)NC(C)CN(C(=O)C(O)(c1ccccc1)C1CCCCC1)C 21275,N1(C(C(CCCC)C)=O)CCCCCC(NC(=O)CN2CC(C)C2)C1 21276,Cc1cncnc1N1CCC(CNC(=O)C(F)(F)c2nccs2)C1 21277,C1(C(N(C(CC)C2CC2)C)=O)CC(F)CN1C(=O)CC1COCCO1 21278,C1(CNC(c2ccc(OC)nc2)=O)CC(C)CN(C(=O)C(C2CCC(=O)N2)C)C1 21279,NS(=O)(=O)C1(C(=O)NCCC2(O)CCN(C(C3C4COCC34)=O)C2)CCC1 21280,Cc1nc2ccc(C(=O)NCC3C4CN(C(c5csc(C)c5)=O)CC34)cc2s1 21281,N1(C(CN(C)C(c2c[nH]c3nccc-3c2)=O)=O)CCC2(CC1)CC2C#N 21282,O=S(=O)(c1ccc(NNC(=O)C2(CF)CC2)cc1)Nc1ccc(O)cc1C(F)(F)F 21283,C1(CNC(C=CC2(C)COC2)=O)CCCCC1NC(c1cnccc1Cl)=O 21284,C1(O)(CN(C)C(c2sccc2NS(C)(=O)=O)=O)CCN(C(=O)C(CO)OC)CC1 21285,c1(NC(N2CCC(CC(=O)OC)C2)=O)nc2ccccc2n1CC#N 21286,c1(C(=O)OCC)cc(CCNC(=O)Cc2nn[nH]n2)nc(O)c1 21287,Cn1nc(C(F)(F)F)c(Br)c1CN1CCCCC1Cc1ccccc1Cl 21288,C1(NC(=O)CCOCCCNC(c2c[nH]ccc2=O)=O)CC(=O)N(C2CC2)C1 21289,C1(C)(CNC(CCCSC)=O)CCC(NC(C2(F)CCCCCC2)=O)C1 21290,C1(NC(C(C)SCC)=O)CCOC1C(=O)NC1CCCC1C(=O)OC 21291,C1(C(N2C(C(=O)NCC3CCOC3)CC=CC2)=O)CC2(C1)CC2(F)F 21292,C1(NC(=O)CCC2CC2)CCC2(CCN(C(c3csc(Cl)c3Cl)=O)CC2)C1 21293,c1(OC)cccc2scc(C(N3CC4CC(NC(=O)CNC=O)CC3C4)=O)c12 21294,c1(OC)[nH]c(=N)ccc1C(=O)NCC1CC2CN(C(=O)Cc3nnc(C)o3)CC12 21295,C1(C2CCN(C(C3CCC(F)CC3)=O)CC2)(NC(C(CC)C(C)C)=O)CCC1 21296,C1(C(F)(F)F)COC(=O)N1.c1(COCC(=O)NCC)nc(C)no1 21297,c1(N(C)C)ccc(CN2CCC(O)C(C(=O)NC(C)CCO)C2)cc1Cl 21298,C1(CNC(=O)NC)CC(COC)N(C(C2(c3ccccc3)CC2)=O)C1.C(C)(C)(C)O 21299,C1(NC(C2(C)COC2)=O)CN(C(=O)C(C)(C)Cc2ccccc2)CCC1F 21300,CC(C(=O)NCC1CCN1C(c1cncc(C(F)(F)F)n1)=O)C(C)(F)F 21301,c1(C(N2C(CNC(=O)C(F)CC3CCC3)CCCC2)=O)cccc(C#CCO)c1 21302,C1(Nc2c(OC)ncc(-c3ccnn3C(C)(C)C)c2)CCC2(CC1)OCCO2 21303,C1(CNC(C=C(CC)CC)=O)(COC)CCCN1C(C1(CCF)CC1)=O 21304,C1(C)(C(N(CC(C)N(C)C(C2CCN(C)S2(=O)=O)=O)C)=O)CCC(F)(F)CC1 21305,C(=O)(CC(=O)N(CC(C)CNC(c1cocc1C)=O)C)OCC 21306,N1(C(C2(NC(=O)Cn3ncnn3)CCOCC2)=O)CCN(C)CC(O)C1 21307,N1(C(C(C)(C)C(F)F)=O)CCCC(O)(CNC(C23CCC(C)(CO2)C3)=O)CC1 21308,c1(C(N2CCCCC2C(=O)NCC(F)(F)F)C(=O)NC)cc2cccnc2s1 21309,c1(NC(c2ccccc2)CCC)nccc(NCCC2(COC)CC2)n1 21310,O=C(CCCc1ccncc1)NC1CC(NC(c2cc(Br)c[nH]2)=O)C1 21311,c1(C(N2CC(C)N(C(C3CCCC34CC4)=O)CC2)=O)cc2c(cn1)CCCC2 21312,c1(CNC(C2CCCN(C3CCC3)C2)C)ccc(I)c(F)c1 21313,C1(CC)CN(C(=O)C(C2CCOCC2)O)CCC1NC(=O)C(O)C(C)(C)C 21314,C(=O)(CC(C)(C)CC(F)(F)F)N1CCCC(N(C(c2cc(C)no2)=O)CCO)C1 21315,C1(NC(CCCc2cc(C)no2)=O)CCN(C(=O)C(C)SC(F)(F)F)CC1O 21316,C(=O)(C1CCCc2ccnn21)N(CCNC(c1nc2nccc(C)n2n1)=O)CC 21317,c1(C(=O)NCC2CCN(C(C=C(C)C(F)F)=O)CC2)ccc2c(C)nn(C)c2n1 21318,c1(-c2cc(NC(C3C(C)OCC3)=O)ncc2)ccc(S(=O)(=O)N2CCCC2)cc1 21319,C1(NC(c2n(C=C)nnc2)=O)CN(C(=O)C2=COCCO2)C(C)(COC)C1 21320,Nc1ccc2c(C(N3CCCC3CNC(c3nccnc3Cl)=O)=O)c[nH]c2c1 21321,C1(C(N(C)CC2CCC(F)(F)C2)=O)CCCN(C(=O)Nc2ccc(Cl)cc2)C1 21322,Cn1[nH]c(=NC(=O)C2CCCN2C(C2(C(F)(F)F)CCC2)=O)cc1Cl 21323,C1(C(N2CC(C)C(F)C2)=O)N(C(c2cc(C(N)=O)c[nH]2)=O)CC12CCCC2 21324,N1(C(c2c(C)nc(CC)o2)=O)CCOC(C)(CNC(=O)CCOC2CC2)C1 21325,N1(C(Cc2c(C)n[nH]c2)=O)CC2CC(NC(c3nnn(C)c3N)=O)C(C2)C1 21326,N1(C(=O)NCC(c2ncn(C)n2)C)CC(S(=O)(=O)N(C)C)C1 21327,C(=O)(CCC(N)=O)NC(C1CCN(C(C(C)NC(C2CCC2)=O)=O)C1)(C)C 21328,C(C)(c1cccc(C(F)(F)F)c1)=CC(=O)NC(CCC)(C)C 21329,C1(c2c(OC)cc(Br)c(F)c2)NC(=O)N(CCC2CC2)C2=C1C(=O)NC(C)C2 21330,C(=O)(CCc1ncc[nH]1)NC1C(NC(CNC(=O)NC)=O)C1 21331,C1(CC=C)CCCN(C(=O)N(CCN(C)C)CC2CCCCC2)C1 21332,C1(NC(CC2ON=C(C)C2)=O)CC2(CCCC2)C1.Cc1nc(C)c(C=O)o1 21333,C1(C2CN(C(=O)C(Cc3ccccc3)n3cnnn3)C2)(NC(C2C(C)C2)=O)CC1 21334,c1(C(CC)C)cc(C(=O)NCc2ncc(-c3cccs3)[nH]2)on1 21335,N1(C(CCCOC)=O)CCc2nc(C3=CCSCC3)sc2C1 21336,c1(C(=O)NC(C)CCNC(=O)C=CC2CCCC2)cnc2ncnn2c1O 21337,N1(C(C#CC(=O)N(C)C)=O)CCN(C(=O)CC2C=CS(=O)(=O)C2)CC1CC(F)F 21338,CCC(C(=O)N1CC(OCC(N)=O)C1)NC(c1cc(CO)[nH]n1)=O 21339,C1(NC(CC(CCC)C)=O)CCC2CN(C(=O)CCC(C)=O)CCC2C1 21340,n1(CC=C)nnnc1C(C1CCC1C(=O)OC(C)(C)C)NCC12CC(CO1)C2 21341,CC(C)(C)C(C#N)C(=O)NCCC1(C)CCN(C(C2CC3(CCC3)C2)=O)C1 21342,c1(CC(=O)OCC)cnn(CC2CC(C(=O)OC)C2)c1 21343,N1(C(C(C)OC)=O)CCC2CN(C(=O)CN3CCP(C)(=O)CC3)C2C1 21344,CCC(C)(C)CC(=O)NC1CCCC(NC(=O)CSCc2ccc(F)cc2)CC1 21345,N1(C(CCc2cc(C)no2)=O)CC(NC(=O)CSS(C)(=O)=O)C(O)C1 21346,C1(F)(CNC(c2c(C)snn2)=O)CCN(C(c2cc(C(C)(C)C)[nH]c2C)=O)C1 21347,Cn1nc(C2CC2)cc1C(C1(C(C)(F)F)CC1)=O 21348,c1(OC)cccc(F)c1C1CCCN1CC(=O)Nc1ccnc(Cl)n1 21349,CC(C)CCCCC(=O)N1CC(C(=O)NCC2CC23CC3)CCC1(C)C 21350,Cc1cc(C(CO)NC(=O)CN(C)C(C2CC=CCC2)=O)no1 21351,CN1CCN(C)C(C(N2CCOCC2C(=O)NC2CCCC2O)=O)C1 21352,n1(C(C)C(C)(C)C)nc(-c2cccc(Cl)c2)nc1C1CC2CC2C1 21353,C=C=CC(C)C(=O)N1CC2C(NC(=O)CC3CCN(C)CC3)C2C1 21354,Cc1csc2ccc(C(N3CCCC3(C)CNC(c3nn(C)cc3C)=O)=O)cc12 21355,N1(C(c2cnn3c2OCC3)=O)CC2CCC(C1)N2C(c1cnc2n1CCC2)=O 21356,C12(CCNC(C3CC(SC)C3)=O)CCC(CC1)N(C(c1cncn(C)c1=O)=O)C2 21357,C(=O)(NNc1ccc(C(=O)C(F)(F)F)cn1)NC(=O)Cc1[nH]nc([N+](=O)[O-])c1Cl 21358,c1(N2CCC(C)(CC)C2)ccc(S(=O)(=O)NCC(c2ncccc2F)(C)C)cn1 21359,CCC(C)(C)C(O)C(=O)N1CC(NC(=O)CSc2ccc(F)c(F)c2)C(C)C1 21360,c1(CC(=O)NCCNC(c2cc(F)cc(N)c2F)=O)ccc(S(=O)C2CC2)cc1 21361,Cc1ccc(C)c(C(N2CC(CNC(=O)CC=CC(C)(C)C)C(O)C2)=O)c1 21362,C1(OCCC)CCN(C(=O)CC2CC(C)N(C(c3cccc(CO)c3)=O)C2)CC1 21363,c1(C(C)(C)O)cc(C(=O)NC2CC(CNC(C3(C)C=CCCC3)=O)C2)ccn1 21364,C1(NC(c2c[nH]nc2-c2ccco2)=O)CCN(C(=O)COC2CCCOC2)CC1 21365,c1(CNC(NC(COC)C(C)C=C(C)C)=NCCCF)cc2c(cc1Cl)OCCO2 21366,C1(NC(CCC=CC)=O)CCCN(C(c2cn(C3COC3)nn2)=O)C1C 21367,c1(CN=C(NC(CC)CC)NC(C)C(C)COC)cc(O)cc(Br)c1 21368,c1(CC(=O)NCC2CC(NC(c3ccsn3)=O)C2)ccc(OC(F)F)cc1 21369,C1(CN(C(C)C(C)(C)NC(C2CCCC2)=O)C(CNC(CC)=O)=O)CCCN1N=O 21370,C12C3CCN(C3C1(C)C)C(=O)C(=O)O2.c1(C)n[nH]c2c1NCCC2.CN(C)C(=O)O 21371,c1(C(N2CC3C(CNCc4c(OCC)nccc4)(C3)C2)=O)ccc(F)cc1C#N 21372,C(CCC(C)(C)C(=O)NC(c1nccn1C)CC)NC(C(CCCC)C)=O 21373,C1(C(=O)NCCOCCCN(C)C(C2SCCS2)=O)CCC1C(F)F 21374,c1(NC(c2ccc(-n3ncc(C)c3)cc2)=O)ccc(Cl)c(Br)c1Cl 21375,N1(C(CSC(C)C)=O)C2CCC1CN(C(=O)C(C)SCc1ccccn1)C2 21376,C1(NC(=O)NC2CCN(c3ncc(C(=O)OC)s3)CC2)CCC(=O)C(C)C1 21377,N#CC1CCN(C(=O)CC2(NC(=O)CC3CCOC3)CC2)C1 21378,c1(C(N2CCC(NC(CCCN(C)C)=O)(CO)CC2)=O)ccc2nonc2c1 21379,CC1CC(NC(c2ccoc2Cl)=O)CN1C(c1c[nH]c(-c2ccccc2)c1)=O 21380,O(N1C(=O)c2ccccc2C1=O)CC(=O)NC(C)CNC(C1(F)CCCCC1)=O 21381,c1(CC)nc(CC(=O)N(C(C)CNC(C2CC2(C)C)=O)C)cs1 21382,N1(C(C2N(N=O)CCC2)=O)CC(NC(=O)C(F)(F)C(F)(F)F)CC2(CC2)C1 21383,N1(C(C(C(C)C)SC)=O)CCC(C=CC(=O)NCCC(C)C(F)F)CC1 21384,c1(OC)cc(C(N2CCC(C)C(CNC(=O)Cn3cc(C)cn3)C2)=O)c(Cl)cn1 21385,C1(NC(C(C=CCCC)O)=O)CC2(C1)CC(NC(C1CCC(C(C)C)CC1)=O)C2 21386,C1(NC(Cc2cccc(OC)c2)=O)CCCN(C(=O)CS(C)(=O)=O)CC1 21387,N1(C(C(=O)N(CCOCC2CC2)C2CC2)CC2CCCC2)CCCC(F)CC1 21388,C(=O)(C(C)(F)C(C)(C)F)NC(CNc1c(F)ccc(C(C)=O)c1)C 21389,CC1=CC(NC(=O)CCC2CC(NC(=O)Cc3ccns3)C2)CCC1 21390,N1(C(c2ccc(OCCC)cc2)=O)CCOCC(NC(=O)CC2CCC(=O)O2)C1 21391,C1(N(C(C2(CC=C)CC=CC2)=O)C)CCCN(C(=O)Cc2nccc(OC)n2)C1 21392,CC(CCNC(C1(S(C)(=O)=O)CC1)=O)CCNC(=O)CSC1CC1 21393,c1(C(N2CCC3CN(C(C(CC=C)CC=C)=O)CC32)=O)cccc2oc(O)nc12 21394,c1(OC)cc(OC)cc(C(N2CC3(NC(=O)CC4CSC4)CC2C3)=O)c1 21395,C(C(C(=O)NC1CCC(=O)NC1=O)C(C)C)NC(c1c(OC)n(C)nc1)=O 21396,c1(N2CCC(=C)C2)ccc(S(=O)(=O)NCCN2CC3CC3C2)cc1Cl 21397,c1(C(N2CCC(c3ccccc3F)C2)C(=O)NCCC2CC2)noc2c1CCC2 21398,N1(C(CC=CC)=O)CC(NC(=O)C(F)n2cccn2)CC(C)(C)C1 21399,c1(C(=O)NCCCNC(C(C(CC)(C)C)OC)=O)c(C)cnc2ccccc12 21400,N1(C(c2c(C)cn(C)c2)=O)Cc2[nH]nc(C(N3CC(F)(CF)C3)=O)c2C1 21401,C(=O)(CCCC(=O)NOC(C)(C)C)NCC(CC)NC(CC=CC)=O 21402,C1(NC(c2cnnn2C2CC2)=O)CC2CC(C1)N(C(C1SC3C=CC1CC3)=O)C2 21403,c1(C(N(CC2N(C(c3cn(CCC=C)nn3)=O)CCC2)CC)=O)cc(Cl)cn1C 21404,N1(CCCC(C)(F)F)CCC2C(O)CC2C1 21405,N1(C(=O)CCF)CCCC2CN(C(=O)CC34CCC(CC3)C4)CCCC12 21406,C(C(F)(C(=O)N1CCCCC1C(C)C)C(C)C)NC(c1nc(CC)oc1)=O 21407,N1(c2cc(NC(c3nc(C)cs3)CC)nc(C)n2)CCC(CC#N)C(F)(F)CC1 21408,N1(C(C2(C)COC2)=O)CC2(CCCCN2C(=O)CN2CCNC2=O)C1 21409,c1(OC)cnccc1C(=O)NC1CCCCC1NC(=O)COCCSC 21410,C1(NC(Cc2cnc(C)s2)=O)CN(C(C2CC3CCC2O3)=O)CC1C 21411,C12(C(=O)NC3CCC(CNC(c4c[nH]nc4F)=O)CC3)CCC(CF)(CC1)CC2 21412,N1(C(c2ccn(CC)n2)=O)CCN(C(c2cc(CCOC(C)C)on2)=O)CC1 21413,c1(N2CCC(S(=O)(=O)NCC3(OC)CCC3)C2)nc(N2CCC2)nc2cc[nH]c12 21414,C=CCC(CNC(=O)CC(CC)C1CCC1)C(=O)NCc1cnc(C)cn1 21415,c1(C(=O)NC2C(C)N(C(c3cnn(C)c3Br)=O)CCC2)nccc2cccnc12 21416,C1(NC(c2c(OC(C)C)nccc2)=O)CN(C(C2CCC3CC23)=O)CC2(CC2)C1 21417,C1(NC(C(CSC)(C)C)=O)CN(C(C2CN(C(N)=O)C2)=O)CC2CC12 21418,O(NC(=O)C(CC#CC)CC)CCCC#C.C(c1ccncc1)=CC(=O)OCC 21419,c1(C(=O)NCC(CC)NC(c2cccc(N)c2C)=O)cccc2[nH]cc(Cl)c12 21420,c1(OC)c(F)ccc(C(N2CCC(C)(NC(=O)C(C)OC(C)(C)C)C2)=O)c1F 21421,c1(C(C)C)noc(CCC(=O)N2CCC2CNC(=O)C(F)(F)c2nccs2)n1 21422,c1(C(N2C(C)C(C(=O)NCC3CC3CO)CCC2)=O)cnc2cc[nH]c2c1 21423,N1(C(C(=Cc2cnc[nH]2)C)=O)CCN(C)C(CNC(=O)CC2CCC(=O)N2)C1 21424,c1(CNC(C2(c3n(C)ncc3)CCOC2)c2nnnn2C)cc2ncccc2o1 21425,C(=O)(C(CCOC)NC(C1CCN(C)C1C)=O)N1CC(N(CC)CC)C1 21426,c1(C(=O)NC(C2CCN(C(c3cc(C)sn3)=O)C2)C)cccc(=O)n1O 21427,c1(C(C)NC(=O)NCC(=O)NCC2CCOC2)ccncc1F 21428,C(=O)(C1CCCc2cncn21)NC(C)CCNC(=O)C(c1cc(F)cc(F)c1)O 21429,C1(C(=O)NC2(CO)CN(C(C=CC(=O)OCC)=O)C2)CC(O)CN1C(N)=O 21430,c1(CN(C(=O)CNc2ccccc2Br)C)cccc(OC(F)(F)C(F)F)c1 21431,C1(COC(C)C(=O)NC2(CCNC(c3cc(C(F)F)cs3)=O)CC2)CCCCO1 21432,C1(NC(=O)CC2CCS(=O)(=O)CC2)CCC2CCN(C(C3CC4CC4C3)=O)C12 21433,C(C)(C)(CCC(=O)N1CCC(c2cn(CC(O)COC)nn2)C12CC2)OC 21434,C1(C(=O)NC2C(NC(=O)CCF)C2)COc2ccccc2C1 21435,C1(O)(CN(C(=O)CCS(C)=O)C)CCN(C(C2(C#N)CC23CCC3)=O)CC1 21436,N=c1cc[nH]cc1CN1CCC(NS(C)(=O)=O)C1.N12CCN(CC1)CC2=O 21437,C1(C)(CNC(CC)=O)CN(C(C23CCCC2CCC3)=O)CC1C 21438,c1(C(N2C3CN(C(C4C(C(=O)OC)C4)=O)C(C3)C2)=O)cccc2[nH]nc(O)c12 21439,N(C1CCCc2sc(Cl)cc21)C(N(CC)Cc1cncn1C)=O 21440,c1(N(C)CC2CCCC(O)C2)cccc2c(Br)cncc12 21441,C1(NC(=O)C(F)=CC2CC2)CN(C(C2CC=CCC2)=O)Cc2ccnn2C1 21442,c1(C(N(CC(C)NC(C(C)(C2CC2)OC)=O)C)=O)cccc2nc(O)oc12 21443,C1(CCCNC(C=CC=CCC)=O)CCCN1C(c1cc(C)c[nH]1)=O 21444,C1(C(=O)NCC2CN(C(C3CN(C(=O)NC)C3)=O)C2)CC(C)(C)O1 21445,C(=O)(C#CC1(C)CCCO1)NCCOC1CCN(C(C(C2CCOCC2)C)=O)C1 21446,C1(NC(CN2CCC(C)CC2)=O)CC2CC1CC2C(=O)NCCCc1cccs1 21447,C1(C)(C(=O)NC(C=C)C2CC2)CCN(C(=O)COC2(C)CCC2)C1 21448,N1(C(CS(=O)(=O)NCC)=O)CCN(C(c2scc(C)c2C)=O)CC1CC 21449,Cc1cc(Cl)ccc1NC(C1C(O)CCN1C(c1cnn(C)c1Cl)=O)=O 21450,N1(C(CN(C(=O)NC)C)=O)CC(CO)(CF)C1.C12(CCCC1)C(=O)N2 21451,c1(C(N2CCP(C)(=O)CC2)C)n[nH]c2ccccc12.C12CN(C1)C(=O)NCCO2 21452,c1(OC)cccc(S(=O)(=O)NNC(=O)c2nccc(C)c2Br)c1 21453,C1(C(=O)NC2(C)CCCCC2)CCC2(CCN(C(C3CCNC(=O)C3)=O)CC2)O1 21454,N1(C(COCCC(C)C)=O)CCC2CN(C(C34CCCC3C4(F)F)=O)CC2CC1 21455,c1(C(=O)NCC2OCCN(C(C3CC(C#N)(O)C3)=O)C2)ccnc2[nH]nnc12 21456,CC1(C)NC(=O)CC1C(=O)NC12CC(C1)N(C(=O)Cn1cc(C3CC3)nn1)C2 21457,c1(OC)ccc2c(c1)OCC(CN1CCCC(C)(C#N)C1)=C2 21458,C12(C(=O)NC3CCN(C(C)=O)C3c3ccccc3)C3C4C1C1C2C3C41C#N 21459,C1(C(=O)NCC(CC(=O)NC)C)CCN(C(c2occc2C(C)C)=O)CCO1 21460,C(=O)(C#CC1(C)CCCO1)NCC(C)CNC(c1ccccc1C1CC1)=O 21461,C1(F)(C(=O)NC2CC(CCNC(C=CC(C)C)=O)C2)CCCOC1 21462,N1(c2nnc(CCC)s2)CCC2(CCCCC2NC(=O)CCC2CCOC2)C1 21463,CCC1=C(C(=O)NC2(CNC(c3ccc(NC(N)=O)cc3)=O)CCC2)SCCO1 21464,C=CCC(C(=O)OC)(C(C)C)NC(C1CCC(C)CC1)=O 21465,c1(C(=O)NC(CC(C)NC(c2ncoc2C2CCC2)=O)C)ccc(F)c(Cl)c1F 21466,N1(C(CCC(=O)NC)=O)CC(C)C(C)(CNC(=O)C(c2ccccc2)N(C)C)C1 21467,C(C(C)(C)CCNC(=O)C(C1CCCN(C(c2cnc(=N)[nH]c2)=O)C1)C)OC 21468,c1(C(N2CC(F)(C(N3CCC(CO)C(O)C3)=O)C2)=O)cnn2ccccc12 21469,N1(C(CCSc2nnc(CN(CCNC(C)=O)CC)o2)=O)CCNC(=O)C1 21470,Brc1c[nH]c2c(-c3nc(CC4CC4)nn3CCc3ccncc3)cnn12 21471,C1(CNC(C(CC)(C)COC)=O)CCC2(CN(C(c3cc(F)cc(Cl)c3)=O)C2)O1 21472,C1(NC(C2C(=C)CC2)=O)CCN(c2cc(C)nc(CC3CC3)n2)CC1O 21473,C1(C(=O)NC2CC(CCC=O)C2)CC(=O)CC(=O)N1.C1(CCC)COCCN1 21474,C1(NC(C(=Cc2cccnc2)C)=O)C2CCC1CN(C(c1ccns1)=O)C2 21475,O=C(C1=COCCO1)NC1CC(NC(C2C3CC4C(C3)C24)=O)C1 21476,Cn1ncc(Cl)c1-c1cc(C(N2CC(c3cn(CC4COC(=O)C4)nn3)C2)=O)on1 21477,C(=O)(C1CCCc2nn[nH]c21)NCC(CNC(=O)COC1CCCOC1)O 21478,C1(C(=O)OCc2ccc(C(=O)OCC)o2)C(Cl)(Cl)C12CC2 21479,C1(C2CC2)(CNC(C(c2cccc(C)c2)C)=O)CCN(C(=O)CCN2CCC2)C1 21480,N1(C(CCC2CCN(C(C3(Cl)C(C(C)=O)C3)=O)C2)=O)CCC(C2CCC2)C1 21481,c1(CC)cc(NC2CN(C(=O)CC(C)c3ccncc3)CC2(C)C)nc(CC)n1 21482,Cc1cccc2c1CCCN2C(=O)NCC1COC(C)(C)OC1 21483,c1(CC(=O)N(C(C(=O)N(CC(O)CF)CC)C)C2CC2)ccc(C)nc1 21484,c1(C(=O)NC)ccc(C(N2CC3C(CNC(c4nn[nH]c4C(C)C)=O)C3C2)=O)cn1 21485,C1(CC(=O)N(C2CCCN(C(c3nc(OC)c(C)s3)=O)C2)C)CC2CCC1CC2 21486,c1(C(=O)NCCCNC(CC(C(CC)C)O)=O)c[nH]c2cccnc2c1=O 21487,N1(C(CC(=O)N(C)C)=O)CCCC2C(NC(c3[nH]nnc3C3CC3)=O)C(C)(C)C12 21488,N#Cc1ccc2c(c1)C(=Cc1cnc(CO)cn1)CC2 21489,C=CCC(O)(CC=C)C(C)NC(C1(C)CNC(=O)N1)=O 21490,C(=O)(C1=NOCC1)N1CC(C(=O)NOC(C)CC)(CC)C1 21491,C(=O)(CCCCCN1CCOCC1)NC(c1cn(CCO)nn1)CCC 21492,C1(C(C)NC(C23CCC2C3)=O)CCN(C(=O)C(F)(F)C2CC2)CC1 21493,N1(C(C2(OC)CC2)=O)CC=CC(NC(c2c[nH]nc2C2CC2)=O)C1 21494,CC(C)C(CNC(C1CC2CC(=O)C1O2)=O)C(=O)N(C(C(N)=O)C1CC1)C 21495,C1(O)(CNC(C(CNC(C=C=C(C)C)=O)OC)=O)CC2C=CC1C2 21496,c1(C(=O)NC23CC2CN(C(c2csc(CC(F)(F)F)n2)=O)C3)coc2c1COC2 21497,C1(C)(C(=O)NC(C2CCCO2)CC)CN(C(=O)CCCCNC(C)=O)C(C)(C)C1 21498,N1(C(C(CC)F)=O)CCN(C(C2(C)CCC(=O)C2)=O)CCC1C 21499,C=CCCC(F)(F)C(=O)NC(CO)CCCCNC(c1cnsn1)=O 21500,c1(C(C(=O)NCCCN(C(CC2(C=C)CC2)=O)CC)(C)OC)ccccc1F 21501,CCCCCCC(C)C(=O)N1CCCC1CNC(=O)CCC1CC1(Cl)Cl 21502,c1(C(=O)NCC(CN(C(Cc2c(C)non2)=O)C)O)ncc[nH]c1=O 21503,c1(CCC(=O)NCCC(=C)CNC(=O)C(=CC2CCCC2)C)cccc(OC)c1 21504,C1(CNC(CC(CC)OC)=O)CN(C(=O)CCc2nc(C)no2)CCC1(F)F 21505,N1(C(c2ccc(CN(CC)CC)o2)=O)CC(CCNC(c2ccsc2)=O)C(C)C1 21506,c1(NCc2nccc(C)c2)ccc2ncc(Br)cc2c1 21507,c1(C(=O)NC(CNC(C2CCC3CC23)=O)CO)cc2c(c([N+](=O)[O-])c1)OCO2 21508,n1(CC)nc(C)c2cc(C(=O)NCC(C)(CO)NC(C3CC4CCC4C3)=O)sc12 21509,N1(CC)CC(NCc2cnc(Cl)c(F)c2)CC(C)C1 21510,N#Cc1ccnc(N2CCCC(C(N3C4CCC3C(N)C4)=O)CC2)c1 21511,C1(COC)CN(C(=O)C=Cc2cccs2)CCN1C(=O)CC(C)(C)F 21512,C=CCC(C)(C)CC(=O)NCCNC(=O)C(c1ccc(OC)cc1)NC(C)=O 21513,C1(CCNC(C2C(C(=O)OC)CCC2)=O)CCN(C(c2nc(O)c(C)s2)=O)CC1 21514,C1(C2CCN(C(=O)CCCCC(F)F)C2)(NC(=O)CCn2cccnc2=O)CC1 21515,N1(C(COCCCOC)=O)CCC2(CC1)CCN(C(C1CCCC1OC)=O)C2 21516,c1(CC(C(=O)NCC(CNC(Cc2nc(C)[nH]n2)=O)CO)C)ccccc1F 21517,c1(C(=O)NC2C(C)(C)N(C(C3CN4CCN3CC4)=O)CC2)cnc2nccn2c1 21518,CC1C(C)N(C(=O)C2=CCOC2)CCN1C(=O)CCCCN1C(=O)CCC1=O 21519,c1(CC(=O)NCC2(O)CN(C(c3oc(C)c(CO)c3)=O)C2)cccc([N+](=O)[O-])c1 21520,CC(C)C(C(=O)NCC(n1cc(-c2cccc(C(F)(F)F)c2)nn1)C)C(C)C 21521,S(=O)(=O)(c1ccc(Cl)nc1C)NCC1CCN(C(CCCC)=O)CC1 21522,N1(C(CCOC2CN(C(c3snc(C)c3N)=O)C2)=O)CC2CC(C)(C)C2C1 21523,C(C(CC(C)C)C(=O)NCCc1c(C)noc1C)NC(C=CCN(CC)CC)=O 21524,c1(OC)ccc(C(=O)NCC(CNC(=O)CCc2cccnc2F)CO)c(C)c1 21525,CC1(C)COCCC1CNC(C1CCCN1Cc1ccccn1)=O 21526,c1(C(=O)NC)ccc(F)c(-c2ccc(NC(C3CCC(O)CC3)=O)c(OC)n2)c1 21527,C1(CC=C)(NC(=O)CCc2ccc(C)s2)CCN(C(C2CCO2)=O)C1 21528,c1(C(N2C(CN(C)C(c3ccon3)=O)COCC2)=O)noc2c1CCCCC2 21529,C1(CC(=O)NCC(C(C)(C)C)NC(c2ccn(C(F)F)n2)=O)Cc2ccccc2O1 21530,Cc1scnc1C(=O)NCC(C)CN(C(=O)CCNC(C1CCC1)=O)C 21531,C=C(Br)CC(=O)N(C)CC1CCN(C(C2CCCC2c2nc(S)n[nH]2)=O)C1 21532,N1(C(=O)Cc2cncc(F)c2)CC2CC(C1)N(C(=O)COc1cccnc1)C2 21533,OC1(CNCc2ccc(-c3nnco3)nc2)CC(O)C12CCC2 21534,Cc1cc(C(=O)NC2CC2CNC(=O)CSC2CCOC2=O)c2ccccc2n1 21535,CCC(CC(=O)NCCCOCCC(=O)NC1C(CO)CC1O)C(C)C 21536,CC1=CC(NC(=O)COC(C)(C)CNC(C2(C)CCCC2)=O)CCC1 21537,CN1CCN(C(C2COCC2NC(=O)C=Cc2cocn2)=O)CC1=O 21538,c1(C(N2CCN(C(C3(C(=O)NC)CCC3)=O)CC2)=O)cncc(Br)c1C 21539,N1(Cc2ccc(OC)c(OCc3ccc(Cl)cc3)c2)CCn2ncc(Cl)c21 21540,C(CCC(=O)NC(c1ccccc1)CNC(=O)Cc1ncccn1)=CC(C)C 21541,Cc1[nH]c(C)c(C(=O)NC2CCCC2NC(C2CC23CCC3)=O)c1C 21542,CC(C(=O)N1CCOCC1)C(=O)N1CC2C(NC(=O)CC34COC(C)(C3)C4)C2C1 21543,C1(NC(=O)CCc2cscn2)CCOCC1NC(=O)CCC(=O)N1CCCCC1 21544,CC1(C(=O)NC2CC(CNC(=O)CC3CCCC34CC4)C2)CC(C#N)C1 21545,CC1CN(C(c2cnc(CNC(=O)C3=CCCCO3)nc2)=O)CC(C)(C)O1 21546,c1(OCC)nn(C)cc1C(N1CCC(N(c2cc(C(C)C)ncn2)C)CC1)=O 21547,C(CCC(CO)NC(=O)CC1CC(O)C1(C)C)NC(c1nc(COC)oc1)=O 21548,N1(C(Cn2c3cccc(C)c3cc2)=O)CCC2(NC(=O)CCF)CCCCCC12 21549,C(=O)(C1=CCCSC1)NC1CCN(CCCC(=O)NCc2cn(C3CC3)nn2)C1 21550,C1(C(N(C2CCCC2)CC(C)C)=O)COCC1NC(=O)CCc1cnn(C)c1 21551,c1(SCC(=O)NCCC(C)NC(c2cn(C3CC3)nn2)=O)nnnn1C 21552,Nc1cc(C(N2CC(NC(=O)CCNC(c3ccsc3)=O)C2)=O)cc(F)c1 21553,CC(C(=O)NCCN(C)C(c1ccns1)=O)C(F)F 21554,c1(-c2ccc(C(=O)NC(CNC(C=C(CCC)C)=O)C(C)C)[nH]2)ccc(Cl)cc1 21555,N1(Cc2c(C)ccnc2)CCC2(CCN(C(C3CC3c3ccc(F)cc3)=O)C2)C1 21556,N1(C(c2cccc(CNC(C(C)(C3(C)CC3)OC)=O)n2)=O)CCOCCC1C 21557,c1(C(N2CCC(NC(CCS(C)=O)=O)(CO)CC2)=O)ccc2c(c1)CC(=O)N2 21558,C1(CC)CCC(NC)C1.C12(CCNC(=O)C(=O)NC)CCCC1C2 21559,CCC1=C(C(=O)N2CCC(CCNC(c3cnsc3)=O)C2)SCCO1 21560,N1(C(CN(C(=O)OC)C)=O)CCCC(NC(=O)CCC2CC(C)C2)CC1 21561,CC1C2CCC(C2)C1C(N1CCCC(C)(C(=O)NC2CC23CC(O)C3)C1)=O 21562,C1(CCNC(C(C)NC(CC)=O)=O)CCN(C(c2cn(C)cn2)=O)C1 21563,C(C(CC(F)(F)F)NC(C1(C)CC1(Cl)Cl)=O)NC(c1c(CC)oc(C)c1)=O 21564,O(NC(=O)CCC1CCC(CC2(C)CC2)C1)C(CNC(=O)CC1CCNC1=O)=O 21565,Cn1ncc2cc(C(N3CC(NC(=O)CC4CCCOC4)C(F)C3)=O)cnc12 21566,N1(C(c2ccn(CC)n2)=O)CCC2CCCC12C(=O)N(C1CCCC(C)(C)C1)C 21567,C12CCN(CCC1(F)F)CC(=O)NC2.C1(F)(C(N2C(C)CCC2)=O)CCOCC1 21568,N1(C(CC(CCC)(C)O)=O)CCOC2(CCN(c3cc(OC)ncn3)CC2)C1 21569,c1(C(=O)NC(CNC(c2cc(C)no2)=O)CO)ccn2ncc(Br)c2c1 21570,c1(C(=O)NCC23C(CN(C(CC)=O)C2)C3)ccc(S(=O)(=O)CC)cc1 21571,C(C(=O)NCC1CC2(CCC2)CN1C(=O)CC(C)CF)(c1ccccc1)=C(C)C 21572,N1(C(CNC(N)=O)=O)CCC(CNC(=O)C(F)C2CC2)CC1 21573,C(=O)(C(C)(C)CC(=O)NCC(CNC(=O)C(C)(O)C(F)(F)F)OC)OC 21574,c1(C(N2CCN(C(C=COCC)=O)C(CF)C2)=O)ccc2c(c1)CCCC2=O 21575,c1(COC)cccc2cccn12.N12CCCN(CC1)C(=O)NC(C1CC1)C2 21576,c1(N2CCCC(N(C(=O)C(C)(C)C(F)(F)F)C)CC2)nc2ccc(F)cc2s1 21577,c1(-c2nc(CCOC)nn2-c2ccn(C(C)C)n2)c[nH]c2cccnc2c1=O 21578,C1(C(=O)NC2C3CCN(C(=O)Cn4cccn4)C23)C2C3CC4C1C1C2CC3C41 21579,Cc1cc(Oc2ccc(-c3noc(-c4c[nH]cc4Br)n3)nc2)ccc1F 21580,N1(C(C2(CC#C)CC2)=O)CCC2(CC1)CC2NC(=O)Cc1nnc(C)s1 21581,N1(C(C2OCC3CCCC23)=O)CC(O)CC2(CCOCC2)C1 21582,c1(C(=O)NC2CN(C(c3cocn3)=O)C3CC23)ccc(-n2cccn2)cc1Cl 21583,N1(C(Cn2ccc(C)n2)=O)CCCCC(CCC(=O)NCC2COCCN2C)C1 21584,c1(C(=O)NC(CNC(CSC)=O)CC)csc2nc(-c3cccs3)nn12 21585,c1(CC)c[nH]nc1C(=O)N(CC(C)N(C(=O)CCc1cccnc1)C)C 21586,C1(CNC(C2C(C=C)C2)=O)CN(C(=O)CCC(=O)OCC)CC12CC2 21587,C1(C(N2CCCCC(CC)C2)=O)CN(C(C2CCCC(=O)C2)=O)CC12CCC2 21588,N1(C(C(CC)CCOC)=O)CCC2(CC2)CC1C(=O)NCC(C)(O)CO 21589,CC(C)CCN(C(=O)C(C1(O)CCC1)CCNC(=O)OC(C)(C)C)CC(C)C 21590,c1(OC)ncccc1-c1ccc(C2CCN(C(c3cnc[nH]3)=O)CC2)cc1 21591,c1(OC)cc(Cl)c(C(N2CCC(C(C)O)C2)C(=O)Nc2ccccc2Cl)cc1Cl 21592,C1(C)(C(=O)NC(C)CNC(=O)CCN2CCP(C)(=O)CC2)CCC(=O)N(C)C1 21593,C1(CCOC)(NC(C2CC3CC3C2)=O)CCN(C(c2ccnc(C)c2)=O)CC1 21594,NCC(Cc1ccc(F)cc1)C(=O)N1CCC(N)(CO)C1 21595,c1(C(=O)NCC(C2CCCOC2)OCC)cnc2ccccn12 21596,C1(NC(CCC(=O)OCC)=O)CN(C(C2CCCOCC2)=O)CC12CCC2 21597,C1(C(=O)NCCc2scc(C(C)C)n2)CCCC1S(C)(=O)=O 21598,c1(OC)cc(C(=O)NCC2N(C(CC3C(C(N)=O)C3)=O)CCC2)on1 21599,C=Cc1cnn(C)c1C(=O)NCC(C1CCC1)NC(=O)CC1CS(=O)(=O)C1 21600,n1(C2CCC(C)C2)nc(CC2CCOCC2)nc1-c1cn(C)nn1 21601,C(c1ccccc1F)=CC(=O)NC1CC(CCNC(C2CC3(C2)CC3F)=O)C1 21602,c1(CC(=O)N(CCN(C(C2CCC(CO)CC2)=O)CC)CC)sc(C)nc1C 21603,C1(C(=O)NCCCCCOC)CCN(C(=O)C2=C(C)CC2)C1C(C)C 21604,CC1(C(N2CCCC(CNC(=O)COc3ccccc3F)C2)=O)CCC(F)(F)C1 21605,C1(C(=O)NC2(C)CN(C(C3CCCS3)=O)C2)CCCCN1C(N)=O.S(C)(=O)(=O)N 21606,N1(C(CSCCOC)=O)CCOC(c2cn(CCCC3CCOC3)nn2)C1 21607,c1(-c2onc(C3CCCC(=O)O3)n2)cc(F)cc(F)c1 21608,N1(C(c2ccn(CC#N)n2)=O)CCC(CNC(c2cccc(C(F)F)c2)=O)CC1 21609,c1(C(N2C(CC)CN(C(c3cc(Br)cn3C)=O)CC2)=O)ccc2n[nH]cc2c1 21610,C(=O)(CC(C)CC(=O)NC(C(=O)N(C)Cc1cc(C)no1)C(C)C)OC 21611,C1(C(=O)NC(c2cncs2)C)C=CCN1C(C1CCOCC1)=O 21612,CC1=NNC(=O)C1CC(=O)NCC1(CNC(C2(C)CCOCC2)=O)CC1 21613,C(=O)(C(F)(F)CCn1cccn1)NCC(C)CN(C)C(c1cc(=O)cc[nH]1)=O 21614,c1(C(N2CC(CCNC(C=CC(C)C)=O)OCC2)=O)cccc2c1C(C#N)C2 21615,N1(C(C2C(CC(C)C)C2)=O)CCC(O)(CCNc2nnsc2C(F)F)C1 21616,O=C(C1CCCc2scnc21)N1CCCNC1=O 21617,CC1CCN(C(C2C(C(F)F)C2(C)C)=O)CCN1C(=O)CSc1ccccc1Cl 21618,C(=O)(C(C)CC(N)=O)NC(CCCNC(C(C(C)O)N(C)C)=O)(C)C 21619,C1(C(=O)NC2(CC=C)CN(C(=O)Cc3csc(Br)n3)C2)CC=C(C)CC1 21620,C(=O)(C1=CCCC1P(C)(C)=O)N(CCN(C(C(CCCC)CC)=O)C(C)C)C 21621,c1(OC)ccc(Br)cc1C1(C(=O)NC2CCN(C(=O)CCCC#N)C2)CC1 21622,CC1C2CC(C2NC(=O)CNC(c2ccccc2F)=O)N1C(c1ccc(Cl)s1)=O 21623,C(=O)(CS(=O)(=O)CC(F)(F)F)NC(C1CCN(C(c2c(OC)nn(C)c2)=O)C1)C 21624,Nc1cnc(Br)cc1C(c1ccc(Oc2ccncc2)cc1)=O 21625,c1(CC)nc(N2CCCC(CNC(C3CC4(CCC4)CO3)=O)CC2)cc(C#N)n1 21626,C1(CNC(C2CC(CC(C)(C)C)C2)=O)CN(C(C2(F)CC=CC2)=O)CC12CCC2 21627,N(C1c2ccccc2OCC1C)c1ncnc(CC)c1I 21628,C(=O)(C(C)S(C)(=O)=O)N(CCCN(C(c1c(CCC)occ1)=O)C)C 21629,C1(C)(CC)C=C(C(=O)N2CC3CC(NC(c4cccc(=O)n4O)=O)C3C2)C1 21630,CCC(CC(=O)NCc1cn(C2CC2)nn1)N(C(=O)C(O)CN1CCCC1)C 21631,CC1CC(NC(C2CCCN(CCNS(C)(=O)=O)C2)=O)CCS1 21632,N1(C(C(C(=O)OCC)(C)C)=O)Cc2cccc(CNC(C3CC(CF)C3)=O)c2C1 21633,C1(C(=O)NC(C(C)C)(C)C)CC(=O)CN1C(=O)CCc1ccncc1 21634,C1(NC(COCC(C)C)=O)CCC2CN(C(=O)CSC(F)F)CCC2C1 21635,c1(NC(c2c(C)noc2)=O)cccc(CC2(CNC(=O)CP(C)(C)=O)CC2)c1 21636,N1(C(=O)CCc2nnc(COC(F)F)o2)CCCC(CN=[N+]=[N-])C1.N1CC=CC1 21637,c1(NC(N2C(C)CC(CNS(C)(=O)=O)C2)=O)cc(Cl)ccc1OCC(=O)O 21638,c1(CC)ccc(CC(N2CCN(Cc3cc(-c4ccccc4)n[nH]3)CC2)=O)cc1 21639,C1(C(N2CC(C(C)NC(C(C)=C3CC3)=O)OCC2)=O)CCC(C(C)C)NC1=O 21640,Cc1nn(C2CCC2)cc1C(=O)NC(C(C)NC(c1ccc(Cl)[nH]1)=O)C(C)C 21641,O=C1CCCC(C(=O)NCCCNC(c2csc(C3CCCCC3)c2)=O)O1 21642,Cc1cc(C(F)(F)F)nc(N2CCCOC(CNC(=O)CC3(CO)CC3)C2)n1 21643,CC1(C)CC(C(=O)N2CCCC2CCC(=O)NCCC2CCCCC2O)=NO1 21644,N1(C(C(c2cnn(C)c2)NC(C=CCC)=O)=O)CCC(C)(O)C(O)C1 21645,c1(NC(C=C(C)CNC(=O)C(CC)C(C)C)=O)cnn2cccnc12 21646,C1(CNC(CCC=C(C)C)=O)CCC2CN(C(c3[nH]nnc3C)=O)CC12 21647,N#CC12CC(C(=O)NC3CC(CC(N4CCCC4CN4CCSCC4)=O)C3)(C1)C2 21648,c1(C(N2CC(C)C(NC(=O)CCC(C)(C)O)C2)=O)cc([N+](=O)[O-])n[nH]1 21649,Cc1ncc([N+](=O)[O-])cc1C(=O)NCCNC(C1CC(C2CCCC2)C1)=O 21650,N1(C(C2C(CCC)CCC2)=O)CCSCC1CCNC(=O)Cn1nnnc1C 21651,C1(C)(CC)CC(NC(=O)C=CC(C)NC(=O)CNc2ccncc2Cl)CCO1 21652,N1(C(Cc2cn(CC)nn2)=O)CCC(NC(=O)CC(F)F)C1c1ccccc1 21653,n1(CC)nc(C(N2CCC(CCNC(C3(SC)CCC3)=O)C2)=O)ccc1=O 21654,C=CCC(C)(CC)C(=O)N1CC=C(CNC(c2sc(C(C)OC)nc2C)=O)CC1 21655,C1(CS(C)(=O)=O)CCCC1(c1nnnn1CCC1CC1)OCC(F)(F)F.C1CNC1 21656,C1(CCC(=O)N(CC(C)(C)NC(C=C(C)C(C)(C)C)=O)C)CCCCN1C 21657,N1(C(C2(C#C)CC2)=O)CC(CNC(=O)CCCN(C)C(C)C)OC2COCC12 21658,c1(C(=O)NC2CCC(CNC(C3NC(=O)OC3)=O)C2)cccc(Cl)c1Br 21659,n1(C(C)C)cnc2c(N3CCC(C)S(=O)CC3)[nH]c(=NCC3(C)CCC3)nc12 21660,c1(C(N2CCN(C(c3c(OC)nccc3)=O)C(CO)C2)=O)nc(O)nc(O)c1N 21661,c1(OC)ccc(Cl)c(C(=O)NCC2CN(C(c3cnc(C4CC4)s3)=O)C2)c1 21662,N1(C(c2n(CC)ncc2)=O)CC2CCCC1(CNC(c1conc1C1CC1)=O)C2 21663,C(c1ccccc1)=CCC(=O)NC(C)(C)CNC(=O)Cc1csnn1 21664,Cc1cc(C(=O)NCCN(C(=O)CCCN2CCCCC2)C(C)C)ccc1Br 21665,C1(C(=O)NCC2CC(NC(C(n3ccc(C)n3)C)=O)C2)CCOC(C)(C)C1 21666,N1(C(c2ccncc2)=O)CC2CCN(C(c3nc(Cl)c(Cl)s3)=O)C2C1 21667,C1(C(=O)NC(CC)(C)CNC(=O)Cc2cn[nH]c2)CC(C)CCO1 21668,Cc1nc(Br)oc1C(=O)N(C1CCCC(NC(C2(CCF)CC2)=O)C1)C 21669,N1(CC)CC2(CN(C(=O)C(c3ccnn3C)NC(=O)C(O)CN(C)C)C2)C1 21670,c1(OC)cc(C)c(C(=O)NC2CC3(C2)CC3NC(=O)CC2CCCN2C)cc1Cl 21671,C1(C(=O)NCc2ccn(CCC)n2)C=CCCN1C(C1CC=CCC1)=O 21672,Cc1ccnc(C(=O)NCC(F)CNC(c2sccc2-n2ccnn2)=O)c1N 21673,C(=O)(CC1OCCc2ccsc21)N1CCN(C(C(CC=C)N(C)C)=O)C(C)C1 21674,c1(C(=O)NCCCN(C(=O)CC(C)F)C(C)C)cc(=O)n(-c2ccccc2)[nH]1 21675,CCC(C(=O)NCC1CCN(C(c2cnnn2C(C)C)=O)C1)C(C)(C)CC 21676,N1(C(CC(=C)I)=O)CCOCC(NC(C23CC(OC)C2C3)=O)C1 21677,C(=O)(C(C)(F)C(C)(C)F)NCCCOCCN(C(c1cnc(C(C)C)nc1)=O)C 21678,C1(C(=O)NCC2CCCN(C(=O)Cc3ccon3)CC2)Cc2n[nH]cc2C(=O)N1 21679,CCC(CNC(=O)CCS(N)(=O)=O)(CC)C(=O)NCC1CCOC(C)(C)C1 21680,Cc1ccc(C(=O)NC(C)CN(C(=O)CC2COC(=O)N2)C)c2c1CCC2 21681,c1(NC(C2NCCN(C(C(C)O)=O)C2)=O)cc(F)c(Cl)c(Cl)c1 21682,c1(CC(=O)N(C2CCN(C(=O)C#CC3CC3)C2)CC)c(Br)ccc(F)c1F 21683,CCC(CC(F)F)C(=O)NC1CCN(C(=O)CCC2CC2)C1 21684,C=C(C)C(C)(O)C(=O)NC1CC1NC(C1(C(=O)OC)CCC1)=O.C1(=O)NO1 21685,c1(C(=O)NCC2C(C)(C)C(NC(C34CSC(C3)C4)=O)C2)ccc2c(c1)OCCO2 21686,N1(C(CCN(C(C)=O)C)=O)CC2CC(C1)CN(S(=O)(=O)c1ccc(F)cc1)C2 21687,C(CCNC(=O)C(C)CO)(C(=O)NCCCN1CC=CC1)OC 21688,c1(CCN(C(=O)COc2ccccc2)CCO)c[nH]c(=NCc2ccncc2)s1 21689,c1(CNCc2c(OC)nc(C)cc2)[nH]c2ccccc2c1Cl 21690,CCC(C)C(C(=O)N1CCC(C(F)(F)F)C(NC(c2ccnn2C)=O)C1)OC 21691,Cc1ccc(CNC(C2CSCCN2C(C2CC2[N+](=O)[O-])=O)=O)nc1 21692,Cc1csc(=O)n1CC(=O)NC(C1CCCC1)CNC(=O)C(C)N=[N+]=[N-] 21693,C1(C2CCOCC2)(C(=O)NCCN(CCC)C(C23CCCC2(C(N)=O)C3)=O)CC1 21694,c1(C(=O)NC(CC(C)NC(C2CCC(=O)N2)=O)C)ncccc1OC(F)F 21695,c1(OC)cc(F)cc(C(N2CCC(N(C)C(C3CC(CC(F)F)C3)=O)C2)=O)c1N 21696,C1(NC(C=CC(C)(C)SC)=O)CCCN(C(C2CCCCCO2)=O)C1 21697,S(=O)(=O)(c1ccc(C(N2C3CN(C(=O)C(C)(C)C)CC23)=O)cc1)N(C)C 21698,C(CO)(CCCCNC(c1ccc(=O)n(CC(C)O)c1)=O)NC(C(C)OCC)=O 21699,C1(COC(C)=O)CCN(C(=O)OC(C)(C)C)CC1C(c1ccncc1Cl)=O 21700,n1(CC)cc(S(=O)(=O)N2CC3CC2CC3NC(=O)Cc2ccc(Cl)cc2Cl)cn1 21701,n1(CC(N2C(CNC(Cn3c(C)ccc3C)=O)CC2)=O)cnc2c1CCCC2 21702,N1(C(c2c(=N)cc[nH]c2)=O)CCCC(NC(c2ccsc2Br)=O)C(F)C1 21703,c1(C(N2CCN(C3CNC3)CC2)=O)csc2c1CCNC2 21704,CC(CC(F)(F)F)C(=O)NC(CC(=O)N(CC(O)C(C)(C)C)C)C(F)(F)F 21705,c1(C(=O)NCC(CC)(CC)NC(=O)CCC(C)(C)C)ccc(C#N)cn1 21706,c1(C(=O)NCC(CNC(CCc2c(C)nn(C)c2)=O)C)ccc2c(c1)CN(C)C2 21707,C(c1cccc(Cl)c1)=C(C)C(=O)NC1CCC(CCNC(=O)COCC2CC2)C1 21708,C1(NC(=O)Cc2ccc(C(F)F)cc2)CC2CN(C(C3C4COCC34)=O)CC2C1 21709,C1(CNC(C2N(CC)CCC2)=O)C2CCC1CN(C(C1CCC1)=O)C2 21710,c1(CC(=O)OC)ccc(C(=O)NC(C)CC(C)NC(=O)Cc2cccs2)c(C)c1 21711,N1(C(CCC=CC)=O)CCC(F)(CNC(C2CCC3(CCC3)O2)=O)CC1 21712,N1(CCCC(=O)OC)CC(C)C(P(C)(C)=O)C1.c1(OC)ccc(OC)c(C(=O)C)c1 21713,c1(C(C(C)NC(c2ccsc2Br)=O)NC(C=C(C)C)=O)ccccc1 21714,C(=O)(CC(C(=O)OCC)C(C)=O)NCC1CCN(C(C(=O)NCC)=O)C1 21715,S(=O)(=O)(c1cccs1)NCC(=O)NC1CC(F)(CNC(c2ccco2)=O)C1 21716,c1(C(N2CCC(NC(C(C#C)(C)C)=O)C(C)C2)=O)nc2ccccn2n1 21717,c1(C(=O)NCCC2(O)CCN(C(C34CCC(C3)C4)=O)C2)nccc2ccccc12 21718,C1(NC(C(F)=CCC)=O)CC2CC(C1)N(C(C1CC1[N+](=O)[O-])=O)C2 21719,C(=O)(CC(CC1CC1)NC(C1C2CN(C)CC12)=O)NCC(=C)Br 21720,N1(C(C(C)(C)F)=O)CCC2(CNC(=O)CCCc3ccc(Cl)cc3)CCCCC12 21721,c1(C(=O)NC23C(CN(C(C(CC)F)=O)C2)C3)nc(C(F)(F)F)ccc1Br 21722,C(C)(C(C(=O)NC(C)C(=O)OC)NC(c1ncccc1Cl)=O)OC 21723,CN1CC(C)(C)CC1C(N1CC2CC(C1)C2NC(=O)C(C)(C)C#N)=O 21724,Cc1ccc(C(=O)NC2CCN(C(=O)CCc3cnn(C)n3)C(C)C2)c(O)c1 21725,c1(CSCC(=O)NC2C(NC(C(C)C)=O)CCC2)ccc(O)cc1 21726,Cc1c(C(=O)NCC2CCCC(NC(C34CCC(C3)C4)=O)C2)cnc2ccnn12 21727,C1(C(C)NC(=O)C(c2ccn(C)c2)C)CCCN(C(C2CCCC2O)=O)C1 21728,N1(CCNC(C2C=CCN2C(c2cc[nH]c2)=O)=O)C(=O)CNC1=O 21729,N1(C(c2c(OC)cncc2)=O)CCC(CNC(C2CC2C)=O)C(O)C1 21730,c1(NC(N(CCC)CCN2CCCC2C)=O)cc(I)c(F)cc1F 21731,CC1CC(NC(c2ccc(C3CC3)nc2)=O)CN(C(c2cnc(S)n2C)=O)C1 21732,CCC(CC)C(C)C(=O)NC(C1(CNC(=O)CC2=CCOCC2)CC1)C 21733,c1(C(C)C)ccc(C(N2CCC(CF)(NC(=O)CC3CCCC3(F)F)C2)=O)cc1 21734,Cc1nc(CC(C)C)sc1C(=O)NCC1CN(C(C2OC(C)CC2C)=O)CCO1 21735,CC(C(O)C(=O)NC1CC(CCNC(=O)Cn2cnnn2)C1)c1ccccc1F 21736,CC1CC(NC(C2CCC2)=O)CCN1C(=O)C(=C1CCCCC1)F 21737,Cc1cc(C)n(-c2ccc(-c3nc(-c4ccc(OC(F)F)nc4)n(C)n3)nc2)n1 21738,C12(CNC(=O)CN3CCNC3=O)CCC1CCN2C(c1ccccc1Cl)=O 21739,C(C)(CCCC(=O)OC)(c1n(CCSCC)nnn1)N.c1(C)ccc(OC)c(C)c1.OC 21740,N1(C(C2=CCC(NC(c3nc(C(C)C)oc3)=O)C2)=O)CCCC(C)(C#N)C1 21741,C(C(C)CN=c1[nH]c(=NC(C)c2cnn(C)c2)[nH]c2ccsc12)OC 21742,N1(C(CCCCOC)=O)CCCC(C)C1CCNC(=O)C=CC1CCOCC1 21743,c1(C(=O)OCC)cc2cc(NCC3CCCC3N)ccc2s1 21744,c1(C(N2C(C(N3CC(CC(C)C)OCC3)=O)CC2)=O)nccc2cc[nH]c12 21745,CC(C)CC(CNC(=O)CC(C)NC(c1ccccc1)=O)NC(C1CC(F)C1)=O 21746,N1(C(C(C=C)C)=O)CCOCC1CC(=O)NC1(CCO)CCCC1 21747,Cc1cc(N)c(C(N2CCC(O)(C(C)NC(c3cc[nH]n3)=O)CC2)=O)cc1C 21748,N1(C(CCCC#C)=O)CCC(O)(CCNC(c2csc(COC)c2)=O)CC1 21749,CC1CN(C(c2ccc(C3CCC3)nc2)=O)CC1NC(C1(F)CCOC1)=O 21750,Cc1ccc(S(=O)(=O)N(CC(N2CC(NC(=O)CC3CCC3)C(O)C2)=O)C)cc1 21751,c1(-c2ccc(F)c(C(N3CCC(NCC)C3)=O)c2F)c(OC)ccc(SC)c1F 21752,c1(C(=O)NCC2N(C(C=Cc3nnc(C(C)C)o3)=O)CC2)cc2scc(Cl)c2[nH]1 21753,c1(C(=O)NCCC2CC(NC(C3ON=C(C(C)C)C3)=O)C2)cncc2c[nH]nc12 21754,S(=O)(=O)(c1cccnc1NCCc1nncs1)NC1C(C)CCCC1 21755,C=CCCCCC(=O)NCC(C(C)C)NC(=O)CN1C(=O)CCCC1=O 21756,C1(C)(CNC(Cc2c(C)nc[nH]2)=O)CCCC1NC(c1cnc(C(F)F)cn1)=O 21757,C=CCC(C(=O)NC1(COC)CC1)OC.N12CCN(CC1)C(=O)C=CC2 21758,c1(-n2ncc(C(N3CC(C)(NC(CCOC)=O)C3)=O)c2)ccc(F)cc1 21759,c1(SCC(=O)NC2C(Nc3cc(OC)nc(SC)n3)C2)nc2ccccc2s1 21760,CCC(C)(C)C(=O)C(=O)NC1CC(C)N(C(=O)CN2CCC2)C1 21761,Cc1ncc(N)cc1C(N1CC(CCNC(c2ccc(Cl)cn2)=O)C(C)C1)=O 21762,c1(SC)ccc([N+](=O)[O-])cc1C(=O)NCCCC(C)(C)NC(=O)CC1(CO)CC1 21763,CCCCC(CNC(c1c(C)nsc1N)=O)NC(=O)CCN(CC)CC 21764,c1(OC)ccc(OC)c(C(=O)NCC2CN(C(c3sncc3C)=O)CCO2)n1 21765,c1(C(N(CCNC(=O)CCc2cccs2)CC)=O)cccc(C2(C)CCO2)c1 21766,CC(C)S(=O)(=O)CC(=O)N1CC(N(C(=O)C(C)NC(N)=O)C)C2(CC2)C1 21767,c1(C(F)(F)F)cc(CNCC2(NC3CCC3)CC2)ccn1 21768,C(=O)(C(COC)CC)NC1(C(N2CCC(C(=O)NC)C2)=O)CC(O)C1 21769,N1(C(CCSCC)=O)CCN(C)CC1C(=O)NCc1nnn(C)n1 21770,c1(C(C)C)cc(N2CCCC2CNC(=O)C(C)C2CC2)n2ncnc2n1 21771,CC1CC(NCC2CCN(C(C)(C)C)CC2CO)CC(C)O1 21772,C(=O)(CC(C)(C)CC(F)(F)F)NCCCNC(c1ncc(OC)nc1)=O 21773,C1(NC(C(C)O)=O)(CO)CCCN(C(C2(c3ccc(Cl)c(Cl)c3)CC2)=O)C1 21774,N1(C(C(C)OCC2CC2)=O)CCCC1C(C)NC(c1ccc(F)s1)=O 21775,c1(CCC(=O)NCCCN(C(C(CCC)NC(C)=O)=O)CC)ccc(C)cc1C 21776,C1(CNC(C(C)NC(C)=O)=O)CCC2(CN(C(=O)C(C)C(C)(F)F)C2)O1 21777,c1(C(N2C(C)(CNC(=O)COC3CCOC3)CCC2)=O)ccn2nccc2c1 21778,C=CCCC(CO)NC(c1nc(CNC(c2ccnc(C)n2)=O)oc1C)=O 21779,C1(NC(C2(CNC(C(C)N(C)C)=O)CCCO2)=O)CC2(C1)CC(O)C2 21780,c1(C(=O)NC2CN(C(CC=C=C)=O)C(C)C2)ccc(SC)c(Br)c1 21781,CCC(C(=O)NCCC1(OC(C)C)CN(C(=O)C(C)c2ccsc2)C1)N(C)C 21782,C1(CN(C(C2C=CCCC2)=O)C2CC2)C2CN(C(=O)COCC(F)F)CC12 21783,C1(NC(C(C)OC2CCOC2)=O)CC2(CCCN(C(C3(O)CCSC3)=O)C2)C1 21784,C(=O)(C#CC1CCCOC1)NCC1=CCN(C(Cc2cc(C)no2)=O)CC1 21785,C1(NC(c2cc(Cl)ccn2)=O)CC2CC1N(C(=O)C(C1(O)CCCC1)F)C2 21786,C1(CC(=O)NCc2cccc(F)c2)CC2(C1)CN(C(=O)Cc1cnns1)C2 21787,C1(C(=O)OC(C(=O)OCCC)C)CC(=O)N(C(c2ccc(F)cc2)C)C1 21788,c1(C(N2CCC(CNC(C(C)OCC(C)C)=O)C2)=O)c2c(c[nH]c1=N)CCC2 21789,N1(C(=O)Cn2cncn2)CC2CN(C(C3(c4cccc(F)c4)CC3)=O)CC2C1 21790,C(c1cc2c(cc1OC)CC(C)O2)=CC(=O)NCC(CC)NC(C1CC1F)=O 21791,c1(C(N(CCCNC(=O)CC(C)C(F)F)CC)=O)cn2cc(C)c(C)cc2n1 21792,C=CCC(C)(C)CC(=O)N1CCC(C)(C)C1C(=O)NC1CCNC(=O)C1 21793,C1(C(=O)NCC2(C(N3CCC3(CO)CO)=O)CC2)COc2ccccc2O1 21794,C1(CC)OCCC1C(=O)NCC1(O)CN(C(c2c[nH]nc2-c2ccnn2C)=O)C1 21795,C12(CNC(C(CCC)=CCC)=O)CCCC1N(C(C1CC(O)CN1C)=O)CC2 21796,N1(C(c2c(CNC(C(C)CO)=O)ccs2)=O)CCC(C)C1c1ccccc1 21797,c1(NC(C(N2CCC(C(=O)OC)C2(C)C)=O)=O)ccc(N=[N+]=[N-])cc1 21798,CCCCC(O)CC(=O)NC1CCC(CNC(c2ccc3c(c2)C(C)CO3)=O)C1 21799,N1(C(C(CC(C)C)=O)=O)CCC2(CC1)CC2CNC(=O)CCCc1cccs1 21800,C1(C(=O)NCC2CN(Cc3c(C)ncs3)C2)CC(=O)N(C)C1c1cccnc1 21801,C1(C(=O)NCc2c(C)cn(C)n2)CN(C(=O)C(CO)C(C)(C)C)CC1C1CC1 21802,n1(C(C)C(N2CC=CC(NC(=O)C(C)(F)F)C2)=O)c(S)nc2ccccc2c1=O 21803,c1(NCC2N(C(Cc3ccc(C(=O)O)cc3)=O)CC2)nc(Br)cnc1Cl 21804,c1(C(N2CCC3(CNC(=O)O3)C2)C(=O)NCCC#N)cn2cc(Cl)ccc2n1 21805,c1(C(=O)NCCCN(C(C(C2CCOCC2)OC)=O)CCO)cn(C)[nH]c1=N 21806,c1(OC)cc(F)c(CNC(c2ccc(-c3cccc4ccnn34)cc2)=O)cc1N 21807,C1(C(=O)NC(CNC(c2sc(CC)c(C)c2)=O)(C)C2CC2)CC2CSCC(C1)C2 21808,C(=O)(CCN=c1[nH]c(=NCCC(C)C(F)F)c2sccc2[nH]1)N(CC)CC 21809,C(=O)(C1CCCn2ccnc21)N1CC2(C(NC(C(CC)OC)=O)CCC2)C1 21810,N1(C(CN(C(=O)CCc2cc(Cl)no2)C)=O)CCN(C(c2ccoc2)=O)C2CC12 21811,CCCC(C(=O)N(CC(CC)NC(c1ocnc1C(C)C)=O)C)C(C)C 21812,N1(C(COCCCC)=O)CCC(CNC(C2CC3CCC2O3)=O)(OC)CC1 21813,O=C(C(F)(F)F)NCC1(Cc2ccccc2)CN(CCOc2ccccn2)C1 21814,N1(C(CC(COC)COC)=O)CCCCC12CN(C(c1cc(O)ncn1)=O)C2 21815,c1(NC2N(C(=O)NC(C(C)C)CN3CCOCC3)CCC2)ccc(C#N)nc1 21816,N(C(=NCCCCn1ccnn1)N1CC=C(F)C1)CCCOC 21817,Cc1nn(C)cc1CC(=O)NCCC1CSCCN1C(=O)CC(C)(C)C1CC1 21818,N1(C(C2C(C)(C)C2C#N)=O)CCC(NC(=O)CSCc2cccnc2)C(CO)C1 21819,C1(C(=O)NCC2CC23CCOC3)C2CC1N(C(=O)C(F)=CC1CC1)C2 21820,c1(C(N2CCC(C(=O)Nc3ccc(C)cc3)C2)=O)cc2c(cc1Cl)NC(=O)C2 21821,C1(n2cc(C(C)C3CC3)nn2)CCN(C(=O)C(n2cc(C(O)C3CC3)nn2)C)CC1 21822,C(=O)(C(C)(C(=O)OC(C)(C)C)OC)NCCN(C(c1cnc(CC)s1)=O)C(C)C 21823,C(=O)(C(c1cccs1)NC(=O)C(C)n1cccn1)N(CCF)CC 21824,c1(SC)nc(Cl)c(CN2CC(C(N3CCCCC3C)=O)CC(F)C2)c(Cl)n1 21825,N1(C(CCN(CCC)C)=O)CCCC(N(CCF)C(c2cc(CC)oc2C)=O)C1 21826,N1(C(C2(OCC)CCOCC2)=O)CC(NC(c2cnccc2C)=O)CC(O)C1 21827,c1(C(N(C)CC2N(C(C(F)=C(C)C)=O)CCCC2)=O)ccc2c(c1)C(=O)C(=O)N2 21828,c1(C(N(CCCN(C(C2C(CC)OCC2)=O)C)C)=O)ccccc1C(C)=O 21829,C(C(C(C)(C)C)NC(c1cc(-c2ccoc2)[nH]n1)=O)NC(c1c(C)ocn1)=O 21830,N1(C(C(CCC)C)=O)CCCCCC1CNC(=O)CCc1c(F)cccc1Cl 21831,CC(C)CC(O)C(=O)N1CCCC(C(C)C(=O)NCCC#CCO)C1 21832,C(=O)(C(C)(O)CC(C)C)NCC(CNC(c1c(C)nc(Br)s1)=O)F 21833,N1(c2n(CC)c(-c3c(C)nn(C)c3OCC3CC3)nn2)CCS(=O)(=O)CC(C)C1 21834,c1(C(=O)NCC2C(NC(C(Cc3ccc(C)cc3)OC)=O)C2)ccc([N+](=O)[O-])s1 21835,N1(C(C(C)CC2CCCC2)=O)CCCC(O)C1.C12CC1CNC2=O 21836,C(=O)(CCC(=O)NC1(C)CCN(C(=O)C(C)OCc2ccncc2)C1)OCC 21837,c1(C(N(C(C)CCNC(C2(C)CC3CC3C2)=O)C)=O)cccc(F)c1N 21838,c1(C(N(C(C)(C)C)CCC)=O)oc(C)nc1C.C12CC3CC3N1C(=O)O2 21839,c1(CC(=O)NC2C=CCN(C(c3ccc(Br)o3)=O)C2)ccccc1CO 21840,CC(C(=O)NC1CC(NC(=O)C(C)N2CCC2)C1)S(C)(=O)=O 21841,c1(C(N(CC(CNC(C2(CC#C)CC2)=O)C)C)=O)cnc(CC)[nH]1 21842,C=CCCCCCCCC(=O)NCCOCCNC(=O)C(c1c(C)n[nH]c1C)C 21843,C=CC(C)(CC)C(=O)NCC1(F)CC(NC(=O)C=CC)C1 21844,CCC(CC(=O)NCC(=O)Nc1cn[nH]c1)N(C(=O)CC1(O)CCOC1)C 21845,c1(C(N2CC(CNC(c3cc(Cl)cs3)=O)C3C2C3)=O)ncc2ccccn12 21846,N1(C(CCNC(COC)=O)=O)CCCN(C(C2CC2[N+](=O)[O-])=O)CC1C 21847,C1(CNC(=O)CC2CCOC2=O)(NC(C2CCSCC2)=O)CC(F)(F)C1 21848,O=C(O)CC1(CNC(N2CCC(c3ccc(O)nc3)C2)=O)CCCc2ccccc21 21849,C(CCCC(=O)NCC1(OC)CCN(C(=O)Cn2cncn2)C1)NC(=O)OC 21850,CC1=C(C(=O)O)N(C(c2ccc3[nH]ncc3c2)=O)CCCC1 21851,c1(C(=O)NCC2C(NC(c3ccc(F)cn3)=O)CC2)cccc(F)c1Br 21852,c1(C(N2CC3C(NC(C4(O)CC(F)(F)C4)=O)C3C2)=O)ccc(Br)cc1F 21853,c1(C(N2CC(CNC(c3cncc(F)c3)=O)C(O)C2)=O)coc2c1C(O)CCC2 21854,N1(C(C2CCC(=C)CC2)=O)CC2(CC2)CC1C(=O)Nc1[nH]cnc1C(N)=O 21855,c1(C(N2CC(C(=O)Nc3cnc(Cl)cc3I)SCC2)=O)c(F)ccc(Cl)c1Cl 21856,c1(C(N2CC(NC(CNC(c3ccc(C)cc3)=O)=O)C2)=O)cc(Br)c(C)cc1F 21857,C(=O)(CCCN=[N+]=[N-])N(CCC(C(C)C)NC(C1(C)CC=CCO1)=O)C 21858,Cc1cc(NCCCCC(C)NC(=O)C(F)(F)CN(C)C)n2nc(C)nc2n1 21859,N1(C(C2(CC)CC2)=O)CCCC2C1CCN2C(c1cn(CC(F)(F)F)cn1)=O 21860,Cc1cc(C(=O)N(C)CC2CCN(C(=O)C(F)C(C)C)CC2)ccn1 21861,c1(OCC)ccc(C(=O)NCC2CC2CNC(C23CCCN2CCC3)=O)c(O)c1 21862,C(=O)(C(C(C)C)n1cccc1)NCCC1CCN(C(c2cc(OCC)no2)=O)C1 21863,c1(NCC(N2CCC=C(Br)C2)=O)ccc(-c2nn[nH]n2)cn1 21864,CCS(=O)c1ccccc1C(=O)NC1CC(NC(C2CC2C)=O)C1 21865,N1(OC(C(C)(C)C)=O)CC(C)N(CCC2(CCOC)CC2)CC1C 21866,CCC(C)C(C)C(=O)N1CC2(CC(CC(=O)NCCOCc3ccccn3)C2)C1 21867,c1(CC)nc(C(=O)NCCC2CN(C(=O)C(COC)N(C)C)CCO2)c(N)s1 21868,c1(C(=O)NCC(CNC(CCCC=C)=O)C)ccn2ncccc12 21869,C(CCC(C)(C)C(=O)N1CCC12CCCC2)NC(c1cn(CC)nc1)=O 21870,c1(CN2CC3(N(C(c4ccc(O)cc4)=O)CC3)C2)c[nH]c2ncccc12 21871,CS(=O)(=NC(=O)c1cnc(-c2ccc(Br)s2)nc1)c1ccncc1 21872,C(CS(C)(=N)=O)NC(C(n1cc(CCC2CCOC2)nn1)C)=O 21873,O=C(C1=CCCOC1)N(C1C2CN(Cc3ccc(=O)oc3)CC12)Cc1ccccc1 21874,C1(CNC(c2ccc(NC)cc2)=O)CC(C(=O)N(C2CC3CC3C2)C)=NO1 21875,c1(CC)oc(C(=O)N(CC(C)NC(=O)C=Cc2ccsc2)CC)cc1C 21876,c1(CN2CCC(C)(C(=O)Nc3[nH]nc(OC)c3C#N)CC2)c(F)ccc(F)c1C 21877,Cc1cc(C(N2CCC(C(C)(C)NC(=O)CSCC(N)=O)C2)=O)cc(C)c1F 21878,c1(N(CCNC(C2(NC(N)=O)CC2)=O)C(C2CCOC2)=O)c(Cl)cccc1Cl 21879,CC(C)C(C(C)NC(c1cn(C(C)C)cn1)=O)NC(=O)CCC1CCC1 21880,Cn1cc(C(C(=O)NCC2(C(C)(C)O)CCC2)NC(=O)CCOC2COC2)nn1 21881,C12(C(N(CCN(C(CCc3cc(C)on3)=O)C)C(C)C)=O)CCCC1CC2 21882,Cc1ccnc(C(=O)N(C2CCN(C(=O)CC3CCC4CC34)CC2)C)c1O 21883,CC1CCN(C(=O)C(N2CCC3CCOC3C2)=O)CCN1 21884,N1(C(C2CC(O)(CC#C)C2)=O)CCOC(CC(=O)NCC2COCC2O)C1 21885,C1(C2(O)CN(C(=O)C(C)OC3CCOC3)C2)(CNC(C(c2cccs2)OCC)=O)CC1 21886,N1(CCCC(C)C#N)CCC(S(C)(=N)=O)C1 21887,N1(CC=C(C)C)CCC(C2CCCO2)C1(C)C.c1(O)ncc(C=O)s1 21888,CP(C)(=O)CC(=O)N1CCOC(CCNC(=O)CC2CCC(=O)O2)C1 21889,c1(C(=O)NC2(CCNC(Cc3c(C)occ3)=O)CCC2)cnc(S)nc1 21890,N1(C(C(CCC)(C)O)=O)C2CCCC1CN(C(C1(OC)CCCCC1)=O)C2 21891,c1(C(=O)NC2CC(N(C(=O)Cc3ccccn3)C)C2)ncncc1C#N 21892,N1(C(C(CCN(C)C)NC(C2C(C)=CCS2)=O)=O)CCCC2(CCCC2)C1 21893,c1(CC(N2C(CCNC(CC3CC(OC)C3)=O)CCC2)=O)cncc(C)c1 21894,C1(NC(COC)=O)COCCN(C(=O)C(C2CCCCCC2)OC)C1 21895,c1(OC)cc(F)c(C(=O)NCC2(C)CN(CC3CNC(=O)CO3)C2)cc1OC 21896,C12(NC(=O)Cc3cnccn3)CCCN(C(C3CC3(Cl)Cl)=O)CC1C2 21897,c1(CC(N2CCC(O)(CNC(c3[nH]cc(CC)c3)=O)C2)=O)cccc2sccc12 21898,c1(C(=O)NC(c2nc(CNC(C3(OC)CCSC3)=O)n[nH]2)C)oc(CC)nc1C 21899,c1(C(=O)NC2C(NC(COCCC=C)=O)CCC2)cc(F)c(C)cc1N 21900,C1(CNC(=O)COCC(F)F)CN(C(c2ccc(Cl)cn2)=O)C2CCN1C2 21901,c1(SC)cc(N2CCSCC2CCNC(=O)CC2CCC(=O)N2)nc(SC)n1 21902,N1(CC)CCN(CC(N2CCC(OC(=O)Nc3ccc(F)cc3)C2)=O)C(=O)C1=O 21903,CC1CC(C(=O)NCC2(F)CN(C(c3c(F)cccc3Br)=O)C2)=NO1 21904,C1(NC(CC2(NC(C(CC)n3ccnc3)=O)CSC2)=O)CN(C)C2(CCC2)C1 21905,C1(CC(=O)NC(CC(C)NC(COCC(=O)OC)=O)C)CCC(=O)N1C 21906,C(C(=O)Nn1cnn(C)c1=S)C1N(C(COCC)=O)CCCC1 21907,C1(C2CCN(C(=O)CCCCCn3cnnn3)C2)(NC(c2c(C)con2)=O)CC1 21908,N1(C(C(N2CCN(C)CC2)C)=O)CC2CC1CN2CC(O)Cn1cccn1 21909,C(C)(C(CC(=O)N1CC(C)CC1(C)C)NC(C1CN(C(C)C)C1)=O)OC 21910,c1(NC(C2CCN(C(=O)OC)CC2)=O)ccc2c(c1)CCC(C)C2 21911,c1(C(=O)NCC2(O)CCN(C(c3c(C(C)C)nn(C)c3)=O)C2)cc2n(n1)CCC2 21912,C1(CNC(c2c(CCCC)ocn2)=O)CC(F)(F)CN1c1nnc(C(=O)OC)s1 21913,C(=O)(CC(C)(C)COC)N(CC(C)(C)NC(C1C(CC)CCC1)=O)C 21914,c1(CN(C)C(C2(CNC(c3coc(Br)c3)=O)CC2)=O)cccc(CO)c1.C1(=O)CN1 21915,N1(C(c2cnc3cnccn23)C(=O)NC(CC)C)CCc2cc(C#N)ccc2C1 21916,N1(C(Cc2cc(C)nn2C)=O)CC(NC(C2(n3cc(Cl)cn3)CC2)=O)CC(C)C1 21917,c1(OCCC)cccc(C(N2CCCCC2CN(C)C(c2cnn(C)n2)=O)=O)c1 21918,C(=O)(NNc1nc(C)c(C)s1)Nc1ccc(C2CCN(CC)CC2)cc1 21919,c1(C(=O)NCC(C)(C)O)n[nH]c2c1CCN(C(c1cccc(F)c1O)=O)C2 21920,C1(C)(NC(C(CCC)O)=O)CCN(C(=O)CCC2CC2(F)F)CC1 21921,c1(C(N2CC(CNC(CN(CC)CC)=O)(OC)C2)=O)c(C)ccc(F)c1N 21922,Cc1cc(N(CC(N2CC(CS(C)(=O)=O)C2)=O)C)nc(NCc2nncn2C)n1 21923,c1(C(=O)NCC2CCC(NC(c3cnnc(Cl)c3)=O)C2)ccc2nn[nH]c2n1 21924,C(=O)(CC(Cl)Cl)N(C)CC=CC(=O)N1CCC1 21925,N1(C(C2CC(C)OC2)=O)CC2CCC1(CNC(C1CCC=CCC1)=O)CC2 21926,c1(C(N2CC(COC)(NC(=O)C(C)OCC(F)(F)F)C2)=O)ccc(C#N)cc1C 21927,N1(C(C(CC)C#N)=O)CCC2(C(=O)NC3(C)CC4CCC3C4)CCCC12 21928,N1(C(c2cnc(OCC)s2)=O)CCC(F)(CNC(=O)CC2CCCC(=O)N2)C1 21929,C1(C(=O)NC2CC(N(C(CCNC(C)=O)=O)C)C2)Cc2ccccc2S1 21930,N1(C(c2c(C)noc2C)=O)CCC(CNC(=O)C(C)(C)c2cnsc2)C(C)C1 21931,Cc1c(Cl)ccc2c(CC(=O)NCCCC3CCCN3C(=O)CC(C)F)coc12 21932,CC1CC(NC(c2ccc(N(C)C(=O)C3CC3)cc2)=O)CN(C(=O)C(F)Cl)C1 21933,c1(C(=O)NC2CN(C(C=C(C)Cl)=O)CC2O)ccc(Br)c(O)n1 21934,C1(CNC(CCCNC(C(c2n(C)ccn2)O)=O)=O)CC2CCCC2C1 21935,CN1CCC2(CCN(C(CCC3CC=CCC3)C(=O)NCC3CCOC3)C2)C1 21936,N1(C(C=CC(C)C)=O)CCC2CC(NC(C3CC(=O)N3)=O)CCC2C1 21937,O=C1CCc2nc(N3CCCC4(NC(C5CCC6(CC6)C5)=O)CCCC34)ccc21 21938,C(=O)(n1nccc1NC(=O)Nc1ccc(O)c(C(=O)O)c1)OC(C)(C)C 21939,C(=O)(C(O)CC(C)C)NCC1(COC)CN(C(=O)CCC2(C#N)CCC2)C1 21940,c1(C2(C)CC2NC(=O)C(N2CCC(OCCO)CC2)=O)cccc(Cl)c1 21941,c1(Oc2nccc(N(C(CN(CCC)CCC)=O)C(C)=O)n2)cc(Cl)cc(Cl)c1 21942,C1(NC(Cc2cccc(C)c2)=O)CN(C(c2ncn(C)c2C)=O)CC(F)(F)C1 21943,C1(C(=O)NC2CCN(C(Cn3c(C)csc3=O)=O)CC2)CS(=O)(=O)CCO1 21944,C(CC(C(C)(C)C)NC(c1ccccn1)=O)N(C)C(c1scnc1C(F)F)=O 21945,C(=O)(C1=CC2(CCOCC2)C1)NCC1CCC(C(=O)NCCCC2C(C)C2)CC1 21946,N1(C(c2c(OC)cc(OC)nc2)=O)CC2CC(C1)N(C(C1CCC3(CC3)C1)=O)C2 21947,CC1C(C(N2CCC(C3OCCCC3NC(=O)C3=NOCC3)CC2)=O)CCN1C 21948,N1(C(CC2COCC(C)O2)=O)CCN(C(c2cccc(C(C)C)c2)=O)C(CO)C1 21949,c1(C(=O)NCC2(N(C)C(=O)OC(C)(C)C)CCOC2)cnn2ccn(C)c12 21950,C(=O)(C1=CC2C=CC(C1)C2)NCCC(C(=O)NC1(CC(C)(C)C)CC1)OC 21951,CC1(C)CCCC(C(N2CCC3(CC3NC(=O)CN3CC4CCC3C4)C2)=O)C1 21952,C(=O)(C(C(C)C)N(C)C)NC1(CC=CC(NOCCCC=C)=O)CCC1 21953,C1(NC(CNC(=O)C2CC2)=O)CCCCC1NC(=O)CNC=O.n12cc(nn1)C2C 21954,c1(CN(CCC)C(=O)NC2CCC2C)ccc(F)cc1 21955,CN1C(=O)C2CN(C(c3ccn(C4CC4)c3)C(=O)NC3CCOCC3)CC2C1=O 21956,c1(C(N2CCCC(c3nccn3C)C2)C(=O)NCCC)ccc2c(c1)OCC2 21957,c1(CCC(=O)NCC(C)NC(C2CC(CF)C2)=O)ccccc1OC(F)(F)F 21958,C1(CC=C)(NC(=O)CC(C)OC)CCN(C(=O)CSC(F)(F)F)C1 21959,Cc1nc(C)c(C(=O)NCC(C2CCCN(C(c3[nH]cnc3C#N)=O)C2)(C)O)s1 21960,c1(-c2nnn(C)n2)ccc(NC2CCOC(c3ccc(F)cc3)C2)cc1Cl 21961,N1(C(=O)CCC2CCC2)CCC2(CC1)CCN(C(C1CC1C(F)F)=O)C2 21962,C(=O)(N=c1cc(C)n(C(C)C)[nH]1)C1(OC)CCN(C(=O)CC2CC=CCC2)C1 21963,N1(C(=O)NCCCOc2ccc(F)cc2)CCS(=O)CC1c1ccccc1 21964,C(=O)(CC(C)C(F)(F)F)NC(CC)CCC(=O)NCC1CC12CCCCC2 21965,Cn1cnc(NC2CC(CCNC(c3cccc[n+]3[O-])=O)C2)c(Br)c1=O 21966,c1(CC(N2CC(NC(C=C(C)Cl)=O)(CO)C2)=O)ccc(-c2nc[nH]n2)cc1 21967,C(C(C)C)(C(O)C(=O)NC(C)(CSC)C(=O)NC(c1cccc(C)n1)C)OC 21968,C1(O)(CC(N2CC(C(=O)NCCCOC)(Sc3ccccc3)C2)=O)CCOCC1 21969,N1(C(C(C)c2ccsn2)=O)CCC(CCNC(C2CCCC2)=O)C(F)(F)CC1 21970,C(=O)(C(CCNC(=O)C(C)c1cc[nH]n1)OC)NCC(C#C)CC 21971,C1(NC(CSCC(N)=O)=O)CN(C(c2sccc2Cl)=O)CC1C(F)F 21972,CN=c1nc(N2CCC(C)(N3CCOCC3)C2)[nH]c(=NC2Cc3ccccc3C2)[nH]1 21973,C1(CC(=O)N(C2(C(NOCCC(C)C)=O)CCC2)C2CC2)CN(C)CCO1 21974,c1(C(N(CCN(C(c2cncc(OCC)c2)=O)C)C)=O)ccc(OC)c(OC)c1 21975,C1(C(=O)NCc2cn(CCNC(CC(C=C)C)=O)nn2)CCOC(C)(CC)C1 21976,N1(C(c2c(CNC(C(CC=CC)CC)=O)nccc2)=O)c2ccccc2CC1C 21977,C1(NC(C2C(C=C)C2)=O)CCC(C)N(C(c2csc(-c3ccccc3F)n2)=O)C1 21978,Cc1cc(C(=O)NC2CCN(Cc3c(C)noc3C)C2)nc(Cl)c1 21979,C1(NC(C2C3C(NC(c4cnc(CC)o4)=O)C4C(C3)C42)=O)C(C)(C)C(O)C1(C)C 21980,C(CC(=O)N(CCNC(C1(n2ccnn2)CC1)=O)C1CC1)=CCC 21981,c1(C(=O)NCCC(C)N(C(C2C(CC)OCC2)=O)C)c[nH]cc(Cl)c1=O 21982,Fc1cc(NCc2c(C(F)(F)F)nn(CC(F)F)c2Cl)cc(Cl)c1 21983,N1(Cc2cccc(C(=O)NCc3c(C)noc3C)c2)CCC2(CC1)OC(=O)NC2C 21984,c1(OC)cc(C2(C(=O)NCC#CCNC(=O)CCCSC)CCCC2)ccc1C 21985,c1(-c2ccc(SCC)s2)c(C(=O)NC)nc2ccccn12 21986,c1(C(N(CC#C)CCC)=O)cc2ccsc2[nH]1 21987,N1(C(c2c(CC)nco2)=O)CC2CCC(N(C(=O)C(C)CC(F)F)C)C2C1 21988,c1(C(N2C(CN(C(=O)C3=C(Cl)CC3)C)COCC2)=O)noc2c1COCC2 21989,C12(O)CCN(C1)C2=O.c1(OC)ccc(C(=O)N(CC(C)C(=O)OC(C)(C)C)C)s1 21990,C1(CNC(c2cncc(NC(c3cocn3)=O)c2)=O)CCc2ccccc2C1 21991,C1(CNC(C(COC)(C)O)=O)CC2CCC1N2C(=O)Cc1ccc(OC)c(O)c1 21992,c1(C(CC)N(C(c2conc2C)C(=O)NCC)CC2CC(F)(F)C2)ccccc1 21993,c1(CC(=O)N(CCC)CCNC(=O)CC2CC2(Cl)Cl)ccnc(Cl)c1F 21994,C1(CCC)CCCN(c2nnc(-c3ccccc3Cl)n2CCC(=O)N(C)C)C1 21995,N1(C(C(C)(C)OC)=O)CCN(C(c2ccc(F)cc2Cl)=O)C(C(C)C)C1 21996,Cc1ccc(C(=O)NCC2(NC(C3CC(F)(F)C3)=O)CCOC2)nc1O 21997,N1(C(CC(=O)NCC)=O)CCN(C(c2c[nH]c(=N)o2)=O)C(C(F)F)C1 21998,CCC(CCC(=O)NC1(CNC(c2ccc(C(=O)OC)c(O)c2)=O)CCC1)OC 21999,N1(C(c2ncc(CC)cn2)=O)CCCC(O)(CNC(C2CCCC(=O)N2C)=O)C1 22000,N1(CC(=O)NCC(C)N(C(c2ccc(Cl)cc2)C(N)=O)C)CCCCCC1 22001,N1(C(C2C(C(=O)O)C23CC3(F)F)=O)CCc2c(I)n[nH]c2C1 22002,N1(C(CCCCOC)=O)C2CCC1CC(CNC(=O)CC1CC(C)=NO1)C2 22003,CCC(C)C(C(=O)NCC(F)F)N(C(C(=O)NCCNC(C)=O)=O)C 22004,C1(CC(C)(C)C)CCN(C(=NCCNC(=O)NC2CC2)NC2CCC2)C1.CS(C)(=O)=O 22005,c1(C(=O)OCC(=O)NCC2C(C(=O)OC)CCC2)cc(C)cc(C)c1 22006,C1(NC(C(C)OCCOCC)=O)CCN(C(c2cnc(S)[nH]2)=O)C1C 22007,CC(C)C(C)(CNC(c1n[nH]cc1CNC(C1C=CC=CC=C1)=O)=O)C(C)C 22008,CN1CCC2(CC1)CN(C(C1CCN(C(C3(C)CC=CC3)=O)CC1(C)C)=O)C2 22009,c1(C(=O)NCC2CC(NC(c3cc(F)cs3)=O)C2)csc(O)n1 22010,C1(C2CCC2)(C(N(CCC)CCNC(=O)C(CCOC)OC)=O)CC1(F)F 22011,c1(OCC)cc(Br)cc(C(=O)NCCNC(=O)CC2C(C)C2(F)F)c1N 22012,N1(C(C(C)Cc2ccc(Cl)cc2)=O)CC2CCC(C1)N2Cc1ccc(F)nc1 22013,c1(NC(CNC(C2(SC)CC2)=O)C(C)C(C)C)ncc(Cl)cc1[N+](=O)[O-] 22014,CS(=O)(=O)c1ccc(S(=O)(=O)N2CCOCC2CNC(c2ccco2)=O)cc1 22015,N1(C(c2ccc(C)nc2)=O)CCC(C2CN(C(c3c[nH]cc(Cl)c3=O)=O)C2)CC1 22016,CCN=C(NCC1(CC)COC1)NC1CC(=O)N(C(C)(C)C)C1 22017,N1(C(CN(CCOC)C2CC2)=O)CCC(C2(NC(=O)CN(C)C)CC2)C1 22018,c1(CNC(CC(C)OC)=O)cnn2c1CN(C(=O)C(c1cccc(N)c1)O)CC2 22019,C1(C(=O)NCCCNC(CC(OCC)OCC)=O)CC(=O)N(C2CC2)C1 22020,c1(C(=O)NCCC(C)NC(c2ccc(C)c(F)c2)=O)ccc2c(n1)OCCO2 22021,c1(CN2C(=O)CN(C(COc3cccc(C)c3)C)C2=O)c(C)nc2ccccn12 22022,C1(C(=O)NCCCN(C(c2c(C)cc(C)cc2C)=O)CC)CCCCC12CCC2 22023,C1(C(=O)NC(CC)C)CC(=O)CN1C(=O)C(c1ccccc1)F 22024,C(CC(C)(C)CC(=O)N1CCN(C(=O)Nc2cc(O)c(F)cc2N)CC1)OC 22025,c1(CCNC(C(C2CCC2)NC(c2cc(Cl)n[nH]2)=O)=O)ccncc1F 22026,c1(C(N2C(CCNC(c3cnnc(O)c3)=O)CCCC2)=O)ccc(O)nc1Cl 22027,Cc1ccc(N(CCC#N)C(=O)COC(C(C)CC(F)(F)F)=O)cc1 22028,c1(C(=O)NCC(C)CN(C)C(c2cc(F)c(N)cc2F)=O)cnc2[nH]cncc1-2 22029,C1(C(C)(C)O)CCCN(C(=O)C(N2CCNCC2)C2CC2)C1 22030,C(=O)(CC(C)(C)C(C)(F)F)N1CCN(C2CCN(C(c3ccccc3)C)CC2)CC1 22031,c1(C(=O)NCC(C)NC(c2c(C)nn(C)c2C)=O)cc(Br)c2ccccc2c1 22032,c1(CNC(C(C2CCCCC2C(C)C)CC)=O)ccc(Cl)c(Cl)c1C 22033,Cc1cc(C)c(C(=O)NCC2CCCCN2C(=O)Cn2ncn(C)c2=O)c(C)c1 22034,N1(C(C2N(C(C(C)=CC3CC3)=O)CCN(C)C2)=O)CCC2CCC(C1)N2C 22035,CCCC(C)(C)C(=O)NC(C1CCN(C(=O)CNS(=O)(=O)N(C)C)C1)C 22036,C1(Cc2nc(C)sc2)CCN(N2CCOCC3(CC3)C2)C1 22037,N#CC12CCC(NC(C3CSCCN3Cc3cnc(Cl)cn3)=O)(CC1)CC2 22038,N1(C(CN2CC(CC)C2)=O)CC2CC2(NC(=O)Cc2cncc(O)c2)C1 22039,c1(C(=O)OCC(F)=C(C)C)ccc2oc(=N)[nH]c2c1 22040,Cc1cnccc1C(=O)NCC1CCC(NC(=O)C(C)C(F)F)CC1 22041,c1(C(=O)NCC23C(CN(C(C(CSC)C)=O)C2)C3)cccc(=O)n1C 22042,C1(CNC(C2CC3CCC2O3)=O)C2CN(C(c3ccc(-c4cccs4)o3)=O)CC12 22043,Cc1cc(C(=O)NC(C2CCCCC2)CNC(=O)C2=CCC2)nn1C(C)C1CC1 22044,CCC1=NOC(C(=O)NC(CCC2CCC2)C(=O)Nc2ccccc2OC)C1 22045,C1(CNC(C(C)c2cccs2)=O)CCN(C(=O)CCS(N)(=O)=O)C1(C)C 22046,Cc1ccc2c(N3CCn4c(O)nnc4C3)nc(=NCCCCC(N)=O)[nH]c2c1 22047,C1(CC(=O)NCCN(C(c2c(C)cc[nH]2)=O)C)CCCCN1C 22048,C(=O)(C(C(C)C)n1cncn1)NCC12CC(NC(C(C3CC3)OC)=O)(C1)C2 22049,CC(C)(C(=O)N1CC(C2CN(C(=O)Cc3ccon3)C2)C1)C1=CCSCC1 22050,C#CCC(C(=O)N(CCCO)CC#C)NC(c1cccnc1)=O 22051,C1(C(N(CC(O)C2CC2)C)=O)CCN(C(c2c[nH]c(C(N)=O)c2)=O)C1(C)C 22052,C1(C)(C(=O)NCC2N(C(C(CNC(C)=O)(C)C)=O)C3CCC2C3)CC(C(C)C)=NO1 22053,Cc1cccc(CSCCNC(C2CCCN2C(=O)Cc2ccccc2I)=O)n1 22054,N1(c2cc(NC(C)C(F)F)ncn2)CCCC2(C1)C(=O)NCCN2C 22055,C(=O)(C1=CNS(=O)(=O)N=C1C)N1CCCC(NC(C(C)=CC)=O)C(F)C1 22056,Cc1ccc(C(N2CCN(C(=O)CSCC(C)C)CC2C(C)C)=O)c(C2CC2)n1 22057,C1(C(=O)NC(CC)CO)CCN(CC2(CO)CC2c2cccc(F)c2)CC1 22058,Cc1cncc(C)c1C(=O)NC1CC(C(F)C(N2CC3CC3(CO)C2)=O)C1 22059,C(=O)(C(F)(F)C1=CCOCC1)NCC(CC=C)NC(C1(CF)CC(F)(F)C1)=O 22060,N1(C(C(CNC(CSCC)=O)N(C)C)=O)CC(C)OC(C)(C)C1C 22061,c1(NC2CN(C(C)C3CC3)C(=O)C2)ccc(S(=O)(=O)NCCC(C)(C)F)cc1Br 22062,N1(C(CSC)=O)CC2CC(NC(c3cnsn3)=O)C1C2.c12ccc(cc1)NC2 22063,N1(C(c2c(C)c(F)ccc2Cl)=O)CC2CC3CC2C1C3NC(c1ccn(C)c1)=O 22064,Cc1ccn2ncc(C(=O)NC3CC(C)N(C(=O)CCCc4ccsc4)C3)c2c1 22065,c1(CCNC(c2cccc(NC(=O)NC)c2)=O)c[nH]c2cc(F)c(Cl)cc12 22066,CCC(C)(CNC(c1ccnc(C)c1C)=O)C(=O)NC1(CCF)CCC1 22067,N1(C(=O)NC)CCN(C(C2CC(NC(c3ccc(F)s3)=O)C(O)C2)=O)CC1 22068,CC1CC2(CCN(C(=O)CC3CCCC3)CC2)CN1C(=O)CCCCC(C)(C)C 22069,Cc1cnn(C(C)C(=O)NC2CCC2NC(c2ccn(Cn3cccn3)n2)=O)c1 22070,C1(O)(CC=C)CCN(C(c2conc2CNC(C2CC(=O)C2)=O)=O)CC1 22071,c1(CN2CCC(O)(C(=O)Nc3cc(O)nc(O)n3)C2)ccc([N+](=O)[O-])cc1O 22072,n1(C(C)C)cnc(C(=O)NC(c2ccnn2C)C(=O)NCC2(C)CC2(C)C)n1 22073,c1(C(N2CC(O)(CCNC(C3CCOC3=O)=O)C2)=O)coc2c1CCCC2 22074,C1(C(C)C(=O)Nc2cnns2)CCN(Cc2scnc2Cl)CC1 22075,CN1CCC2CN(C(C3(NC(C4CN(C(N)=O)C4)=O)CCOCC3)=O)CC2C1 22076,C(=O)(CCCC(=O)N1CCN(C(=O)CC2CCCSC2)C(C2CCC2)C1)N(C)C 22077,C1(c2scc(C)n2)COCCC1C(=O)OC.n12ccnc1CN2C.CC 22078,c1(CSCCC)ccc(C(=O)NC2(CNC(C3CCOC3)=O)CCOC2)o1 22079,c1(C(C(=O)NC(CNC(COCCCC)=O)(C)C)O)ccc(F)c(Br)c1 22080,Cc1oc(C(=O)NCC2CC(O)(CNC(c3sccc3Cl)=O)C2)cc1CO 22081,c1(C(=O)NCC2C(NC(c3cc(OC)n[nH]3)=O)C2)c(Cl)cc(C(F)(F)F)cc1Cl 22082,C1(CSC)C(=O)Nc2noc1n2.c1(OC)ccccc1 22083,C(=O)(CCS(N)(=O)=O)NC(CC(C)C)CNC(=O)CCC(=O)NC1CCCC1 22084,C(=O)(CC(C)C1CC1)NC(CN(C(=O)C(C)(C)OCC(F)(F)F)CC)C 22085,c1(C(=O)NC2CN(C(C3(CC)CCOC3)=O)CC(F)C2)c(O)ccc(F)c1F 22086,C(c1c(C)coc1C)=CC(N1C(CCNC(C2(CCCC)CCC2)=O)CCC1)=O 22087,Cc1ncccc1C=CC(=O)NC1(CN(C)C(c2nccn2C)=O)CC1 22088,c1(NC(c2ncnn2C)C)[nH]c(=NCCc2ccncc2Br)nc2scnc12 22089,N1(C(c2nc[nH]n2)=O)CC2CCC1C1CN(C(c3ccn(C(F)F)n3)=O)CC21 22090,C(C(C(=O)NC1COC1)N1CCN(C(c2ccncc2)=O)CC1)(C1CC1)OC 22091,c1(OCC)c(C(N2CCC(NC(=O)Cc3ccc(C)c(Cl)c3)C2)=O)cccc1F 22092,C1(NC(C2CCC(CC)CC2)=O)CCN(C(=O)C(C)(C)COC(C)C)CC1CO 22093,CC(=O)C(C)CC(C)C(=O)N1CCC(C)(C)CC1C(=O)NCC(CO)C(C)(C)C 22094,c1(CN2CCC(C(N3CC4CC4C3)=O)CC2)cccc2ccnn12 22095,C1(CCNC(=O)C=CI)CCN(C(C23CC(CN2C2CC2)C3)=O)CC1 22096,C12(C(=O)OCC)C(NC(C34CC(C)(C3)OC4(C)C)=O)C3CCC1C2C3 22097,Cc1cccc(C)c1C(N1CCC(C)C(CC(N2CCSC(C)(C)C2)=O)C1)=O 22098,c1(CC)nc(C(N2CCCC2CC(C)(C)C)C(=O)NCCC#N)cs1 22099,C(C(C)(C)CC(=O)NC(C)(C)CC(N1CC2(C1)CC2(F)F)=O)OC(C)=O 22100,c1(OC)cc(Br)c(C(N2CCCC2)CNC(=O)C(=O)c2ccco2)cc1O 22101,C1(CC=C)(NC(c2cnc(CC)s2)=O)CN(C(c2cc(C(F)F)cs2)=O)C1 22102,Cc1cc(C)c(CN2CCC(N(C(=O)C(F)(F)Cl)C)C2)cc1C 22103,c1(CC)ncc(C(=O)NC2CCCN(C(=O)CCC(F)(F)F)C2CC)c(C)n1 22104,c1(CCC)onc(CN(C)Cc2cccs2)c1CC 22105,C1(NC(=O)CC(F)F)CC2CC1CN(C(c1cnnc(O)c1)=O)C2 22106,Cc1cccc2c1CCC2NC(c1cnc2n1C(C)CCC2)=O 22107,N1(C(CC2C(C)(C)OCC2)=O)CC2CCC(C1)N2C(C12CCCN1CCC2)=O 22108,CC(C)CC(CNC(=O)CC1CCC(=O)C1C)C(=O)NCC(C1CC1)N(C)C 22109,Cc1cc(C(=O)N(C)Cc2ccn(C)n2)nn1CC(F)(F)F 22110,c1(C(N2CC(N(C(C3CN(CC(C)C)C3)=O)C)C2)=O)ccc2c(O)ncnc2c1 22111,N1(C(c2[nH]cc(C)c2)=O)CCN(C(C23CCCC2C3(F)F)=O)CC(O)C1 22112,c1(C(=O)NCCCCC2CN(C(C(C(C)O)(F)F)=O)C2)cc2ccsc2n1C 22113,c1(C(=O)NC)ncoc1C1CN(N(C(C)C(=O)OC)CC)C1.C1(C=O)CCCS1 22114,N1(C(C2(CC)CCC2)=O)CCC2(CCN(C(C3CCC(C4CCCO4)O3)=O)C2)C1 22115,C=C(Cl)CCC(=O)NC(C)C(C(C)C)NC(=O)CC=CCc1ccccc1 22116,C(=O)(C1CCc2nccn21)NC(C)C(=O)NOC1CCCCO1 22117,C(N=c1[nH]c(N2CCC(c3nncs3)C2)nc(=N)[nH]1)c1cn(CC)nn1 22118,C1(CC)CN(C(C2(O)CC3CC2C3)=O)CC2(CCCOC2)O1 22119,C12(NC(C(C)=CC3CC3)=O)CCC1CN(C(c1ccsc1C)=O)C2 22120,Cc1cc(NCCCCC(C)NC(c2c(F)cccc2F)=O)n2nc(C)nc2n1 22121,C(=O)(CS(=O)(=O)N1CCOCC1CNC(c1cccnc1C)=O)OCC 22122,c1(N2CCOCC(C(N3CC4CC3CS4=O)=O)C2)ncc2[nH]ncc2n1 22123,c1(C(CC)C(=O)NCC(C)N(C)C(c2ccn(C)c2)=O)ccc(Cl)cc1 22124,CC1CCC(NC(=O)Cc2cn[nH]c2)CN1C(c1ccc(O)nc1Cl)=O 22125,Cc1cc(NC(C23CC2CN(C(c2ccno2)=O)C3)=O)c(F)c(Br)c1 22126,C1(NC(C2C(=C)C2)=O)COC2(C1)CN(C(c1cccc3nncn13)=O)C2 22127,N1(C(C)=O)CCC(CNC(c2cccc(NC3CC3)c2)=O)C(c2ccccc2)C1 22128,C1(CC(=O)NCC(CC=C)NC(=O)Cn2cnc(C)cc2=O)CCCCC(=O)N1 22129,c1(CNC2CCC(C(=O)NCc3ncn(C)c3)CC2)c(Br)ccc(Cl)c1F 22130,N1(Cc2cc(Cl)c(Br)nc2)CCC2(CCSCC2)C1 22131,c1(C(=O)NC2(C(=O)OC)CC2(C)C)cc(Br)ccc1Cl 22132,C(=O)(CS(=O)CCC(F)(F)F)N1C2(CNC(CC=CCC)=O)CCC1CC2 22133,c1(C2C(C(=O)NCC(C)(C)C(C)(C)C)C2)c(F)cccc1F.C(=O)(CCC(=O)O)N 22134,N1(C(C(CCCC)C)=O)CCC2CCCC12C(=O)NCC1CC2(CCC2)C1 22135,c1(C(=O)NC2CCN(C(c3cccnc3)CC)CC2)cnc2onc(C)c2c1 22136,C1(C(N(CCCNC(c2c(OC)nsc2)=O)C2CC2)=O)CCSC(C)C1 22137,Cc1cnc(C(N2CCCC(CN(C)CCc3cnn(C)c3)C2)=O)cn1 22138,c1(C(N(C)C2CC2)=O)ccc(NC(C2CCCN2C(=O)C2CC2)=O)cc1 22139,C(C)(C(=O)N1CCC(N(CCO)C(C2CC(C)C2)=O)CC1)(C(C)C)OC 22140,C(CCN=c1cccc(S(=O)(=O)N(C)Cc2cccc(F)c2F)[nH]1)OC(C)C 22141,C(=O)(CCCCC(=O)NOC(C)(C)C)N1CCC(C(=O)OC)(NC2(C)CSC2)C1 22142,C(=O)(C1=CCCOCC1)NC1CCCC(CC(=O)NOCCCC2CC2)C1 22143,Cc1cc(C)c(CNC(=O)C(c2ccoc2)NC(c2cccc(O)n2)=O)cn1 22144,c1(C(=O)NC2(CNC(C(CC)(C)C)=O)CC2)c(C)nn2c1NCCC2 22145,C1(N(C(C2(SCC)CC(O)C2)=O)C)CC2CCC(C1)N2C(=O)CCCCN(C)C 22146,N1(C(CCC2C(=O)NC(=O)N2)=O)CCC(NC(c2cnccn2)=O)C2CC12 22147,C1(C(=O)NCC(C)N(C(c2cc(C)n(C)c2C)=O)C)CN(C)CCN(C)C1 22148,N1(C(c2c(C)snc2)=O)CCC(NC(=O)CC(C)c2cccnc2)C(F)(F)CC1 22149,C1(C(=O)Nc2ccc(OC)cc2)CCCCC1(C)NC(=O)CCOC1CCCC1 22150,c1(C(N2CCN(S(CCCC)(=O)=O)CC2)=O)cc(NC(C)=O)ccc1C 22151,C#Cc1ccc(C(N2CCCC(CC(N)=O)C2)C(=O)NCCC2CC2)cc1OC 22152,c1(C(C)C)conc1C(=O)N(C)CC=CC(N1CCCC1C(O)CO)=O 22153,N1(C(C2C3CN(C(CCC(C)OCC)=O)CC32)=O)CCCC12CCCC2 22154,Cc1ccc(C2C(=O)N2)cc1.C(=O)(CCCC1CC1)NCC(O)COCC1CC1 22155,c1(CC(=O)NCC2C(NC(Cc3c(C)cccc3)=O)C2)ccc2nonc2c1 22156,N1(C(C2C(CC)N(C(=O)C(CN(C)C)N(C)C)CC2)=O)CC(F)CC(F)C1 22157,C1(N(CCOC)C(c2ccncc2)=O)CCN(C(=O)C(C)(C)n2cccn2)CC1 22158,c1(C(=O)OC)cccc(C(=O)N(N2CCN(Cc3nc(Br)cs3)CC2)C)c1 22159,C1(CNC(N(c2ccccc2)CCNS(C)(=O)=O)=O)CCC(F)C1 22160,C1(Nc2ccc(COC(C3CCOCC3)=O)cc2)CCC2CC1CN2 22161,c1(CC(=O)NC2CCN(C(=O)C(=O)NCC3CC3)CC2)ccc2c(c1)CC2 22162,c1(C(N(C2CCN(C(=O)Cc3cnn(C4CC4)c3)C2)CC)=O)cc(OC)ncn1 22163,c1(C(N2C(C)C(C)N(C(=O)CN3CC4CC4C3)CC2)=O)cccc2c1CCC2=O 22164,c1(C(=O)NC2(C(N3CC(C)(CC=C)C3)=O)CCCCC2)cnc(C)c(C#N)c1 22165,N1(C(Cc2ccc(C)s2)=O)CCN(C(=O)C=Cc2ccoc2)C(C)C1C 22166,C(=O)(C(C)CCCC(C)C)N1C(CCNC(=O)C=C(C)C)CC(OC)C1 22167,c1(CC)cc(=NCC2(C)CCC(NC(c3ccon3)=O)CC2)[nH]cn1 22168,C1(NC(c2ccnc(C)c2N)=O)CN(C(=O)CCCF)C2(CCCCCC2)C1 22169,c1(C(=O)NCCC(C(C)C)NC(=O)CC2NC(=O)NC2=O)ccc2[nH]ccc2n1 22170,N1(C(C(n2ccc(C3CC3)n2)C)=O)CC2(C1)CN(C(=O)C(C)CF)CC2CO 22171,C1(CC(=O)NCC(O)CNC(=O)CC2CCCC2)(CC)CCOCC1 22172,c1(C(N2CCCC(c3cn(-c4ccc(Cl)cc4)nn3)C2)=O)cc2scc(Cl)c2[nH]1 22173,C1(C(N2CC(F)CC(OC)C2)=O)CCN(C(C2CCCCO2)=O)C(C)(C)C1 22174,c1(C(=O)OC)cnc(C(N2CCC(CC(=O)NC(C3CCOCC3)C)C2)=O)cn1 22175,N1(C(C2CCN(C)C2=O)=O)C2CCC1CN(C(=O)C1=CCCS1)C2 22176,C12(CNC(CC(C)C3CCCO3)=O)CC(NC(c3ccc(O)nc3)=O)(C1)C(C)O2 22177,CCCCCC(C)CC(=O)NCC1C2CN(C(=O)C(c3ccc(C)o3)C)CC12 22178,N1(C(c2cc(C(=O)OC)on2)=O)CCC2(CC(NC(c3n[nH]cc3C)=O)C2)C1 22179,CC1OCCCC1C(=O)NC(C)CNC(c1cccc(OC(C)(C)C)c1)=O 22180,C1(O)(CNC(NC(C)C)=NCc2ccnn2CC2CCCO2)CCC(C)CC1 22181,C1(C)(C(N(C2CCC(OC)C2)C)=O)CCN(C(=O)CCc2cnc(C)o2)CC1 22182,N1(C(CNC(C2C(C)C2)=O)=O)CC(C(=O)NC2(CO)CC(CO)C2)CC(C)(C)C1 22183,C(C(CNC(C1C(C)C1C)=O)CO)NC(CC1(OC)CC1)=O 22184,CC1c2cc(CNC(=O)C(=O)N(c3ncnc4c3ccn4C)C)ccc2OC1C 22185,C(=O)(C(C)(C)CC(=O)NC(C)C(C)NC(c1cc(=O)cc(Cl)[nH]1)=O)OCC 22186,C1(NC(C2CCC(=O)N2)=O)COCCN(C(C2CCCCS2(=O)=O)=O)C1 22187,c1(CN2CC(F)(C(=O)NCCc3ccc(OC)cc3)C2)cc(F)cc(Br)c1Cl 22188,C(=O)(CC(F)(F)C(F)F)N1CCC(C(F)F)(CNC(C2(C)CCNC(=O)C2)=O)C1 22189,N1(C(c2c(CC)csc2)=O)CC2CCCC2(NC(C2OCCC2(C)C)=O)C1 22190,N1(C(c2ccc(SCC)nc2)=O)CCC(OC)C(C)C1 22191,Cc1cn(C(C)(C)C(=O)NCC(=C2CN(C(c3cc(C(N)=O)[nH]n3)=O)C2)F)cn1 22192,C(C(=O)NC1CCC(NC(C2(N3CCCC3)CC2)=O)CC1)(C(C)(C)C)NC(C)=O 22193,C1(CNC(CCC)=O)CC2(CCOCC2)CN1C(=O)CCSCCCC 22194,S(=O)(=O)(CC(=O)NC1(C)CC(C(=O)NC2CC23CCC3)C1)NCC 22195,N1(C(C(C)NC(=O)NC)=O)CCN(C(=O)C(C)=C(C)C)CC1CC1CC1 22196,Cc1cc(C(N2CCOCC2CS(C)(=O)=O)=O)ccc1C#N 22197,N1(C(c2c(CC)oc(C)c2)=O)CC(Nc2ncncc2Cl)CC(F)C1 22198,C(=O)(C(C)S(C)(=O)=O)NCCN1CCN(C(c2c(OCC#C)nccc2)=O)CC1 22199,c1(C(N2CCN(C(=O)CC3CCN(CCF)C3)CC2)=O)c(F)ccnc1Cl 22200,C1(S(N)(=O)=O)(C(=O)NCC(C)N(C)C(c2cc(Cl)cn2C)=O)CCC1 22201,c1(C(=O)NCC2CC(F)CN2C(C2CCCC23CC3)=O)cnn2cnnc2c1 22202,Cc1nc(C(C)NC(c2cccnc2-n2nccn2)=O)c(C)o1 22203,c1(CCC)c(C(N2CCN(CCOCCC(C)C)CC2)=O)nnn1CC 22204,C1(N(C)C(C2CCOC2)=O)CCCN(C(c2cc(O)ccc2Br)=O)CC1 22205,C(=O)(C(O)CCC(F)(F)F)N1C(CN(C(=O)CCc2ncc(C)[nH]2)CC)CCC1 22206,C1(NC(C2OCCC(C)(C)C2)=O)CN(C(=O)CC2CCC(C)(C)C2)CC12CCC2 22207,N(C1CCC(NC(C2(n3ccnn3)CC2)=O)c2ccccc21)C(C(CCC)C)=O 22208,CC(C)C(CC(=O)NC1CCC(C2CC2)C1)NC(=O)CC1C(C)(C)C1(C)C 22209,C1(NC(CC(CCC)O)=O)CCCCN(C(c2cccc3cnsc23)=O)CC1 22210,c1(-c2nn(C(C)C3CC3)c(C(OC(F)(F)F)F)n2)ccc(F)c(Cl)c1 22211,C1(CCNC(Cn2ccc(C)n2)=O)CCN(C(C2CC2C(C)(F)F)=O)CC1 22212,C1(C(=O)NC(c2cc[nH]n2)C)CC2CCCC2N1C(C1CC12CCCC2)=O 22213,N1(C(CC2(CSC)CC2)=O)CC2CCN(C(c3cncc(O)c3)=O)CC(C2)C1 22214,C1(NC(CCC(N)=O)=O)CC2(CCN(C(c3cncc(OC(F)F)c3)=O)CC2)C1 22215,c1(CC(=O)NCC(C)CN(C(=O)Cn2cnc(C#N)n2)C)cc(F)ccc1F 22216,c1(NC(C2(c3ccccc3)CCC2)=O)cncn1C(F)(F)F 22217,N1(CC(N2CC(CC(C)NC(C3C4CNC(=O)C34)=O)C2)=O)CCN(C2CC2)C1=O 22218,CC#CC1CCN(C(c2c[nH]nc2CNC(=O)C(O)C(C(C)C)OC)=O)CC1 22219,C1(CNc2ccccc2)CCN(c2ccnc(NCc3ccc(Cl)o3)n2)CC1 22220,N1(C(C(C2CC2)OCC)=O)CCC(C)(NC(=O)Cc2ccn(C3CCCC3)n2)C1 22221,c1(OC)cccc(F)c1C(=O)NCC1CN(C(=O)Cc2csc(C)n2)CCC1C 22222,C(=O)(C(O)CC(F)(F)F)NCC1N(C(CSc2nc(C)[nH]n2)=O)CCCC1 22223,C1(CCNC(c2c(C(C)C)noc2)=O)CCCCN1C(=O)C=CC1CCOCC1 22224,c1(C(=O)NCC(CNC(C2CC(C#N)C2)=O)F)nc2ncccn2n1 22225,C1(C(N2CCC(C(=O)OC)C2)=O)(OC)CCN(C(C2CC(F)CN2C)=O)C1 22226,Cc1c(C(N2CCOC(C(=O)NCC(C3CCCC3)C)C2)=O)cnn1C 22227,C1(NC(C(C)C2CCCC2)=O)CCCCCN(C(c2cn3ccnc3cn2)=O)C1 22228,c1(OC)ccc(C=CC(=O)NC2CCCCC2CNC(C2CC2C)=O)c(OC)c1 22229,Cc1cc(NC(=O)NC2CC2(F)F)cc(F)c1Br 22230,Clc1cc2c(cc1Br)CCN(c1nc3c(Br)csc3s1)C2 22231,c1(CN(C(=O)CN2Cc3ncnc(N(C)C)c3C2)C)cccc2ccccc12 22232,c1(C(C(=O)NCCSC)N(CCC(C)(C)C)C)ccnc(Br)c1 22233,N1(C(C2CC(=C)C2)=O)CC(CNC(c2ncccc2C(C)=O)=O)C(O)C1 22234,C1(CC=C)(NC(C2CCCN2C(C)C)=O)CCCN(C(c2cc(OC)cs2)=O)C1 22235,C12(CNC(CCOCCC)=O)CC1CN(C(=O)C(C)Oc1ccccc1OC)C2 22236,Nc1cc(C(=O)NCCNC(=O)C(c2ccccc2)C2CC2)cc(F)c1Cl 22237,N1(C(c2c(CC)c[nH]n2)=O)CCN(C(c2cnc(C)cn2)=O)CC1CCOC 22238,CCC(CCC(=O)N(C(C)CC(N)=O)C)NC(C1(C)CCCCC1)=O 22239,C#Cc1cccc(C(=O)NCC2COC(CNC(=O)C(C)(C)c3ccsc3)C2)c1 22240,C1(NC(=O)Nc2ccc(OCCCC)c(Cl)c2)CCC(S(C)(=O)=O)C1 22241,CCCCC(CNC(=O)C(C)(C)NC(=O)C1CC1)OC.C12=CC(=O)N(CC1)CC2 22242,c1(OC)cc(C(N2CCN(C(C3CCCCN3C(C)=O)=O)CC2C)=O)cnc1C 22243,c1(CNC(C2(C(C)NC(CCOC(C)=O)=O)CC2)=O)n[nH]cc1C 22244,N1(C(CCc2cc(OC)no2)=O)CCC(CO)(CNC(=O)C(C)C(F)F)C1 22245,c1(-c2c(F)cc(C)cc2F)ccc2c(C(=O)NCC(C)(C)C(N)=O)nn(C)c2c1 22246,c1(C(N(C(CNC(c2ccc(C(OC)OC)o2)=O)C)C)=O)occ2c1CCOC2 22247,CON1CCC(NC(C2(NC(=O)COCC3CCOC3)CC2(C)C)=O)CC1 22248,c1(C(=O)NC2CC(NC(C3(CC)CCNC3=O)=O)C2)cn2cccc(Br)c2n1 22249,c1(C(=O)NCCCC(C)NC(c2c[nH]ccc2=N)=O)cnc(C(F)(F)F)[nH]c1=N 22250,Cc1cc(C(=O)NC2CC(C(=O)N(CCC(C)(C)C)C)C2(C)C)c(C)s1 22251,CC(CNC(=O)C(O)Cn1cncn1)C(F)C(=O)NCC(F)CO 22252,C(=O)(CS(=O)(=O)C(C)C)N1CCC(N(C(=O)CCn2ccnc2C)CC#C)CC1 22253,c1(NCC2(C(C)C)CC2)[nH]c(=NC2CC3(C2)CC3(C)C)nc2c1cnn2C 22254,N1(C(c2ccn(C3CC3)n2)C(=O)NC(CC)C)CCc2c(cc(C#N)n2C)C1 22255,C1(CC(=O)NCC(C)(CO)NC(=O)C=CC2CCCO2)CCCCCCC1 22256,CC(c1ccc(F)cc1)=CC(N1CC(NC(c2c[nH]nc2[N+](=O)[O-])=O)C(C)C1)=O 22257,N1(C(=O)NC2(C)CCCC2)CCCC2CN(C(c3cc(N)ccn3)=O)CCC12 22258,C(=O)(C1=CC2CCCC12)NC1CCC(NC(CSCCC(C)C)=O)C1 22259,C1(C(N(C)CCOCCN(C(=O)C(F)(F)c2cscn2)C)=O)CCCC(F)C1 22260,CC1CC(C2CN(C(C3CCC3NC(c3ccnnc3)=O)=O)C2)=NO1 22261,C1(n2ccc(C)n2)CCC(N=c2cc[nH]cc2S(=O)(=O)NCC=CCl)C1 22262,N1(C(c2c(C)nn(C)c2)=O)CCC2CN(S(=O)(=O)c3ccccc3F)CC2CC1 22263,CC1(Cn2cc(NC(=O)NC3C4COC(C)(C)OCC34)cn2)CCC2(CC1)CC2 22264,c1(OCC)nc(Cl)ccc1C(N1CC(NC(c2cc(C)c(C)nn2)=O)C(C)C1)=O 22265,c1(C(=O)NCC(c2ccccc2F)(F)F)c[nH]c2cc(Cl)ccc12 22266,N1(C(CCCC(C)NC(c2ccc(C)c(C)n2)=O)=O)CC2(C)CC1CCO2 22267,Cc1cnccc1C(C)C(N1CC(NC(=O)CCc2cncnc2)CC1C)=O 22268,CC1(F)CN(C(=O)C=CBr)CCN(C(C2CC(C(F)(F)F)CO2)=O)C1 22269,N1(C(C(C)C2CCCO2)=O)C(CNC(c2n[nH]cc2Cl)=O)CC2COCC12 22270,c1(C(=O)NC2CCC3CCC23)n[nH]c2c1CN(C(c1cnc(Cl)s1)=O)C2 22271,CC1(C)CC(O)CCN(C(c2cc(F)sc2)C(=O)NC2CCOCC2)C1 22272,c1(C(C(=O)NC2CC(CCNC(c3ccsc3)=O)C2)SC)ccccc1 22273,c1(OCC(=O)NC2CN(C(=O)C(F)F)CC2C(F)F)ccc(C2CCC2)cc1 22274,CC1CCN(C(C2CC(c3ccccc3)O2)=O)CCN1C(c1ccccn1)=O 22275,N1(C(C(C)N(C)C(C2CC2(C)C(F)F)=O)=O)CC(CN(C)C)C(O)C1 22276,C1(N(C(C(COCC)C)=O)C)CN(C(=O)CNS(C)(=O)=O)CC1F 22277,n1(C(C)C)cc(Br)cc1C(=O)NC(C)CCNC(C1(O)CCSC1)=O 22278,Cc1c(C(N2CC3(C2)CN(c2nc(Cl)ncc2F)C3)=O)cccc1O 22279,c1(C(=O)NCC2N(C(C3C(C)OCC3)=O)CC2)c(N)cccc1Cl 22280,c1(C2(NC(C(C)NC(COC)=O)=O)CC2)ccc(C)cc1.C12CC1CNC2=O 22281,CCCCC(C(=O)NCC1CC(C)=NO1)NC(=O)Cc1cnns1 22282,C1(C(=O)NC(C)CN(C)C(c2ccccc2)c2ccccc2)(OC)CC(C)(C)C1 22283,CCC(C)CC(C(=O)N1CC(OCCF)C1)NC(=O)C1=CCOCC1 22284,N1(C(Cc2cccc(OC)n2)=O)CCC(C)(C)C(NC(c2cccnc2S)=O)C1 22285,c1(C(NC(NCC(C2COC(C)(C)O2)O)=NCC2CC2)C2CC2)ccc(Cl)cc1F 22286,Cc1ccc(C=CCNC2CCN2C(=O)OC(C)(C)C)cn1 22287,CC(C(C)CO)NC(=O)CCN(C(c1cnns1)=O)C1CC1 22288,Cc1cc(C(=O)NC(CNC(C2(S(C)(=O)=O)CCCC2)=O)C2CC2)ncc1C#N 22289,c1(CC(=O)NC2COCCN(C(=O)CC3(O)CCOC3)C2)nc2c([nH]1)CCCC2 22290,Cc1cc(NC(=O)C(C2CCOCC2)O)ccc1NC(=O)C(N1CCCC1)C1CC1 22291,C1(C(=O)NCC(C)(C)OCCNC(C(C)Cn2ccnc2)=O)NC(=O)OC1C 22292,N1(C(Cn2cc(C(C)O)nn2)=O)CC(NC(c2cccn2C)=O)C2CCCCC12 22293,C=CCC(CNC(=O)C(C)OCC1CC1)C(=O)NC1(CO)CC2CCCC12 22294,N1(C(COC(C)=O)=O)CCC2(CC1)CC(N1CCC(F)(F)C(O)C1)C2 22295,c1(C(C)=O)cc(C(=O)NC2CC(C)(NC(c3sc(C4CC4)nc3C)=O)C2)c(C)o1 22296,C(C(F)(F)CNC(=O)CCCNC(=O)CC1(C)CC1)OC 22297,c1(C(=O)NCCC(C)NC(=O)C(=Cc2c[nH]cn2)F)cc2c(Cl)cc(Cl)cc2[nH]1 22298,CC(C)C(C)C(CNC(c1cccc(C2(F)COC2)c1)=O)NC(=O)C1=COCC1 22299,OC1(F)CCN(C(=NCC2CC23CCSCC3)NC2CC2)CC1 22300,C1(OC)CN(C(=O)CC2CCOC2=O)CC1NC(C1(NC2CC2)CCC1)=O 22301,c1(OC)cc(C)c(C(=O)NC(CNC(=O)Cc2cnccc2C)C2CC2)c(C)c1 22302,Cc1nn(C)c(C)c1C(N1CCCC(C(=O)NC2CC(=O)N(C)C2)CC1)=O 22303,Cc1cc(CC(=O)NCC(C)(CO)NC(=O)CNC(=O)CCCCl)n[nH]1 22304,N1(C(C=CCCC)=O)Cc2occ(C(N3CCC3C(C)O)=O)c2C1 22305,c1(N2CC(C)(NC(C(C(C)O)C)=O)C2)nc2cc(Cl)cc(Cl)c2o1 22306,CC(C)(CO)C(=O)N1CCC(C)(CNC(C2CCOC2c2ccncc2)=O)C1 22307,N1(C(=O)CCc2sccc2Br)CCN(c2ccc(-n3cc(CO)nn3)cc2)CC1 22308,CC1CN(C(c2ccc(OCC(N)=O)cc2)=O)CC1NC(=O)CCC1CC1(Cl)Cl 22309,C1(NC(C(CCOCC)C)=O)CN(C(c2cc3ccccc3[nH]2)=O)CC(C)(C)C1 22310,c1(NC(c2c(Cl)ccc(OC)c2)=O)ccc(S(C)(=O)=O)cc1Cl 22311,n1(CC(=O)NCC2CC2NC(C2CC2c2cccc(Cl)c2)=O)cccnc1=O 22312,C12(C(=O)NCCCc3cc(C)no3)CCCC1CCN2C(c1n[nH]c(=N)[nH]1)=O 22313,c1(C(=O)NCc2cn(C3CN(C(c4n(C)c(O)nc4)=O)C3)nn2)ccc(O)c(Cl)n1 22314,c1(C(N2CCC2CN(C(C2CCCC(=O)N2)=O)C2CC2)C)ccc(F)cc1 22315,N1(C(c2c(SCC)cncc2)=O)CC2CC(NC(c3c(C)nn(C)c3C)=O)C2C1 22316,c1(C(=O)NCCC(C)NC(C(OC)OC)=O)ccc2cccnn12 22317,C1(C(=O)NC2CCN(C(c3ccc(C)cc3N)=O)C(C)C2)(OC)CCS(=O)(=O)C1 22318,N1(C(CCC(C)O)=O)CC(NC(c2coc(C3CCC3)n2)=O)CC2(CC2)C1 22319,N1(C(c2cn(CC)nc2C)=O)CC(NC(=O)Cc2ccns2)C(N=[N+]=[N-])C1 22320,Cc1ncnc(N2CC3CC3(CNC(c3cc(F)ccc3Cl)=O)C2)c1Br 22321,C(c1cnc(C)s1)=CC(=O)NCC1(CNC(C(C=CCCC)O)=O)CC1(F)F 22322,CC(=Cn1ccnn1)C(=O)N=S1(=O)CCC2(CC1)CN(C(C1CC1Cl)=O)CCO2 22323,c1(NC(CC)C)ccc(S(=O)(=O)NCCc2ccsc2)cc1Br 22324,Cc1nn(C)c(C)c1NC(c1nc(Nc2nccc(C#N)n2)cn1C)=O 22325,C1(CC)CCCC(CNCC2(Cn3cnc(C(N)=O)c3)CC2)CC1 22326,C1(O)(C(C)NC(=O)CNC(=O)Nc2nc[nH]n2)CCN(C(=O)S)CC1.C(C)(C)C 22327,CC1OCCC1CN(C(=O)CNC(c1cscc1Cl)=O)C 22328,c1(C(=O)NC2C(OC)CN(C(C3CCN(C4CC4)C3=O)=O)C2)ccc(F)cc1O 22329,N1(C(C=C(C)Cl)=O)CC2C(NC(=O)CCSc3ccccn3)C2C1 22330,C=CC(C)(C)CC(=O)NC1COCCN(C(C2(c3ccccn3)CC2)=O)C1 22331,Cc1c(C(N2CC3C(NC(=O)COC(F)(F)F)CC3C2)=O)cccc1F 22332,N1(C(c2c(C)nc(C(C)C)o2)=O)CC(NC(c2ccnc(CO)c2)=O)C2CC2C1 22333,C=CCC(CC(=O)NC(CCC)c1nn[nH]n1)NC(=O)CCCF 22334,C(=O)(CS(=O)(=O)NCC1CC1)NCCCN(C(=O)C(F)(F)c1cncs1)CC 22335,N1(C(C2CC(C#C)(O)C2)=O)CCC(O)C(N(C)C(c2cnsn2)=O)C1 22336,c1(C(=O)NCC2CC(NC(c3cccnn3)=O)C2)cnc(S)nc1 22337,C12(CNC(COCC#C)=O)CCC(CC1)N2C(C1(C)CNC(=O)C1)=O 22338,n1(CCCC)c(C)cc(C=C(C#N)C(=O)Nc2c(C(N)=O)noc2C)c1C 22339,N1(C(=O)C=Cc2ccccc2)CCC(C(=O)NCCCNC2COC(=O)C2)C(O)C1 22340,c1(CC(=O)NCCN(C(c2c(C)cc(SC)s2)=O)C(C)C)ccc2c[nH]nc2c1 22341,N1(C(CC)CC)CC2C(CNC(=O)OCC)(C1)C(F)(F)C2.C(C)(C)C 22342,CCCCCCC(F)C(=O)NC1CCC12CCN(C(=O)CCSCC(N)=O)CC2 22343,N1(C(C(F)=CC)=O)CCC(NC(=O)CC2CCCN2CC)C1 22344,c1(C2(CNC(=O)Nc3cc(C)c(F)cn3)CC2)ccc2c(c1)OCCO2 22345,C1(C(N2C(C(N)=O)CC2)=O)C=CCN(C(=O)CC2OCCCO2)C1 22346,C(=O)(C(C(C)(C)O)Nc1ccc(-c2cccnc2C#N)cc1)OC(C)(C)C 22347,c1(N2CCCC3(CC(NC(=O)C4CCCc5ccnn54)C3)C2)nc2ncc(Cl)cc2s1 22348,N#Cc1cc(F)ccc1C(N1CCN(C(C2CCSCC2)=O)C2CC12)=O 22349,Cc1ccc(CC(N2CCCC(O)(CNC(=O)C(C(C)O)N(C)C)C2)=O)cc1C 22350,N1(C(c2c(C)ccnn2)=O)CCN(C(=O)C(C)(F)C(C)(C)F)CC12CCC2 22351,C(=O)(CCC(CC)NC(=O)C1CC1)NC1C(C#C)CCC1 22352,n1(CC)cc(CC(=O)NC(C(=O)NC(C)CC2CCC2)C2CCOC2)cn1 22353,CC(C1CCCCC1)=CC(=O)NC1CN(C(=O)CCOC2CC2)CCC1C 22354,c1(C(=O)NC2CC(F)(CNC(C(n3ccc(C)n3)(C)C)=O)C2)cccn(C)c1=O 22355,C(C)(CNC(c1ccc(O)c(C)c1)=O)(CC(C)C)NC(C1C(C=C)CC1)=O 22356,n1(CC(=O)NC2CCC(NC(C(CC)O)=O)C2)nc(-c2ccccc2)oc1=O 22357,c1(CNC(c2cnc(S)nc2)=O)ccc(C(=O)NCCC(O)CCO)cc1 22358,c1(CNC2(CCC)CCNC2=O)ccc2n[nH]cc2c1.C12CC(CCO1)NC2=O 22359,N1(C(C(CC#C)(C)NC(=O)CCC#CC)=O)CC2(CNC(=O)C2)C1 22360,N1(C(C=C(C)C(C)C)=O)CCC(O)(C(C)NC(=O)CCOC(C)CC(C)C)CC1 22361,C1(C(=O)NC(CC)C(C)(F)F)CN(C(=O)C(C)O)CC1C1CC1 22362,c1(C(=O)NC2(C)CC(NC(=O)CC3COC4CC3C4)C2)cc([N+](=O)[O-])ccc1Cl 22363,C(C(C)(C)C(=O)NCCC(C)CCNC(=O)C=C1CCCC1)OCC 22364,CC1(C)CN(C(=O)C=CC=CCO)CC(CNC(=O)CC2CC3(CCC3)C2)O1 22365,Cc1ncc(Cl)c(C(N2CC3C(CNC(=O)C(C)(C)O)C3C2)=O)n1 22366,N1(C(C2(F)CCN(C(C3CCN(CC)C3)=O)CC2)=O)CC(C)N(C)CC1C 22367,c1(C(N2CC(C(=O)NC(c3ccc(OC)nc3)C)OCC2)=O)cccc(C#N)c1 22368,c12cc(c(C)o1)S(=O)(=O)NC2=O.N1(CCC)C(=O)CCC1C(=O)NC 22369,C(=O)(C1=NN2CCCN=C2N1)N(C1CN(C(CN(CC)CC)=O)CC1(C)C)C 22370,C1(CNC(C(CC)(C)C)=O)C(O)C(O)CN1C(=O)C=Cc1ccnn1C 22371,c1(CC)nn(C)c(NC(C2C3CN(C(=O)CCS(=O)(=O)N(C)C)CC23)=O)c1Cl 22372,c1(C(=O)NC2C3CN(C(C4(CF)CC4(F)F)=O)CC23)cccc2cnccc12 22373,C1(C2CC2)(C(=O)NC2C(C=C)COC2)CN(C(C23CCC(C2)C3)=O)C1 22374,C1(NC(c2cnc3cccnn23)=O)CCc2nnc(C(F)(F)F)n2C1 22375,N1(C(CNC(C(C)(C)C)=O)=O)CCC2CCCC12C(N1CCCC(C)(CO)C1)=O 22376,Cc1nsc(N)c1C(=O)NC1CCCC(CNC(=O)C(F)(F)c2ncccn2)C1 22377,C1(CCCNC(=O)CSc2cccnc2)CCCCN1C(c1cccnc1)=O 22378,c1(CC(N2CCC(N(C(CC(CC)OC)=O)C)C2)=O)c(F)cccc1Cl 22379,C1(CC(=O)NCC(C23CCC(CC2)C3)NC(c2ccon2)=O)CCCNC1=O 22380,CC1CN(Cc2ccccc2Br)CCN1C(C1CC=CCO1)=O 22381,C1(C)(CCC(=O)NCCC)CN(C(=O)CC2CC2(C)C)C1.c1nocc1C(C)C 22382,C(CNC(C1CC1c1ncc[nH]1)=O)(CC(=O)N1CCOC(C2CCC2)C1)OC 22383,N1(C(C(CC)OC)=O)CCOC(C(=O)NCC2(F)CC(CO)C2)CC1 22384,CCC(C(=O)OC)C(=O)NC1CC=C(C(=O)NCCc2nc(C)no2)C1 22385,c1(NC(CC(=O)N2CCCC2)c2cccnc2)ncnc2[nH]cc(Cl)c12 22386,Cc1ccc2c(C(N3CC(CNC(c4ccc5nc[nH]c5c4)=O)C3)=O)n[nH]c2c1 22387,C1(COC)(CNC(=O)CC#N)CCN(C(=O)Cc2ncccc2C)C1 22388,c1(C(=O)NCCC2(O)CN(C(C34CCCC3CC4)=O)C2)cnc2n1CCOC2 22389,S(=O)(=O)(CCN=c1ccnc(NCC(c2nc(C)cs2)(C)C)[nH]1)NCC 22390,N1(CCCC)CCCC(NC(c2ccc(C(C)C)cc2)C(N)=O)C1 22391,C(=O)(C1=CNC2=NCCCC2=C1)N1C2C(NC(c3ccc(C)o3)=O)CC(CC2)C1 22392,c1(OCOC)cccc(C(=O)NC(C)CNC(=O)C(F)C(C)C)c1 22393,Cn1cc(C(N2CCC(CNC(c3nocc3C3CC3)=O)C2)=O)nc1C(F)F 22394,N1(C(CNC(C2C(C)C2)=O)=O)CCCC1CC(N1CCC(OCC2CCC2)C1)=O 22395,c1(C(=O)NC(C)CNC(=O)CCC2CCCC2)ccc2cccnc2n1 22396,C(=O)(C1=C(Cl)CCC(C)C1)NCC1(NC(C2CCCC(C(=O)OC)C2)=O)CCC1 22397,C1(NC(=O)CC2CC(CF)C2)CCCC(C(=O)NCC=Cc2cccc(F)c2)CC1 22398,c1(CC)nc(=NCC(C)(C(C)C)OC2COC(C)C2)s[nH]1 22399,CC(C(=O)N1CCC(C(CO)NC(=O)C(C)(F)c2ccon2)CC1)S(N)(=O)=O 22400,N1(C(c2cn(CC)nn2)=O)CC2(CCC2NC(=O)CC2CC3(CCC3)C2)C1 22401,Cc1ccc(C2(C(N3CCC(NC(C4CC4C#N)=O)C3)=O)CCOCC2)cc1 22402,C1(=O)C(CC(F)F)NC(=O)CC2CN(C2)CC2CCCN1C2.CCOCC 22403,CC1=C(C(=O)OCC(=O)NC(C2N(C)CCCC2(C)C)(C)C)C(=O)OC1(C)C 22404,CC1CC(NC(=O)C(C)(C)N2CCOCC2)CCN1C(C1C(F)(F)C12CC2)=O 22405,C1(NC(CCOCC)=O)CN(C(=O)C=CC2CCOC2)CC12CC2 22406,c1(CC)c(C(=O)NC(CN(C(=O)CC(C)C(F)F)C)CC)cccc1C 22407,c1(C(=O)NC2CC3CC(NC(CCCOC)=O)CC3C2)ccc2c(c1)ncn2C 22408,C1(NC(C2N(CC)CCC2)=O)CN(C(c2cccc(=O)n2C)=O)C(C)(C)C1 22409,c1(C(N(C(CNC(C2C(OC)C2)=O)C)C)=O)ccc(-c2ccccc2)[nH]1 22410,N1(CC)CCC(NC(C2CCOCC2NC(C2CC2Cl)=O)=O)C1=O 22411,C12(NC(CC3(OC)CC3)=O)CCCC(NC(=O)CCc3nccn3C)(C1)C2 22412,C(C)(C(O)C(=O)NCC(C)(C)NC(=O)CN(S(=O)(=O)CC)C)OC.OC 22413,C(=O)(C#CC(C)(C)C)N(CC(CNC(CC(C)n1ccnc1)=O)O)C 22414,N1(C(=O)CSc2nc[nH]n2)CCC2(NC(=O)CC3CCSCC3)CCCC12 22415,N1(C(C2(C)CC(C)C2)=O)CCC(C2(O)CN(C(C3C4COCC34)=O)C2)CC1 22416,c1(CC)cc(F)ccc1CC(=O)N(CC(CC)NC(=O)Cc1ncoc1C)C 22417,C1(NC(=O)CC2=CCCC2)CCC2(CCCN2C(C2COC2)=O)CC1 22418,c1(CSc2nc3ccc(C(=O)OC)cc3o2)nc2ccc(Br)cc2n1C 22419,C1(F)(C(NOC(C(=O)NCc2ncc(COC)s2)C)=O)CCCCC1 22420,c1(C(N(C(C)CNC(=O)CN2CC3CC3C2)CC)=O)cn(C)cn1 22421,c1(OC)cccc(CC(C)(C)NCc2c[nH]nc2C(F)(F)F)c1 22422,n1(C(C)C)ccc(C(N2CCC2CNC(c2nc(Cl)cs2)=O)=O)n1 22423,N1(C(CCC#C)=O)CC(CCNC(c2ccnc(Cn3cnnc3)c2)=O)OC(C)C1 22424,C1(C(N2CC(C)(CO)C2)=O)C2CCC(C2)N1C(C1(C)CC(C#N)C1)=O 22425,N1(C(C(C)C#N)=O)CC(C2CCCN(C(C3CC(c4ccccn4)=NO3)=O)C2)C1 22426,Cc1[nH]ccc1C(=O)NCc1cn(CC(N2CCC2CC(=O)N(C)C)=O)nn1 22427,N1(C(C(=O)NCc2cnn(Cc3ccccc3)c2)=O)CCC(CO)C(F)C1 22428,C1(NCC(=O)Nc2c(CC)cco2)CCN(C(=O)C=CCOC)C(C)C1 22429,c1(C(=O)NCC2CC(CNC(C3CCN(CC)CC3)=O)OC2)nccc(C)c1F 22430,Cc1cc(C)[nH]c(=NCC2(NC(c3cccn4c(O)nnc34)=O)CC2)n1 22431,C1(CC(=O)NC(C(C)(C)NC(c2cncc(COC)c2)=O)C)NC(=O)CNC1=O 22432,CC(N=c1cc(C(F)(F)F)nc(Cl)[nH]1)C1CCCN(C(=O)C=Cc2nccs2)C1 22433,CCCCC(O)CC(=O)NCc1cn(CC2(C(=O)O)CC(OC)C2)nn1 22434,n1(CCC)cc(Cl)c(C(=O)NC2(CCNC(C3CCCC3(C)C)=O)CCCC2)n1 22435,c1(C(N2CC3C(NC(c4c(OC)n[nH]c4)=O)C3C2)=O)cc(Br)cc2cc[nH]c12 22436,c1(CC(c2ccccc2)N2CCOCC2)cc(Cl)cs1.C12(COC1)CNC(=O)N2 22437,CCS(=O)c1ccccc1C(=O)NCC(C)(CO)NC(c1nc(O)c(C)s1)=O 22438,C(C)(C(C(=O)NCCN(C)C1CC1)NC(c1nc(C)oc1C)=O)OC 22439,N1(CCC)CCC(C(=O)NC2C3CC(NC(=O)Cc4ccsc4)CC23)CC1 22440,Cc1ccc2c(c1)C(C(=O)OCCCN1CCCCC1)OCC2 22441,N1(C(C2CC(C)(C)C2)=O)CC(CNC(=O)CC2=CCCCC2)C2(CCOCC2)C1 22442,c1(NC2CC(C(C)C)C2)ccc(NC(=O)CCCCC2CC2)cc1C(F)(F)F 22443,N1(C(C(CC)(C)C)=O)CCC(NC(=O)Cc2cc(Cl)ccc2O)C(C)C1 22444,c1(C(=O)NCC(C)NC(c2c(C)nn(C3CC3)c2)=O)cnn2c(N)ccnc12 22445,C(=O)(C(=O)C(C)(C)C)NC(C(C)NC(=O)CSc1cccc(F)c1)C 22446,N1(C(=O)CN2CCOCC2)CCCC(CCC(=O)NCC23CC(CO)(CO2)C3)C1 22447,c1(SCCC(=O)NC2(CC=C)CN(C(=O)C(C)CO)C2)ccc(C#N)cc1 22448,C(C(CC(C)C)C(=O)N(C(C)CNC(c1cnc(Cl)n1C)=O)C)OC 22449,Cc1cc(N2CCC(C(C)NC(C3CCCC(O)C3)=O)C2)c(Br)cc1[N+](=O)[O-] 22450,c1(C(=O)NCC2(NC(=O)C3=CCSC3)CC2)c(Cl)ccc(Br)c1F 22451,C12(NC(CN(C)C)=O)CCCCCC1N(C(c1coc(Br)n1)=O)CC2 22452,Cc1cnn(C)c1C(=O)N(C(C)(C(=O)N1CCC(C(N)=O)C1)C1CC1)C 22453,C1(CN(C(C(C2CC2)OC)=O)C)CCCN(C(=O)CCCOC(C)(C)C)C1 22454,CC1(C)CC(NC(=O)C2=NOCC2)CN(C(c2ccnn2CC2CC2)=O)C1 22455,c1(OC)cc(-n2c(Cn3nc(C)cc3C)nnc2SCCC(F)(F)F)cc(F)c1 22456,c1(-c2c(C)c(N3CCn4c(C)cnc4C3)ncn2)cccc2c1OCCO2 22457,CC(C)(O)C(F)C(=O)NCC1CCCC1C(N1CC2(CCC2O)C1)=O 22458,Cc1cc2nc(NCC3CC4(CC(NC(=O)C(F)(F)Br)C4)C3)cc(=O)n2o1 22459,N1(C(c2cc(CSC)on2)=O)CCC(F)CC1C(=O)NCC(C)C(C)(F)F 22460,C1(NC(c2n(CC#C)ccc2)=O)CN(C(=O)C(F)CC)CC2CC12 22461,N1(C(C2CC3(CC(NC(C(CC(C)(C)C)OC)=O)C3)C2)=O)CCC2(CCC(O)C2)C1 22462,C1(NC(C(c2ccc(F)cc2)C)=O)C2CC(CN(C(C3CC=CC3)=O)C2)C1CO 22463,N1(C(c2ccc(NC(C)=O)cn2)=O)CCCC(NC(=O)C(F)(F)CC2CC2)C1C 22464,C(=O)(C(C)CC(F)F)N1CC(CCNC(c2c(C)[nH]c(=N)s2)=O)C1 22465,C(=O)(C(C)CC(C)(F)F)NC(CCNC(CCc1ccc(OC)cc1)=O)C(C)C 22466,C(CCCC(C)C)N(C(CCC1N(C(c2c(C)scn2)=O)CCC1)=O)C 22467,C1(C(=O)NCCC(=O)NC2CC2)(CNC(C23CSCC2C3)=O)CCCCC1 22468,c1(CC(C)NC(=O)Nc2cncc(C(C)(C)C)c2)nc2ccccc2s1 22469,N1(C(c2c(C)cc(SC)o2)=O)CC(NC(=O)Cc2coc(C)n2)CC1(C)C 22470,C1(CC=C)(NC(=O)CN(C)CCOC)CN(C(=O)C(=O)N(C)C)C1 22471,c1(CNC(C(C2CCN(C(=O)CCNS(C)(=O)=O)CC2)C)=O)ccc(O)c(O)c1 22472,c1(CC(=O)NCCN(C(C=C(CC)C)=O)CCOC)cccc(C(C)OC)c1 22473,N=c1ncn(CC(=O)NC(CC2CC2)C(=O)NCCC2CC(F)C2)[nH]1 22474,C1(NC(C2(N(C)C)CCCC2)=O)CN(C(=O)CC2CCC23CCC3)CC1C(F)F 22475,CCC(CC)(CC)C(=O)N1CC(O)(c2cn(-c3ccc(C(C)(C)C)cc3)nn2)C1 22476,CCC(CC)CC(=O)NCC12CC1CN(C(=O)CC1(C)CC1(F)F)C2 22477,C12(C(N3CCC(C)(NC(C=C(C)Cl)=O)CC3)=O)CCOC1CC(=O)NC2 22478,C(=O)(C(COC)OCc1ccccc1)NCCCNC(C=CC(CC)=CC)=O 22479,c1(N(CCC#N)C)nc(=NC2CC(N3CCC3)C2)[nH]c2cc[nH]c12 22480,c1(C(C)C)ncncc1C(=O)NCC1CC(NC(=O)CC(C)C2CC2)C1 22481,N1(C(CC2(OC)CCC2)=O)CCOCC(NC(c2cc(Br)no2)=O)C1 22482,c1(C(N2C3CC(NC(C(C(=C)C)(C)C)=O)C(C3)C2)=O)ccc([N+](=O)[O-])c(C)n1 22483,C1(NC(CC2C(C)CC2)=O)CCCCN(C(=O)C(C)(C)C2CCCCO2)C1 22484,C1(C(N2C(C(=O)NCC)CCC2)=O)CCCN(C(C2CC3(CSC3)C2)=O)CC1 22485,c1(C(=O)NCC(C)(C2CC2)NC(c2ccc(CC)[nH]2)=O)ccc(=O)n(C(C)C)c1 22486,c1(CCC(=O)NCC2(C(=O)OC)CC2(F)F)cccc(F)c1Br 22487,C1(NC(=O)C=CC2CCOC2)CN(c2nnco2)CCC12CCC2 22488,N1(C(CCCC)C(=O)Nc2ccccc2CC)CCS(=O)(=O)C(C)C1C 22489,C(=O)(CC(C)(C)C(=O)N1CC2C(CNC(C3CCS(=O)CC3)=O)C2C1)OCC 22490,O(NC(=O)C(CC(=C)C)NC(C1CCC2CC1CO2)=O)CC#C 22491,c1(NCC)ncc(C(=O)NC23CC(CNC(=O)C#CC(C)C)(C2)C3)cc1Cl 22492,c1(CC(=O)NCC23CC(NC(C(COC)N(C)C)=O)(C2)C3)c(O)ncnc1O 22493,c1(NCCC(C)(C)c2ccccc2)csc(Cl)c1 22494,CCCC(C)CC(=O)NCC(C)N(C(c1ocnc1-c1ccccc1)=O)CC 22495,c1(OCC)cccnc1C(=O)NCCC(C)N(C(=O)C=Cc1ccc[nH]1)C 22496,C1(C)(CNC(C(CC)O)=O)COCCN(C(c2cc(F)c(O)c(Cl)c2)=O)C1 22497,c1(C(=O)NC2C(CN(C(=O)Cn3ccc(C(F)F)n3)C)CCC2)nsnc1O 22498,N1(CC2CC(C)OC2)CC2(CN(C(=O)OC)C(c3cnn(C)c3Cl)=O)CC1CO2 22499,C=C(C)C(C)(C)C(=O)NCC1CCC1NC(=O)C(CO)N(C)C 22500,c1(C(=O)NCC(CO)NC(C(C2CC2)OC)=O)c[nH]c(=N)nc1C 22501,c1(C(=O)NC2(C)CC(C(N3CCCN(C(C)=O)CC3)=O)C2)cc2ccccn2c1 22502,CC(C)CC(O)C(=O)NC1(C(=O)NC2CCCCCC2C)CC1(C)C 22503,CC(CC(C)(C)C)C(F)C(=O)NCC1C2CN(C(=O)CCCn3ccnn3)CC12 22504,N=c1[nH]c2cccc(C(=O)NC3C4CN(C(c5cscc5Cl)=O)CC34)c2o1 22505,C=C(Cl)C(C)(C)C(=O)NC(C1CCCCN1C(=O)CN1CCC(C)(C)C1)C 22506,CCCCCC(O)C(=O)N1CC=CC1CNC(=O)CNC(C1CCC1)=O 22507,c1(C(C)OC(C2CC(CCC)C2)=O)ccc(Cl)nc1 22508,C(=O)(C1CCCn2cnnc21)N(CCC(C(C)(C)C)NC(C)=O)C 22509,C1(C(=O)NCc2cn(-c3cncc(C(F)(F)F)c3)nn2)(OCC)CC2CCC1C2 22510,c1(C(C)(C)C)cncc(NC(C2CN(C(=O)C3CC3)CCN2)=O)c1 22511,C1(C(=O)NCc2n(CC)nnn2)N(C(=O)C(C)n2cccn2)CCCC1(C)C 22512,c1(C(N2CC(Cn3cc(C(C)OC)nn3)C2)=O)ccc2nc(Cl)nn2c1 22513,c1(C(=O)NCC2CCCC(NC(C(CC)C(C)C)=O)C2)ncnc2c1CCC2 22514,c1(C(N(C(C)CN(C)C(C2(F)CC=CCC2)=O)C)=O)ccc([N+](=O)[O-])[nH]1 22515,N1(C(CCN(C(C)=O)C)=O)CC2CC(NC(C3(C(F)F)CCN(C)CC3)=O)C1C2 22516,N1(C(c2n[nH]c(C)c2O)=O)CCC(C2CC2)(CNC(=O)COc2ccccc2)C1 22517,C1(NC(C(COC)(C)OC)=O)CC(C)CN(C(=O)Cc2cnc(Cl)cc2C)C1 22518,N1(C(CN(C(=O)COCC2CCCO2)CC#C)=O)CC2COC(=O)C2C1 22519,N1(C(C23C(CN(C(C(CC#C)C4CC4)=O)C2)C3)=O)CCCSCC1C 22520,c1(C(N2CCC(O)(CCNC(CSCC=C)=O)C2)=O)cccc(C(N)=O)c1F 22521,c1(OCC)nc(N2CCC(N(C)C(c3sc(CSC)nc3C)=O)C2)ncc1C 22522,C1(C)(C(=O)NCC2CC(NC(c3c(C)cnn3C(C)C)=O)C2)CCCNS1(=O)=O 22523,N1(C(CC(C)(C)C)=O)CCC2CN(C(c3cc(F)cc(F)c3O)=O)CCC2C1 22524,C1(C(=O)Nc2cnc(I)cn2)CCN(Cc2ccc(OCCO)cc2)CC1O 22525,C(C(O)(C(F)(F)F)c1ccccc1Cl)NC(=O)NC(C(C)F)C(=O)O 22526,N1(C(c2c(CCC)n[nH]c2)=O)CC=CC(NC(c2cnco2)=O)C1 22527,Cc1cc(C)n(CC2CCN(C(=O)N(C)CC3(O)CCCCC3)CC2)n1 22528,C(=O)(CS(=O)(=O)CC1CCCO1)NCC(C(C)(C)C)NC(=O)C=C1CCCC1 22529,c1(C(=O)NCCC2CCN(C(C(CC)=CCCC)=O)C2)cncc2ncccc12 22530,C(CCC)(C(=O)NCC(C)CNC(C1(CC(C)C)CCCC1)=O)=CCC 22531,c1(-n2cc(CNCC3CCCN(C(C(COC)O)=O)C3)nn2)ccc(C)c(Cl)c1 22532,Cc1cc(C)n(CC(N2CCC(N(C)C(c3cccc(CS(C)=O)c3)=O)C2)=O)n1 22533,C1(C(=O)NC(C(=O)OC)C)CN(C(c2ccc(COC(C)=O)s2)=O)CCC1O 22534,N1(C(C(F)=CCC)=O)CC(C)N(C(c2ccc(C3OCCO3)cc2)=O)CC1C 22535,O=C(C1=CCCCO1)Nc1cccc(CNC(C2CCN(C3COC3)C2)=O)c1 22536,N1(C(CC=CC)=O)CCC(C)(CC(=O)N(C(C2CCC2)C)CC)C1 22537,N1(C(c2ccn(CCNC(C3(CC)CCC3)=O)c2)=O)CC(S(N)(=O)=O)C1 22538,CC1(CNC(C2CC3C=CC2C32CC2)=O)COCCN(C(=O)CC2CC(=O)C2)C1 22539,N1(C(CSCC)=O)CC2CCCC2(CNC(=O)C2=NOC(c3ccccc3)C2)C1 22540,c1(NC(=O)NC(c2ccccn2)Cc2cccc(C)c2)cc(F)c(I)c(F)c1 22541,N1(C(c2c(C)nsc2)=O)CC(NC(c2ncc(Cl)c(N)c2Cl)=O)CC2(CCC2)C1 22542,C(CN=c1[nH]cc2ccnc-2[nH]1)=CCNC(c1cc2sccc2[nH]1)=O 22543,C1(C(=O)NC(CC)C(N)=O)CCN(C(C2CC(=O)NC2(C)C)=O)C12CCC2 22544,C1(N(C)C(C2C=CCS2)=O)CN(C(c2cc(Cl)c[nH]2)=O)CCC1O 22545,C1(N(C(=O)C(O)C2CN(C(C3CCCC3F)=O)C2)CC)CCCCC1 22546,CC(C)CCCC(C)CCNC(=O)N(C(C)(C)C)Cc1ccc(Cl)cc1 22547,c1(C(N2C(C)CC(CNC(C3(C)CCNC3=O)=O)CC2)=O)cnn2ncccc12 22548,C(=O)(C(C)(O)COC)NC1CC(C)(NC(c2ccc(CC)cc2)=O)C1 22549,c1(CNC(C(=O)OC)(C)COC)cc2c(cc1OC)CCC2 22550,C1(C(=O)NCCC(N)=O)CCC(NC(=O)Cc2cccc(Cl)n2)CO1 22551,Cc1cc(NC(=O)C(C)CNC(=O)Cc2cnccc2C)c(C)c(C)c1 22552,N1(C(C2(C)CCCOC2)=O)CCOC2(CCN(C(C3CCC4CC4C3)=O)C2)C1 22553,C1(C(=O)NCC2CC(O)C2O)(NC(c2cnn(C3CC3)c2)=O)CC(O)C1 22554,O=C(CC(F)(F)F)NCC1CC(NC(=O)CCCOc2cccnc2)C1 22555,c1(CC(=O)NC2C=CCN(c3nc(C)nc(Cl)c3)C2)c(C)[nH]c2ccccc12 22556,c1(C(N2CC(C(C)NC(C34CC(C3)C4)=O)C2)=O)cc(O)c(O)c(O)c1 22557,C1(C(N2CC(NC(CN(C(C)=O)C)=O)(CO)C2)=O)CCC(=O)N1C 22558,C1(COC)(NC(=O)Cc2cc[nH]n2)CCN(C(=O)C(C)NC(C)(C)C)CC1 22559,C1(NC(c2nccc(CC)c2)=O)CC2CC1N(C(c1ccc(F)c(N)c1)=O)C2 22560,c1(C(=O)NCc2sc(Cl)nc2Cl)ccc(=O)n(Cc2ccccc2Cl)c1 22561,C=CCC(CNC(=O)CC1(C#N)CC1)C(=O)NC(C)Cc1nncn1C 22562,C(=O)(C1=CC2(CCOCC2)C1)NC.C(=O)(C(CO)C(C)(C)C)NCC(C)CC(=O)N 22563,C(C(C)(C(=O)N(CC(O)CNC(c1n[nH]cc1I)=O)C)OC)OC 22564,N1(C(C(C2CCC2)NC(c2c(OC)ccnc2)=O)=O)CCC(C)C(F)(F)C1 22565,N1(S(=O)(=O)c2cnccc2N2C3CCC2CC3)Cc2ccccc2CC1CO 22566,N1(C(c2c(OC)cc(N)cc2)=O)C2CCC1CN(C(=O)CC1CCCN(C)C1)C2 22567,C1(NC(COC(C)=O)=O)CC(CNC(c2ccc([N+](=O)[O-])[nH]2)=O)C12CCC2 22568,CN1CCCC1(C)C(=O)NCc1cccc(NC(C2CC2F)=O)c1 22569,N1(C(c2ncc(NC)nc2)=O)CC(C)C(C)(CNC(=O)COC(C)C)C1 22570,Cc1ccc(NC(C2C=CC(NC(=O)Cc3c(F)cccc3F)C2)=O)c(CO)n1 22571,Cc1cc(C(N2CCCCC2CNC(=O)CNC(=O)C(C)C)=O)cc(C(F)F)c1 22572,Cc1oc([N+](=O)[O-])cc1C(=O)NCCC(C)(C)NC(=O)C(=Cc1cscn1)F 22573,C(=O)(C1=C(C)S(=O)(=O)CC1)NC1CN(C(c2c(C#C)c[nH]n2)=O)C(C)(CC)C1 22574,C1(C)(C(N2CCC(CNC(c3c(OC)c(F)ncc3)=O)C2)=O)CCCCCCC1 22575,c1(C(=O)NC23CC(CNC(C4(CCOC)CCC4)=O)(C2)C3)ccc(O)c(CO)c1 22576,N1(C(c2cnnc(C)c2C)=O)CCOC2CN(C(C3CCN(C)C(=O)C3)=O)CC12 22577,C1(NC(C23CC(COC)(OC2)C3)=O)CN(C(c2ccc(CSC)o2)=O)CCC1C 22578,Cc1cc(C(N2CCN(C)CC2CNC(c2c(Cl)nsc2Cl)=O)=O)cc(=O)n1C 22579,c1(C(=O)NC2CC(NC(CCCOC)=O)C2)cc(C)c(Br)cc1C 22580,N1(C(c2[nH]cc(C)c2)=O)CCN(C(=O)C=Cc2cnc[nH]2)CC1C#N 22581,C#CCC(C(=O)NCC1(NC(=O)C=CC2CCCCC2)CCOC1)C1CC1 22582,C1(NC(C(=O)NC(C)C)=O)CCC2(CC1)CN(C(C1OCCO1)=O)C2 22583,CCC(CC)(CC)C(=O)NC1CN(C(=O)CS(=O)(=O)CC)CC1O 22584,C1(S(C)(=O)=O)(C(=O)NC2CC(NC(c3nc(OC)nc(O)c3)=O)C2)CC(O)C1 22585,C#CC1CCN(C(=O)C(Cc2cn[nH]c2)NC(=O)CCCN(C)C(C)=O)C1 22586,Cc1cn2c(C)c(C(=O)NCCNC(=O)CCCOC(C)(C)C)nc2s1 22587,C1(C(=O)NCCC(=O)OCC)CCC(O)CN1C(c1cccc(O)c1)=O 22588,S(=O)(=O)(c1ccccc1Br)N1CCC(C(N2CCCC(C#C)CC2)=O)CC1 22589,c1(C(=O)NCC(C)NC(=O)CC2CC3CC3C2)ccccc1 22590,CC1COC2(C1)CN(C(=O)C(C1(C)CC1)NC(C1CN(C)CCO1)=O)C2 22591,C1(C2CC2)(CNC(COCCC=C)=O)CCN(C(c2cn(C)nc2Cl)=O)C1 22592,N1(C(C(C(CC)O)(F)F)=O)CCc2nc[nH]c2C12CCN(c1ncncc1C)C2 22593,C1(CSCC(=O)NCC2CC2NC(=O)CC2(C(F)(F)F)CC2)CCCO1 22594,Cc1nc(N(C2CCC(NC(C3CCC(=O)NC3)=O)CC2)C)cc(C(C)C)n1 22595,C1(O)(CNC(C(C)OCC=C)=O)CC(N=c2[nH]c3c(C)cccc3o2)C1 22596,C1(NC(c2cc(Cl)nnc2O)=O)CN(C(=O)CSCC(F)(F)F)CC1C1CC1 22597,CC(C)(CC#N)C(=O)N1CCN(C(c2ccnn2CCF)=O)C(CF)C1 22598,C1(F)(C(N2C(C(=O)OC)CC2C)=O)CCN(C(C2(C)CCNC2=O)=O)C1 22599,N1(C(C2(CCC)CC2)=O)CCC(F)(F)C(CNC(C2(N(C)C)CC2)=O)C1 22600,CC1=CC(C)CN(c2nccc(N(C)Cc3cc(C)nc(C)n3)n2)C1 22601,c1(C(=O)NCC(CNC(Cn2ccc(C)cc2=O)=O)(C)C)cncc2nc[nH]c12 22602,C(C1=NOC2COCC12)NC(C1(CCNC(C(C)SC(C)C)=O)CCC1)=O 22603,C1(C(=O)NCCCSC(F)F)CCCCN(C(C2CC3(CSC3)C2)=O)C1 22604,c1(C(N(C)CC2N(C(C(C=C)C)=O)CCCC2)=O)cc(CC)ccc1F 22605,CCC(C)(C)CCCC(=O)NC(CC)CCCC(=O)NC1(C2CC2)CC1 22606,c1(C(N(C2CCN(Cc3cc(OC)ns3)C2)C)=O)cc(F)c2ncccc2c1 22607,C1(CC)C(C(=O)N(C)Cc2nc[nH]n2)CCN1C(C1CC(F)(F)C1)=O 22608,C1(CNC(c2cc(Cl)sc2C(F)F)=O)CCN(C(=O)C(=O)NC2CC2)CC1(F)F 22609,C(C(C)C(C)(C)C)N(C(C)C)C(C1CCCN(CCc2ccccn2)C1)=O 22610,C1(NC(C2(OC)CCN(C(C(CC)N(C)C)=O)C2)=O)CCCOC12CCC2 22611,c1(C(=O)NCCCCN(C)C(C2CC(=O)N(O)C2)=O)coc2c(F)cccc12 22612,C1(C(=O)NCC2N(C(C=Cc3ccc(CC)o3)=O)CCC2C)CC(S(C)(=O)=O)C1 22613,CCC(CO)CCNC(=O)C(C)C(C)NC(=O)CCC1CC(C)C1 22614,C=CCC(CC)C(=O)N1C2CCC1C(CNC(=O)C(Br)=C(C)C)C2 22615,c1(C(=O)NCCCN(C(CCNC(N)=O)=O)C2CCCC2)nocc1Cl 22616,c1(OC)ccc(CN2CCCC(CNC(=O)C(N3CCC(OC)C3)=O)C2)cc1 22617,c1(CC)c(NC(C2CC(NCc3n[nH]c(C)c3C)C2)=O)cnn1C 22618,c1(OC)ccc(C(=O)NCC(C(C)C)NC(=O)Cc2cnn(C)c2)c(C)c1OC 22619,c1(C(N2C3C(NC(C(c4ccccc4)OC)=O)C(C3)C2)=O)ccc(=O)n(O)c1 22620,c1(CC(N2C(C)CC(CNC(=O)C(C)(C)CC#N)CC2)=O)ccccc1S(C)(=O)=O 22621,C1(O)(C(C)NC(C2(CO)CCCCC2)=O)CCN(C(c2nccnc2N)=O)CC1 22622,c1(C(N2CCOC(CNC(C3(O)COC3)=O)C2)=O)ccnc(Cl)c1O 22623,CC1=C(C(=O)NC(C2CCN(C(c3ncccc3N(C)C)=O)C2)C)CCO1 22624,Cc1cccc(C(N2CC(CC(=O)N(CC(C)C(F)(F)F)C)C(C)C2)=O)c1O 22625,c1(C(=O)NC(C)(C)CCNC(c2cc(CCO)on2)=O)ccnc(F)c1O 22626,N1(C(c2cncc(NC)c2)=O)CCC2(COC(CNC(=O)C(F)CC(C)C)C2)C1 22627,C(CN=C(NCC(F)F)N1CCP(C)(=O)CC1)c1cc(OC)ns1 22628,N(C(=S)N1CC(S(=O)(=O)C2CC2)C1)C(c1ccccc1)C 22629,C(C)(C(C(=O)NCc1nccn1C1CC1)C(C)C)NC(C#CC(C)C)=O 22630,c1(C(N2CC(NC(c3[nH]n(C)c(=O)n3)=O)C(O)C2)=O)occ2c1CCOC2 22631,C(CNC(c1cc(CN(C)C)c[nH]1)=O)(CC(C)C)NC(c1c(CCC)occ1)=O 22632,c1(N(CCC(=O)NC)C)nc(=NCC(CO)C2CCC2)[nH]c2cccnc12 22633,c12cccc(c1)CNC(=O)N2.c1(COCC(=O)OC)nnc(-c2cccnc2)s1 22634,N1(C(CC(=C)Br)=O)CCC(NC(=O)CSCCCC)C(F)C1 22635,c12ccccc1CS(=O)C2C.N#CCCCN 22636,N1(C(=O)Nc2c(C)cn(-c3ccc(F)cc3)n2)CC2CC1CN2c1ccccc1 22637,C12CCCC1C(C(=O)NCCCF)N2C.C(=O)(CCC1CC1CC1CC1)OCC 22638,C(=O)(C1=CCCOCC1)N1CCC(N(C(C2C3CC4C(C3)C24)=O)CC2CC2)CC1 22639,C=CCC(CC)C(=O)NC1CN(C(c2cn(C(C)C)nn2)=O)CC1(C)C 22640,C1(C2CCN(C(c3ccc(C#N)nc3O)=O)CC2)(NC(C(OC)OC)=O)CCC1 22641,c1(C(=O)NC2CC(C)(NC(CNC(CC)=O)=O)C2)cc(F)c2c(c1)CCC2 22642,C(C(=O)NCC1CC(O)CN1C(=O)C=Cc1cnccn1)(C(C)C)OC 22643,c1(C(C(=O)N(C2CCCCC2)CCNC(CCC(N)=O)=O)O)ccc(F)c(F)c1F 22644,C(CO)(CCCNC(=O)C(c1cnn(C)c1)=O)NC(C(C)C1CCCC1)=O 22645,c1(C(=O)NC(CCNC(c2n(CC)nnc2)=O)C)cc2c(s1)CCOC2 22646,N1(C(c2ccc(C#C)cn2)=O)CCC2(CC(NC(=O)C3=NOCC3)CO2)C1 22647,c1(OCC(=O)OCCC2CCN(C(=O)OC(C)(C)C)C2)nc2cc(F)ccc2s1 22648,c1(C(C(=O)NC)c2nn[nH]n2)ccc(Br)cc1ON1CCC(O)C(C)C1 22649,N1(C(C(CCC)C#N)=O)CC2CCC(C(N3CCc4c[nH]nc4C3)=O)(C2)C1 22650,c1(CCCCC)ccc(C(N2CC(OC)CC2C(N2C3COCC2C3)=O)=O)cc1 22651,C1(C(=O)NCCC2CCN(C(=O)CCc3ncc[nH]3)C2)CCCC(CF)C1 22652,C(CCCC(CO)NC(=O)Cc1cc(C)[nH]n1)NC(c1c(C)cc(CC)o1)=O 22653,C1(NCc2cccc(C)c2)CC12CCN(Cc1cc(C(=O)O)cc(C)c1)C2 22654,C1(C(=O)NCC2(O)CN(C(c3c(C)cnn3C)=O)C2)CCC2(C1)CC2(F)F 22655,N1(C(CCP(C)(C)=O)=O)CCOC2CN(C(=O)C=C(C3CC3)C3CC3)CC12 22656,N1(C(=O)COCCc2ccccc2)CCC2(CCCN2C(C2CCCO2)=O)C1 22657,Cc1cnsc1C(=O)NC1(C(=O)NOCC2CC(=C)C2)CCC1 22658,C1(CC(C)NC(C2C(F)(C(=O)OC)C2)=O)CCN(C(c2ccon2)=O)CC1 22659,N1(C(COC(C)(C)C)=O)CC(O)CC1C(=O)NCCN=[N+]=[N-] 22660,c1(OCC#C)ccc(C(=O)NC(CCN(C(=O)C(O)CN(C)C)C)C(C)C)cc1 22661,c1(C(=O)NCC2C(C)CCN(C(C)=O)C2)cc2c(c(S(N)(=O)=O)c1)CCC2 22662,C1(NC(C(C=C)(C)C)=O)CCC2(CC1)CN(C(C1(CC(F)(F)F)CC1)=O)C2 22663,c1(C(=O)OC)nc(Nc2nc(C)c(C(=O)NCCC3COCCO3)s2)oc1C 22664,N1(C(C(=O)NCC=C)CCc2ccco2)CC2C(OC)CS(=O)(=O)C2C1 22665,C1(CN(C(c2n(CC#C)ccc2)=O)C)CCCCN1C(c1cnsc1)=O 22666,c1(C(N(C2CCN(C(C3C(OC)(OC)CC3)=O)C2)C)=O)cnc(SC)nc1O 22667,C1(C(N(CC(O)CF)C)=O)C(C)CCN1C(=O)C(C(C)C)SC 22668,C1(NC(=O)NC(c2c(I)cnn2C)C(C)C)CC2(C1)CC(N(C)C)C2 22669,CC(CS(=O)(=O)c1ccccc1)NCc1nnc2cccnn12 22670,c1(SCCC#N)cc(-c2cccs2)n2nccc2n1 22671,C(=O)(CCC(CF)CF)NC(C(C(=O)NC(C1CCCC1)CC)(C)C)C 22672,N1(C(c2nc(CC)[nH]n2)=O)CC(NC(=O)CSCc2ccccn2)CC(C)C1 22673,c1(C(C(=O)NCCC(CNC(=O)C=CCO)O)O)cc(F)c(F)cc1F 22674,C12(C(N3CCC(OCCNC(C(C)n4cnnn4)=O)C3)=O)CCCCC1C2(F)F 22675,c1(C(=O)NC2CC3CN(C(CCN(C)CC)=O)C2C3)c(F)cc(C)cc1Br 22676,Cc1nnc2cnc(C(=O)NC(C)CN(C(=O)C(C)(O)CC(C)C)C)cn12 22677,Cc1oc(C)c(C(=O)NCc2ccc(C(=O)NOCC3CCCO3)s2)c1C 22678,C1(C(N(CCC(=O)NC(C2CCCO2)(C)C)C)=O)COCC1C(N)=O 22679,c1(C(=O)NCC(C)CNC(C2CCCN2C(=O)C2CC2)=O)cncc2[nH]ccc12 22680,N1(C(Cc2cc(C)no2)=O)CCC(CNC(C2CCC(C)(C)O2)=O)C(F)(F)C1 22681,C1(CNC(CCCCNC(N)=O)=O)CCN(C(=O)CC2CCCOC2)CC1(F)F 22682,c1(OC)ccc2c(C(=O)NC3CC(C)CN(C(c4[nH]ccc4C)=O)C3)c[nH]c2c1 22683,Cc1nc(NCC(CC(C)C)NC(c2nc(Cl)ccc2F)=O)cc(O)n1 22684,N1(C(CC2CC(C)C2)=O)CCC(C)(C)C(C(=O)NCC2(C)CC(C)(C)C2)C1 22685,c1(OC)ccc(F)cc1C(=O)NCCN(C(=O)CN(c1cnccn1)C)C 22686,N1(C2C(NC(C(CC)F)=O)CCC2)CCN(C(C2CC(O)C2)=O)CC1 22687,C(=O)(C1c2ccccc2CCN1CC(c1cc(Cl)ccc1Br)=O)OC 22688,C=C(C)CC(C(=O)N1CCC(C)(N(CCCO)CC)C1)NC(C)=O 22689,CC1CN2CCN1C(C(N1CCCC1C1CCN(C(=O)CC3CC3(Cl)Cl)C1)=O)C2 22690,N1(C(CCN(CC)CC)=O)CC(O)CCC1C(=O)NCc1ncn(C)n1 22691,Cc1cc(=NCC23CCCCC2C3)[nH]c(=NCCc2ccc(Br)c(F)c2)[nH]1 22692,N1(C(c2ccc(C)c(Cl)c2Cl)=O)CCCC2CCN(C(c3ccncn3)=O)CC12 22693,c1(OCC)ccc(C)nc1C(=O)NCC1CN(C(=O)CC2COC(=O)C2)C1 22694,N1(C(CSCC#C)=O)CC2CCC1CN2C(=O)Cc1c[nH]c2ccccc12 22695,CCCC(CC)CC(=O)NC1C2CN(C(=O)CC3OCCOC3(C)C)CC12 22696,c1(C(N2CCC(NC(CCn3c(C)ncc3)=O)C2)=O)cc2scc(C)c2[nH]1 22697,C=CC1(C(=O)N(CCOCC)CC)CCN(C(=O)CCCn2cccc2)C1 22698,c1(C(=O)NCC2(F)CCC(NC(c3ncn(C)c3)=O)C2)ccnc2ncccc12 22699,C12(C(N3C(CNC(c4cccc(COC)n4)=O)COCC3)=O)CC1CCC2(F)F 22700,N1(C(C2=C(C)CC2)=O)CC2COCC2(C(=O)N(C2CCCC(O)C2)C)C1 22701,O=C1CCC2(CCCN(C(C34CC(c5cnccn5)(C3)C4)=O)C2)N1 22702,c1(C(=O)NCCN(C(=O)C=CC(=O)N(C)C)C)cccc(N(CCO)CC)c1 22703,c1(CC(=O)NCC(C)(C2CCC2)NC(CC2(OC)CC2)=O)nc(F)c(F)cc1F 22704,c1(C(N2CC(C(=O)NCC(C)(C)C3CC3)(COC)C2)=O)ccc2cccnn12 22705,Cc1coc(C2CC2)c1C(=O)NCC1CC(NC(c2coc(CF)n2)=O)C1(C)C 22706,C#Cc1ccc(C(N2CCC(NC(c3cc(O)ncc3Br)=O)C2C)=O)nc1 22707,CC1CCn2c(C(=O)NCCCOCCCNC(C3CCC(=O)N3)=O)cnc2C1 22708,Cc1ccc2occ(C(=O)NC3CCC(CNC(c4cscc4C)=O)CC3)c2c1 22709,C1(NC(c2n(CC)cnn2)=O)CC2(CCCN(C(c3ccsc3C)=O)C2)C1 22710,c1(C(C)C)ccccc1CC(=O)NCC(C)(CO)NC(=O)C(C)SC(C)C 22711,C1(C(N2CC3C(NC(C4(C)CCOCC4)=O)(C3)C2)=O)CN2CCN1CC2 22712,c1(C(N2CC(O)(CCNC(C3CC(=O)N3)=O)C2)=O)noc2cc(F)ccc12 22713,n1(CC(=O)NCCNC(C23CNC(CO2)C3)=O)cc([N+](=O)[O-])cn1 22714,N1(C(c2c3ccc(C)cc3no2)=O)CC2CCCC(C1)N(C(=O)C=CBr)C2 22715,CCCCCC(F)C(=O)N1CC2CC1C2C(N1CCC2CC12C)=O 22716,N1(C(CCC2(NC(c3c(CC)cno3)=O)CCC2)=O)CC(C)SC(C)C1 22717,C12CCN(CC1F)C2=O.c1(CNC(C(C)OCCN(C)C)=O)c[nH]cc1C(F)(F)F 22718,N1(C(C2CC(C(=O)OC)C2)=O)CCOC2(CCC(F)(F)CC2)C1 22719,N1(c2scc(C(N3C(CNC(C4C(CO)C4(F)F)=O)CC3)=O)n2)CCCNC1=O 22720,c1(C(C)=O)ccc(C(=O)NC(C)(C)CCN(C(=O)CCS(C)=O)C)cc1 22721,CCCC(C(=O)NCC1(c2nn[nH]n2)CCCCC1)OCC 22722,c1(CN(C(CC2CCN(C(=O)Nc3nnc(C)o3)CC2)C)C)ccccc1C#N 22723,CC(C)C(O)C(=O)NC1CC12CC(NC(=O)C=Cc1ccsc1Br)C2 22724,O=C(CC1=CCN(C(C2(O)CCOC2)=O)CC1)Nc1cncc(C2CC2)c1 22725,c1(C(=O)NCc2occc2C(=O)NC2CN(c3ccncc3)C2)ncc(F)cc1F 22726,c1(C(C(=O)OC)C)ccc2c(c1)nc(NCC(c1cc(Cl)cc(Cl)c1)O)n2C 22727,C1(C(=O)NC(CC)CNC(c2ccc(CC3CC3)cc2)=O)CC(C)(C)OC1(C)C 22728,CC1=C(C)CC(C(N2CCOC(C(=O)NCC3(O)CCC(C)(C)C3)C2)=O)CC1 22729,c1(OC)cc(C(=O)NCC#CCNC(=O)CCc2ccc(Cl)nc2)ncn1 22730,C1(C(N(C)Cc2ccc(Br)s2)=O)CCCN(CCC(=O)Nc2ccccc2Cl)C1 22731,CCC(CC(=O)N1CCC(CCNC(=O)C(C)(CC)OC)C1)C1CCC1 22732,CC1(C)Cc2cccc(C(=O)NCC3CC(NC(C4(C)CC4)=O)C3)c2O1 22733,Cc1ccn2cnc(C(N3CCN(C(C4CCC4)=O)C(C)(C)CC3)=O)c2c1 22734,C(=O)(CC(C)(C)CC(=O)N(C1CN(C(=O)C(O)c2ccco2)CC1(C)C)C)OC 22735,N1(C(c2ccc(C)c(CO)c2)=O)CCC(C(=O)N2CCN(C)C(=O)C2C)=C(F)C1 22736,c1(C(N(C2CCN(C(=O)C=CS(C)=O)C2)CC)=O)ccccc1Cl 22737,C1(CNC(CSCC(C)C)=O)CC2(CCC2)CN1C(=O)CC(C)n1cccn1 22738,O=C(C#CC1CC1)Nc1ncn(-c2ccccc2)n1 22739,C1(C(N2CCCC2Cn2cc(C(c3nccn3C)O)nn2)=O)(CC)CCCC1O 22740,C1(NC(Cc2nc(CC)sc2)=O)CCN(C(c2ccncc2Cl)=O)C(C)C1 22741,c1(C(=O)NCC(C2(O)CN(C(C(C=C)O)=O)C2)(C)C)nc2ncccc2cc1C 22742,CCCC(O)CC(=O)N(C1CCCN(C(c2nccn2C(C)C)=O)C1)C 22743,C1(C(N2CC(O)(C(F)C(=O)N(C(C)C(F)F)C)C2)=O)(CC)CCOC1 22744,C1(C(=O)NCC(CNC(c2ccc(C3CC3)cc2F)=O)O)CC2(COCCO2)C1 22745,N1(C(CCCCC(=O)NC)=O)CCC2(C1)CN(C(=O)C(F)n1ccnc1)CCO2 22746,N1(CC(C)OC(=O)Nc2noc(C)c2C)CCSC(C)(C)C1 22747,S(=O)(=O)(c1ccc(=NCc2csc3cc(Cl)ccc23)[nH]c1)NC1C(C)CN(C)C1 22748,CCC(CO)(C(=O)N1CC=CC(C(=O)NOC(C)C)C1)OC 22749,Cc1cc(NC(C2CCCN(C(c3ccc(C)c(F)c3)=O)C2)=O)c(=O)n(C)c1 22750,c1(OCC(=O)NCCC(C)NC(=O)C(C)(Cl)Cl)ccc(F)cc1 22751,C1(CC(=O)NC(CNC(C2(COC)CCC2)=O)(C)C2CC2)C=NN(C)C1=O 22752,c1(CC=C)ccccc1C(=O)NC(C)(CSC)C(=O)NCCOC(F)F 22753,C(C(C(C)(C)C)NC(=O)Cn1c(C)csc1=O)NC(C1C(CC)C1)=O 22754,C(=O)(C(O)C(C)(C)C)N1C(C(=O)NC(COC)COC)CC2CC21 22755,C1(NC(CCC=CC)=O)CCN(C(C2(CO)CCCCO2)=O)CC1CC 22756,C1(C2CCC(=O)NC2)(C(N(C)CC2(O)CN(C(=O)C(F)C(F)(F)F)C2)=O)CCC1 22757,c1(C(N2C(C3CCCN(C(CCCC#C)=O)C3)CCCC2)=O)ccc(N)cc1F 22758,C1(C(=O)Nc2ccc(CC(F)CO)cc2)CNCCS(=O)(=O)C1 22759,c1(CC(=O)NCC2CC(NC(c3c(=N)cc[nH]c3)=O)C2)cc(O)nc(O)n1 22760,c1(CN(C)C(c2cnn[nH]2)=O)cnn2c1CN(C(=O)CC1CC1C(F)(F)F)CC2 22761,C(C)(C(=O)NC1(CN(C)C)CC1)(N(C(C(C)C1CCCC1)=O)C)C1CC1 22762,C1(NC(c2ccc([N+](=O)[O-])nc2)=O)COC2(CCN(C(C3CCC3)=O)CC2)C1 22763,C1(C(=O)NC(COC)C(C)(C)C)CCCCCCN1C(=O)C(F)CCC(C)C 22764,c1(C(N2C(C(=O)NCC)CCC2)=O)cc(OC)ncc1-c1cc(C)sc1C 22765,C1(OC)CC(NC(c2cncc(F)c2C)=O)CN(C(c2ccnc(C)c2C)=O)C1 22766,C1(=O)C(CCF)NCCCN1.C=CCC(=O)N(C1(NC(=O)OC(C)(C)C)CC1)C 22767,C1(CNC(c2cn(CC)nc2)=O)CCC(NC(=O)CN2CCSCC2)CC1 22768,C1(NC(C2CCC(C)(C)OC2)=O)CC1C1CCN(C(c2ccoc2Cl)=O)CC1 22769,c1(NCC2(C)N(C(=O)OC(C)(C)C)CC(OC)C2)oc2ccccc2c1Cl.OCC 22770,O=C(CC(Cc1cccs1)NC(=O)Cc1cc[nH]c1)NCc1ccc[nH]1 22771,c1(N2C(C(=O)Nc3c(C(=O)OC)nsc3)COCC2)ncc(C)c(C)n1 22772,c1(OC)cncc(NC(CC2(NC(C3(NC(N)=O)CC3)=O)CCC2)=O)n1 22773,CCCC(C(=O)NCC1CCC(NC(=O)C=Cc2nc(C)cs2)CC1)NC(C)=O 22774,N1(C(CC(C)(C)C#N)=O)CC2CC1CCC2NC(c1scnc1C1CC1)=O 22775,c1(OCC)ccc(-c2ccc(NC(=O)Nc3cc(C)cc(C)c3)nc2)c(C)c1 22776,N1(C(c2c(C)cccc2C)=O)CC2CCC(C1)C(NC(C1CC(F)(F)CS1)=O)C2 22777,N1(C(c2cn(CCOC)nc2)=O)CCOC2(CCN(C(=O)C3=COCC3)CC2)C1 22778,C1(NC(CCCC#C)=O)CCN(C(=O)COc2ccc(C)cc2C(C)C)CC1C 22779,Cc1c(C(=O)NC(CC2CC2)C(N2CC3C=CC2CC3)=O)cccc1C#N 22780,CC1CC=C(C(=O)NC(CC2CC2)C(=O)NCCCn2cnnc2)CC1 22781,C1(C)(C(N2CC(SCC)C2)=O)CCCN(C(=O)CC(F)(F)F)C1 22782,c1(C(N(CC(C)NC(C(COC)N(C)C)=O)C)=O)sc(C)c(Br)c1OC 22783,C1(NC(C(C)S(N)(=O)=O)=O)CN(C(=O)CCc2cnn[nH]2)CCC1(C)C 22784,c1(C(=O)Nc2cccc(N3CCCS3(=O)=O)c2)cccc(-c2ccccn2)c1F 22785,Cc1c(C(=O)NC(C)(C)C(=O)NCc2ccccc2)nc(O)c2ccccc12 22786,N1(C(CC2OCC(C)(C)OC2)=O)CC2(C1)CN(C(C1CCC(=O)N1)=O)CCO2 22787,c1(OCC=C)ccccc1C(N1CCCC1(C)C(=O)NCc1ccccn1)=O 22788,C1(CNC(C=CC(C)=O)=O)CC2CCC(C1)N2C(=O)CCCc1cccnc1 22789,Cc1ccc(C(F)C(N2CCCCC2CCNC(=O)CSCCC#N)=O)cc1 22790,C1C2CN(C=O)CC12.O=C(C(O)CN1CCCC1)NC1CCCCC1 22791,C1(C(=O)NC)CCN(C(C2(COC)CN(C(c3ccn(C4CC4)n3)=O)C2)=O)C1 22792,N#Cc1c(Cl)ccc(NC(C2CN(Cc3ccnc(O)c3)CC(F)(F)C2)=O)c1Cl 22793,C1(NC(C=CC=CCC)=O)CCC(O)CN(C(=O)CCC2CCN(C)C2)C1 22794,c1(C(=O)NCC(CNC(Cc2c(C)n(C)cn2)=O)C)ccc(S(N)(=O)=O)nc1 22795,CC(CC(C)(C)C)C(=O)NCc1ncc(C(=O)NCC2(O)CCN(C)C2)cn1 22796,C(CNC(=O)NC(c1cc(C)c(F)c(C)c1)C)(CCS(C)(=O)=O)OC 22797,N1(C(c2cnn(CC)n2)=O)CCCC(NC(c2cccc(C)c2Cl)=O)CC1 22798,C1(CC)CN(C(c2c(C)nn(C)c2N2CCCC2)=O)CCC1NC(=O)C(F)F 22799,c1(C(N(CC(CC)NC(C=CC)=O)CC)=O)cnn2cccc(Br)c12 22800,N1(CC(=O)NC2C(NCC(=O)NC3CC(C(F)F)C3)CCC2)CCOCC1 22801,C1(CN(C(=O)CCCNC(C)=O)CC)CCN(C(c2cc(C)cs2)=O)CC1 22802,CC1CCc2sc(C(N3CCC(NC(=O)CN(S(C)(=O)=O)C)C3)=O)cc2C1 22803,c1(NC(C(c2cc(C(=O)OC)ccn2)N(CC=C)C(C)C)=O)ccc(F)cc1C 22804,C(=O)(CC(O)C(C)C)NCC1(C(=O)N(CCC(C)O)C)CC(=C)C1 22805,C1(CN(C)Cc2cnn(C)c2)CCN(C(=O)C(C2CCOCC2)=O)CC1 22806,C(=O)(C1CCCn2cnnc21)NCC1(F)CCN(C(c2nc(C)nc(O)c2)=O)C1 22807,C1(CNC(c2cnn(CC(C)C)c2C(F)F)=O)CN(C2CC2)CCC1(C)C 22808,c1(C(N2CCC(C3N(CC#C)CCC3)CC2)=O)cc(C#N)[nH]c1C 22809,C1(C(N(C)CC2(CC(C)C)CC2)=O)CC2(CCN(C(C3CCCCS3)=O)C2)C1 22810,C(=O)(C(C)CC(=O)N1CC(C)(C(=O)Nc2cncc(OC)c2)C1)OC 22811,c1(NC(C(=O)N(C)Cc2c(OC(F)F)cccc2Cl)=O)cccc2c1CCC2 22812,c1(C(C)(C)C)nc(=NCC2CCCCN2C(=O)Cn2cncn2)s[nH]1 22813,C1(NC(c2cc(C)ncc2)=O)CCN(C(C2OCCCO2)=O)CC1F 22814,c1(NC(CSCC(=O)OC)=O)c(Cl)cc(OC)cc1Cl.c1(C)nnc(C)o1 22815,CCC(C)C(C)C(=O)N(C)CC1CCCCN1C(=O)C(C)CC1CCCC1 22816,CC(C)(C(=O)NCCC1CN(C(C2CCS2(=O)=O)=O)C1)c1ccccc1 22817,Cc1cc(N2CCC(NCCC3CCNC3=O)CC2)ccn1 22818,n1(CC(N2CCCC(N(C(C3CC3CF)=O)CC)C2)=O)cc([N+](=O)[O-])cn1 22819,Cc1cc(Cl)c(C(=O)NC2CC3CC(NC(C4C5(CC5)C45CC5)=O)C3C2)cc1C 22820,Cc1ccc(CN2CCCC2CC(N2CCCC(C)C2)=O)cc1[N+](=O)[O-] 22821,c1(C(=O)NCC(C)(C)NC(CC(=C)C)=O)ccc(CC)nc1C 22822,Cc1nc2nccc(C(=O)NC3CCCC(CNC(C4CN(C)C4)=O)C3)n2n1 22823,N1(C(CC(C)N(C)C)=O)CCC2(CCCN2C(c2cnc(C3CCC3)s2)=O)C1 22824,c1(C(=O)NC2(CO)CCN(C(=O)CC3C=CCC3)C2)cccc2ccsc12 22825,Cc1ccncc1C=CC(=O)NC1CC(NC(=O)C(=C2CCCCC2)F)CC1O 22826,CC(CCCCNC(C1CCOC1C1CC1)=O)NC(c1ccc(F)nc1)=O 22827,C1(CNC(C2CCCC2(F)F)=O)COCCN1C(c1ncccc1O)=O 22828,C1(C)(C(=O)Nc2c(C)cc(Cl)cc2)CN(C(=O)C(C)OC(C)(C)C)C(C)(C)C1 22829,C1(C(N(CCN(C(=O)CC2CCC(=O)N2)C(C)C)C)=O)CCNC(=O)C1 22830,N1(C(CCC(C)C)=O)CCC2(CCCCN(C(=O)Cn3cc(C4CC4)nn3)C2)C1 22831,C1(C(=O)NCCCNC(C(C)NC(c2ccco2)=O)=O)C(C)(C)OC1(C)C 22832,CCCC(CC(C)C)C(=O)N1CC=CC1C(=O)NCC(=O)OC 22833,c1(NC(CCC(=C)C)C)ccc(S(=O)(=O)NCc2cscc2C2CC2)cn1 22834,C1(C(=O)NCCC2COCCN2C(c2cnc(SC)n2C)=O)(CC)CC(C)(C)C1 22835,Cc1nc2cncc(C(=O)NC34CCCN(C(=O)CCNC(N)=O)CC3C4)c2[nH]1 22836,C(=O)(C1=NOC(C)(C)C1)NCC1(NC(C2C(c3c(C)cccc3)C2)=O)CC1 22837,C(=O)(CCCc1ccncc1)N(CC(CC)NC(=O)C(C)(C)C1CC1)C 22838,N1(C(C(C)(C)CF)=O)CCC2(CCCC2CNC(c2ccnc(O)c2)=O)CC1 22839,S(=O)(=O)(c1c[nH]c(C(=O)NCC2CC(C)N(C(c3cnns3)=O)C2)c1)NC(C)C 22840,CC1CCN(C(c2cccn3ccnc23)=O)C(C)C1NC(c1nn(C)cc1Cl)=O 22841,N1(C(c2cccc(CC)n2)=O)CCOC2CN(C(=O)C(=O)CCC(C)C)CC12 22842,c1(CNCC23N(C=O)CCC2CC3)nccn2nccc12.c1(CO)ccccc1 22843,C(=O)(C1=Cc2ccccc2OC1)N(CC(C)NC(=O)C(N1CCCCC1=O)C)C 22844,c1(OCCCC)ccc(C(=O)NCCCc2cn(CCC(F)(F)Cl)nn2)cc1 22845,c1(C(C(N2C(CCOC)CN(C(=O)CC3CC3)CC2)=O)C)ccc2c(c1)OCO2 22846,c1(C(C)=O)cc(O)cc(O)c1C(=O)N(C)C.C123C4CC1C1C(C4C21)NC3=O 22847,c1(OC)cc(CN2CCC(C(=O)Nc3ncn(C)n3)C(O)C2)c(Br)cn1 22848,c1(C(=O)NCC2C(NC(C3(CC#C)CCCC3)=O)C2)cnc2[nH]cnc2c1 22849,C(CNC(C1(C(F)F)CC1)=O)(C(C)C(C)C)NC(c1cc(C)c(C)[nH]1)=O 22850,N1(C(C(C)OC2CCCCCC2)=O)CCCC2(NC(=O)CC3(C)CC3)CCCC12 22851,C1(C(=O)NC2CC2)CC(F)CN1C(=O)CCCCc1cn(C2CCOC2)nn1 22852,N1(C(c2cn(CC)nc2)=O)CCC(C)(C)C1CC(N1CC(C)(C#N)C1)=O 22853,S(=O)(=O)(c1cccc(-c2nnc(SCCO)o2)c1)N(C)C1CC1 22854,C1(NC(Cc2c(C)cco2)=O)CN(C(=O)CC2CCCOC2)CC2(CC2)C1 22855,C(C1C(C(=O)N(C)CCOCCNC(c2sc(CO)nc2C)=O)C1(C)C)=C(C)C 22856,O=S(c1ccc(NC2COc3ccccc32)cc1)C(F)(F)F 22857,c1(C(=O)NC2CC3(CN(C(C4(SC)CC4)=O)C3)C2)cc2nc[nH]c2cn1 22858,CCC(CC)CC(=O)OCc1nn(C)c(Br)c1C 22859,C1(C(=O)NC(C)C(=O)N(C)CCN(C)C(C2CC(O)C2)=O)CCCCC1 22860,Cc1ccc([N+](=O)[O-])c(C(=O)NC2CCCN(C(c3c(C)nsc3C)=O)C2)c1C 22861,CCC(CC)CCCC(=O)NC(C1(O)CCN(C(c2noc(CC)c2C)=O)C1)C 22862,C1(NC(c2csc(Cl)n2)=O)CC(O)CN(C(c2ccc(OCC3CC3)nc2)=O)C1 22863,C12(C(=O)NC(CC=C)CO)COCC1CN(C(c1cnns1)=O)C2 22864,N1(C(C(CCC)(C)O)=O)CC(=O)NC2(CCOCC2)C1 22865,C1(NC(C2(N=[N+]=[N-])CC2)=O)CCCN(C(c2cc(C(F)(F)F)cs2)=O)C1 22866,C=CCC(C)(C)CC(=O)NCCC1CCC(NC(c2cc3ncccc3s2)=O)C1 22867,C1(NC(c2nc(C)sc2)=O)CN(C(C2C=CCC2)=O)CC12CCS(=O)(=O)CC2 22868,C(=O)(C(O)C1=CCCCC1)N1CC(C)(OCC(N2CC3CCCC2C3)=O)C1 22869,C1(C(N2C(CNC(c3ccnc(C)n3)=O)CCCC2)=O)CCc2ccccc2O1 22870,C1(C(C)NC(=O)Cc2cn[nH]c2)CCN(C(c2cnnn2C2CCCC2)=O)CC1 22871,N1(C(c2c(C)ccnc2)=O)CCC2(CC1)CC(NC(C1CCN(C)C1C)=O)C2 22872,c1(OC)c(CC(=O)NCCN(CC(C)O)C(C2CCCCS2)=O)cccc1F 22873,C(CC(=O)NCC1(COC)CC1)(C(C)C)NC(c1ccn(CC)c1C)=O 22874,c1(C(=O)NCC2CN(C(C3C(CCOC)C3)=O)C2)ccc(O)c(CC(C)C)c1 22875,C(C)(N=c1cc(C)nc(C(F)F)[nH]1)c1[nH]nc(NC(=O)OC(C)(C)C)n1 22876,N1(C(CC2(CN(C)C)CCC2)=O)CCC(C(F)F)(CNC(C2CCCCC2)=O)C1 22877,c1(C(=O)NCC(C)N(C(=O)Cc2cccs2)CC)cc(CNC(C)=O)on1 22878,CCC(C)(C)C(C)NC(C1CCN1C(=O)C(C)NC=O)=O 22879,C=CC1OCCC1C(=O)NCCC1CC(NC(=O)CCC2CC2C)C1 22880,c1(OCC)cc(Cl)ccc1C(N1CCN(C(=O)CCC=CBr)CC1CF)=O 22881,Cc1cn(C)nc1C(=O)NC(CC1CCCC1)C(=O)NC1CCOCC1F 22882,C(=O)(C1COc2ccccc21)NC1CCN(c2ncnc(C)c2Br)CC(C)(C)C1 22883,CC(C)C(O)C(C)C(=O)NCC(O)CC(N1CC2CC(C1)N(C)C2)=O 22884,N1(C(c2[nH]cc(C(C)(C)C)c2)=O)CCC2CN(C(c3ncc(F)cn3)=O)C2C1 22885,C(=O)(CC(O)CC(C)C)N1CCN(C(C(CCCOC)C)=O)CC1c1ccco1 22886,c1(C(N2CC(CNC(CC=C=C)=O)C(O)C2)=O)c(-n2cccn2)cccc1F 22887,c1(C(=O)NC2C(NC(=O)CC3CC4(CC4)CO3)CCC2)ccc2c(c1)CNC2=O 22888,C#CCCC(O)C(=O)N1CC(F)CC1CNC(C1(S(N)(=O)=O)CC1)=O 22889,c1(C(=O)NC2C(F)CCN(C(C3CC(=C)C3)=O)C2)ccc2nc(C(F)F)[nH]c2c1 22890,C1(NC(=O)C(O)C2CCC2)CC=C(C(=O)NC2CCCCC2O)C1 22891,c1(C(=O)NCC(C(C)(C)C)NC(C(C)OCC#C)=O)ccc(C#N)c(O)c1 22892,N1(C(CC2(OC)CCC2)=O)CCCC(C)(C)C1C(N1CC(O)C(O)C1)=O 22893,c1(C(=O)NCC2(F)CN(C(C3C4CCOCC34)=O)C2)ccc2ncnc(O)c2c1 22894,CCCCCCCCCCCCCCCOC(C1CC(=O)NC2(CCC2)C1)=O 22895,c1(CCCNC(C2CCC(F)CN2)=O)ncc(Cl)cc1Cl 22896,c1(-n2cnc(C(N3CCC(NC(CCC=C)=O)C3)=O)n2)ncccc1F 22897,N1(C(c2cc(Cl)nc(Cl)c2)C(=O)NC)CCc2[nH]nc(CO)c2C1 22898,c1(CN(C2CCCC2)C2CC2)cc(CCNC(=O)CC2CC(COC)C2)on1 22899,Cc1oc(CNC(C2CN(C)C2)=O)nc1C(=O)N(C)CCC1CCC1 22900,c1(C(=O)NCC2(CN(C)C)CCC2)ccccc1-n1cc(CCS(N)(=O)=O)nn1 22901,C12(C(N(CC(CCC)C)C)=O)C(NC(c3cocn3)=O)C3CC1C2C3 22902,N1(C(CO[Si](C)(C)C)=O)CC(O)CC1CNC(C1(C(F)(F)F)CC=CC1)=O 22903,C12(COC)CC(C(=O)NCCCC3CCCN3C(=O)C(C)CSC)(CO1)C2 22904,C1(CC(=O)NCC(O)C2(Cl)CC2)CCCN1C(c1cnsn1)=O 22905,c1(OCC)cc(CN(C)Cc2noc(C3CNC3)n2)cc(F)c1 22906,Cc1nnn(CC(=O)NCCC(=O)NCc2ccn(C3CC3)n2)n1 22907,N1(C(C(C)(C)NC)=O)CCC2(CC1)CC2NC(c1cnn(CCCOC)c1)=O 22908,c1(CC)nc[nH]c1C(=O)NCCCn1cc(CCC2CCCCO2)nn1 22909,Cc1csc(Cl)c1C(=O)NCC1CN(C(=O)CC(c2cccc(F)c2)O)CC1C 22910,c1(C(=O)NC2CCC(CC(=O)NC3(CC=C)CC=CC3)CC2)cc2ccccn2n1 22911,c1(OC)ncccc1-c1cn(C2CCC(C(N3CCC(CC4CC4)C3)=O)C2)nn1 22912,c1(C(=O)NC(CN(C(C(CCC)O)=O)C)(C)C)nn(C)c2ccc(Br)cc12 22913,CC(C)CC(C(=O)N1CCCC(CNc2ncccc2C#N)C1)C(N)=O 22914,N1(C(c2occ(C)c2)=O)CC2OCCN(C(C3CCCCS3(=O)=O)=O)C2C1 22915,N1(Cc2cc(C(=O)OC)c(F)cc2)CCc2c(C(N3CCCC3C)=O)cccc2C1 22916,N1(C(CCCCC)=O)CC2(C1)CN(C(C1CCCC1)=O)CC2CO 22917,C(=O)(C(CCCC)C(C)C)N1CCC(C(=O)NCCOCC=C)C1CC 22918,C1(NC(=O)CCOCC(F)F)CCCC(NC(c2coc(C3CCC3)n2)=O)C1 22919,Cc1cn2c(C(=O)NCC3CC3CNC(=O)C=C3CCOCC3)c(C)nc2s1 22920,CC1(C)C(NC(=O)C(=O)NCc2ccc(Cl)cc2)CCN1C(=O)C(O)CC1CC1 22921,N1(C(C(CCC(C)C)F)=O)CC(C)CN(C(=O)C=Cc2ccc(=N)[nH]c2)C(C)C1 22922,c1(C(=O)NC2C(NC(C3=CCCC3C)=O)CCC2)cc2c(s1)CCCCCC2 22923,N#Cc1ccc(NC(C2CN(C(=O)CCc3ccccc3F)CCS2)=O)cc1Cl 22924,N1(C(CC=C)=O)CCC(N(C)C(C2CCN(c3cnn(C)c3)C2=O)=O)C2(CC2)C1 22925,C(=O)(C(CCC(C)C)NC(C1CC2(CC(=O)C2)C1)=O)N1CCN(CCOC)CC1 22926,CC(O)CCC(=O)N(C1CCC(NC(=O)CCc2ccccc2C(N)=O)CC1)C 22927,C1(CC#C)(C(=O)NC2CCC2NC(C2CN(c3nncs3)C2)=O)CCCCO1 22928,C1(C)(CC)CC(NC(c2cc(N)cc(O)n2)=O)CN1C(=O)CSc1ccccn1 22929,c1(C(=O)NCC(C(=O)NC2CCN(CCCSC)C2)OC)ccc(F)cc1C 22930,CC(C)CC(C(=O)NC(COC(C)C)C(=O)NC1CC(C)(C)OC1(C)C)C(N)=O 22931,C(=O)(CC(CNC(c1ccc(C2CC2)o1)=O)C1CCC1)NCC(CC)(C)O 22932,Cc1ccc(C(=O)NC2CN(C(C3CC(n4cnnc4)C3)=O)C2)cc1Cl 22933,c1(C(N(CCN(C(CCC)=O)C)C)=O)c(NC(C2CC2C)=O)sc(C)c1C 22934,c1(C(=O)OCC23COC(CF)(C2)C3)sc2sccc2c1Cl.C(=O)C1CC1 22935,CCCCC(CNC(c1cc(C#N)c[nH]1)=O)NC(=O)COCC1CCOC1 22936,c1(N2CC(CC)OCC2)cc(C(C)=O)ccc1Br 22937,CC1=C(C(=O)NC2CC2CNC(C2(C)CCC2)=O)CCCC1 22938,N1(C(C(COCC)C)=O)CC(N(C)C(c2cnc(SC)nc2O)=O)C2(CC2)C1 22939,c1(OC)cc(C(=O)O)ccc1NC(=O)C(N1CC(C)CC(C)C1)=O 22940,c1(C(c2n(CCOC)nnn2)NCC(c2cccs2)C)nc(C)c(C)[nH]1 22941,CC1CCN(C(=O)CNC(N)=O)CCN1C(C1C2CCN1CC2)=O 22942,c1(CNc2c(C(=O)NCC)nccc2)oc2ccccc2c1C 22943,C(c1ccc2c(c1)COCC2)=CC(N1CC2CCN(C(C(C)C)=O)CC21)=O 22944,N1(c2nnc(C)s2)CCC2CC(C(N3CCC(c4nncn4C)CC3)=O)C2C1 22945,C1(C2CCC2)(C(N2CCC(CNC(c3cc(C4CC4)[nH]n3)=O)(CO)C2)=O)CC1 22946,N1(C(c2c(C(C)C)nn(C)c2)=O)C(CNC(=O)COCC2CC2)CC2COCC12 22947,c1(CNC(CN2CCP(CC)(=O)CC2)=O)ccc2c(c1)CCN2S(C)(=O)=O 22948,CC12CC(C(N3CCC(F)(CNC(=O)C4=CCCOC4)C3)=O)(CCO1)C2 22949,C1(NC(C2C(CC)C2)=O)CCC2(CC1)CCN(C(=O)C(C)C(C)COC)C2 22950,N#CC1(C(=O)NCC2(CCNC(c3cc(C4CC4)cs3)=O)CC2)CCCO1 22951,C(C)(C)(CCC(=O)N1CCCC(COC)(NC(=O)Cc2ccco2)C1)OC 22952,C12(C(=O)NCC3CN(C(C4CCCC45CCC5)=O)CCO3)C3CC(CC13)C2(F)F 22953,c1(C(=O)NCCN(CCCN(C)C)C(C2C(C)C2C)=O)csc(Cl)c1 22954,N1(C(c2ccc(SC)o2)=O)CCCC2CN(C(c3noc4c3COCC4)=O)CCC12 22955,C=CC(C(=O)NC(C1CCCN1C(C1CC1(C)C)=O)C)OC 22956,CC(C(=O)N1CCC(C(C)C(=O)N(C2CC2)Cc2ccoc2)C1)C(F)F 22957,C(C1c2ccccc2CCN1C(C1CCCS(=O)(=O)C1)=O)NC(COCC)=O 22958,Cc1ccc(F)cc1CN(C1C2CCC1CNC2)C(c1ccnc(C(N)=O)c1)=O 22959,C(=O)(C(C)(O)CCN(C)C)N1C2C(CNC(C=CCCC)=O)C(C2)C1 22960,C1(C(N2C(CN(C(c3c(CC)non3)=O)C)CCCC2)=O)Cc2ccncc2C1 22961,c1(C(=O)OC(c2ccc(F)cn2)CC)cc(C(F)F)cc(C(F)(F)F)c1 22962,S(=O)(=O)(c1ccc(F)c(F)c1)N1CCC(NCc2ccc(CC)nc2)C1 22963,Cc1cc(O)ncc1C(=O)NCCC1CC(C(=O)NCCC(F)(F)F)C1 22964,CC1(C#N)CCN(C(=NC2CCC2)NC2CCN(S(C)(=O)=O)C2)CC1 22965,CCC(C)C(O)C(C)C(=O)NCC(C)=CC(N1CCC(O)(C(F)F)C1)=O 22966,c1(C(N2CCC(C3(NC(C4CC4(F)F)=O)CC3)C2)=O)ccc2ncccc2n1 22967,N1(C(c2n[nH]c(CC)c2Cl)=O)CCCC(O)(CNC(C2CC23CC3)=O)CC1 22968,N1(C(c2c(CC)cns2)=O)CC(N(C(=O)C(C2CC2)SC)C)C2(CC2)C1 22969,N1(C(C=CC(=O)OCC)=O)CCN(C(c2coc(Br)c2)=O)C(CF)C1 22970,c1(CC(N2CC(CNC(C(C)C)=O)OCC2)=O)ccc2ccncc2c1 22971,CCCC(C)(O)CNC(C1(CNC(=O)C(n2ccc(C)n2)C)CC2(CC2)C1)=O 22972,C1(C(C(=O)O)NC(c2nc(CCP(C)(C)=O)sc2)=O)CC2C=CC1C2 22973,C1(N(C(=O)CN(C)C2CC2)C)CCN(Cc2nccc(CO)n2)CC1 22974,c1(SC)ccc(CN(C(c2cc(C)ns2)C(=O)NCC2CCCO2)C)cc1 22975,C=C(CNC(=O)C(C)(C)C1CCCC1)CCN(C(=O)CC1(C(F)(F)F)CC1)CC 22976,C(C(=O)N(C1CCN(C(C2(OC)CCCC2)=O)C1)CC)(C(C)C)SCC 22977,C1(CNC(C(CC=CCC)C)=O)CN(C(c2cc(Cl)nn2C)=O)CC1(F)F 22978,c1(C(=O)NCCC2CN(C(C3CCCS3)=O)CCO2)coc2c1COC2 22979,N1(C(c2cn(CC=C)nc2)=O)CC(O)CC1CNC(C1CC1C(=O)NC)=O 22980,Cc1nc2[nH]c(C(N3CC4CCC(NC(=O)CCNC(N)=O)(C4)C3)=O)cc2s1 22981,N1(C(C(C)OCC(F)(F)F)=O)CCC2(CC1)CC2CNC(=O)CN1CC(C)(C)C1 22982,Cc1cc(NCCc2ncc(Br)cn2)ncc1S(=O)(=O)NC(C)(C)C1CC1 22983,C1(NC(C2C(NC(CCc3n(C)ccn3)=O)COC2)=O)CCCCC12CC2 22984,N1(C(c2cc(OC)nc(F)c2)=O)CCN(C(c2c[nH]nc2C(C)C)=O)CC(O)C1 22985,c1(NC(=O)NCCC(COCC2C(COC)C2)C(F)(F)F)ccc(F)cc1 22986,C1(NC(=O)C2=CCCOC2)CC2CCC1N(C(c1ccc(N3CCC3)nc1)=O)C2 22987,N1(C(c2c(-c3cn(C)nc3)onc2)=O)CC=C(CCNC(=O)C=C2CCC2)CC1 22988,C1(O)(C(C)NC(C(C)OCC=C)=O)CN(C(=O)C=Cc2ccc[nH]2)C1 22989,c12ccccc1O2.C(=O)(CCCOC(=O)Cc1ccccc1)OCC 22990,c1(C(N2CCCC(CCNC(C(CN(CC)CC)F)=O)C2)=O)cnc(O)cc1O 22991,c1(C(N2C(CN(C(C(CSC)(C)C)=O)C)COCC2)=O)nsc2ccc(C)cc12 22992,c1(NC(C2CC2C(=O)Nc2ccc(C3CC3)cc2)=O)cncc(C2CC2)c1 22993,c1(CNC(CN(C)C(c2nnc(-c3c(F)cccc3F)s2)=O)=O)cc2c(s1)CCC2 22994,CC1CCC(C)N1CC(=O)N(CC(N)=O)C(c1ccc(N(C)C)cc1)=O 22995,c1(C(CNC(=O)CCc2ccsc2Cl)NC(=O)C=CCF)cccc(F)c1F 22996,N1(CCC(=O)NC2CC(C)(NC(C3C=CCCC3)=O)C2)CCCS1(=O)=O 22997,c1(C(=O)NC2(CCCCNC(c3c(C)nns3)=O)CC2)cc2ccccc2n1C 22998,Cc1cccc(SCC(=O)NCC(C(C)C)NC(=O)C(C)(C)N2CCOCC2)c1 22999,c1(CC(=O)OC)ccccc1C(=O)NC1(CNC(=O)C(F)CC2CCCC2)CC1 23000,C1(C(N(CC(CN(C(=O)CC2CC(F)(F)C2)C)O)C)=O)CCC(F)(F)CC1 23001,CC(C)CC(F)C(=O)NCC1C2CCC(C2)N1C(C1(CCOCCO)CCC1)=O 23002,c1(OC)cc(F)cc(C=CC(=O)N(C(C)CNC(=O)C2=CCOC2)C)c1 23003,CCC(C)(CCNC(c1nocc1C)=O)NC(=O)COC1(C)CCCC1 23004,N1(C(c2cc(CCC)ncc2)=O)CCCC(C2CC2NC(C2CC=CCO2)=O)C1 23005,c1(CN(C(=O)C(C2CCC2)NC(C2C=CCS2)=O)C)ncc[nH]1 23006,C(=O)(C(C(C)(C)S(=O)(=O)N1CCC(CCC#N)CC1)NC(=O)OC(C)(C)C)NC 23007,N1(C(C(C)(C)NC(C2C(C)C2)=O)=O)CCc2ncccc2C1 23008,N1(C(C2CCC(=O)N2)=O)CC2CC3CC2C1C3NC(=O)C(F)C1CCOC1 23009,CC(C)(O)C(C(=O)NOC1CC1)NC(c1ccc(=O)n(C)c1)=O 23010,C(=O)(C(O)CCCC)N(C)CC1OCCN(C(C2(C=C)CC2)=O)C1 23011,N1(C(C=CC)=O)CCC2CN(C(C3CCN(c4nccn4C)C3)=O)C2C1 23012,C1(C(N(C(C)CNC(C2(CCF)CC2)=O)C)=O)CCC(NS(C)(=O)=O)C1 23013,c1(NCc2cc(C)cc(N)c2)cc(Br)ccc1S(=O)(=O)N1CCCNC(=O)CC1 23014,N1(C(c2n[nH]cc2Br)C(=O)NCc2cccc(OC)c2)CCNC(=O)C1C(C)C 23015,C123CC(C1)(C(C)O2)N3.C1(C(N(C2CCC2)CC)=O)CN(CC(C)C)C1 23016,c1(C(=O)NC2CCC3CCN(C(CCOCC)=O)C32)cc2c(=O)[nH]c(C)cn2n1 23017,C1(OC)CN2CCCC2(C(=O)NC2CC(NC(c3c(Cl)cccc3Cl)=O)C2)C1 23018,N1(C(COCc2onc(CC)n2)=O)CC2CN(C(c3coc(C#N)c3)=O)CC2C1 23019,N1(C(C=C(CC)CC)=O)CC(CNC(C2(CO)CCOCC2)=O)C2(CCC2)C1 23020,N1(C(C2(CC=C)CCCN2C(=O)C(CC)NC(N)=O)=O)CC(F)(F)C(F)(F)C1 23021,C#Cc1ccc(C(=O)NCC2CCN2C(C2CNC(=O)N2)=O)cc1F 23022,CC1=CCSC1C(=O)NCC(C1CC1)NC(c1cnc(C(C)C)[nH]1)=O 23023,Cc1ncnc(C(N2CCC(NC(=O)CC3C=CCCC3)C2(C)C)=O)c1C 23024,C1(NC(CC)=O)(CNC(C2CCN2S(C)(=O)=O)=O)CCC(C)(C)CC1 23025,C1(O)(CC(N)=O)CCN(C(c2cccnc2O)C(=O)Nc2ccccc2Cl)CC1 23026,c1(C(N2C(CNC(C3N(C)CCCC3)=O)CC(O)C2)=O)ccc(N)c(Cl)n1 23027,C1(CN(C(CC(=O)OCC)=O)C)CN(C(C2(C)CCN(C)C2)=O)CCO1 23028,c1(C(=O)NCc2cn(C3CCN(C(C=C(CC)C)=O)C3)nn2)ccccc1C 23029,Cc1cc(N2CC(F)(F)CC2CNC(=O)C(c2cccnc2)O)n2ncnc2n1 23030,S(=O)(=O)(c1ccccc1Cl)NCC(=O)NCCN(C)C(c1ccns1)=O 23031,c1(CC(N2CCN(CC3CCCN(C(COC)=O)C3)CC2)=O)csc2nccn12 23032,S(=O)(=O)(c1cccc(=NCC(C)c2cccs2)[nH]1)NCCCCCC(=O)NC 23033,N1(S(CCOC)(=O)=O)CCC(N=c2nc[nH]n3cc(Br)cc23)C1 23034,C1(NC(c2ccn(C(C)C)n2)=O)CC(CNC(c2cc(C(N)=O)cs2)=O)C1(C)C 23035,C1(CNC(c2cccc(C)n2)=O)CN(C(=O)C(C)(C)C2CCCO2)CCN1C 23036,C1(C(C)C)CCC(NC(c2nc(NS(=O)(=O)CC#N)cn2C)=O)CC1 23037,C1(NC(CCCCCC)=O)CC2CN(C(c3cc(C)n(C(C)C)c3)=O)CC2C1 23038,c1(C(=O)NCC2OCCCN(C(C(C(C)C)F)=O)C2)ccc2c(c1)C(C)(C)CO2 23039,C1(S(N)(=O)=O)(C(=O)NCCCNC(C2(C(=O)OCC)CC2)=O)CC1 23040,C(=O)(CC(C)CNC(C1CCC(=O)N1)=O)NCc1nnc(CC)s1 23041,C(CO)(C(F)(F)F)NC(C(Cc1cc[nH]n1)NC(=O)CCn1cncn1)=O 23042,N1(C(C=C(C)c2cccs2)=O)CCN(C(c2ccc3cc[nH]c3n2)=O)CCC1C 23043,C1(C(N2C(CCNC(c3nc(C4CC4)cs3)=O)CCC2)=O)CCC2(CCC2)C1 23044,c1(OC)cccc(C(N2CCC(CF)(NC(=O)Cn3cccn3)C2)=O)c1 23045,c1(NC(C2C3CC2N(C(c2cnc(Cl)cc2I)=O)C3)=O)nc(Br)ccc1Cl 23046,N1(C(CC(C(C)C)O)=O)CC(C)(CNC(=O)COCCCN(C)C)CC1(C)C 23047,C#CCCCCC(=O)NCC(CC(=O)N(CC(=O)OC)CC1CC1)C1CCC1 23048,N1(C(CC#C)=O)CCN(C(c2[nH]c(C)cc2C)=O)CC1CC1CC1 23049,Nc1ccc(NC(N2CC(CC(=O)C(=O)O)C2)=O)cc1Cl 23050,c1(C(=O)NC(C2CCCC2)CNC(C2(CC)COC2)=O)ccc(F)c(C)c1Cl 23051,C1(C(=O)NCCC2CCN(C(=O)C(C3CCC3)C3CCC3)C2)CC(F)C(=O)N1 23052,c1(CNC(c2cc(CC)on2)=O)ccc(CNC(C2(C)COC2)=O)cc1F 23053,C1(CC(=O)NCC(C)NC(c2nnc(C(C)(C)C)o2)=O)CCOCC1 23054,c1(SC)cc(F)ccc1C(=O)NCCOCCNC(=O)COCC(F)F 23055,C1(N(C(CSC)=O)CCO)CCN(C(c2cc(SCC3CCC3)c[nH]2)=O)C1 23056,N1(C(C(CC)O)=O)CCN(C)CC1C(=O)NOCC(C)(C)O 23057,CN1CC(NC(=O)Cc2c[nH]c3cc(F)ccc23)CCc2ccccc21 23058,c1(C(C(N2CC(N(C(CCC#C)=O)C)C2)=O)C)cccc(Br)c1 23059,c1(C(N2CCCC3CN(C(C(COC)O)=O)CC32)=O)cc(F)c2ncccc2c1 23060,c1(C(=O)NCCC(=O)NC(C(C)NC(c2ccsc2Cl)=O)(C)C)ncc(F)cn1 23061,Cc1ccc(-c2cn(C(CC)CC3CC(C)CCN3C(=O)C(O)C(F)F)nn2)c(Cl)n1 23062,c1(C(N2CC(NC(C3C(C(C)C)C3)=O)C3(C2)CC3)=O)cc(Cl)cc2ccncc12 23063,N1(C(CCCOC(C)C)=O)CC2(CC(NC(c3csc4cncn34)=O)C2)C1 23064,C1(N(C(C2C(OCC)C2)=O)CC)CCN(C(=O)Cc2cccc(F)c2)CC1 23065,N1(C(C(CCCOC)NC(=O)CCC(C)SC)=O)CCC2(CCC(OC)C2)C1 23066,CN1CC2C(CCN2C(c2cc3n[nH]cc3cc2Cl)=O)C2=CCC1CC2 23067,C(CN=c1nc2scnc2c(NC2CC2C2CCCC2)[nH]1)NC(=O)NCC 23068,Cc1ccc(C(C#N)C(=O)N(c2cnncc2C)C2CC3(CNC3)C2)nc1 23069,c1(C(=O)NCC2C(C)CCN(C(C34CC(C)(C3)C4)=O)C2)ccc2nn[nH]c2n1 23070,c1(C(N2CCCN(C(C3CC4CCC3O4)=O)CC2)=O)ncc(F)cc1F 23071,n1(C(C)C)cc(C(=O)NC(C2CCOC2)CNC(c2cc(C(F)F)no2)=O)nn1 23072,N1(C(c2c(OC)cc(F)cc2)=O)CCCN(C(=O)CC(C)C)C(C)C1 23073,C1(NC(C2CCOCC23CCC3)=O)CC2CCC1CN(C(=O)C1=COCCC1)C2 23074,c1(NC2CCN(C(=O)Oc3ccc(C)cc3)C2)cc(C(F)F)c(Br)cn1 23075,C1(C(=O)NCC2C(CNC(Cn3ccc(C)c3)=O)C2)CCC2(CC2)C1 23076,C1(C(N2CCC(CCC(=O)NC(c3n(CC)ncn3)C)C2)=O)CC2(C1)CC21CC1 23077,N1(C(C2COC(=O)O2)=O)C(CNC(C2(C(F)F)CC2)=O)CC2COCC12 23078,C1(CC(=O)Nc2cccc(Oc3nccs3)c2)CCC2(CCCC2)CC1 23079,N1(C(c2cnc(C(C)C)nc2)=O)CC(NC(C2CCCC2O)=O)CC(C)(C)C1 23080,N1(C(c2c(C)ccnn2)=O)C2CCCC1CN(C(c1cnc(O)cc1O)=O)C2 23081,CCS(=O)CC(=O)NCC1COCC1NC(=O)CSc1cn[nH]c1 23082,c1(CC)c(C(=O)NCC2CCC(C(=O)NC3(CCO)CCC3)O2)nnn1C 23083,C(=O)(C(CNC(C12COCC1C2)=O)CC(C)C)NCC(CC)(C)C 23084,Cc1cc(C(=O)NC(C)CCNC(=O)C=Cc2cnccc2C)ccc1C#N 23085,c1(-c2cc3c(cc2)N(C(COCC)=O)CC3)ccc2c(c1)n(C)c(=O)n2C 23086,c1(CNC(c2occc2CNC(C2C=CCCC2)=O)=O)ccc2n[nH]cc2c1 23087,c1(C(N(CCC(C)NC(c2csnn2)=O)C)=O)ncccc1C1CC1 23088,n1(CC)c(C)cc(C(=O)N(CC(C)NC(=O)C(C)(O)Cc2ccccc2)C)c1C 23089,C1(CCNC(N(C(C)CN2CCOCC2)C)=O)CCCS1(=O)=O 23090,c1(C(C)(C)C)nc(=NC2CCN(C(=O)C(c3ccc(Cl)cc3)(C)C)C2)s[nH]1 23091,CC(O)C(C)(C)C(=O)N(C)CC1CN(C(=O)CC2(N(C)C)CCCC2)CC12CC2 23092,C1(F)(C(=O)NCC23CC(CNC(C(CC)COC)=O)(OC2)C3)CCC(F)(F)CC1 23093,c1(CC)[nH]c(=N)sc1CNC(=O)C=CBr.N12CC(CC1C)SCC2=O 23094,C(=O)(C#CC1CCCCO1)N(CCCNC(C(CSC)C)=O)C 23095,C1(C(C)C(=O)NCc2cccc(Cl)c2)CCN(C(C2CCC(=O)C2)=O)CC1 23096,C#CC1(O)CC(C(=O)N(C2CCN(C(=O)CCc3ccc(C)s3)CC2)CCO)C1 23097,CCC(CCOC)C(=O)NC12CCC(C1)N(C(c1sccc1-n1ccnn1)=O)C2 23098,CC1CN(C(C2CC3C=CC2C3)=O)CC1NC(c1cnn(C)c1N)=O 23099,N1(c2ccc(S(=O)(=O)NC3CCOC4(CCC4)C3)cn2)CCOCC2(CCCC2)C1 23100,N1(C(c2ncc(C)c(C)c2)=O)CC(NC(=O)CC2CCCCN2C)C2(CCC2)C1 23101,N1(C(c2cn(C(C)(C)C)nn2)=O)CC2(NC(=O)C(c3ccc(F)cc3)F)CC1C2 23102,C1(N(C(c2c(C)ocn2)=O)C)CCCC(N(C)C(c2ccon2)=O)C1 23103,C1(C(c2ncc(C)o2)NCc2nnnn2C2CC2)CCCCCC1 23104,Cc1cccc(C(N2CCOCC2CCNC(=O)CC2CCC23CCC3)=O)c1F 23105,C1(NC(CC2C(CNC(c3ccc(CC)s3)=O)C2)=O)CC2(CCC2)C1OC 23106,Cc1onc(Cl)c1NC(=O)C(=O)NCc1nccn1C(C)(C)C 23107,C1(NC(COC(C)C)=O)C2CC1N(C(c1ccnc(CN(C)C)c1)=O)C2 23108,C1(NC(C=C(C)Cn2cncn2)=O)CN(C(=O)CN(C)S(N)(=O)=O)CC1C 23109,C1(n2cc(CNC)nn2)CCCN(C(=O)C(C)(C)c2ccc(Cl)s2)C1 23110,C1(C(N2C(C(CNC(C3C(C)OCCC3)=O)(C)C)CCC2)=O)CC2CC1C1CC21 23111,C1(CC)CN(C(c2sccc2Cl)=O)CCN1C(=O)Cc1ccc(Cl)nc1 23112,c1(C(N2CC(CNC(C(c3c(C)cncc3)C)=O)C2)=O)cc2c(s1)CCSC2 23113,c1(CC(N2CCCC(NC(C3C(C=C)C3)=O)CCC2)=O)ccc2c(c1)CCCO2 23114,c1(C(N(C(CNC(C2(C(=O)OC)CC2C)=O)C)C)=O)cc(C)c(C)[nH]1 23115,c1(C(=O)NCCCCCN(C(CC2CCC(C)O2)=O)C)ccc(Cl)c(F)c1N 23116,C1(CC)C(NC(=O)C=C2CCC(C)C2)CCN1C(c1oc(C(F)(F)F)nc1C)=O 23117,C1(CCC)(NC(=O)CCOCC2CCCO2)CCN(C(=O)C(C)=C2CCC2)CC1 23118,c1(NC(c2nnnn2C2CCOC2)C2CC(OC)C2)ccc2nn(CO)cc2c1 23119,Cc1cc(C(=O)O)cc(C(=O)NCCNC(c2c(C)cccc2Cl)=O)c1 23120,C(C(=O)N1CCC(CO)(NC(=O)Cn2nnc(C3CC3)n2)C1)(C(C)C)OCC 23121,C(C(C)(CCO)Nc1cn(CC2(CC(C)C)CNC(=O)C2)nn1)OC 23122,CC(C)CCC(O)C(=O)NC1CCN(C(=O)CC2(O)CCCCC2)CC1F 23123,N1(C(C2N(CC)CC2)=O)CC=C(C(C)(C)C(=O)NCCCOCC(F)F)C1 23124,c1(C(N2CC(C)(CNC(C(C3CC3)OC)=O)C2)=O)cc2c(cc1Br)OCCO2 23125,c1(CNC2C(C(=O)Nc3ncc(C)nc3)C2)cc(I)ccc1O 23126,c1(C(C)C(N2CCCC(F)CC2)=O)ccc(S(=O)(=O)N2CCCC2)cc1 23127,C(=O)(C1CSc2ccccc21)NCCC1CC(NC(c2c(CC)nn(C)c2)=O)C1 23128,N1(C(C(c2cnn(C)c2)C)=O)CCOC(C(=O)NC2COCC2CN(C)C)C1 23129,C(=O)(C(F)(F)CC(C)C)NC1CC2(C(NC(c3c(C)n(C)nn3)=O)C2)C1 23130,C1(C2CC2)(NC(c2c(C)cc(CC)o2)=O)CCN(C(C2CCCNS2(=O)=O)=O)C1 23131,CC1(NC(C2CCC(n3cc(-c4cncnc4)nn3)CC2)=O)CCCC1O 23132,c1(C(N2CCN(C(C=Cc3c(C)cncc3)=O)CC2)=O)c(Cl)cccc1[N+](=O)[O-] 23133,c1(N2CC(C(C)C)C(O)CC2)nc(=NCC(C(C)C)N(C)C)[nH]c2c1COCC2 23134,C1(CNC(c2ncncc2Cl)=O)CCCCN1C(=O)Cc1cccc(Br)c1 23135,c1(NC)cnncc1C(N1CCC(C(=O)NCC(C)C#N)(C(C)C)C1)=O 23136,c1(N(CCOCCN(C(c2ccc(SC)cc2)=O)C)C)cc(Cl)nc(SC)n1 23137,C1(NC(c2cc(OCC)ncc2)=O)CN(C(=O)C(O)CC(N)=O)CC1(C)C 23138,N1(C(c2cncs2)=O)CC2CCC1C1CN(C(C3(CO)CCC3)=O)CC21 23139,c1(C(=O)NCC2CCCN(C(C3(O)C(C)(C)C3)=O)CC2)nc2ccccn2c1F 23140,c1(C(N(CC(CNC(C2C(C)OCCC2)=O)(C)C)C)=O)nccc2cccnc12 23141,C(CNC(=O)C=Cc1ncc[nH]1)(CCCC)NC(C1(CC#C)CCCO1)=O 23142,C1(NC(C2(CC=C)COC2)=O)CCN(C(=O)C(F)(F)c2ccccn2)CC1 23143,CC1=C(C(=O)N2CCN(C(C3(C4CCCO4)CC3)=O)C(C(C)C)C2)CCS1(=O)=O 23144,C#CCC(C)(CC)C(=O)N(C)CCNC(=O)CCC1CCCN1C 23145,CCCC(CC(C)C)C(=O)N1CCC(C(=O)NCc2nocc2CC)CC1 23146,N1(C(c2ccc(C(=O)OC)o2)=O)CC(NC(=O)Cc2csc(C)n2)C(F)C1 23147,CC1=C(C)C(OC(c2cnc(C3CC3)nc2)=O)CCC1 23148,c1(N2C(c3nc(C)[nH]n3)CCC2)nccc(N(CC(C)CO)C)n1 23149,C12(C(N3CCC(N(C(c4c(C)cc(SC)o4)=O)C)C3)=O)CCC(CC1)C2(C)C 23150,C1(C2CCCO2)(C(N(C(C)CNC(=O)C(C)(C)O)C)=O)CCCCC1 23151,c1(CNC(C(CSC)n2cc(CNC(C3CCC3)=O)nn2)=O)c(C)[nH]c(C)c1C 23152,c1(COC)ccc(C(N2CCCC(CCNC(c3ccc(Cl)nn3)=O)C2)=O)cc1 23153,C(=O)(C1=CC2(CCN(C(=O)CC3(CSC)CC3)C2)C1)N(CC(CC)C)CC 23154,N1(C(C2=CC(C)C2)=O)CCN(C(c2coc3ccccc23)=O)CC(O)C1 23155,c1(OCC)c(-n2cc(NC(C)=O)nn2)cccc1F.C1(C)CCC(=O)N1CC 23156,Cc1ccc([N+](=O)[O-])c(NC(C2CCCN(Cc3ccc(Br)o3)CC2)=O)n1 23157,C1(C(=O)NCCS(CC)(=O)=O)CN(C(=O)CCC2CCCO2)C2(CCC2)C1 23158,C1(C)(CNC(c2c(C)nncc2)=O)CCCN(C(=O)C(C)C2CCC2)C1 23159,C1(CNC(c2c(Cl)nc(OC)s2)=O)CCCCN(C(=O)C(C#N)C2CC2)CC1 23160,C1(CCC(=O)N(CCCNC(=O)CCOc2ccccc2)C)CCCC(=O)N1 23161,CCC(C)C(C(=O)NC(C)CNC(c1cccc(NC(N)=O)c1)=O)NC(=O)OC 23162,C1C(F)(F)CCC(=O)N(C)CC(O)Cc2cn1nn2.C1(C)CC1.CO 23163,c1(C(N(CCNC(COC2(C#C)COC2)=O)C)=O)cc2c(s1)CC(C)CC2C 23164,C(=O)(CCC#Cc1ccccc1)NC1CC(N(C)C(c2ccn(C3CC3)n2)=O)C1 23165,C1(CNC(CC2CC(C)(C)C2)=O)CCCCN(C(=O)CC2CCCO2)CC1 23166,C1(C(=O)NCC(C)CNC(c2sc(C(C)C)nc2C)=O)(COC)CC=CCC1 23167,CC1Oc2c(C(=O)NC3(CCNC(c4cccs4)=O)CC3)cccc2NC1=O 23168,N1(C(c2sc(CC)c(C)c2)=O)CC2CCC(NC(c3cnsn3)=O)(C2)C1 23169,Cc1c(C(N2CC(NC(=O)C(C)(F)F)CCC2C)=O)cnc2ncnn12 23170,CCCCCC=CCC(=O)NC(C)CC(C)NC(=O)CSC(F)F 23171,N1(c2c(C)nccn2)CCC(O)C(C(=O)NCC2CCCC(=O)N2C)C1 23172,C#Cc1ccc(NC(=O)C(CCC)NC(=O)C(CC)=CC)cn1 23173,N1(C(=O)NC(c2ccc3c(c2)OCCO3)C(F)(F)F)CC(=O)NCCNC(=O)C1 23174,C(=O)(C(O)CC1CCCC1)N1CC(CC(C)NC(=O)C(C2CCCCC2)O)C1 23175,N1(C(CSc2nc(C)sc2)=O)CC2(CCN2C(=O)CCCCNC(N)=O)C1 23176,CCCCC(O)CCC(=O)NC(CNC(c1ccc2nc(S)[nH]c2c1)=O)C(C)C 23177,C1(C(=O)NC2(C)CN(C(C3CCCN(C(C)=O)C3)=O)C2)CC2CC1CC2(F)F 23178,N(C1CCc2c(Br)cccc21)C(C1CC1C(=O)Nc1cccc2nc(O)oc12)=O 23179,C1(C(N2CCC(C(=O)Nc3ccc(CC)c(Br)c3)CC2)=O)Cc2ccccc2C1 23180,c1(CNC(Cn2ncc(CC)c2)=O)cccc(C(=O)NCc2[nH]nnc2C)c1 23181,C1(C(N(CCCN2CCNCC2)C)=O)CC2(CCO1)CC(F)(F)C2 23182,c1(-c2nnc(COC(C3CC3c3ccncc3)=O)o2)ccc(F)cc1 23183,c1(OCCC(=O)NCC2CCCN2C(c2nn[nH]c2Cl)=O)ccccc1F 23184,CC1CCCC(C(=O)NC2(C)CC(C(=O)NCC3CC3C3CCC3)C2)C1 23185,N1(C(=O)NCCc2ccon2)CCC2(CC1)CC2c1cccnc1 23186,Cc1ncnc(C(=O)N(CC(C)N(C(=O)CN2CCN(C(C)C)CC2)C)C)c1C 23187,C1(NC(c2cnn(CC)n2)=O)CCC2(CC1)CC2NC(=O)CCc1cccs1 23188,c1(CC(=O)NC(C)C(CO)NC(c2nn(C)cc2N)=O)cnc2cccnn12 23189,S(=O)(=O)(c1c(C)sc(C)c1C)NCC(CCCC)NC(=O)NC(C)(C)C 23190,C1(COC(C2N(C(=O)OC(C)(C)C)CCCCCC2)=O)CCCCN1S(N)(=O)=O 23191,N1(CC)CCC(NC(=O)C(CC2CCC2)NC(=O)CSc2cn[nH]c2)C(C)C1 23192,O=C1CCc2cc(-c3ccnc(C(=O)NCCc4ccc(O)cc4)c3)ccc2N1 23193,O=C(C1=CCCCCC1)NCC12CCC1CN(C(c1nncs1)=O)C2 23194,CC(CC(=O)NCC1(F)CCN(C(c2cnc(Cl)cc2N)=O)C1)C(C)(C)C 23195,C1(NC(CCc2c(C)cccc2)=O)CC(O)CN(C(c2cc(CO)oc2C)=O)C1 23196,c1(C(=O)OC)cnn2c1CC(Nc1nn3cc(CC(C)C)nc3s1)CC2 23197,C(=O)(C(CC(C)C)C(C)C)NC(C(=O)NC1CC(COC)C1)c1cccs1 23198,Cc1ccccc1C1(C(=O)NC2CC(NC(C3(C)CC3C(=O)O)=O)C2)CCCC1 23199,c1(NC2(NC(CC3C(CNC(CSC)=O)C3)=O)CCC2)c(Cl)nsc1Cl 23200,C12(NC(c3ccc(CC)c(C)c3)=O)CCCC1N(C(c1cncn1C)=O)CC2 23201,c1(C(N2CCN(C(C3C(C)(C)NC(=O)C3)=O)C(CO)C2)=O)cnn2ncccc12 23202,C(=O)(C1Cc2ccc(F)cc21)N1CC2(CN(C(CS(CC(=O)OC)(=O)=O)=O)C2)C1 23203,N1(C(C(=O)NCCCC2CC2)C2C(C)C2)C=CCCCC1 23204,Cc1cc(CNC(=O)NC2(n3cnnn3)CCCCC2)cnc1Br 23205,C12(NC(Cc3c(C)ocn3)=O)CCCN(C(c3ccc(Cl)c(F)c3F)=O)CC1C2 23206,C(=O)(C1=NOC(C(C)(C)C)C1)N1CCCC(N(C(C2C3CCC(F)C23)=O)CC)C1 23207,N1(C(C(COCC)n2cc(C3CCCC4CC34)nn2)=O)CCN(C)C(C(F)F)C1 23208,c1(C(=O)NCC2N(C(C(C)Cc3cnn(C)c3)=O)CC2)c(Br)nnn1C 23209,C1(C(N(CC(C)(O)C2CC2)C)=O)C=CCCN1C(c1sccc1F)=O 23210,C(F)(c1ccccc1)=CC(=O)NC(CNC(C(COC)OC)=O)CC(C)C 23211,Cc1ncncc1C(N1CC(NC(C2CCCCC2)=O)C(C)C1)=O 23212,C1(NC(N(CCN2CCN(C(C(=O)NC)C)CC2)C)=O)CC2CCC1CC2 23213,c1(CCNC(CN2CCCC(CNC(CC)=O)C2)=O)ccc2cnccc2c1 23214,C1(C(=O)NC(CC#C)CC)CC(=O)N(C)C1c1ccc(F)cc1 23215,Cc1ccc2c(c1)C(NC(C1CC1c1cccc(Br)c1)=O)CCCN2CC(C)O 23216,N1CC=C(c2cccc3ccccc23)CC1.c1(C(=O)O)cccc2c([N+](=O)[O-])c[nH]c12 23217,C(CN=c1cc(C)nc(Cc2ccccc2F)[nH]1)NC(CN(CCC)C1CC1)=O 23218,c1(CC(=O)NC(Cn2cc(C3(C)CCCO3)nn2)CC2CC2)c(F)cccc1Br 23219,N1(C(CC(C)C)=O)C(CNC(c2cnccc2CN2CCOCC2)=O)CC2CC12 23220,CC(C)C(C(=O)N1CCN(C)CC1)C(C)NC(c1ccc(O)nc1)=O 23221,C(=O)(C(F)CC(C)(C)NC(=O)CC1CC2CCC1C2)NC(c1ccc(C)cc1)C 23222,c1(NC)ccc([N+](=O)[O-])cc1C(N1CCC2(CCCN2C(=O)C=CCF)C1)=O 23223,C(C1COCc2ccccc21)c1nnc(N2C(C)(C)SCC2)n1CC#N 23224,C1(NC(N2CC(C(=O)NCC(C=C)O)C2)=O)CC(=O)N(c2ccccc2)C1 23225,CC1ON=C(C(=O)N2CC(NC(=O)Cc3c(Cl)cnn3C)C(C3CC3)C2)C1C 23226,C#Cc1cccc(NC(=O)C(=O)NC2(c3ccc(Br)s3)CCC2)c1 23227,N1(CC(CC)OC)CC(C)N(c2ccccc2)CC1C 23228,C1(NC(C)=O)CCC(C(N2CCC(NC(c3cn(C(C)C)cc3C)=O)C2C)=O)CC1 23229,N1(C(c2c(C)n[nH]c2)=O)CC2CC1(CNC(=O)C(C)(O)Cc1ccccc1)C2 23230,c1(CC)nnc(=NCC2CCCC2NC(c2sc(C)nc2C)=O)[nH]c1CC 23231,N1(C(C=CC=CC)=O)CCc2ccccc2C1CNC(=O)CCc1scnc1C 23232,N1(C(c2ccc(CC)c(F)c2)=O)CC2CCCC2(NC(c2cc(Cl)c(Cl)[nH]2)=O)C1 23233,c1(CCC)ccccc1C(=O)CNC(=O)C(C)Oc1ccc(F)nc1 23234,c1(NC(C(CC)(C)CNC(=O)C(C)CN(C)C)=O)cnc2ccnn2c1 23235,C(=O)(C1=CC2CCCC12)NCC1C2N(C(c3cccc(CC)c3N)=O)C(CC2)C1 23236,N1(C(c2c(C)cc(F)s2)=O)CCCC2(CCCN2C(c2cncs2)=O)C1 23237,N1(C(C2(CNC(C(C)=NOCC#N)=O)CCCO2)=O)CC[Si](C)(C)CC1 23238,c1(CN(CCOC)Cc2ccccc2C)c(-c2cncc(Cl)c2)ncn1C 23239,Cc1cccc(C)c1CC(N1CCCC(NC(C2(O)CCC2)=O)C1)=O 23240,CC1=C(C(=O)NCC2CCCN(C(=O)CCCc3nccs3)C2)CCC(C)(C)C1 23241,c1(C(N2C(CNC(c3noc(CC)c3C)=O)C=CC2)=O)ccc(P(C)(C)=O)cn1 23242,C1(CNC(C2C=CCC2)=O)CCN(C(=O)Cc2ncc(F)cc2F)CC1(F)F 23243,S(=O)(=O)(c1cccnc1N1CCC(CN2CCC(C)C2)CC1)N(CCCCC)C 23244,N1(C(C2(c3c(C)cccc3)CC2)=O)CC2CC(NC(=O)C(C)SC(C)C)C1C2 23245,c1(CNCC2(C(=O)NC3C(NC(CCOCCCC)=O)C3)CC2)cc(C)no1 23246,Cn1nc(CN2CCC(Nc3ncccc3C(F)(F)F)C2)c2c1CCCC2 23247,c1(N2CCC(NC(c3nc(Cl)ccc3F)=O)(CF)C2)ncc([N+](=O)[O-])cc1Br 23248,C(=O)(C1=CS(=O)CCC1)N1C(CC(=O)NC)CN(C(=O)C(C)(C)C(F)F)CC1 23249,N1(C(COCCSC)=O)CCC2(NC(C3CCN(C)C(=O)C3)=O)CCCCCC12 23250,C1(C(N(CC(CC)NC(=O)CC2COC(=O)C2)C)=O)CC2(CCC(F)(F)CC2)C1 23251,N1(C(CC(CCC)NC(c2oc(C)nc2CC)=O)=O)CCC2(CCCCC2)C1 23252,CCC(CC(F)(F)F)C(=O)N1CC2(CNC(C3CCC(C)CC3)=O)CC1CO2 23253,c1(C(=O)NCCN(CCC)C(C2CCCC23CC3)=O)ccc(C(F)(F)F)cn1 23254,c1(C(=O)NCC(CN(C(c2ccsc2Cl)=O)CC)(C)C)cc2sc(C)cc2[nH]1 23255,N1(C(CCCC(=O)N(C)C)=O)CC2CCC1CN2C(c1ncccc1Cl)=O 23256,CC1(C)CCC(CNC(C2(C)CCCS2(=O)=O)=O)N(CC(N2CCOCC2)=O)C1 23257,N1(C(c2nc(C(C)C)oc2)=O)CCn2nc(C(=O)N(c3ccccn3)C)cc2C1 23258,c1(C(=O)NCC2CC2C(=O)Nc2cncc(Cl)c2)ccnc(O)c1 23259,O=C(C1CCCn2c(Br)cnc21)NC12CC(C1)N(C(C1CC1F)=O)C2 23260,C1(NC(C2(COC)CN(C(c3cn(CC=C)nn3)=O)C2)=O)CCc2ncnn2C1 23261,C(C(=O)N=S(C)(=O)c1cnn(CC(F)(F)F)c1)c1onc(N(C)C)n1 23262,C#CCCCC(=O)NC1CCOC(C2CCN(C(=O)Cn3ccsc3=N)CC2)C1 23263,CCS(=O)(=O)CC(=O)N1CCC(N(CCO)N(N(C)C)C)C1.c1(C=O)ccncc1 23264,N1(Cc2cc(C)ncc2)CC2CN(C(c3cccc(C)c3I)=O)CC12 23265,c1(C(=O)NC2C(NC(C3(C)CC4CC4C3)=O)CCOC2)cc2nn[nH]c2cc1F 23266,Cc1nnc2n1CC(C(=O)NC1CC1NC(=O)CCc1cc(Cl)no1)C2 23267,c1(CC(=O)OCCCC2N(C(=O)OC(C)(C)C)CCC2)ccc(F)cc1 23268,C1(CN(C(=O)C=CI)C)COCCN1C(=O)Cn1cnnc1O 23269,N1(C(C2(C#C)CC2)=O)CCC(C(=O)Nc2cnccc2C)C(C)(C)C1 23270,C(=O)(C(O)CC(N)=O)NCCCOCCC(N1CCC(=CC#C)CC1)=O 23271,C(=O)(CCC(C)NC(C1CC2(CC2)CO1)=O)NCC(CSC)(C)C 23272,Cc1cc(C(=O)NCC2CCC2NC(C2(Cl)CC2)=O)sc1Br 23273,c1(N2CC(O)(CNC(c3nn(C(CC)CC)c(C)c3)=O)C2)cc(O)nc(=O)n1C 23274,N1(C(CCc2ccc(C)o2)=O)CC(NC(c2onc(C)c2C)=O)CC(F)C1 23275,C1(CC)(CO)CCCN(C(C2(C)CCCN2C(c2coc(C(C)C)n2)=O)=O)C1 23276,CC(C)CCC(C(=O)NCCCc1ncn(C)n1)NC(C1CC1(F)Cl)=O 23277,N1(C(CC(CC(C)C)C)=O)CCN(C(C2CC3CCC2C3)=O)CC2(C)CCCC12 23278,C1(NC(c2cccc(C(=O)NC)n2)=O)CN(C(=O)Cc2nocc2C)CC1(C)C 23279,C1(Nc2cc(CC(C)C)ncn2)CCN(C(=O)CC2(C)CC2(F)Cl)CC1C 23280,CC1CCN2N=C(C(=O)NC(C3CN(C(c4ccnn4C(F)F)=O)C3)C)NC2=N1 23281,N1(C(=O)OC(C)(C)C)CC(CNCC2CC(C)(C)CO2)C(F)C1 23282,c1(C(C(=O)NCC=C)N(c2cc(Br)ccc2OC)C)cn2c(Br)cnc2s1 23283,N1(C(C(CC)N(C)C)=O)CCCC(C)(CNC(=O)CCc2cnco2)C1 23284,N(C1CCCc2ccc(F)cc21)C(C(CC)OC1CCCCC1)=O 23285,c1(NCc2[nH]nc(CSC)n2)nccc(=NCc2ccnc(C#N)c2)[nH]1 23286,CC1OC2(C(=O)OCC3CC(C#N)(Oc4ccccc4)C3)CCC1CC2 23287,N1(C(c2cc(C)c(F)cn2)=O)CC2CCCC2(C(=O)NCC2(F)CCOCC2)C1 23288,N#CC1CN(C(=O)C=Cc2ccc(O)cc2Cl)CCN1C(=O)C=Cc1ccoc1 23289,C1(CC)CN(C(C2CCCC2F)=O)CC1C(=O)NC1CCCC1CN(C)C 23290,C1(C(=O)NCCN(C(CC(CC=C)(C)C)=O)CCC)CC12CCC1(CC1)CC2 23291,N1(c2nccc(C(=O)Nc3ccccc3)c2)CC(C(=O)O)OCC12CCOC2 23292,C(=O)(C1=CS(=O)(=O)CCC1)NC1C2(CN(C(c3cn(CC=C)nn3)=O)C2)CCC1 23293,C1(c2ccccc2)(C(N(C)CCNC(=O)COC2CCOCC2)=O)C=CCCC1 23294,C1(NC(C(C)CCO)=O)COC2(C1)CN(C(=O)Cn1nc3c(n1)CCCC3)C2 23295,CC1(C)NC(=O)CC1C(=O)NCC1CC(NC(=O)CC2CC3CCC2CC3)C1 23296,c1(OC)ccc(C(N2CC(CO)(NC(=O)Cc3sc(S)nc3C)C2)=O)c(OC)n1 23297,C1(F)(C(N(CC(C)N(C(C(c2cc(F)cc(F)c2)C)=O)C)C)=O)CCN(C)CC1 23298,N1(C(CCOCC)=O)CC2CC1C2NC(c1nn(CC)cc1Br)=O 23299,N1(Cc2cn(CCCNC(c3conc3C(F)(F)F)=O)nn2)C(=O)CNC1=O 23300,Cc1nccc(C(=O)NCCC2(C(=O)NC3CC3C)CC2)c1N 23301,C#CC1(C(=O)N(CCCCN(C(=O)C(F)(F)c2nc(C)cs2)C)C)CCCC1 23302,C(=O)(C(F)C(=O)N1CC(F)CC1C(=O)NC(CC)C1CC1)OCC 23303,CC1CN(C(=O)C=Cc2ccco2)CC2(CCN(C(C3CCC(C)(C)O3)=O)C2)O1 23304,O=C(C#CC1CC1)NC1CC2(C1)CC2NC(C1CCCCS1)=O 23305,O=C(N=c1[nH]nc2n1CCCC2)N1CCC(Cc2cccnc2)C1 23306,CCCS(=O)(=O)CC(=O)N1CCN(CC2CCN(C(=O)CSC(F)F)CC2)CC1 23307,Cc1cc(=NCc2cc(NC(=O)C(C)C)on2)[nH]c(N2CCc3ncncc3C2)n1 23308,c1(C(=O)NCCc2ccc(C(N(C)C)=O)cc2)c(F)ccc2n[nH]cc12 23309,N1(C(C(CC)NC(C)=O)=O)CCC(C2CCCN(C(=O)C(C)C(C)(C)C)C2)CC1 23310,N1(C(CC(CCC)C)=O)CC2CCC(N(C)C(c3ncc(F)cc3C)=O)C2C1 23311,N=C1NC(=O)C(CC(=O)NCC2(CNC(=O)C(O)Cc3cnc[nH]3)CC2(F)F)S1 23312,C1(CNC(c2c(CC)ncs2)=O)C(O)C(O)CN1C(=O)CN1CCCC1=O 23313,CC12CC(C(=O)NC3CC(O)CN(C(c4cnc(C(F)F)s4)=O)C3)(C1)C(C)(C)O2 23314,C(=O)(C#CC1CCOCC1)NC(C1CCCN1C(c1cc(C(F)(F)F)n[nH]1)=O)C 23315,C1(C)(C(=O)NCCN(C(CC=CC=C)=O)Cc2ccccc2)CC(OC)CN1C 23316,c1(CC(N2CC(NC(C3CC(C)(C)OC3)=O)C3(C2)CC3)=O)ncn2c1COCC2 23317,C1(CNC(CCC=C(C)C)=O)CC2(CC2)CN1C(C1CC(C2CC2)=NO1)=O 23318,c1(C(N(CC(C)NC(C(CSC)C)=O)C)=O)cc2ccc(Cl)cc2c(O)n1 23319,N1(C(C(c2ccc(C)cn2)(F)F)=O)CCCC(NC(c2cccs2)=O)C1C 23320,C1(CNC(c2c(C)[nH]cc2)=O)CN2CCCCC2CN1C(c1ccn(C)n1)=O 23321,c1(C(N2C(C)CC(CNC(COc3cccc(C)c3)=O)C2)=O)cc(O)nc(Cl)c1 23322,c1(C(=O)NC2CCN(C(C(CC)NC(C)=O)=O)CC2F)cc2n(n1)CCNC2=O 23323,N1(C(C(=O)NCCCC)C2CCC2C(F)(F)F)CCCC(C2CCC2)C1 23324,c1(C(=O)NC2CC(F)(CNC(C3C(C)C3)=O)C2)cccc(C(F)(F)F)c1 23325,CC1=NNC(=O)C1CC(=O)NCC1(CN(C)C(c2ccn(CC(C)C)n2)=O)CC1 23326,CCCC(CNC(=O)CC1CCN(C(=O)CC2(COC)CC2)C1(C)C)CCO 23327,C(=O)(CS(=O)(=O)CC(C)C)NC1(CCNC(c2ccnc(C)n2)=O)CC1 23328,C(CCCCCCCO)=CCO.C1(C(C)N(C(=O)C2CC2)C)CN(C(=O)O)C1 23329,C1(CCOC)CN(C(=O)CC2(NC(C)=O)CC2)CCN1C(C1CS(=O)C1)=O 23330,CC1CCCN1CCCn1cc(C2CC=CCC2)nn1 23331,C=CC1(CC(N2CCC2C(=O)OC)=O)CN(C(=O)C(CN(C)C)CC)C1 23332,N(C(=NCCc1csc(C)n1)NC1CC(c2ccccc2C)C1)C(C=C)C 23333,n1(CC)cc2ccc(C(=O)N(C)CCNC(=O)CNC(C3CC3C)=O)cc2n1 23334,c1(N2CC(C(C)NC(C3(C)CCC(=O)N3)=O)C2)nc(Cl)nc2[nH]c(O)nc12 23335,C1(NC(=O)Cn2cccc2)CC2CC1CC2C(N1CC2(C1)CN(C1CC1)C2)=O 23336,c1(C(N2CC(c3ccc(C)cc3)OC(C)C2)C2CCC2)c(O)ncc2c1CCC2 23337,N1(C(c2cc(CC)ncc2)=O)CC2ON=C(CNC(=O)C=CBr)C2C1 23338,c1(CCC)nccn1CC(=O)NCC(C1CC1)NC(C1(C(C)(F)F)CC1)=O 23339,Cc1nscc1CC(=O)N(C1CCC(NC(=O)COC(C)C)C1)C 23340,c1(N2C(C)C(NC(=O)CC3(CO)CC3)CCC2)ncc2ccnc-2[nH]1 23341,N1(C(C(N2CCN(C)CC2)C)=O)CC2CN(C(C3(Br)CC3)=O)CC(C1)O2 23342,c1(SCC)cccc(C(=O)NC2(C)CCN(C(c3nnc(S)n3C)=O)C2)c1 23343,CC(C(O)C(F)F)NC(=O)C(c1ccco1)NC(=O)CC1(C)CCOC1 23344,C(C1=CCCSC1)(c1nnnn1C1CCOCC1)NCCCCC(C(C)C)O 23345,C1(c2nnnn2-c2ccc(Cl)cc2F)(NCc2c(C)noc2)CCOC(C(C)C)C1 23346,N1(C(C(C)COCCOC)=O)CCC(C)(C)C1NC(=O)Cc1ccc(C)c(Cl)c1 23347,N1(C(C2(COC)CC2(F)F)=O)CC2CCCC(NC(=O)C=CCO)(C2)C1 23348,N1(C(C(CC=C)C(C)C)=O)CC2(CCN(C(c3cc(C)c[nH]3)=O)CC2)CC1C 23349,N1(C(C2C(OCC)C2)=O)CC2CCN(C(=O)CCc3cc(C)nn3C)CC2C1 23350,c1(NC(CN(C)Cc2coc(Br)n2)=O)cccc2c1OCC2 23351,C(CC(C)(C)CC(=O)NC(CC(C)C)C(=O)Nc1ccc(O)c(Cl)c1)OC 23352,C1(NC(=O)C2=NOCC2)CCCOC12CCN(C(=O)Cc1ccc(O)cn1)CC2 23353,CC1(C)CC(C(=O)NCC(CC(=O)N(CC2CC2)CC2CC2)C2CCC2)CCO1 23354,c1(OCCOC)ccc(Cl)cc1C(=O)NCC1CN(C(=O)C(C)CF)CCO1 23355,CC(C)C(C)CC(=O)N1CC(C)CCC1C(=O)Nc1cc(Cl)cnc1O 23356,c1(OC)nccc(Br)c1C(=O)N(C)CCNC(C1CCSC(C)C1)=O 23357,N1(C(c2nc(C)oc2)=O)Cc2[nH][nH]c(=NC(=O)c3cc(Br)ccc3Cl)c2C1 23358,c1(C(N2CCC(OCCNC(CCC#CC)=O)C2)=O)cc(C)c(O)c(C)c1 23359,c1(OC)[nH]c(=N)nc2sc(C(=O)NCCCNC(C34CCC3CC4)=O)cc12 23360,CCCCC(CNC(=O)CCSc1ccccc1)NC(=O)CCC1CCCN1C 23361,C(=O)(C1=NNC(=O)CC1)NC1CN(C(C2C(C)(C)OCC2)=O)CC(O)C1 23362,C1(O)(C(C)NC(=O)Cn2cccc2)CCN(C(=O)Cc2ccc(Br)cc2)CC1 23363,C1(C(=O)NC(C)CCNC(=O)C(C(C)O)N(C)C)(COC)CCCCO1 23364,CC1=C(C(=O)N2CCCC(NC(c3cc(F)ccc3Cl)=O)C2C)CCC1 23365,c1(NC)cccc(C(=O)NC(C)C(c2ccccc2)NC(=O)C(C)SC)n1 23366,c1(OCC#C)ncccc1C(=O)NCC1CC(NC(c2cnn(CC=C)c2)=O)C1 23367,S(=O)(=O)(c1cccc2c(Cl)ccnc12)NCCN1CCC(NC)CC1 23368,C(C(CNC(c1ccn(C(F)F)n1)=O)C(F)(F)F)NC(c1cn(C(C)C)nn1)=O 23369,c1(C(=O)NC23C(CN(C(c4n[nH]c(CC)c4Cl)=O)C2)CC3)cc(F)cc(F)c1O 23370,CC1(NC(=O)C(C2CCOCC2)O)CCCN(C(=O)CSCc2ccccc2)C1 23371,c1(C(=O)NCC2(O)CN(C(C(C)NC(CC)(C)C)=O)C2)cc(Br)cn1C 23372,CC1(C)CC(NC(c2ccco2)=O)CN(C(C2CC2(F)F)=O)C1 23373,c1(CCC(=O)N(C2CN(C(CN(C)Cc3ccccc3)=O)C2)C)cnc(O)[nH]1 23374,c1(OC)cccc(C(=O)NCC2(NC(C3C=C3C)=O)CCOCC2)c1[N+](=O)[O-] 23375,C=C1CC2(C1)CC(C(=O)NCC(C)CNC(=O)C(O)C(C)CC)C2 23376,C(=O)(CC(C1CC(F)(F)C1)NC(c1ncoc1C(F)F)=O)OCC 23377,c1(C(=O)OCCC(=O)Nc2ccc(OCC)cc2C)cnc2ccccn12 23378,N1(C(C(C(C)C)CNC(C2(C)CCC3CC3C2)=O)=O)CCCOC(C)(C)C1 23379,C1(CC)CCC(C)CN1C(c1c[nH]nc1CNC(c1cnc(Cl)s1)=O)=O 23380,C1(N(C(=O)CCc2cn[nH]c2)C)CCCN(C(=O)C(C)(C)c2ccccn2)CC1 23381,C1(O)(CC)CCC(NC(=O)CC(C)(C)CNC(C2CCCOC2)=O)CC1 23382,N1(C(C2CCCN(CCC)C2)=O)CCC(NC(=O)CN2CCCCCC2)C(F)C1 23383,CC1CCN(C(=O)Cn2cnnc2)C1CNC(C1(C)CC1Br)=O 23384,c1(C(=O)OC)cc(CC(=O)NC(C)CNC(c2[nH]ccc2C2CC2)=O)cs1 23385,c1(C(=O)OC)cncc(C(=O)NC2COCC2Cc2ccccc2)c1 23386,C1(C(=O)NCC(C)(C)OCCNC(=O)Cc2ccc(Cl)cc2)CCC2CC2CC1 23387,N1(C(C(C)NC(COC)=O)=O)CC2CC1C2CNC(C1(C)CC1(F)F)=O 23388,c1(-c2nc(Cc3ccc(C)nc3)n(C3CCS(=O)(=O)C3)n2)ccc2nc[nH]c2c1 23389,c1(C(N2CCN(C(C(n3ccc(C)n3)C)=O)CC2CF)=O)ccc(O)c(C)c1C 23390,C1(NC(=O)Cn2cccn2)CN(C(c2ccnc(Cl)c2F)=O)CC1(F)F 23391,n1(CCCNC(COCCCOC)=O)cc(C(=O)NCC2CCOC2)nn1 23392,C1(OC)(CO)CCN(C(c2cn(CCNC(=O)C3=CCCC3)nn2)=O)C1 23393,CC1(C)CN(C(c2cnc(C(F)F)nc2)=O)CC1NC(C1(CCF)CCC1)=O 23394,C1(CC2(O)CCN(C3CC(=O)N(CC)C3=O)CC2)COC2(CCCC2)O1 23395,C1(C(N(CCCC)CC)=O)CN(C(C2CCCOC2)=O)C(C)(C)C1 23396,C12(OC)CCC(C(N3CC(CNC(=O)CN(C)S(N)(=O)=O)C(O)C3)=O)(CC1)CC2 23397,c1(C(=O)NC2CC3CC(NC(C(C(C)(C)O)F)=O)C2C3)ccn2cccc2c1 23398,C(=O)(C(O)(C(C)C)C(F)(F)F)N1CCCCC(NC(c2c(C)scc2)=O)C1 23399,N1(C(=O)NCCNc2ncco2)CCN(C(=O)CC2(C(F)(F)F)CC2)CC1 23400,c1(CNC(C2C(=C)CC2)=O)ccc(CNC(=O)CC2CCCC23CC3)c(F)c1 23401,C(=O)(C(CC(F)F)NC(=O)Nc1cc(C)cnn1)OCC 23402,N1(C(C(C)C)=O)CCN(C2CCC(NC(=O)C(N3CCC(C)(O)C3)=O)C2)CC1 23403,c1(C(=O)NCC(C)(CNC(C2CCNC2=O)=O)OC)cccc([N+](=O)[O-])c1 23404,N1(C(CCC2CC(C)C2)=O)CCC(NC(c2cn(C(C)C)nn2)=O)C12CCC2 23405,C1(NC(C2N(CCC(C)C)CCC2)=O)CN(C(=O)Cn2nccn2)CC1CO 23406,N1(C(C(C(C)O)C)=O)CCC(C2(NC(c3ccnc(O)c3)=O)CC2)C1 23407,C1(NC(C)(C)COC(c2ccco2)=O)CC2(C1)CC(C#N)C2 23408,C(=O)(CC(F)(F)C(F)F)N1CCC(NC(c2cc(COC)oc2C)=O)C(F)C1 23409,C(=O)(C(O)(C(C)C)C(F)(F)F)NCCOCCN(C(CCn1ccc(C)n1)=O)C 23410,C1(C(C)N(C(=O)C(O)C2CC2)C)CN(C(C2(C(=O)N(C)C)CC2)=O)C1 23411,CC1CC(NC(c2cccn2C)=O)CN1C(C1CC1C)=O 23412,C1(N(CC(=O)Oc2cccc(C)c2)C)CCC12CCN(C(=O)OC(C)(C)C)CC2 23413,c1(NC(C2CCCN2C(=O)CN2CCOC2=O)=O)cnc2ccccc2c1Cl 23414,Nc1cncc(C(=O)NCC2CCCCN2C(c2cc(C(F)(F)F)ccn2)=O)n1 23415,C1(C(=O)NCCC(C)N(C)C(c2ccc(CC#N)cc2)=O)CS(=O)(=O)CC12CC2 23416,Cc1c[nH]cc(C(=O)NCC(F)CNC(c2ccc(N)c(F)n2)=O)c1=O 23417,C1(NC(COCc2onc(C)n2)=O)CN(C(C2CCN2C2CCCC2)=O)CC1F 23418,Cc1cc(C(N2CCN(C(c3ccc(Br)c(O)n3)=O)C3CC23)=O)nc(C)c1 23419,Cc1cnc2n1CC(C(N1CCCOC(CNC(C3CCSCC3)=O)C1)=O)CC2 23420,N1(C(CSCC)=O)CCN(C(=O)Cc2cn3ccsc3n2)C(C(F)F)C1 23421,c1(C(=O)NC2CN(C(C(c3cccc(C)c3)(C)C)=O)C2)ccc(F)c2[nH]ccc12 23422,c1(C(=O)NC(C)CC(N)=O)cccnc1CNC(c1nn(C)cc1Cl)=O 23423,C=CCC(Cc1ccccc1)NC(=O)Nc1ncsc1-c1ccccc1 23424,C1(CCC(=O)NC(CNC(C2CC(OC)C2)=O)(C)C)CCCCO1 23425,c1(OC)cc(OC)nc(N2CC(C(=O)NCC(=O)N(C)C)CC(F)C2)n1 23426,N1(C(c2c(C)cc(O)cc2)=O)CCC2CC(NC(=O)C3=CC(C)(C)C3)CCC2C1 23427,N1(C(C2CC(OC)(OC)C2)=O)CCC(C)C(C(=O)N(CCCO)C2CC2)C1 23428,N1(Cc2cn(C)c(=O)cn2)CC(n2cc(-c3cccc(Cl)n3)nn2)CCC1(C)C 23429,CCCCC(C(=O)NC(C)CCCCNC(C)=O)N1CCCS1(=O)=O 23430,CC(F)(F)CCCC(=O)NCCCCNC(C1OCC1(C)C)=O 23431,C1(CN(C(=O)C(F)=C2CCC2)C)CCCN(C(=O)CCOCC2CC2)C1 23432,C(=O)(CCCCCc1ccc(O)cc1)NC1C(NC(C(C)CN(C)C)=O)COC1 23433,NC(=O)CCC(C(=O)NCc1ccc2occc2c1)n1cc(-c2cccs2)nn1 23434,CC1(C)CCC(C(=O)NC2(CNC(=O)CSc3ccccc3Cl)CC2)CO1 23435,CC(C)CCCC(=O)N1CCCCC1CCN(C)C(c1cc(CC(C)C)c[nH]1)=O 23436,CC(C)(F)CCC(=O)NCC(F)CNC(c1cccc(Cl)c1O)=O 23437,N#Cc1ccccc1C=CC(=O)NCC1(NC(c2n[nH]cc2F)=O)CCOC1 23438,Cc1cc(C#N)nc(N2CCC(N(C)C(c3ccn4ccnc4n3)=O)C2)n1 23439,C1(N(C(=O)C(C)NC(=O)C2CC2)CCC)CCN(C(=O)CCC(=O)OC)CC1 23440,CCC(CC(F)F)C(=O)NC(C)(C)CNC(=O)C(C(C)C)NS(=O)(=O)C1CC1 23441,C1(NC(C(C)=C2CC2)=O)CN(C(c2ccc([N+](=O)[O-])c(C)c2)=O)C2CCCCC12 23442,c1(C(=O)NC(c2ccc(C)cc2)CC(=O)OCC)cc(F)cc2c1CCC2 23443,Cc1ccc(Cl)c(C(N2CC3(CCC3)CC2CNC(C2(CF)CC2)=O)=O)c1N 23444,c1(OC)cnc(Cl)cc1C(=O)NC1(CO)CN(C(C2CCCC(=O)N2C)=O)C1 23445,N1(C(c2ncn(CC)n2)=O)CCOCC(C(=O)N(CC(C)SC)C)C1 23446,c1(NC(COc2ccc(CNC3C(CC)CCC3)cc2)=O)nc(O)sc1C 23447,C1(C(N(C2CCN(C(c3nccnc3Cl)=O)C2)CC)=O)CCC(C)(CC)O1 23448,c1(N2CC3N(C(C4(O)CC4)=O)C(CC3)CC2)nc2ccc(F)cc2s1 23449,C12CCCN(C1)NC2.n1(C(C)CN(c2cnns2)C)nnnc1C(C)(C)C 23450,CC(CC#N)C(=O)N1CC(n2cc(C(C)N(C)C)nn2)C1 23451,C(=O)(CC1=CCN(C)CC1)NCCC(C(N1C(C)CS(=O)(=O)CC1)=O)O 23452,N1(C(c2cn(CC3(C)CC3)nn2)(C)C)CCCN(C(C2CCCC2CF)=O)CC1 23453,C1(C(C)C)CN(C(c2cc(-c3ccc(-c4nsc(=N)[nH]4)cc3)[nH]n2)=O)CCO1 23454,c1(CN(C(C)C)C(=O)NCC2CC(O)C2)ccccc1.C1(C)CCCO1 23455,C#CC1CN(C(=O)CC2CCCCN2C(=O)CC2CCC(=O)C2)CCN1C 23456,Cc1nc2cncc(C(=O)NC3CCN(C(=O)C(C)(F)C(C)(C)F)CC3)c2[nH]1 23457,C=CC(C)(C)C(=O)Nc1cccc(CNC(c2ccnn2-c2ccncc2)=O)c1 23458,c1(OC)c(C)cc(C(=O)NC2CCCC(N(C(=O)CSC3CC3)C)C2)cc1C 23459,N1(C(C=CC(=O)OCC)=O)C2CCCC1CC(NC(C1CC1CC)=O)C2 23460,c1(C(N(C(C)C(=O)NC2CC(C(=O)NOCC)C2)CCC)=O)cc(C)ccc1C 23461,N1(CC)C2CCC1CN(C(=O)CCCCN1CCCCC1)C2 23462,c1(C(=O)NCCN(C(C2C(CC)C2)=O)CC2CC2)cccc(Cl)c1O 23463,c1(C(=O)NC2C(NC(=O)CC3C=CCCC3)C2)c[nH]c2ccc(Br)cc12 23464,c1(C(=O)NCCN(C(c2cc(O)n(C)n2)=O)CC)ccccc1-c1ccccc1 23465,c1(N(CC(C)C)C(=O)NC(C)(C)C2CC2)cccn(O)c1=O 23466,c1(C(N2CC(SC)C(NC(=O)C(O)C(C)C)C2)=O)cc(S(N)(=O)=O)cnc1C 23467,N1(C(C(C(CC)C)OC)=O)C2CCC1CN(c1ncnc(Cl)c1OC)CC2 23468,C(=O)(C(O)C(C)SC)NCCN(C(Cc1nnc(C)o1)=O)Cc1cccc(Cl)c1 23469,C(=O)(CC1OCCc2ccsc21)N1C2CC(CNC(C(C)=CC)=O)C1CC2 23470,Cc1csc(C(C)CNC(=O)C=Cc2ncc[nH]2)n1 23471,c1(NC(C2(C)N(Cc3c(C)nc[nH]3)CC2)=O)cccc(C(O)C2CC2)c1C 23472,N1(C(CSCCNC(Cc2n(C)nnc2)=O)=O)CC2CC2C2CC12 23473,n1(C2(C(N(CCC)CCNC(=O)CCCN3CCCCC3)=O)CC2)ncn(C)c1=O 23474,C(=O)(CCC(CF)CF)NC(c1ccccc1)C(N1CCC(COC)C1)=O 23475,N1(C(c2occc2C2CC2)=O)CC2C3CCC(C2C1)N(C(=O)CCF)C3.CN 23476,N1(C(C2C(OC)CCC2)=O)CCC2(CCN(C(=O)CN3CCCCC3)CC2)C1 23477,c1(C(C)C(N2CCCC2C2CCN(C(C3CN(C)C3)=O)C2)=O)ccc(F)cc1Cl 23478,Cc1cc(Cl)cc(C(N2CCCOC(CNC(C3CC4(CCC4)C3)=O)C2)=O)c1C 23479,c1(C(=O)NCCN(C(=O)CC23COC(C2)C3)CC)ccc(C(F)F)s1 23480,N1(C(C(C)(C)SC)=O)CC2CS(=O)(=O)CC2(NC(c2ccc3cccnn23)=O)C1 23481,N1(C(C(COC)O)=O)CCOCC(F)(CNC(=O)CCc2ccccn2)C1 23482,CCS(=O)(=O)CC(=O)N1CCN(C(=O)CC2C=CS(=O)(=O)C2)C(CO)C1 23483,c1(CC)ccc(C(=O)NCC2COCC2NC(c2c(C)cncc2C)=O)cc1Cl 23484,C1(CC(=O)N(CCCNC(C2CC2F)=O)CC)COCCO1 23485,C1(CC)CN(C(=O)CCC(F)F)CCC1NC(c1cc(-c2ccncc2)on1)=O 23486,C1(NC(c2c(C)nn(C(C)(C)C)c2)=O)CC2CCC1N(c1ncncc1C#N)C2 23487,C1(O)(C(=O)NCC(C)CNC(=O)C(n2ccc(C(F)(F)F)n2)C)CCCCCC1 23488,C1(CNC(C(C2(O)CCOCC2)(C)C)=O)CN(C(C2CSCCS2)=O)C(C)(C)C1 23489,c1(CC(N2C(CNC(c3[nH]cc(CC)c3)=O)C(C)CC2)=O)ccc(O)cc1Cl 23490,CCCC(C(C)(C)C)NC(=O)CC(C)(C)NC(C1CCCN1C(C)=O)=O 23491,c1(CC)ccccc1OCC(N1CCCC1CNC(=O)C(C)(C)c1cnco1)=O 23492,CCCC(C(F)(F)F)NC(C1CCCC(NC(C2(Cl)CC2)=O)CC1)=O 23493,C1(OC2CN(C(CCN(CC)CC)=O)C2)CCN(C(=O)CC2CCOC2C)CC1 23494,c1(C(=O)NC2C(CNC(c3ccc(CC)[nH]3)=O)C2)ccc(NC)cc1Cl 23495,N1(C(C(C(C)C)O)=O)CC2=C(C1)CN(C(c1cccnc1-n1nccn1)=O)C2 23496,C1(C(=O)NC(C#C)C2CCC2)CC(NC(c2ccc([N+](=O)[O-])o2)=O)C12CCC2 23497,c1(C(=O)NCC2(NC(CC(C=C)(C)O)=O)CCCC2)n[nH]c2cccc(OC)c12 23498,Cc1cc(C(=O)N(CCC(C(C)C)NC(=O)CC2CCCO2)C)c(C)nc1C 23499,O=C(CC1CCc2ccccc21)NC1COC2CN(C(=O)Cc3csnn3)CC12 23500,CC1CCN(C(=O)C(F)CC2CC2)CCN1C(=O)CC1NC(=O)NC1=O 23501,c1(C(=O)NC23CC(NC(C4C(C)(CC)C4)=O)(C2)C3)cc(F)cc(F)c1N 23502,CC(C)CS(=O)(=O)CC(=O)N1CC(NC(=O)CCc2cscn2)CC1(C)C 23503,Cc1cccc(CCC(=O)NCCN(C(=O)CC2CCCN(C)C2)CC2CC2)c1 23504,c1(C(c2n(C(CC)(C)C)nnn2)NC2CCCCCC2)cn2cc(C)ccc2n1 23505,CC1CN(C(c2cccc(=O)n2C)=O)CC(C)C1NC(=O)Cc1cccs1 23506,C=C1COCCN(C(=O)CC(CC)N(C(=O)Cn2cnnn2)C)C1 23507,C(=O)(C#CC1CCOC1)N1C(CC)CN(C(c2cc(N)cnc2C)=O)CC1 23508,CCCC(C(=O)NC(CC)C(c1ccc(OCC)cc1)=O)N(C)C 23509,N1(C(C2(N(C)C)CCC2)=O)CCCC(CNC(=O)CCc2cnco2)C1 23510,c1(NCC(C2CCCCO2)(C)NC(=O)C)ncc(Cl)cn1.c1(C)ncoc1C1CC1 23511,C1(NC(=O)NCC(=O)Nc2c(CC#N)cccc2)CCCC(C)(C)C1 23512,c1(NC(C(N2CCC(CO)CC2C)c2nc(COC)sc2)=O)c(C)cccc1C 23513,O=S(=O)(c1ccc(NCC2=CCCC2)cc1Br)NCc1cscc1-c1ccccc1 23514,N1(C(CN(C(=O)OC)C)=O)CCC2(COC(CNC(c3ccccc3)=O)C2)C1 23515,c1(CNC(C2(N(C(C3CC(C)OCC3)=O)C3CC3)CCC2)=O)cc(F)ccc1O 23516,c1(C(=O)NCC2(NC(C(C(CC)C)C)=O)CC(OC)C2)cc2cccnc2[nH]1 23517,CCCC(C)(C)C(=O)NCCC1(C)CCN(C(c2cn(C(C)C)nn2)=O)C1 23518,CC(O)CCCCCC(=O)N1C(CNC(=O)C=C2CCCC2)CC2CCCC12 23519,C12CCCC(C1)NC(=O)CN2C(C1(N(C)C)CC1)=O.c1(CSC)ccccc1 23520,Cc1oc(Br)cc1C(N1CCC(O)C1c1cccc(Br)c1)=O 23521,C(C)(C(C(C)C)NC(c1ccc(SC)o1)=O)NC(c1ccn(CCCC)n1)=O 23522,c1(NCC(N2CCCCC2)C)nc(N2CC3CCC(CC3)C2)nc2ncn(C)c12 23523,S(=O)(=O)(c1cnc(N(C)Cc2conc2C2CC2)cc1C)N(CCF)CC 23524,c1(C(N(CC(=O)N(C(CN(C(C)=O)C)C)C)CC2CC2)=O)cn[nH]c1 23525,O=C(NNC(=O)C1CCC1)N1CCC(C(=O)NC)C1.c1(C(=O)CN)cccc(Cl)c1.C(CNCC)S.O 23526,N1(C(C2N(CC)CC2)=O)CC(C2(NC(c3cccc(CO)c3)=O)CC2)C1 23527,c1(C(N2CCC(C)(NC(c3ccc(COC)cn3)=O)C2)=O)ccc2occc2c1 23528,c1(OCC)cc(C(=O)NCC2CC(OC)C(=O)NC2)cnc1O.O(C)OC.O 23529,N1(C(=O)NC(C)CN2CCCCC2)CCC(c2nc(-c3ccccc3)no2)CC1 23530,N1(C(c2nncc(C)c2)=O)CC2CC(NC(=O)C(c3ccc(F)cc3F)C)C2C1 23531,C1(Nc2ccc(Br)cc2)CCN(N2CCOC3CCCCC23)C1 23532,CC(C)(O)C(F)(F)C(=O)N1CC(NC(C2CCC23CCOCC3)=O)C1 23533,CC(C)S(=O)(=O)CC(=O)N1CC2(CCN(C(c3ccn(O)c(=O)c3)=O)C2)C1 23534,c1(OC)nc(=NCC(C2CCCCC2)NC(=O)C=C(C)C(C)C)[nH]c2[nH]cnc12 23535,N1(C(c2cnc(C)o2)=O)CC2CCCC2C1C(=O)NCC(O)CF 23536,C(CCSC)(C(=O)N(C)CC1(NC(=O)CC2CSCCS2)CC1)OC 23537,c1(C(N(CCCNC(=O)CN(C2CCSC2)C)C)=O)ccc2c(n1)CCC2 23538,c1(C(N2CCN(C(=O)CCN3CCCC3)C(C3CC3)C2)=O)ccn2nccc2n1 23539,CC1(C)CN(C(c2cnns2)=O)CC1NC(=O)CNC(C1CCCC1)=O 23540,C1(C(=O)NCC#CCOC)(CNC(C2CCC(C)(C)C2)=O)CC12CCC2 23541,C(=O)(C1=NOC(CNC(c2cccc(CO)c2)=O)C1)NC(C(=O)N(C)CC)C 23542,N1(C(CC2(COC)CC2)=O)CCCC(C)(C)C1CNC(c1ccc(C)c(F)c1)=O 23543,N1(C(C(CC#C)O)=O)CC2CCC(C1)N2C(=O)CC(C)(C)COC 23544,c1(N2CCCCC(CNC(CC)=O)C2)cc2nnc(-c3ccccc3)n2cn1 23545,C(=O)(C1=CCC(F)(F)CC1)N(CCCNC(C1(COC)CCCOC1)=O)C(C)C 23546,c1(C(=O)NC2CC(C)N(C(=O)C(C)(C)CCC#N)C2)ccc2nc(CO)[nH]c2c1 23547,C1(C(N2CCC(F)(CNC(c3ncn(C)n3)=O)CC2)=O)CC2CCCCN2C1 23548,C(=O)(C(CCC(N)=O)n1cc(CCc2nn[nH]n2)nn1)NC(C12CC(CO1)C2)C 23549,Cc1ccc(CCC(=O)NC2CCCC2NC(C2(O)CCOC2)=O)c(Br)c1 23550,c1(C(N(C)CCC2CCO2)=O)ccc(-n2cccn2)cc1 23551,C1(C(=O)NOCCC(F)F)CCCCCCN1C(C1C2CCC(F)(F)C12)=O 23552,Cc1cc(C(=O)NC(C(C)NC(c2cnco2)=O)C(C)C)cc(N)c1Cl 23553,N1(C(CCOCCOCC)=O)CC2ON=C(CNC(c3cnn(C)c3)=O)C2C1 23554,C1(NC(C(n2cc(C)nc2)(C)C)=O)CN(C(c2ccncc2)=O)CCC1CO 23555,Cc1nn(C)c(C)c1-c1cn(C2CCCC2NC(C2CCC(=O)N(C)C2)=O)nn1 23556,C(=O)(C(CC(C)C)N(C(=O)CN1CC(=O)NC1=O)C)NCc1c(C)non1 23557,CCC(C(=O)N1CC(CNC(=O)CC(C)=C(C)C)(OC)C1)C(C)(C)CC 23558,N(C1CCc2ccc(Cl)nc21)C(=O)NC1(C)CCCC(F)(F)C1 23559,n1(CC)cnc(C(=O)NCc2occc2C(=O)N(C2CC2(C)C)C)n1 23560,CCC(C)(C)C(=O)C(=O)N1CCCC1C(C)(C)NC(=O)CC1CC1(C)C 23561,N1(C(CC(OCC)OCC)=O)CC(NC(c2ccc(Br)nc2Br)=O)C(C#N)C1 23562,S(=O)(=O)(c1c[nH]c(=NCCN2CCS(=O)(=O)CC2)cc1C)N1CC(C)=C(C)CC1 23563,CC(C)S(=O)(=O)CC(=O)N1CCCC(N(CCCOCC(F)F)C)C1 23564,C1(C(N2CCC(NC(CC=CC)=O)C23CC3)=O)CC(c2ccccc2F)=NO1 23565,N1(C(c2n[nH]cc2-c2ccccc2)=O)CCN2C(=O)OCC2C1 23566,Cc1cnccc1C(=O)NCCC1CCC(NC(=O)C#CC2CC2)C1 23567,C1(C(=O)NC(CC(C)NC(c2cn(C(C)C)nn2)=O)C)CCC(C(N)=O)CC1 23568,c1(CC)ccc(N)c(C(N2CC3C(CNC(=O)CC4C(C)C4(F)F)C3C2)=O)c1 23569,N1(C(CC=CC=C)=O)CCN(C)CC1C(=O)NCC(C)C(F)F 23570,C1(C)(NC(=O)C(O)CC(CCOC)SC)CCCN1C.c1(-c2c[nH]nn2)ccccc1 23571,N1(C(COCCCC#C)=O)CCC(NC(C2CCC(=O)N2CC)=O)C1(C)C 23572,C(=O)(CC(C)(C)CC(=O)N1CCC1CNC(C1CCN(C2CCC2)C1)=O)OC 23573,c1(NC(C)=O)c(C(=O)NCC2C=CC(NC(=O)CN3CCCC3)C2)cccc1C 23574,C1(NC(=O)CCn2ccnn2)CCC(NC(=O)C(C2CC(F)(F)C2)O)C1 23575,C1(NC(C2(C)CCCNCC2)=O)C2CC3COC1C3C2 23576,c1(C(=O)NOC2CCN(C(c3ncc[nH]3)=O)C2)cnn(C2CC2)c1 23577,c1(NC(C2CC23CN(Cc2scnc2Cl)C3)=O)cc2ccccn2n1 23578,Cc1ccc(C(c2nnnn2-c2ccccc2C)NC(C)(C)C)c(Br)c1 23579,N1(C(C2CCN(C(=O)OC)CC2)=O)CCC(C)(C)C1CNC(=O)C(C)N1CCC1 23580,CCCC(CC)CC(=O)NCC(O)CN(C)C(c1ccoc1CC)=O 23581,CC(c1ccccc1)=CC(N1CCC(C)(NC(C2(C3CCCO3)CC2)=O)CC1)=O 23582,N1(C(C(C)NC(N)=O)=O)CCC(N(C(=O)CN(C2CCCC2)C)C)C1 23583,N1(Cc2cnc(C)[nH]2)CCCC2(CCN(C(c3ncc(OCF)cn3)=O)C2)C1 23584,N1(CC(C=C)Cc2ccc(OC)c(OC(F)F)c2)CCc2[nH]nc(C(F)(F)F)c2C1 23585,C#CCCC(C(=O)NCCN(CCCC)C)NC(c1cc[nH]c1C)=O 23586,CCC(C)(COC)C(=O)NCc1ncoc1C1CN(C(C2CCN(C)C2=O)=O)C1 23587,N1(C(C(C)CC(F)F)=O)CC(C)(C)OCC1CNC(=O)CC1CC2CCC1O2 23588,Cc1cccc(CCC(=O)NCC(CNC(=O)CCc2cnoc2)CO)c1Br 23589,N1(C(c2c(CNC(C=Cc3n(C)cnc3)=O)ccs2)=O)CCC(N=[N+]=[N-])C(O)C1 23590,N1(C(c2c(C)ccnc2)=O)CCN(C(=O)CCC2CCCC(=O)N2)C(C2CC2)C1 23591,c1(C(=O)NC(C2CCN(C(c3cnco3)=O)C2)(C)C)ccn2nccc2n1 23592,S(=O)(=O)(c1cc(C(N)=O)ccc1F)N(C)Cc1c[nH]nc1C(F)F 23593,C1(NC(c2cncnc2)=O)CCCC(NC(C2OCCCO2)=O)CC1 23594,CCCC(C)(C)CN=c1[nH]c2c(c(=NCCC3CC(C)CC(C)(C)C3)[nH]1)CSC2 23595,N1(C(C2CC(CCC)C2)=O)CCN(C(=O)C(N)=O)C(C2CCC2)C1 23596,C1(C#CC(=O)N2CC(NC(C3CCC(C#N)CC3)=O)C(C)C2)(CC)COC1 23597,c1(C(C)C)cccc(C(N2CCC(F)(C(=O)NC(c3ccccc3)C#N)C2)=O)c1 23598,O(C1CCOc2c(F)cc(F)cc21)C(=O)CCCCc1cnn[nH]1 23599,Cc1cc(C(=O)N(CCNC(c2cnc[nH]2)=O)CCN2CCCC2)c(O)nn1 23600,c1(CC)ncccc1C(=O)N(C)Cc1cncc(Br)c1 23601,N1(C(c2c(Cl)cn(CCC)n2)=O)CC(NC(=O)COCC(C)C)CC1(C)CC 23602,C=CCC(CC(F)F)NC(=O)CC1CCCCC1NC(C1CCCSC1C)=O 23603,c1(C(=O)N(C2CCCCC2)CCNC(C2(F)CCCC2)=O)cc(F)cc(F)c1 23604,C#Cc1cccc(C(N2CCN(CCNC(=O)CC3CCC(O)C3)CC2)=O)c1C 23605,C1(OC)CC2CN(C(C3OCCC3CNC(=O)CCCC(OC)OC)=O)CC12 23606,C(=O)(CCCCCC(C)(C)C)NC1CC2(C(NC(c3c(C)cc(N)cc3)=O)C2)C1 23607,C12(C(=O)NCC(C(C)C)OC)CCCC1CCN2C(C1CC2C=CC1O2)=O 23608,CC(C)C(C)CCNC(=O)C(C(C)O)NC(=O)CN1C(=O)CNC1=O 23609,Cc1ccc(Cl)c(O)c1C(N1CC(NC(c2ccc(F)s2)=O)CC(C)C1)=O 23610,N1(C(C(CC(=C)C)C)=O)CCC2(CC1)CN(C(c1ccc3scnc3c1)=O)C2 23611,C1(NC(C=C(C)C)=O)(CNC(=O)C(C)Cc2ccncc2)CCCCC1 23612,c1(C(=O)Nc2cncc(OC)n2)cc2cc(-c3ccnc(F)c3)cnc2[nH]1 23613,C(=O)(C(C)C(CC)CC)NC1(CC=C)CCN(c2nc(CC)nc(C)c2Br)CC1 23614,Cc1cc(C(=O)N(C(C)CNC(=O)CC2CCCOCC2)C)cnc1O 23615,C1(NC(C(N2CCOCC2)C)=O)CC2(CCCN(C(C3C(C)C3C)=O)C2)C1 23616,C12(C(=O)NC3CC(C)(NC(C(C)OCCOC)=O)C3)CC3CC1C2C3 23617,N1(C(CC2CC(C)(C)OC2=O)=O)CC2CC(C1)CN(C(=O)C=Cc1ncc[nH]1)C2 23618,C1(NC(c2c(C(C)=O)cccc2)=O)COC2CNCC12 23619,C12(NC(C(C=CC)O)=O)CC(C)(C1)OC21CN(C(C2CC(F)C2)=O)C1 23620,Cc1cccc(Cl)c1CN1CC(O)(CNC(=O)CC2CCOC(C(C)C)C2)C1 23621,N1(C(C)=O)CCC(C)(C(=O)NCC2CC(C)N(C(C3CNC(=O)N3C)=O)C2)CC1 23622,CCCCC(C)C(=O)N(CC(CC)NC(=O)C(C)(C)CO)C 23623,N1(C(C(CC(=C)C)NC(C2CCC(C3CC3)C2)=O)=O)CCc2oc(C)nc2C1 23624,C#Cc1ccc(CC(=O)NC(C2CN(c3cc(C(F)F)ncn3)C2)C)cc1 23625,C1(NC(CNC(CC)=O)=O)CC2CN(C(c3cc(C)ccc3C)=O)CC12 23626,c1(OC)cccc(C(N2CCC(C(C)(C)NC(=O)CSC(F)(F)F)C2)=O)c1 23627,Cc1cc(NC(C2(CNC(=O)Cn3c(O)nnc3O)CC23CCC3)=O)c(C)cc1O 23628,CN(C)NC(=O)CCC(=O)N1CC2(CCN(C(c3ccc(CO)cc3)=O)CC2)C1 23629,c1(C(=O)NCC(C2CC2)NC(CN2CCP(C)(=O)CC2)=O)c(O)ccc(Cl)c1F 23630,C(=O)(C1CCCc2sccc21)NC1CCN(C(CCc2nnc(C)n2C)=O)C1 23631,c1(NC(c2cnc(-c3ccc(Cl)s3)s2)=O)c(O)cccc1O 23632,CC(C(=O)NC1(CNc2nc3ccc(F)cc3o2)CCOCC1)C(C)S(C)(=O)=O 23633,c1(C(C)C)cccc(C(=O)NC)c1.c12nc(nn1CCCN(C)C)C(C)(C)CS2 23634,c1(C(=O)NCC2(C)CCN(C(C34CCC(F)(CC3)C4)=O)C2)noc2ncccc12 23635,Cc1cc(CNC(c2coc(CNC(=O)CC3CCN(C)C3)n2)=O)sn1 23636,Cc1c(C(C)NC(=O)C(=O)N(C)C)oc2ccccc12.N12CCOCC(C1)C2=O 23637,CC1CN(C(=O)CC2(O)CCOCC2)CC1CNC(c1ccn(C)n1)=O 23638,CC(C(F)(F)C(F)(F)F)=CC(=O)N(CCCNC(c1cnn(C)c1Cl)=O)C 23639,N1(C(c2c(C#C)c[nH]n2)=O)CCCC(O)(CNC(=O)COC2CCC2)CC1 23640,c1(CNC(c2nnnn2C2CC2)C2(COC)CC2C2CCCCO2)cc(Cl)no1 23641,Cc1oc(CO)cc1C(N1CCN(C(C2CNC(=O)C2)=O)CC1)=O 23642,N1(C(Cc2cnc(C)[nH]2)=O)CC2CCC1C1CN(C(=O)C=CC3CC3)CC21 23643,C1(CCNC(CN(C)C2CC2)=O)CCN(C(C2CC3C(C2)C3(F)F)=O)CC1(F)F 23644,C(C(C#C)CC(C)(C)C)C(=O)N.N1CCCC(F)(c2n(C3(C(C)C)CC3)cnn2)C1 23645,C1(C(N2CCC(n3cc(C(C)N(C)C)nn3)CC2)=O)CCC2(CCC2)C1 23646,C12(CNC(CCOCCCOC)=O)CCN(C(=O)CC(C)(C)C)CC1C2 23647,c1(OC)ncnc(C)c1C(=O)NCC1CCN1C(C1CC(F)(F)C1)=O 23648,c1(C(=O)NC(CNC(C(C)(CO)NC(C)=O)=O)C2CCC2)ccc(C)c(C)c1O 23649,c1(C(=O)NCC=CCC(=O)Nc2cnn(CSC3CC3)c2)cc(C(F)F)no1 23650,C1(C(N(CCCCCNC(=O)CCN2CCCCC2=O)C)=O)CCC2(CCOC2)O1 23651,c1(C(=O)NC(C(=O)N(CC(C)O)CC2CC2)C)cc(CO)on1 23652,C1(O)(C(CNC(CCN(C)CC)=O)C)CCN(C(c2cc(CO)n(C)n2)=O)C1 23653,Cc1oc(C)c(C(N2CC(N(C(=O)CC3CC4COCC34)C)C2)=O)c1C 23654,c1(C(C)NC(C2CCN2C(C2(C)COC2)=O)=O)nnc(O)o1 23655,N1(C(c2ccc(OC)nc2F)=O)CCCC2(CCCN2C(C2CNC(=O)N2)=O)C1 23656,N1(C(c2cc(C)nc(C)c2)=O)CC(C)CN(C(c2nc(Cl)sc2Cl)=O)C(C)C1 23657,N1(C(c2cnc(OC)s2)=O)CC2CCC1C(CNC(=O)CCCC(N)=O)C2 23658,Cc1cc(Br)ccc1CNC(C1CCCCN1C(c1ccc(C)n1C)=O)=O 23659,c1(C(=O)NCCN(C(=O)CC(O)c2ccccc2)CCOC)nocc1C 23660,C1(CC(=O)NCCC2CCN(C(C3(C)CCCC3)=O)C2)CCCC1(F)F 23661,C1(NC(c2cnsn2)=O)CCC12CCN(C(c1onc3c1CCCC3)=O)CC2 23662,N1(C(C(C2CN(C(C3CCCCCC3)=O)C2)O)=O)CCN2CCCCC1C2 23663,c1(C(N(c2cc(C)c(Cl)cc2)C)=O)ccc2c(c1)COC2 23664,N1(C(C)=O)CCCC(C)(C(=O)N(C2(c3ccc(Br)cc3)CC2)C)C1 23665,c1(N2CC3CC(NC(c4cccc(C(C)C)n4)=O)C3C2)ncnc2c1CCO2 23666,N1(C(Cc2cc(CC)nn2C)=O)CCC(NC(=O)C(F)F)C(CC)C1 23667,N1(C(=O)OCC2CC2)CCC(O)(C(=O)OC(C)(C)C)C1.CCC1C(=O)N1 23668,N1(C(=O)Nc2n(C)nc(C)c2Br)CCCc2ncccc2C1 23669,C(C(=O)NOCCN(C)C)N(C(=O)CC1(C)OCCO1)C(C)C 23670,c1(OC)cc(F)c(S(=O)(=O)NC2CCCC2P(C)(C)=O)cc1OC 23671,c1(CC(=O)NC2CC(NC(C(n3cc(C)nc3)(C)C)=O)C2)cccc2nonc12 23672,S(=O)(=O)(c1c[nH]c(C(=O)NC2CCN(C(=O)C(C)(C)C#N)C2)c1)NCC 23673,N1(C(C)=O)CCCC(O)(CCNC(=O)C(C)(Cl)Cl)C1 23674,C(=O)(C(O)CC(F)F)NC(C1CCN(C(Cn2nc(C)c(Cl)c2)=O)CC1)(C)C 23675,C(=O)(C1=CCC(NC(c2cnn(C)c2Cl)=O)C1)N(C)CC1CC(F)(F)C1 23676,CC(C)(C)C(CN=c1ccn2ccnc2[nH]1)NC(=O)C(C)(C)c1cccnc1 23677,N1(C(Cc2scc(C)c2)=O)CC2(CNC(=O)C(C)n3cncn3)CC1CO2 23678,C12(CNC(c3ncc(Cl)cn3)=O)CC1CN(C(=O)CCCn1cccc1)C2 23679,C1(C(=O)NC2CCC(CCCC)C2)CCNC(C2CC2)C1 23680,N1(C(c2ccc(SC)o2)=O)CC(C)(C)C(NC(c2n[nH]cc2F)=O)C(C)(C)C1 23681,C(CO)(CCCO)C(=O)NCC(C)(C)Cn1cc(-c2cn[nH]c2)nn1 23682,N1(C(=O)OC(C)(C)C)CC2COCC2(C(=O)NC(C)(C)CN2CCOCC2)C1 23683,c1(C(=O)NC2C(CNC(C34CCC(OC)C3C4)=O)C2)[nH]c2ccccc2c1C 23684,c1(-c2cn(C3CC4(C(N5CCCC(SC)C5)=O)C3C4)nn2)ccccc1C#N 23685,c1(CC(N2CCC3C(NC(C4CC(CCO)C4)=O)C32)=O)ccc(F)cc1[N+](=O)[O-] 23686,C1(C(N2CCCC(F)(C(N)=O)C2)C(=O)NCCCCCC)CC12CCOCC2 23687,C(=O)(C(C)(C)CC(C)=O)NCC(=O)NCC(=O)NCC(C(CC)C)(C)O 23688,C1(CC(=O)NCC2(F)CN(C(C3(C)CCCOC3)=O)C2)CN2CCN1CC2 23689,CC1(C)CN(C(c2cc(CO)[nH]n2)=O)CC1CNC(C1CC1C#N)=O 23690,N1(C(C(C)OCCCC)=O)CC(C(N2CC(C(C)(C)O)C2)=O)CC(C)C1 23691,C(=O)(C#CC1CCCCO1)NCCN(C(C)C)C(c1ccc(OCCF)cc1)=O 23692,c1(C(N2C(C(C)NC(C3CC(C#N)C3)=O)CCCC2)=O)cc2cc(F)ccc2o1 23693,CCCCC(F)C(=O)N1CCCCC1C1CCN(C(c2ccc(F)cn2)=O)C1 23694,NS(=O)(=O)c1ccnc(C(=O)NCC(CO)NC(=O)CC2CN3CCN2CC3)c1 23695,Cc1ccc(C(C)C)cc1OCC(=O)NCC(CC(C)C)NC(=O)C1=CSCS1 23696,C1(C(N2C3CN(C(c4ncn(C)c4)=O)C(CC3)C2)=O)CCC(S(C)(=O)=O)CC1 23697,N1(C(COCCCC(C)C)=O)CCC2(C1)CN(C(C1CC1C(F)F)=O)C2 23698,CCC(O)CCN=c1[nH]c(N2CCN(Cc3cnsc3)CC2)nc2cccnc12 23699,c1(CC)nc(C(N2CCC(C(C)NC(c3cncs3)=O)C2)=O)co1 23700,c1(C(=O)NC(CC(C)NC(=O)Cn2ccnn2)C)ccc(-c2csnn2)cc1 23701,N1(C(c2ccc(C)nc2)=O)CCC2C(C1)CN2C(=O)CCn1ccc(O)nc1=O 23702,C(CC(C)C(=O)NCC(C)NC(c1c(C)nsc1I)=O)OC 23703,C12(NC(C=CC(=O)OCC)=O)CC1CN(Cc1cccc(CO)n1)C2 23704,C1(CC(=O)NCc2cccc(O)c2)CCCCN1C(=O)CN1C(=O)CNC1=O 23705,C1(NC(CC2C(=O)NCC2)=O)CC2CC(C1)N(C(=O)Cc1cnsc1)C2 23706,C12(C(N3CC4C(NC(c5cc(O)ccc5Cl)=O)C4C3)=O)CC3CC1C2C3O 23707,N1(C(C(COC)C)=O)CCC2(CCC(NC(C3CCC(F)C3)=O)CC2)CC1 23708,c1(C(=O)NC(C)CNC(=O)CC2CC3CC3C2)c(Cl)csc1Cl 23709,CC1CN(C(=O)Cc2cc(C3CC3)no2)CC1NC(c1cc(Br)c[nH]1)=O 23710,C(=O)(C(CCC)N(C)C)NCC(C)(C)NC(COCCOCC=C)=O 23711,C(=O)(CC(C)C(C)(C)NC(C1CC(C)(CC)C1)=O)NCC1(CO)C(C=C)C1 23712,N12CCC(CC1)C2=O.c1(NCc2onc(C(=O)OCC)n2)nccnc1SC 23713,c1(CC(=O)N(C(C)C(C)(C)O)C)ccc(NC(=O)OC(C)(C)C)nc1 23714,C1(NC(C(C2CCC2)OCC)=O)CN(C(c2ncccc2SC)=O)CC1C 23715,c1(C(=O)NC(C(C)NC(C2C=C(C)CS2)=O)C)cn2cccnc2n1 23716,c1(C(N2CC=C(CO)CC2)C(=O)NCCC2(C)CC2)noc2ccccc12 23717,c1(C(N2CC3(CCN(C(=O)CCC4CC4)C3)C2)=O)ccc(Cl)c2cccnc12 23718,c1(OC)ccccc1OCC(=O)NC(CNC(c1cn(C)nc1C)=O)C1CCC1 23719,CC(CC(=O)N1CCC(CNC(=O)C(c2cc(F)cc(F)c2)O)C1)C(C)(C)C 23720,c1(C(N2CCN(C(=O)C#CC3CCCCC3)CC2)=O)cnc2ncnc(O)c2c1 23721,Cc1ccc(C2(C(=O)NCc3c[nH]c(C#N)c3)CC2)cc1.C12CCCN1C(=O)N2 23722,C(C(C)(C)C(F)(F)F)N(C)C(=O)OC(C)(C)C.C12CN(C1)C(=O)N2 23723,CC1=C(C(=O)NC2CC3CC(NC(=O)C(O)CN(C)C)CC23)SCCO1 23724,N1(C(c2nn(CC)c(O)c2)=O)CCC2(CC1)CC2CNC(=O)CC(O)CC(C)C 23725,C1(C(=O)NCC2C3CN(C(C4(C)CCCCC4)=O)C2C3)CS(=O)(=O)CC(=O)N1 23726,O=C1CCN(C(C23CC(CO2)N(C(=O)C(C)(C)C2CCCO2)C3)=O)CCN1 23727,N1(C(c2c(C)nc(O)[nH]2)=O)CCC(NC(c2cc(C(F)(F)F)no2)=O)CC1C 23728,CC1CC(C(=O)NCc2ccc(C(=O)NOCC3(C)CCC3)cc2)CC(C)C1 23729,N1(C(C2C(OC(C)=O)C2)=O)C2CCC(C(=O)NC3(CC(C)C)CC3)C1CC2 23730,C(CC(C)C(F)(F)F)NC(C(CNC(C(F)=CCC)=O)NC(C)=O)=O 23731,Cc1nn(CC(=O)NCCCC(=O)NCCC2CCCO2)c(=O)o1 23732,C1(CNC(C2C(=O)NCC2)=O)CC2CC2N1C(c1ccn(CC(F)F)n1)=O 23733,n1(CC(=O)NCC(CNC(C2CC3CCC(C2)O3)=O)OC)nc(C)c(C)c1C 23734,C1(NC(C2(C)CC(NC(c3c(C)noc3)=O)C2)=O)CCOC2(CCC2)C1 23735,C1(O)(CN(C(=O)C(F)=CC2CC2)C)CCN(C(c2ccc(C(C)(C)C)[nH]2)=O)C1 23736,c1(C(=O)NC2(CCNC(C3C(C)CCC3)=O)CCC2)cc2c(F)c(F)ccc2[nH]1 23737,c1(C(=O)NCC(CN(C)CC2CCC(=O)N2)O)ccc(C(F)(F)F)cc1[N+](=O)[O-] 23738,c1(C(N(C2CCN(C(c3conc3C(C)C)=O)C2)CC)=O)cc(C(F)(F)F)co1 23739,C1(F)(CNC(c2ccc(C#C)cc2OC)=O)CC2CCC(C1)N2C(=O)C=C(C)C 23740,Cc1cc(C)n(-c2ccc(-c3nc(-c4ccn(C)c4)n(CCC(C)C)n3)nc2)n1 23741,c1(C(=O)NC2(C)CCN(C(c3c(CC)con3)=O)C2)cnc2c(c1)CNC(=O)N2 23742,C(=O)(C(O)CCNC(=O)C(O)C1CCCC1)NC(C1CCCC1O)C 23743,C1(CNC(Cn2c(C(C)C)ncc2)=O)COCCN1C(=O)CN(C)C(=O)C1CC1 23744,N1(C(C(CSC)C)=O)CC(NC(=O)C(CO)NC(=O)C(F)(F)F)CC(F)C1 23745,c1(SC(C(=O)NC2CC(CNC(Cn3nnc(C)n3)=O)C2)C)ccc(C#N)cc1 23746,N1(C(C=C(CC)C)=O)CC(NC(c2cnc(C)nc2C2CC2)=O)CCC1C 23747,CC(C)CC(F)C(=O)NCC1(C)CN(C(c2cc([N+](=O)[O-])c[nH]2)=O)CC1C 23748,N1(C(C(C)(Cl)Cl)=O)CCCC2(CCCN2C(c2cnc3ccccn23)=O)C1 23749,C1(COC)(NC(C23CC4CC2C3C4)=O)CCN(C(=O)C(c2ccc(O)cc2)F)C1 23750,N1(C(c2cnc(C)s2)=O)CC2(CC(NC(c3n[nH]c(C)c3Br)=O)CO2)C1 23751,c1(C(=O)NCC2(F)CCN(C(CCCCC#C)=O)CC2)cc(N)cc(C)c1F 23752,N1(C(c2c(CC)nc(C)[nH]2)=O)CC(NC(C2(C)CCN(C)C2)=O)CC12CCC2 23753,c1(CC)cc(C(=O)NC2(C)CCN(C(C3(c4ccnn4C)CC3)=O)C2)ccc1C 23754,c1(CCC(=O)N(CCC)CCNC(=O)CC(C)(O)COC)ccc2ncsc2c1 23755,C1(C(=O)NC(CNC(C=C(C)c2ccco2)=O)CC(C)C)CN(C)CC(C)O1 23756,N1(C(CC(C=C)CC)=O)CC(C)CN(C(=O)CCCc2cnn[nH]2)C(C)C1 23757,N1(C(Cc2ccc(C)s2)=O)CCC(C2CC2)C1CNC(=O)COc1ccsn1 23758,c1(C(=O)NC2CCN(Cc3cc(F)ccc3Br)CC2)ccc([N+](=O)[O-])c(Br)c1 23759,CCC(CC)CCCC(=O)NC(CC1CCC1)C(N1CC(O)CC1CO)=O 23760,CC(C(=O)NC1C=CC(C(=O)NC(C)C(=O)NCCF)C1)C(F)F 23761,C1(OC)CC(CNC(c2csnc2C)=O)N(C(C2CC(N(C)C)C2)=O)C1 23762,c1(-c2ncc(NC(CC3(C#N)CNC3)=O)s2)ccccc1OC(F)(F)F 23763,N1(C(C2(C#N)CCC2)=O)CCC2(CCCC2NC(C23CCCC2C3)=O)CC1 23764,CCCC(C(O)C(=O)NCC1(O)CCN(C)C1)NC(c1ccccc1CC)=O 23765,N1(C(c2ccc(OC)cc2F)=O)C2CCC1CC(NC(=O)C(C)CS(C)(=O)=O)C2 23766,C=CCCCC(C(=O)Nc1cccc2c1CCO2)NC(=O)CC1C=CCCC1 23767,c1(CC(=O)OCC)cnc(SC)[nH]c1=NCCCCNc1cc(F)ccc1F 23768,N1(C(c2c(N)cnc(Cl)c2)=O)CCCC(NC(=O)C=C2CCOCC2)C(F)C1 23769,C(C(C)(C(=O)NC(CNC(c1cc(Cl)c[nH]1)=O)C(C)C)OC)OC 23770,c1(CC(N2C(CCN(C(CC(CC)SC)=O)C)CCCC2)=O)ccc(C)c(C)c1 23771,Cc1c(C(=O)NCCCC(C)NC(C2CCCS2)=O)ccc(Br)c1F 23772,C1(CC=C)(C(=O)NC2CC(C(C)NC(c3cscc3Cl)=O)C2)CCOC1 23773,N1(C(C2(C)CCOC2)=O)CCC(C(F)F)(CNC(c2ncc(F)cn2)=O)C1 23774,C(=O)(C(C)Cn1ccc(C)n1)NCCCN(C(=O)C(C)c1ccon1)CC 23775,C1(C(=O)NC(CNC(c2c(C)cc(F)s2)=O)C(C)(C)C)SC2C=CC1CC2 23776,C#CC1(O)CCN(C(=O)C=CCN(C(=O)C(C)(C)C(=O)OC)C)CC1 23777,c1(CC(C)OC(=O)OC(C)(C)C)ccccc1Cl.S1(=O)(=O)CCN1C 23778,c1(C(=O)NC(C)C(C)(C)NC(=O)CC2COCCN2C)cccc(C(C)(F)F)n1 23779,N1(C(C(=O)NCC(C)N(C(=O)CCOCCCOC)CC)CC)C(=O)CCC1=O 23780,Cc1cnccc1CN1CCCC(CNC(C2C3CN(CC#N)CC23)=O)C1 23781,Cn1cnc2nc(N3CCC4(C3)CC4(F)F)nc(NCCCc3nc[nH]n3)c12 23782,Cc1nc2cccc(C(N3CC=CC(NC(C4(Cl)CC4(C)C)=O)C3)=O)c2s1 23783,C(=O)(C(C(F)(F)F)=Cc1ccccc1)NC(C)CNC(c1cc(C(N)=O)no1)=O 23784,N1(C(c2cnn(C)c2Cl)=O)CCCC(NC(=O)CC2CCC(C(F)(F)F)O2)CC1 23785,Cc1cc(NC2(F)CC2)ccc1C(=O)NCCCC(C)NC(=O)C1=CCCC1 23786,C(=O)(C(C)(CC1CCC1)OC)NCC1C(NC(CCNS(CC)(=O)=O)=O)CC1 23787,Cc1nnc2ccc(C(N3CCC(NC(=O)CC4(C)CC4(Cl)Cl)C3(C)C)=O)cn12 23788,c1(C(N2CCC(C(C)NC(C=C=C(C)C)=O)C2)=O)cccc2c[nH]nc12 23789,C(=O)(CC(O)CC(C)(C)C)NCCN(CC(C(C)C)OC)C(=O)COCC(C)(C)C 23790,C1(C(C)NC(=O)COCCN(C)C)CN(C(=O)CC2(CO)CCOCC2)CCO1 23791,Cc1nn(CC(=O)NC2CC3C(NC(=O)C(c4cnccn4)C)C3C2)c(=O)o1 23792,c1(CC(=O)NCC(C)CN(C(=O)CC2(c3ccon3)CCC2)C)ccc(F)cn1 23793,N1(C(C(C(C)O)(C)C)=O)CC2COCC2(C(=O)NCc2ccc(Cl)cc2)C1 23794,c1(C(C(=O)N(C(C)C)CCNC(=O)C(C)(C)C)C)c(F)cccc1F 23795,C1(C)(C(N2CCN(CCCNC(C(C(C)C)F)=O)CC2)=O)CCCCC1(F)F 23796,C1(C(=O)NCCCOC2CCN(C(C3OCC(C)C3)=O)CC2)CC(C(C)C)=NO1 23797,C(C(CCC)C(=O)NCc1ccc(CC)s1)NC(C(C=C)O)=O 23798,c1(C(N2CCN(C(CC(C=C)C)=O)CC2C2CC2)=O)ccn2ncc(C)c2n1 23799,N1(C(CSC)=O)CC2(C)CC1C2NC(c1ccc(=O)n(C(C)C)c1)=O 23800,C(C)(C)(C(=O)N1CCC(CCNC(=O)Cc2[nH]cnc2C)C1)OCC 23801,c1(C(=O)NC2CC(C)N(C(=O)CC3COCCO3)C2)ncc(Cl)cc1Cl 23802,c1(C(=O)NC2C(CCCC)CCC2)ccc(F)c2cccnc12 23803,c1(CC)ncsc1C(=O)NC1(CN(C(=O)CC(F)F)C)CC1 23804,CCCCC(Cc1ccccn1)NC(=O)NC(c1cccnc1)c1cccnc1 23805,C1(C(N2CC(C(C(=O)NC3C=CC(CO)C3)OC)C2)=O)CC(C)(CO)C1 23806,N1(C(c2c(SC)csc2)=O)CCC2CN(C(c3ncc(C)cc3C)=O)CC12 23807,C1(NC(CCOC(C)C)=O)CC2CCC1CN2C(=O)CC1(C#N)CCOCC1 23808,Cc1c(C(=O)NS(=O)(=O)c2cc(Br)c(Br)s2)cc([N+](=O)[O-])cc1I 23809,CCC(C)C(O)C(=O)NCC1(NC(=O)C2=NOC(C3(O)COC3)C2)CCCC1 23810,c1(C(=O)NC(C(CO)NC(c2cccc(C(C)=O)c2)=O)C)onc2c1CCCC2 23811,N1(CC(=O)N2C3CCC(CC3)C2=O)CCC(CO)C(F)(F)C1.CC(C)C(=O)ON(C)C 23812,C=CC(C)CC(=O)NCC1(OC)CN(C(=O)Cc2ncn(C(C)C)n2)C1 23813,c1(CC(=O)NC(CNC(COCCOC)=O)C2CC2)ccc(C(F)(F)F)cc1 23814,c1(OC)nc(Cl)cc(=NC(=O)C2CC2C(=O)Nc2ncc(C)c(Cl)n2)[nH]1 23815,c1(C(N(CC)CC2CCCN2C(=O)C=CS(C)=O)=O)cnn2cccnc12 23816,c1(C(N2CC(C)(CNC(c3c(C)c[nH]n3)=O)OCC2)=O)cc2c(s1)CCCC2 23817,c1(C(N2CCN(Cc3c(C)n[nH]c3C)CC2)=O)ccc(O)c(C(=O)C(C)C)c1 23818,S(=O)(=O)(c1cccnc1[N+](=O)[O-])N(C)CP(C)(C)=O 23819,c1(C(=O)NCCCN(C(=O)Cn2nccc2C)CC)ccc(CC(C)C)s1 23820,N1(C(CCOCC)=O)CC(CNC(=O)CN2CCSCC2)CC(C)(C)C1 23821,C1(O)(C(C)NC(Cc2c(C)scc2)=O)CCN(C(c2n[nH]c(C3CC3)c2C)=O)C1 23822,C1(C(=O)NCC(CNC(C2(CCOC)CC2)=O)C)Cc2cc(F)ccc2O1 23823,C1(C)(CNC(CCNC(Cc2c(C)noc2C)=O)=O)CC2CCC1C2 23824,N1(C(C=CC(CC)=CC)=O)CC2CCC1C2NC(C1C=CCC1)=O 23825,C1(N(C)C(c2ccc(C3CC3)o2)=O)CCC2CN(C(=O)Cc3nccn3C)CC12 23826,S(=O)(=O)(c1cnccc1N1CCS(=O)(=O)C(CO)C1)NC(c1ccc(Br)cc1)C 23827,C1(NC(CC=C)=O)CN(C(=O)CC)Cc2nccn2C1 23828,c1(C(C(=O)NCCCOC)N(C(C#C)C)C)c(Br)c(C)nn1C 23829,c1(NC(CC)CO)cc(Br)ccc1S(=O)(=O)NC1CCCN(C)C1 23830,CCCC(C)CC(=O)N1CCCC1(C)C(=O)N(CCCOCC)C 23831,C1(C2CCOCC2)(Nc2cccc(Cn3c(C)csc3=O)c2)CC1 23832,N1(C(c2c(C)ncn2C)=O)CCC(NC(C2(O)CC2)=O)C(c2ccccc2)CC1 23833,CCC(c1cccc(Cl)c1)=CC(=O)NCCCCN(C)C(C1CCCN1CC)=O 23834,C(=O)(C(O)CCCC)NC(C1(O)CCN(C(CSCCC)=O)C1)C 23835,N1(C(C(C2CCCC2)OCC)=O)CCC(CNC(c2cnc(O)o2)=O)CC1C 23836,N1(C(C=CC=CC)=O)CCN(C(=O)Cn2c(C)c(C)sc2=O)C(c2ncc[nH]2)C1 23837,Cc1cc(C(=O)NCC(C)(CC(C)C)NC(=O)C(C)Cn2ccnc2)c(C)cn1 23838,Cc1cc(C(C)C(=O)N(C)CC2CN(C(c3cncs3)=O)C2)cc(F)c1 23839,N1(C(c2nc(C)n(C)c2C)=O)CC(C)OC2(CCN(C(=O)C(N)=O)C2)C1 23840,N1(C(=O)NCC23CC(C(F)F)(CO2)C3)CC=CC12CCCC2 23841,C(=O)(CS(=O)CCC(F)(F)F)N1CCC(NC(C(CC)=CCCC)=O)CC1C 23842,c1(C(=O)NCC(CC)NC(c2cn(CCF)nn2)=O)c(OC(F)F)cccc1F 23843,c1(C(=O)NCC2(NC(CCC=C)=O)CCC2)sc2nc(C)nc(C)c2c1C 23844,Cc1ccc(-n2ccnc2)c(C(=O)NC2C=CCN(C(C3CC3C)=O)C2)c1 23845,c1(OCC(N2CC(C3CCN(C(=O)C(F)=CCCF)CC3)C2)=O)cccc(O)c1 23846,Cc1cc(=N)[nH]cc1C(=O)NC1CC(C)N(C(c2cn(CCF)nn2)=O)C1 23847,CC1=CC2CCCC(C1)N2C(=O)NCCCNC1CCC1 23848,CC#CCC(C(=O)Nc1ccc(O)cc1C)NC(=O)C(C)NC(=O)CC 23849,C1(C(N2CC(C)C2C(=O)NCCC2=CCOCC2)=O)CC2CCC(C1)N2C 23850,c1(C(=O)NC(CCNC(C(CCCOC)C)=O)C)cccc2c1C1CCC2CC1 23851,N1(C(C2(CCNC(C(C(CC)C)OC)=O)CC2)=O)CC2C=CCC(C2)C1 23852,c1(OC)c(Cl)nc[nH]c1=NCC1(CNC(c2cc(C(F)F)ncn2)=O)CCCC1 23853,C12(C(=O)NCc3ccc(C)c(Cl)c3)CCC(CC1)N(C(=O)C(O)CC(F)(F)F)C2 23854,c1(NCC(C2CCCCC2)NC(C2C(C)(Br)C2)=O)cnc2ccccc2n1 23855,S(=O)(=O)(c1c(C)ccc2nonc12)NC(CC)C(c1ccc(F)cc1)=O 23856,c1(OC)ccc(Cl)cc1NC(=O)CC1CCC(C)(C)CO1 23857,N1(C(=O)NCCCCCC)CC(Cc2cc(-c3ccccc3)n[nH]2)C(C)C1 23858,CCS(=O)(=O)CCNC(C1(C(C)NC(c2cnnc(O)c2)=O)CC1)=O 23859,c1(OC)ccccc1C(CNC(C1CCC(C)(C)C1)=O)NC(c1ccoc1)=O 23860,c1(CC2(NCCc3c(OC)cccc3OC)CCC2)ncc2c(ncn2C)n1 23861,N1(C(C(CCCC)C)=O)CCCC2CN(C(C3CN(CC(C)C)C3)=O)CC12 23862,C1(C(=O)NC(c2ccn(C)n2)C)(NC(Cc2c(C)ccs2)=O)CCN(C)C1 23863,C(C)(CNC(=O)C(n1nc(C)cc1C)C)(C(C)C)NC(Cn1ncc(CC)c1)=O 23864,N1(C(c2c(CC)cccc2)C(=O)NC)CCc2cc(C)cc(C)c2C1 23865,C1(CNC(c2n(CC)ncc2)=O)CC(OC)CN1C(c1cn(C2CC2)nn1)=O 23866,C(=O)(C1=CCCOC1)NC12C(CN(C(C(C)(C)CC3CC3)=O)C1)C2 23867,c1(C(=O)NCC2N(C(C(C(CC)C)O)=O)CC(F)C2)c2n(c(=O)n1C)CCCC2 23868,Cc1ccc(C(F)C(=O)NCC(=O)N(C)CC2CCOCC2)cc1 23869,Cc1nccc(CCC(=O)NCC2CCCCN(C(C3(C)CCCCO3)=O)C2)n1 23870,CCCCC(C(=O)NC)NC(C12CC1CCN2C(c1cc(C)ccc1O)=O)=O 23871,c1(NC(c2ncc(COC)[nH]2)c2nnnn2C(C)CC)ncc(OC)cc1C 23872,n1(C(CC)C)ccc(=NC(=O)c2ccc(C3CCCN3)s2)[nH]1 23873,C1(CNC(CC2(C)CC2)=O)CN(C(=O)Cc2cc[nH]c2)CCO1 23874,C(=O)(CCCCC(F)F)N(CCNC(c1nc(COC)sc1)=O)C(C)C 23875,C(=O)(C#CC(C)(C)C)N1C(C)(C(=O)NC(CCCC)C)C=CC1 23876,CC(CN=C(NCC1(N2CCCC2)CCCC1)NC1CCCC1)CC(F)(F)F 23877,N1(C(C(c2ccnn2C)NC(Cn2c(C)ccn2)=O)=O)CCC(C2CCC2)CC1 23878,C(=O)(CCC(F)(F)F)NC(C1(O)CCN(C(c2nn(C)cc2Cl)=O)C1)C 23879,C1(C)(NC(CCOc2ccc(C)cc2)=O)CCN(C(C2CC=CCC2)=O)CC1 23880,c1(OC)cc(CCNC(=O)C(F)(F)c2ccncc2)ccc1I 23881,N1(C(COC(C)=O)=O)CC2CCC2(CC(=O)NC(C)(CO)C2CCC2)C1 23882,N1(C(C(C2CCOC2)OC)=O)CC(C)(NC(=O)COC2CCCCC2)C1 23883,C(=O)(C(F)C(C)CNC(c1cncc(OC)n1)=O)NCc1n(CC)cnn1 23884,c1(OCC(=O)NC2(C)CN(C(C(CC3CCC3)OC)=O)C2)ccccc1C 23885,N1(C(CCC(=O)OC(C)(C)C)=O)CC2(C1)CN(C(c1cnn(CCF)c1)=O)C2 23886,N1(C(c2c(C)nn(C)c2C)=O)CC(NC(c2cnn(CCO)c2)=O)CC2(CC2)C1 23887,C1(CNC(c2c(COC)cco2)=O)C2CCCC1N(C(=O)Cc1csc(Cl)c1)C2 23888,CCCCCCCC(F)C(=O)N1CC(O)(CNC(C2CC3CCC2O3)=O)C1 23889,Cc1c(C(N2CCCC2C(C)NC(C2CCCN2C)=O)=O)cnn1CCO 23890,S(=O)(=O)(c1cccc(=NCc2ccn(CC)n2)[nH]1)NCCC(CC=C)(C)C 23891,N1(C(C(C)N(C(=O)C2=NOCC2)C)=O)CC(F)CC1C 23892,C1(OC)CN(C(=O)C(c2ccccc2)O)CC1CNC(=O)C(C)(C)OC 23893,C(CNC(=O)Cc1c(Cl)cnn1C)(CCCC)NC(CSCC=C)=O 23894,C(c1ccc(F)cc1F)=CC(=O)NCCC1(NC(C(CCSC)OC)=O)CCC1 23895,C(=O)(CCCCC(=O)OC(C)(C)C)N1CC(N(C(C2CC(C)OCC2)=O)C)C1 23896,C(=O)(C1=CC2C=CC(C1)C2)NC(COCC)C(=O)NC1CC(O)C(O)C1 23897,C(C)(C)(CCN=c1nc(C#N)[nH]cc1Cl)NC(c1ccc(OC)cn1)=O 23898,C1(C(=O)Nc2nc(C(F)(F)F)cs2)CN(Cc2occc2Br)CCN1 23899,C1(C(=O)NCCC2CCC(NC(Cn3c(C)ccc3C)=O)C2)CC(S(C)(=O)=O)C1 23900,Fc1ccccc1C(F)(F)CCCOCC1CCOC1 23901,c1(C(N(CC(CNC(COC(C)=O)=O)C)C)=O)c(Br)c(C)nn1C 23902,CC1SCCCC1C(=O)NC1CCN(C(=O)C=Cc2cnccn2)CC1 23903,N1(C(C(C)(C)O)=O)CCC(C2CCN(C(C3(CCCF)CC3)=O)CC2)C1 23904,N1(C(CCCOCC=C)=O)C2CCC1C(C(N1CCC(C(C)CO)CC1)=O)C2 23905,N1(C(CCSCCC)=O)CCN(C(=O)Cc2nocc2C(C)C)CCC1C 23906,C=CC(CC)CC(=O)NCC1(O)CCN(C(c2cnc(C)c(OC)c2)=O)C1 23907,CCC(C)CCC(=O)N1CCC(CNC(c2cncnc2C)=O)C1(C)C 23908,C(C)(C(=O)NCCN(CC(N1CCCC1)C)C(=O)C1CC1)OCC(C)C 23909,C#Cc1cc(NC(C2CC2CC(C)C)=O)ccc1C.C1C(N(C)C)C(=O)N1 23910,Cc1nsc(CN(C(=O)CC2C(NC(C3CC(=C4CC4)C3)=O)CC2O)C)n1 23911,C1(C(=O)NCCC(=O)NCC#C)CCCC(NC(=O)CN(CC)CC)CC1 23912,C1(NC(C(C)C2CC2)=O)CN(C(c2cc3scnc3[nH]2)=O)CC12CCOCC2 23913,c1(C(=O)NCC2(O)CCN(C(C3(SC)CC3)=O)C2)cnc2nc(C)ccc2c1O 23914,N1(C(C(CCCC)O)=O)CCOC2(C1)CN(C(=O)C(O)Cc1ccc(O)cc1)C2 23915,c1(C(=O)NCC2CCCN2C(c2ccc(O)cc2)=O)cc(Br)cc2c1OCC2 23916,C1(NC(c2ccn(C(C)C)n2)=O)CC(C(N2CC(O)(C(N)=O)C2)=O)C12CCC2 23917,c1(C(=O)OC)cc(Br)cc(C)c1NC1CN(C(=O)CCc2ncc[nH]2)CC12CC2 23918,Cc1ncnc(C(N2CCCC(NC(C3(F)CCCOC3)=O)C2)=O)c1C 23919,Cc1noc(C)c1CC(C)C(=O)N(C)CC1CN(C(C2CC3C=CC2C3)=O)C1 23920,N1(C(c2cc(C)c(C)o2)=O)CCC(C)(CNC(=O)CCNC(C2CC2C)=O)CC1 23921,C1(CN(C)C(C2C3CCCOC23)=O)COCCN1C(C1CC(N2CCCC2)C1)=O 23922,C(N=c1[nH]c2ccc(Cl)cc2[nH]1)C1(OC(F)F)CCCCC1.CO 23923,CCC(C)(C)CC(=O)NCC1OCCC1C(=O)Nc1cc(OC)ccc1O 23924,n1(CC)cc(C(=O)NC(c2cccnc2)C(=O)NCC2CCCS2)c(C)n1 23925,C(=O)(CCCCCn1cc(-c2ccccc2C(C)=O)nn1)N1C(CC)CC(C)C1 23926,c1(NC(CNC(C2CC(=C)C2)=O)=O)ccc(CC(C)C)nc1 23927,C1(c2nn[nH]n2)(C(=O)NC(c2noc(-c3ccc(Br)cc3)n2)C)CC[Si](C)(C)CC1 23928,c1(CC)cccc(C(=O)NC(C(=O)NC)C2CN(C(=O)CCN3CCCC3)C2)c1 23929,N1(C(C2(OC)CCC2)=O)CC(CC(=O)NCCn2nc(C)cc2C)C2(CC2)C1 23930,c1(C(=O)NCC2C(C)CCN(C(=O)CCc3cnc[nH]3)C2)cccc2nncn12 23931,CC(C)C(C)(C)C(=O)NCc1cc(C(=O)NC(C2(CO)CC2)C)n[nH]1 23932,O=S(=O)(c1ccc(NCC2(CO)CCCCO2)cc1Br)NCc1cc(F)ccc1F 23933,C1(NC(C(CC=C)CC)=O)CCC2(CC1)CC(NC(C1CC(CC)C1)=O)C2 23934,c1(SCC(=O)NCC2(OC)CCN(C(C(CC)SC)=O)C2)nc2ccccc2[nH]1 23935,c1(C(N2CCN(C(C(CCC)N(C)C)=O)C(C)C2)=O)sc2ccccc2c1Cl 23936,CC1(C)CCCC(CC(=O)NCC(C)(O)CNC(C2CC(O)C2)=O)C1 23937,CC1CC(C(N2CCCN(C(C3CC(NS(C)(=O)=O)C3)=O)CC2)=O)CCC1=O 23938,N1(C(c2cc(OCC)no2)=O)CC(C(=O)NC(c2ccccn2)C)C(F)C1 23939,c1(CC)nnc(CNC(c2cc(-c3ccccc3)on2)=O)s1 23940,C1(NC(COCCOC)=O)CC(NC(c2sccc2C#N)=O)C12CCC2 23941,C1(NC(CC(C)O)=O)CN(C(c2ccc([N+](=O)[O-])[nH]2)=O)CC1(C)C 23942,C(c1cccc(F)c1)=CC(=O)NC(CNC(=O)C(F)(F)CC1CC1)CO 23943,C1(C(=O)NC(C(=O)NCCCC)C)OCCOC1C 23944,CCS(=O)(=O)CC(=O)NC(C)(CNC(c1c(C2CC2)noc1C)=O)c1ccccc1 23945,c1(NS(C)=O)ccc(C2C(C(=O)NC(=O)CN(C)C(C3CC3)C3CC3)C2)cc1 23946,Cc1c(CC(=O)NCC2CC2CNC(=O)CC2CCOCC2)cccc1[N+](=O)[O-] 23947,N1(C(C2(CCC)CC2)=O)CCC(NC(=O)CC2CC(C)=NO2)C2(CCC2)C1 23948,N1(C(CCCC=CC2C(CCCC(=O)NC)C2)=O)CCn2nc(C)cc2C1 23949,C1(N)(CC)CCN(CC2CC(=O)CCO2)C1 23950,N1(C(C2(C=C)CCC2)=O)CC2C(NC(=O)CCCc3ccc(O)cc3)C2C1 23951,Cn1nnc2ccc(C(N3CCCC3c3ccc[nH]3)=O)cc12 23952,Cn1cnc(C#N)c1C(=O)NC(c1cccc(Cl)c1)CNC(=O)CS(C)(=O)=O 23953,CCC(C)C(C(=O)NCCC1=CCCCC1)N(C)C(c1cccc(OC)n1)=O 23954,c1(C(=O)NCCC2CCC(NC(CC3N(C)CCC3)=O)C2)nccc2occc12 23955,C(CC1CC1)(C(=O)NOC1CCC(O)C1O)NC(CC(COC)C)=O 23956,N1(C(C2C(C)N(C)CC2)=O)CCC2CN(C(=O)CNS(N)(=O)=O)C(C)C12 23957,c1(COc2c(C(CC)=O)cc(F)cc2)cccc2c1OCC2 23958,C(C(=O)N1CC(NC(=O)Cc2c(F)cncc2Cl)CC(O)C1)(C(C)(C)C)SC 23959,c1(OC)cc(NCc2cc(O)nc(O)n2)nc(OCCOC)n1 23960,c1(-c2c(OCCC)ccnc2)ccc2c(c1)CN(Cc1cnc(O)c(Br)c1)C2 23961,C1(C(N2C(C(=O)O)(CC)CCC2)=O)CN(C(c2cnc(C)s2)=O)CCC1O 23962,C12(CC(=O)N(C)CC3CCC(CNC(C(=O)NCC)=O)CC3)CCC(CC1)OC2 23963,CCC(CC)C(C(=O)N1CCC(F)(F)C(CNC(C2CC3(CCC3)C2)=O)C1)OC 23964,N1(C(CCC(=C)C)=O)CCS(=O)(=O)C(CCNC(c2coc(CC3CC3)n2)=O)C1 23965,c1(CNC(C2(CO)CC3C=CC2C3)=O)cc(O)ccc1O 23966,c1(C(N(CCN(C(C2C(C(C)C)C2)=O)C(C)C)C)=O)c[nH]nc1-c1cnn(C)c1 23967,c1(OC)ccc(C(=O)NC2CC(C)CN(C(c3c(C)cnn3C)=O)C2)c(F)c1Cl 23968,O1NC(=O)C(CCSC)NC(=O)CCC1.C1(C(=O)OC)CC1(C)C(F)F 23969,C1(NC(CC(C)SC)=O)CCN(C(C2CC(C)(c3ccccc3)C2)=O)CCC1(F)F 23970,c1(C(=O)NCC2C3CN(C(C4=CC(C)(C)C4)=O)CC32)[nH]cc2c1CCC2 23971,C(=O)(C(F)C(=O)NCCCOCCCCNC(=O)Cc1ccc(O)cc1)OCC 23972,c1(CCOC(c2cnn(CC)c2C(F)(F)F)=O)ccc(Br)cc1OC 23973,C1(CC(=O)NC(C)CNC(c2n[nH]cc2Br)=O)CCCCN1C 23974,CCC(C)CCCCC(=O)N(C1CCCN(C(c2cnc(S)n2C)=O)C1)C 23975,Cn1ncc2c(NC3CC4CN(C(C5C6CC7C(C6=O)C57)=O)CC34)ncnc12 23976,C(=O)(CCCCNC(=O)CCc1ccn(C)n1)N(C)CCC1CCC1 23977,CCC(C)CCCCC(=O)N1CCC(CC(C)NC(=O)CCCOC(C)=O)CC1 23978,CS(C)(=O)=Nc1ccc(C(N2CCN(C(=O)C(C3CCCO3)C3CC3)CC2)=O)s1 23979,C1(C(=O)NOCC2CCCO2)(C(C)C)CCCN1C(=O)C(C1CCOCC1)O 23980,c1(C(N(CC(CNC(C(C)=C(C)C)=O)C)C)=O)c(C)c[nH]c1CC(N)=O 23981,c1(SCc2n(-c3c(OC)nccc3)nc(CC(C)C)n2)cc2c(OC)cccc2[nH]1 23982,C#CC1(O)CC(C(=O)N(C(C)CNC(c2cc(CC)[nH]n2)=O)CC)C1 23983,Cc1cc(Cl)cnc1-c1cn(CCCC(=O)N(CC(C)(C)S(C)(=O)=O)C)nn1 23984,c1(OC)ccc(C2(C(=O)N(CCCCNC(=O)CN(C)C3CC3)C)CCC2)cn1 23985,C1(C(N2CC(C3(NC(C(c4ccnn4C)C)=O)CC3)C2)=O)CS(=O)(=O)CC(=O)N1 23986,N=c1cc(C(N2CCN(C(=O)C=CC3CCOC3)CC2CCO)=O)[nH]c(=N)[nH]1 23987,Cc1nc(-c2ccccc2)sc1C(=O)NC1(CCNC(C2(C)CC2(F)F)=O)CC1 23988,C1(NC(c2ccc(F)c(Cl)c2F)=O)CN(C(C2SCCS2)=O)CC12CCOCC2 23989,c1(C(=O)NCC2(F)CC(NC(C(C(C)C)F)=O)C2)sccc1S(C)(=O)=O 23990,c1(OCC=C)ncccc1OC(c1nnn(C)n1)c1nnnn1CCCC 23991,c1(OCC)ccnc(C(N2CC(CCNC(C3(OC)CCOC3)=O)C(C)C2)=O)c1 23992,C1(NC(c2ccc(N(C)C)c(F)c2)=O)CN(C(C2(C)C=CCC2)=O)CC1C1CC1 23993,CCCC(CCC)C(=O)N1CCC(CC(C)NC(C2CC(C)CC(C)C2)=O)CC1 23994,C1(C(C(=O)N(C(COC)C)C)C)CCN(C(c2ccns2)=O)C1 23995,n1(CCC=C)c(N(C2CN(C(=O)OC(C)(C)C)C2)C)nnc1-c1coc(C)n1 23996,c1(OCC(N2CCN(C(c3ccc(CO)cc3)=O)C3CC23)=O)ccc(Cl)c(F)c1 23997,c1(C(=O)NC(CC)(CNC(C2(C)CSC2)=O)CC)ccc2occc2c1 23998,c1(NC(C(C)N(C(C(CC)O)=O)C2CC2)=O)cnccc1C 23999,N1(C(C(CCC)C)=O)CCN(C(c2cc(C(N)=O)c[nH]2)=O)C2CCC12 24000,C(=O)(C1=C(C)N(CC)C(=O)NC1c1ccc(Br)cc1OC)N1C(CC)CCC1 24001,c1(C(=O)NC2(CF)CCN(C(C(C)N3CCC3)=O)C2)ncc2cc(Cl)ccn12 24002,N1(C(C2C(c3n(C)cnc3)C2)=O)CCCC2(CCN(C(=O)Cn3ccnn3)C2)C1 24003,CP(C)(=O)c1cncc(CNC(=O)NC(c2ncccc2F)c2ccccc2)c1 24004,C#CCC(CC(=O)N1CCOCC1C(C)(C)C)NC(=O)C(=O)N(C)C 24005,C=CC(C)(C)CC(=O)NC12COC(C1)C(NC(C1CCCC1(F)F)=O)C2 24006,C(CCCC(=O)NCC(CO)ON)N(C(Cc1n(C)nnc1)=O)C 24007,c1(C(=O)NCC(CNC(C2=C(C)OCCS2)=O)CO)ccc2c(c1)OC(C)(C)C2 24008,C1(C(=O)OCC2CC(=O)N(C(c3ccsc3)=O)C2)CCCN(C2CCCC2)C1 24009,n1(CC(=O)NC2CN(C(c3ccc(NC(C)=O)nc3)=O)C2)c(C)cc(C)nc1=O 24010,c1(OCCNC(=O)C(c2ccc(I)cc2)F)c(F)cc(Cl)cc1F 24011,c1(C(=O)NCC(CNC(=O)Cc2cncc(C)c2)OC)cnn2c1NCCC2 24012,N1(C(C(C)Sc2ccccc2)=O)CCCC12CN(C(c1ccccc1)=O)C2 24013,N1(C(C(C)=C2CCC2)=O)CCCC(C)(NC(=O)C(=Cc2cnn(C)c2)C)C1 24014,C(=O)(CCC(=O)C(C)(C)C)NCC1C(C)CCCN1C(C1CCCCC1(C)C)=O 24015,c1(C(N2CC(CNC(C=CC=CCC)=O)C(F)(F)C2)=O)c(S(C)(=O)=O)cnn1C 24016,C12COC(C)(C)CN1C2.c1(C(=O)NC2C(=C(C)C)CCCC2)ccc(O)c(F)c1 24017,N1(C(CCC(C)=O)=O)CCC2(CCCN2C(c2nn(C)c(C)c2Br)=O)CC1 24018,N1(C(CCNC(=O)OC)=O)CC(C(C)C)CC1CNC(=O)CC1CCCC12CC2 24019,C1(CC(=O)NC(C#C)C(C)C)CCCCN1C(=O)C(C)NC(=O)CC 24020,C1(NC(c2cc(C)sc2C)=O)CC12CCN(C(c1nccnc1N)=O)C2 24021,N1(C(CC(=O)NCC)=O)CCC2CC(NC(=O)C(C)SC)CCC2C1 24022,N1(C(c2ccnc(C)n2)=O)CC2CC(NC(c3csc(C(C)(C)C)n3)=O)CC2C1 24023,C1(NC(c2c(SC)csc2)=O)CC2CCC1(NC(=O)CC(C)(C)C#N)C2 24024,C(=O)(C(C)CC(F)(F)F)NCCCCCNC(c1ccc(OCC(C)C)nc1)=O 24025,c1(CC(=O)NCCC(CNC(C(CC)C)=O)O)cccc2cnccc12 24026,CCCCC(C)(F)C(=O)NC(CC(=O)NCC(O)C1CCC1)C1CC1 24027,c1(NC(=O)CC2CC(O)CN2C(C2CCCSC2)=O)cc(O)cc(F)c1 24028,CC1CN(C(=O)CNC(N)=O)C(C)CN1C(c1cc(N)cnc1Br)=O 24029,Cc1c(NCc2nocc2Br)ncnc1NC1CCCCC1C(N)=O 24030,N1(C(c2n(C)c(Cl)c(Cl)c2)=O)CCC2(CCCCC2NC(=O)Cc2cnc[nH]2)C1 24031,CCC(CC(=O)NC1CCC(C)N(C(c2nc(C)sc2C)=O)C1)CC(C)C 24032,c1(C(=O)NCCN(C(c2cc(C)ccc2N)=O)CC)coc2c(Cl)cccc12 24033,c1(N(C(C(C)C(F)(F)CN)=O)C2CCCCC2)c(Cl)cc(Cl)cc1C#N 24034,N1(C(CCC2(C)CCC(=O)N2)=O)CC2CCC(C1)C(NC(=O)CC1CC1)C2 24035,C12(C(=O)NC(CCOC)CNC(c3ccsc3SC)=O)CCC(OC)C1C2 24036,C1(CNC(C2(NC(C)=O)CCCC2)=O)CN(C(c2ncncc2Cl)=O)CC1C 24037,Cc1ccc2c(C(=O)N(C3C4CN(C(C5CCC(F)CC5)=O)CC34)C)onc2c1 24038,C=CCCC(C(=O)NCCC(O)C(=O)OC)NC(C1CCCCS1)=O 24039,c1(C(=O)NC2C(NC(CC3(C=C)CCC3)=O)CCCC2)cc(F)c2[nH]nnc2c1 24040,c1(OC)cc(C(N2CCCC2CNC(C2C(C#N)C2(C)C)=O)=O)cc(Cl)c1 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24058,N1(C(C2CC(C)(C(=O)OC)C2)=O)CC(NC(=O)Cc2cc(C)on2)C(O)C1 24059,CC1C(NC(c2c[nH]nc2C2CCC2)=O)CC2CCC1N2C(c1ccccc1)=O 24060,c1(CN(C2CCC2)C(C)=O)ccc(NC(=O)N(C)CC2(C)CCCO2)cc1 24061,C(=O)(C(C)CC(C)(C)C)NCCCC(CO)NC(C(COCC)SC)=O 24062,C1(NC(C2(CC=C)CC2)=O)CS(=O)(=O)C2CN(C(C3CC(OC)C3)=O)CC12 24063,N1(C(CC(C=C)(C)O)=O)CCC2(CC1)CC(NC(=O)C=Cc1ccc(SC)s1)C2 24064,c1(OCC=C)ccc(NC(C23CC(C(=O)NCC(C)C)(C2)C3)=O)cc1 24065,C1(C(N2C(C)(CNC(c3c(C)noc3C)=O)CCC2)=O)CC(C2CC2)=NO1 24066,C12(CNC(c3c(C)cccc3)=O)CCCC1CCN2C(=O)Cc1cnn(C)c1C 24067,c1(OC)cc(OC)cc(CN2CCC(O)C(C(=O)Nc3ccc(C)cc3F)C2)c1 24068,C1(CC(=O)NC2CC(C)OC2=O)CC(C)(C)CN1C(=O)CCC1CCCCC1 24069,c1(CNC2(c3nnnn3C3CCCCC3)CC(C)(CBr)C2)ccc(C#N)cn1 24070,C(=O)(C(C#N)C(C)C)NCC1(C(=O)NCCc2ncc[nH]2)CC(=C)C1 24071,C1(C(N2CCC(c3nn[nH]n3)C2)=O)(COC)CN(C(=O)C(Cl)=CCl)C1 24072,Cc1nc2sccn2c1C(=O)NC1CN(C(c2cccc3ccoc23)=O)C1 24073,C1(NC(CCC=C(C)C)=O)CN(C(=O)C2=CC(C)(C)C2)C2CCCCC12 24074,C(=O)(C1=CCCCC1C)NCCCCCNC(c1cc(COC)cn1C)=O 24075,C(CC(O)C(=O)N(C1CC(NC(=O)CCSc2ccccc2)C1)C)SC 24076,c1(CC(=O)NCCOCCN(C(=O)C(O)CF)C)ccccc1OC(F)F 24077,c1(N(CCCC(F)(F)F)C)nc2c(c(=NCC3(c4n[nH]c(=N)s4)CC3)[nH]1)CCC2 24078,c1(COC(C2CC(=C(F)F)C2)=O)cccc2ncccc12 24079,C1(C(N2CC(=C(CNC(CC(C)n3cccn3)=O)F)C2)=O)Cc2ccccc2O1 24080,c1(C(=O)NCC(COC)O)n[nH]cc1CNC(=O)CN1CCCC1C 24081,C1(C)(C(=O)NC2(C)CCCN(c3cc(C(C)C)ncn3)C2)CC(C2CC2)=NO1 24082,c1(C(N2CCC(O)(CN(C(C3C(OCC)C3)=O)C)C2)=O)cnc2cnccc2c1 24083,C(=O)(N1CC(O)CCO1)C1CC(=C)CN1C(=O)C(O)CC[S+](C)C 24084,C1(C)(C(=O)NC(CNC(c2cc(CC)c(CC)o2)=O)C)CCC2(CC1)OCCO2 24085,C1(C)(C(=O)NC2CCC(CNC(c3cc(CC)oc3C)=O)C2)CC(C(C)C)=NO1 24086,C1(C(N(C(C#C)C2CCC2)C)=O)CC(F)(F)CN1C(=O)CC1CCC(=O)C1 24087,CC1CCCC(CCNC(=O)CC2CC(O)CN2C(c2cnn(CCO)c2)=O)C1 24088,N1(C(C(OC)OC)=O)CC(CNC(=O)C2=NOC(C)C2)C(F)(F)C1 24089,N1(C(C(CCCCC)C)=O)CCCC2(CCCN2C(c2cccnc2C)=O)CC1 24090,Cc1nn(-c2ccccc2)cc1NC(=O)NC1C2CN(CC(O)C(F)(F)F)CC12 24091,Cc1cc(C)c(CC(=O)NCC(F)CNC(=O)C(c2ccccc2)=O)s1 24092,C(CC(O)C(=O)N1CC=CC1CNC(=O)CSC(C)C)SC 24093,C12(NC(C3CC4CCC3C4)=O)CCC(CC1)N(C(c1cnc3occc3c1)=O)C2 24094,n1(CC)nnc(C(=O)NCc2csc(CNC(c3cc[nH]n3)=O)n2)c1C 24095,c1(C(=O)NC2C(NC(CC3CC(=O)NC3)=O)CCC2)cccc2nccnc12 24096,Cc1nc(C2CC2)ncc1C(=O)NC(CCNC(=O)C(C)NS(C)(=O)=O)C(C)C 24097,CC(C)(C)CCCC(=O)NC1CCC(CCNC(c2cnn(C(C)(C)C)c2)=O)C1 24098,c1(CNC(C2C(C(C)C)CCC2)=O)nc2c(s1)CN(C(=O)C(C)CC(N)=O)CC2 24099,CC1CCCN(C(C2(C)CCCN2C(C2COCC(C)O2)=O)=O)C1CO 24100,N1(C(C2(C(F)(F)F)CC2)=O)CCC2CN(C(=O)C(F)(F)Cl)CC2C1 24101,Cc1cc(O)c(F)cc1NC(C1CCN(C(c2cscc2Cl)=O)C1C(C)C)=O 24102,N1(C(CCCC=C)=O)CC(C(N2CCCC2CSC)=O)C2(CC2)C1 24103,CC(CCC(=O)N1CCOC(CCO)C1)NC(=O)C=C1CCC1 24104,N1(C(CNC(C)=O)=O)CC(C(N)=O)(CNC(C2(c3ccno3)CCC2)=O)C1 24105,Cc1coc(C)c1C=CC(N1CC(O)(CCNC(C2COC(C)C2)=O)C1)=O 24106,C1(N(C(C=CC)=O)C)CN(C(=O)C(C)N(CC(F)(F)F)C)CC1(C)C 24107,c1(C(c2nnnn2CCCCCC)NCC(=C)Cl)cnn(C2CC2)c1.C1CCCO1 24108,c1(CC)[nH]nc(C(=O)NC2(CCNC(C3CN(C)C(=O)N3)=O)CCCC2)c1C 24109,C1(C(N(C2CCN(C(=O)OC(C)(C)C)CC2)C2CC2)=O)SC2C=CC1CC2 24110,CC(C)C(C)CC(=O)NCC1CCCC(CNC(=O)C=Cc2ccncn2)C1 24111,C1(C(N(C)CC2CCCC(NC(=O)CN3CCSCC3)C2)=O)CC2(CCCC2)C1 24112,Cc1c(C(N2CCN(C(c3c(Cl)cnn3C)=O)C3CC23)=O)cccc1O 24113,c1(COC)ccc(C(=O)NCC2CC(CNC(=O)CCc3cncn3C)CO2)o1 24114,N1(C(c2c(CC)ccc(Br)c2)=O)CCCN(C(=O)CC2CC(C)C2)CC1C 24115,c1(C(N(CCN(C)Cc2cn(CC3CCCC3)nn2)C)=O)nnc(O)nc1O 24116,C(=O)(CC(C1CC1)C1CC1)C(=O)CC1CCCN1C(=O)CCCn1cccc1.N 24117,S(=O)(=O)(c1cnc(NCCN2CCC(F)(F)C2)c(Cl)c1)N(C(C(OC)OC)C)C 24118,C1(C)(C(=O)NCCCNC(C2(C)CC(C(F)(F)F)C2)=O)CC2CC2C1 24119,C(=O)(C(O)CC(F)F)N1CC(O)(CCNC(CCC2C(C)=NOC2=O)=O)C1 24120,C1(CCOCC)CCCCC1NC(C1(CC)CN(C(C2CCCO2)=O)C1)=O 24121,C1(NC(C(C)OCC)=O)CC2CCC1CC2NC(c1cc(F)cnc1OC)=O 24122,N1(C(CS(CC)=O)=O)CC2N(C(c3ccc(C4CC4)nn3)=O)CCC2(C)C1 24123,c1(CNC(=O)NC(C2CC3CC3CC2C)C)ccc(F)c2c1CCC2 24124,c1(C(=O)OCC)c[nH]c(=NC(C(C)NC(=O)C2=CCCOC2)C(C)C)cn1 24125,C1(C(=O)NC2C(C)N(C(c3cc(Cl)cc(Cl)c3N)=O)CC2)OCC2COCCC12 24126,N1(C(COCCOCC#C)=O)CCCC12CCCN(C(=O)C=CC)C2 24127,CC1(C)C2CCC(C2)C1(C)C(=O)NCc1ccccc1CNC(c1csnn1)=O 24128,C1(C(=O)NN(CCCCC(C)O)C(c2cn(C3CC3)nn2)=O)C2CC3C(C2=O)C13 24129,c1(C(=O)NC(C)C=CC(=O)N(C2CCCC2)CCO)ccc2c(c1)CC2 24130,c1(C(=O)NCC(C)NC(C=CCOC)=O)cc(C)ccc1S(N)(=O)=O 24131,c1(C(=O)CN(C(C(CNC(C2(CC)CC2)=O)N(C)C)=O)C)ccncc1N=[N+]=[N-] 24132,c1(CC(N2C(C(C)(C)NC(C3CC4C=CC3C4)=O)CCC2)=O)cccc(Cl)c1Cl 24133,N1(C(C2(CC)COC2)=O)CCC(C2CCCN(C(=O)C=CCO)C2)CC1 24134,N1(C(c2c(C#C)c[nH]n2)=O)CCC(C2CC2)C1CNC(C1C=C(C)CS1)=O 24135,CC1CN=C(NC(C2CCCN2C(=O)OCc2ccccc2)=O)S1 24136,c1(C(C)C)ccc(C=CC(=O)NC23CCC2CN(C(=O)CC2CC(F)C2)C3)cc1 24137,Cc1nc2cnn(C)c2cc1C(N1CCC(=CCNC(=O)C(C)O)CC1)=O 24138,c1(C(=O)NCCC(CNC(c2ccnn(C)c2=O)=O)O)c2c(nn1C)CCSC2 24139,CC1CC(NC(C2CN(C)C(=O)N2)=O)CCN1Cc1cnc(-c2ccccc2)[nH]1 24140,c1(-c2ncc(C(C)NC3CCOC(C(=O)O)C3)s2)ccccc1F 24141,C1(O)(C(N(CCN(CCN(C(C)C)C(c2ccccc2)=O)C)C)=O)CC2CCC1C2 24142,C(=O)(C1=C(C#N)CCC1)NC(CC(=C)Cl)C(=O)N1CCCC(F)(CO)C1 24143,c1(C(N2CCCC(CNC(C3C(CC)CCO3)=O)C2)=O)cc2cc[nH]c(=O)c2s1 24144,C1(C(=O)NC2(C(=O)NCC3(OC)CCCC3)CC2C)CCC(=O)N(C)C1 24145,c1(C(N(CCCCCNC(C(CC)N(CC)CC)=O)C)=O)cc(C)ccc1F 24146,C1(C(=O)NCC2(F)CCN(C(=O)Cc3cccnc3)C2)Cc2cscc2C1 24147,CCC(CC(=O)NC(C)(CO)C(=O)NC1(CC(=O)OC)CC1)SC 24148,c1(CC(=O)NC2CCCCC2NC(c2csc(CC3CC3)n2)=O)ccc(O)cc1 24149,C12(C(N3CCCC(N(C(CCC(=O)NCC)=O)C)C3)=O)CCC(C1)C(C)(C)O2 24150,C(=O)(CCCCCF)NCc1c(C(=O)NCC2(OCC)CCOC2)nco1 24151,C1(C(=O)OCc2nnc(C)o2)CC(F)(F)CS1 24152,C1(C)(C(N(CCCN(C)C)CC)=O)CCCN(C(C2CCOCC2)=O)C1 24153,C1(C(COC(C2CCN(CC(=O)Cc3ccccc3)C2)=O)=O)CC2CCC1C2 24154,CC1(C)CCCC1CCNC(=O)C(=O)Nc1ccc(CN2CCCCC2)cc1 24155,S(=O)(=O)(c1ccc(N(C(C)CCC(C)C)C)cc1Br)NC(c1scc(CC)n1)C 24156,O=S1CCC(N=c2nc3sccc3c(N(CC=CCn3cncn3)CCO)[nH]2)C1 24157,C(=O)(CCS(N)(=O)=O)NCC(CCNC(=O)C(c1cccc(C)c1)O)OC 24158,N1(C(C(COCC)N=[N+]=[N-])=O)CCC2CN(C(C3CN(C4CCC4)C3)=O)CCC12 24159,Cc1ccn(CC(=O)NCC2(NC(c3cn(C)c(=O)cn3)=O)CCCC2)c(=O)c1 24160,c1(NC(c2ccc(Cl)nc2)C)[nH]c(=NCc2cc(N)ccc2F)nc2scnc12 24161,CCC(C)(CO)C(=O)NC1CCCCCC1NC(=O)Cn1cc(C(=O)NC)nn1 24162,N1(C(C(CC)OC)=O)CCN(C(C2CCC(C)(OC)CC2)=O)C2(CCC2)C1 24163,N1(C(C(C(C)C)OCC)=O)Cc2nccn2CC(NC(=O)C2=CCC(C)(C)C2)C1 24164,c1(C(=O)NC(CCC)C)cccc(-n2cc(-c3cnccn3)nn2)c1 24165,N1(c2nc(NCC(C)(C)C)c3c(n2)scc3)CCCC(C2CC2(F)F)C1 24166,c1(CC)cc(C(=O)NC(C2(O)CCN(C(C3(OC)CCOCC3)=O)C2)C)sc1C 24167,C(=O)(CCC(C(=O)N(CCCNC(c1cnn[nH]1)=O)C)N(C)C)OC 24168,c1(C(=O)NC23C(CN(C(CC#N)=O)C2)C3)ccc(N=Nc2ccc(O)cc2)cc1 24169,CC1CN(C(=O)Cc2cscn2)CCC1NC(c1ccc(C(C)(C)C)cc1N)=O 24170,C1(C(=O)NC2CCC(NC(C3(CSC)CCC3)=O)CC2)OCC2CCCC12 24171,c1(NC(C2CC2C(=O)NC2C3COCC23)=O)ncc(Cl)nc1Cl 24172,N1(C(CCP(C)(C)=O)=O)CCCC2C1CCCN2C(c1cc2cccnn2c1)=O 24173,C1(C(=O)NCCN(CCC)C(C2(CCC)CC2)=O)CCn2cnnc2C1 24174,c1(C(=O)NC2C(NC(C3CCC(C(=O)OC)CC3)=O)CC2)cc(SC)cc(F)c1 24175,C1(C)(CNC(C(C)OCc2ccc(OC)cc2)=O)CN(C(c2cccs2)=O)CCO1 24176,c1(CNC(N2CCC(c3ccncn3)C2)=O)cc(O)ccc1F 24177,N1(C(c2c(OC)c[nH]n2)=O)CC2OCCN(C(C3CC34CCSCC4)=O)C2C1 24178,C1(N(C)C(C2CC(C)(O)C2)=O)CCCN(C(C2CC23CC(F)(F)C3)=O)CC1 24179,c1(CNC(C(COC)OC)=O)ccc(CC(C)NC(c2c[nH]c(C#N)c2)=O)cc1 24180,C(=O)(C(O)C(C)(C)C)N1CCC(CC=C)(C(=O)NCc2cncnc2)C1 24181,C12(NC(=O)Cn3cncn3)CC(CNC(C3(N4CCOCC4)CCCC3)=O)(C1)C2 24182,CC1CCn2cc(C(=O)NCCC3=CCN(C(=O)Cc4nc[nH]n4)CC3)nc2C1 24183,c1(C(=O)NC2CC(C)(COC)N(C(=O)C=CCF)C2)cc(=O)n2nccc2[nH]1 24184,N1(C(C2C(C)OCCC2)=O)CCCC(CO)(NC(c2cccc(N)c2)=O)C1 24185,C=CC(C)(C)CCN=C(NC1CCC1)NC1CCN(C(=O)NC2CC2)C1 24186,c1(C(=O)NC(C2CCCN(C(=O)CCC(F)(F)F)C2)C)cc2cccn2c(O)n1 24187,C12CCCN(C1)C(=O)CNC(=O)C(N(C)C)CNC(=O)N2.C(C)(C)(C)NC(N)=O 24188,Cc1ccccc1C(C)(C)CNC1CCOC(c2ccc(F)cc2)C1 24189,c1(C2(C(=O)NC(C)CC3CN(C(=O)CC4CSC4)C3)CC2)ccncc1 24190,C(CC(O)CNC(C1(c2ccccc2)CC1(F)F)=O)NC(c1coc(Cl)n1)=O 24191,C1(CNC(C=Cc2n(CC)ncc2)=O)CCC12CCN(C(C1(CC)CC1)=O)CC2 24192,CCCCC(C)CCC(=O)NC1(COC)CN(C(=O)C(CC)N(C)C)C1 24193,c1(C(N2CC(O)(C(C)NC(c3cc(Br)no3)=O)C2)=O)ccc2c(c1)CCC2=O 24194,Cc1cc(C(=O)NCC2(NC(=O)C(C)OCCC(C)C)CCC2)c(O)c(C)n1 24195,c1(CCC(=O)NC2CN(C(c3c(C)n[nH]c3)=O)C(C)CC2)n[nH]c2c1CCCC2 24196,CS(=O)(=O)CCC(=O)NC1(CF)CCN(C(=O)COc2cccc(CSC)c2)C1 24197,S(=O)(=O)(c1cc(Br)ccc1Br)N(C)CC1CN(C(c2ccnc(Cl)c2F)=O)C1 24198,c1(CCNC(C2(OCOC)CCOCC2)c2n(CCC)nnn2)cncc(F)c1 24199,C(=O)(CC1=CCN(C(=O)C(c2cccnc2)O)CC1)NC(CCCC)(C)C 24200,C1(CC=C)(NC(c2ccccn2)=O)CN(C(c2nc(C(=O)OC)cs2)=O)C1 24201,O=C1NCCC2CCN(C(c3cc4occc4s3)C(=O)NCc3ccco3)C12 24202,c1(-n2cc(C(C)N(C)C(C3(CO)CCCCO3)=O)nn2)cccc2c1OCO2 24203,c1(OC)cc(F)c(C(=O)NC2CCN(c3ccc(Cl)c(Cl)c3)C2=O)cc1OC 24204,c1(OC)ccc(CC(=O)NC2(CCCNC(=O)CC3CCCCN3C)CC2)cn1 24205,C1(C(=O)NC2C(CC(=O)NC(C3(CO)CCC3)C)C(O)C2)CC2C=CC1O2 24206,Cc1c(C(=O)NC(C2CCCN2C(=O)Cn2cnc(=N)[nH]2)(C)C)ccn1C1CC1 24207,C1(C(c2nnnn2CCSC)NCc2conc2C)(CC)CCOCC1 24208,N1(CC)CCC(C(=O)N(C)CC=CC(=O)NC2CC2C)C1 24209,n1(CC)ncn(NC(=O)Cn2cc(CNC(=O)CC3COCCO3)nn2)c1=O 24210,C1(CNC(=O)C=CC2CC2)CC2CN(C(=O)C(c3ccccc3F)O)CC12 24211,c1(C(NNC(=O)C2CC(N)C2)=O)csc(S(=O)(=O)N2CCOCC2)c1 24212,C1(C(C)(C)C)CC(C(=O)N2CCC(CO)C(NC(c3csc(CO)n3)=O)C2)=NO1 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24230,C(=O)(C(F)C(C)(F)F)N1CC(C)(OCC(=O)N(C)CC2CC2(F)F)C1 24231,C(C1=CCN(C(=O)Cc2ccc(Br)cc2F)CC1)NC(Cn1c(C)cnc1)=O 24232,C(=O)(CC(C)C(F)F)NCCCC1CCN(C(C2(CC)CC(F)(F)C2)=O)CC1 24233,c1(C(=O)NC(CC2CCOCC2)C(=O)N2CCC2CO)ncnc(O)c1F 24234,c1(C(=O)NC2CC(N(C(c3cnc(OCC)s3)=O)C)C2)nccc(OC)c1N 24235,CC(C)C(C)N=c1[nH]c(N2CNC(=O)C2)nc2c1CCCC2 24236,c1(C(CC)NCC2CCC(C)O2)ccc(O)c(Br)c1 24237,c1(C(N(CCC)CCNC(=O)C(C)C2CCOC2)=O)c(F)ccc2nc[nH]c12 24238,C(CC(C(C)C)(c1nnnn1CC(F)F)Nc1ccc(CO)c(F)c1)OC 24239,C(CCC(=O)N1CC(C(N)=O)C1)(C(C)C)NC(C=Cc1cc(C)no1)=O 24240,c1(C(=O)NCCC2(C)CCN(C(=O)CCC3CC3)C2)ccn2ccnc2c1 24241,Cc1cc(C(=O)NCC2(CNC(=O)C=Cc3cncs3)CC2(F)F)ccc1O 24242,CC1C2CC(C2NC(C2CCC(F)(F)CC2)=O)N1C(c1c[nH]c(=O)cn1)=O 24243,C1(CC)CN(C(=O)C(C2CCCCC2)O)CCN1C(c1cc(C)n(C)c1)=O 24244,N1(C(C(CC)OC)=O)CCN(C(c2cc(S(C)(=O)=O)co2)=O)C2CCC12 24245,C1(C(N2CC(C)C(N=[N+]=[N-])C2)=O)CC(F)(F)C12CCCC2 24246,c1(C(=O)NC2C3(CC(NC(=O)COCC(F)F)C3)C2)ccc2cnnn2c1 24247,C1(NC(C2CCCC(NC(CC3(C#N)CC3)=O)C2)=O)CC2(CNC(=O)O2)C1 24248,CC1CCN(C(=O)CCc2c(F)cccc2F)CC1NC(=O)C=C1CCCCC1 24249,N1(CC(=O)NCC2(O)CN(C(c3c(N)cc(Cl)nc3)=O)C2)CCCCCCC1=O 24250,C1(NC(c2c(Cl)cn(CC)n2)=O)COCCN(C(=O)C(C)Cn2ccnc2)C1 24251,c1(C(=O)NC(C(=O)NC(CCOCC)C)c2cccs2)cc2ccccc2o1 24252,C(C)(C(=O)NCC1CC(SCCC(=O)S(=O)(=O)CCC(N)=O)C1)OCCOC 24253,N1(C(C2CC(=C)C2)=O)CCC(CF)(NC(c2cnc(C3OCCO3)s2)=O)C1 24254,c1(N2CC(C)(C)SCC2)nc(N2CCOC(C)(C3CC3)C2)nc2c1SCC2 24255,C1(CC)CCCCC1C(N1CCC1(C)C)C(=O)Nc1ccccc1Cl 24256,c1(CC(=O)NCC2C(NC(CNC(C3C(C)C3)=O)=O)CC2)ccc(C2CC2)cc1 24257,Cc1c(CC(=O)NCC2(CCNC(=O)CC3CC=CC3)CC2)ncn1C 24258,N1(C(C(=O)NCC)=O)CC2COCCC2(NC(c2ccnn2CCOC)=O)C1 24259,Cc1cccc(C(=O)N(C2CCC(NC(C3CN(C)CCO3)=O)CC2)C)n1 24260,N1(Cc2c(C(=O)O)cccc2)CCC2(CCC(C(=O)NC(C)(CO)CO)O2)CC1 24261,c1(C(N(CCN(C(CC(COC)C)=O)C(C)C)C)=O)ccc(S(N)(=O)=O)cc1N 24262,C1(C(N2CCC(OCCNC(C(C=C)O)=O)C2)=O)CCC2C(CC1)C2(F)F 24263,N1(C(c2c(C)ccs2)=O)CCC(NC(=O)C(c2ccc(F)cc2F)C)C(F)C1 24264,C=CC(CC(=O)NC(C1CCN(C(=O)CC(F)(F)F)CC1)(C)C)c1ccccc1 24265,C(=O)(C1=C(Cl)CCC1)N(C1CCN(C(=O)C(c2cccnc2)OC)CC1)CCC 24266,c1(OCC=C)ccc(Cl)nc1C(=O)NC1CCCCC1NC(=O)C(O)C(C)(C)C 24267,c1(CC(=O)NC2CC2CNC(C2CS(=O)(=O)C2)=O)cc(F)c(F)cc1F 24268,C(C(C)C(F)C(=O)N1CC(OCC(F)F)C1)NC(c1cc(CCC)[nH]n1)=O 24269,C1(C(=O)NCC2(C)CCN(C(c3nccc(CC)c3)=O)C2)CCCCS1(=O)=O 24270,c1(C(=O)OC)cnc(NCC2CC(C)N(C(=O)CN(S(C)(=O)=O)C)C2)nc1 24271,c1(C(C(N2CCC(O)(C(C)C)C2)=O)(F)F)ccc2c(c1)OCO2 24272,Cc1cncc(C(=O)NCC2CC2CNC(c2ccc(=N)[nH]c2Cl)=O)c1Cl 24273,N1(C(c2cc(C)nn2C)=O)CCN(C(c2c(C)coc2C)=O)CC12CC2 24274,c1(OC)ccc2nc(N3CC(NC(C4(C)COC4)=O)C(C)(C)C3)sc2n1 24275,N1(C(c2cccn(C3CCSC3)c2=O)=O)CCS(=O)(=O)N2CCCC12 24276,Cc1cc(C)nc(CNC(=O)CCCC(C)NC(=O)CC2C=NN(C)C2=O)n1 24277,Cc1ccc(Br)c(F)c1C(N1CC2CN(C(c3ccc(O)c(I)c3)=O)CC2C1)=O 24278,C(=O)(CC(O)C(C)C)NC(CCOC)C(=O)NC12CC1CN(C)C2 24279,N1(C(CN(C(=O)C(O)C(C)CC)CCC)=O)CC2(COCC(=O)N2)C1 24280,c1(C(=O)NC2CC(NC(CN3C(C)CC3)=O)C2)cnn(CCO)c1N 24281,N1(C(=O)NCc2c(CC)ccc(F)c2)CCc2cc(OC)ccc2C1C 24282,c1(C(N(C2CCN(C(C3CC=CCO3)=O)C2)CC)=O)nc(OC(C)C)ccc1Cl 24283,c1(C2(C(=O)NCCNC(C3(C#N)CC3C(F)(F)F)=O)CC2)ccc(O)cc1 24284,C(C(=O)N1CC(NC(=O)CC2(CO)CCC2)C(C)C1)(C(C)(C)C)NC(C)=O 24285,c1(C(=O)NC2(CNC(=O)CC3CCCS3(=O)=O)CCCC2)cccc2nsnc12 24286,C1(C(=O)NCCCN(C(C(C)SCC)=O)CCO)CCCC1n1ccnn1 24287,C(C(CC(C)C)C(=O)N(C)Cc1c(C)cnn1C)NC(CC(C=C)C)=O 24288,C1(NC(C(CC)N(CC)CC)=O)COCCC1NC(c1cnc(C2CC2)s1)=O 24289,N1(C(C(CC)C)=O)CCN(C(=O)CNC(c2ccccc2C)=O)CC1 24290,c1(CC)cccc(C(=O)NCC2CCCN(C(=O)CN(C)C(C)=O)C2)c1N 24291,c1(OCCNC(CC(CC)N(C)CCO)=O)ccccc1C#N 24292,C1(C(=O)NC(CC)CC2CCOCC2)CCC(C2CCC2)CC1 24293,c1(CC)ccc(C(=O)NCCC2(C)CCN(C(c3ocnc3C3CC3)=O)C2)cc1 24294,N1(C(c2c(COC)noc2)=O)CC2CC(NC(=O)C(C)CCO)C2C1 24295,c1(C(=O)NC2CCC(CNC(C3(COC)CC(=C)C3)=O)C2)c(F)cc(Cl)cc1F 24296,N1(C(c2n(CC)ncc2)=O)CC2(CC2)CC1C(N1CCC(N2CCC2)C1)=O 24297,C(=O)(CCCCCN=[N+]=[N-])N1CC(CC)N(C(=O)CC(C)c2cnn(C)c2)CC1 24298,CCC(C)C(O)CC(=O)NCC(CC(=O)N1CCOCC1CC)OC 24299,c1(C(=O)NCC(CN(C(C(C)SCC)=O)C)O)ccn(CCN(C)C)n1 24300,c1(CCC)cccc(C(=O)NC2CCCC2CNC(c2ocnc2C)=O)c1 24301,N1(C(c2c(SC)snn2)=O)CC(NC(C2(C(C)(C)C)CCCCC2)=O)C(C)C1 24302,c1(C(N2CCC(C)(CNC(C3CC(SC)C3)=O)CC2)=O)cc2cc(Cl)cnc2[nH]1 24303,CC1(C)CCCOC1CC(N1CCOC(CNC(C2CC(Cl)(Cl)C2)=O)C1)=O 24304,N1(C(C(C2CCC2)OC)=O)CC(CNC(C2CCCCC2O)=O)C(C)C1 24305,Cc1cc(C(N2CCC(N(C(=O)CCCc3sccc3C)C)CC2)=O)[nH]c1C#N 24306,C1(C(N2CCC(N(C(C(c3ccccc3F)C)=O)CCO)C2)=O)C(C)(C)C1(F)F 24307,Nc1ccc(CCCC(=O)NC2CCOC(CNC(=O)COC(F)(F)F)C2)cc1 24308,Cc1ccc(S(=O)(=O)N2CCN(CC(=O)NC3CCCC3)CC2)nc1 24309,Cc1ncnc(C(N2CC3(C(=O)NOCCC(C)C)CC2CO3)=O)c1C 24310,C=CC1CCCCN1C(=O)Cn1cc(CNC(c2cc(C(C)=O)c[nH]2)=O)nn1 24311,c1(C(=O)NC(C2(CNC(C3(CCOC)CCC3)=O)CC2)C)ccc(C)cc1 24312,c1(CC(=O)NC(CNC(C2C(CC)CCO2)=O)(C)CC)cnn2ccccc12 24313,N1(C(c2n(CC)ccc2)=O)CC(N(C(=O)C=Cc2cc[nH]c2)C)C2(CC2)C1 24314,c1(N2CC(OC)C(F)C2)nc(Nc2cc(N)ccc2F)c2cnn(C)c2n1 24315,n1(CCC)cc(C(=O)NCC2(NC(=O)CC3CCNC3=O)CCC2)c(C)n1 24316,Cc1ccc2c(C(=O)NC3CCN(C(=O)C#CC4CC4)C(C)C3)n[nH]c2c1 24317,c1(NC=O)ccc(C)cc1.C1(C2(CC(=O)NCCN(C=O)C)CC2)(COC)CC1 24318,c1(C(=O)NCC(CC)NC(CCCCOCCC=C)=O)ccc(S(N)(=O)=O)[nH]1 24319,N1(C(c2c(C)ncc(Cl)c2)=O)CC2(CCN(C(=O)C3=CCCCC3)CC2)CC1C 24320,N1(C(C(C)OCCC(C)C)=O)CCCN(C(c2cnc3c[nH]nc3c2)=O)C(C)C1 24321,C1(CC)CCOC1C(=O)NC1CC(NC(=O)CC2(O)CCCC2)C1 24322,N1(C(CC(C(C)C)O)=O)CCCCC12CC(NC(=O)COC1CCCOC1)C2 24323,C1(C(C(=O)N(CC(O)CN(C)C(c2cc(O)cs2)=O)C)O)CCS(=O)(=O)CC1 24324,Cn1cc(C(=O)NC2CC3(C2)CC3NC(C23COCC2C3)=O)ncc1=O 24325,C(=O)(CC(F)(F)F)NC(C)C(=O)NCC1(NC(c2coc(CO)c2)=O)CC1 24326,CC(N=c1[nH]c(N(C)CCC2CN(C)C2)nc2c1CCC2)c1nnc2n1CCC2 24327,N1(C(=O)CC2CCSC2)CCCC(n2cc(COc3ccc(Br)cc3)nn2)C1 24328,C1(CNC(c2cnc(CC(C)C)[nH]2)=O)CCC(CNC(C2CCN(C)C2)=O)CC1 24329,FC1(F)CCC1C1c2nnnn2CCN1.C(C1=NOCC1)N1CCOCC1 24330,C(=O)(C1CCc2c[nH]nc21)NC(C(NOCC)=O)c1ccccc1 24331,C(C)(CCC(=O)NC1CC1CNC(c1cnc(-c2ccccc2Cl)nc1)=O)OC 24332,C1(CNC(COCCN(C)C)=O)CC2(CCN(C(C3(CC(F)F)CC3)=O)CC2)CO1 24333,c1(C(c2n(CCC)nnn2)Nc2conc2C)c(F)ccc(Br)c1Cl 24334,C1(NC(CN(C)CCO)=O)CC2CN(C(=O)C(c3ccccc3)N(C)C)CC2C1 24335,C1(CC)CCN(C(C2CCCC2F)=O)C1CNC(c1ccnnc1O)=O 24336,c1(C(N2CC3(CN(C(c4c(C)coc4C)=O)C3)C2)=O)cc(N)c(O)c(F)c1 24337,C(=O)(C1=NOC(C)C1)NCC1(C)CC(NC(Cc2c(C)cco2)=O)C1 24338,C1(C(=O)NC(C)C(C)NC(c2cnoc2-c2ccoc2)=O)CCCC2(CC2)C1 24339,C=CC(CC)CC(=O)NCCOCCNC(=O)C=Cc1ccc(C)cc1 24340,n1(C(CC)C)ccc(=NC(=O)CC(CC(C)C)NC(C2C=CCCC2)=O)[nH]1 24341,N1(C(C(C)Cc2ccco2)=O)CCC(OC2(C(=O)NCCN(C)C)CC2)CC1 24342,N1(C(c2c(COC)cc[nH]2)=O)CC2CC(N(C(=O)Cc3ccns3)CC)CC(C2)C1 24343,N1(CCCNC(C(C)OC)=O)CCC(NC(=O)C(C)(F)F)C1 24344,C(=O)(C1CCCc2scnc21)NC1CN(C(c2n(C)c(O)nc2)=O)CC1O 24345,C(C)(CN=c1cc(COC)nc[nH]1)(C(C)C)NC(c1ccc(CC)cc1)=O 24346,C(C)(CSC)(C(=O)NC(c1cccnc1O)C)NC(C1CC(=C)C1)=O 24347,C1(C(N(CCC(=O)OC)C)=O)CCC(CNC(=O)CCc2nncn2C)O1 24348,C(=O)(C(CC)(CC)c1ccccc1)NC(CCCC)CNC(=O)CCN(C)CC 24349,C1(C(=O)NCCN(C(=O)CN(C)Cc2ccccc2)C(C)C)CN(C)CC(C)O1 24350,C1(CNS(CCSc2c(COCC)cccc2)(=O)=O)COC2(CCCCC2)O1 24351,Nc1cccc(C(N2CCN(C(c3ccnc(-n4cccn4)c3)=O)CC2)=O)c1O 24352,C(C(F)(C(=O)N(C1CCCC(C)C1)CC)C(C)C)NC(COCCC=C)=O 24353,N1(C(C2C(C)(C)C2(F)F)=O)CCC(NC(c2ccnc(N(C)C)c2)=O)C12CCC2 24354,N(C(=NCCF)NC(C)CCN1CCCCCC1)CC1(CC)COC1 24355,C#CCCCCCCCNC(=O)C(CC#C)NC(=O)CNC(=O)CC 24356,C12(C(N(CCCN(C(C(C3CCCC3)OCC)=O)C)C)=O)CC(C3CC3)(C1)C2 24357,C1(C(NOC(C(C)C)CO)=O)COC(=O)N1C.C1(=O)C(CO)N1 24358,C1(NC(=NCC=C)NCCS(=O)(=O)NC(C)(C)C)CC2(C1)CC(F)(F)C2 24359,N1(C(CCC(C)OCC)=O)CCC(C2CCCN(C(=O)C(=O)C(C)CC)C2)CC1 24360,C12(NC(c3ccc(C)cc3)=O)CC(CNC(=O)CC(O)C(C)C)(C1)OC2(C)C 24361,c1(C(C)NC(=O)NCC(c2scc(C)n2)C)ccc(Br)nc1C 24362,N1(C(c2n(CC)cnn2)=O)CCCCC(N=c2ccc(C(F)(F)F)n[nH]2)C1 24363,C1(NC(c2cnc(CC)[nH]2)=O)(CNC(c2cc3c(s2)CCC3)=O)CC2CCC1C2 24364,c1(C(=O)NCCC2N(C(C(N3CCOCC3)C)=O)CCC2)cc2ccccn2n1 24365,C1(C(=O)NCC(C2CCC2)OCC)CC(O)CN1C(c1ncccc1Cl)=O 24366,C(=O)(C(CO)C(C)(C)C)N1CC(CCNC(=O)Cn2ccc(O)nc2=O)(OC)C1 24367,N1(C(CCCC#C)=O)CCC(C(=O)NCC2(O)CCC(C)C2)C12CCC2 24368,c1(CC(=O)NCCC2CCCN2C(=O)CCc2cn[nH]c2)cn(C2CC2)cn1 24369,c1(C(=O)NCC2CN(C(c3cnc(C(C)(C)C)s3)=O)C3C2C3)cc(Cl)ccc1Cl 24370,N1(C(C(COC)OC)=O)CC(CNC(c2cccc(-n3cccc3)c2)=O)CC1C 24371,Cn1cc(C=CC(=O)NCCC2(NC(C3CC4C=CC3C4)=O)CCC2)nn1 24372,N1(C(c2cnc(C)c(N)c2)=O)CCC2(CCCC2CNC(C2(Cl)CC2)=O)CC1 24373,c1(C(=O)NCC2C(CNC(C(C)(C)OC(C)C)=O)C2)cn2c(n1)CCCC2 24374,Cc1c(F)ccc(-c2cn(C3CN(C(c4scnc4C(F)(F)F)=O)C3)nn2)c1Cl 24375,c1(OC)ccc2ccnc(C(C)NS(=O)(=O)CCCOCCOC)c2c1 24376,C(N=c1nc2c(ncn2C)c(NC2CC2c2c(Cl)cccc2Cl)[nH]1)c1c(C)nc[nH]1 24377,Fc1cc(Cc2nc(C3CCOCC3)nn2CC2CCCO2)ccc1Cl 24378,N1(C(c2ncc(CC3CC3)s2)C(=O)NCCOCC)CCOC(C2CCC2)C1 24379,C1(CNC(c2ccc(OCC)cc2)=O)CCC(C)CN1C(c1cnnc(O)c1)=O 24380,C1(CCNC(c2c(C)ocn2)=O)CCCN(C(C2CCCOCC2)=O)C1 24381,c1(CSC)cccc(C(N2CCC2CNC(=O)C(C(C)C)NS(C)(=O)=O)=O)c1 24382,C1(NC(C(c2cccnc2)C)=O)CC12CCN(C(C1CC(N=[N+]=[N-])C1)=O)C2 24383,C1(CC)(CC)CC(NC(C2CC2C2CC2)=O)CN1C(=O)CCCF 24384,C(C(=O)NC(C1CCCC1)CNC(=O)CC1CC1(Cl)Cl)(C(C)C)NC(C)=O 24385,c1(C(=O)NCCCC(C)NC(c2cncn2C)=O)cccc2c(O)nncc12 24386,N1(CC)CC(C(N2CCC2CNC(C2(c3ccsc3)CC2)=O)=O)CC1=O 24387,Cc1ccc(CO)cc1NC(=O)CC1CCCC1CNC(=O)CN1CSCC1=O 24388,N(C(=NCC(C)OC(C)(C)C)NCc1cccc(N2CCOCC2)c1)C1C(C)C1 24389,CCC(CC(=O)NC1CC=C(C(=O)NCCCC2CCC2)C1)C(F)F 24390,C1(C(N(C(CCC=C)C)C)=O)(NC(c2cccc(Cl)c2)=O)CCCCC1 24391,c1(C(N2CCC(NC(C(C=C)O)=O)C(O)C2)=O)c(C)cc(O)cc1C 24392,Cc1cc(C(N2CC3(NC(c4csc(CO)n4)=O)CCC2CC3)=O)cc(N)c1O 24393,C1(C(N2CC(NC(CCSCC(C)C)=O)C3(C2)CC3)=O)CCC2(CC1)CC(O)C2 24394,C(=O)(C1=NNC(=O)CC1)NC1C(NC(c2c(C)ccnc2O)=O)CCCC1 24395,CC1(C)CN(C(=O)C2=CCCCO2)CC1C(=O)NC1CC2C=CC1C2 24396,c1(OC)cccc(C(=O)NCC(C)CNC(c2cnc(CC(C)C)s2)=O)c1N 24397,c1(C(N2CC(C(=O)NC3C(CC=C)COC3)C(OC)C2)=O)cncc(C=C)c1 24398,C#Cc1ccc(C(=O)NC(C2CCCN2C(c2ccc(=O)n(O)c2)=O)(C)C)nc1 24399,C(=O)(CC(C)C(C)(C)C)NCC1N(C(C(CC(=O)OC(C)(C)C)O)=O)CCC1 24400,c1(NC(C2C(C(N(CC#C)C)=O)C2)=O)cc(Br)cc(F)c1OC 24401,c1(C(=O)NCC2C(CNC(C(C)SCC)=O)C2)c[nH]c2c(C)c(C)ccc2c1=O 24402,Cc1c(C(=O)NCC2(CNC(=O)C(C)CS(C)=O)CCC2)ccc2c1CCC2 24403,c12cccc(c1)CC(=O)N2.C(=O)(C1=CCCC1)N1CC(C)(OCC=C(C)C)C1 24404,c1(C(N(C2CC3CNC2C3)C(=O)CN2CCCC2)C)nc(OC)cc(OC)n1 24405,CC1COCCCN1C(C1CC(O)CN1C(=O)Cn1cnnc1)=O 24406,c1(C(=O)NC2CN(C(C(C)OCC)=O)CC2C2CC2)c(C)[nH]cc([N+](=O)[O-])c1=O 24407,N1(C(C2C(NC(=O)Cc3ccccc3[N+](=O)[O-])C2)=O)CCc2cc(O)ccc2C1 24408,C1(C(=O)OC)C(F)(F)C12CC(C(=O)NC13CC1CN(C(=O)C(F)(F)C(F)F)C3)C2 24409,c1(C(=O)NC2(CCCNC(C34C=CC(CC3)C4)=O)CC2)cccc2nsnc12 24410,Cc1n[nH]c(C)c1C(N1CCCC1CCC(=O)NCC1CCC1CO)=O 24411,CC1(C(=O)NCC2CCN(C(C3(F)CC3)=O)CC2)CCc2ccccc21 24412,N1(C(COC(C)=O)=O)CC=C(C(C)(C)C(=O)N(C)CC2OCCC2(C)C)C1 24413,C1(CNC(c2cn(C(F)(F)CO)nn2)=O)CCN(C(=O)Cc2ccoc2)CC1 24414,C1(C(=O)NCC2(c3ccccc3)OCCO2)Cc2ccncc2C1 24415,C(CC(C(=O)NCc1ccc(F)cc1)NC(C1CCS1(=O)=O)=O)=CC 24416,C12(NC(C3OCCC(C)C3)=O)CC(CNc3cc(CC4CC4)ncn3)(C1)OC2C 24417,Cc1ccnc(C(=O)NCc2ncc(C(=O)NC(C)Cn3cccn3)cn2)c1F 24418,c1(OC)cc(CN2CCC2C(=O)NCC2CCCC2)cc(F)c1OC 24419,c1(CNC(=N)NC(c2cccc(Cl)c2)C(F)F)ccccc1Br 24420,N1(C(C(CC2CCCC2)NC(c2nc(C)oc2C)=O)=O)CCCC12CCCOC2 24421,c1(N(C)CC)ncnc2c1ncn2CC(CSC)(CC)CC.c12ccc(o1)CN2 24422,c1(CCOC)cn(C(N2CC(CO)C2)=O)nn1 24423,CC1CC(c2nnnn2Cc2nnn(C)n2)(NCC2CC(C(F)(F)F)C2)CS1 24424,N1(C(C2CC(C)(CC)C2)=O)CC=C(CC(=O)N2CC(F)(F)CC2CO)CC1 24425,N1(C(C(c2ccccc2F)C)=O)CCN(C(=O)CC=C(Cl)Cl)C2(CC2)C1 24426,N1(C(CC2CCC(=O)C2)=O)CC2CCC1CN2C(C1C2C=CSC12)=O 24427,C1(C(=O)NC(CNC(c2nc(C)sc2)=O)(C)Cn2cccn2)CCC(O)CN1C 24428,Cc1nc2ccc(-c3cncnc3C(=O)NCc3nccnc3C)cc2[nH]1 24429,N1(CCC(N2CC(F)(C(=O)OCC)C3(C2)CCC3)=O)CCc2ccccc2C1 24430,C1(C(=O)OC(C)C(=O)Nc2cccc([N+](=O)[O-])c2)NCCC12CCCCC2 24431,Cc1csc2c(NC3CCC(NC(=O)CC4CCC(C(N)=O)O4)CC3)ncnc12 24432,c1(C(CNC(c2ccnc(C)n2)=O)NC(C2CCCN2C)=O)cc(F)cc(Cl)c1 24433,c1(OC)ccc(C(N2CCCC2CNC(=O)Cc2cccnc2C)=O)cc1O 24434,C(=O)(CC(C)(C)C(F)F)N(C1CCN(C(c2cnn(C3CCC3)c2)=O)C1)C 24435,C(CC(CC)C(=O)N1CCCC(NC(C2CCC(N(C)C)CC2)=O)C1)=CC 24436,N=c1[nH]n(CC(=O)NCCNC(C2CCCCC2O)=O)cc1Br 24437,c1(C(N2CCC(NC(C)=O)C2)C(=O)NC(C)(C)C)c(C)nc2sc(C)nn12 24438,C1(NC(c2sc(C)c(O)n2)=O)CCCC2CN(C(=O)C=Cc3cccs3)CC12 24439,C1(c2ccccc2)(CNC(=O)NC(c2ccc[nH]2)C2CC2)CCCO1 24440,c1(C(=O)NCCC2CC(NC(c3cncc(CO)c3)=O)C2)cnc2n1CCS2 24441,CC(C)C(C(=O)N1CCCC(C(=O)N(CCC(=O)O)CCO)C1)c1ccncc1 24442,CC1COc2c(C(=O)NC3CN(C(c4ccc5c(c4)nnn5C)=O)C3)cnn2C1 24443,Cc1cc(C(=O)NCCNCC2CC3CCCC3C2)cn(C)c1=O 24444,n1(CC)nc(C)cc1C(=O)NCc1ocnc1C(=O)N(C12CC(C1)C2)C 24445,c1(CCC(=O)NC2CCN(C(=O)C=C(Cl)Cl)C2C(F)(F)F)cncc(F)c1 24446,Cc1ccc(-c2ocnc2C(=O)Nc2cncs2)s1 24447,C1(C(N(CC(CNC(CCOCC#C)=O)C)C)=O)COCCN1C 24448,CN=c1[nH]ccc(C(N2CCC(C)(C)C2CNC(C2CCC(C)CC2)=O)=O)c1N 24449,c1ccc(C(=O)N(C)CC=CC(=O)NCCN2CC(COC)C2)s1.CC=C 24450,CCCCC(CNC(=O)Cn1cc(CO)nn1)NC(C1CCN1C1CCCC1)=O 24451,C#CC1CCCC(c2nnnn2C2CCCC2)(NC2(C)CCC(C)=C(C)C2)C1 24452,c1(C(=O)NCCCN(C(C2C(C)C2(F)F)=O)C2CC2)cccc(C2CCCC2)c1 24453,c1(C(=O)OC)cnc2nncn2c1C.N1(C(C23CC(O)(C2)C3)=O)CCC(Cl)=C(Cl)C1 24454,N1(C(C2CCCC(OC)C2)=O)CC2(CCN(C(=O)C(C)NC=O)C2)C1 24455,N1(C(C(COC)(F)F)=O)CCCCC2(CCN(C(c3cnc(N(C)C)s3)=O)C2)C1 24456,c1(CC)ccc(C(=O)NCCC2CCN(C(=O)CCCC#N)C2)cc1Br 24457,C1(C(=O)NC2CC(CC)(CC)C2)CN(C(=O)CC(C)SC)CC1N=[N+]=[N-] 24458,c1(NC(c2cn(C3CCCCC3)nn2)=O)ccc2c(O)ncnc2c1 24459,C(=O)(C(C)C(F)(F)C(F)F)NC1(CCCNC(c2cc(CC)c(F)cc2)=O)CC1 24460,Cn1c(C(=O)NCC2CCCC(NC(=O)C=C3CCC3)C2)cc2ccsc12 24461,c1(C(=O)NC2CCCN(C(c3n(CC#C)ccc3)=O)C2)cc2n(c1)CCC2 24462,n1(CC(=O)NCCCNC(CC2CCCC(C)(C)C2)=O)sc2ccccc2c1=O 24463,CC1CN(C)CC1NC(C1CCN(C(c2ccoc2Cl)=O)C1C)=O 24464,c1(C(N2C(C(C)=O)C(C)(C)C2)=O)ccc2nnn(C(C)(C)C)c2c1 24465,CC1CCNC(=O)C1NC(C1CCC(CNC(=O)C=Cc2ccco2)O1)=O 24466,C(CC)(CCCC(=O)NCc1ccc(O)cc1)NC(C1(OCC)CCCC1)=O 24467,CCCCC(CO)NC(=O)CC1CC(NC(=O)CN2CCNC(=O)C2)C1(C)C 24468,C1(C(=O)NCCCN(CC)CC)(NC(=O)CCN(C)C)CCOC1 24469,Cc1cc(Cl)c(C(=O)NCC2(C)CCCN2C(=O)CSCc2ccncc2)cn1 24470,c1(CC(C)NC(C(N2CC(CC)C(C(F)(F)F)C2)=O)=O)cc(CC)ncn1 24471,c1(NCCSC(C)C)[nH]c(=NCC(c2ccccc2)N(C)C)nc2c1ncn2C 24472,CC1CCCC(N=c2nc(N3CC4C=CCC(C4)C3)c3c([nH]2)CCC3)C1 24473,C1(COC)(NC(c2cocc2C)=O)CCN(C(=O)C(C#N)C(C)C)CC1 24474,c1(C(=O)NC(CC(C)NC(CCOCC(C)C)=O)C)ccc(F)cn1 24475,c1(CNC(CC2C(CC)C2)=O)csc(C(=O)Nc2ccsc2CC)c1 24476,CCC(C)C(C(=O)NC(C)CCSC)N(C)C(c1cccc(C)c1C)=O 24477,C1(C(N2C(CNC(=O)CN3CSCC3=O)CCCC2)=O)CCC=CCCC1 24478,N1(C(c2cccc(CC)c2)C(=O)NC)Cc2nccn2CC(C(=O)OC)C1 24479,C(=O)(CCC(CF)CF)N1CC(CC(C(=O)NCCC2CC(O)C2)F)C1 24480,C1(NC(c2c(C)scc2)=O)CN(C(C2CCC2C(C)(C)C)=O)C2(CCC2)C1 24481,C(CS(=O)(=O)CC(=O)NC(C)(C)CC(F)C(=O)NCc1nnnn1C)OC 24482,C1(C(=O)NC2COCC2F)(COC)CCCNCC1 24483,c1(CC(=O)NC2(C(=O)OC)CCC2COC)ccc(OC(C)C)cc1Cl 24484,Cc1c[nH]c(C#N)nc1=NCC1CCCN(C(=O)C2=CC3(CCOC3)C2)CC1 24485,Cc1ncc2n1CCC(C(=O)NC(C)CNC(=O)CCc1ccc(CO)cc1)C2 24486,C1(C(N2C(C(=O)NCCC(C)(C)C)CSCC2)=O)CC1C1(C)COC1 24487,c1(C(C(=O)NC(C)CN(C(=O)CSC(=N)N)C)C)cccc(O)c1 24488,C(C(CC(C)C)C(=O)N(C)Cc1ccncc1)NC(C(CCC)CC)=O 24489,Cc1cccc(C(O)C(=O)NCC2(CNC(C3(N(C)C)CC3)=O)CCCC2)c1F 24490,N1(C(c2cc(C3(C)CC3)n[nH]2)=O)CCC2(CCC2NC(c2ccoc2Cl)=O)CC1 24491,c1(CCCC(=O)NC(CNC(C2CCOC2)=O)C2CCC2)ccccc1Cl 24492,C(=O)(C1=C(F)CN(C(=O)CN2CCC(OC)C2)CC1)N1CC(CCC)OCC1 24493,C(=O)(CC(C)(C)C1CCCCC1)NCC(CCOC)NC(=O)C(F)OC 24494,C1(C(=O)NC(c2ccc(C(F)(F)F)cc2)CO)CC(c2c(F)cccc2F)=NO1 24495,N1(C(CC(C(C)C)NC(CC(=O)OCC)=O)=O)CCn2ccnc2C1C 24496,c1(C(=O)NCC(C2CC2)NC(CC2C(C)(C)C2)=O)cocc1Br 24497,N1(C(c2ccc(C)cc2)=O)CCC(NC(C2CCC(CO)CC2)=O)C(F)C1 24498,C=CC1(CC(=O)NCC(C2CCN(C(C3CCC(=O)O3)=O)CC2)F)CCCCC1 24499,n1(C(C=C)C)nc(-c2ccoc2)nc1-c1cccc(-c2ccncc2)n1 24500,C(=O)(C(F)C(C)CNC(c1ccc(F)c(O)c1)=O)N1C(COC)C=CC1 24501,C(=O)(C(C)(C)C(=O)Nc1cc(F)cc(F)c1)NCC1(O)CCN(C(C=CC)=O)C1 24502,Cc1ccc(F)cc1C(N1CC2CC1C2NC(=O)CC1(O)CCCCCC1)=O 24503,C(=O)(C(C(C)(C)C)NC(C1CC(=O)N(OC)C1)=O)NC(COC(C)=O)CO 24504,Cc1c(Br)cnn1CC(=O)NCCC(C)N(C(=O)C=C1CCOCC1)C 24505,CC(C)CS(=O)(=O)CCC(=O)NCC(C)CN(C(=O)CP(C)(C)=O)C 24506,CC1(C)CC(CC(N2CC(CC(F)F)C2)=O)N(CCNC(=O)CO)C1 24507,C1(C(=O)NC(C)COCC2CC2)CC(F)(F)CN1C(=O)CCC1CC1 24508,CCCCCC(CC)C(=O)NCC1CN(C(=O)CCCOC(C)C)C2(CCC2)C1 24509,c1(N2CCN(C(c3cc(Cl)nnc3O)=O)CC2)ncc([N+](=O)[O-])cn1 24510,N1(C(=O)CC2C=CC(NC(C3(C(N)=O)CC3)=O)C2)CC=CC12CCCCC2 24511,N1(C(c2cc(F)cc(C)c2N)=O)CCOC2(C1)CN(C(=O)OC(C)(C)C)C2 24512,Cc1cc(CCC(N2CCOC(CN(C(=O)C(C3CC3)C3CC3)C)C2)=O)nn1C 24513,N1(CC(=O)N(C)CCn2cccn2)CCCC(NC(c2coc(C3CC3)c2)=O)C1 24514,N1(C(=O)Nc2nc3ncc(C(=O)OC)cc3o2)Cc2ccc(F)cc2CC1C 24515,C1(C(=O)NCCN(C(C(CC=C)C(C)C)=O)C)CCOC2(CCOCC2)C1 24516,c1(C(=O)NC2CC(CNC(Cc3nnc(C)n3C)=O)CC2O)c(C)ncnc1O 24517,c1(C(C)=O)ccc(S(=O)(=O)N2CC(O)CC2C(=O)Nc2ccc(F)cc2O)cc1 24518,C1(NS(CC=C)(=O)=O)CC2(C1)CN(C(c1cc(I)ccc1O)=O)C2 24519,C1(CC(=O)NCCCC(C)NC(Cc2cccc(OC)c2)=O)CCCC(C#N)C1 24520,CC1(C)CN(C(=O)CCn2ccnc2)CC(C)(C)C1NC(c1ccc[nH]1)=O 24521,C1(NC(=O)CN2CCOCC2)CCN(C(=O)CCc2cn[nH]c2)CC1F 24522,C(=O)(CC(O)CC(C)C)N1C(CCC)CN(C(=O)CCC(C)(F)F)CC1 24523,c1(OC)cc(F)c(C(N2CCC3(C2)CN(C(C2C=CCCC2)=O)C3)=O)cc1F 24524,C1(c2c(C)cco2)NC(=S)N(Cc2ccco2)C2=C1C(=O)NC2C 24525,C(C(=O)N1OC2CCC1CC2)N(C)CCNC(=O)C(F)C1CCCC1 24526,C1(N2C(c3nc(C)nc(=N)[nH]3)CCC2)CCC2(CC1)OCCO2 24527,C(C)(CCCNC(=O)C(C)Sc1nncn1C)NC(C1(CCC=C)CC1)=O 24528,c1(NCc2c(OCC)cccc2)ccc(NC(c2ccccc2OC)=O)cc1F 24529,Cc1ccc(C(F)(F)C(N2CC(NC(c3cnc(C)o3)=O)C(C)C2)=O)cc1 24530,C1(CNC(c2c(CC)nc(C)o2)=O)CN(C(=O)C(CCSC)OC)C2(CCC2)C1 24531,C=C=C(C)CC(=O)N1CCC(O)(C(C)NC(=O)Cc2c(C)n[nH]c2C)C1 24532,CCCC(C)CC(=O)N1CC(NC(=O)CCCc2ccccc2)C(O)C1 24533,N1(C(c2cccc(CC)c2)=O)CCN2C(=O)C(NC(=O)Cc3cncs3)CC2C1 24534,c1(C(N(CC(N2CC=C(COC)CC2)=O)CC)=O)ccc(=O)oc1 24535,N1(Cc2nccc(C(=O)OC)c2)CCC(NC(=O)Cn2cc(Cl)cn2)C(C)(C)C1 24536,C(=O)(C(O)C(C)CC)NCC1(CCNC(CNS(CCCC)(=O)=O)=O)CC1 24537,N1(C(C(C2CCOC2)NC(C2CCC3(CC3)C2)=O)=O)CC2CC2C2CC12 24538,c1(NC(CCS(CC)=O)=O)sc2c(c1C(=O)Nc1ccc(C#N)nc1)CCCC2 24539,c1(OC2(C(=O)NCC(c3cccc(F)c3)C)CC2)ccc(Cl)cc1 24540,N1(C(=O)CCC2CCCN2Cc2cncc(Cl)c2)CCc2c(Cl)ccc(Br)c2C1 24541,N#Cc1c(N2CCC(F)(CNC(C34CC=CCN3CCC4)=O)CC2)cccc1F 24542,c1(C(N2CCC(O)(CCNC(C(C)C)=O)C2)=O)nc(N(C)C)nc(=N)[nH]1 24543,Fc1cc(Cl)cnc1-c1nnc(N2CC3CN(CC(F)(F)F)C3C2)n1C 24544,C(=O)(C(C)(CNC(=O)CCc1nc(O)n[nH]1)CC)NCC(N(OCC)C)=O 24545,C(=O)(C(C)C(C)CC)N(CC(CNC(c1nc(C(=O)NCC=C)sc1)=O)(C)C)C 24546,c1(C(=O)NCC2OCCCN(C(COCCC#C)=O)C2)cccc2nc(O)[nH]c12 24547,N1(C(CC(=O)NC)=O)CCC2(CC1)CCN(C(c1ccc(CC(C)C)cc1)=O)C2 24548,c1(C(=O)NC23CCN(C(=O)CCc4nc(O)n[nH]4)CC2C3)ccc2ccsc2c1 24549,N1(C(CCCOC)=O)CC2CCCC(N(C(=O)CC3CCCC34CC4)C)C2C1 24550,CC#CCCCC(=O)NCCOCCCNC(=O)C(c1ccn(C)n1)C 24551,C(=O)(C(CCC(C)C)NC(c1ccnn1CCC)=O)NC(C=C)C1CCC1 24552,CCC(O)C(C)C(=O)N1CCCC1CN(C)C(C1CN(C2CCOC2)C1)=O 24553,c1(OC)ccc2nc(N3CC(CO)(NC(c4c[nH]nc4C4CC4)=O)C3)sc2c1 24554,N1(C(c2c(SC)cn(C)n2)=O)CC(C)(CNC(=O)C(F)(F)C2CC2)CC1(C)C 24555,N1(C(C2=CC(C)(C)C2)=O)CC2(C1)CN(C(c1cccc(=O)n1O)=O)CC2CO 24556,CCC(C)(CO)C(=O)NC1CC(CNC(=O)C(C(C)C)n2cnc(C)c2)C1 24557,C1(NC(CCN(C(=O)COc2ccncc2)CC#C)=O)CCC(C(C)O)CC1 24558,c1(OC)cccnc1C(=O)N(C(CNC(=O)CCSc1nnnn1C)C1CC1)C 24559,N1(C(C2N(C)CCOC2)=O)C(CC(N2CC3C(C(N)=O)C3C2)=O)C2CCCC12 24560,C(C(C)(O)CC)NC(C(N(C(C1C(=C)C1C(=O)OC)=O)C)C1CC1)=O 24561,CC1CC(NC(=O)CC2CC(O)C23CCC3)CCN1C(c1ccc(N)c(O)c1)=O 24562,C(=O)(C(C)(C)C(C)(C)C)NCC1(C(=O)NCc2cccc(C)c2O)CC1 24563,Cc1ncnc(C)c1CC(N1CCC(F)C(NC(C2CCC3CC2CO3)=O)C1)=O 24564,C1(C(=O)NCCC(C)(C)N(C)C)(CF)CCN(C(=O)CN2CC=CC2)C1 24565,N1(C(C2C(C)CCN2C(=O)CCC(N)=O)=O)CC2(CCCCCC2)C1 24566,c1(C(N2CC(CCCCNC(CC(C=C)CC)=O)C2)=O)[nH]nc2c1COC2(C)C 24567,c1(-c2c(C)ccs2)ccc2c(c1NC(=O)Cn1cc(Br)cn1)OCO2 24568,C1(NC(C=CC(C)(C)SC)=O)CC2CC(C1)CN(C(=O)Cc1ccc(O)cc1)C2 24569,N1(C(C2(CNC(=O)Cn3cccc3)CCCCC2)=O)CC2CCCC(C2)C1 24570,CCC(F)(F)C(=O)N1CCOC(CCNC(c2cnnn2C2CCOCC2)=O)C1 24571,N1(C(C(C)CN)=O)CCOC2(CCCN(C(c3cc(Cl)c(Cl)c(Cl)c3)=O)C2)C1 24572,c1(OC(C)C(=O)NC2(CCNC(=O)CCC3(C)CC3(F)F)CCC2)cccnc1 24573,N12CCC(OC(C)C)(C1)C2=O.C1(=O)C(C(=O)C(C)=O)NCCN1.C(C)(C)(C)N 24574,Cc1ccccc1C(C)C(N1CCC(CN(c2nccs2)C)CC1)=O 24575,c1(C(N2CC(OC)C(NC(=O)CCC3CCOCC3)C2)=O)ncc(N)cc1C 24576,N1(C(C=C(C)Cl)=O)CC(CNC(C23CCC(C)(CC2)CO3)=O)CC12CCOCC2 24577,CCC(CCC(=O)NC1CC1CNC(C1CC1C1CCCC1)=O)OC 24578,C1(C(N2CC(OC)(CNC(=O)C(C)(C)c3ccccn3)C2)=O)CC1C1CCCC1 24579,C(CCC(=O)N1CC2(CC2)CC1CO)(C(C)C)NC(Cc1cncc(C)c1)=O 24580,c1(C(=O)NCC(CC)(CC)NC(=O)C(O)CN(C)C)nc2n(c1Cl)CCCC2 24581,N1(CC(=O)NCC(C(=O)NC2CC2F)OC)CCC(=O)CC1 24582,CC1CC(CNC(c2ccn(C3CCC3)n2)=O)CN1C(c1cncc(F)c1)=O 24583,c1(C(N2CCC(N(C(=O)CC3CCOC3)CCC)C2)=O)cccc2c1OCCO2 24584,c1(CN(C(=O)Cc2ccnn2C2CCOCC2)C)cccc2c1OC(F)(F)O2 24585,N1(C(c2c(CC)c[nH]n2)=O)CC2CCCN(C(=O)C(C)O)C2C1 24586,N1(C(CN(C)C)=O)CCn2ncc(C(=O)NCc3ccc4cc[nH]c4n3)c2C1 24587,C1(NC(CC2CC(NC(c3cn(C)nn3)=O)C2)=O)CC2CCCC(C1)C2 24588,c1(C(C(=O)NCC(C)NC(C2CC2[N+](=O)[O-])=O)C)cncc(F)c1 24589,Cc1cc(C(=O)NC(c2ccccc2)C(C)NC(=O)CCC2CC2)nc(O)n1 24590,N1(C(C2(NC(C3CCC(C)O3)=O)CCCC2)=O)CC2(CCCC2)C1 24591,N1(C(C(CC)OC)=O)CCCC(F)(C(=O)Nc2cn(C)nc2C#N)C1 24592,C1(C(=O)N(CC)Cc2ccc(C)o2)(OCC)CCN(C(C)CO)CC1 24593,N1(C(C(C)c2ccco2)=O)CCCN(C(c2ccc(Br)s2)=O)CC1CO 24594,C1(NC(=O)C=Cc2cnc[nH]2)CC2CC(NC(=O)CCc3cc[nH]n3)CC2C1 24595,Cc1cc(C(=O)NCCC2(C)CCN(C(c3nnn(C)c3N)=O)CC2)ncc1Cl 24596,C(C1CCN(C(C2CCCC(=O)N2C)=O)CC1)=CC(=O)NCc1c(CC)nccn1 24597,C1(N(C)C)CCC(N=c2ccnc(NCc3ccc(C#N)cc3)[nH]2)CC1 24598,Cc1nc(-c2ccn(C)n2)sc1CC(N1CC(NC(=O)C(C)C(C)C)C1)=O 24599,c1(C(=O)NC(C)CNC(=O)C2=CCCCC2)cc2c(Br)cc(F)cc2[nH]1 24600,c1(C(=O)NC2(CNC(Cc3cc(C)on3)=O)CCC2)cc2c(C)cc(F)cc2[nH]1 24601,N1(CC)CCOC(C(N2CCOC(CNC(=O)CC(F)(F)Br)C2)=O)C1 24602,CCN=C(NCC(CO)C(C)(C)C)N1CCC(COc2cccc(C)n2)CC1 24603,C(=O)(CC(C(F)F)NC(c1c(O)noc1C)=O)Nc1ccc(OC)nc1 24604,Cc1oc(C)c(C(=O)NCCC(O)CNC(c2cnn(C(C)(C)C)c2C)=O)c1C 24605,Cc1ccc(F)c(CC(C)NC(c2cccc3[nH]ncc23)=O)c1F 24606,N1(C(C2CC(N(C)C)C2)=O)CCC(NC(C2CCC(F)(F)CC2)=O)C(O)C1 24607,N1(C(CN(CCC)C)=O)CC(C(=O)NCc2ccnc(Cl)c2)C2(CCC2)C1 24608,C1(CCCC(=O)NC2(CCNC(=O)CSc3nc[nH]n3)CC2)CCCC(=O)N1 24609,C(C)(C)(CCC(=O)NCc1ccoc1)NC(C(CC)NC(N)=O)=O 24610,Cc1nccc(C(=O)NCCOC2CCN(C(C3CCC(C)NC3=O)=O)C2)c1C 24611,c1(C(=O)NCC2C(C)CN(C(c3cccc(C(N)=O)c3)=O)C2)c(F)ccnc1F 24612,N1(C(C(CC)NC(c2cnnn2C)=O)=O)CCOC(C)CC1 24613,C1(CNC(CSCC)=O)CCC(C)CN1C(c1ccnn1CC(C)C)=O 24614,C1(c2c(CC)n[nH]c2)CCCN(C(c2ccc(C(n3ccnc3)=O)cc2)=O)C1 24615,C1(NC(=O)C(O)C2CCCC2)CC2CN(C(c3occc3C3CC3)=O)CC2C1 24616,C(C)(C(C(=O)NCCCc1nncs1)C(C)C)NC(c1nc(CCC)oc1)=O 24617,c1(C(=O)NCC(CC)NC(=O)C(Cc2ccccc2)n2cnnn2)cscc1C 24618,C(C1CC(=O)Nc2ccccc21)NC(=NCC)NC1CCS(=O)(=O)C1 24619,Cc1ccc(-c2nc(CC3CCCCC3C)n(C3CCC3)n2)cc1Br 24620,C12(C(N(CC(CN(C(=O)C(=O)Cc3ccccc3)C)O)C)=O)CCOC(C)(C1)C2 24621,Cc1c(COCCC#N)ncnc1N(CCCN(C)C(C)C)C.c1(O)ccc(F)cc1 24622,N1(C(CC=C=C)=O)Cc2ccnn2CC(NC(=O)C(C)CCOC)C1 24623,C(=O)(C(C)(C(F)(F)F)c1ccccc1)N(C)CCNC(C1CCCCC1O)=O 24624,N1(C(CC=CC(C)(C)C)=O)Cc2ccccc2C(NC(=O)CC2CCC2(F)F)C1 24625,CC(C)C(C)(C)C(=O)NCC(CC1CCCC1)C(=O)N(C1CCCN(C)C1)C 24626,c1(C(=O)NC2(c3cn(C(CC=C)CC)nn3)CCC2)ccc2occc2c1 24627,c1(N2CC(CC(C)C)OCC2)nc(=NCC2(CC#N)CC2)[nH]c2ccc(Cl)cc12 24628,N1(C(C(C(C)C)NC(=O)OC)=O)CCCC(O)(CNC(C2SCCS2)=O)CC1 24629,C1(C(C)NC(C2(CC)CCC2)=O)CCCN(C(=O)CN2CCCC2=O)C1 24630,Cc1occc1C(=O)NC1CC(C)(NC(c2ccon2)=O)C1 24631,CC1(C)CN(C2CC(n3cncn3)C2)C1c1nccn1Cc1ccccc1Cl 24632,C1(CCN(C(CC(C)F)=O)C)CCN(C(=O)CC2CCC23CCC3)CC1 24633,c1(NC(C2N(C(c3cnc(C)nc3C)=O)C3C(C2)C3)=O)ccc(O)c([N+](=O)[O-])c1 24634,c1(C(=O)NCCC(C)NC(c2cc[nH]n2)=O)cc2c(s1)CCCNC2=O 24635,c1(C(N(C(C)CNC(=O)C(C)(O)CC)CC)=O)ccnc(CO)c1 24636,c1(NC(C)C)ccc(C(=O)N(C)CC2CCCN2C(c2ncc(Cl)n2C)=O)cc1 24637,c1(CNC(=O)NCC(c2ccccc2)C2CCC2)cc2c(s1)CCCC2 24638,C1(F)(c2cn(CCC(C)C)nn2)CCN(C(C2CC3(CC3)CO2)=O)C1 24639,C1(C(N2CC(SCC)C2)=O)C(NC(=O)COCC2CCCO2)C1(C)C 24640,N(C(=NCCC(C)=O)NCC(=O)NC)C1CCCC(C#C)(O)C1 24641,Cc1cn2c(n1)CC(C(=O)NCC1CC13CCN(C(c1nncs1)=O)CC3)C2 24642,C(=O)(CCCC(F)(F)F)NC1CN(C(C2C(C)(C)C(F)(F)C2)=O)CC12CC2 24643,c1(N(C(C2CCC2)=O)CC2(CCC=C)CC2)nnn(C)c1N 24644,N1(C(c2cnc(SC)s2)=O)CCOCC1CCNC(=O)C=Cc1cnc[nH]1 24645,C1(C(N2CCCCC2CNC(=O)C(C)NC(=O)NC(C)C)=O)(CC)CCCCC1 24646,N1(C(C=CC)=O)CC2CC1CN2C(=O)CC1NC(=O)CNC1=O 24647,Cn1cc2c(n1)C(O)CC1(CCN(C(N3CCC4(CCC4(CCOC)C)C3)=O)CC1)O2 24648,c1(C(=O)NC2CCCN(C(C3C(C)C3)=O)C2)ccc2c(c1)CC2 24649,c1(C(N2CCC(COC)(NC(=O)C(C)SC(C)C)C2)=O)ccc2c(c1)NC(=O)C2 24650,C1(NC(C(C)NC(CC)=O)=O)CC2(C1)CN(C(c1cc3ccsc3s1)=O)C2 24651,C1(CC(C(=O)NCCOC)N2CCCC2CCNC(C)=O)CCC(C)(C)CC1 24652,N1(C(CC(COC)C)=O)CCCC2CN(C(c3ncc(C)cc3C)=O)CCC12 24653,N1(C(c2cc(C(=O)OC)oc2C)=O)CCCC2(CCN(C(=O)C(F)C(C)C)C2)C1 24654,c1(CC)cccc(C(=O)NC(C2CCN(C(=O)CS(=O)(=O)N(C)C)C2)C)c1O 24655,N1(C(Cc2c(C)cco2)=O)CCCC12CCN(C(C1(CC(F)(F)F)CC1)=O)C2 24656,c1(CC(=O)NCCN(C(c2cnn(-c3ccccn3)c2)=O)CC)ncncc1Cl 24657,N1(CC)CCC(N(C(=O)C=CC(c2ccc(Cl)cc2)=O)C)C(C)C1 24658,C1(C(N2CC(OCC)(CNC(=O)CCS(C)=O)C2)=O)CCCCC1(F)F 24659,c1(-c2cn(C3CC(NC(=O)Cn4cccnc4=O)C3)nn2)cccc(Cl)c1Cl 24660,C#CCCC(O)C(=O)N(C1CCN(C(=O)COc2ccsc2)C1)CCC 24661,N1(C(CC(CC)OC)=O)CCCN(C(=O)C(COC)C(F)(F)F)CC1C 24662,N1(C(CC(C)(F)F)=O)CC2CC(NC(c3ccnc(-n4cccc4)c3)=O)CC1C2 24663,C1(NC(C(C)=C2CC2)=O)CC2(C1)CN(C(C1(C(C)C)CC1)=O)C2 24664,CC(C)CC(C)C(=O)NC1(C)CC(NC(=O)C(N2CCC(C(=O)NC)CC2)=O)C1 24665,C1(C)(C(=O)NC(CC)CN(C(c2ccc(SCC(C)C)o2)=O)CC)CCNC1=O 24666,N1(C(C2C(CC)CCO2)=O)CCN(C(c2c(C)cc(C)nc2S)=O)CC(O)C1 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24684,N12CCC(C)(CC1)NC2=O.c12nocc1C2C.n1(C2(C(=O)NF)CC2)ccnn1 24685,C12(C(N3C(C)(CC)CC3)=O)CC(C)(CN1C(=O)CCCn1cccc1)C2 24686,CC(F)(F)CCC(=O)NN1CCCC1C(=O)NCC1(CO)CCOCC1 24687,c1(C(=O)NCC2(NC(C=CC(C)(C)C)=O)CCCC2)cc(O)c2ccccc2c1 24688,C1(C(=O)NC2CCC(OC)C2)CCN(C(=O)CCc2cnco2)C1C 24689,C1(C(=O)NCCNS(CC)(=O)=O)C=CCN(C(C2(OC)CCOCC2)=O)C1 24690,C1(C(=O)NCC(C)N(C2CCN(CC(F)(F)F)C2=O)C)CC(=O)N(C)C1 24691,O=S(=O)(c1cccc(F)c1)NC(c1ccc(NCc2cccc(CO)n2)cc1)=O 24692,c1(OCC)ccc(C(=O)NC2CCC2NC(=O)CC(n2nc(C)cc2C)C)nc1 24693,CC1CCC(C)N(c2nnc(-c3ccc(CCn4ccnn4)cc3)n2CCN)C1 24694,c1(C(N2CCN(C(C3C(C)(C)C3)=O)C3(C2)CC3)=O)c[nH]c2nc(F)ccc12 24695,c1(C(=O)NC2CCN(C(c3cccc4nccn34)=O)C2)ccc2c(c1)COCO2 24696,C1(C(=O)NC(CN(C(CS(=O)(=O)NC)=O)C)C)CCCC(=O)N1C 24697,C12(c3ccc(C)cc3)CN(C(=O)N(C)CCF)CC(CO)(C1)C2 24698,Cc1c(-c2cccnc2C(N2CCCC3CCCCC23)=O)cccc1S(C)(=O)=O 24699,N1(C(C#CC)=O)CCC(CN(C(=O)CC(c2ccc(C(C)C)cc2)C)C)CC1 24700,C(C(=O)NCC1CC(C)N(C(=O)CCn2cnnn2)C1)(C(C)C)OCC 24701,Cc1ccc(C(=O)NC2(C)CCN(C(C3(C)CCN(C)C3)=O)CC2)c(C)c1 24702,c1(C(=O)NCC(CCC)NC(c2cnn3c2OCC3)=O)ccn2nccc2c1 24703,C(CCC(CO)NC(c1cn(C)nc1C1CC1)=O)NC(Cc1ccn(C)n1)=O 24704,c1(OC)ccccc1C(N1CC2CC1C2NC(c1cnn(C2CCC2)c1)=O)=O 24705,c1(C(N(CCCNC(C2CC3(CC3)CO2)=O)CC)=O)cc(Cl)c(N)cc1F 24706,n1(CCC(N2CC(C(N(CC#N)CC#N)=O)C(O)CC2)=O)ccc2ccccc12 24707,N1(C(C2(C)CC2)=O)CC2(CC(NC(=O)C(c3ccc(Br)cc3)(C)C)C2)C1 24708,N1(C(c2ccoc2)=O)CCCCC1C1CCCN(Cc2nc(C(F)F)no2)C1 24709,C1(C2CCN(C)CC2)(C(=O)NC2C(OC)CN(C(C3CCCC3(F)F)=O)C2)CC1 24710,C(=O)(C(C)N(OC)C(=O)CCCCCN(C)C(C1CCCC(F)C1)=O)OC 24711,CC(C)CCN=C(NCc1cccc(Cl)c1Cl)N1CCC(OC2CCCC2)CC1 24712,CCS(=O)(=O)C=CC(=O)N1CCC(CCNC(c2cncc(N)c2)=O)C1 24713,N1(C=O)CCn2nc(C)c(Br)c2C1.c1(NC(NCNCC)=S)coc(C)c1 24714,c1(C(N(CCOC)CCNC(C2CC3CCC2C3)=O)=O)cc(F)c(F)cc1Cl 24715,c1(C(=O)NC2CC(NC(C3C(COC)(COC)C3)=O)C2)cc(C)nnc1O 24716,N(C(=NCc1ccco1)NCC1(O)CCSC1)CC(C1CCCCC1)(C)C 24717,C#CC(CNC(=O)CC1(N(C)C(C23CCC(C2)C3)=O)CC1)CC(C)(C)C 24718,N1(C(C2N(CCC)CCC2)=O)CCN(C(c2cccc(C3CC3)c2)=O)C2CCC12 24719,N1(C(C(c2c(C)noc2C)C)=O)CCCC2CN(C(c3nonc3N)=O)CCC12 24720,c1(NC)cnncc1C(N1CCC(O)(CN(C)C(C2CC=CCC2C)=O)C1)=O 24721,c1(N2CCCC(CC=CC)C2)nc(N2CCC(O)CC2)nc2c1CCCC2 24722,N1(C(C2CN(C)C2)=O)CCC12CCCN(C(c1ccnc(OC(C)(C)C)c1)=O)C2 24723,N1(C(C(C=C=C)C)=O)CC2COCCC2(NC(c2ccc([N+](=O)[O-])[nH]2)=O)C1 24724,N1(C(c2cnc(O)nc2O)=O)CC(C2CCCN(C(C3CC34CCCC4)=O)C2)C1 24725,N1(C(C(C)OCCC=C)=O)CCCCCC1C(=O)NCC1(OC)CC1 24726,c1(C(N2C(COC(=O)NC)CCC2)=O)cc(Br)ccc1O 24727,CCC(CO)C(=O)NCCCCCn1cc(COCCN(C)C)nn1 24728,C(=O)(CCCCC(=O)N(C)CC1(CNC(c2cnc(N)cn2)=O)CC1)NC 24729,Cn1cc(N)c(C(=O)N(C2CCN(C(c3ccc(Cl)s3)=O)C2)CCO)n1 24730,S(=O)(=O)(c1ccnc(NC(c2cncc(CN)c2)=O)c1)NC 24731,c1(C(=O)NC2(CC=C)CN(C(=O)C(c3nc(C)cs3)C)C2)cc2ccccn2c1 24732,c1(CC(=O)N(CCC(C)NC(C2CC2C(c2ccccc2)=O)=O)C)ccccc1 24733,C1(CC(=O)NCCC2CN(C(CCc3n(C)cnc3)=O)C2)CCC=CCC1 24734,Cc1ccc(F)c(OCC(=O)N(CC(C)N(C)C(c2ncn3c2CCC3)=O)C)c1 24735,C1(C#N)(C(=O)NCC(C(C)(C)C)NC(c2cnn(C(F)F)c2)=O)CC2CC2C1 24736,n1(CC(N2CC(N(C)CC)C2)=O)cc(CNC(=O)C(C2CCOC2)OC)nn1 24737,Cc1cc(Br)cc(C(N2C3CCC2C(NC(=O)CN(C)C2CC2)C3)=O)c1N 24738,c1(C(=O)NC2C(C)CCN(C(c3cnc(C)o3)=O)C2)cc2c([nH]1)CCCC2 24739,N1(C(c2c(CC)occ2)=O)CCC2CCN(C(c3ccnn3C(F)F)=O)CC2C1 24740,c1(N2CC(NC(c3cccc(C#C)c3)=O)C(C#N)C2)ncnc2sc(Br)cc12 24741,Cc1c(C(=O)NCCOCCNC(=O)CC(C)n2ccnc2)ccn1C(C)C 24742,CCCC(C(=O)N1CC(NC(C2COCCOC2)=O)CC1CO)OC 24743,c1(OC)cc(N(C)C)ccc1C(=O)NC(C)CN(C(=O)C(C)CC1CCC1)C 24744,CC1(C)COc2cc(C(N3CCSCC3CNC(=O)C[PH](C)(CC)c3ccccc3)=O)nn2C1 24745,c1(-c2nc(N(C(C)=O)C(c3nccnc3Br)=O)sc2)cn(C)nc1C(F)(F)F 24746,N1(C(c2c(OC)csc2)=O)CC(C)(CNC(C2CC3CCC2CC3)=O)CC1(C)C 24747,C1(C(=O)NCC(CNC(C(C)Cc2ccncc2)=O)F)C2CC3C(C2=O)C13 24748,N1(C(C(CC#C)NC(=O)CCC(F)(F)F)=O)CC(C)(C)CCC1C 24749,C1(C(N2C3CCN(C3)C(=O)C3C(C3C)OC2=O)=O)CC(=O)CO1.C1(CC)CCC1 24750,Cc1ncc(N)cc1C(=O)N(C1CCCN(C(C2CC3CCC2CC3)=O)CC1)C 24751,CN1CCN(C(=O)C(C)(C)CC2CC2)CC1C(=O)NCC1C2CCCC12 24752,c1(C(N(C(C)CNC(=O)CN(C)C(C)C)CC)=O)cccc(C2CC2)c1 24753,C1(C(=O)NCC2(CO)CN(C(=O)CC3(O)CCCCC3)C2)CS(=O)(=O)CC12CC2 24754,C1(C(=O)NC(CC=C)CO)CN(C(c2ccns2)=O)CC1C(C)C 24755,C1(C(=O)NC2CCCCN(C(c3ccco3)=O)C2)CCC2C(CC1)C2(F)F 24756,c1(C(=O)NC2CCC(C)N(C(c3cncc(F)c3Cl)=O)C2)cnc2ccnn2c1 24757,C(=O)(C1Cc2ccccc21)NC(C(=O)NCCc1ccc(C)nc1)CCN(C)C 24758,N1(C(c2[nH]cc(C)c2)=O)CC(C)CC1C(=O)Nc1cccc(F)n1 24759,C1(C(=O)NC(CNC(c2n(C)cnn2)=O)C(C)(C)C)CCCCN1N=O 24760,N1(C(C2CN(C(c3cc(C)n(C)n3)=O)CC2F)=O)CC(O)CC(O)C1 24761,c1(OC)cc(Cl)ccc1NC(=O)NCC(N1CC(=O)NC(C)C1)(C)C 24762,N1(C(C(C)(C)C2CC2)=O)CCOCC(NC(C2(CSC3CC3)CCC2)=O)C1 24763,N1(C(C(C)(CSC)NC(C(CC#C)C2CC2)=O)=O)CCOCC(=C)C1 24764,C=CCCCC(C(=O)NOCC1(C)CCC1)NC(c1csc(C)c1)=O 24765,Cc1cc(CC(=O)NC(C)CCNC(=O)CC2CCOC(C(C)C)C2)c(C)o1 24766,c1(CN(c2ccccc2)C(C(C)Nc2ccccc2)=O)c(Cl)nc2sccn12 24767,N1(C(C2=CCC(NC(C(CCC)=CCC)=O)C2)=O)CC2CCCCC12C 24768,C1(C(=O)NC(C2CCCC2)CNC(C2NC(=O)OC2)=O)CCS(=O)CC1 24769,CC1(C)CC2(CN1Cc1cccc(OCC(F)F)c1)CC(F)(F)C2 24770,c1(C(N(C(CNC(Cc2cncc(C)c2)=O)C)C)C)cccc2ccccc12 24771,N1(C(c2c(C)cc(C(F)F)o2)=O)CC(NC(c2cc(N)cc(O)c2)=O)CC(O)C1 24772,N1(C(c2nccc(N(C)C)c2)=O)CC2(C1)CN(C(=O)COC1CCOC1)C2 24773,CC1CCc2nc(C(N3CCC(N(C)C(c4cccs4)=O)C3)=O)ccc2C1 24774,CCCC(CCC)CCCC(=O)N(CCCNC(=O)CC(C)(CC)C(=O)OC)CC 24775,n1(CC(=O)NC2C(NC(C(C)C(F)(F)F)=O)CCCC2)ccc(=O)n(C)c1=O 24776,N1(C(C(C)CC(C)(C)C)=O)CCC2(CC1)CCN(C(C1CNC(=O)N1)=O)CC2 24777,c1(C(N2CCC(CN(C(Cc3nc(C)sc3)=O)C)CC2)=O)cc2c(ncn2C)s1 24778,N1(C(c2csc(-c3ccccn3)n2)=O)CCC2C(CCCN2C(=O)C2CC2)C1 24779,N1(C(CNC(CNC(C(CCC)N(C)C)=O)=O)=O)CC(OC)CC(C)C1 24780,CC1CCN2N=C(C(=O)NCC3CCN3C(c3ncccn3)=O)NC2=N1 24781,C1(c2cc(C)no2)CCCCCN1C(=O)CC1CCN(C(C2CC(O)C2)=O)C1 24782,CCC(CC)C(C)C(=O)NCC1C2CN(C(C3CCC(C)=C(C)C3)=O)CC12 24783,c1(CNC(CC2(C)CCN(C(=O)C(F)(F)C3CCCC3)C2)=O)cnc(O)c(F)c1 24784,C1(CCOC)CCCN(C(c2ccc(NCC(N)=O)cc2)=O)C1.C1(C)CC(=O)N1 24785,N1(C(C(CC)N(C)C)=O)CCC2CCCC12C(=O)N(C)CCn1cccn1 24786,c1(-c2c(C)ccnc2)cccc2c(C(=O)NCCCO)n[nH]c12 24787,C1(C(=O)NC(C(C)NC(c2ccn(C3CCCC3)n2)=O)CO)CCOC(C)(C)C1 24788,c1(C(=O)NCC2N(C(CNC(C)=O)=O)CCCC2)ncc(Cl)cc1Br 24789,C1(C(=O)NCC(CO)NC(c2ccc(C(=O)OC)cc2)=O)CC(C)(C)CN1C 24790,C1(CC(N2CCC(OCC)CC2)=O)CN(C(=O)CN2CC(=O)NC2=O)CCC1C 24791,N1(C(c2ccc(C#C)cc2OC)=O)CCCC12CCCN(C(C1(F)CC1C)=O)C2 24792,O=C(CCCC(F)F)NCCC12CCC1CN(C(=O)CCn1cc(Cl)cn1)C2 24793,C1(NC(=O)NC2(C)CCCC2Nc2ccccn2)CCC2(CC1)CC2C(=O)O 24794,N1(C(CCOCC#C)=O)CC=CC1CNC(=O)C(C)OCCN(C)C 24795,Cc1ccn2ncc(C(=O)NC(CNC(=O)COCC3CC3)CC(F)(F)F)c2c1 24796,N1(C(CCc2c(C)ncs2)=O)CCN(C(=O)CCn2cc(Cl)cn2)C(C)CC1C 24797,C12(CC(=O)NCC(CNC(c3cc(COC)[nH]n3)=O)C)CCC(CC1)C2(C)C 24798,Cc1c[nH]cc(Br)c1=NC(=O)C1CCCCN1C(=O)COc1ccccc1 24799,c1(C(=O)NCC(=O)NCC(=O)NC2CCCC(OC)C2)ccc(P(C)(C)=O)o1 24800,c1(C(=O)OC)ccc(C(=O)NCC(C)NC(=O)CCC(C)SC)cc1Cl 24801,c1(C(=O)NCC(CC)NC(=O)Cc2cc(F)ccc2Cl)cc(F)c2cn[nH]c2c1 24802,c1(OCC=C)cccc2[nH]c(C(=O)N(C(C)CNCC)Cc3cncs3)cc12 24803,C1(NC(=O)COCC2CCC2)CC(F)(CNC(c2cc(Cl)no2)=O)C1 24804,c1(C(=O)NC(C)CCNC(=O)C(C2CCCCC2)C)nnn(C)c1N 24805,c1(SC)nc(N(C)CC2CCCN(C(c3cscc3Cl)=O)C2)cc(C)n1 24806,c1cc(C(C)(C)C)cc(C(C)(C)C)c1CC#N.c1(C2C(OC)CC2)ccc(C)cc1 24807,Cc1cnncc1C(=O)NCC1CCC1C(=O)NCC1CN2CCC1C2.C(C)(C)(C)S 24808,C1(NC(c2ccncc2Br)=O)CN(C(C2CCCCO2)=O)CC(F)(F)C1 24809,C(=O)(CC(C)(O)C(F)(F)F)N1CC(C(C)NC(c2c(C)cc(C)[nH]2)=O)OCC1 24810,c1(CNC(CCSCCC)=O)ccc(CN(C)C(c2ccncc2F)=O)cc1 24811,CS(=O)(=O)C1(C(N2CC3CC(NC(=O)CCOC4CC4)C2C3)=O)CCC1 24812,CC1CN(C(=O)C(F)(F)c2cscn2)CCC1N(C(=O)CSC(F)F)C 24813,c1(NC(c2ccc(F)cc2)CC(=O)N2CCC(OCCO)C2)c(Br)ccnc1Cl 24814,Cc1n[nH]cc1CC(=O)NC(CO)C(C)NC(=O)CC(C)n1cccn1 24815,Cc1ncnc(C)c1NC(=O)C(C1CCN(C(=O)CC(O)C(C)C)CC1)C 24816,C1(F)(C(N(C(CCN(CC)Cc2ccc(C)cc2)=O)C)=O)CC12CCCCC2 24817,C1(C(N2C(C(C)C)CN(C(=O)Cc3nncs3)CC2)=O)CCC(=O)C(C)C1(C)C 24818,C(=O)(CC(C)C(F)F)N1CCC(CN(C(c2ccnc(C(F)F)c2)=O)CC)CC1 24819,CCC(C)(C#N)C(=O)NCc1ccc(C(=O)NC2(CO)CC(F)(F)C2)cn1 24820,c1(C(=O)NC(CNC(=O)C(F)OC(F)(F)F)C2CC2)cc2c([nH]1)CCOC2 24821,S(=O)(=O)(c1ccc(CC(=O)NCC#CCNC(=O)CC#N)cc1)NCC 24822,Cc1cnn(C)c1CNC(=O)Nc1nnc(N(C)C)s1 24823,C1(NC(C2CCCCCN2C(C2CC(F)(F)C2)=O)=O)C2CCC(F)(F)C12 24824,CON=CC(=O)N1CCC(C(=O)NCC2CC2c2ccco2)O1 24825,N1(Cc2ccc(C)c(C)c2)CC2C3CCC(C2C1)N(C(=O)CC1CCCCC1)C3 24826,c1(NC(N(CCN2CCCCC2)CC)=O)ccc2c(=N)[nH][nH]c2c1 24827,CCCCC(CNC(C12CCC(C1)C2)=O)NC(c1ccsn1)=O 24828,N1(C(C(c2ccccc2)=O)=O)CC(NC(C2CCCSS2)=O)CC2(CCC2)C1 24829,CCC(C)(CO)C(=O)N1CCCOC(CCNC(=O)CCC(=O)N(C)C(C)C)C1 24830,Cc1cccc(-n2nnc(CC3CC(F)CN3C(=O)OC(C)(C)C)c2C(C)C)c1 24831,c1(N2CCC3(CN(C)C3)C2)ccc(Br)c(S(=O)(=O)NCC2C(CO)C2(C)C)n1 24832,CC(C)C(C)(C(N)=O)NC(C1CC2CC2N1C(C1CCC2(CC2)C1)=O)=O 24833,c1(N2CCC(NC(N3CCCCC3c3nccs3)=O)C2)ccc(Br)nc1 24834,c1(OC)ccccc1C(=O)NCC(=O)NC1CC1NC(C1CC(O)(C(F)F)C1)=O 24835,c1(C(N2CC(CC(C)NC(=O)CCc3nncn3C)C2)=O)cc(N)cc(O)c1 24836,c1(C(N(C(CC)C)CCn2nc(C3CC3)cc2C)=O)ccc(C=O)cc1 24837,c1(CC)nn(C)cc1C(=O)N(CC(CC)NC(=O)C(C)Cc1cccc(F)c1)C 24838,c1(C(=O)NC2C(NC(=O)Cn3cnnc3)C2)cncc2c[nH]nc12 24839,C(c1ccc2cc(OC)ccc2c1)=CC(=O)NCCNC(CCC(=C)C)=O 24840,c1(C(=O)NCc2c(C3CCN(C(C)=O)C3)n[nH]c2)cccn2c(C)nnc12 24841,Cc1csc(=NCC(=O)N2CCC3CCCC23CNC(=O)C(=O)NC2CC2)[nH]1 24842,C(=O)(C1CCCc2nc[nH]c21)NCC(CNC(c1nc(OCC)sn1)=O)(C)OC 24843,C1(C(=O)NCCCN(C(C2(C)CCCO2)=O)C2CC2)CCc2ncncc2C1 24844,c1(OC)cc(N2CC3CN(C(c4ccco4)=O)C3C2)nc(C)n1 24845,CC1(CCCO)CCN(C(C2(NC(c3cn(CCO)nn3)=O)CCC2)=O)CC1 24846,C=CCC(CNC(=O)C(C1CCOCC1)F)C(=O)N(C1CC=CCC1)CCF 24847,c1(C(N2C(C3CCN(C(CCC(C)C)=O)CC3)CCC2)=O)ccc2n[nH]cc2c1 24848,N1(C(c2c(C)nn(CC(F)F)c2)=O)CC(NC(=O)C=Cc2cnc[nH]2)CC(O)C1 24849,C(=O)(C(O)CC1CC1)N(CCNC(C(C)OCC1CC1)=O)CCc1ccccc1 24850,C(CNC(=O)CCCN(C)C(C)C)(C(C)(C)C)NC(CCN(C(C)=O)C)=O.CCO 24851,Cc1nn(C)cc1C(=O)NCC(C1CCCCC1)NC(=O)C(F)=CCCF 24852,C(=O)(CS(=O)(=O)CC(F)(F)F)NCC(C1CC1)NC(C1(CC#C)CCOCC1)=O 24853,Cc1n[nH]c(C)c1C(C)C(=O)N(CC)CC1CCCN1C(=O)CC1CCOCC1 24854,c1(NC(C2N(C(CC(C)c3ccccc3)=O)CC=C2)=O)nc(Cl)c(Br)cc1O 24855,N1(C(C(OC)OC)=O)CCCC(NC(c2ccc(OC)cc2C(F)(F)F)=O)CC1 24856,C(=O)(C(COC)CC(C)C)N1CCC(NC(CC2(OC)CCCCC2)=O)(CO)C1 24857,C1(CNC(C(C)n2cccn2)=O)CC2CC2N1C(=O)C=CCN1CCOCC1 24858,Cc1cccnc1CC(=O)NC1CC(C(=O)N(CCC#N)C2CC2)C1(C)C 24859,c1(OC)cc(F)c(CC(=O)NCCNC(c2cnc(C(F)(F)F)s2)=O)c(Cl)c1 24860,c1(C(C(=O)NCC2(F)CN(C(C3CC(OC)C3)=O)C2)(C)F)ccc(F)cc1 24861,c1(C(=O)NCC2CN(Cc3cn[nH]c3)CCO2)c(C(F)(F)F)cccc1Br 24862,c1(C(=O)NC2CC(C)(CNC(CC=C)=O)C2)cccc(OC)c1 24863,Cc1ccc(C(=O)NCc2cc(C(=O)NCC3(O)CSC3)no2)c(C)c1 24864,c1(OCC)cc(C(=O)NC(C(=O)OCc2ccccc2)C2CC2)ccn1 24865,C#CCC(C)(C(=O)NCC(CCC)OCC)NC(=O)C(CC)C(=O)OC 24866,O=C(C1=NOCC1)N1CCC(C2CCCCN2C(c2n[nH]cc2Cl)=O)C1 24867,C(CCCCCN=C(NCC(c1ccccc1F)O)NC1CC(F)C1)SC 24868,C1(NC(CNC(N)=O)=O)CCCOC12CCN(C(C1(C3CC3)CC1)=O)CC2 24869,c1(-c2cn(C3(C(=O)OC)CN(C(C4(C)CNC(=O)C4)=O)C3)nn2)cc(OC)nn1C 24870,c1(CN2CC3C(C(=O)Nc4cnc(C)nc4Cl)C3C2)c(F)ccc(Cl)c1Cl 24871,c1(CNC(c2cc(=O)cc[nH]2)=O)cccc(NC(C2OCCCO2)=O)c1 24872,c1(C(N(CC(CC)NC(C2C3CC(=O)CC23)=O)C)=O)nc(C)oc1C 24873,C(C(=O)N(CC(=O)NCc1nonc1C)CC(C)C)(C(C)C)SCC 24874,c1(OC)ccccc1OC(C)C(=O)NCCC(C)N(C)C(c1c[nH]c(C#N)c1)=O 24875,C1(OCC(=O)OC)CCN(C(C2CN(C(c3ocnc3C)=O)CCS2)=O)CC1 24876,C#CC1(O)CC(C(N2CC(F)CC2C(=O)N(CC=C)CCO)=O)C1 24877,C12(C(N3CC(CCO)(CC)C3)=O)CCCC1CCN2C(=O)CCC1(C)N=N1 24878,CN1CCC(CC(=O)NC(C)(CNC(=O)CN(C2CCC2)C)C2CCC2)CC1 24879,N1(C(C2CC23CCCC3)=O)CC2CCC1C(CNc1cc(F)ncn1)C2 24880,C1(NC(c2cc(C(C)C)[nH]n2)=O)CC2CC1N(C(C1(C(F)F)CCC1)=O)C2 24881,CCC(C(=O)N1CC(CCNC(c2ccn(C)c2C)=O)C(C)C1)C(C)C 24882,Cc1cc(C(N2C3CC2CN(C(c2c(O)cccc2O)=O)C3)=O)cc(Br)c1 24883,Cc1ccc2cc(C(N3CCCC(NC(c4coc5c4COC5)=O)C3)=O)cn2c1 24884,c1(CN2C(C(=O)OCC)CCC2NCc2ccccc2)ccc2c(c1F)CCC2 24885,Cc1cc(Cl)c(C(=O)NC(C)(CNC(=O)CC2(O)CCCOC2)CO)cn1 24886,c1(OC)cc(C=CC(N2CCC(NC(=O)C(F)CC3CCCC3)C2)=O)sn1 24887,c1(N(c2cc(=N)[nH]cc2)C(c2cc(F)ncc2Br)=O)ccc2c(c1)CNC2 24888,N#Cc1ccc(Cl)c(C(=O)NCCNC(C2CCOC2c2ccccc2)=O)c1 24889,O=C(C(Cc1ccccc1)NC(=O)C1CC1)Nc1nnc(Cc2ccccc2)s1 24890,C1(NC(CCCSC)=O)CCC2CCN(C(=O)C=Cc3cncn3C)C1C2 24891,c1(C(=O)NCC2C3CN(Cc4cccc(C)c4Br)CC32)ccc2scnc2c1 24892,C1(N(C(=O)CCN(CCO)C(c2ccc(CO)o2)=O)C)CCC(CC(C)(C)C)C1 24893,Cn1nc(C(=O)NC(CNC(c2cnoc2-c2ccccc2)=O)C2CC2)cc1Cl 24894,CC1CC2(C(N3CC(SC(C)(C)C)C3)=O)CC12 24895,C1(=CCC)CCN(C(=O)C(C)=CCNC(=O)C(F)C2CCC2)C1 24896,c1(C(=O)NC(CN(C(c2ccc(F)c(O)c2)=O)CC)C)ccc(C)cc1OC 24897,N1(C(c2ccc(SC)cc2)=O)CCC(NC(=O)CN2C(=O)COC2=O)C1(C)C 24898,CC(CC(=O)N1CCC(N(CC(C)C)C(C2CCC(O)C2)=O)CC1)C(F)(F)F 24899,C=CC(CC(=O)N1CC(O)(CNC(c2oc(CC)nc2C)=O)C1)c1ccccc1 24900,c1(C(N2CC(O)(CNC(CCC(=C)C)=O)C2)=O)nc(Cl)ccc1Cl 24901,c1(OCC)ccc(CN(C=O)C(c2ccccc2)CC2CCC2(F)F)c(C)c1 24902,N1(C(CC2CCN(C(CNC(N)=O)=O)CC2)=O)CCCC(C2CCC2)C1 24903,c1(CN2CCC(NC(c3c(C)ccnc3)=O)C(O)C2)ccc(F)c(C#N)c1 24904,C12(C(N(C3CCCC(NC(c4coc(C5CC5)n4)=O)C3)C)=O)CCC(CC1)C2 24905,C(C(=O)NCCCC(C)NC(=O)CCNC(c1ccco1)=O)(C(C)(C)C)SC 24906,Nc1nc(C(=O)NCCS(=O)(=O)NCc2c(Cl)nsc2Cl)ccc1O 24907,C=CC(C)(O)CC(=O)N1CCC(C(C)(C)C(=O)NC2CCOC2C)C1 24908,N1(C(Cc2c(C)non2)=O)CCC(C)(C(N2CCC(OCC(N)=O)C2)=O)C1 24909,CC(O)C(C)C(=O)NC1(CNC(=O)CCCc2cccs2)CC1 24910,N1(C(COCCC#C)=O)C2CCC1CN(C(=O)CN1C(=O)NC(C)(C)C1=O)C2 24911,C(=O)(CCCCC#N)NCC1CN(C(C=CCOC)=O)C(C)C1 24912,C1(NC(C(CC)OCC)=O)CC2CC(C1)N(C(c1ccnc(Cl)c1N)=O)C2 24913,c1(OC)nc(Cl)ccc1C(N1CCCCC(NC(C2CCN(C)C(C)C2)=O)C1)=O 24914,C1(O)(C(N2CC(C)N(C(=O)CCCN=[N+]=[N-])CCC2)=O)CCc2ccccc2C1 24915,C(=O)(CCCC(N)=O)N1CCC(NC(C2C(C)C2(F)F)=O)C1C1CC1 24916,CCN=c1[nH]cc(C(=O)N(CCC(c2cccs2)NC(c2cnoc2C)=O)C)s1 24917,CCC(C)(COC)C(=O)NC1C=CCC(C(=O)NCC(C)C(C)O)C1 24918,C1(C)(C(N(C(CCNC(C(C(C)C)n2cnnc2)=O)C)C)=O)CC2CCC(C1)S2 24919,N1(C(C2CCN(c3ccccc3)C2)=O)CCc2sccc2C1c1ccc(Cl)cc1 24920,c1(C(=O)NCC2CCCN2C(=O)C2=CCS(=O)(=O)C2)ncnc2ccccc12 24921,Cc1cnc(C(N2CC3CC2C3C(=O)NCC2CCC(C)(C)O2)=O)c(F)c1 24922,c1(OC)ccc(C)cc1C(=O)NCCCN(CCO)C(C1CCC1C(=O)OC)=O 24923,c1(C(CN(C)Cc2snc(C)n2)O)ccc(Cl)c(Cl)c1 24924,N1(C(c2nc(OCC)oc2)=O)CCC(C)(C)C1CNC(=O)C(C)(C)CO 24925,c1(CC(N2CCSC3CCC23)C(=O)NCC2CC(=C)C2)ccc(OC)c(OC)c1 24926,Cc1cccc(CN(C(C2C3CCN2CC3)=O)Cc2cccnc2)c1 24927,N1(C(c2n[nH]c(C)c2C)=O)CC(C)(C(=O)NCC(c2ccccc2)O)CC1(C)C 24928,C1(C(=O)NC(C2CCCN2C(=O)CC2CCC(=O)O2)(C)C)CCc2cncn2C1 24929,C=C=CC(C)C(=O)NC1(C(F)F)CC(NC(=O)CCCOCCOC)C1 24930,N1(C(c2ccc(C3CC3)s2)=O)CC2CCCC(N=c3ccnc(CO)[nH]3)C2C1 24931,CCC(CCCC(=O)N1CC2COCC2O1)NC(C1(F)C(C)(C)C1(C)C)=O 24932,N1(C(CCCOC(C)=O)=O)CCN(C(=O)C(CO)NC(N)=O)CC1c1cn[nH]c1 24933,CC1CCN(C(C2CC(F)(CO)C2)=O)CC1NC(c1ccoc1Cl)=O 24934,N1(C(C(=O)NC(C(=O)OC)C)c2ccoc2)CC(c2cccc(Cl)c2)OCC1C 24935,CCCCC(C)C(=O)NCCn1cc(CNC(=O)CSc2ccc(Cl)cc2)nn1 24936,c1(C(N2CC=CC(NC(C(NOC)=O)=O)C2)=O)cccc2c(C)coc12 24937,C=CC(CCC)CC(=O)N1CC=CC1C(=O)NCCOC1(C)CCCC1 24938,C1(NC(C2CC(=C)C2)=O)CC2CCC1CN(C(c1cn(C3CCOC3)cn1)=O)C2 24939,C(=O)(CCC(C)(C)O)NC(C(C)C)CNC(=O)Cc1ccc(C(N)=O)cc1 24940,C1(COC)(NC(=O)CCNC(N)=O)CCN(C(C2CC3(CSC3)C2)=O)C1 24941,N1(C(C(CC(F)F)NC(c2c(C)ncs2)=O)=O)CC2C3CCC(C3)C12 24942,c1(CC(=O)NCCOC2CCN(C(COCC(=C)C)=O)C2)cnn(C)c1C 24943,C1(C(=O)NC(C(=O)NCC(C)(C)SC)(C)C2CCC2)Cc2ccccc2C1 24944,c1(C(N(C2CCN(C(=O)CCc3ncco3)CC2)C)=O)ccc(F)c2c1OCC2 24945,O=C(CC1CCOc2ccccc21)NC1CN(C(c2nccc(Br)c2)=O)C1 24946,Cc1cc(-c2cncc(C(N3CCN(C(C)(C)C)CC3)=O)n2)c(C)cc1O 24947,C1(C(C2(C(C)(C)[N+](=O)[O-])CC2)C)CCCCC1NC(N1CC(c2cc[nH]n2)C1)=O 24948,CCC(CNC(=O)C(C)(C)c1ccccc1)(CC)NC(=O)CN(C1CCSC1)C 24949,C1(CC)CN(C)CCCN1C(=O)C(CC(N)=O)NC(=O)C(C(C)OC)N(C)C 24950,c1(NC(C2CCN(Cc3sc(Br)nc3Br)CC2O)=O)ccc2c(c1)C(=O)CCC2 24951,c1(OCCC)ccc(CN(C(=O)C(CC)SC(C)=O)C(C)(C)C)cc1 24952,C1(OC)CC(C(=O)N(C2CC3CNC2C3)CCc2csc(C)n2)CCC1O 24953,Cc1cc(CNC(=O)C(CC2CCCC2)NC(=O)C(C)C#N)no1 24954,c1(C(C(N2C(CCCCCC)CCCC2)=O)(F)F)ccc(Cl)c(Br)c1 24955,CC1(CNC(c2cc[nH]n2)=O)CCCN1C(=O)C=CCO 24956,C=CC1(C(=O)NCc2ocnc2C(=O)NCC2CC(N(C)C)C2)CCOCC1 24957,c1(C(N(CC(C)CNC(=O)CCCn2ccccc2=O)C)=O)cc(Cl)ccc1N 24958,CCCC(C)C(=O)NC1CC(F)(C(=O)OC(C)(C)C)C1.C12CCC1CNC2=O 24959,C1(N(C)C)CCC(C(N2CC(C(N)=O)(CNC(c3n[nH]cc3C(N)=O)=O)C2)=O)CC1 24960,n1(CC)cnnc1CNC(=O)C(C1CC1)N(C(=O)Cc1nonc1C)C 24961,N1(CCC(C)C)CC(C(=O)NC(C)(C)C(C)NC(c2ccc(F)cc2)=O)CC1=O 24962,C1(NC(CCNC(C)=O)=O)CC2(CCN(C(C3CC3Cl)=O)CC2)C1 24963,c1(CCC)ccc(N)c(C(=O)NCC=CCNC(=O)C=CC2CCC2)c1 24964,C1(C(=O)OCC)CN(C(=O)C(Br)=C(C)C)CC1C1CC1 24965,N1(C(c2c(Cl)cn(C)n2)=O)CCCC2CN(c3nc4ccc(Br)cc4s3)CCC12 24966,C=CCC(CC=C)C(=O)NC(CN(C)C)C(=O)NCC(=O)OCC 24967,C1(CNC(C=C(CC)C)=O)CN(C(c2cc(C)[nH]n2)=O)CC12CCC2 24968,C(CC(O)CCc1ccccc1)C1(NC(CC(=C)Br)=O)CC1 24969,c12cc(c(F)c(F)c1)NC2=O.C1(=CC(=O)NCC(CC)OC)CCSCC1 24970,N1(C(c2cccc(OC)n2)=O)CC(CC(=O)NC2CC(F)(F)C2(C)C)C2(CC2)C1 24971,N1(C(C(COC(C)(C)C)(C)C)=O)CC2CC(NC(=O)CCC3CCOC3)C1C2 24972,c1(NC(=O)N(C2C(C(N3CCCC(O)C3)C)C2)CCCl)ccccc1O 24973,N1(C(c2cc(C)n(C)c2)=O)CC2CCN(C(c3ccnc4cc[nH]c34)=O)C2C1C 24974,C1(NC(c2cn(CCC)nc2)=O)CS(=O)(=O)CC1NC(=O)C=Cc1csc(C)n1 24975,c1(C(N2CCC(NC(c3c(CC)cno3)=O)C23CC3)=O)noc2c(F)cccc12 24976,C(=O)(C(C)(C)CN1CCOCC1)NCC(CO)NC(C1(CCCC)CC1)=O 24977,Cc1ccnc2sc(C(=O)NCC3CC3NC(=O)Cc3ccc(O)c(F)c3)c(C)c12 24978,CC1CN(C(C2CCC(C(C)(C)O)CC2)=O)CCC1CNC(C1(C)CC1Br)=O 24979,C(=O)(CCOCCCN(C(C(=O)COC)c1cnsc1)CC1CC1)OCC 24980,C12(C(=O)NCC3C(NC(CN(CC)CC)=O)CCCC3)CCCN(CC1)C2 24981,CC(C)CC(CNC(C1OCCC1C(C)C)=O)C(=O)Nc1ccccc1N=[N+]=[N-] 24982,c1(CC)onc(C(N2CCOC(C(=O)NCC(C)(O)CO)C2)=O)c1C 24983,C1(NC(c2n(C)c(S)nc2)=O)CN(C(c2noc3c2CCCC3)=O)CCC1(C)C 24984,C(C(O)CC(=O)NC1(CCCCO)CC1)NC(C(C)(C)NC(C)=O)=O 24985,CN1Cc2cc(NC(C3C=CCN3C(=O)Nc3ccccc3Cl)=O)ccc2C1=O 24986,C(c1c(C)nn(C)c1Cl)=CC(=O)NC1C(OC)CN(C(c2cc(=O)cc[nH]2)=O)C1 24987,C1(NC(C(C2CC2)OC)=O)CCN(C(c2cn(CC(=O)N(C)C)nn2)=O)C1C1CC1 24988,C(C(c1ccccc1)NC(=O)CCF)(C(C)C)NC(c1c(OC)nsc1)=O 24989,C(C(=O)NCC1CC(NC(=O)Cc2csc(C(F)(F)F)n2)C1)(C(C)O)NC(C)=O 24990,C1(C(=O)NCC2(C)CCOCC2)C2CC3C(C2NC(=O)CC2CCCC(=O)N2)C13 24991,c1(Nc2nc(-c3ccc(OC)nc3OC)sc2)ncnc2c1ccn2C 24992,C(=O)(C1=Cc2cc(Br)ccc2OC1)NC1CCN(C(C)=O)CCC1(F)F 24993,c1(CN2CCC3(C(C(=O)Nc4ncc(Br)s4)C3)CC2)c(F)c(F)cc(F)c1F 24994,c1(OC)ccc(CC(=O)NCC2(C(=O)NOCCN(C)C)CCCOC2)cc1 24995,CCC(C)(CC)NC(C1CC(CCNC(=O)CC(=O)N(C)C)C1)=O 24996,C1(NC2CCC(C(C)(C)C)CC2)CCCCN(C(=O)Cc2ccnc(Cl)c2)C1 24997,C1(C(=O)NC2C(OCC)CCCC2)CC12CCN(C1CCN(C)CC1C)CC2 24998,C(=O)(C(C)CS(=O)(=O)NC1CCC(CC(C)(C)C)C1)OC 24999,CCC(c1ccccc1)=CC(N1CCC(C)C1CNC(c1c(C)coc1C)=O)=O 25000,C1(CNC(CCN(CC#C)C(C2CC(C)CO2)=O)=O)CCCOCC1 25001,c1(C(C(=O)NC)N(C)Cc2ccc(C(C)C)cc2)cc(C)c(Br)c(Cl)n1 25002,N1(C(C2(OC)CCN(C(c3c[nH]c(=O)cn3)=O)C2)=O)CCCCC(CO)C1 25003,N1(C(Cc2cc(C)[nH]n2)=O)CCC2(CCN(C(c3cc(Cl)c(N)c(Cl)c3)=O)C2)C1 25004,C1(C(=O)NCCCN(C(c2c(N)cccc2Cl)=O)CC)CCn2c(cnc2C)C1 25005,C(N=c1cc(NCCCn2ccnc2)nc[nH]1)c1cc(Cl)nc(=N)[nH]1 25006,C1(C(=O)NC2CN(C(C(C)OCC=C)=O)C(CO)C2)CC12CCOCC2 25007,C1(NC(c2ccsn2)=O)COCCN(C(=O)CCc2ccsc2)C1 25008,c1(CC(=O)N(CCCCN(C(CC=CC=C)=O)C)C)cc(F)cc(Br)c1 25009,C(=O)(C1SCc2cccnc21)NCC=CCNC(c1cc(CCC)[nH]n1)=O 25010,C(=O)(C1CCc2c(F)cccc21)NCc1cc(OC)ns1 25011,C1(C(=O)NC2C(C(=O)NC(C=C)(C)C)OCC2)CCOC(C)C1 25012,C(=O)(C(C)(C)CNC(=O)CCCOC(C)C)NCC(C1CC1)OCC 25013,c1(C(=O)NC2(C3N(C(C(F)=CC)=O)CCC3)CC2)cccc(C(F)(F)F)c1OC 25014,c1(OC)cc(I)c(C(N2C3CCC2CC(c2cnn(C)c2)C3)=O)cc1OC 25015,c1(CNC(=O)CN(C(=O)CCc2cnco2)CC2CC2Cl)nncs1 25016,N1(C(C2C(C)(C)C2(F)F)=O)CCC(CNC(=O)Cn2ncc(O)nc2=O)C(O)C1 25017,N1(CC(CNC(=O)NC2CC(CSC)C2)O)CCCC(C)C1 25018,c1(C(=O)NC2C(C)(C)N(C(=O)CCCC#N)CC2)ccc([N+](=O)[O-])cc1Cl 25019,C=CCC(C(=O)NCC(C)N(C(c1[nH]nc2ncccc12)=O)CC)C(C)C 25020,c1(C(=O)NC2CC(NC(CS(CC)=O)=O)C2)cc(O)nc2cc(F)ccc12 25021,C1(NC(CN(C(=O)CN2CCCC2C)C(C)C)=O)COCCOC1 25022,C(C(CNC(=O)CC1CCN(C(c2nc[nH]n2)=O)C1)C(C)C)OC 25023,C1(CCC(=O)NC(CCCNC(C(C)NC(CC)(C)C)=O)C)CCCC(O)C1 25024,c1(C(N2CC(O)(CNC(c3ncn(C(C)(C)C)c3)=O)C2)=O)ccc2c(c1)COC2 25025,C1(C(=O)Nc2c(OC)c(N)ccc2)CS(=O)(=O)C2CN(C(C)=O)CC12 25026,CC1(C2CC2)CCCN1C(C1CCC(NC(=O)CCC2CC2(F)F)C1)=O 25027,C1(n2cnnn2)(C(=O)NCCC(C)NC(=O)C(C)(C)NS(C)(=O)=O)CCOCC1 25028,Cc1cc[nH]c(=N)c1C(=O)NC(CNC(=O)C(C)c1cccs1)C1CC1 25029,c1(OC)ccc([N+](=O)[O-])c(C(N2CC(F)CC2C(=O)NCC2CCOC2)=O)c1 25030,C1(C(N2C(C(=O)OC)CCC2)=O)COCCN(C(c2cnc(C)n2C)=O)C1 25031,S(=O)(=O)(c1cc(C)ccc1C)N(CC(CC)CC(C)C)C1CC2CNCC12 25032,c1(OC)ncc(C(N2CCCCC2C2CCN(C(c3ccsn3)=O)C2)=O)cc1F 25033,c1(OC(C)C)cc(OC)cc(CN2CCN(CCO)CC2)c1.N1(C)CCN(C)CC1 25034,c1(C(=O)NC(CNC(C(C(C)C)(C)O)=O)CO)coc(S(N)(=O)=O)c1 25035,CCCCC(CC)C(=O)N1CCCC(N(C(c2ccc(C)nc2C)=O)CC)CC1 25036,C1(OCC)CN(C(=O)C(=Cc2c[nH]cn2)F)CC1CNC(c1cn(C)nc1Cl)=O 25037,c1(C(N2CCCC(NC(C3CC3(F)F)=O)C2)=O)c(OC(F)F)cccc1Br 25038,c1(C(=O)NC2C(CNC(c3scc(OC)c3)=O)CCC2)n[nH]c2ccccc12 25039,Cc1cc(C(=O)NCC2CCCC2C(N2CCCC(C#N)C2)=O)cc(O)n1 25040,c1(C(N2C(CNC(Cc3c(C)csc3Cl)=O)CC2)=O)ccc2c(c1)CCNC2=O 25041,CC(C)(C)C(C(=O)N1CCC(NC(=O)CC2CCC3CC23)CC1)N1CCOC1=O 25042,Cc1ccc(C)c(C(=O)NCc2ccc(C(=O)N(C3CCCC(O)C3)C)s2)c1 25043,N1(C(CC(C)(C)F)=O)CCC2CCCC12CNC(=O)COCC1CC1 25044,c1(N(c2ccc(F)cc2)CCC#N)ccc2ccccc2c1O 25045,c1(CC)cc(C(=O)NC(C)CN2CCN(C(=O)C=CC(C)C)CC2)cn(C)c1=O 25046,N1(C(C(C2CCN(C(CCCOCCC)=O)C2)C)=O)CCCC2C(O)CC12 25047,N1(c2ccnc(NCCS(CC)=O)n2)CC(C)(C)C(F)(F)C1 25048,c1(C(=O)NC(CCC)C(N2CC(O)CC(C)(C)C2)=O)ccc(C#N)c(C)c1 25049,C1(NC(C(C)C(C)O)=O)CC2CCCC(C1)C2NC(=O)Cn1ccc(O)nc1=O 25050,C(CCCC(C)(C)C(=O)NNC(=O)C1CCCS1)NC(C1(C=C)CCOCC1)=O 25051,Cc1nc(=N)[nH]c(C)c1C(N1CC(NC(c2ccc(C(C)C)cn2)=O)C(C)C1)=O 25052,c1(C(=O)NC2C(NC(C3(C(C)(C)C)CCCC3)=O)C2)cccc(CCO)c1 25053,C(=O)(CC(C)C(F)(F)F)N1C(C(N2C(COC)COCC2)=O)CC2CC21 25054,C1(F)(CNC(C(C2CCC(=O)N2)C)=O)CCN(C(=O)CC2SC(=N)NC2=O)CC1 25055,N1(C(C2CCCC(C(N)=O)C2)=O)CCCC(C)(CNC(c2ccc(CO)s2)=O)C1 25056,N1(C(C2CCCN2C2CC2)=O)CCCCC(N=c2ccc([N+](=O)[O-])c(O)[nH]2)C1 25057,NS(=O)(=O)CC(=O)NC1CN(C(c2cccc(C3(O)COC3)c2)=O)C2CC12 25058,c1(CNC(c2cc(C)sc2C)c2nnnn2C2CCOC2)cn(C)c(=O)nc1O 25059,N1(C(C(C=C)O)=O)CC(C2CCCN(C(c3ccc([N+](=O)[O-])cc3F)=O)C2)C1 25060,Cc1ccc(C)c(C(C)N(C)Cc2cc(-c3ccccc3)[nH]n2)c1 25061,c1(C(N(CCN(C)C(C2CCc3ccnn3C2)=O)C)=O)cncc2ccsc12 25062,C1(NC(c2c(C)ccnn2)=O)C(C)(C)CN(C(c2cnsc2C)=O)CC1(C)C 25063,C(=O)(CC(C)(C)CC(=O)NCC1(C2CC2)CCN(C(=O)Cc2ccsc2)C1)OC 25064,C(=O)(C1=NOC2(CCC2)C1)N1C(CNC(c2occc2Cl)=O)CC(O)C1 25065,C(=O)(C(F)CCC(C)C)NC(CC(=C)C)C(=O)NC(c1cccnc1)CC 25066,N1(C(c2n(C)cnc2)=O)CCCC(C(=O)N(C(C)(C)C)CCO)C1 25067,C(=O)(C1CCCCc2ccccc21)N1CC(O)(C(C)NC(CCCOC)=O)C1 25068,c1(C(=O)NCCCCC2CN(C(C3N(CC)CC3)=O)C2)cc(N2CCCC2)ccn1 25069,NS(=O)(=O)CC(=O)NCCCN1CCC(NC(=O)CC(F)(F)F)C1 25070,c1(NC(C(=O)NCC(F)(F)F)=O)ccc2nc(Cn3ccccc3=O)[nH]c2c1 25071,c1(CC)[nH]nc(C(=O)NC(CCC2CCC2)C(=O)NC(c2cnc(C)s2)C)c1C 25072,N1(C(C2(COC)CC=CC2)=O)CC2OCC(C(=O)N(C)CC#N)C2C1 25073,CC(c1cccnc1)=CC(=O)NCC1CC2CCC1N2C(=O)Cn1ccc(C)n1 25074,c1(C(=O)NCCN(C(=O)C(=O)NOC)CCC)ccnc(OC(C)(C)C)c1 25075,c1(C(N2CCC(NC(Cc3c(C)ocn3)=O)C2)=O)cc(O)cc(Br)c1 25076,CC(CC(=O)NCC1C(C(=O)NC(CC(N)=O)C2CC2)C1(C)C)C(F)F 25077,CCCC(CC1CCCC1)C(=O)NCC1CCN(CC(O)COC)CC1 25078,c1(OC)cc(F)c(F)cc1C(N1CCC(C)(C(N)=O)CC1)=O 25079,c1(OC)ccc(C(=O)N(C)CCNC(=O)C(C)S(N)(=O)=O)cc1S(=O)(=O)NC1CC1 25080,C(=O)(C(C(C)(C)C)NC(=O)C(C)C)NCCC1(NC(CCC(C)OC)=O)CCC1 25081,C(=O)(C(C)(C)C(O)CC)N1CCC(CC=C)(NC(c2cc3c(s2)CCC3)=O)CC1 25082,c1(C(N(CCNC(c2cc3ccccn3n2)=O)CC)=O)ccc([N+](=O)[O-])cc1Cl 25083,C1(C(=O)NC2(CCO)CN(C(CC3(NC(C)=O)CC3)=O)C2)CCOCC12CCC2 25084,CCCC(C(=O)NC1CCCN(C(c2ccc(F)c(C(F)F)c2)=O)C1C)C(C)C 25085,Cc1nn(CCO)c(C)c1C(=O)NCC(C)(C)OCCNC(=O)CCC1(C)CC1 25086,CC1CCC(NC(c2ccc(C#N)n2C)=O)CN1C(c1cnc(C2CC2)nc1)=O 25087,C1(C(N2C(CNC(c3c(C)ccc(OC)n3)=O)C=CC2)=O)CC2(CCOCC2)C1 25088,N1(C(CCC(=C)C)=O)CCCC(CO)(NC(=O)CCSc2ccc(C#N)cc2)C1 25089,C1(NC(=O)CC(F)(F)F)CC2(C1)CC(NC(c1ccc(SC(F)F)cc1)=O)C2 25090,CC1(C)C(C(N2CC(CNC(=O)C(c3ccccc3)O)C2)=O)CCS1(=O)=O 25091,c1(C(C2(OC)CCOC2)NC(CCC)C2CCCC2)nnnn1CCC1CC1 25092,CC1CN(C(=O)COCC2CC2)CCN1C(C1CCCCN1C1COC1)=O 25093,C1(NC(=O)NCC=O)CC2CN(C(C(CC)NC(C)=O)=O)CC2C1.C1CCCC1 25094,c1(C(N2CCCC(CCNC(C(COC)O)=O)C2)=O)cc(C)cc(Cl)c1 25095,C1=C(CNCc2ccc(-c3ccco3)cc2)OCCO1 25096,C1(C(=O)NC(C2CCN(C(CC(C)C)=O)C2)C)Cc2ccccc2N1C 25097,c1(OCCCC)ccc(C(=O)NCC2C=CCN2C(=O)CCNC(=O)C2CC2)cc1 25098,c1(OC)csc(C(N2CCOC(CNC(C3CCCC3C)=O)C2)=O)c1OC 25099,c1(C(=O)NC(C(C)NC(c2ccn(C3CC3)n2)=O)C)c(F)cccc1Cl 25100,c1(OC)cnc(F)c(C(=O)N(C(C)CN(C)C(c2cncc(COC)c2)=O)C)c1 25101,S(=O)(=O)(c1cnn(C)c1)N1CC(C(=O)NCC(C)CN(C(=O)C(C)C(F)F)C)C1 25102,CCC(C)CC(=O)C(=O)N(CCC(=O)NC(C1CCOC1)CO)C 25103,CC1(C)CCCOC1C(=O)NCCCC(=O)NCc1cccc(O)n1 25104,N1(C2CC(CCC)C2)CCCCC(C(=O)NCC(N2CCN(C)CC2)C)C1 25105,C12(C(N3CC(O)(CC(=O)OC)C3)=O)CCN(C(C3(C)C=CCCC3)=O)CCC1C2 25106,C1(CCNC(CCCOCCOC)=O)CCCN(C(=O)Cn2cnnc2)CC1 25107,CC(C(=O)NC1CC(C(F)(F)F)CN(C(=O)CCc2cnn(C)c2)C1)S(N)(=O)=O 25108,N1(C(CC)=O)CC2CCC1C1CN(C(c3ccnc(OCC(F)F)c3)=O)CC21 25109,CCCCCCCC(=O)NC1C(C)CCN(C(=O)COc2ccc(F)cn2)C1C 25110,CC1CCN2N=C(C(=O)NCCN(C(=O)C(C)NC(=O)C3CC3)C3CC3)NC2=N1 25111,c1(C(=O)NC2CCCC(NC(CCSCCC)=O)C2)cc(C)c2c(c1)CCC2 25112,c1(CNC(c2n(CCC)nnn2)c2cc(CSC)no2)ccc(C(=O)OC)cc1 25113,N1(C(CN(C(=O)CCC2CC(C)C2)CC)=O)CC(CO)OCC1C 25114,C1(CNC(CC=C(C)C)=O)CN(C(=O)C(C2CCCCCC2)C)CC12CCC2 25115,C(=O)(CC(C)CC(C)(C)C)NCC1=CCN(C(c2c(NC(C)=O)cccn2)=O)CC1 25116,N1(C(C(C)OCCC=C)=O)CCCC1C=CC(=O)NCc1ccc(C)cc1 25117,Cc1noc(C(C)C)c1C(=O)NC1CCCC1CNC(=O)CC1CCC=CCC1 25118,c1(C(N2CCCC(C)C2CNC(C2CC3(C2)CC3F)=O)=O)ccc2nonc2c1 25119,c1(C(C)NC(CCN(C(C(COC)OC)=O)CCO)=O)ccncc1F 25120,N1(C(C(C)n2cnnn2)=O)CC2CCCC(C1)N2C(c1cnc(F)c(F)c1)=O 25121,c1(CC(N2C(C)(C)CC(NC(=O)CCCC3CC3)C2)=O)n[nH]c2c1CCCC2 25122,c1(C(=O)NCCC(=C)CNC(=O)C(C)CC2CC2)ccc(Cl)c(N2CCNC2=O)c1 25123,C1(=CC(=O)NCCCCCCNC(=O)Cc2csnn2)CN2CCC1CC2 25124,CC1CCN(C(C2(O)CC2)=O)CC1NC(c1coc(-c2ccccc2)n1)=O 25125,C#CCCC(O)C(=O)NCC(c1ccccc1)N(C(=O)Cc1sc(C)nc1C)C 25126,Cc1scc(CNC(=O)CC(O)CNC(C2CC3C=CC2O3)=O)c1C 25127,c1(OC)ncc(C(=O)N(C(C)CN(C(=O)C(O)C2CC2)C)C)c(C)n1 25128,O=S(=O)(c1cnn2ccc(=NCC3OCc4ccccc43)[nH]c12)NCCC=CBr 25129,C(=O)(N=c1[nH]nc(CC2CC2)s1)NCCOC(CNC(C)=O)(C)C 25130,c1(CNC(c2nc(C)oc2C)=O)cc2n(n1)CCN(C(=O)CC1CCC1)C2 25131,CCCC(C(=O)N1CC(OC)C(NC(=O)C(=O)N=S(C)(C)=O)C1)S(N)(=O)=O 25132,CC(CC#N)C(=O)NC(C(N1CCC(C(F)F)CC1)=O)c1ccco1 25133,CC1CC(CO)CCN1C(=O)CN(C(=O)NNC(=O)c1ccc(Cl)cc1)C1CC1 25134,CCC(C(=O)N1CC(CNC(=O)CC2CCOC2=O)C1)N(C)C 25135,N1(C(CNC(CCC)=O)=O)CCCC1CC(c1ccco1)=O 25136,N1(C(C2(OC)CCCC2)=O)C2CCCC1CC(NC(=O)C(C1CC1)SC)C2 25137,Cc1[nH]nc2cc(C(N3CC4CC3CN4C(C3CCS3(=O)=O)=O)=O)ccc12 25138,C1(C2CC2)(OC)CN(C(=O)C(C2CCOC2)NC(c2cn[nH]c2)=O)C1 25139,CC1CCN(CC2CCN(C(=O)OC(C)(C)C)C(C)C2)CC1C 25140,C1(C)(NC(C=CC(C)NC(c2cn(CC)nn2)=O)=O)CC(F)(F)C1 25141,C=CC(C)(C)CC(=O)N1CC(F)(F)CC1CCNC(=O)C(C)COC 25142,N1(C(=O)OC(C)(C)C)CC2CCCC2C1NC(=O)Nc1cc(Br)cc(CO)n1 25143,C1(CC(=O)NC2CN(C(c3ccc(C)o3)=O)C2)COCCOC1 25144,C(=O)(C(C)CC(N)=O)N1CCC(C(=O)N(C)CCc2nccs2)(CC)C1 25145,c1(CNC(COCC=C)=O)ccc(CC(=O)NC2(C)CS(=O)(=O)C2)cc1 25146,C(=O)(CC(C)C(F)F)N1CC(OC)C(NC(=O)Cc2ccc(F)c(F)c2)C1 25147,C(CC(C)N=c1[nH]c(N2CCC(CN(C)C3CC3)CC2)nc2c1CC(C)CC2)OC 25148,C=C(C)C1CN(C(=O)C(O)C(CCC)NC(=O)CC2CCCC2)CCO1 25149,N#Cc1cc(NCCc2cccc(F)n2)cc([N+](=O)[O-])c1Cl 25150,C(c1ccc(F)c(F)c1)=CC(=O)NCCCCC(C)NC(=O)C(C)CC1CCC1 25151,Cc1nc(C(=O)NCCC(O)CNC(=O)C(C)(C)CS(C)(=O)=O)ccc1[N+](=O)[O-] 25152,N1(CCSC(C)C)CCSCC1C 25153,Cn1ncc(Cl)c1C(c1nnnn1-c1ccon1)NC1CCC1COC(C)(C)C 25154,c1(C(C=CC(N2CC(NC(C(C)Cc3ccco3)=O)C2)=O)=O)cccc(Cl)c1Cl 25155,C(=O)(CCCCN(C)C(c1cnnn1C)=O)N(CCN=[N+]=[N-])C 25156,Cc1cc(O)cc(C)c1CS(=O)(=O)Oc1ccccn1.N1(C)CCC(ON)CC1 25157,C1(C(=O)NCC(CNC(C(C=C)OC)=O)(C)OC)CN(C)CC(C)O1 25158,C(=O)(C(CCCC#N)N(C)C)NCC1(OCC)CCOC1 25159,Cn1ncc(Cl)c1C(=O)NCCC1CCCN1C(C1CN(C2CCOCC2)C1)=O 25160,C1(C)(COC)CCN(C(=O)C(C)NC(C2CCCCC(=O)N2)=O)CC1 25161,N1(C(C(C(C)C)O)=O)CC2(COC(CNC(C3C4CCC(C4)C3(C)C)=O)C2)C1 25162,C(CC(C(=O)NC1(SC)CCC1)OC)NC(=O)CC1C(N(C)C)CC1O 25163,CC1CC(CNC(c2ccc(=N)[nH]c2)=O)CN1C(=O)CCN1CCCC1 25164,C(CCOCCO)(C(=O)N(CC(O)C(C)(C)C)C)NC(C(C)=C(CC)C)=O 25165,C1(C2CCN(Cc3ncc(C)s3)CC2)(NC(C(C(CC)C)OC)=O)CC1 25166,C(C)(CNC(C1SCC=C1C)=O)(CC(C)C)NC(C(C=C)OC)=O 25167,C(=O)(C(C(C)(C)C)N(C)C)NC(C(C)C)(C)CNC(=O)Cn1ccnc1C(C)C 25168,C(C(CC(=O)N(C1CCOCC1OC)C)NC(c1cncc(CO)c1)=O)OC 25169,CC(=O)CCC(=O)NC(CC1CCC1)C(N1CCC(F)(CF)C1)=O 25170,c1(C(=O)OCC)ccc(=NCCCOCCc2nccc3ccccc23)[nH]c1 25171,c1(C(N2CCCC(c3cc[nH]n3)C2)C(=O)NCC=C)cc(OC)c(OC)cc1F 25172,C1(NC(N(C(c2ccc(Cl)cc2)C)C2CC2)=O)COCCC1N 25173,CON(CCO)C(=O)CC(C(F)F)NC(=O)CC1CCOCC1 25174,C1(C(=O)NCC(CNC(C(N2CCC(O)CC2)C)=O)O)CCCCC1(F)F 25175,c1(C(=O)NCC#CCNC(c2c(C(C)C)n(C)nc2)=O)cc(Cl)c(Cl)cc1O 25176,CCCCCCCC(=O)N1CC(C)C(NC(=O)C(O)Cc2cnc[nH]2)C(C)C1 25177,CC1(CCNC(=O)C=Cc2cnc[nH]2)CCN(C(c2nccnc2N)=O)C1 25178,C1(NC(c2n(CC)ncc2)=O)CC2CCC1N(C(=O)COCc1ccccc1)C2 25179,C1(NCc2cn(C)nc2Cl)CC(O)C12CC(F)(F)C2 25180,Cc1ncccc1C(=O)N(CC(C)(C)C(=O)NCC1(n2nccn2)CC1)C 25181,c1(CC(N2CCC(CC(=O)NC(C3CCC3)C)C2)=O)c(F)cccc1F 25182,c1(CC(N2CC(NC(CC(CCC)O)=O)C3(C2)CC3)=O)c[nH]c2cccc(Cl)c12 25183,N1(C(C(C)(C)F)=O)CCC2C(CCN2C(=O)C(C)(O)C(F)(F)F)C1 25184,c1(CC)ccc(C(N2CCC(CCNC(c3cn(CC)nn3)=O)C2)=O)c(O)c1 25185,CCC(CC)CCC(=O)N(C1C2CN(C(=O)C(C)CC(N)=O)CC12)C 25186,C(=O)(CN=S(C)(C)=O)NC1C(CN(C(C(C)Sc2ccccc2)=O)CC(=O)OC)C1 25187,c1(CN2CC3N(C(c4c(OC)cncc4)=O)C3C2)c(C)cc(C)cc1C 25188,c1(COC)cc(C(=O)NC(C)(CNC(=O)Cc2nccn2C)C2CC2)no1 25189,O=C1COc2cccc(C(=O)NCC3CN(C(C4CC4C(=O)O)=O)CCO3)c2N1 25190,CC1(CNC(=O)CC2(O)CCOC2)CCCC1NC(c1cnn(C2CCC2)c1)=O 25191,c1(C(N(CC(CC)NC(=O)CCCCN(C)C)C)=O)cc(O)n(CC)n1 25192,C1(CC#C)(C(=O)N(CC(C)CN(C(c2ccco2)=O)NCC2CC2)C)CCCCO1 25193,N1(C(Cc2cc(C)sc2C)=O)CC2(CCN(C(c3cc(F)ccc3Cl)=O)C2)C1 25194,C1(CNC(=O)CNC(=O)C(O)C2CC2)CCCN1C(=O)CCCN1CCOCC1 25195,N1(C(C(C)(C)n2ccc(C3CC3)n2)=O)CCC2(CCC2)CC1 25196,C#Cc1cccc(NC(=O)CC(C)CNC(=O)CCSCC(F)F)c1 25197,C1(NC(CN2C(=O)CN(C)C2=O)=O)CCC2(CC1)CC2Nc1ncncc1Cl 25198,C(=O)(C(CC(C)C)C(N)=O)NCCCN(C(c1ccc(CC)cc1F)=O)C 25199,c1(CC)cc(C(N2CC=CC2C(=O)NCc2cc(N(C)C)ccn2)=O)n(C)n1 25200,C1(CCC)CCCCN1C(c1cnc(-c2ccc(Br)cc2)s1)=O 25201,N1(C(CC(C)(C)O)=O)CCC(C2CCCN(C(c3ccc(N)cc3F)=O)C2)CC1 25202,C1(NC(COC(C)=O)=O)CC2(C1)CC2NC(=O)COc1cnn(C)c1 25203,CC1(C)CCCC(O)(C(=O)NCC2CCCC(NC(c3ccnc(O)c3)=O)C2)C1 25204,C(C)(CCCNC(c1csc(CC(F)(F)F)n1)=O)NC(C1CC(SC)C1)=O 25205,N1(c2n(CCSCC=C)c(-c3ccc(C)s3)nn2)CCCC(O)(CCOC)C1 25206,CC1CCN(C(C2CCCC2(C)O)=O)C1c1cn(-c2cccc(OCCO)c2)nn1 25207,C1(O)(CNC(c2c(C)snn2)=O)CCN(C(c2cccc(Cl)c2)=O)CC1 25208,C(N=c1nc2sccc2c(NC2CC(C)CC(C)(C)C2)[nH]1)c1cc(C)cc(C)c1 25209,CCC(CC)(CCC(=O)N1CC(OCCNC(=O)CC2CCCC2)C1)[N+](=O)[O-] 25210,C1(C(=O)NCCOC2CCN(C(=O)C(F)n3ccnc3)C2)CC2(C1)CC21CC1 25211,Nc1cc(C(N2CCC(CF)(NC(=O)Cc3ccc(F)c(Cl)c3)C2)=O)cc(N)c1 25212,N1(C(CCC(=O)c2ccc(F)cc2)=O)CC2(CCCC2)c2cc(C3CC3)ccc21 25213,C1(C(=O)NCCn2cc(C(N3C(CC)CCC3)=O)nc2)CCC(C)=C(C)C1 25214,C#Cc1cnn(C)c1C(N1CC(C)(NC(=O)CC2CC(O)C2(C)C)C1)=O 25215,n1(C(C(=O)NC2CCC(F)(CNC(C(C)=CC)=O)C2)C)cnc2ccccc12 25216,C1(C)(C(=O)NCCN(C)C(c2ccnc(F)c2F)=O)Cc2ccccc2NC1=O 25217,C12(C(=O)NC(CCCC=C)C)CC(CN(C(c3ncc(CC)cn3)=O)C1)C2 25218,C1(C(=O)NCCNC(CN(CCC)C(=O)C2CC2)=O)CC12CCC2 25219,c1(NCC)scnc1C(=O)NCCN(C1CCCC1)C(C1OCCC1C(C)C)=O 25220,N1(C(c2cnc(CC)s2)=O)C2CCC1CC(N(C)C(c1cc(C)ncc1C)=O)C2 25221,CCC(CNC(=O)CC1CC2(CC2)CO1)(CC)NC(=O)C(C)O 25222,N1(C(CCNC(=O)OC)=O)CC2(CCC(NC(=O)C(C)C(O)CC(C)C)CC2)C1 25223,Cc1nn(C)c(N)c1C(N1CCC(OCC(=O)NC(C)C(O)C(C)C)C1)=O 25224,C(=O)(CC(C)(C)C(C)(F)F)N(CC(C)NC(c1ccc(NC(N)=O)cc1)=O)CC 25225,c1(C(=O)NC(C)(C)C(C)NC(=O)C(F)=C(C)C)ccc(C2(CCC)CCC2)cc1 25226,CCCC(CC(C)C)C(=O)N1C(C(=O)NCCC(=O)OC(C)C)C2CC(O)C1C2 25227,C1(C(C)NC(c2cnc[nH]2)=O)CN(C(=O)C(N)=O)CC1O 25228,N1(C2CN(C(=O)CC3CC3(Cl)Cl)C2)CC(NC(c2cc[nH]c2C2CC2)=O)CC1=O 25229,CCCCC(O)C(=O)NC1(CCNC(c2[nH]ccc2C2CC2)=O)CCCC1 25230,Cn1cc(-c2cnn3cccnc23)cc(C(N2CCCC2C(F)(F)F)=O)c1=O 25231,S(=O)(=O)(c1c[nH]ccc1=NC1COCC(C)(C)C1)N(CC(CC)C)CC 25232,C1(NC(c2n(CC=C)nnn2)c2cc(C)on2)CCn2nnnc2C1 25233,C1(C(=O)NC2(CN(C)C(C34CCC(C3)C4)=O)CC2)CCCC2(CCCCC2)C1 25234,c1(C(N2CCC(NC(COCC#C)=O)C(O)C2)=O)cc(C)c2[nH]nnc2c1 25235,CC1CC(C(=O)NCCC2CC(NC(=O)C3=CCCCO3)C2)CC(C)C1 25236,C1(=C(CO)NC(=O)CC2CCOCC2)CCN(C(=O)CCCOCCCO)CC1 25237,c1(C(C)(C)C)[nH]cnc1C(=O)NCC(C1CC1)NC(c1cn(C(C)(C)C)cn1)=O 25238,CC(C)C(C)(CNC(=O)Cc1csc(-c2ccoc2)n1)NC(C1CCCOC1)=O 25239,c1(C(N(CC(CNC(C2(C#C)CCOCC2)=O)O)C)=O)cc2n(c1)CCOC2 25240,C1(NC(C2CC23CCC3)=O)CCC(O)CN(C(c2ccc(-c3csnn3)cc2)=O)C1 25241,N1(C(c2c(C)c[nH]c2)=O)CC2CCCC(C1)N2Cc1cc(Cl)ccc1F 25242,C1(N(C(c2cc(C)oc2)C(=O)N(C)C)CC2CCCO2)CCCN(CC2CC2)C1C 25243,c1(C(=O)NCCCCN(C(=O)CSCc2cscn2)C)cccc(C(C)(C)C)c1 25244,c1(C(N(CCNC(c2ccc(Br)o2)=O)CC)=O)ccncc1Br 25245,C1(C(=O)NC(CNC(=O)CCCn2ccnc2)C(C)C)(CSC)CCN(C)CC1 25246,c1(CCC)cc(C(=O)NC2CN(C(=O)CCC(=O)OCC)CC2C)ccn1 25247,C1(CC(=O)NCC2C(NC(CN(C)CCO)=O)CCC2)CCC(F)(F)CC1 25248,N1(C2C(c3cn(C(C)(C)C(=O)O)nn3)(C)C2)CCC(S)CC1.C(=O)C(F)(F)F 25249,C1(C2CC2)(C(=O)NCC(C(C)C)OC)CN(C(=O)C=Cc2cn(C)nn2)C1 25250,Cn1ncnc1CNC(c1ocnc1C1CC1)c1nnnn1C 25251,c1(SC)c(C(N(c2ccc(C(C)C)cc2)CC2CNC2)=O)cnn1C 25252,c1(C(=O)NC2CC(N(C(C34CC(C(C)C)(C3)C4)=O)C)C2)cn(C)[nH]c1=N 25253,C1(NC(C(N2CCCCC2)C)=O)CC(NC(=O)Cc2nnc(S)n2C)C12CCC2 25254,N1(CC)CC2CC1CN2C(C1(COC)C=CCN1C(c1oc(C)cc1C)=O)=O 25255,C1(NC(CC(C)c2ccco2)=O)COC2(C1)CN(C(=O)CC1CC(F)C1)C2 25256,C(C)(CNC(=O)C(O)CC1CC1)(CC(C)C)NC(c1[nH]cc(C)c1)=O 25257,Cn1ccc2cccc(C(=O)NC3(C)CCN(C(c4sccc4F)=O)C3)c12 25258,C(CCN(C)C(c1c(C)noc1C)=O)(C(C)(C)C)NC(c1cncc(C)n1)=O 25259,C(=O)(CCCCCCNC(c1cocn1)=O)Nc1c(C)ncnc1.CCOCC=C 25260,CCCCC(C)CCC(=O)NC(COC(C)C)C(=O)N(C(CO)C1CC1)C 25261,N1(C(C2N(CC)CCC2)=O)CC(C)(C)C(NC(C2CCOCC2)=O)C(C)(C)C1 25262,N1(C(=O)NC2(CC)CC(NC(=O)OC(C)(C)C)C2)CCC2(CC1)CC2N 25263,c1(NC(CC2CCCN(C(C(CC=C)C)=O)C2)=O)ccc(Cl)nc1CC 25264,c1(C(N(CCNC(C=C(CC)C)=O)CCOC)=O)cccc(F)c1Br 25265,CCC(O)C(F)(F)C(=O)NCC(C1CCN(C(c2ccncc2F)=O)CC1)(C)C 25266,C1(CC)C(C(=O)NC2CCN(C(=O)CCCn3nc(C)nc3C)C2C)CCN1C 25267,C12(CC(N3CCC4CN(C(CC=C)=O)CC4C3)=O)CC3CC(C)(C1)CC(C)(C3)C2 25268,C(=O)(C(C)C(O)C(C)C)N(CC(COC)C)C.C(=O)C(C)(C)C1CCCC1 25269,N1(C(c2c(OC)scc2)=O)CCC(C2(NC(c3[nH]nnc3C)=O)CC2)C1 25270,c1(C(=O)NC(CNC(CC(C)F)=O)C)nc(Br)c2c(F)cccn12 25271,N1(C(CCc2ccc(C)o2)=O)CCCC2CN(C(=O)C(C)(C)C(C)(C)O)CCC12 25272,S(=O)(=O)(c1cccc(Cl)c1F)NC1CC(C(=O)NC(c2cccnc2)C)C1 25273,c1(C(CO)NC2CC(C)(CC)C2)ccc(F)cc1F 25274,N1(S(CC)(=O)=O)CCC(NC(=NCc2noc(C(N)=O)n2)NC(C)CC)CC1 25275,C(CC(=O)N(C)CCNC(=O)C(C)OC(C)C)OCC1C(C)C1 25276,C1(F)(CNC(=O)Cc2c[nH]nc2O)CCCN(C(C2(CC3CC3)CCCO2)=O)C1 25277,c1(C(N2C3CN(C(C4(C=C)CC4)=O)C(C3)C2)=O)cc2ccc(OC)cc2s1 25278,C(CCCCC(=O)NCC1CCCC(C)(C)C1)N(C(=O)C1=CCCCC1)C 25279,CC1(C)CN(C(c2c(O)cc(F)cc2F)=O)CCN(C(=O)C(F)(F)CCCO)C1 25280,C(=O)(C1=C(C#N)CCC1)NC(C1CCCN(C(c2c(C)nc(N(C)C)s2)=O)C1)C 25281,c1(C(N2C3C(NC(=O)CCC4CCCO4)C(C3)C2)=O)n[nH]c2c1CCC2 25282,C1(NC(CCCN(C(C)C)C)=O)CC2CC(C1)CN(C(C1(O)CC(C)(C)C1)=O)C2 25283,O=C1CC2CN(C(C3CC34CCN(C(C3CC3F)=O)CC4)=O)CC2CN1 25284,C=C=CCCC(=O)N1CC(O)CC1CNC(=O)C(CC)n1ccc(C2CC2)n1 25285,n1(CC)cc(Br)cc1C(=O)OCc1nnc(C2CC2)o1 25286,Cn1cc(Cl)c(C(N2CC(O)(CCNC(C34COCC3C4)=O)C2)=O)n1 25287,C1(CC)CCN(C(c2[nH]ccc2CNC(=O)CCCCSC)=O)C1C 25288,c1(CN2CCN(c3nc(SC)c(Br)cn3)C(CC#N)C2)cc([N+](=O)[O-])ccc1O 25289,C1(CNC(C=CC=CCC)=O)CCC(N(C)C(C2CCOC2)=O)CC1 25290,N1(C(c2c(CC)c[nH]c2)=O)CCC(C)C(NC(C2(F)CCC(=O)CC2)=O)C1C 25291,N(C(=NCCc1cn2c(n1)SCC2)NC1CCCC1)CCC1(CC)CCCCC1 25292,c1(C(N2CC(C)C(NC(=O)COCC(F)F)C2)=O)cccc2ccnn12 25293,C#Cc1c[nH]nc1C(=O)NC(C)CC(C)NC(=O)Cc1ccc(F)cc1 25294,C1(C(=O)OC)CC2(C1)CC(C(=O)NCC(CNC(=O)CSC(F)(F)F)CO)C2 25295,C1(NC(C(c2cncnc2)C)=O)(CO)CCCN(C(c2cc(Cl)no2)=O)C1 25296,Cc1nc(N(C)C)sc1C(=O)NC1CCC(CCNC(C2(O)CCSC2)=O)C1 25297,C=Cc1cnn(C)c1C(=O)NCc1cccc(NC(C2(C)CCC(C)C2)=O)c1 25298,C1(NC(C(C)N(C(C)=O)C)=O)CC(C(=O)N(CC(c2nn[nH]n2)C)C)C1(C)C 25299,C1(C(N2C(C3(NC(COCCC)=O)CC3)CCC2)=O)CC(=O)N(CC(F)(F)F)C1 25300,CCCCCC(O)CC(=O)N1CCOC(CNC(=O)CC2CC=CCC2)C1 25301,c1(CNC(C2CCOC2)=O)cccc(OC)c1.C12CCN(C1)N(CCOC)C2=O 25302,C(=O)(C(Cn1cccn1)NC(=O)CC1CCCC1)N(CC#C)CCO 25303,C1(NC(C2N(C(=O)OC)CCC2)=O)CC2CC1CN(C(c1ccc(F)cn1)=O)C2 25304,c1(NC(C2CC2Cc2cccnc2)=O)cnn(Cc2ccccc2)c1 25305,c1(CC)nc(C(N2CCC(CCNC(C34CC(O)C3C4)=O)C2)=O)co1 25306,N1(C(C2N(CCC)CCC2)=O)CCCC(C(=O)NCCN2CC(OC)C2)C1 25307,Cc1ccc(C(=O)NCC(C2CCCC2)NC(C2CN(C)C(=O)N2)=O)cc1C 25308,c1(N2CC(C(C)NC(c3cc(SC)ncc3)=O)OCC2)ncnc2cnccc12 25309,c1(C(=O)NC(CCNC(C(C)SC(C)C)=O)C)ccc2c(c1)NC(=O)CN2C 25310,N1(C(C=CCC(C)(C)NC(c2cnn(C)c2Cl)=O)=O)CCC(O)(CO)CC1 25311,c1(OC)nc(=NCc2cc(C(=O)O)co2)[nH]c2ccsc12 25312,N1(C(C=COCC)=O)CC(NC(c2nc3cccnc3s2)=O)CC12CCCOC2 25313,c1(C(=O)NCc2c(C(N3C(C)(CCC)CC3)=O)occ2)nc(C)ccc1C 25314,C1(CNC(CC(CCOC)(C)C)=O)CCC2CN(C(=O)C3=CCCO3)CCC2C1 25315,C(=O)(C(CNC(=O)Cc1cncn1C)N(C)C)NCC(N(C)C)C1CC1 25316,S1(=O)(=O)c2ccc(c(Cl)c2)N1CC(F)CO.c1(NC(CC)(C)C)cccc(OCF)c1 25317,c1(C(=O)NC(CNC(c2c(SC)cc(F)cc2)=O)(C)C)cc2ccc(F)cc2o1 25318,C(=O)(C1OCCc2c(O)cccc21)NCC1(C)CC(NC(=O)C(N)=O)C1 25319,c1(OC)c(NC(=O)C(C)NC(c2cc(=N)[nH][nH]2)=O)cccc1F 25320,C1(NC(C2(CC#C)CC=CCC2)=O)COC2(C1)CN(C(=O)Cc1cccnc1)C2 25321,C(=O)(C1CC(O)c2ccccc21)N1C(CN(C(CC(CC)(C)C)=O)C)CCC1 25322,C1(CNC(C(C)OC2CCCC2)=O)C(C2CC2)CCN1C(=O)CC(C)(F)F 25323,Cc1ccc2c(c1)C(C(=O)NC1CC1NC(=O)Cc1ccc(C#N)cc1)OCC2 25324,CC1(CN=c2ccnc(NCC3CCCCO3)[nH]2)CCCCC1(F)F 25325,Cc1cccc2[nH]cc(C(=O)NCC3CC3NC(c3nnc(O)cc3O)=O)c12 25326,C1(NC(C2CC(O)(CC#C)C2)=O)CCC2(CCN(C(=O)CC(C)CC)C2)C1 25327,c1(C(C)N)ccc(N(CC(=O)NCCCC#N)C(=O)CC)cc1 25328,Cc1cc(C(N2CCC(N(CCO)C(c3cn[nH]c3)=O)C2)=O)n2ncnc2n1 25329,c1(-c2ccc(C(N3C(C(C)NC(C=CC)=O)CCC3)=O)s2)cccc(F)c1 25330,Cc1cccc(OCC(=O)NC(CNC(=O)C2=CCCSC2)CO)c1C 25331,C1(O)(CCNC(c2c(CC)scc2)=O)CCCN(C(=O)CC2CC=CCC2)C1 25332,C1(NC(C(CC=C)OC)=O)CC(NC(C23COCC(C2)C3)=O)C12CCC2 25333,C1(Cn2cnc(C(N)=O)n2)CCN(Cc2cn(CC3CCC(=O)O3)nn2)CC1 25334,c1(CC(=O)OCC)cc2n(n1)CCN(C(=O)CN1CCCNS1(=O)=O)C2 25335,C1(F)(CNC(=O)C(F)=CC2CC2)COCCN(C(c2ncsc2C2CC2)=O)C1 25336,C1(C2=CCN(C(=O)Cc3c(C)ncnc3C)CC2)(C(=O)OC)CCC1 25337,O(NC(=O)C(CC(N)=O)NC(c1csc(C#N)c1)=O)CC(C(C)C)O 25338,C1(C)(CNC(CC2N(C(CCn3ccc(C)n3)=O)CC(F)C2)=O)NC(=O)NC1=O 25339,c1(SCC(=O)NC(CNC(C(CC)F)=O)(C)CO)cccc(C(F)(F)F)c1 25340,c1(C(=O)NC2CCC(NC(c3c(CC)cccn3)=O)CC2)cc(C)c(F)cc1Cl 25341,N1(C(c2ccc(C(C)C)s2)=O)CCC12CN(C(=O)CC13CCCC1C3)C2 25342,CC1(CNC(=O)CCC2(NC(=O)C=CC(=O)N(C)C)CCCC2)CCCCC1O 25343,c1(C(=O)NC(c2cn(CCCCCO)nn2)C)ccn(CC2CCC2)n1 25344,N1(CCn2ncc(C)c2)CCC(C)C1c1cn(CCCCc2ccccc2)nn1 25345,C12(CCCCO1)CC2.C(CC(=O)NCCSC)OCCCNC(COC)=O.OCO 25346,C1(CNC(C2C(C)=C2)=O)C2CN(C(=O)COc3ccccc3)CC12 25347,C(CN=C(NCCN1CCOCC1)N1CCC(C(C)(C)C)C1)c1n(C)ncn1 25348,C#CC1CN(C(=O)CC2CCC(C)(C)O2)CCN1C(c1nnsc1SC)=O 25349,N1(CC)CCC(CNC(=O)CC2C=CC(NC(=O)C=C3CCOCC3)C2)CC1 25350,N1(C(C2N(CC)C(=O)CC2)=O)CCOC2(CCN(C(C3CC3C3CC3C)=O)C2)C1 25351,c1(CC)nc(N2C3CN(S(=O)(=O)Cc4ccc(F)cc4)CC23)ncc1F 25352,C(C(CC(=O)N1CCC1c1cccnc1)C1CCC1)NC(=O)C(C1(O)CCCC1)F 25353,C1(CNC(c2c(C)nn[nH]2)=O)CC(F)CN1C(c1sccc1C(F)F)=O 25354,C1(O)(CNC(=O)CSc2ccncc2)CCCN(C(C2(F)CCOC2)=O)C1 25355,N1(C(c2c(C)ncc(N)c2)=O)CCC(C2CCCN(C(=O)C(C)O)CCC2)CC1 25356,c1(C(=O)NC2CC(CCNC(CC(COC)C)=O)C2)cnn2ccccc12 25357,C(=O)(CC1=CCOCC1)N1CC(C)C(CC(N2CCN(C)CC2CO)=O)C1 25358,c1(C(=O)NC2CN(C(C(CCC)N(C)C)=O)C2)ccc(C(C)C)cc1F 25359,CC1(C(=O)NCC(C2CCN(C(=O)CCC3CCC3)CC2)F)CCNC1=O 25360,c1(NCC2(O)CCCN(C(C(CC)OC)=O)C2)c(C#N)cnc2c(Cl)cccc12 25361,Cc1cc(C(=O)NC(CNC(=O)NC2CC(O)(C(N3CCCC3)=O)C2)CO)sn1 25362,C(=O)(CCCCC(C)(C)C)NC(C(C(C)C)NC(=O)C=Cc1ccc(F)cc1)C 25363,N1(C(c2ccc(C)nc2C2CC2)=O)CC(C)N(C(=O)CN(C)C(N)=O)CC1C 25364,CC(C)(CS(C)(=O)=O)C(=O)NCC1(C(F)F)CCN(C(=O)Cn2ncnn2)C1 25365,C1(C(NOCc2cn(CC3CCC(=O)O3)nn2)=O)CC2CCCC2C1 25366,CC(CC(C)NC(=O)CNC(=O)C(CO)N(C)C)NC(=O)NCC1CCCCC1 25367,C1(COC)CCCCN1C(=O)CCN(C(=O)CCc1ccc[nH]1)C(C)C 25368,CC(C)(F)CCC(=O)NCC1(C)CCCN1C(C1COC(=O)O1)=O 25369,CCCCS(=O)(=O)CC(=O)NC1(CNc2ccncc2[N+](=O)[O-])CCCC1 25370,C1(C(=O)NCC(COC)NC(c2cnc(C3CC3)s2)=O)CNC(=O)N1C 25371,C=CCC(C)(C(F)F)NC(=O)CCn1cc(-c2ccc(C)cc2C)nn1 25372,C1(NC(c2ccn(CCOC)n2)=O)CN(C(=O)CNS(=O)(=O)C2CC2)CC1C 25373,S(=O)(=O)(c1ccc(OCCBr)cc1O)NC1(NCc2ccc(OC)nc2)CCC1 25374,Cc1cc2[nH]c(C(=O)NCC(C(C)C)NC(=O)CCCCCN(C)C)cc2o1 25375,c1(C(=O)NCC(C2CCCC2)C)cn(CCNC(c2cc[nH]n2)=O)cn1 25376,N1(C(CCN(C(C)=O)C)=O)CCC(C2CCN(C(c3ncc(Cl)cc3F)=O)C2)C1 25377,N1(C(c2n(CCC)ccc2)=O)CC(CNC(C2(C)CCCCC2)=O)CC12CCC2 25378,N12CCN(CC1)CC(C)NC2=O.C1(NC(CC=CCC)=O)CCC(C)CC1 25379,n1(CCNC(CCCn2cc(COC)nn2)=O)cc[nH]c(=O)c1=O 25380,c1(C(=O)NCCC2OCCCN(C(CC(CC)(F)F)=O)C2)cc(S(N)(=O)=O)c[nH]1 25381,c1(C(C)NC(=O)NCc2cccc(F)n2)cccc(Cl)c1Cl 25382,Cc1cc(C)c(C(=O)NCCC2CCN(C(=O)C(c3ccccc3)O)C2)s1 25383,C1(C(=O)NCC(CNC(C2CCC(OC)C2)=O)(C)C)C2CCC3(COC(=O)C13)O2 25384,Cc1cnc(C(N2CCC(C)C(NC(c3cccnc3O)=O)C2)=O)c(F)c1 25385,C(=O)(C(C(C)O)NC(C)=O)NC(CC)CN(C(=O)C(C)c1ccon1)C 25386,C1(C(N2C(C(=O)OC)CCC2C(C)C)C(=O)NC)CCC2(CC2)C1 25387,C1(C(N(CCN(C(=O)CCCCc2ccccc2)C)C)=O)CCC(C)(F)CC1 25388,Cc1nsc(C(N2CCCCC2CC(=O)NCC2CC(F)(F)C2)=O)c1N 25389,N1(C(c2c(COC)cc[nH]2)=O)CCCC(CCC(N2CCC2(CO)CO)=O)C1 25390,Cc1nc(NCC(C)(C)C)cc(=NCc2ccc3ncsc3c2)[nH]1 25391,c1(C(N2CCCC(NC(c3ncn(CC)n3)=O)C2)=O)c(C)oc(C)c1Br 25392,C(CNC(c1cnc(SC)s1)=O)(C(C)(C)C)NC(c1cn(CC(CC)O)nn1)=O 25393,Cc1cc(F)cnc1C(=O)NCC1(CC(=O)NCC(C2CC(C)(C)C2)O)CC1 25394,C1(C(N2C(CCNC(=O)COC3CCCCC3)CCC2)=O)CCCC2(CCC2)O1 25395,N1(C(c2c(CNC(C(C)SC(C)C)=O)nccc2)=O)CCc2nnnn2CC1 25396,C1(O)(CNC(C2CCN(C(C)=O)C2)=O)CCN(C(c2cnoc2C2CC2)=O)CC1 25397,c1(C(=O)NCC2(C)CCCC2NC(C2(O)CC2(C)C)=O)nnc(O)cc1O 25398,C1(CNC(=O)NC(c2ccc(N(C)C)cc2)CN(C)C)Cc2ccccc2O1 25399,c1(C(=O)NC23CC(CNC(c4c(CC)occ4C)=O)(C2)C3)ccc2c(c1)CCO2 25400,N1(C(c2c(OC)nsc2OC)=O)CCCC(CNC(c2csnc2Cl)=O)CC1 25401,C(=O)(CCCC(C)(c1nnnn1C1CCCC1)NCc1ncc(Cl)n1C)OC 25402,C1(N(C(CCCOC)=O)C)CC2CCC(C1)N2C(C12CCCC1C2(F)F)=O 25403,C(CC=O)(CC)NC(C=CCCC)=O.C12(F)CC1C(=O)NC2=O 25404,N1(C(c2cc(CNC(c3ccco3)=O)no2)=O)CC2CC1CO2 25405,N1(C(C(CC(=C)C)C)=O)CCC2CCN(C(c3c[nH]c4nccc-4c3)=O)C2C1 25406,C1(SCC(=O)NCC(=O)NC2(C#N)CC2)CCOCO1 25407,C(=O)(C1=C(CC)OCCS1)NCC(C1CC1)NC(c1oc(CC)c(C)c1)=O 25408,C(=O)(CC1CS(=O)(=O)C1)NC1CC(NC(c2c(=N)c(Br)c[nH]c2)=O)C1 25409,C(C(C)CC(=O)N1CCCCC1C(C)(C)CNC(c1cc(C#N)on1)=O)OC 25410,N1(C(C2(CNC(c3ccc(C)o3)=O)CCCO2)=O)CCCC(C)CC1 25411,c1(CNC(C2(Cl)C(C(C)=O)C2)=O)cncc(C(=O)NC2CCCC2(F)F)c1 25412,C1(OC)CCC2(C(N3CCCC(C(=O)NC4(c5cccnc5)CC4)C3)=O)CC12 25413,c1(CCC)cc(C(=O)NCC(O)CCNC(=O)Cc2cccn2C)ccn1 25414,CC1c2cc(O)ccc2CCN1C(=O)C(=O)Nc1snc(-c2ccccc2)c1Cl 25415,c1(C(=O)NCC2C3CN(C(C4(CCCC)CC4)=O)CC32)cc(CC)nnc1C 25416,c1(CCC(=O)NC2CN(C(CCC(=C)Cl)=O)CC(C)C2)cccc(S(N)(=O)=O)c1 25417,C1(CNC(C2(CC#C)CCC2)=O)CN(C(C2(OC)CCC2)=O)CC(C)(C)O1 25418,C1(C(C)NC(=O)CN2CCCC2=O)CCN(C(C2COC(=O)N2)=O)CC1 25419,C1(NC(C(CC)O)=O)CC2(C1)CC(C(=O)NC(c1ccc(O)nc1)C)C2 25420,Cc1cc(CN2CCC(C(C)NC(C3COCCN3C)=O)CC2)ncn1 25421,N1(C(c2cc(C(C)(C)C)no2)=O)CCC2(CC1)CC2C(=O)O 25422,N1(C(CN(C2CC2)CC)=O)CC2CN(C(C34CCC(C3)OC4C)=O)CC(C1)O2 25423,CS(=O)(=O)C(CNC(=O)CSCC(F)F)CNC(C1CC2CC2C1)=O 25424,C12(CC(=O)N(C3CCN(C(c4ccc(CC#N)cc4)=O)C3)C)COCC(C1)C2 25425,N1(C(CCc2onc(CCC)n2)=O)CCC(NC(c2cc(Cl)cn2C)=O)CC1C 25426,N#Cc1c(N2CC(NC(=O)C(O)CC3CCNCC3)C2)sc2c1CCCC2 25427,c1(OC)ccc(CNC(C)C(=O)NC23CC(C(=O)OC)(C2)C(C)O3)cc1OC 25428,C(=O)(C1SCCc2sccc21)OC(C(C)(CN(C)C)NCCC#N)C 25429,C12(NC(c3cnc(=N)[nH]c3)=O)CCN(C(c3cnn(C4CC4)c3)=O)CC1C2 25430,Cn1ccc(=O)cc1C(N1CCOCC(C(=O)NCCc2ccc(O)cc2)C1)=O 25431,C(=O)(C1CCCc2nn[nH]c21)N1CC2CC(NC(=O)Cn3ncccc3=O)C2C1 25432,Cc1cc(C(N2CCC(NC(=O)C(=O)N(C)C)C(CO)CC2)=O)cc(C)c1C#N 25433,c1(C(N2C(CNC(c3c(C)ccc(OC)c3)=O)CC2)=O)cn(C)c2ncccc12 25434,CCCCCC(O)C(=O)NC(C)CN(C(=O)C(c1ccc(=O)n(C)c1)(F)F)C 25435,N1(C(c2cc(C)sc2)=O)CC(C)CN(C(c2ccn(C)c2C)=O)C(C)C1 25436,C1(CC(=O)NC(C)CC(=O)OC)(OC)CN(C(c2cnn(C(C)C)c2)=O)C1 25437,c1(CC)c(C(=O)NC2COCCC2C(=O)NCc2cccnc2)ccn1C 25438,c1(C(=O)NCC2N(C(C(c3scc(C)n3)(F)F)=O)CC2)nc(C2CC2)oc1C 25439,Cn1c(NCC2(CNC(=O)CC=C(Cl)Cl)CCC2)cc(=O)n(C)c1=O 25440,c1(C(=O)NC2C(C)(CC)C2)cc(CNC(C2(CC)CCCC2)=O)[nH]n1 25441,N1(C(C2(S(C)(=O)=O)CCC2)=O)CC2CCC1CN2C(=O)CN1CC2C=CC1C2 25442,CC1CCCC1NC(=O)CCCN(C(=O)CC1CCCC1)C 25443,c1(CNC(c2cc(C)[nH]n2)C)ccc(CN2CCC(C)CC2)cc1 25444,N1(C(Cc2n(C)nc(Br)c2)=O)CCC(NC(=O)CCc2ccoc2)C12CC2 25445,C1(SC)CC(CC(=O)N(C(C)CCNC(=O)C=CBr)C)C1 25446,N1(C(COC)=O)CC(OC)C(NC(=O)Cn2cc(-c3ccc(C)cc3)nn2)C1 25447,c1(C(=O)NCC(CO)NC(CC(CC)C2CC2)=O)cc(C)ccc1C 25448,N1(C(CC=C)=O)CCC2CCCC12C(=O)NC(c1ccnn1C)C 25449,S(=O)(=O)(c1ccc(C(=O)NC2CC(NC(C3CC3(F)F)=O)C2)cc1)N(CC)CC 25450,CS(=O)C1CN(C(=O)CC2CCN2C(c2csc(Cl)n2)=O)C1 25451,c1(C(=O)NCCCC2(CNC(C(C)N(C)C)=O)CCCC2)cnc2ccoc2c1 25452,C1(C(N(C)CCc2ccccc2)=O)CC12CCN(C(C1CCC1C#N)=O)C2 25453,C=CC1(C(=O)NC2CCC(NC(=O)C(C)=CCC)CC2)CCCCC1 25454,C(=O)(CCCN=[N+]=[N-])N1CCC(N(C(=O)Cc2occc2C)CCOC)CC1 25455,c1(-c2cn(C3C(NC(Cc4c(C)non4)=O)CCC3)nn2)cccc(Cl)c1Cl 25456,C1(CNC(CCc2n(C)cnc2)=O)C(O)C(O)CN1C(C1CCNC(=O)C1)=O 25457,c1(C(N2CC(C)C(NC(=O)COCCN(C)C)C2)=O)cnc2c(c1)COC2 25458,C1(NC(C2(OCC)CCOC2)=O)CCCCN(C(=O)Cc2cncnc2O)C1 25459,C(=O)(CC(CC(C)C)NC(C12CCC(C)(C1)OC2)=O)N1CC(C)(CC=C)C1 25460,N1(CCC)C(=O)CCC1C(=O)NCC1(CN(C(=O)C(CCC)N(C)C)C)CC1 25461,C1(C)(C(=O)NC2C(NC(C)=O)CCC2)Cc2ccc(Br)cc2C(=O)O1 25462,Cc1ncncc1NC(C1CC1NCc1cccc(C(F)(F)F)c1)=O 25463,N1(C(C(CC2CC2)NC(Cc2n(C)ccn2)=O)=O)CCC12CC(C(N)=O)C2 25464,C1(C(=O)NCCC2(OC)CN(C(C3CC34CC(O)C4)=O)C2)(CC)CNC(=O)C1 25465,Cc1cc(C(=O)NC(C)CNC(=O)Cc2cccc(C3CC3)c2)cc(Br)c1 25466,C1(NC(C(C(C)C)(C)C)=O)CC2CCC1CN(C(=O)CC1CCCCC1O)C2 25467,c1(C(N(CCNC(Cc2ccc(C)c(C)c2)=O)C2CC2)=O)cc2ccncc2s1 25468,N1(C(c2c(C)cn(C)c2)=O)CCC(F)C(NC(c2cc(C)n(C(C)(C)C)n2)=O)C1 25469,c1(COC)cc(C(=O)NCCN(CC(C)O)C(=O)CN(C2CCSC2)C)sc1C 25470,Cc1nn(C)c(C)c1CCC(=O)NCCOCCCN(C)C(C1CCCOC1)=O 25471,c1(C(=O)NC2CCCN(C(c3n(CC)cc(Cl)c3)=O)CC2)cc(O)cc(N)c1C 25472,N1(C(CCCC(=C)C)=O)C2CCCC1CN(C(C1CCc3n[nH]cc3C1)=O)CC2 25473,C1(C(=O)NCCC2CC(C)C2)CN(C(C2(C)CCCC2O)=O)CC1(F)F 25474,N1(C(c2ccc(C)nc2O)=O)CC2(C1)CN(C(=O)C(C1CC1)C1CC1)CCO2 25475,C1(C(N2C3C(NC(CN(CCC)C)=O)C(C3)C2)=O)CCCC2CCCN12 25476,c1(C(=O)NCCN(C(C(CC#C)O)=O)C2CC2)ccc(OC)c(C)c1 25477,c1(NC(C2N(C(COC)=O)CC2)=O)ccc([N+](=O)[O-])c(C(=O)OC)c1 25478,N1(C(c2cc(C)[nH]n2)=O)CCN(Cc2ccc(-c3cccs3)o2)CC1 25479,c1(OC)cc(N)c(C(N2CC(NC(=O)Cn3cncn3)C3CC23)=O)cc1F 25480,C1(C(N2CC(S(C)(=N)=O)C2)=O)(NC(c2scc(OC)c2)=O)CCC(C)(C)C1 25481,c1(N2CC(N(C(c3ccn(CCOC)n3)=O)C)C2)ncnc2[nH]c(C)nc12 25482,c1(C(=O)NCC2CC(NC(C(C=CC)O)=O)C2)cc2n(n1)CCCC2O 25483,Cc1ncc(Cl)cc1NC(=O)COC(C1CC1c1ccc(C2CCCCC2)o1)=O 25484,c1(CNC(C2C3CN(C(c4nc(C)nc(O)c4)=O)CC32)=O)ccc(Cl)c(C)c1F 25485,C(=O)(CC(C)C(C)C)NC(COCC)C(=O)NC1CCC(CC)CC1 25486,C(=O)(CC(C)(C)N(C)C(C1(Cl)CC1)=O)N1C(CC)CCC1 25487,C1(C#N)(C(=O)NCC(C)(C)NC(c2c(C)n[nH]c2)=O)C(C#N)C1(C)C 25488,C1(C(=O)NC2CCCC(NC(c3cccnc3)=O)C2)CCCC12CCC2 25489,N1(Cc2ccc(C(=O)OC)cc2)CCCC(C)(CNC(C2CC(C)=NO2)=O)C1 25490,C=CCC(CNC(=O)C(C#N)CCC)C(=O)N1CCC(OC(C)=O)C1 25491,c12cc(ncn1)N(C1CNCC1C#N)C2=O.c1(CC)cc(Cl)sc1Cl 25492,c12ccc3nc(sc3c1)CN2.C(CC(=O)N(C)C)(c1cccs1)OC(C)=O 25493,C1(CNC(c2ccc(Cl)[nH]2)=O)CC(F)CN1C(C1CCS(=O)(=O)C1)=O 25494,CN1CCC(=CC(=O)NC2CC(CCNC(c3n[nH]cc3Br)=O)C2)CC1 25495,Cc1nc(C(C)NCC2CN(C)CCO2)ccc1OC(C)C 25496,CC1(CNC(c2cc(Cl)ccc2F)=O)CN(C(C2CCOC2=O)=O)CCO1 25497,C=CCCC(C(=O)N1CCOC(C)(C)C1)NC(=O)CCn1cnnn1 25498,c1(C(N2CC(CNC(c3cc(OC)ncn3)=O)C3C2C3)=O)ccc(F)c(F)c1F 25499,C123CC1CN(C2)C(=O)NC3=O.C(CC(C)C)(c1ncnn1C)CC.C(=O)(NCC)N 25500,N1(C(C2C(C)N(C)CC2)=O)CCC2(CCC2NC(c2cc(C(N)=O)co2)=O)CC1 25501,Cc1cc(C(N2CCC2CNC(=O)Cn2nnc(=N)[nH]2)=O)cc(C)c1C 25502,CC(C)(C)CCCC(=O)NC1CCCCC1NC(C1CC2(C)CC1CO2)=O 25503,C1(C(=O)NC(CCSC)C)CCN(C(=O)CCCC2CCCO2)O1 25504,C1(CNC(CC2CC(OCC)C2)=O)CCN(C(=O)CC2(C)CCC2)C1 25505,c1(C(=O)NCC2(F)CC(CNC(C(CCC)N(C)C)=O)C2)c(C)nn(C)c1N 25506,c1(C(N2CC3(CCC(NC(CC=C)=O)C3)C2)=O)cc(C)cc([N+](=O)[O-])c1 25507,C(=O)(C1Cc2c(Cl)cccc21)NC1C(F)CCN(C(c2ccc(CC)s2)=O)C1 25508,c1(N2CCC(NC(CC=C)=O)(CO)C2)nc(O)c2cnn(-c3ccccc3)c2n1 25509,C(=O)(C1CCc2c[nH]nc21)N1CCC(CC(=O)Nc2cc(C)nc(O)c2)C1 25510,c1(CCC(=O)NCCC(C)NC(C(C)SC)=O)ccccc1Cl 25511,C(=O)(C(C)(CCC(F)(F)F)c1ccccc1)NCc1nc(C)c(C)[nH]1 25512,c1(C(N(CC(C)CNC(c2cnsc2)=O)C)=O)cc2c(nc1O)CCCC2=O 25513,C1(n2ncc(C)c2)CCN(C(=O)C(=O)Nc2cnn(CC3CCCOC3)c2)CC1 25514,c1(C(N2CC(c3nc(C4CC4)no3)C2)=O)cc(C2(CO)CC2)ccc1Cl 25515,C1(NC(c2nc[nH]c3nccc2-3)=O)CN(C(C2CSC2)=O)C2CCCCC12 25516,C=CCC(CNC(C1CCC2CC12)=O)C(=O)NCC1(CC)CCCCO1 25517,C1(N(C(=O)CCc2cnoc2)CC)CCCN(C(=O)CC=C(C)C)C1 25518,c1(COC)nc(NCCc2c[nH]nc2O)cc(=NC2CCCC(C)C2)[nH]1 25519,c1(SCC(=O)N(C(C)CC(C)C)C2(C(C)C)CC2)ccccc1 25520,C1(NC(c2cc(CCNC(CCSCCC)=O)on2)=O)CC(CO)C2CC12 25521,c1(OCC)nc(C(=O)NCC2CN(C(C3(C)CC3)=O)CC2OC)cc(O)n1 25522,N1(C(CNC(C(C)OCCOC)=O)C)CCc2sccc2C1 25523,C(CCCCC(=O)NCC(CNC(C1CC(C)(C)O1)=O)OC)OCC 25524,N1(C(C(C)(CO)OC)=O)CC2(CNC(=O)Cc3nc(C4CC4)cs3)CC1CO2 25525,N1(C(c2cccc(C(F)(F)F)n2)C(=O)NC)CC(N=[N+]=[N-])CCC1(C)C 25526,C=CCCCCCC(=O)N1CCC2(C(=O)NCCn3nc(C)cc3CC)CC2C1 25527,n1(CC(=O)N(CC(CO)(CO)NC(C(CC)C)=O)C)c(C)nc2ccccc12 25528,CC1CCN(CC(C)(C)CNC2(c3ccc(C(=O)N(C)C)cc3)CC2(F)F)CC1 25529,c1(OCC)ccc([N+](=O)[O-])c(C(=O)NCC(O)CNC(=O)CCCCCOC)c1 25530,C1(CNC(=O)CC2CCCSC2)CCCC(CNC(C2C(C)CCO2)=O)C1 25531,CC1(C)COc2c(C(=O)NCC3CC3NC(c3csc(C#N)c3)=O)cccc21 25532,N1(C(c2nccc(C#C)c2)=O)CC2CCCCC2(NC(c2cnco2)=O)C1 25533,c1(C(C(=O)N(CCCNC(c2cccc(CC)n2)=O)C)C)ccc(Cl)c(Cl)c1 25534,C1(CN(C(C2CC2CC(C)C)=O)CC)CCCCN1C(=O)CC1(OC)CCC1 25535,Cc1ccc(OC(C)C)cc1NC(c1cnn(C2CCOCC2)c1C)=O 25536,N1(C(c2c(CCC)cccc2)=O)CC2CCC2(CCNC(=O)C2=CCCCC2)C1 25537,C(=O)(CCCCCC(=O)NC(C)CNC(=O)CC1CCC2(CC1)CC2)OC 25538,C1(OCC)CCN(C(=O)C=CC(C)(C)NC(=O)CCOC(C)=O)CC1C 25539,C12(CCNC(CCc3c(C)noc3)=O)CCC1CN(C(c1cncs1)=O)C2 25540,Cc1cc(CNC(=O)NCc2ccc(CC(C)C)cc2)ccc1O 25541,CCCC(O)CC(=O)NC1CN(C(c2ccnn2CCC(F)(F)F)=O)CC1O 25542,c1(C(=O)NCCc2cn(-c3n(C)nnc3)nn2)cc2cc(Br)cn2cn1 25543,n12cc(c(=O)cc1C)C(=O)NC1CCCCC1CC2.C(=O)(CCS(N)(=O)=O)OC 25544,c1(C(=O)NCCC2CC(NC(c3nn(C)c(O)c3)=O)C2)cnc2ncccn12 25545,C12(NC(C(C)(N(C(=O)C=Cc3ccoc3)C)C3CC3)=O)CCN(CC1)CC2 25546,c1(NCC(CCCC)NC(=O)Cn2ccnn2)ccc([N+](=O)[O-])cn1 25547,N1(C(C(C(=O)OCC)OC)=O)CCC2(CCN(C(c3coc(Cl)c3)=O)CC2)C1 25548,C1(OC)(CNC(N2CCCCC2CN(C)C)=O)CCCSC1 25549,C1(NC(c2n[nH]cc2Br)=O)CC2CC(NC(C3CC34CC4)=O)C2C1 25550,C1(C#N)(C(N(C2CC(c3cn(C4(O)CCOCC4)nn3)C2)C)=O)CC2CCC1C2 25551,CS(=O)c1ccccc1C(=O)NC1C=CC(CNC(=O)Cc2ccns2)C1 25552,C(CC(CC)(CC)NC(=O)C(C)NC=O)NC(c1cn(CCC)nn1)=O 25553,c1(NC(=O)NCC2(C#N)CC2)ccc(C(F)(F)F)cc1Cl 25554,C=CC1(c2ccccc2)CCN(C(C2C(c3onc(C)n3)N(C)C(=O)C2)=O)C1 25555,Cc1cc(N2CCCC(CNC(C3(C4CCC4)CCC3)=O)C2)nc(C)n1 25556,c1(C(N2CCN(C(C(C)OCc3ccc(C)cc3)=O)CC2)=O)cnc(F)cc1C 25557,c1(CCN(c2nnnn2-c2ccccc2)C)ccc(Cl)c(Cl)c1.C1(C)CC2CC1C2 25558,c1(NC(=O)CC2COCCN2C(=O)NC2CCC(CO)CC2)cnnc(Cl)c1Cl 25559,C1(NC(CC2CC(C)N(C(=O)CC3CCSCC3)C2)=O)CCCC(O)CC1 25560,CCC(C)C(C(=O)N1CCCC1(C)CNC(C1CCOC1)=O)OC 25561,c1(-c2c(CC)noc2)nc(Cc2cccnc2)nn1C(C)COc1ccccc1 25562,c1(CC(N2CC(CC(C)NC(c3c(CCC)n[nH]c3)=O)C2)=O)cnccc1OC 25563,c1(OC)cc(C(=O)NCCCCNC(=O)C(F)Cc2ccccc2)c(O)c(Cl)c1 25564,c1(C(=O)NC(C(C)C)CNC(=O)C2=CCOC2)c(C(F)(F)F)cccc1F 25565,C1(NC(C2CCN(C(C(C)C)=O)CC2)=O)CN(C(C2(CO)COC2)=O)C(C)(C)C1 25566,N1(C(c2c(C)scn2)=O)CC(C)CN(C(c2ncncc2Cl)=O)C(C)C1 25567,N#Cc1cc(C(N2CC(NC(C3CC(F)(CO)C3)=O)C(C3CC3)C2)=O)ccc1F 25568,N1(C(CC(=O)NCC)=O)CCC(NC(=O)CCSc2ccccc2)C1C 25569,c1(C(=O)Nc2ccc(-c3cccc(CN(C)C)c3)cc2O)cccc2occc12 25570,Cc1cc(NC(C2CC2CNC(C23CCN(CC2)CC3)=O)=O)cnc1C 25571,C1(N(C(CC(C)C2CCCO2)=O)C)CCC(CNC(=O)CCc2cccs2)CC1 25572,c1(CN(c2ccc(CNC(c3ccncn3)=O)cn2)C)cc(F)c(F)c(F)c1 25573,c1(C(=O)NCc2cccc(C(F)(F)F)n2)cc2ncccc2o1.C12CC1NC2=O 25574,C1(CC(=O)N(Cc2c(C(=O)NC3(C)CCCC3)nco2)C2CC2)CC(O)C1(C)C 25575,CCS(=O)c1ccccc1C(N1CCCN(CCNC(C2CC2C)=O)CC1)=O 25576,N1(C(C(CC#C)C)=O)CCC2(CC1)CC(NC(=O)C(C)(C)CCC)CO2 25577,C1(NC(c2c(C(N)=O)coc2)=O)CCCN(C(C2CC3OC2C2CC32)=O)CC1 25578,Cc1nc(N)c(CC(=O)NCC(C)(O)CNC(=O)CC(C)N(C)C)c(O)n1 25579,Cc1nc2cc(C(=O)NCC(CNC(c3cn(C)cn3)=O)CO)cnc2[nH]1 25580,c1(C(=O)NC2C=CC(CNC(COCCCCC)=O)C2)cccc(C#N)c1F 25581,C(C)(CNC(C1(C2(C)OCCO2)CC1)=O)(CC)NC(C1C(=C)CC1)=O 25582,N1(CC)CCCN(C(c2ccccc2C(F)(F)F)C(=O)NC2CCOC2)CC1 25583,Cc1cc(F)cc2[nH]c(C(=O)N(CC(C)O)CCNC(c3cnnn3C)=O)cc12 25584,c1(C(=O)NC2CN(C(Cc3nc(=N)[nH][nH]3)=O)CC2O)cccc2ccccc12 25585,n1(C(C)C)cnc2c(NC(c3ccnn3C)C)[nH]c(=NC3CCOC(C)C3)nc12 25586,Cc1ccn2c(C(=O)NCCCNC(c3cccc(O)c3Cl)=O)cnc2c1C 25587,N1(C(C(C)N(C(CC(C)OCC)=O)C2CC2)=O)CCN(C(=O)CO)CC1 25588,C1(C(N2CC(O)(C3CC3)C2)=O)CCN(C(C2CCCC2)=O)C12CCC2 25589,n1(CC(=O)NCC2(NC(C=CC)=O)CC3CCC2C3)cc([N+](=O)[O-])ccc1=O 25590,Cc1ccccc1OCC(=O)NC1CN(C(=O)CCC2NC(=O)NC2=O)CC1O 25591,c1(C(=O)NC2CC(N(C)C(C3CC34CCCC4)=O)C2)c[nH]c2ccc(Cl)cc12 25592,c1(C(=O)NCCC(C)NC(C2COC(=O)N2C)=O)ccc(SC(F)(F)F)cc1 25593,C1(C(=O)NCCCN(C(C(C)SC)=O)C(C)C)CC(=O)N(c2ccccc2)C1 25594,N1(C(COC2CC(N(C)C)C2)=O)CC2CC1CN2C(C1C2CCC(=O)C12)=O 25595,C(=O)(CC(C)C(C)(C)NC(=O)C(CCC)C1CCC1)NCCCCCCC=C 25596,C(=O)(C1=C(Cl)CCC1)N(CCC)CCNC(=O)CNC(c1cnccn1)=O 25597,N1(C(C=C2CCC(C)C2)=O)CCC(C2(NC(c3cc(F)c(F)c(F)c3)=O)CC2)C1 25598,c1(C(N(S(C)(=O)=O)CC2CCCCC2CN)=O)ccccc1NC1CCC1 25599,N1(Cc2cn(CCCCCN)nn2)CCOc2ncccc21 25600,C1(CNC(COCC=C)=O)CC(C)N(C(=O)Cc2cnccc2C)C1 25601,CC(CC(=O)N1CCN(CC(N2CC(F)(F)CCC2C)=O)CC1)C(C)(C)C 25602,c1(C(=O)OC)cc(C)cnc1N(CC(O)CN(C(=O)C=Cc1cccnc1)C)C 25603,c1(C(N2CCC(C3CCCO3)C2)=O)cnc(N2CCNCC2)nc1 25604,C(CN=C(NCc1c(Br)cnn1C)NC1CCN(C2CC2)CC1)N(C)CC 25605,C1(CNC(C2(CCCC)CC2)=O)CCCCCN1C(c1ccccc1OC)=O 25606,CN1CC(C)(C)CC1C(=O)NCC1CCC(C(=O)NCCC(F)(F)Cl)O1 25607,Cc1cc(O)c(C(=O)NCCCN(C(=O)COCCCF)C)cc1Br 25608,C(CC(F)F)(C(=O)N(CC)CC1CCOC1)NC(C=CCC)=O 25609,C=CCN=C(NCc1ccc(F)cc1)NC1CCCN(CC(F)F)C1 25610,N1(C(CCC(=O)C2CC2)=O)CC2CN(C(=O)C3=CCOCC3)CC2C(F)(F)C1 25611,N1(C(=O)CCc2ccoc2)CC2CN(C(c3ncc(Cl)s3)=O)CC2C1 25612,Cc1ncnc(C(N2CCC(C(C)NC(c3n[nH]cc3C3CC3)=O)C2)=O)c1C 25613,N1(C(COCCC)=O)CCC(NC(C2CCCN2C(N)=O)=O)C12CCC2 25614,N1(C(C(C)NC(C)=O)=O)CCC(C2OCCC2NC(c2ccns2)=O)CC1 25615,C(C(F)(F)F)(C1CCCCC1)NC(=O)NC(c1cscn1)C 25616,N1(C(C(C)(C)C2CCOC2)=O)CC2C(CNC(=O)C(N)=O)C2C1 25617,Cc1ccc(C=CC(=O)NCC(O)CN(C(=O)CN2CCCCC2)C)c(C)c1 25618,c1(C(=O)NCCN(C(C=C(CCN(C)C)Cl)=O)CC2CC2)cnc(C(F)F)nc1 25619,C1(F)(CNC(CCOCC#C)=O)CCN(C(C2CC2C2CC2)=O)C1 25620,C(=O)(C(C)C1=CCCC1)N(C)CC1CN(C(CSC(C)C)=O)CC12CC2 25621,CC(C)CC(CCO)NC(=O)CC1CN(C(C2(O)CCCCCC2)=O)CC1C 25622,C1(O)(CN(C)C(=O)C2CC2)CCN(C(c2scnc2C2CC2)=O)C1 25623,CC1CN(C(=O)C(c2cccs2)NC(c2cncc(CO)c2)=O)CCS1=O 25624,C(CNC(c1ccc(N2CCC2=O)cc1)=O)(CCS(C)(=O)=O)OC 25625,C1(C(N2CC3C(CNC(CNC(C(C)(C)C)=O)=O)C3C2)=O)CC2(CCOCC2)C1 25626,C1(C(=O)NC(CNC(C2CC(CF)C2)=O)C2CCC2)(COC)CCC1 25627,C(=O)(C1=NNC(=O)CC1)NC1CCC(C(N(C(C)C)C2CC2)=O)C1 25628,C1(NC(C(C(C)C)OCC)=O)CN(C(c2csc3nccn23)=O)CCC1C 25629,C(C1CCCCC1)=CC(=O)NC1(C2N(C(C3CC(N(C)CC)C3)=O)CCC2)CC1 25630,N1(Cc2ccc(C(=O)OC)[nH]2)CC2CCN(C(c3ccc(C#N)s3)=O)CC2C1 25631,N1(C(C2CCN(C(c3cnc(CC)nc3)=O)CC2)=O)CCC2C(O)CC12 25632,c1(C(=O)NCC2N(C(CCC)=O)CCCC2C)cc2ccccn2c1 25633,Cc1cc(C(N2CC3CC2CC3CNC(=O)C2=COCCC2)=O)c(S(N)(=O)=O)s1 25634,N1(C(c2cc(C)c(C(N)=O)cn2)=O)CC2CCC1C(CNC(C1(CO)CC1)=O)C2 25635,c1(C(C)C)cccc(CNC(c2cnccc2Cl)c2nnnn2CC2(C)CC2)c1 25636,N1(C(C2(CNC(C(C)OCC)=O)CCC2)=O)CC2COCC2C1 25637,c1(CCC(=O)N(C2CCC(NC(c3c(C)nc[nH]3)=O)CC2)C)ccc(C#N)cc1 25638,Cc1ccc(F)cc1CC(=O)NC(C)CN(C(=O)CCOC1CCCC1)C 25639,C1(N(C(=O)CN2CCS(=O)CC2)C)CN(C(C2CCCCCC2)=O)CC12CC2 25640,C=CCC(C(=O)NC(C)CC(C)(C)OC)NC(C1(CO)CCCCC1)=O 25641,c1(C(=O)NC(CCSC(C)C)CO)ccc(=O)n(-c2ccccc2)c1 25642,S(=O)(=O)(c1cccc(=NCC2CCOCN2CC)[nH]1)NCCC(CC)(C)C 25643,c1(N2CC(CN(C(=O)CCNS(C)(=O)=O)C)OCC2)ncc([N+](=O)[O-])cn1 25644,C1(C(=O)NC(CCOC)CNC(=O)CC2(OC)CCC2)Cc2nccn2C1 25645,Cc1nn(C)c(C)c1C(=O)C(=O)NC(CNC(c1cc[nH]c(=N)c1)=O)C(C)(C)C 25646,C1(C#CC(=O)NC2CC(NC(c3nc(C)c(C)[nH]c3=O)=O)C2)(CC)COC1 25647,CC(CCCO)N=c1cc[nH]cc1S(=O)(=O)NCc1cccc([N+](=O)[O-])c1 25648,Cc1cc(C(=O)NC2CC3CCC2N(C(C2(C(C)C)CCC2)=O)C3)cc(C)c1Cl 25649,c1(CNC(C2(NC(c3nc(Cl)cs3)=O)CCC2)=O)cccc(F)c1O 25650,C1(CC(=O)N(CCNC(Cc2c(C)con2)=O)C)CCOC(C(C)C)C1 25651,C1(NC(c2n(CC)nnn2)C(C)(C)C2CCOCC2)C=C(c2ccccc2)C1 25652,CCCC(CCCNC(C1CCCCC1O)=O)NC(c1cc(CC)no1)=O 25653,C1(NC(c2n(CC)ccc2)=O)(CF)CCN(C(=O)C=C(C)C(C)C)C1 25654,N1(C(=O)NC2(C(=O)OCC)CCC2)CC(NC2CCC=CCC2)C(C)C1 25655,c1(C(=O)NCCNC(CCc2c(C)nn(C)c2C)=O)nc(=N)[nH]c2ccccc12 25656,C(C(=O)Nn1cnnc1C)C1CN(C(Cc2c(C)ncs2)=O)C(C)(C)C1 25657,C(C(CC(C)C)C(=O)N(C1CCCC1O)C)NC(c1cc(C)oc1)=O 25658,C(=O)(C1=NN(C)C(=O)CC1)N1CC(NC(CC2C(C)CCO2)=O)CC2(C1)CC2 25659,C1(CNC(=O)C=Cc2cccs2)CCN(C(c2cn(C(F)F)cn2)=O)CC1 25660,c1(CCC(=O)NC(C)CNC(=O)COc2ccccc2CO)ccc(C#N)cc1 25661,C(=O)(CCC(C)(C)N(C)C)NC1CC(CNC(c2ncc(OC)cn2)=O)C1(C)C 25662,N1(C(CNC(=N)N)=O)CC2(CCCC2NC(=O)Cc2c(Cl)cccc2Cl)C1 25663,C1(CNC(c2c(C)nn[nH]2)=O)CC(O)CN1C(=O)CCCCN(C)C 25664,c1(CC)ccc(C(=O)NCc2csnc2N(C(C2CCC2C2CCC2)=O)CC)cc1 25665,C1(CNC(CC(C)SC)=O)CN(C(C2CC=CCC2)=O)CCC1C 25666,CCCCC(CC(=O)NC1CC2OCCCC12)NC(c1cccc(CC)n1)=O 25667,CC1CCN(C(=O)CC(C)(C)C#N)C(C)C1NC(=O)Cc1c(F)cncc1Cl 25668,C(c1cc2ccccc2o1)=CC(N1CCC(CN(C(CN(CCC)C)=O)C)C1)=O 25669,c1(C(=O)NCC(CC=C)NC(C2CC(O)CN2C)=O)c(F)ccc(C)c1Cl 25670,N1(C(C(C2CCOCC2)OC)=O)CCC(C(F)CNC(=O)CSC)CC1 25671,c1(OC)cnc(C(F)(F)F)cc1C(=O)NC1(CO)CCN(C(C2(O)CCC2)=O)C1 25672,N1(CN(CCNC(C2CCC(n3cc(CO)nn3)C2)=O)C2CC2)C(=O)CCC1=O 25673,C=C(C(=O)NC1CC1C(=O)Nc1cc(F)ccn1)C(F)(F)F 25674,c1(C(N(CCCNC(CC=CC=C)=O)C(C)C)=O)cc(O)cc(C#N)c1 25675,Cc1ccc(C)c(C(N2CC3C(CNC(C4(c5ccccc5)CC4)=O)C3C2)=O)n1 25676,C1(NC(C23OCC(C(C)C)(C2)C3)=O)CN(C(=O)C(C)CC(F)(F)F)C2(CCC2)C1 25677,CC1CN(C(=O)C(N2C(C)CCC2C)C)CCN1C(=O)CCCC(C)O 25678,CCCC(CCC)=Cc1nc(C2(C(=O)N(C)C)CC2)no1 25679,N1(C(C(C2CCOCC2)OCC)=O)CCC12CN(C(=O)C(CC)NC(N)=O)C2 25680,Cn1nc(C(F)F)cc1C(N1CCCC(CNC(=O)CC2CCNC2=O)C1)=O 25681,N1(C(CCC#C)=O)CC(N(C(=O)C(C)N(C)C)C)C2(CC2)C1 25682,N1(C(CSCC#C)=O)CC(C(N2CCc3nc[nH]c3C2)=O)CC(C)(C)C1 25683,C1(C(N(CCN(C(CCOCCCOC)=O)C(C)C)C)=O)CCC(N=[N+]=[N-])CC1 25684,N1(C(C2CCC(=C)CC2)=O)CCC2(CC(NC(=O)CCOCC(C)C)C2)C1 25685,C=CC1COCC1NC(=O)C(O)CCNC(=O)CCOCC(F)F 25686,CC(C)CC(C(=O)NCC1C2CCOCC12)N(S(C)(=O)=O)C1CC1 25687,c1(NC(C2CC(C)CN2Cc2sccc2Br)=O)nc2ccc([N+](=O)[O-])cc2[nH]1 25688,C12(c3cn(C(C4(CO)CCCO4)C)nn3)COC(CN1C(C1CC(O)CO1)=O)C2 25689,c1(C(C)=O)ccc(C(=O)NCC=CCC(=O)NCCCCCC)[nH]1 25690,c1(CN(C(CC2CC2)=O)C)cccc(C)c1.C(c1ccsc1)=CC(=O)NC 25691,C(CC(N)=O)(C(=O)N1CCCC1CC(N)=O)NC(C(C)n1ccnn1)=O 25692,C1(NC(c2occ(C)c2)=O)CCCCCCC1NC(c1cnn(C2CC2)c1)=O 25693,c1(C(C)O)ncc(C(N2CCC2CNC(=O)C(C)OC2CCCCC2)=O)s1 25694,O(NC(=O)CC1(C)CCN1C(=O)NC)CC(=O)NCC(CC)OC 25695,C(C(CC)(CC)C(=O)NC1CCN(C(C)=O)CC1C)NC(Cc1cn(CC)nn1)=O 25696,C1(N(C(=O)CCNC(=O)C(C)(C)C)CC)CCc2ccccc2NC1=O 25697,N1(C(C=NOC)=O)CC2CCC1C1CN(C(=O)CCn3cc[nH]c(=O)c3=O)CC21 25698,CN1C(=O)NCC1C(=O)NC(C1CCCC1)CNC(=O)C=CC1CCOC1 25699,C#CCCC(O)C(=O)N(C1CN(C(=O)C2=CSCCO2)C1)C 25700,O(P(=O)(CCCNC(=O)C(n1cc(C2(OC)CNOC2)nn1)C)OCC)CC 25701,Nc1nccnc1C(=O)NC1CC1NC(C1COCC1Cc1ccccc1)=O 25702,CC1C(NC(C2CN(C)C(=O)N2)=O)CC2CCC1N2C(c1ccsc1C(F)F)=O 25703,c1(C(N(C2CCN(C(CCc3cc(C)nn3C)=O)C2)C)=O)ccc(F)c(F)c1 25704,c1(C(N(C2CCN(C(c3scc(C)c3)=O)CC2)CCO)=O)ccn2ncccc12 25705,C12CC3CCC1(C3)C(=O)N2.C(F)(F)(C(F)(F)F)c1cc(NCC=CCSC)no1 25706,N1(CCC(=O)NCC2(C(=O)NOCC3CCOC3)CCCO2)CCCCC1 25707,C(COCc1ccccc1)(C(=O)N1CC(c2noc(C(F)F)n2)C1)N(C)C 25708,N1(C(CN(C(C(C)OCC2CC2)=O)C2CCC2)=O)CCC(O)C(C)(C)C1 25709,c1(C(N2CCCC(F)(CNC(c3ccncc3F)=O)C2)=O)cccc2nn[nH]c12 25710,Cc1nc(C(=O)NCC(c2ccccc2F)NC(=O)C=CC2CCCC2)c(C)s1 25711,N1(C(C=C(C)C2CC2)=O)CCOC(C)(CNC(=O)C(c2ccc(Cl)s2)=O)C1 25712,N1(C(c2cccc(I)c2)C(=O)NCCOC)CCCC(O)(c2ccccc2)CC1 25713,n1(CC)ncc2cc(C(=O)NC(CNC(c3nocc3Cl)=O)CC(C)C)cnc12 25714,c1(-c2nc(C(CC)CC)nn2Cc2cccs2)cnc2n1CCCCC2 25715,C(CCC(C)(C)C(=O)NCC1CCC2(CCC2)C1)NC(COCCOCC#C)=O 25716,C#CCCCCC(=O)N1CCC(CO)C(NC(c2cccnc2C)=O)C1 25717,C1(CC(=O)O)CCN(CC(c2ccccc2Br)O)C2(CC2)C1 25718,CCCC(C(=O)NCc1cc(C)ns1)NC(=O)CC1CCOC1(C)C 25719,C1(CCN2CCCC(O)C2)CC(C(=O)NC(C2(C)CCCC2)=O)=CC1O 25720,CCCC(CCC)CC(=O)NC(C(=O)NCCCC1CCOC1)c1ccco1 25721,c1(C(=O)NC2CN(C(C(CCC)N(C)C)=O)C2)nc2ccccc2[nH]1 25722,c1(C(=O)Nc2cc(C(=O)OC)c(C)nc2)cc2c(=O)n(C)c(=O)n(C)c2s1 25723,N1(C(C(CCSC)O)=O)CC(NC(c2ccc(C)s2)=O)C(C2CC2)C1 25724,c1(C(=O)NCC2C(C)(C)C(NC(=O)Cc3cc(Cl)cs3)C2)ccc2c(c1)CC2 25725,C1(CNC(C(C(C)O)C)=O)(CO)CCN(C(=O)CCCc2cnn[nH]2)CC1 25726,N1(C(CCC2C(C)(C)C2)=O)CCC(OCCNC(c2cocc2Br)=O)C1 25727,C1(NC(C2CC(C)CC(C)C2)=O)CCOC12CCN(C(=O)OC(C)(C)C)CC2 25728,C1(C(=O)O)CN(C(c2cnco2)=O)C2(CCC2)C1.C1CN1 25729,c1(C(=O)NCCC2(CNC(C3(O)C(C)(C)C3)=O)CC2)cccc(OC(F)F)n1 25730,C(CCN=c1[nH]c(=NCC2COC(C)(C)CO2)[nH]c2c1CSC2)NC(C)=O 25731,c1(C(N(CC)CC2CCCN2C(c2occc2F)=O)=O)[nH]c(O)nc1C 25732,c1(N(C)CC2(C)CC2)nc(=NCC2(C)CCC(=O)N2C)[nH]c2c1CSC2 25733,c1(C(N(CC(CC)NC(=O)CSC(F)F)C)=O)ccc(-c2ccncc2)s1 25734,c1(C(N2CCC(CNC(C(=C(C)C3CC3)F)=O)C2)=O)cn2cnnc2cn1 25735,C(=O)(C(CCC=C)NC(c1cc(C)cc(O)c1)=O)NC(CC#C)C(=O)NC 25736,N1(CC2(CNC(C(C)(C3CC3)OC)=O)CC2)CCC(NC(=O)C=CCF)CC1 25737,Cc1nc2c(C(=O)NCC3CCCN3C(=O)C=Cc3sccc3C)cccc2o1 25738,c1(CC(=O)OC2CCCN(c3cccc(F)c3)C2=O)ncc(F)cc1F 25739,c1(CC2N(CCC(=O)OC)CCC2C)ncc(C)cc1Cl 25740,Cc1cccc(C(C(C)C)NC(c2cccc(C(N)=O)c2)=O)c1 25741,C1(CNC(C(C)NC(=O)C2CC2)=O)CN(C(c2ccccn2)=O)CC1(F)F 25742,N1(C(CCC)=O)CCCC2(CCN(C(=O)C=Cc3ccc(N(C)C)cc3)CC2)C1 25743,CCCCC(C(=O)Nn1cnnc1C)NC(c1ccc(C#N)c(C)n1)=O 25744,CC1=C(C(=O)NC(CCN(C(=O)CC2CCCC23CC3)C)C(C)(C)C)CCO1 25745,CC1CCN(C(c2cc(Cl)nnc2O)=O)CCN1C(C1C2CCC1CC2)=O 25746,N1(C(C(C)NS(C)(=O)=O)=O)CCCC(O)(CNC(=O)CCn2ccnn2)C1 25747,N1(C(C(=Cc2cccnc2)C)=O)CC(NC(=O)CCCNC(N)=O)CCC1C 25748,C(=O)(C(O)CC(C)(C)C)NC1(NCCNC(CCCOC(C)=O)=O)CCCSC1 25749,Cn1cc2c(C(=O)NC3CCCN(C(=O)CCc4nc(=N)[nH][nH]4)C3)cccc2n1 25750,CC1CC(CCNC(c2cccs2)CO)C1 25751,CC1CCc2[nH]c3c(C(C)NCC4CC4c4ccsc4)cccc3c2C1 25752,c1(SC)ccc(C=CC(=O)NCC2CC2CNC(=O)CCOC2CC2)s1.C(C)(=O)NCC 25753,S(=O)(=O)(c1ccc(Nc2cn(C)nc2OC)nc1)NC1CCC(NC)C1 25754,n1(CC(=O)OC(CNC(C(C)OCC)=O)C)cc(Cn2ccnc2)nn1 25755,N1(C(C)C)C(=O)CCC1C(=O)NCC1C2CC1N(C(=O)COC1(C)CCCC1)C2 25756,Cc1nc2ccsc2c(=NCCOC(=O)Cc2ccc(F)cc2)[nH]1 25757,C1(C(=O)NCCOC(C)C)(CNC(C2CC(OC)C2)=O)CCCCC1 25758,N1(Cc2cccc(C#N)n2)Cc2ccc(NC(C3CC(O)CN3)=O)cc2C1 25759,C1(N(C(C(C(=C)C)(C)C)=O)C)CC2CCC(C1)N2C(=O)C1=CC2CCCC12 25760,CCC(CC)CCC(=O)N1CCOC(C(C)NC(=O)C#CC2CCC2)C1 25761,N1(C(C(N2CCC(c3nc(=N)[nH][nH]3)C2)=O)=O)CCC2(CC1)CC2CO 25762,N1(C(C(CC#C)NC(c2scnc2CC)=O)=O)CC2C3CCC(O3)C2C1 25763,C1(NC(C23OCC(CC)(C2)C3)=O)CCN(C(c2cc(Cl)c(Cl)s2)=O)CC1F 25764,C1(C2CCC2)(SCC(C2CCCC2)OC)CC1 25765,C1(C(=O)NCCCC(C)NC(=O)Cc2cccc(F)c2)COCC2(CCC2)O1 25766,N1(C(c2c(C)sc(Cl)n2)=O)CCN(C(c2ncc[nH]2)=O)CC(O)C1 25767,N1(C(=O)CCC=Cc2ccccc2)CCN(C(=O)Cn2cnnc2)CC(O)C1 25768,c1(C(=O)Nc2cc(F)ccc2F)n[nH]c2c1CN(C(C1(F)CC1)=O)CC2 25769,C1(C(=O)NCc2cc(=N)[nH]cn2)(COC)Cc2ccccc2C1 25770,CCCCCC(C)CC(=O)NC1CN(C(=O)CN(C)S(=O)(=O)N(C)C)CC1O 25771,c1(C(N(C(CN(C(c2c(C)cccn2)=O)C)C)C)=O)ccc(F)c2occc12 25772,c1(C(C)=O)cc(C(N2CCC(F)(CNC(c3cnnn3C)=O)C2)=O)oc1C 25773,c12cncnc1C(=O)N2.N1(C(C2C(CC)CCO2)=O)CC2C(COC)C2C1 25774,C(CO)(CCCCNC(C1CC(F)C(=O)N1)=O)NC(c1coc(Cl)n1)=O 25775,N1(C(c2n(C)[nH]c(=N)c2)=O)CCCC1C1CCCCN1C(c1cc(=O)cc[nH]1)=O 25776,CCS(=O)CC(=O)NCCCC(C)(C)NC(=O)C(C)NC(c1ccoc1)=O 25777,CC1CN(C(=O)CCc2ncc[nH]2)CCCN1C(c1cncc(CO)c1)=O 25778,CN1CCN(c2nccc(=NCC3CC3(F)F)[nH]2)CC1(C)C 25779,c1(C(N2CC(C(C)NC(c3c(C)ccnc3O)=O)C2)=O)cccc2[nH]ccc12 25780,C(C)(c1ccc(OC)cc1)=CC(=O)N(C1CCCN(C(CC(CCC)O)=O)C1)C 25781,C1(c2ccc(C(=O)OCC)o2)CCN(Cc2cc(C(F)F)no2)CC1 25782,Cc1cc(C(=O)NCC2CCC(NC(c3csnn3)=O)CC2)cc(CC2CC2)n1 25783,c1(CC)cc(C(=O)NC2CC(NC(c3nn(C)cc3N)=O)CC2O)n(C)n1 25784,c1(C(=O)NCC(CC)NC(C2(c3ccsc3)CC2)=O)[nH]ncc1Cl 25785,N1(C(C2CC(=O)N(Cc3ccc(Cl)cc3)C2)=O)C2CCC1CC1(C2)CC1(F)F 25786,c1(C(N2C(CCNC(C3CC3C(C)(C)C)=O)CC(OC)C2)=O)cccc(O)c1Cl 25787,CCCS(=O)(=O)CC(=O)N(CC)CC1CCN(C(C2(F)CC2C)=O)CC1 25788,CC(C)CC(C(=O)NC1CC1CNC(=O)Cn1cc([N+](=O)[O-])cn1)C(C)C 25789,c1(C(=O)NC23C(CN(C(CSC)=O)C2)C3)c(Cl)oc2ccccc12 25790,C(=O)(CCCCCC#N)NC(C)CC(C)NC(c1cccc(OC(F)F)c1)=O 25791,C(=O)(C1=C(Cl)CCOC1)N1CCC(C(=O)NCC(CC)C(C)(F)F)C1 25792,C(=O)(CC(C)(C)O)N(CC(=O)NC(C)Cn1cncn1)CCOC 25793,CC1(C)CC(NC(=O)CCC2CCOCC2)CN1C(=O)CN1CCCCCC1 25794,N1(C(C(CCC)NC(N)=O)=O)CCN(C(c2cc(Br)cnc2C)=O)C(C)C1 25795,C1(C(C)NC(=O)C(=Cc2cn(C)cn2)F)CN(C(=O)C(O)C2CCC2)CCO1 25796,n1(CCC(=O)NCC2CC2NC(=O)CCC2CCCCC2)cnc([N+](=O)[O-])c1 25797,C1(C(C)NC(C(C)(C)OC)=O)CCCN(C(=O)CC(C)(F)F)C1 25798,C=CCCC(C(=O)NC(C(N)=O)C1CCCC1)NC(c1cc(Cl)n[nH]1)=O 25799,Cc1cc(C(=O)NCC(C)NC(C2CNC(=O)CC2(C)C)=O)c(Cl)cc1F 25800,c1(C(N2CC(CCNC(C(CCCC)C)=O)C(C)C2)=O)nccn2cc(C)nc12 25801,N1(N(C(c2cc(OC)cc(CC)c2)C(=O)NC2CC2)C)CC2C3C=CC(O3)C2C1 25802,C1(C2CN(C(c3nnc(C)s3)=O)C2)CN(C(c2coc(C(F)F)c2)=O)CCO1 25803,N1(C(c2cc(CCCC)oc2C)=O)CC2(C1)CN(C(=O)C(C)(C)CCC)C2 25804,C1(C)(NC(C(C2CN(C(c3cccc(CC)n3)=O)C2)OC)=O)CCCCC1C 25805,C1(NC(C(=Cc2ccncc2)C)=O)CS(=O)(=O)CC1NC(c1cnc[nH]1)=O 25806,Nc1cc(F)ccc1C(=O)NCC(O)CNC(C1CCC(CCO)CC1)=O 25807,C1(NC(c2c(CC)cno2)=O)C(C)CCN(C(c2nc(C)c(C)nc2C)=O)C1C 25808,CS(=O)(=O)CC(=O)NC1CCOC(C(=O)NOCC(=O)OC(C)(C)C)C1 25809,N1(C(CC(CC)(F)F)=O)Cc2nccn2CC(NC(=O)C(F)C(F)(F)F)C1 25810,c1(C(=O)NC2CCCCCN(C(C3C(=C)CC3)=O)C2)n[nH]c2cc(Br)ccc12 25811,Cn1cnc(I)c1C(N1CCC(c2nc[nH]n2)CC1)C(=O)NC1(C)CC1 25812,Cc1cncc(C=CC(=O)NC2(CNC(C3(CCO)CC3)=O)CCC2)c1 25813,Cc1[nH]nc(C(=O)N(C)CC2CN(C(c3ocnc3C(F)(F)F)=O)CCO2)c1F 25814,C(=O)(CCCC(C)O)NCC(C)(C)Nc1nccc(CC(=O)OC)n1 25815,N1(C(c2cc(COC)no2)=O)CC2CN(C(=O)C(C)CS(C)(=O)=O)CC2C1 25816,c1(C(=O)NCC2CC(C)(C)CN2C(=O)Cn2cnc(=N)[nH]2)cc2c[nH]cnc-2n1 25817,Cc1c(C(N2CCC2CNC(=O)C(F)CC(C)C)=O)sc2[nH]cnc(=S)c12 25818,c1(C(=O)NC(CN(C(c2c[nH]cc(Cl)c2=O)=O)CC)C)n[nH]c2cc(Cl)ccc12 25819,N1(C(CCOC)=O)CCC(NC(c2cc(C(C)C)n(C)n2)=O)C1c1ccccc1 25820,N1(C(C2C(C)C2C)=O)CC2CC1(CNC(=O)C(C)(C)c1nccs1)C2 25821,CC1CCn2cc(C(=O)NCC(CO)NC(c3c[nH]c(Br)c3)=O)nc2C1 25822,N1(C(c2ccc(CO)nc2)=O)CC=CC(C(N2C(CO)CCC2CO)=O)C1 25823,CCCCS(=O)(=O)CC(=O)NCCCN1CCN(C(=O)C2=CS(=O)CCC2)CC1 25824,C#Cc1ccc(C(=O)NC2CCN(C(c3c(C)ncn3C)=O)CC2O)c(OC)c1 25825,C1(CNC(C2CN(C(N)=O)C2)=O)CN(C(c2cc(F)ccc2Cl)=O)CC12CC2 25826,C1(C(N(CC(C)(C)N(C)C)C)=O)C2CC2CN1C(=O)C(C)OC1CCCC1 25827,C1(NC(c2ccn(C)n2)=O)CN(CC(C2CC(C(C)(C)C)=NO2)=O)CC2(CC2)C1 25828,N(C1COc2ccccc21)CCOC(C)C(=O)NC(CCSC)C(=O)N.CO 25829,c1(C(C)(C)C)cccc(C(c2nnnn2C2CCCC2)NCCc2cccs2)c1 25830,N1(C(C)C(=O)NC(=O)Nc2nccs2)CCCC(C(=O)Nc2cc(O)n(C)n2)C1 25831,N1(C(=O)NCCc2c(C)ncs2)CCCC(NCCO)C1 25832,C(C)(C)(C#Cc1cn(-c2ccncc2OCC)nn1)NC(C(CC)CC(C)C)=O 25833,C(C)(CCCCNC(C12CC(C)(C1)C2)=O)NC(c1c(C)ocn1)=O 25834,C1(C(N(C)CCNC(c2sncc2Br)=O)=O)CN2CCC1CC2 25835,c1(NC(C2N(C(c3ccc(C)c(F)c3)=O)CC2)=O)cc(F)c(O)cc1C 25836,Cc1ccccc1C1(C(N2CC(O)(C(C)NC(c3nn[nH]c3Cl)=O)C2)=O)CC1 25837,C1(C(=O)NC2(CNC(CCSCC(N)=O)=O)CCCC2)CCOC(C(F)(F)F)C1 25838,N1(C(CCCS(C)(=O)=O)=O)CCC2(CC1)CCN(c1ncns1)C2 25839,c1(C(=O)NC(C2CN(C(=O)CCCCC(N)=O)CCO2)C)cc(Cl)c(F)cc1F 25840,c1(NC(C(C)(C)CCl)=O)ccn2c(C(F)(F)F)nnc2c1 25841,c1(C(=O)NC2CCCCN(C(CC(=C=C)C)=O)C2)c(F)cc(O)cc1F 25842,c1(C(N(CC(CC)NC(=O)C2=CC(C)(C)C2)CC)=O)ccc2c(c1)C(=O)NC2=O 25843,c1(OCCC(=O)NC2(CC=C)CCN(C(C3C=CCC3)=O)C2)cc(Cl)ccc1Cl 25844,N1(C(CCNC2C3(CC(N)C3)C2)=O)CC(=O)Nc2ccccc21 25845,c1(CC)nn(C)cc1C(=O)NCC=C1CCN(C(C2(OC)CCCC2)=O)CC1 25846,c1(OC)ccc(F)c(C(=O)NC2CC3(C2)CC3NC(c2nccc(C)n2)=O)c1 25847,C1(NC(CCc2c(C)noc2)=O)CC(C)N(c2nc(-c3ccccc3)ns2)C1 25848,N1(C(C2C(OC)CN(C(=O)CCC(C)C)C2)=O)CC(O)C(O)C1CO 25849,S(=O)(=O)(c1ccccc1F)NCC(=O)NC(CNC(CCCCNC(C)=O)=O)C 25850,c1(C(=O)NC(CNC(C(C)C2CC2)=O)(C)C2CCC2)cc(-c2cnn(C)c2)on1 25851,c1(NC(=O)Nc2cc(C)c(F)c(Cl)c2)ccc(S(=O)(=O)NC(C)(C)C)cc1 25852,C1(C(=O)NCC(CC)(C)C)CN(C(c2ccc(O)nc2C)=O)CC1(C)C 25853,C1(NC(CCCC2(C)N=N2)=O)CCN(CC2CCC(C(=O)NO)CC2)CC1CO 25854,C(C(C)(C)C(C)(C)O)NC(C1N(C(C(C)=CCC)=O)CCC=C1)=O 25855,N1(C(c2nnn(C)n2)=O)C2CCC1CC(NC(=O)CCC1CC1)C2 25856,C(=O)(C1CCc2nccn21)NCCCCCCC(=O)N1CC2CC(N(C)C)C2C1 25857,C12(CNC(c3cc4ccncc4[nH]3)=O)CCC(CN(C(c3ccns3)=O)C1)C2 25858,C1(CNC(c2cc(C(C)C)no2)=O)CC(C)CN(C(=O)C(CO)N(C)C)C1 25859,c1(OCC)c(O)ccnc1NC(c1ccccc1)C(F)F 25860,c1(C(=O)NC(C)C(C)NC(=O)C(N)=O)cc2occc2s1 25861,C(=O)(C(CO)C(C)(C)C)N(C(CNC(CCCC=C)=O)C1CC1)C 25862,c1(OC)ccc(C(N2CC(F)CC2C(=O)Nc2ccnc(Br)c2)=O)c(Br)n1 25863,C=CC(CCC)CC(=O)N1CC2C(CNC(c3cc(C4CCCC4)[nH]n3)=O)C2C1 25864,C(C(O)CC(=O)NCC1(O)CCC1)NC(CNC(CC(C)C)=O)=O 25865,N#Cc1cnccc1N1CCCC1CNC(C1(CN2CCCC2)CC1)=O 25866,c1(C(=O)NCC2C(C)CN2C(=O)CC2OCCC2(C)C)cc2ccccn2c1 25867,c1(C(=O)OC)c[nH]c(=NC(CNC(=O)Cc2cnnn2C)C(C)C)cn1 25868,Cc1oc(S(C)(=O)=O)cc1C(=O)NC(C(C)NC(c1ccc(F)s1)=O)C(C)C 25869,N1(C(=O)CCc2cc(F)ccn2)CCC2C1CCN2C(C12CC(CO)(C1)C2)=O 25870,c1(NC(c2c(CC)cc(Br)cc2)=O)ccc(S(=O)(=O)N2CCOCC2)cc1 25871,CC(C)CC(CNC(=O)C1=C(Cl)CCC1)C(=O)N(C1CCCC(O)C1)C 25872,Cc1ccc2[nH]c(=NC(C)C3CCN(C(C4CCC=CCCC4)=O)CC3)sc2n1 25873,c1(CNC(c2c(CC)onc2)=O)cccc2c1CN(C(=O)COCP(C)(C)=O)C2 25874,N1(C(Cc2cc(C)cc(Cl)c2)=O)CCCc2c(O)cccc21 25875,C(=O)(CS(=O)(=O)CC1CCCO1)N1CCC(N(C(=O)CCCc2cccs2)C)C1 25876,c1(SC)ccc(C)c(C(N2CCCCC2CCN(C)C(c2nnc(C)s2)=O)=O)c1 25877,N1(C(C(C)OC(C)C)=O)CCN(CC(=O)Nc2scnc2Br)C(=O)C1 25878,Cc1ncc(CC(=O)NCC(C(C)C)NC(=O)C(C)CSC(F)(F)F)[nH]1 25879,c1(C(=O)Nc2cc(-n3cc(CC(O)CO)nn3)ccn2)c(F)cccc1Br 25880,N1(CC(=O)NC(C)CCN(C(=O)C(=O)C(C)(C)C)C)C(=O)c2ccccc2C1=O 25881,c1(NC(C2CCCC(NC(c3cccc(F)n3)=O)C2)=O)cc(Cl)ncc1[N+](=O)[O-] 25882,c1(C(N2CC(C)(C)C(NC(=O)Cc3nc(=N)[nH][nH]3)C2)=O)ncnc2c1CCCC2 25883,CCCC(C)(C)CC(=O)NC(C1(O)CN(C(c2ccsc2SC)=O)C1)C 25884,Cc1ccc2cc(C(=O)NC3CCCN(C(c4ccn(C)c4)=O)C3)nn2c1 25885,C1(OC)CN(C(=O)CC2(O)CCOCC2)CC1NC(C1(n2nccn2)CC1)=O 25886,c1(C(=O)NC2C(NC(CC(CC)C(C)C)=O)CC2)c[nH]c2cccc(Cl)c12 25887,CN1CC2C(c3ccc(Cl)s3)CCCN2C(=O)NC1=O 25888,c1(C(N(C2(C(=O)NCC(COCC)O)CC2)C)=O)sccc1Cl 25889,c1(C(N(CC(CN(C)C)O)C)=O)sccc1CNC(c1cnn(C2CC2)c1)=O 25890,C1(NC(CN(C(=O)CC(C)n2cccc2)CCC)=O)CC12CCOCC2 25891,c1(NCc2ccc([N+](=O)[O-])o2)ccc(S(=O)(=O)NC2CCN(CCF)C2)cn1 25892,c1(C(=O)NC(CCN(C(C(C)CC(N)=O)=O)C)C(C)(C)C)ccc2occc2c1 25893,CN1CC2CCC(NC(c3ccc(-c4ccc(C(N)=O)o4)cc3)=O)C2C1 25894,c1(C(C(=O)NCC(C)CN(C(=O)CCC2(C#N)CCC2)C)O)cnn(C)c1 25895,c1(C(=O)NC2CCCC(CNC(C(C)(F)F)=O)C2)ncc(C(N)=O)cc1Cl 25896,c1(C2C(C(N3C(CN(C(C4CCC(CC)O4)=O)C)CCC3)=O)C2)cccc(C)c1 25897,N1(C(c2ncc(OCC)nc2)=O)CC2CN(C(=O)CCc3cccc(C)n3)C2C1 25898,c1(CN(C2CC(C)C2)CCC(=O)N2CC(OC(C)=O)C2)c(C(F)(F)F)cnn1C 25899,CCCC(C(=O)NC(C(=O)N1CCC(CC2CCC2)C1)C(C)OC)OCC 25900,C1(CN(C(C2(COC)CCOC2)=O)C)CCN(C(=O)CC(C)c2ccco2)CC1 25901,Brc1cc(I)c(CNCc2nc(C3CCCCO3)n[nH]2)s1 25902,n1(CC(N2C(CC(=O)NCc3nccs3)CC2)=O)ccc2ccccc12 25903,N1(C(CSc2cc(C)sc2C)=O)CC(NC(c2nc(C)n(C)n2)=O)C(C)(C)C1 25904,c1(C(=O)NC(CCSC)C)ccc(NCCC(F)(F)Cl)cc1 25905,Cc1nc(O)nc(C)c1CC(N1CC(C)C(C)(CNC(c2cnsc2C)=O)C1)=O 25906,c1(NC(N2CCOC(C3CC3)C2)=O)ccc(N2CCCCC2)cc1N1CCOC1=O 25907,Cc1nnc(CC(N2CC(NC(c3cnc(C)s3)=O)C2)=O)o1 25908,CC(Cc1cnc[nH]1)N=c1[nH]c(N(C)Cc2ccc(Br)c(F)c2)nc2ccsc12 25909,Cc1cccc(C(=O)NC2CC(O)CN(C(=O)CN3CCC(C)(C)CC3)C2)c1C 25910,N1(C(c2n(C)ccn2)=O)CC2(CC(NC(C3(C(F)F)CC3)=O)CO2)C1 25911,CC1CCc2sc(C(N3CCC(CNC(c4csc(Cl)c4)=O)C3)=O)cc2C1 25912,c1(C(N2CCC3C(CCN3C(C3C=CCN3)=O)C2)=O)c(Cl)ccc2c1OCO2 25913,c1(CNC2CCC(C(=O)NCc3cn[nH]c3)C2)ccccc1C(F)(F)F 25914,C(CC(C)(C)C)(C(=O)NC(C)C(=O)Nc1cc(C)c(F)c(C)c1)OC 25915,c1(NC)ccccc1C(=O)N(CC(C)NC(=O)CCC1CCCN1C=O)C 25916,C(C(C)(F)C(C)(C)F)NC(CCCN(C(c1n(CC)c(O)nc1)=O)C)=O 25917,C1(CC=C)(NC(c2cocn2)=O)CC2CCC(C1)N2C(=O)CCN1CCCC1 25918,N1(Cc2nc(C#C)sc2)CCCN(C(=O)Cc2ccccc2)CC1 25919,N(C1CN(C(c2cncn2C2CC2)=O)Cc2ccccc21)C(CSCC#C)=O 25920,C(=O)(C(C(C)(C)C)NC(C1CN(C(c2ccc(C)c(F)c2)=O)CC1(F)F)=O)NC 25921,C(C(C)(C)CN(CC(CO)OCC)C)NC(c1nnn(-c2ccccc2)n1)=O 25922,c1(OC)cncc(C=CC(=O)NC2(CN(C(=O)CN3CCCC3C)C)CC2)c1 25923,Cc1cc(C(=O)NC2CCCC2NC(c2ccnc(O)c2)=O)nc(O)n1 25924,c1(C(N2CCC(n3ccnc3)C2)C(=O)NCC)ccc(Oc2ccccc2)nc1 25925,c1(CC)cc(C(=O)NCC(CC)NC(C2CCCCC2(C)C)=O)ccc1OC 25926,c1(C(N2CC(C(=O)Nc3cc(Br)cc(Br)c3)C(O)CC2)=O)cccc2c1CCC2 25927,CCC(CCC(=O)NCC(CC(=O)NCC(C)(CC)CO)C1CCC1)OC 25928,C1(CNC(CC2CCN(C)C2=O)=O)CCCN(C(C2(CC(F)(F)F)CC2)=O)CC1 25929,C(C1=CCN(C(C2CCC(F)CC2)=O)CC1)NC(C(C)C1CCCO1)=O 25930,C(=O)(CCCCCCCCN(C)C)NCC(C)NC(c1cc(C(F)(F)F)no1)=O 25931,c1(OC)cc(OC)c2c(c1)CCN(C(=O)C(C)Sc1cc(Cl)cc(Cl)c1)C2(C)C 25932,c1(SC)ncc(N)c(C(N2CC(NC(=O)Cn3cc(C4CC4)cn3)C(F)C2)=O)n1 25933,CCCCCCCCCCCCN(C(=O)CC1CCN1C(=O)OC(C)(C)C)C 25934,c1(C(N(C2C(C)CCC2)CCc2ccccc2)=O)cn2c(n1)CCCC2 25935,CC(C)(CNC(C1CCS1(=O)=O)=O)C(=O)NOCC=CCl 25936,c1(CC(=O)NC2CN(C(C(F)=CCC)=O)C2)ccc2c(c1)CCOC2 25937,C1(CNC(CCc2onc(C(C)C)n2)=O)CN(C(=O)C=CS(C)=O)CC(C)(C)O1 25938,c1(C(=O)NC2C(CNC(=O)CCOC3COC3)C2)cccc(=O)o1 25939,C1(C(=O)NC(C2CC(NC(C3COCCC3(F)F)=O)C2)C)CC2(C1)OCCO2 25940,c1(C(N2CCC(N(C(=O)CCc3cccnc3C)CC)C2)=O)cc(C)ccc1N 25941,C12(C(=O)NC3CCCN(C(C(CSC)OC)=O)C3)C3C4C1C1C2C3C41C(N)=O 25942,C1(NC(Cc2c(C)ncs2)=O)C2CC3C(C2)C13C(=O)NCCC1CC=CCC1 25943,c1(C(N2CC3(C)C(CC2)C3(F)F)=O)cc2c(nc1O)CCC(C(C)C)C2 25944,CCC(C)(CNC(=O)C=Cc1ccccc1)C(=O)NC(C)Cc1ccco1 25945,C(=O)(CS(=O)(=O)CC(=O)NCC1CCN1C(=O)Cn1nc(C)nc1C)OC 25946,C(C(C)(C)C#CC(=O)N1CC(O)(C(F)(F)F)C1)NC(C(CC#C)C1CC1)=O 25947,CC1(C)CN(C(=O)C=Cc2cncs2)CC(CNC(=O)C(F)(F)CC2CC2)O1 25948,N1(C(CC2(C)CCOCC2)=O)CC2CC(NC(=O)CCN3CCOCC3)C(C2)C1 25949,Cn1cnc2c(N3CCCCC(NC(=O)Cc4cnoc4)C3)nc(Cl)nc12 25950,Cc1nc[nH]c1CC(=O)NCC1CCC1NC(=O)Cc1csc(NS(C)(=O)=O)n1 25951,C(=O)(C(=O)N=c1cc(C)o[nH]1)NCC1C(F)(F)CCN(C(C(C)SCC)=O)C1 25952,c1(C(=O)NCCC(CCC)C)cc(C(N)=O)cc([N+](=O)[O-])c1 25953,Cc1nn2ccccc2c1C(=O)NC(CNC(C1CC1C(N)=O)=O)CC(F)(F)F 25954,N1(C(c2cc(OC)ns2)=O)CC(NC(=O)Cn2cnc(C#N)n2)C2CCCC2C1 25955,C(=O)(C(CNC(c1ncncc1Cl)=O)CC1CCCC1)NCCOCC(C)C 25956,N1(C(c2ccc(N)c(O)c2)=O)CC(NC(c2cc(Cl)c(Cl)s2)=O)CC12CCC2 25957,c1(OCCNC(=O)CC(O)c2ccccc2)ccccc1Sc1ccc(F)cc1 25958,C12(CNC(=O)C(C3CC3)C3CC3)CCCC1N(C(=O)Cn1cnnc1)CCC2 25959,Cc1nc(N(C)CCN(C(=O)CC2NC(=O)NC2=O)C)c(C)c(Cl)n1 25960,C1(C(C)(C)O)(CNC(c2ccnn2CC(F)F)=O)CN(C(c2ccccc2)=O)C1 25961,c1(C(N(C)CC2CC(F)CN2C(=O)C(F)=C2CCCC2)=O)cc(N)ccc1O 25962,c1(CCC(N2CCC(CN(C(C3C(C)OCCO3)=O)C)C2)=O)ccc(C#N)cc1 25963,c1(C(CC(=O)NC2CC(F)(CNC(c3c(SC)ccs3)=O)C2)O)ccc(Cl)cc1 25964,C1(C(N2CCOC(c3cn[nH]c3)C2)C(=O)NCC(=C)C)CC(C)(C)OC(C)(C)C1 25965,c1(CC(=O)NC(CNC(COCCOCC)=O)(C)C2CCC2)coc(C(F)F)n1 25966,C1(C(N(CC(=C)C)CC)=O)CCN(C(c2cnn(C)c2Cl)=O)C1(C)C 25967,CC(C)S(=O)(=O)C1CCN(C(CCCCC#N)c2nnnn2CC2CC2)CC1 25968,C1(CCNC(C2CCN2C2CCCC2)=O)CSCCN1C(C1CCC(F)(F)C1)=O 25969,C1(NC(C2(C#C)CCN(C(c3cc(CC)nn3C)=O)C2)=O)CC2C(O)C(O)CC12 25970,c1(C(N2CC(C)C(CC(=O)NC3COC4(CCC4)C3)C2)=O)coc2c1COC2 25971,c1(C2(C(=O)NCCCCN(C(C(c3ccc(C)s3)C)=O)C)CC2)cccc(F)c1 25972,N1(C(C(Br)=C(C)C)=O)CCC2(CCN(C(c3ccc4nc[nH]c4c3F)=O)C2)C1 25973,N1(C(c2scc(CNC(C3CN(C)C3)=O)c2)=O)CCCC2CC12.OC 25974,N1(C(c2c(OC)cccn2)=O)CCC2CN(C(c3ccnc(C)c3N)=O)C(C)C12 25975,C(C)(C(=O)NOC(C)C(=O)OC)NC(c1c(CCC)[nH]cc1)=O 25976,C=CCCCCCCCC(=O)N(CC(CC)NC(c1ncc(OC)cn1)=O)C 25977,c1(C(N2CCC3CN(C(C(F)=CCC)=O)CC3C2)=O)n[nH]c2c1CC(C)OC2C 25978,C1(NC(C(C(C)C)N(C)C)=O)CN(C(=O)C=CBr)CC1C1CC1 25979,C(=O)(C(C)(C)C(F)F)NC(C(C(C)C)Nc1ncc(F)cn1)C 25980,c1(NCC2CCN(CC#N)C2)cc(=NCc2ccc(-n3ccnc3)cc2)[nH]cn1 25981,C1(C#N)(C(N2C(CNC(C3(C)CC4CC4C3)=O)CCCC2)=O)CC(F)(F)C1 25982,c1(CNC(C(C)OCCCC)=O)cnn(C)c1CN(C(C1(N(C)C)CCC1)=O)CCC 25983,c1(C(=O)NCC(C)CNC(c2cc(N)cnc2Cl)=O)ccc2cnn(C)c2c1 25984,C12(NC(c3cc4c(O)nnn4cn3)=O)CC(CO)(C1)OC21COC1 25985,N1(CC)CC2(C1)SCCC2N=c1[nH]c(=N)[nH]c(=NC(C)c2ccc(F)c(F)c2)[nH]1 25986,c1(C(=O)NCC(CNC(C2C(C=C)OCCC2)=O)C)cc(F)cc2nn[nH]c12 25987,C(C1=NOC2CN(C(=O)CC3CC3)CC12)NC(c1cc(CC)c(C)cc1)=O 25988,C=CC(CC(=O)NCCCCNC(C1CC1OCC)=O)c1ccccc1 25989,N1(C(C(CN(C)C)(C)C)=O)CCC(C2CC2)(CNC(=O)CCCC2CCCO2)C1 25990,c1(C(C(C)(C)C)N(C)C)nc(-c2cncnc2)nn1-c1ccccc1 25991,C1(NC(c2cnc(CC)o2)=O)CCCN(C(C2(c3cccs3)CC2)=O)CC1F 25992,Cc1nc(NC(C2CCCN2Cc2ccncc2O)=O)cnc1Cl 25993,C1(C(N(CCCNC(C2CCCCC2C(N)=O)=O)CC)=O)CCC(C)(C)CO1 25994,N1(C(C(CCNC(C(CC)NC(C)=O)=O)O)=O)CC(O)CC12CCOC2 25995,N1(C(CC2(C)CCOC2)=O)CC2CC1CC2CNC(=O)CCC1CCCOC1 25996,C1(NC(COC)C(=O)OC)CN(C(=O)OC(C)(C)C)CC2(CC2)C1 25997,O=C(C#Cc1ccc(Cl)cc1)N1CCN(CCNCc2cc(F)c(Cl)cc2Cl)CC1 25998,N1(C(=O)CN2CSCC2=O)CC(NC2(CC(F)(F)F)CC2)CC12CCOCC2 25999,c1(C(=O)NCCCC(C)(C)NC(=O)CC2CCOCC2)ccc2nonc2c1 26000,c1(N2CC(C)C=C(C)C2)nc(NCCc2c[nH]nc2C2CC2)c2ccsc2n1 26001,C(=O)(CC(CNC(=O)C(C)OCC1CCCC1)OC)N1C(C=C)CC1 26002,N1(C(CC2(OCC)CCC2)=O)CC(C(=O)N(C2CCOC(C)C2)C)C2(CC2)C1 26003,C(CN=c1[nH]c(=NC2CC2C(C)(C)C)c2ccccc2[nH]1)c1c(C)nc(C)s1 26004,N1(C(=O)OC(C)(C)C)CC=C(CO)CC1.c12c[nH]nc1NC2=O 26005,C1(CC)C(NC(c2cc(O)nc(Cl)c2)=O)CCCN1C(=O)CCS(N)(=O)=O 26006,c1(NCC(CCC)(F)F)ccc(Cl)cc1N1CCN(C)CC1 26007,CN1CCCCC(C(N2CC=CC(NC(c3csc(C(F)(F)F)c3)=O)C2)=O)C1=O 26008,CCCC(CC(C)C)C(=O)NOC(CC(C)C)C(=O)N1CC(CO)C2(CC2)C1 26009,CCC(C)C(=O)NNC(=O)c1nnn(C)c1-c1ccc(N(C)C)c(C)c1 26010,N1(C(C2C(CC)OCC2)=O)CC(OC)C(NC(=O)CC23CCCC2C3)C1 26011,c1(CC(C(=O)N(CCCN(C)C(c2ocnc2C2CC2)=O)C)O)ccccc1Cl 26012,N1(C(c2ccc(F)cc2F)=O)CC2CC1CCC2NC(C1(CO)CCCC1)=O 26013,C=CC1CCCN1C(=O)CC(N1CCN(C(=O)OC(C)(C)C)CC1)C1CC1 26014,C(=O)(CCC(C)(C)C#N)NCCCC(C)NC(C(C)(CO)OC)=O 26015,N12CC3C(C3C1)C(=O)OC2=O.C1(O)(CN(c2ccccc2)C(C)(C)C)CCCCC1 26016,c1(C(=O)NC(C(=O)NC)C(C)C)cc(C(F)(F)F)ncc1Br 26017,c1(CC(N2C(CNC(c3c(C)nco3)=O)CCCC2)=O)cc2ccccc2s1 26018,Cc1ccc(C(N2CCOCC2CC(=O)NCC2COCCO2)=O)nc1O 26019,c1(CC(N2C3C(NC(C4CC(C)SCC4)=O)C(C3)C2)=O)ccccc1[N+](=O)[O-] 26020,C(=O)(C(CC(C)C)ONC(C1CC2C=CC1CC2)=O)NCCC(CC)O 26021,C1(CC(=O)NCCN(C(=O)C=C=C(C)C)CCOC)CCCCN1C 26022,[N-]=[N+]=NC1CCCCC1C(=O)NCC1CC(F)(F)CN1C(=O)CC1C=CCC1 26023,CCCCCC(O)CC(=O)NCC1CC(NC(=O)C2=CCCC2(C)C)C1 26024,C1(C(=O)NC2(CNC(=O)Cc3ccccc3F)CC2)CC2C=CCC(C1)C2 26025,c1(C(C(=O)NC2C(NC(C(c3ccc(Cl)cc3)C)=O)C2)(C)C)ccc(O)cc1 26026,c1(N2CCC(CC)(CO)C2)nc(N2CCCC(F)(F)CC2)nc2ccc(Cl)cc12 26027,C1(C(N2CC(CCCCC)C2)=O)CCCC(NC(C2(F)CC=CCC2)=O)CC1 26028,c1(CC)ccc(F)cc1C(=O)NCC12CCC(C1)N(C(C1(CCO)CC1)=O)C2 26029,CN1CC2CCC(C1)N2C(C1CCC(O)CN1C(=O)C1=C(Cl)CCOC1)=O 26030,CC1=C(C(=O)N2CCC(N(C)C(C3CCC(N(C)C)C3)=O)C2)CCCO1 26031,N1(C(Cn2c(C)cc(C)n2)=O)CCOC2CN(C(c3nocc3Cl)=O)CC12 26032,c1(CC(=O)NCC(CC)(C)NC(c2ncoc2C)=O)cc(Br)ccc1F 26033,c1(C(=O)NC2CC(C)(CNC(C(CC)C)=O)C2)[nH]c(C2CC2)nc1C 26034,C(=O)(CC(C)(C)CC)N1CCC(CC=C)(NC(C2CCN(C3CC3)C2=O)=O)C1 26035,c1(CC)ncc(S(=O)(=O)NC2(c3nnnn3C)CC(C)N(C)C2)s1 26036,N1(C(Cc2ccc(C)cc2)=O)CCCC(NC(=O)Cn2cnnc2)CC1 26037,C1(CNC(C(C)NC(N)=O)=O)(CO)CCN(C(=O)C=CCF)CC1 26038,Cc1cc(C2CCN(S(=O)(=O)CCC(O)COc3ccccc3C)C2)cc(C)c1 26039,N1(Cc2occ(C)c2)CCOCC12CN(C(=O)OC(C)(C)C)C2 26040,c1(NC(C2(F)CN(C(c3ccc(C)c(O)c3)=O)C2)=O)c(Br)cccc1[N+](=O)[O-] 26041,N1(Cc2cc(C)c(F)nc2)CCN(C(c2cc(F)ncc2Br)=O)C(C#N)C1 26042,c1(OC)cc(C(=O)OC2CCCN(C(N3CCCCC3=O)=O)C2)cc(Br)c1 26043,N1(C(C2(C)N(C)CC(OC)C2)=O)CCCC(C2CC2NC(c2scnc2C)=O)C1 26044,N1(S(=O)(=O)CCc2ccccc2)C2CN(c3ccncn3)CC12 26045,N1(C(C2CC(NC(C3(C)CCNC3=O)=O)C2)=O)CC(O)C(C2CC2)C1 26046,N1(C(CCC#C)=O)CC2(CCCCN(C(=O)C(C)C3CCCO3)C2)C1 26047,N1(C(c2c(CC)occ2C)=O)CCCCC(NC(=O)C(C(C)(C)C)N(C)C)C1 26048,Cc1cnc(C=CC(=O)NC2COCC2NC(=O)CC2COCC2O)[nH]1 26049,c1(OC)cc(C)ccc1C(=O)NC(C1CCN(C(=O)CC=CC(C)(C)C)C1)(C)C 26050,N1(C(CC2C(OC)CC2)=O)CCN(C(c2cocn2)=O)C(c2ncc[nH]2)C1 26051,C1(CNC(C2(C(C)C)CC2)=O)CCC2(CN(C(=O)Cn3ccnn3)C2)O1 26052,C(=O)(C1CCc2c[nH]nc21)NC1(C(=O)NC(C2CCCCC2)C)CSC1 26053,N1(C(CCC#CC)=O)CCCC(C(=O)N(C)CC2CCOC2)CC1 26054,c1(C(C(=O)NCC2N(C(C)=O)CCCC2)=O)cc(S(N)(=O)=O)cn1C 26055,Cc1[nH]nc(C(=O)NCC2CCCN(C(C3CC3C)=O)C2)c1C 26056,C1(CCC)CN(C(=O)C(C)CN2CCCCC2)CCN1C(=O)C(C)C#N 26057,c1(C(=O)NCCCCN(C)C(C2CC2c2cccs2)=O)c[nH]nc1C(C)(F)F 26058,N1(C(Cc2cnc(C)o2)=O)CCCC2(NC(=O)CSc3nccn3C)CC2C1 26059,c1(C(N2CCN(C(c3ccn(CC)c3C)=O)C(C)C2)=O)nc[nH]c2ncnc1-2 26060,N1(C(Cn2c(N)cc(C)n2)=O)CCCC(N(C)C(c2ccccc2O)=O)CC1 26061,c1(C(C)C(=O)NCC2(CNC(=O)CC3CC(F)C3)CC2)ccc(F)c(Cl)c1 26062,c1(-c2ccc(SC)cc2C)ccc2oc(C(=O)NC(CC)C(F)(F)F)cc2c1 26063,c1(C(=O)OC)noc(C(C)NC(c2cscc2C)c2nnnn2C(C)C)n1 26064,c1(NC(c2c(OC)cncc2)C)ccc(S(=O)(=O)NCC2C3CCCOC23)cn1 26065,c1(CC)[nH]nc(C(=O)NCC(C)CN(C(=O)C(C)(Cl)Cl)C)c1Cl 26066,N1(C(c2c(C)occ2)=O)CCN(C(c2csnc2Cl)=O)CC1CF 26067,C1(CNC(CCC(=O)C2CCCCC2)=O)CCCN(C(=O)COCC2CC2)CC1 26068,c1(C(N2CCC(=CCNC(C(C(C)C)C)=O)CC2)=O)c(F)ccc2occc12 26069,O=S1(=O)CCc2cc(NS(=O)(=O)c3cnc(-c4ccccc4)nc3)ccc21 26070,Cc1ncc(S(N)(=O)=O)cc1C(=O)NC1CCCCC1NC(=O)C1=C(Cl)CC1 26071,C1(CC)CN(C(=O)CN2CC(C)(OC)C2)CCN1C(=O)C(O)CSC 26072,c1(C(N2CC(C(=O)NCc3cc(C)on3)OCC2)=O)cc(Cl)cnc1Cl 26073,C#CCC(C)(C(=O)N1CCC(CN(C)C)C1(C)C)NC(c1ccc(F)c(C)c1)=O 26074,C(=O)(C1=COCCO1)NC1C(CNC(c2cc(C(C)=O)cn2C)=O)C1 26075,N1(C(CN(C(=O)CC2CC3CCC2C3)CC#C)=O)CCC(C(=O)OC)CC1 26076,C1(C(C)C)(NC(=O)CCn2cc(-c3cscn3)nn2)CCOCC1 26077,c1(NC2CCCN(C(CC(CC)CN(C)C)=O)C2)c(F)cccc1[N+](=O)[O-] 26078,C1(O)(CCNC(CNC(=O)NC)=O)CCCN(C(c2sc(C#N)cc2Cl)=O)C1 26079,c1(N(C2CCCN(C(=O)C(C)(O)C3CC3)C2)C)ccc(Cl)cc1[N+](=O)[O-] 26080,C1(OCC)COCCC1NC(C1CCCOCC1)c1nnnn1C1CC1 26081,c1(C(=O)NC2C(NC(CSC(C)(C)C)=O)CS(=O)(=O)C2)ccc2nncn2c1 26082,N1(C(C2(N(C(C(C)N(C(C)=O)C)=O)C)CC2)=O)CCC(CO)C1(C)C 26083,C1(CNC(CCc2n(C)cnc2)=O)CCN(C(=O)CCCNC(N)=O)C1(C)C 26084,S(=O)(=O)(c1ccc2ccccc2c1)Nc1ccn(C)n1.C1(=O)CCN1 26085,C(=O)(CP(C)(C)=O)NCC(CN(C(=O)C(C)O)CC)(C)C 26086,CCCCCCC(CC)C(=O)NCC1COCCN(c2nccn3nnnc23)C1 26087,C(N=c1[nH]c(=NC(CCO)c2ccccc2F)[nH]c2c1SCC2)C1(C)CCC1 26088,C1(COCC(C)NC(c2ccc(Cl)o2)c2nnnn2C2CC2)CCC(F)(F)CC1 26089,N1(C(=O)Cc2cnc(-c3ccco3)s2)CCC2C(CCCN2C(C2COC2)=O)C1 26090,C(=O)(C1CCCc2ncc(C)n21)N1C(CNC(c2c(OC)ccc(OC)n2)=O)CC1 26091,CCS(=O)CC(=O)NC(C)(CNC(=O)CN(c1cccc(Cl)c1)S(C)(=O)=O)C1CC1 26092,CCC(C)C(C)(O)CNC(C1CC(C)CN(C(=O)Cc2ccc[nH]2)C1)=O 26093,c1(-c2cn(CCC)nc2)nc(=NCc2ccn(CCCOC)n2)[nH]cc1Br 26094,CCCCCCCCC(=O)NC(C)CN(C(=O)Cn1cc(F)ccc1=O)CC 26095,C1(NC(C(=O)NC(C)C)=O)CCC(F)(CNC(c2csc(Cl)c2)=O)C1 26096,C1(C(=O)NC2CC3(CN(C(Cc4c(C)non4)=O)C3)C2)CCCC1S(C)(=O)=O 26097,C1(CNC(CS(CC)=O)=O)N(C(c2cc(Cl)cc(F)c2)=O)CCC1(C)C 26098,c1(NC)ccc(Cl)c(C(N2CC(C)(C)CC2CNC(C2CCC(O)CC2)=O)=O)c1 26099,C1(C(=O)NCC2N(C(CC3CN(C)C3)=O)CC(F)C2)CC1C1CCCC1 26100,N1(C(CC2(C=C)CC2)=O)CC2CC(NC(=O)C(C)(C)F)CC2C1 26101,N1(C(C(C)CO)=O)CCCCC1CCC(N1CCC(C(N)=O)C1)=O 26102,C(=O)(C1(C)CCc2ccccc21)NCC1C(NC(C(C)(C)C2CCC2)=O)CCC1 26103,N1(CC)CCC(n2nc(-c3cncc(F)c3)nc2COC)CC1 26104,C1(N(C(COC(C)=O)=O)C)CCCC(NC(=O)Cc2cnn(C)c2C)C1 26105,C1(CNC(C2CCN(C(C(C)SCCCC)=O)C2C)=O)CC(C(=O)NC)=NO1 26106,C1(CC(=O)NC2CC2NC(c2cncc(CO)c2)=O)CN2CCN1CC2 26107,C1(C(C2(O)CN3CCC2CC3)=O)CC2CC(NC(=O)NC3C4CC5C(C4)C35)C1C2 26108,[N-]=[N+]=NC1(C(=O)NCC(O)CF)CCN(C(=O)CC2CCOC2=O)C1 26109,S(=O)(=O)(CCC(F)(F)F)NC(C1CN(C(C2CC2(F)F)=O)CC1F)=O 26110,c1(N2CCC(CC)(NC(=O)C3=CCCS3)CC2)c(Br)cccc1[N+](=O)[O-] 26111,c1(CC)nc(CC(=O)NCC2CN(C(C3CC3Cl)=O)C2)cs1 26112,C1(OCC)(OC)CCC(C(c2nnnn2CCC2CC2)NC(C)CC(C)C)C1 26113,N1(C(CC2(C)CCN2C(=O)CC2CC(F)(F)C2)=O)CCOC(C)(CO)C1 26114,C1(C(=O)NCc2cn(CC#C)nc2)C2CCC(C2)C1NC(c1cccn1CC)=O 26115,N1(C(c2cnn(C(C)C)c2F)=O)CC2CC(NC(c3cc4scnc4[nH]3)=O)C1C2 26116,N1(C(CC2(NC(c3c(CC)noc3)=O)CCCCC2)=O)CCNC(=O)C1CC 26117,C1(NC(COC2C(C)CCCC2)=O)CCN(C(=O)CS(C)(=O)=O)CC1O 26118,C1(NC(C(CC)C)=O)CCC2(CC1)CN(C(c1cscc1Cl)=O)CCO2 26119,C(CC(C)NC(=O)CCC1CC1(C)C)N(C(COC)=O)C 26120,C(CC(C(=O)NOCC1(C)CCC1)NC(C1CC2(CCCO2)C1)=O)=CC 26121,c1(C(N(CCCNC(=O)CN2CCOCC2=O)C(C)C)=O)cc2ccsc2n1C 26122,c1(C(C)N(C2CS(=O)(=O)C2)C(=O)C2CC2)cccc(F)c1 26123,CC(N=c1cc(C(F)(F)F)nc(Cl)[nH]1)C(c1ccccc1)NC(=O)C(C)O 26124,C1(NC(c2c(C)nc(CCC)s2)=O)CC2(CCN(C(=O)CCOC(C)C)C2)C1 26125,Cc1cccc(C(=O)NCC2(CNC(=O)C=Cc3cncs3)CCCC2)c1O 26126,N1(C(C2N(C(C)=O)CC(O)C2)=O)CCN(C(=O)C(F)(F)C(C)O)CC1CO 26127,c1(C(=O)NC2CCN(C(c3nc(CC)oc3)=O)C2(C)C)ccc2c(c1)CCCC2 26128,C1(NC(C2CC(=C)C2)=O)CCCCC1CNC(=O)CCC1(C)CC1 26129,Cc1ccc(CC(=O)NC(CNC(C2CC(n3ccnc3)C2)=O)C2CC2)cc1C 26130,c1(CC(=O)NCC(C)CN(C(=O)Cc2cnns2)C)cccc(OC(F)(F)F)c1 26131,C1(C(=O)OC)CC(OC)CN(C(=O)C(C)OC(C)(C)C)C1.c1(C=O)ccccc1 26132,CCC(C)CCC(=O)NCCOC1CN(C(=O)CCCc2ccc(C)s2)C1 26133,c1(C(N2C(CCNC(C3CCO3)=O)CCC2)=O)csc2ccc(F)cc12 26134,N1(C(c2c[nH]c(=NC)s2)=O)CC(NC(=O)C(Br)=C(C)C)CC(C)(C)C1 26135,c1(C(=O)NCC2C3N(C(C4CC(OC)C4)=O)C(CC3)C2)c(Cl)c([N+](=O)[O-])nn1C 26136,C1(NC(c2cc[nH]n2)=O)CCCC2CN(C(=O)Cc3csc(C(F)(F)F)n3)CC12 26137,C1(C)(CNC(C2C(CNC(c3cc(COC)no3)=O)C2)=O)CNC(=O)O1 26138,C1(NC(C(CC)(F)F)=O)(CNC(c2ccnn2COC)=O)CCCCC1C 26139,c1(SC)c(C(=O)NC(C2CCOC2)CNC(=O)CN2CCCC2=O)cccc1F 26140,c1(OC)cccc2nc(C(=O)Nc3cc(F)c(Cl)cc3Cl)sc12 26141,N1(C(C2C(NC(c3ccccc3)=O)CCCC2)=O)C2CCC1CC(O)C2 26142,c1(N2CCC(C(C)NC(C(C)Oc3cccnc3)=O)C2)nc(Cl)c(C#N)s1 26143,C1(C(=O)NCCCc2n(C)nnn2)CCN(C(c2ccc(=O)n(C)c2)=O)C1(C)C 26144,C1(N(C(CC2CN(C(C(C)n3cccn3)=O)C2)=O)C)CCN(C2CC2)C1 26145,C1(CC(=O)NCC2CCCO2)CCN(C(C2CCCC2)=O)C1.C(C(=O)O)N 26146,c1(C(=O)NC(CC)(C)CCNC23COCC2C3(F)F)ccc(OC)nc1OC 26147,NS(=O)(=O)CCC(=O)NCCC1(CNC(=O)CC2CCC(O)C2)CC1 26148,C1(C)(CNC(COCC(=C)C)=O)CCC(NC(c2ccn(CC)c(=O)c2)=O)CC1 26149,c1(C(C(N2C(CNC(CCC(=O)NC)=O)C=CC2)=O)C)ccc(F)c(F)c1 26150,CC1CCN(C(C2(F)CCN(C(=O)CCN3CCC3)CC2)=O)CC1O 26151,C(C1CN(C(c2coc(C(F)F)c2)=O)CC1C(=O)NC1(CO)CCCC1)=CC 26152,CCCCC(CC)C(=O)NC1CN(C(c2cccc(C(N)=O)n2)=O)CC12CC2 26153,C(=O)(C(C(C)(C)C)n1ccnn1)N(C)CC1(CNC(COC)=O)CC1 26154,C(=O)(CS(=O)(=O)C1CC1)NCC1N(C(C2C(C)(C(F)F)C2)=O)CC=C1 26155,c1(OC)ccc(C(C)NC(=O)N(C)CC2(F)CCOCC2)cc1S(N)(=O)=O 26156,N1(C(c2c(Cl)ccc(C#C)c2)=O)CC2(C1)C(NC(=O)C=CC(C)C)CCS2(=O)=O 26157,Cc1nc2c(CN3CCN(c4cccc(S(C)(=O)=O)c4)CC3)cccn2c1Br 26158,N1(C(=O)CN2CCOCC2)CC(C2CCCCN(C(=O)C(F)(F)CO)C2)C1 26159,CON1CCC(C(N2CCCC2CC(=O)NC(C)CN(C)C(C)C)=O)CC1 26160,C1(NC(=O)CCC2CC(NC(=O)CC(Cl)Cl)C2)C=CC(CO)C1 26161,c1(OC)cc(OC)cc(C(C#N)NC(c2ncoc2C(C)C)=O)c1 26162,CC1CCC(CNC(=O)COCC2CCCO2)CN1C(=O)C=Cc1nccs1 26163,Cc1sc(Cl)nc1C(=O)NCC1CCN(C(C2CC3(CC3)CO2)=O)CC1 26164,N1(C(COC(CC)C)=O)CCN(c2ccc([N+](=O)[O-])cc2C(C)=O)CC(C)(F)C1 26165,C1(NC(=O)C=Cc2ccccc2)CN(C(=O)CCCN2CCCCC2)CC12CC2 26166,N1(C(c2ccc(CCC)cc2)=O)CCC(NC(=O)CC2CCCC23CC3)C1(C)C 26167,c1(C(N(CC(C)NC(=O)C(C)(C)CCCF)C)=O)nnn2ccccc12 26168,N=c1ncc(C(=O)NCC2(CNC(=O)CCF)CCC2)c[nH]1 26169,C(CNC(=O)CNS(=O)(=O)C1CC1)(C(C)C(C)C)NC(C1(OC)CCCCC1)=O 26170,N1(C(C(CC)C(F)(F)F)=O)CC2(C=C(C(=O)NCC3CCSC3)CO2)C1 26171,Cc1cc(C)n(CCCCNC(=O)CC2CCN(C(c3ccco3)=O)C2)n1 26172,C(C#N)(C(=O)C(C)(C)CNC(c1cnn2cccc(CO)c12)=O)c1scc(C)n1 26173,c1(OC)cc(C(=O)NC23CCC(CN(C(C4CC4(F)F)=O)C2)C3)sc1S(N)(=O)=O 26174,N1(C(C=CC(CC)=CC)=O)CC(O)(C2(CNC(c3ccc(=NC)[nH]c3)=O)CC2)C1 26175,Cc1nscc1C(=O)NC(Cc1cc[nH]n1)C(=O)NC(c1nncs1)C 26176,N1(C(CN(S(CC)(=O)=O)C)=O)CC(C(C)(C)O)(CNC(=O)CC(C)OC)C1 26177,c1(N2CC(OCC)(CNC(=O)CC(O)c3ccccc3)C2)ccnc(CO)n1 26178,S(=O)(=O)(c1cnccc1NCC(C1CCCCC1)F)NC1(C)CCOCC1 26179,c1(C(=O)NCC(C)N(C(=O)COc2ccc(F)cc2)C)cnc(Cl)cn1 26180,C(Cn1cccn1)(C(=O)NC(c1nc(=O)o[nH]1)C)NC(C(C)=C(C)C)=O 26181,c1(C(=O)NC2C(C3CCN(C(C(C=C)O)=O)CC3)C2)ccc2nccc(C)c2c1 26182,c1(CC(=O)NC(CO)C2CC2)cc(Cl)ccc1Br.c12ncccc1NC2=O 26183,C1(NC(C(C)(C)SC)=O)CC2CN(C(C3CC3(F)F)=O)CC12 26184,C(CC(C(=O)N1CCC(C)(C(N)=O)C1)NC(c1cccc[n+]1[O-])=O)N(C)C 26185,c1(C(N2C(CC)C(C(=O)N(C3CC3C3CC3)C)CC2)=O)cccc(C)c1N 26186,C1(CCC)CN(C(=O)Cc2csc(Cl)n2)CCN1C(=O)C(C)OCC 26187,N=c1[nH]c(CCC(=O)NCCOC2CN(C(C3CC3Cl)=O)C2)cs1 26188,Cc1cc(C(c2nnnn2C2COC2)NCCn2ncc(Br)n2)ccn1 26189,C1(C(=O)NCC2N(C(C)(C)C)CC2)C=CCN(C(=O)CN2CC(=O)NC2=O)C1 26190,CCCC(C(=O)NC(C)C(=O)NCC(C)(CC)CC)NC(N)=O 26191,N1(c2nc(C)c(F)cn2)CCc2ccc(NC(=O)CC3COCCO3)cc2C1 26192,n1(CC(=O)NC2CN(C(C=C(CC)C)=O)CC2C2CC2)ccc2ccc(F)cc12 26193,c1(C(=O)NCC(=O)N(CCNC(C2CCCC(=O)O2)=O)CC)cc(F)cc(F)c1 26194,N1(C(C2C(C)C2C)=O)CC(N(C)C(c2cccc(F)c2F)=O)C(C)(C)C1 26195,C1(CNC(C(C)(C)SC)=O)CN(C(=O)CCc2nnc(C(C)C)o2)CC(C)O1 26196,c1(CC(=O)NC(C2CC=CCC2)C(=O)NCCN(C(=O)OC)C)ccccn1 26197,CC(CC(N)=O)C(=O)NC1CC(NC(c2cc(C3CC3)nn2-c2ccccc2)=O)C1 26198,N1(C(c2n(CC#C)ccc2)=O)CC2CCC2(CC(=O)N(CC)CC)C1 26199,c1(CC(=O)NCC2(NC(c3cccc(F)c3O)=O)COC2)nc2ncccn2n1 26200,N1(C(N=c2ccn(-c3ccnc(C)c3Cl)[nH]2)=O)CC(F)(F)CC2CCCCC12 26201,Cc1cc2c(cc1C)C(C(=O)N1CCC(C(C3CC3)N(C)C)CC1)CO2.C(=O)N 26202,N1(C(C(C)=C2CC2)=O)CCN(C(=O)CNC(C2CCC2)=O)CC1CS(C)(=O)=O 26203,Cc1cccc(C)c1CCC(=O)NC1CC12CC(NC(=O)CC13CCCC1C3)C2 26204,CCC(C)C(O)C(=O)NC1CCN(CCNC(=O)C(F)(F)C2CCCC2)CC1 26205,CC1(C)CC2(CC(C(N3CCN(C(c4ccccc4Cl)=O)CC(CO)C3)=O)C2)C1 26206,CC(C)C(CN(C)C)C(=O)N1CCOCC(NC(=O)CCCN=[N+]=[N-])C1 26207,c1(C(N2CC3C(CNC(C(C)=C(C)C)=O)(C3)C2)=O)cccc2cccc(O)c12 26208,c1(C(N2CCC(c3cccc(C#N)c3)C2)=O)c(F)ccc2c1OCO2 26209,c1(NC(c2ccc(CF)cc2)c2n(C(CC)C)nnn2)ccccc1OC 26210,C=Cc1ccc(C(N2CCC(C(=O)NC(C)CN3CCCC3)(OC)C2)=O)cc1 26211,C(=O)(CC(O)CC(C)(C)C)NCC#CCNC(C(CSC)c1ccccc1)=O 26212,c1(C(=O)NC(CCCNC(CSCC#C)=O)C)ccc(Cl)c(Cl)c1C 26213,C1(NC(C2(C)CC(=C)C2)=O)CCC(F)(CNC(=O)COCC2CCCCO2)C1 26214,CC(C)C(F)(F)CC(=O)N1CCCC(N(C)C(c2ccc(Cl)cc2)=O)C1 26215,c1(OC)cc(C=CC(N2CC(F)CC2CNC(c2cnc(Cl)s2)=O)=O)ccc1N 26216,Cc1cc(C(=O)NC2CCN(C(=O)CN3CSCC3=O)CC2F)c2[nH]cnc2c1 26217,C1(COC)CN(C(=O)N(C)Cc2nnc(CO)s2)CCO1 26218,C1(C(=O)NCCCN(C(c2ccc(CC(C)C)s2)=O)C(C)C)CCCCCCC1 26219,c1(C(N2C(C(C)NC(C3(C)CS(=O)(=O)C3)=O)CCC2)=O)cn(C)c2ccccc12 26220,N1(C(C(CC)(C)O)=O)CCC2(CCCC(CNC(C3(C(F)F)CCC3)=O)O2)CC1 26221,c1(NC(C2N(C(CSCC#C)=O)CC2C)=O)cncc([N+](=O)[O-])c1 26222,C1(NC(C(CCSC)OC)=O)CCC2(CCN(C(C3CC=CC3)=O)CC2)C1 26223,c1(C(N2CC(NC(c3ccc4sncc4c3)=O)C2)=O)cnn2cc(Br)cnc12 26224,N1(C(c2n(C(CC)CC)ncc2)=O)CC2C(CNC(c3ccc(Br)o3)=O)C2C1 26225,c1(OC)cc(C)c(C(=O)NCC2(F)CCN(C(C3COC(=O)N3)=O)C2)cn1 26226,C1(NC(c2c(CC=C)cccc2)=O)CN(C(=O)C(O)C=CC)CC12CCC2 26227,C1(NC(c2c(C)nc(C(C)C)s2)=O)(CNC(=O)COC(F)(F)F)CCCCC1C 26228,C=CCC(CC=C)C(=O)N1CCC(C(=O)NC2(C)CCC(C)(C)CC2)CC1C 26229,Cn1nnc2cc(C(=O)NC3CN(C(c4ccon4)=O)CC3C3CC3)ccc12 26230,C1(C(N(C2CC(NC(C3(C(F)F)CCC3)=O)C2)C)=O)CCCOC1 26231,c1(OC)ccc(C(CNC(c2snc(Cl)c2Cl)=O)NC(=O)CCC#N)cc1 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26250,O=C1Cc2c(C(N3CC4(CC4C(N4CC(F)C(F)C4)=O)C3)=O)cccc2N1 26251,C1(NC(C(OCC)OCC)=O)CCN(C(=O)CC2CC(C(C)(C)C)C2)CC1CO 26252,c1(C(N(CCCNC(CC(CCC)C)=O)CC)=O)csc(=NC2CC2)[nH]1 26253,c1(C(C(=O)NCC(CN(C(=O)Cc2cncs2)CC)(C)C)O)ccc(Cl)cc1F 26254,C(=O)(N1CC(O)CCO1)C1CCCN(C(c2cncc(CO)c2)=O)CC1 26255,C(C1(C)CCOCC1)=CC(=O)NCC(CNC(CCN(CC(C(C)C)C)C)=O)O 26256,c1(CC(=O)NC2CCC2NC(C(C)NC(=O)OC(C)(C)C)=O)cn(C)nn1 26257,CCC(CC(F)(F)F)C(=O)N1CC2CC3CC2C1C3NC(=O)CCCS(N)(=O)=O 26258,n1(CCC)cc(C(=O)N(CCCNC(=O)CNC(=O)NCC)C)cn1 26259,Cc1sc2nc(CN(C)CC3CCCN3C(C3CCC4CC4C3)=O)nc(O)c2c1C 26260,N1(C(CCCCCCC)=O)CC(CO)C2(C1)CN(C(=O)C(C)(C)c1ccsc1)C2 26261,c1(C(=O)NCC2N(C(CCc3ccc(C4C(C)C4)o3)=O)CC2)cc(C)ccc1F 26262,C1(c2n(Cc3cn(CC)nn3)ccn2)CCCCCCC1.c12ccc(s1)CC2C 26263,N1(C(CN(C)CC)=O)CC2CCCC1C2CNC(=O)C(C)(C)n1cccn1 26264,N1(C(c2n(C)ncc2I)=O)CC2(C1)SCCC2NC(C1CC12CCSCC2)=O 26265,c1(C(N(C)CCNC(=O)CCCn2cccn2)=O)ccc(OCC2CC2)cc1 26266,c1(C(N2CCC3CCN(C(=O)C4=CCC4)C3C2)=O)cc2cc(F)ccc2[nH]1 26267,c1(C(=O)NC2C3(NC(c4cc(C)nn4C)=O)CCC(C2)C3)cccc2[nH]ncc12 26268,CCCCCC(O)CC(=O)N1CCN(C(c2sccc2F)=O)CC1CF 26269,Cc1cnc(C(N2CCOC(CCNC(=O)C(C)(C)C(C)O)C2)=O)nc1 26270,c1(CN=C(NCc2cc(C)on2)NC(c2ccn(C)c2)C)cn(C)c(=O)nc1O 26271,CCC(CC)(CCNC(=O)C=NOC)NC(C1CCC1n1cccn1)=O 26272,c1(C(N=c2cc(CC(C)C)o[nH]2)=O)ccc2nnn(O)c2c1 26273,c1(C(N(CC(C)NC(Cc2c(C)cco2)=O)C)=O)[nH]c2cc(F)cc(F)c2c1C 26274,C(C1=CCN(C(=O)COCC(F)F)CC1)NC(C1C(C)(C(C)C)C1)=O 26275,C(=O)(CCC(C)N(C)C)N(CC(CNC(CSCCC(C)C)=O)(C)C)C 26276,C1(C(=O)NC2(C)CCCN(C(=O)CNS(N)(=O)=O)C2)CC2CC1CC2(F)F 26277,CCCCC(CC)CC(=O)NC1CN(C)CCN1C(=O)COC1(C)CCCC1 26278,N1(C(C2(CNC(CCC3(C)CC3)=O)CC23CCC3)=O)CCC(C2CCC2)C1 26279,C(=O)(CCC(=O)NCC)NCC1(NC(CC=CCC)=O)CCC1 26280,N1(C(C(CN(C)C)NC(=O)COCCCF)=O)CCCN(CCO)CC1 26281,C1(n2cc(C3CCN(C)C3)nn2)C=CCC(C(=O)NCC2CCSCC2)C1 26282,C(C(C)(CNC(c1cscc1Cl)=O)OC)NC(C(C)OCCCC)=O 26283,CC(C)C(CCNC(c1ccc(N(C)C)cn1)=O)NC(=O)CCN1CCCCC1 26284,c1(C(N2C(CNC(=O)CC3CCCCC3)C=CC2)=O)ccn2ccnc2n1 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26302,Cc1c(OC(F)(F)F)cccc1Br.C12CN(CCO1)C(=O)C2 26303,C1(NC(C2CC(NC(C(NOC)=O)=O)C2(C)C)=O)CC2CCCC2C1 26304,C1(C(N2CCC(C)C2CNC(c2ccoc2)=O)=O)CCCNS1(=O)=O 26305,Cc1ccc(C)c(C(=O)NC2CC2CNC(=O)C(C)Sc2nncn2C)c1 26306,c1(C(CNC(c2n(CCCSCC)nnn2)CCOC)F)ccc(Br)cc1 26307,N=c1[nH]cc(C(=O)NCCC2(CC(=O)NCC(O)C(=O)OC)CC2)o1 26308,Cc1oc(-n2cccc2)c(C#N)c1C(=O)NCC1CCCN1C(=O)CC1CC1 26309,Cc1ccc(N)c(C)c1C(N1CC2CCCC2(NC(C2CCC(O)CC2)=O)C1)=O 26310,C1(CC)CCCC(N=c2[nH]c(=NCC3(CN(C)C)CC3)[nH]c3c2CSC3)C1.C1CC1 26311,c1(NC(c2nc(Nc3nc(OC)nc(OC)n3)sc2)=O)ccc2ccsc2c1 26312,N1(C(C(CCC)O)=O)CC2(CCN(C(C3CCCCO3)=O)CC2)CC1C 26313,Cc1cc(C(N2CCC(C)C2CNC(=O)Cn2ccsc2=N)=O)cc(F)c1 26314,C1(C(N(C2CCCC2)CCNC(c2ccc(CC)o2)=O)=O)CC(C)CC(C)(C)C1 26315,c1(CC(=O)NCC(C2CC2)NC(C(C)OCCC=C)=O)ccc([N+](=O)[O-])c(N)c1 26316,C=CC(C)CC(=O)N(C1CCN(C(c2cc(C)sn2)=O)C1)CC 26317,N1(C(=O)NC(CC)C(C2CC2)Sc2ccccc2)CC2(CSCBr)CC2(C(F)(F)F)C1 26318,CCCCC(O)C(=O)N1CC(NC(c2nccc(C)n2)=O)C(CC2CC2)C1 26319,N1(C(CC2C(NC(c3n(C)nc(O)c3)=O)CCCC2)=O)CCOC2CCCC12 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26355,c1(OC)cc(F)c(C(=O)NCC2CCCCC2NC(C2CC(F)(F)C2)=O)c(F)c1 26356,c1(CNC(c2ncc(Cl)n2C)C(=O)OC)cccnc1N1CCN(C)CC1 26357,CC(C)C(F)(CNC(=O)C(F)C(F)(F)F)C(=O)N1CCC2(CC2)C1 26358,c1(CC)nc(C(=O)N(C2CCC(NC(=O)COCc3cc(C)on3)C2)C)co1 26359,C#Cc1ccc(CC(N2CCN(C(c3cccnn3)=O)C(CO)C2)=O)cc1 26360,N1(C2N(C(C(COC)NC(C)=O)=O)CCC2)CCCC(C)C1 26361,C1(NC(CSC)=O)C2CC1N(C(=O)CCC(=O)N(C)C(C)C)C2C 26362,Cc1csc2ncc(C(N3CCC(NC(C4CCC(F)(F)CO4)=O)C3)=O)c(=O)n12 26363,c1(OC(C2(CC=CC)CC2)=O)ncnc2[nH]cc(C)c12.c12ccc(cc1F)NC2 26364,N1(C(COCC=C)=O)CCCC1C1(C(=O)NCC=Cc2ccsc2)CC1 26365,C1(C(=O)OC)CC(C)N1C(C1(NC(c2cnc(C(C)C)o2)=O)CC1)=O 26366,c1(C(=O)NC2CCN(C(C(CC=C)C)=O)CC2F)ccc2c(c1)C(=O)NCC2 26367,c1(CC)cc(C(N2CCOCC2CCNC(=O)CC2C=CCCC2)=O)cc(O)n1 26368,c1(C(N(CC(CN(C(=O)C(F)n2cccn2)C)O)C)=O)ccccc1N(C)C 26369,C1(NC(C(C)(C)SC)=O)CN(C(c2cncc(C(C)(F)F)c2)=O)CC1C(F)F 26370,C1(CC)CCN(C(C2CCC2C(N)=O)=O)C1C(=O)NCCCC1(C)CC1 26371,c1(CC(=O)NCC(CN(C(C2C(CC)CCC2)=O)C)C)ccc2ccccc2c1 26372,C(C(O)CC(=O)Nc1cccc(C)c1)NC(COCCOC)=O 26373,C1(C(N2C(CNC(C(CC)N(C)C)=O)CCCC2)=O)OC2CCC1CC2 26374,C1(OCCNC(C2(C(F)(F)F)CCC2)=O)CCN(C(c2coc(O)n2)=O)CC1 26375,c1(C(=O)NCC2(NC(CN(C(COC)=O)C)=O)CC2)cn2c(n1)CCC(C)C2 26376,C(=O)(C(C)(C)CC=C)N1CCCC(CNC(C(CC=C)OC)=O)C1 26377,C(=O)(C(CCS(C)=O)N(C)C)NC1CCN(C(CCCOC)=O)C1(C)C 26378,C12(C(=O)NC(C)CNC(C3COC(=O)N3C)=O)CC3CC(C)(C1)CC(C)(C3)C2 26379,C1(NC(C(CC=C)C)=O)CCN(c2ncc(Br)cn2)CC1C 26380,c1(OCCC)ccc(C(=O)NC2(CNC(C3SCCCS3)=O)CC2)cc1N 26381,c1(C(=O)NCCN2CCN(C(C=CCCC)=O)CC2)c[nH]c2cnccc12 26382,c1(C(c2n(C)nnn2)NCc2cnoc2C(C)(C)C)nn(C)cc1I 26383,c1(OC)c(C)cc(NC(C2(O)CCN(C(=O)C(O)C(C)(C)C)C2)=O)cc1C 26384,Cc1ccc(SC(C)C)c(NC(=O)C(=O)Nc2c(C)noc2-c2ccccc2)c1 26385,C1(C(=O)NCC(C)(O)CNC(=O)Cc2csc(Cl)c2)CCOCC12CCC2 26386,C(CC(O)C(=O)N1CCC(C)(CC(=O)NCC2CCC(=O)O2)C1)SC 26387,c1(-c2cn(CCN(C(=O)C(C)NC(N)=O)CC)nn2)cccc(N)c1C#N 26388,C1(OC)CCCC1CNC(c1cn(CCNC(C2CNC(=O)N2)=O)nn1)=O 26389,c1(OC)c(C(=O)NCC(C(C)C)NC(c2ncc(F)cc2F)=O)ccnc1F 26390,C(CCCCCC(=O)N(CC(=O)N(C)C)C)NC(C(C=C)CC)=O 26391,C1(COC)CCCCN(C(=O)C(N2CCSCC2C)=O)C1 26392,CC1CC(NC(=O)C=Cc2ccc(Br)s2)CN(C(=O)C(C)NC(N)=O)C1 26393,c1(NC(c2ccc(Br)c(Cl)c2)c2n(C(C(=O)OC)C)nnn2)ccc(Br)c(C)c1 26394,C1(C(=O)NC(c2ncnn2C)C)CN(C(=O)CN2CCC(F)CC2)C2(CCC2)C1 26395,c1(NC(C)=O)ncc(S(=O)(=O)N2CCCC2c2cc(F)cc(Br)c2)s1 26396,CCC(F)(F)C(=O)NCC1CCN1C(=O)CCN1CCNC(=O)C1 26397,N(C(=NCC1CCN1c1ccccc1F)NC(C1CC1)C1CC1)C1CC(F)C1 26398,C=CCCCC(C(=O)NOCCCOCC)NC(c1nscc1C)=O 26399,C=CCCCC(=O)NCC1(CNC(C2CCC(C)CC2)=O)CC1(F)F 26400,c1(C(=O)NCC(C)CNC(=O)CC(C)(C)O)ccc(F)c2ncccc12 26401,C(=O)(CS(=O)(=O)CC(=O)N(C)CC1CCCN1C(=O)C(C)CC(C)C)OC 26402,c1(OC)cccc(CC(O)C(=O)N(C)CC2CN(C(C3CCC(=O)N3)=O)C2)c1 26403,c1(CC)cc(C(N2CCCC2c2ccc(F)cc2)C(=O)NC(C)(C)C)ccc1Br 26404,N1(C(c2cnn(C)c2C(C)(F)F)=O)CCC(NC(C2CC2CF)=O)CC(O)C1 26405,C1(C)(C(=O)OCC)CN(S(=O)(=O)CC2OCCC2CC)CCO1 26406,C1(CNC(=O)CN2CC3CC3C2)C(C2CC2)CCN1c1cc(O)nc(O)n1 26407,N1(C(CC2CC(OC)C2)=O)CC(NC(C2(CC(C)C)CCCC2)=O)CC1(C)C 26408,N1(C(CC(=O)OC)=O)CCC2C1CCCN2C(c1ccc([N+](=O)[O-])c(C)c1)=O 26409,C1(C(C(=O)NCC(=C)C)N(CC(=O)NC)CC)CCSC1(C)C 26410,CCCCCC(O)C(=O)NCC1CN(C(=O)C(=O)NCCOCCOC)CCO1 26411,N1(C(c2c(C)cno2)=O)CC2CC(NC(=O)CCOC3CCOC3)C1C2 26412,c1(C(=O)NC2CN(C(=O)C=Cc3cncs3)C2)cc(F)ccc1Cl 26413,C1(C)(C(N(CC(C(=O)NC)C)C)=O)CCN(C(=O)CCOCC(F)F)C1 26414,C12(C(N3CC(n4cc(C(c5cn(C)nn5)N)nn4)C3)=O)C(C(=O)O)C3CC1C2C3.CC 26415,c1(C(=O)NC2CC(NC(c3cnc(C)[nH]3)=O)C2)c(C)[nH]c(-c2ccc(C)o2)nc1=O 26416,N1(C(C(CC)F)=O)CCc2nc(NC(=O)CNC(=O)NCc3ccco3)sc2C1 26417,c1(-c2scc(C(=O)OCC=CC=CC)n2)cccc(Cl)c1 26418,CC(C)C(F)(F)CC(=O)NC1CC(CNC(c2ccc(O)nc2)=O)C12CCC2 26419,c1(CNC(C(CC)C)=O)ccc2c(c1)CCN(C(C1(C)CCN(C(C)=O)C1)=O)C2 26420,N1(C(C)=O)CC2COCCC2(NC(c2cccc([N+](=O)[O-])c2Br)=O)C1 26421,C1(C(=O)NC(CNC(C(CC)C2CCC(=O)N2)=O)C)CCC(OC)CC1 26422,c1(C(=O)NCC2CCN(Cc3cscn3)CC2)cncc(N2CCCC2)n1 26423,c1(N2CCN(C(=O)NC)CC2)nc(=NC2CCCSCC2)[nH]c2c1COC2 26424,N1(C(C2(C)COC2)=O)CCC2(NC(c3ccc(-c4cccs4)[nH]3)=O)CC2C1 26425,c1(C(CNC(c2c(C)cncc2)=O)NC(c2ncccc2N)=O)cc(F)cc(Cl)c1 26426,C1(C(N(C2CN(C(c3cnc(C(F)F)nc3)=O)CC2F)C)=O)CCC(C)(C)CC1 26427,n1(C(C(=O)NC2CC(NC(C3C(C(=O)OC)CC3)=O)C2)C)cc2c(n1)CCCC2 26428,c1(C(N2CCC(NC(C3(CC)CCNC3=O)=O)CC2)=O)cnc2sccc2c1 26429,C#CC1CC2CCC1N(C(=O)CC1(OC)CN(C(c3cnn(C)c3CC)=O)C1)C2 26430,CC1(C)OC2(C(N3CC(OCCNC(=O)CCn4cccn4)C3)=O)CCC1CC2 26431,C1(CNC(C2(C)CC(=C)C2)=O)C(C)CCN1c1ccnc(C(C)CC)n1 26432,C1(C)(CNC(C(C)NS(CCC)(=O)=O)=O)COCCN(C(=O)CNC(=O)OC)C1 26433,C1(c2nc(C3(C(C)C4CC4)CC3)on2)(c2nn[nH]n2)CCCCCC1 26434,C1(C(=O)NCC2CC(O)CN2C(c2cn(C)c(C)n2)=O)(COC)CCOCC1 26435,N1(CC2CCN(C(=O)OC(C)(C)C)C2)CC(CO)C2(CC2)C1 26436,C12(COCC)CC(C(N3CCC(C)(CNC(=O)CC=C(C)C)C3)=O)(CO1)C2 26437,c1(C(N2C(C)CC(NC(c3cnn(C)c3C3CC3)=O)C2)=O)cc(Cl)ncc1O 26438,C1(CNC(c2c(SC)ccs2)=O)C(C)CCCN1C(=O)CC1CCCC(F)(F)C1 26439,C1(NC(CN(CCC)C)=O)(CNC(C2(CC#N)CCOC2)=O)CCCC1 26440,CC1CC(C(=O)NCC2(NC(=O)CS(N)(=O)=O)CCCCC2)CCS1(=O)=O 26441,C(=O)(CCCC(F)F)NCC(CCCC)NC(=O)CN1CCCC1C 26442,C1(F)(CNC(c2cnsc2)=O)CC(NC(C2CC2(F)F)=O)C1 26443,C1(C(=O)NCCC(CNC(=O)C(C)O)OC)CCCOCC1 26444,C=C(C)CCCC(=O)NCC=CCNC(=O)C(C)c1cncs1 26445,c1(C(=O)OC)ccncc1C(=O)NC1CCCCC1NC(C1CC12CCC2)=O 26446,CC1CCN(CC(=O)NCCN(C(=O)CC2CCSCC2)CC2CC2)C1 26447,C(CCCCCF)N(C(=O)C(n1cc(CCCS(N)(=O)=O)nn1)C)CC 26448,c1(C(N(CC(C)(C)O)C2CC2)=O)cc(CO)ncn1.C1(=O)C(F)CC2CN1C2 26449,c1(C(=O)NC2(C)CN(C(c3nc(C(=O)OC)sc3)=O)C2)cncc(N=[N+]=[N-])c1 26450,CCC(C)(CC)C(=O)OC(C)(C)C.C12CC(=NO1)CCc1nc(no1)CN2 26451,N1(CC)CCCCC1C(=O)NCC1CCCCN1C(C1(O)CCCCC1)=O 26452,CC(O)CCCCCC(=O)N1CCN(C(=O)C(F)C(F)(F)F)C2(CCC2)C1 26453,c1(C(C)(C)C(=O)NCC2(O)CC(NC(C3CCCO3)=O)C2)cccc(Cl)c1F 26454,c1(C(=O)NCCC2N(C(C3=CCCC3C)=O)CCSC2)n[nH]c2ccc(F)cc12 26455,N1(Cc2cccc(OC)c2)CCC(O)(C(=O)NC2CCOCC2F)CC1 26456,C1(C(=O)NC)CN(C(=O)CN(C)C(=O)C2CC2)CC1(C)C 26457,C1(CNC(Cn2c(C)ccn2)=O)CN(C(=O)CC2C=CCC2)CC1(C)C 26458,c1(CO)ccc(N)cc1.C12(N)CC(CC3(C(=O)COCC)CC3)(C1)C2.C1(=O)CN1 26459,c1(C(=O)NC(C2(O)CCN(C(=O)CCc3ccccc3O)C2)C)cnccc1Cl 26460,C(C)(N=c1ccc(Br)c(S(=O)(=O)N2CCCC2CO)[nH]1)c1ncc(C)s1 26461,c1(C(C(N2CCCN(c3ccccc3C#N)CC2)C)=O)ccc2c(c1)CCC2 26462,c1(OCC)cccc(F)c1C(=O)NC(C)C(=O)O 26463,c1(OCC(=O)Nc2nc(CC)nc(C(C)(C)C)c2)c(Cl)cc(Cl)cc1Cl 26464,CCC(CC)CCC(=O)N1CCC(NC(c2cncc(F)c2Cl)=O)C(F)C1 26465,C1(NC(C(=O)NCCOC)=O)CCC(CCNC(=O)CC2CCOC2)C1 26466,c1(NC(=NCC(=C)C)NC2CC2C2CCCC2)ccc(S(N)(=O)=O)nc1OC 26467,C1(NC(Cc2c(C)nn(C)c2)=O)CCS(=O)(=O)C12CN(C(=O)C(O)C1CCC1)C2 26468,c1(OC)cc(C=CC(=O)Nc2ccn(C)c(=O)c2C)ccc1OCC(N)=O 26469,c1(CC)cc(C(N2CC(CC(F)C(=O)NCCCc3cc(C)[nH]n3)C2)=O)ccn1 26470,C1(NC(C2CC(C)(CC)C2)=O)CCCC2CN(C(=O)C=Cc3ccccc3)CC12 26471,c1(CCC(=O)NC2(CNC(C3CC(Cl)(Cl)C3)=O)CC2)cnc2ncccn12 26472,c1(C(=O)NCC2N(C(C(C3CCOC3)OC)=O)CCC2)c(F)cc(C#N)cc1F 26473,c1(C(N(CC(C)NC(C2CCCSC2)=O)CC)=O)cc(SC)ccc1Cl 26474,C1(C(=O)NCCSC)(CNC(=O)CCN(C)C)CCCCC1 26475,CCCCC(CNC(C1C2CCC12)=O)NC(=O)CCc1nccs1 26476,Cc1cccc(OCCC(N2CC(O)(C(C)NC(c3c(C)nsc3C)=O)C2)=O)c1 26477,N1(C(CC2N(C)CCC2)=O)CCC(NC(c2ccnc(O)c2F)=O)C(CO)C1 26478,C1(C)(NC(C(CC2CCC2)NC(CC(CC)O)=O)=O)C(C)(C)C1(C)C 26479,c1(C(=O)NC(c2cccc(Cl)c2)C)ncccc1CNC(C1CC1CO)=O 26480,c1(C(=O)NC(CN(C(=O)Cc2ccon2)C)(C)C)ncc(Cc2ccccc2)s1 26481,C(=O)(C(C(=O)N1CCC(CN(C)C(c2cncn2C(C)C)=O)C1)OC)OC 26482,C1(CC)(NC(c2ccnc(C(C)(C)C)c2)=O)CCCN(C(c2snnc2C)=O)C1 26483,c1(C(=O)Nc2c(C)cc(NC(C3CCC(=O)N3)=O)cc2)c(Br)ccc2c1CCC2 26484,C1(NC(C(c2ccccn2)C)=O)CN(C(c2cccc(Cl)c2)=O)C2CCCCC12 26485,C(CCNC(=O)CCC=CC(C)C)(C(C)C)NC(CCSCC)=O 26486,c1(C(=O)NCC2CC(OC)(OC)C2)sc(Br)c(C)c1C 26487,Cn1nc(C(=O)NCCC2(CNC(=O)CCc3ccc(=N)[nH]c3)CC2)ccc1=O 26488,C(CN=c1cc(C)nc(N2CCOC3(CCSC3)C2)[nH]1)(c1ccccc1)OC 26489,C1(C(=O)NC23C(CN(C(CC4(C)CCC4)=O)C2)C3)CC2CCCC(C1)C2 26490,c1(C(=O)NCC(CNC(c2ncc(C)c(C)c2)=O)O)ccn2ccccc12 26491,C1(C(=O)NCCOCCN(C(Cc2ccc(CC)cc2)=O)C)CC2C(C1)C2(C)C 26492,S(=O)(=O)(c1ccc(NC(c2ncc(Br)cc2C)C)c(C#N)c1)NC(CC=C)CC 26493,c1(OC)nccc(C(=O)NC2CCCN(C(=O)C(C)CC(F)F)C2C)c1F 26494,C(=O)(CCCC(=O)OC)N(C1CCN(C(C(C(C)C)OCC)=O)CC1)CCO 26495,c1(CC)nc(N2CC3CC(NC(=O)C(C)C)CC3C2)c(C)c(Cl)n1 26496,C#CC1CCCN(C(C2(C(C)NC(=O)C=Cc3ccoc3)CC2)=O)C1 26497,c1(OC)cc(F)ccc1C(N1CC(C)(C)CC1CNC(=O)CCCC1CC1C)=O 26498,c1(C(N2CCC(NC(CN3C(C)CC3)=O)CC2C)=O)cccc2[nH]ccc12 26499,Cc1ccnc2nc(C(=O)NC3CN(C(C4CC4(C)Br)=O)CC4(CC4)C3)nn12 26500,Cc1ccc(C(=O)NC(C)CCCNC(c2coc(CO)c2)=O)cc1S(N)(=O)=O 26501,C(=O)(CC(C)C(C)(C)C)N1C(C(C)C)CN(C(=O)CCCc2ccccn2)CC1 26502,N1(C(CC(CC)C)=O)CCC(CNC(=O)C=Cc2ccc(Cl)s2)C12CC2 26503,N1(C(C(COC)OC)=O)CC(C(=O)N(CCCC(C)(F)F)C)CCC1C 26504,C(=O)(C#CC1(C)COC1)N1CC(CC(=O)NCc2cc(C)nn2C)OCC1 26505,c1(C(N(C2CC(CNC(=O)CSc3nncs3)C2)C)=O)cccc(=O)n1C 26506,c1(C(N2CC(C(C)NC(C(COC)(C)O)=O)OCC2)=O)cncc2[nH]ccc12 26507,CC(C)CC(C)CC(=O)N(C1CCC(Cc2nccn2C)CC1)CC.c1(=O)c(=O)[nH]1 26508,C(=O)(C1=CCCOCC1)NC(CC)(CC)CCNC(=O)Cc1c(C)nn(C)c1C 26509,CCC(C)C(C(=O)N1CCC(n2cc(Cn3cncn3)nn2)C(O)C1)N(C)C 26510,N1(C(c2c(C)nn(C)c2Br)=O)CCN(C(C2CCC(O)C2)=O)CC(O)C1 26511,C1(N(C)C)CCCN(C(C2C=CCN(C(=O)C=Cc3ccnn3C)C2)=O)C1 26512,C1(C(=O)NC2C(C)N(C(c3ccn(C4CCC4)n3)=O)CC2)CC2(COC(=O)N2)C1 26513,N1(CCNC(c2cnc(S)[nH]2)=O)CCN(C(c2csc(-c3cnc[nH]3)n2)=O)CC1 26514,c1(C(N2C(CC(=O)NC3CC=C(C)CC3)CCC2)=O)ncn2ccccc12 26515,CP(C)(=O)CC(=O)N1CC2(NC(C3CN(C(C4CCCCC4)=O)C3)=O)CC1C2 26516,C1(C(N(CC#C)Cc2cccnc2)=O)CCCC(C(F)(F)F)C1 26517,c1(Cc2c(-c3ccc(OCC)c(CO)c3)nccc2)cc(OC)c(C)cc1C 26518,C1(CNC(=O)C2=CCOC2)CCN(C(=O)C2=C(Cl)CCC2)CC1(F)F 26519,CCC(C(=O)NC(C)(CNC(c1cc(C2CCCCC2)[nH]n1)=O)CO)C(C)C 26520,N1(C(C(=O)NCCC)CC2CC(F)(F)C2)CCC(C2CCCCC2)CC1 26521,c1(CC(=O)NCCn2cc(CC(CC)(C)O)nn2)cccc(F)c1Cl 26522,C1(NC(=O)COC(=O)CO)CCN(CCNC(c2cocn2)=O)CC1 26523,c1(CN2CCC(CCNC(C(COCC)C)=O)C2)cccc(S(C)(=O)=O)c1 26524,CC1CC(C)N(C(c2ccns2)=O)CCN1C(c1ccc(CC2CC2)cc1)=O 26525,N1(CC2(C(=O)OCC)CCC2)CCC(Nc2cn(C)cn2)C1c1ccccc1 26526,CC1CC(NC(C2CC2C#N)=O)CCN1C(c1cnn(C2CC2)c1Cl)=O 26527,c1(C(=O)NCC2(NC(=O)CC(F)(F)F)CCC2)cc2c(nn1)CCC2 26528,n1(CC)cnc2[nH]c(=NC3CC3CC)nc(N3CCCC(OC)C3)c12 26529,C1(CNC(C(C)(C)O)=O)CC(C)(C)CCC1NC(=O)COc1ccsn1 26530,c1(C(=O)NC(CC)CN(C(=O)C=CC2CC2)C)cccc(NC(N)=O)c1 26531,C1(CC(=O)N(CCCO)CC)CC(NC(C2(C3CC3)CC2)=O)C(O)C1 26532,c1(OC)ncc(Cl)c(C(N2CC(N(C)C(c3ccccn3)=O)C(O)C2)=O)c1Cl 26533,c1(C(=O)OC)ccc2c(c1)C(C(=O)N1CCC(NC(=O)COCCF)C1)CC2 26534,C1(CNC(c2ncccc2Cl)=O)CN(C(=O)C2=CC(O)CCC2)CC12CCC2 26535,C#CC1(CNC(C2(NC(c3ncc(F)cc3F)=O)CCSC2)=O)CCOCC1 26536,c1(OC)ccc(F)cc1CCC(N1CCCC1CNC(c1cc(O)nn1C)=O)=O 26537,C1(C(=O)NCC(C)(C)C#N)CCCC(NC(=O)CC(C)(C)C)CC1 26538,c1(SCC(=O)NC(C(CO)NC(C(F)OC)=O)C)nc(C)nc2sc(C)c(C)c12 26539,c1(C(N)=O)cccc(C(N2CC3(CNC(=O)CCOCCF)CCC2C3)=O)c1N 26540,C1(C(=O)NC(CCOC)CO)C=CCCN1C(=O)Cc1cc(C)cs1 26541,C=CCC(CNC(C1(C2CC2)CC1)=O)NC(c1c[nH]nc1-c1ccnn1C)=O 26542,N1(CC(C)C)CCC(C(=O)NCC(C(C)(C)C)NC(=O)C=CC2CCCO2)CC1 26543,C1(NC(C2(COC)C=CCN2C(=O)CC(C)n2ccnc2)=O)C2CCCCCC12 26544,CCCC(C#N)C(=O)NCC1(O)CCCN(C(c2c(C)cnn2C)=O)C1 26545,C(=O)(CCC(C)(C)C(=O)N(CCNC(C1CCCCC1F)=O)C1CC1)OC 26546,N1(C(c2ccc(NC(C(C)C)=O)cc2)=O)CCN(C(=O)C2CC2)CC1CC1CC1 26547,c1(C(=O)NCC2N(C(CC(C)C(F)F)=O)CC(F)(F)C2)cc2ccccn2n1 26548,N1(C2CC3CN(C(c4nccs4)=O)C2C3)CCc2ccc(Br)cc2C1 26549,c1(C(N(C2CN(C(C3C(CC)CCCC3)=O)C2)C)=O)cc2c(C)ccc(F)c2[nH]1 26550,C(c1ccccc1OC)=CC(=O)NCC1CCC(NC(C(CC=C)C)=O)C1 26551,N1(C(C(CSC)C)=O)CC(C(=O)NCC2(C(C)C)CC2)CC1(C)C 26552,N#Cc1c(Cl)cc(-c2cn(CCNC(C3(O)CCC3)=O)nn2)cc1Cl 26553,CC1(CNC(C2C3COCC23)=O)CCN(C(C2(C(N)=O)CCC2)=O)C1 26554,N1(Cc2cccc(C)c2)CCC(C)C(NC(c2cc(C3CC3)nn2C)=O)C1 26555,C1(NC(COCC=C)=O)CCCC(NC(c2cccc(CCN(C)C)c2)=O)C1 26556,CCC(C)(C#N)C(=O)N(C)CCNC(=O)CNC(c1ccccc1N(C)C)=O 26557,c1(OC)ncc(C(N2CC(NS(=O)(=O)C(F)(F)F)CC(F)C2)=O)cc1Br 26558,c1(N(C(N2CC(=C(C)C)C2)=O)CC2CC2)cccc([N+](=O)[O-])c1 26559,N=c1nc[nH]n1CC(N1CC(CC(F)C(=O)NCC2C=CCC2)C1)=O 26560,N1(CCN(c2cc(Nc3cc(C)cc(C)n3)ncn2)CC)CC(C)N(C)CC1C 26561,N1(C(c2n(CC)ncc2)=O)CCN(C(c2nocc2Cl)=O)C(c2cccnc2)C1 26562,N1(CCC)CC(C(=O)NC(C2CCN(C(=O)Cn3cncc3C)CC2)C)CC1=O 26563,N1(C(c2c(NC(C)C)cccc2)=O)CC2CCC1C(CNC(C1(C)CC1F)=O)C2 26564,c1(OCC)cccc(C(=O)NCC(CO)NC(c2cc3scnc3[nH]2)=O)c1N 26565,C1(CC=C)(NC(c2ccc(F)o2)=O)CCN(C(C2OCC2(C)C)=O)CC1 26566,S(=O)(=O)(CC(=O)NCC1(F)CC(NC(c2cccn2CC)=O)C1)NCC 26567,CCC(CCCC(=O)N1CCN2CCC1C2)NC(C1(O)CCSC1)=O 26568,c1(CC(=O)OCC)csc(=NCc2c(Br)cnn2C)[nH]1 26569,c1(C(=O)NCCN(C2CCCCCC2)C(CC(C)OC)=O)cn(C)nc1Cl 26570,C1(CNC(CC(C=C)C)=O)CCC2(CCC2)CN1C(=O)C(c1ccn(C)n1)C 26571,C(=O)(C#CC(C)(C)C)NC1(CC(=O)NCc2nnn(CC)n2)CCCCC1 26572,CCS(=O)c1ccccc1C(N1CCN(C(=O)CP(C)(C)=O)C(CC2CC2)C1)=O 26573,C1(c2cn(CCOC)nn2)C(C)CCN1C(c1ccc(C(C)=O)s1)=O 26574,c1(OC)ccc(S(=O)(=O)N2CCOCC2C2CC2)cc1CC(=O)O 26575,CCCCCC(F)C(=O)N(CC(N1CCc2ncsc2C1)=O)CCOC 26576,C1(CC)CN(Cc2ncn(C(C)C)n2)CCN1C(=O)CC1CCCN1 26577,c1(NCCCSC(C)(C)C)ccc(C(F)(F)Cl)cc1 26578,N1(C(CCCOC(C)(C)C)=O)CC2(C=C(C(=O)N3CC(F)CC3CO)CO2)C1 26579,C1(C(N(CC(F)F)C)=O)CCN(C(=O)COCC2CCCO2)CC1(C)C 26580,C1(O)(CCNC(CCN(C(C2C(C)(C)C2)=O)CCO)=O)CCOC1 26581,c1(OC)ccc(N)c(C(=O)NCC2CCCN2C(=O)CCC(C)(C)OC)c1 26582,C1(C)(C(=O)NC(c2ccncc2F)C)CC(C#N)C1.C12CCC(O1)C(=O)NOC2 26583,N1(c2nnc(C(CC)(C)C)o2)CC(C)CN(C(c2ccc([N+](=O)[O-])s2)=O)CC1C 26584,c1(C(N2CCCC(N(C(c3cc(OC)cs3)=O)CC)C2)=O)cc(C)c(C)cn1 26585,c1(C(N(CC(C)NC(C2(SC)CCCCC2)=O)CC)=O)cc2cc(C)ccc2[nH]1 26586,C(=O)(CC1=CCOCC1)NCC1C(NC(C(C)(c2cccs2)N(C)C)=O)C1 26587,C(=O)(C(C)S(=O)(=O)C(C)C)N1CCC(OC)(CNC(C2(CO)CC=CC2)=O)CC1 26588,c1(-c2nc(C(CC)C)nn2C2CCCC2(C)C)cc(F)cc2nccnc12 26589,C1(CNC(CCC)=O)CCC12CCN(C(=O)COc1ccc(Cl)cc1C)CC2 26590,C1(=O)C(c2ccccc2)CN1.S(C)(=O)(=O)N(CCN(CC)CC)C(C)C 26591,c1(NC(C2CC2C(=O)Nc2cc(Br)cnc2Br)=O)c(Cl)cnnc1Cl 26592,c1(NC(C2(C)CN(C(c3c(C#C)cccc3)=O)C2)=O)cc(Br)c(F)cc1C 26593,N1(C(CCC(C)C)=O)CCN(C(c2cc3n(n2)CCNC3=O)=O)C2COCC12 26594,c1(C(N2CCC(CNC(c3c(CC)scc3)=O)C2)=O)n[nH]c2c1COC2 26595,N1(C(C(C=CC)O)=O)CCC2CCCC12C(=O)NC1CCC2CCC12 26596,N1(C(C(CC)C)=O)CCC2CN(C(=O)C3=C(C)OCC3)CC2CC1 26597,N1(C(CCC(C)(C)NC(=O)C2CCc3c[nH]nc32)=O)CC(O)C2(CCCC2)C1 26598,C(=O)(C(F)(F)C(C)(C)O)N(C(C)CN(C)C)C.C(c1ccccc1)=CCC1CC1 26599,C1(F)(CNC(Cc2cc(C)sc2)=O)COCCN(C(C2COCC2(C)C)=O)C1 26600,C#CCC(C)(CC)C(=O)NCCN(C(c1cnc(C2CCC2)o1)=O)C(C)C 26601,C#Cc1ccc(C(=O)NC(Cn2cncn2)C(=O)NCC2C=CCC2)cc1 26602,Cc1c(O)ccc(C(=O)NC2CCC2CNC(=O)C(C2CCC2)C2CCC2)c1C 26603,c1(C(=O)NCC23N(C(C4C(C)(C)CCC4)=O)C(CC2)CC3)ccsc1S(C)(=O)=O 26604,c1(C(=O)NC(C(C)NC(=O)C(F)OC(F)(F)F)CO)ccn(C)c1C1CCC1 26605,c1(NC(C2CN(Cc3cccc(F)n3)CCC2O)=O)cccc2nc(O)ccc12 26606,CC1(C)CCN(C(c2cncnc2)=O)CC1NC(c1cc(-c2ccoc2)[nH]n1)=O 26607,c1(CNCC(c2ccc(F)cc2)OCC)cc2ccncc2[nH]1 26608,c1(-c2nc(CC(c3cccc(Br)c3)OCC)oc2)nc(CSC)nn1C1CC1 26609,c1(CC(=O)N(C(C)CCNC(=O)CCC2CC2(C)C)C)cncnc1O 26610,C1(C(=O)OC(C)(C)C)CCCCN1C(=O)NC.C1(C(=O)NCC(C)N)CNC(=O)C1 26611,N1(C(c2c(C)con2)C(=O)NC(c2ccccc2)C)CC(C)(C)C1C(C)C 26612,C1(C(=O)NC(c2ccsc2)C)CN(C(=O)C(=O)NC2CC2)CCC1(C)C 26613,c1(OC)cc(C(=O)NCC2(CNC(=O)C(C)N(C)C)CCC2)cc(Br)c1 26614,C12(C(=O)NC3C(NC(CC=CC=C)=O)CCCC3)CCC(CC)(C1)OC2 26615,C(C(=O)Nn1cnnc1)(C(C)CC)NC(c1cc(=NC)[nH]cc1)=O 26616,C(=O)(CCC(C(C)C)NC(c1ocnc1C1CC1)=O)N(CC(=C)C)CC(=C)C 26617,C1(N(C(=O)COC2CCC2)CCO)CCN(C(C2CCOC2c2ccccc2)=O)C1 26618,N1(C(c2n(CC)ncc2)=O)C2CCC1C(NC(=O)Cc1nn(C)cc1Br)C2 26619,N1(C(c2c(C)n(C)nc2)=O)CCC2(CCCN2C(=O)CCCc2cccs2)C1 26620,CC(C)CC(C(=O)NC(CNC(C1(n2ccnn2)CC1)=O)C(C)C)N(C)C 26621,C1(C)(CC)CC(C(=O)N(CCNC(c2coc(C3CC3)n2)=O)CC)CCO1 26622,c1(C(=O)NC(CC)CNC(=O)C(C(C)C)NS(C)(=O)=O)ccc2nc(C)oc2c1 26623,S(=O)(=O)(c1ccc(Br)cc1N(C)Cc1cccc(Cl)c1)NCC1OCC(C)C1 26624,N1(C(CCC(=O)NCC)=O)CC(NC(C2CC=CC2)=O)CC(F)C1 26625,c1(C(=O)NC(C)CCNC(C2(CO)CC2)=O)cn(C)cc1C(F)(F)F 26626,C12(C(=O)NCC3N(C(c4c(C)n[nH]c4C)=O)CCC3)CCC(CC1)C(C)O2 26627,N1(C(Cn2ccc(C)n2)=O)CC(NC(c2ccc(-c3ccco3)s2)=O)C2(CC2)C1 26628,c1(C(=O)NCC(CC)NC(=O)C(O)CC2CC2)cc(F)n(C)n1 26629,N1(C(CCC=C)=O)CC2CC(C(=O)NCCc3cccnc3OC)C(C2)C1 26630,C(C1=CCN(C(=O)C2=CCCOC2)CC1)NC(CCCc1ccc(CC)cc1)=O 26631,N1(C(Cc2ccc(C)o2)=O)CC2CN(C(=O)CC3CC(N(C)C)C3)CC(C1)O2 26632,c1(C(N(CC(O)CNC(=O)CN2CCNC(=O)C2)C)=O)cc2nc[nH]c2cc1F 26633,N1(C(CC)=O)C2CCC1CC(CNC(c1ccccc1O)=O)C2 26634,C(=O)(C(C)(CC)C(=O)OCC)NCCC1CCN(C(CC=CC=C)=O)C1 26635,c1(C(N(CC(C)NC(=O)CC2OCCC2C)C)=O)cnn(CCF)c1 26636,CCC(CC(C)C)C(=O)N1CC(C(=O)NCc2ccccn2)C2(CC2)C1 26637,Cc1ccc(Br)c(C(=O)NC23CC2CN(C(=O)COCC(C)(C)C)C3)c1 26638,C1(CNC(c2c(C)nco2)=O)CN(C(C2CC2c2sccc2C)=O)CC12CCC2 26639,c1(NC(C(=O)NCCCCSC)=O)ccc(Br)cc1-n1cncn1 26640,C1(C2(O)CN(C(c3nccc(Cl)c3F)=O)C2)(CNC(C2CCC3(CC3)C2)=O)CC1 26641,CN1CCCC(C)(C(N2CC(NC(C3CCCN3N=O)=O)C(C)(C)C2)=O)C1 26642,C1(NC(C(C)=C(CC)C)=O)CC(CNC(=O)C(F)=C(C)C)C12CCC2 26643,c1(CC)[nH]c(C(=O)NCC(C)(CO)NC(c2cc(C)nn2C)=O)nc1Cl 26644,c1(NC(C2(F)CN(C(CCOCC)=O)C2)=O)ccccc1N(C)C 26645,C1(CNC(C(=O)NCc2n(C)nnc2)=O)CCC(C)(C)CO1 26646,c1(CC)cccnc1-c1nc(CC2CC3(CC3)C2)nn1-c1ccc(C(C)C)cc1 26647,c1(CC)noc2ncc(C(=O)NC3CC4CC(C3)N(CC(C)OC)C4)cc12 26648,Cc1cnc2n1CC(C(N1CC(N(C)C(C3SCCCS3)=O)C3(CC3)C1)=O)CC2 26649,N1(C(=O)CC2(O)CCOC2)Cc2n[nH]cc2C1C(=O)N1CC2CCCC2C1 26650,c1(C(COC(C(C)(C)C2CCOC2)=O)=O)ncn2c1OCC2 26651,c1(OC)ccc(C=NOCC(=O)NC2CC2CNC(=O)Cc2cc(C)cs2)cc1 26652,c1(OC)cc(C)c(C(N2CCCC(C)(NC(C3CC4(CC4)CO3)=O)C2)=O)cn1 26653,N1(CC(=O)NC(C(=O)NCCC(=O)NC(C)C)C2CC2)CCCCC1=O 26654,c1(CCN(C(C(=O)NCCO)C2CC(OCOC)C2)C)ccc(F)cc1.COC 26655,C1(NC(c2cncc(C)c2Cl)=O)CCN(C(=O)CCOCC2CC2)CC1(C)C 26656,Cc1nn(C)cc1C(=O)N(CCCNC(=O)C(C)Sc1ccc(Cl)cc1)CCO 26657,CC(C(O)C(=O)NC1(C(=O)Nc2ccc(N(C)C)nc2)CCC1)c1ccccc1 26658,c1(N)c(I)cc([N+](=O)[O-])cc1I.C(=O)(CCCCCCCO)C(=O)CC1CNC1 26659,N1(C(C(C2(O)CN(C(c3cnn(C)c3Cl)=O)C2)F)=O)CC2(CNC(=O)C2)C1 26660,C1(C(N(C)CC2N(C(CCc3cc(OC)no3)=O)CCC2)=O)CC(C)OC(C)C1 26661,N1(C(c2c(F)ccc(C)c2O)=O)C2CCC1CC(F)(CNC(C1CC13CC3)=O)C2 26662,C1(C(N(CC(=O)NCc2c(C)scn2)C(C)C)=O)CCCC(F)C1 26663,N1(C(CNC(COC)=O)=O)CCC(c2n[nH]c(CNC(=O)C=CC3CC3)n2)CC1 26664,C(=O)(C(O)CC(C)(C)C)NCC1(C(C)(C)O)CN(C(C=C(CC)CC)=O)C1 26665,C1(CNC(COCC#C)=O)CCN(C(=O)Cc2cc(C)no2)CC1CC 26666,N1(C(C(C2CC2)NC(c2cc(C)c(C)nc2)=O)=O)CC2(C1)CN(C)CCO2 26667,c1(C(=O)NC23CCCC(NC(CC=CC)=O)(C2)C3)ccc(Cl)c(F)c1N 26668,c1(N2CCCC(CN(C(C3(OC)CCCOC3)=O)C)C2)cccc(F)c1[N+](=O)[O-] 26669,C12(CC13CCC3)C(=O)NC2.C12(CNC(C3CN(C(=O)NC)C3)=O)COCC1C2 26670,c1(C(=O)NCCN(C(CN(C)CC)=O)Cc2ccccc2)cc(C(C)C)nn1C 26671,N1(C(c2nccc(C)c2)=O)C2CCC(C2)C1CNC(=O)COCc1ccccc1 26672,c1(C(N(CCN(C(=O)Cc2cc(Cl)ccc2F)C)C)=O)cncc([N+](=O)[O-])c1 26673,N1(CC(N2C(C(N3CCC(CO)C3)=O)C=CC2)=O)C(=O)CCC1=O 26674,C(=O)(C1OCCc2ccccc21)N(CCNC(CC(C)OC)=O)CC1CC1 26675,C=Cc1ccc(C(=O)NCCCC(C)NC(=O)C(C)(C)C#N)cc1 26676,C1(NC(C(COC)C)=O)CN(C(C2CC(S(C)(=O)=O)C2)=O)CC12CCC2 26677,Cc1cc(C(N2CC(NC(=O)C(=O)NCC(F)F)C2)=O)c(C)cn1 26678,C1(CN(C(C(C)NS(CC)(=O)=O)=O)C)CN(C(c2cc(Br)n[nH]2)=O)CCO1 26679,C#CCC(CC(=O)N1CCCC1C(C)CC)NC(c1cc(O)ccc1F)=O 26680,N1(C(CCCC(C)C)=O)CC2(CCN(C(=O)C(c3ccccn3)C)C2)C1 26681,c1(C(=O)OC2CCN(CC(C(=O)NC)O)C2)ccc(F)cc1Cl 26682,C12(NC(c3c(C)nsc3)=O)CCN(C(c3cnc(N)cn3)=O)CCC1C2 26683,C1(CCN(C(COCc2onc(C)n2)=O)C)CCCCN1C(C1CC1F)=O 26684,CC1CC2(CC2)CN1C(C1OCCC1CNC(=O)Cc1cccnc1O)=O 26685,S(=O)(=O)(c1ccc(I)cc1)N1CCN(C(C(C)=O)=O)C2C1C2 26686,N1(C(C(CCC)(C)C)=O)CCC2(CC1)CC(CNC(=O)CC(C)CC)C2 26687,C1(NC(C2(CC)CCCO2)=O)CCC(O)CN(C(c2cc(C)no2)=O)C1 26688,C=CCCCC(C(=O)NCC1CN(C(=O)OC)C1)NC(=O)C(C)CC(=C)C 26689,CC(C)(C)CC(O)C(=O)NC(c1cccc(O)c1)CO 26690,c1(CCC(=O)NCCC2C(C)CCO2)nc2ccccc2oc1=O 26691,N1(C(c2c(SC)ccs2)=O)CCOCC1CNC(=O)C(C)Oc1ccc(F)cc1 26692,c1(C(N2CC3N(C(C(C(C)C)SC)=O)C(CC3)C2)=O)n[nH]c2c1CC(F)(F)CC2 26693,C(CN=c1cc[nH]cc1S(=O)(=O)N1CCC(C)(CO)C1)N(C)N(C)C 26694,C(CC(=O)NC1CC(NC(=O)C(C)=C2CCC2)C1)=CCC 26695,c1(C(=O)NC(C)CCNC(C2COCCN2C)=O)cccc2nc(O)[nH]c12 26696,c1(C(=O)NC2(C)CCN(C(C(C(C)(C)O)F)=O)C2)cc(O)c2ccoc2c1 26697,c1(C(c2n(C(C(=O)OC)C)nnn2)NCCC(N)=O)ccc(OC(F)F)cc1 26698,C1(C(N(CC(F)F)CC)=O)CN(C(=O)CCC2(C)CC2)CC1C(C)C 26699,N1(C(C=C(CC)C)=O)CC2CC3CC2C1C3NC(=O)CCc1ccccc1OC 26700,C1(NC(C2C(C)=CCS2)=O)CCN(C(=O)CCc2ncnn2C)CC1O 26701,c1(C(C)OC(C)=O)nc(-c2cccc(Cl)n2)nn1CC(C)C 26702,C(C(F)(F)C(=O)O)N(C(=O)C(c1ccc(F)cc1)CO)C 26703,C1(C(N(C2(C(=O)NC3(CCO)CCOC3)CC2)C)=O)CCCCC1(F)F 26704,C(CC(C)(C)CC(=O)NCC1(CNC(c2cc(C3CC3)cnn2)=O)CCC1)OC 26705,C1(NC(=O)CCC2CCCCO2)CCN(c2nnc(C(F)F)o2)CC1O 26706,Cc1cccc(C(N2CC(CNC(=O)Cc3ccc(F)cc3)C3CC23)=O)n1 26707,C=CCCCC(C(=O)NC1CCn2nnnc2C1)NC(C1CCC1)=O 26708,Cc1cn2cc(C(=O)NCC3(CNC(c4cn(C)nc4C)=O)CC3)sc2n1 26709,c1(CCNC(=O)NC(c2ccccc2Cl)C)c[nH]c2ccc(O)cc12 26710,Cn1cnc2c(C(=O)Nc3cccc(Cc4ccc(C#N)cc4)c3)ccnc12 26711,CCC(CCOC)C(=O)N1CC(OC)C(C(=O)NCCCCN(C)C(C)C)C1 26712,C1(COC)(CNC(=O)Cc2ccccc2C)CCCN1C(=O)C(C(C)C)NC=O 26713,N1(c2ncc(C(=O)OCC)nc2)CCN(C(=O)CN(C2CC2)CC)C(C)C1 26714,CC1(C)CN(C(C2CCCCS2(=O)=O)=O)CCC1NC(c1cc(F)cnc1Cl)=O 26715,c1(C(=O)NCCC(=C)CNC(=O)CCCN=[N+]=[N-])ccc(S(=O)(=O)C(C)C)cc1 26716,N1(C(CC=C=C)=O)CCC(C2CCN(C(c3cc(C#N)c[nH]3)=O)CC2)C1 26717,Cn1cc(CNC(=O)C(C2CC2)NC(c2cnns2)=O)nn1 26718,C(=O)(C1=CCC(C)CC1)N(CC(CNC(CCC#C)=O)(C)C)CC 26719,c1(COC)ccc(C(=O)N(CC(O)CNC(c2cc(C)ccc2O)=O)C)cc1F 26720,C1(NC(C(CC=C)C)=O)CN(C(c2cccc(F)c2NC)=O)Cc2ccnn2C1 26721,N1(C(c2c(CC)c[nH]n2)=O)CCCCC1C1(NC(c2ccc(C)n2C)=O)CC1 26722,N1(C(C2CC(C(=O)OC)C2)=O)C2CCC1CC(CNC(c1occ(C)c1C)=O)C2 26723,C1(NC(CC(CN(C)C)O)=O)CCN(C(c2cc(F)ccc2Cl)=O)C12CC2 26724,C(=O)(C1=CCCCC1C)NC(CN(C(c1c(OC)cc(O)nc1)=O)C)C 26725,C=CCC(C)C(=O)N1CCOC(CCCNC(=O)CCc2nncs2)C1 26726,c1(C(C(=O)NCCCNC(CC(C)CN(C)C)=O)O)ccc(Cl)c(Br)c1 26727,c1(C(=O)NCC(CNC(c2ccn(CC(C)C)n2)=O)F)cccc2c1CCOC2 26728,c1(C(N2CC(C(N)=O)(CNC(C3C(CC)CCC3)=O)C2)=O)nc(CC)ncc1Cl 26729,C(C(C)(C)CC(=O)N1CCC(N(C)C(c2ncccc2O)=O)C1)OC(C)=O 26730,C1(C(=O)NCC=CC(=O)N(CCCCC=C)C)CC2(CC2)CO1 26731,N1(CC)C(=O)CCC1CC(=O)NC1CN(C(C2(c3n[nH]cc3C)CC2)=O)CC1O 26732,C(=O)(CCCC(=O)NC12CC(CC(C)C)(C1)C2)NN1CCCC1C(=O)NC(C)C 26733,N1(C(C(C)C)=O)Cc2ccc(O)cc2CC1C(=O)Nc1ccc2ocnc2c1 26734,c1(C(N(C2CCN(C(=O)COc3cccnc3)C2)CC)=O)ccc2cccnn12 26735,c1(C(N2CC(NC(C3C(C)(C)CC3)=O)CC3(C2)CC3)=O)[nH]c2ccccc2c1Cl 26736,CC(C(=O)NO)NC(c1nc(CO)cs1)c1nnnn1C1CCC1 26737,c1(CC(C(N2CCC(CNC(C3CC(CF)C3)=O)C2)=O)O)cc(Cl)cc(Cl)c1 26738,C(=O)(CS(=O)(=O)C12CC(C1)C2)N(C)CC1(O)CN(C(C2CC(C)C2)=O)C1 26739,c1(C(N(CCNC(=O)Cc2sc(O)nc2O)CC)=O)c[nH]c(C)c(Br)c1=O 26740,C1(C(N2CC(C)(CC=C)C2)=O)CCCCCC1NC(c1nc(Cl)oc1C)=O 26741,Cc1snnc1C(=O)N(CCNC(C1CC(C(F)(F)F)CO1)=O)C1CC1 26742,N1(Cc2cc(C)sc2C)CC2(CCC(CNC(C3(C(F)F)CCOCC3)=O)O2)C1 26743,c1(CC(=O)N(CCC(=O)NC(C=C)C2CC2)C)cc(C)on1 26744,c1(CNC(CC)=O)ccc(CN(C(=O)CC=CC(C)(C)C)C)cc1 26745,c1(C(=O)NC2CN(C(Cn3nnc(C)n3)=O)C(C)CC2)cnn2ccc(O)nc12 26746,N1(C(C(COC)N(C)C)=O)CC(CNC(=O)Cc2c(C)n[nH]c2C)C(C)C1 26747,c1(C(=O)NCCNC(C(N2CCCC(O)C2)C)=O)c(Cl)cc(Br)cc1Cl 26748,c1(CC(=O)NCCCN(C(=O)CNS(C)(=O)=O)C(C)C)nccc2ccccc12 26749,C1(NC(C2CCCN2C(c2ncccn2)=O)=O)CCOC12CCCC2 26750,c1(C(n2cc(CC3CCN3C(=O)NCC3CCCC3)nn2)C)ccccc1 26751,C(CC(C)(C)C#N)(c1n(CCOC)nnn1)NCCC(=O)NCC(C)C 26752,COn1cnc(C)c1C(=O)NC1CC(=O)N(C2CN(C(C3CC3C#N)=O)C2)C1 26753,n1(CC)ncc(Cl)c1C(=O)NCC(O)CN(C)C(C1CC1C(C)(C)C)=O 26754,N1(C(CSCCC(C)C)=O)CCCCCCC1C(=O)N(C)CC1CC1C 26755,c1(OC)cc(Br)c(NC(C2CC2C(=O)NCC(C)(C)C(N)=O)=O)cc1C 26756,C(=O)(C(C(C)(C)C)N1CCNC1=O)N1C(C)C(NC(c2cc(N)ccn2)=O)CC1 26757,n1(C(C)(C)C)nnc2c1CCC(C(=O)Nc1ncc(O)c(=N)[nH]1)C2 26758,c1(C(N2CCC(C)(N3CCCC3)C2)C(=O)NCCC)cc(Cl)cc(Cl)c1Br 26759,O=S1(=O)CCC2(CCN(C3CCN(c4c(Cl)cccc4Cl)C3=O)CCO2)CC1 26760,Cn1nnc2c1CCC(C(=O)NCC1(C)CC(NC(c3cnc(Cl)s3)=O)C1)C2 26761,CC1CN(C(=O)CCc2cccc(C#N)c2)C(C)CN1C(=O)CCc1nc[nH]n1 26762,c1(CC(N2C(CNC(C(C)CC(C)(F)F)=O)CC2)=O)cc(F)cc2c1OCOC2 26763,C(=O)(CC(C)CF)NC(C)CCN(C)C(c1c[nH]nc1-c1cnn(C)c1)=O 26764,N1(C(C(C)N(C(c2c(CC)c[nH]n2)=O)C2CC2)=O)CC2(C1)OC(=O)NC2C 26765,C=CCC(C)(C)CNC(c1conc1C(C)NC(c1cnccc1OCC)=O)=O 26766,CN=c1cc(C(N2CC=CC2CNC(=O)C(COC)COC)=O)cc[nH]1 26767,CC(CC(=O)N1CCN(C(=O)C(C)(C)N=[N+]=[N-])CC12CC2)CC(C)(C)C 26768,C1(C(=O)NCC(COC)OC)CC12CC(NC(c1ccc(=N)[nH]c1)=O)C2 26769,N1(C(c2c(C)scc2)=O)CC2COCC2(C(=O)N(CC(C)C#N)C2CC2)C1 26770,Cc1cc(C(=O)N(CCC(=O)N(C)Cc2ccco2)CCO)nc(O)c1 26771,c1(-c2c(C(N(C(C)C)CCc3ccccc3)=O)ccnc2)ccc(F)c(CO)c1 26772,Cc1nc(O)nc(C)c1C(=O)NC1CC(C)N(C(c2ccc(N)c(Cl)n2)=O)C1 26773,CC1CN(C(c2cc(O)nc(O)c2)=O)CCC1NC(=O)CCc1ccc(N)cc1 26774,C(=O)(CCCC(=O)NCc1cnc(Cl)cc1F)NC 26775,CC1CN(C(C2CC2c2ccccc2)=O)CCC1NC(c1cnnn1C)=O 26776,C1(F)(C(=O)NCC(C(C)C)NC(=O)Cn2cnc(C(N)=O)n2)C2CCCC12 26777,N1(S(CC)(=O)=O)CCCC(C(=O)NC(C)CNC(=O)CC2COCCO2)C1 26778,c1(CN2CCC(NC(CCC)=O)CC2)cc(CN=[N+]=[N-])cc(N=[N+]=[N-])c1 26779,N1(C(C2CC(F)(F)C2)=O)CCCC(NC(C2(CC3CC3)CC2)=O)C1 26780,C=C(Cl)CCC(=O)NC1CCN(C(c2cncc(N(C)C)n2)=O)C1 26781,N1(C(C(C)C=Cc2ccccc2)=O)CC2CCC1C(NC(=O)C(C)(F)F)C2 26782,N1(C(C2C(CC)OCC2)=O)CCC2(CC1)CC(NC(c1cc(Br)nn1C)=O)C2 26783,c1(C(=O)NCC(CNC(=O)C(O)Cc2ccccc2)OC)ccnc2c1CCO2 26784,C(=O)(C(CC(C)C)C(C)C)NCC1(Nc2nc(CC)nc(C)c2)CCCCC1C 26785,c1(C(=O)NCC2(O)CN(C(=O)CCc3cn[nH]c3)C2)csc2cccc(F)c12 26786,c1(C(=O)NCC2(C(C)(C)C)CN(C(=O)CC3CCCC3(F)F)C2)cccc(=O)n1C 26787,c1(C(N2C(C)(CNC(C(CCCC)C)=O)CCC2)=O)cn2nc(OC)ccc2n1 26788,CC1CC(C(=O)NC2CCC(CNC(=O)COc3cnn(C)c3)CC2)=NO1 26789,N1(C(c2c(C)nc(C(F)(F)F)o2)=O)CCC2C(C1)CN2C(=O)Cn1nnc(=O)[nH]1 26790,C1(CC)CC(C(=O)NCC(C)(C)NC(c2ccc(CCOC)cc2)=O)CC(=O)N1 26791,C(=O)(C(C)(CC)CO)NCCn1cc(-c2ccc(C3C(C(=O)OC)C3)cc2)nn1 26792,c1(C(N2CCCC(NC(C(CC)NC(C)=O)=O)C2)=O)cc2cccnc2[nH]1 26793,CCC1=NOC(CC(=O)NCC2C=CCN2C(c2csc(C)c2)=O)C1 26794,Cc1ncc(C(=O)NC(C2CCCC2)CNC(=O)C(F)Cc2ccccc2)[nH]1 26795,N1(C(c2c(C(C)=O)ccs2)=O)Cc2nccn2CC(NC(C2CN(C(C)=O)C2)=O)C1 26796,c1(C(C(=O)NCC(CNC(COC(CC)(C)C)=O)C)C)cccc(F)c1 26797,c1(CC(=O)NCCCC(C)NC(C2OCCCO2)=O)c(Cl)cccc1Br 26798,O=C(CN=c1cc[nH]cc1)NCCC(O)CNC(c1ccc(O)nn1)=O 26799,N1(C(COCC)=O)CCN(C(C23CCC(CO2)C3)=O)CC1C1CC1 26800,S(=O)(=O)(c1ccc(=NCc2ccnc(OC)c2)[nH]c1)NC(c1ccccn1)CC 26801,c1(NC(C(C2CCN(C(c3cccc(C)c3)=O)CC2)C)=O)cc(Br)c(Cl)cc1F 26802,C1(CC(=O)NC2(CCNC(C=CC(=O)OCC)=O)CCC2)CCOC1(C)C 26803,C(=O)(C(C#N)C(C)(C)C)N1CCN(CCC(C(C)C)(F)F)CC1 26804,c1(CC(N2CC3CCN(C(COCCC#C)=O)C3C2)=O)oc2ccccc2c1C 26805,CCC(C)(CC1CCCCC1)C(=O)N1CCN(C(=O)C(F)F)CC1 26806,c1(-c2c(C(=O)NCC(C)NC(=O)Cc3cccnc3N)c[nH]n2)ccccc1F 26807,N1(C(C(C#C)(C)C)=O)CCC2CCN(C(C3CNC(=O)C3)=O)C2C1 26808,C=CC(C)(O)CCCC(C)C(=O)N1CCCN(C(c2cc(Br)co2)=O)CC1 26809,C(=O)(C1=C(C#N)CCC1)N1CC2(C1)C(=O)N2.C(C(=O)OC)(C1CC1)OC 26810,c1(C(CC(=O)Nc2cncc(Cl)c2)NC2C(OCC)CCC2)ccc(F)c(F)c1 26811,c1(C(N(C)CCNC(=O)CSCC(F)(F)F)=O)cccc2c1COC2 26812,C(c1cccnc1)=CC(N1C(C(C)NC(C2CC=CCC2)=O)CCC1)=O 26813,C(CCC(C)(F)F)N(C(=O)CN(C(=O)CC1CC2CC2C1)C1CCC1)C 26814,C12(CNC(=O)CCn3ccnn3)CC1CN(C(c1nccnc1C(F)(F)F)=O)C2 26815,C(CN=c1[nH]c2c(c(=NCCCC3CC3(Cl)Cl)[nH]1)CC(C)CC2)c1nc(C)sc1 26816,O=C(Nn1ccnn1)C1C(c2ccccc2O)C1(F)F 26817,C(=O)(C(CC(C)C)CC(C)C)N1CC2(NC(C(CC=C)(C)C)=O)CC1(COC)C2 26818,C=C(Cl)CCC(=O)N1CC(CNC(c2cnc(-c3cnn(C)c3)s2)=O)C(C)C1 26819,C(CC1=CCN(C)CC1)NC(C1(CC#C)CCN(C(C2CCN(C)C2C)=O)C1)=O 26820,Cc1ccc(C(=O)CCC(=O)N(C)CC2CN(C(c3cnccn3)=O)C2)cc1 26821,Cc1onc(C(=O)NC2CCN(C(c3cnn(CC(F)F)c3C)=O)C2)c1[N+](=O)[O-] 26822,Cc1cc(C(=O)NCC2CN(C(c3ccc(F)cc3)=O)CCC2C)cc(C)c1O 26823,C#CCCCC(=O)N1CCN(C2CN(Cc3cnc(Cl)nc3)C2)CC1 26824,C(=O)(C(C)C(O)C(C)CC)N1C2C(C(=O)NCCCCC)CC(C=C2)C1 26825,C1(CNC(=O)CSCc2ccccn2)COCCN(C(=O)Cc2cn[nH]c2)C1 26826,N1(C(=O)N)CC(CCO)OCC1C.c1(C(NOC)=O)ccc(C(N)=O)cc1 26827,N1(C(c2c(C)ccnc2)=O)CCC(NC(=O)C(F)(F)c2csc(Cl)c2)C(O)C1 26828,c1(NC(C(c2cc(C)ccc2I)N(CCC(N)=O)CC)=O)c(C)cccc1C 26829,C1(C)(C(=O)NC2CCC(N(C(C=C(C)Cl)=O)C)C2)COC(=O)OC1 26830,CCC(C)C(C)C(=O)N1CCC(NC(=O)CCN(C(=O)C(C#N)CC)C)C1 26831,C(C1=NOC2CN(C(c3cc(C#N)c[nH]3)=O)CC12)NC(CSC(C)C)=O 26832,N1(C(C(C2CC2)OC)=O)CC(CNC(=O)CN(CC(=O)NC(C)C)C)C2(CC2)C1 26833,C(CC(=O)NC1CCC1CC1CCC1)(OC)OCC.C12CC1CCNC2=O 26834,CCC(C)C(C(=O)NCC=CCNC(=O)C(c1ccc(C(F)(F)F)cc1)O)OC 26835,N1(C(CCCCOCCC=C)=O)CC2(C1)C(NC(=O)C(O)C1CC1)CCS2(=O)=O 26836,Cc1cccc(CO)c1C(N1CCC(CO)C(NC(=O)C(F)n2ccnc2)C1)=O 26837,CCC(C(=O)NC(CNC(=O)C(C)C(=O)N1CCOCC1)(CC)CC)C(C)C 26838,CCC(C)(C#N)C(=O)NCCCOCCCNC(C1CCCC(C(N)=O)C1)=O 26839,C1(C(=O)NC(c2ccccc2)CNC(c2ccoc2Cl)=O)CCCCO1 26840,N1(C(C2C=CCC2)=O)CCN(C(=O)Cc2ccon2)C(c2ccccc2Cl)C1 26841,Cc1cc2cc(C(=O)NCC34CC3CN(C(C3(O)CC3)=O)C4)c(Cl)cc2[nH]1 26842,C1(C(=O)NCC2N(C(CC3(C=C)CC3)=O)CC(C)CC2)(CO)CC2CCC1CC2 26843,N1(CC)CC(C(=O)NCC(C2CC2)N(C(=O)CN2C(=O)CNC2=O)C)CC1=O 26844,O(P(C)(=O)CNC(C1(OC)CCN(C(=O)C(C2CC2)OC)C1)=O)CC 26845,C1(C(=O)NCCCN(C(c2coc(CO)c2)=O)CC)CC(C(F)(F)F)CO1 26846,C1(NC(C2CCC3CC23)=O)CN(C(c2cccc3[nH]ccc23)=O)CCC12CCC2 26847,N1(C(Cc2cc(OC)no2)=O)CCCCC(CNC(c2cc(OC)cc(C)n2)=O)C1 26848,C(C(CC(C)C)NC(c1ccc(C(C)(C)C)o1)=O)NC(C1(COCC)CC1)=O 26849,C1(C(N2CCN(CC)CC2)=O)CNC(=O)CN1C(c1ccc[n+]([O-])c1)=O 26850,C1(CNC(C=CCCC)=O)CC2CCC1N(C(C1CCC1OCC)=O)C2 26851,c1(NC)ccc(Cl)c(C(N2CCC(NC(C3CCCC34CCC4)=O)C2CO)=O)c1 26852,N1(C(C(C)CC2CCC2)=O)CC2(CCCN(C(=O)C=CC3(C)CCOCC3)C2)C1 26853,c1(OCC(=O)NC(C2(F)CCN(C(=O)CN3CCC3C)C2)C)ccc(F)nc1 26854,c1(C(=O)NC(C)CC2CN(C(=O)CN3CCCC3=O)C2)ccc(CF)cc1 26855,c1(NC(c2cc(-c3cc(C)cc(F)c3F)ncc2)=O)ccc2ncnc(O)c2c1 26856,C#Cc1ccc(C(=O)NC(CNC(c2cccn2C)=O)CC)o1 26857,c1(C(N2CC(NC(c3nc(CC)oc3C)=O)C(C(F)F)C2)=O)cc(C)nc(O)n1 26858,C1(C(=O)Nc2c(C)ncnc2)CC2CCC1N2C(C1CCC1C#N)=O 26859,N1(C(C(C=C)O)=O)CCC(CCCCNC(=O)C(n2ccc(C)n2)C)CC1 26860,S(=O)(=O)(c1cc(C(=O)NC2CC3(C2)CN(C(C24CC(C)(C2)C4)=O)C3)co1)NC 26861,Cc1cc(C(N2CCC(C)(NC(=O)CC3CCC(C)(C)O3)C2)=O)ccc1Cl 26862,c1(C(=O)NCC2C(NC(c3cc4[nH]ccc4s3)=O)C2)cc2cc(Cl)cnc2[nH]1 26863,CCC(C)(COC)C(=O)N1CCCC(CNC(c2nocc2C)=O)CC1 26864,C(C(=O)NOCC(N1CCC(C(C)(C)C)C1)=O)=CC 26865,C1(C)(COC)CC(NC(C2(CCF)CC2)=O)CN1C(c1ccc(C)cc1C)=O 26866,c1(NC(c2c(C)cccn2)C)nc(N(C)CC2CCC(=O)N2)c2ccsc2n1 26867,N1(C(c2cc(C)cnc2OC)C(=O)NCC=C)CCc2n[nH]cc2C1 26868,N1(c2c3ncn(C(C4CCC(C)C4)CO)c3ncn2)CC=C(c2cccs2)CC1 26869,CC1CN(C(CN(C)Cc2ccc(OC(F)F)cc2)=O)CC(C)O1 26870,C1(NC(c2cc(CC)oc2C)=O)(CO)CCCN(C(=O)C(F)=C(C)C)C1 26871,c1(CNC(CCC=CC)=O)ncccc1C(N1CCC(Cc2ccccc2)C1)=O 26872,c1(OC)cc2c(cc1NC(=O)Cc1c(F)cc(Cl)cc1Br)OCO2 26873,c1(CN(C(CC2CCOC2)CO)C=O)cccc(COc2ccccc2)c1 26874,Cc1cc(F)ccc1CNC(=O)NC1(CF)CCCC1 26875,CC1CCN(C(=O)CC2(C)CN(C(=O)CS(=O)(=O)NCc3ccccc3)C2)CC1 26876,N1(C(CCC(C)C)=O)CCCCC2C1CCCN2C(C1CCNC(=O)C1)=O 26877,C1(NC(CC2C(C)=NN(C)C2=O)=O)CN(C(=O)CCC2CC2)CC1C1CC1 26878,Cc1cc(C(=O)N(CCCNC(c2cnn(C3CC3)c2)=O)C)cn1C(C)C 26879,C(CCC(C(=O)NCCC(O)C1CCC1)NC(c1cc(C)c(C)cn1)=O)OC 26880,CCCC(C(=O)NCC(CNC(c1ccc(OCC(=O)NC)cc1)=O)CO)OC 26881,N1(S(Cc2c(C)nns2)(=O)=O)CC(=O)NC(C)C1 26882,c1(C(=O)NC2C(C(=O)NCc3ncc(C)s3)C2)c(Cl)ccc(Br)c1F 26883,c1(C(N2CC(CC)C(NC(c3cc(COC)no3)=O)C2)=O)ccc(N)c(Cl)n1 26884,C(=O)(C1=Cc2ccccc2C1C)NC(CCOC)CNC(c1nc(Cl)cs1)=O 26885,Cc1ccc(C=CC(N2CCCC(C(C)NC(=O)CC(F)(F)F)C2)=O)cc1Cl 26886,Cc1c(C(N2CC=CCC2C(=O)NOCC(C)O)=O)nnn1C 26887,c1(C(=O)OC)nccnc1N1CCCC(C(C)NC(=O)CSCC(N)=O)C1 26888,C1(CC)CN(C(c2ccnn2C2CCC2)=O)CCC1NC(=O)CC(C)(F)F 26889,N1(C(C2N(C(c3ncc(C)cc3F)=O)CC(O)CC2)=O)CC2(C)COCC2(C)C1 26890,c1(C(=O)NCC(CNC(Cc2c(C)ccs2)=O)F)ccc2c(c1)NC(=O)C2(C)C 26891,C#Cc1cc(F)c(C(=O)N(C2CCC(NC(c3csc(C#N)c3)=O)C2)C)cc1F 26892,CCC(CC)(CC)C(=O)N1CCC(OCCCNC(=O)CC2CCC2(C)C)CC1 26893,c1(CNC(C2ON=C(CC)C2)=O)nn(C)c2c1CN(C(=O)C=C(C)C(F)F)CC2 26894,C1(NC(c2nc(SC)nc(O)c2)=O)CCC2(CC1)CC(O)C2 26895,Cn1cc2cc(C(=O)NC3C=CC(CNC(=O)Cn4nccn4)C3)ccc2n1 26896,C(CCC(C(=O)N(C)Cc1nncn1C)NC(c1csnc1Cl)=O)OC 26897,c1(NC(C(=O)OC2CCCC2O)=O)ccccc1C(=O)OC(=O)C1CCC1 26898,Cc1ccc(C(=O)NCCC(O)CNC(C2CC(O)C2)=O)c(N)n1 26899,c1(C(=O)NC(C)(C)CC2C(CNC(c3nc(COC)sc3)=O)C2)nc(O)sc1C 26900,N1(C(c2ccc(C)nc2)=O)CC2CCN(C(=O)COCP(C)(C)=O)C2C1C 26901,C(CCCC(=O)NC1CC1)N(C)CCNC(CCF)C(=O)N(C)C.C(=O)O 26902,N1(c2ccnc(C(=O)OCC)n2)CCC(C)C(NC(=O)C(F)C(C)C)C1C 26903,C1(CC(N2CCC(NC(C)=O)C2)=O)CCN(C(=O)Cc2cnnn2C)CC1 26904,c1(COC2CCCN(C(CNC=O)=O)C2)cccc2cncn12 26905,N1(C(C2C(=C)C2)=O)CC=C(C(=O)NCC2Cc3nccn3C2)CC1 26906,c1(C(=O)NC(C(=O)NC(C2CCOCC2)C)Cn2cccn2)cccc(CO)n1 26907,c1(CCC)cc(C(=O)NCC(O)C(=O)NCCCC(C)O)n[nH]1 26908,Cc1nc(C=CC(=O)NC2(CCCNC(C3(C(C)(F)F)CCC3)=O)CC2)cs1 26909,C1(C)(C(=O)NCC(CN(C)C(c2csc(-c3ccco3)n2)=O)O)C(C)(C)C1(C)C 26910,C1(C(=O)NCCC2N(C(c3cn(CC)nc3)=O)CCCC2)CC2CCCCCC12 26911,C1(C)(CC(=O)N(CCOC(C)=O)C)CCN1C(=O)CC(=O)N(C)C 26912,C1(C(=O)Nc2cccc(Cl)c2C)(CC)CCN(C(=O)CC2CCC(=O)NC2)CC1 26913,N1(C(c2cnc(SC)s2)=O)CC2CN(C(c3ccc(C)nc3)=O)C2C1 26914,C1(NC(C(C)(C)OC(C)=O)=O)CCCC1(C)NC(=O)C=C(C)Cl 26915,C1(c2nnnn2CC)(CC(c2ccc(NC(CC)=O)cc2)=O)CCCC2(CC2)C1 26916,C1(C(N2C3CC(NC(C4(C#C)CCC4)=O)CC2CC3)=O)CCc2c(n[nH]c2C)C1 26917,N1(C(=O)OC(C)(C)C)CCC(NCCC2CCN(Cc3ccccc3)C2)C(O)C1 26918,CCCCCCCC(=O)NC(CC)CCC(=O)N(C)CC1CCOCC1 26919,C1(C(N2CCC(CCC(=O)NC(c3nccs3)CC)C2)=O)CCCC1C1CC1 26920,CC(C)S(=O)c1ccc(C(=O)NCC2(O)CN(C(C3C(C)C3C)=O)C2)cc1 26921,N1(C(C(C)NC(CC)=O)=O)CCC12CN(C(=O)C(C)(C)c1cc[nH]n1)C2 26922,O=C1Cc2c(C(N3CC(NC(C45CC(O)C4C5)=O)C3)=O)cccc2N1 26923,C1(NC(CCCC)=O)CCN(C(c2ccc(C#N)s2)=O)CC1C 26924,C1(NC(c2ccc(C(F)F)o2)=O)(CNC(C2(Cl)CC23CCC3)=O)CCCCC1 26925,C1(NC(C(CSC)C)=O)CCN(C(c2cc[nH]c(=N)n2)=O)C1C 26926,c1(C(=O)NC2CC(C)(C)CN(C(C3CC3(C)C)=O)C2)cccc2nc(CO)[nH]c12 26927,N1(C(CC2C(C)CCC2)=O)CCCC(C)(CNC(c2scnc2C(C)(C)C)=O)C1 26928,N1(C(c2cscn2)=O)CC2(C(N3CC4(CC(CO)CO4)C3)=O)CC1CCO2 26929,N1(C(c2c(C)n(C)nn2)=O)CC(F)(F)CC1CCNC(=O)C1=C(Cl)CC1 26930,c1(C2(C)CC2)cc(C(N2CCC(CCNC(=O)C(CO)N(C)C)C2)=O)[nH]n1 26931,N1(C(CC(C)(C)C#N)=O)CC2CCC1CN2C(c1cccc2nccn12)=O 26932,C1(NC(=O)CCN2CCC2)CN(C(c2cnc(O)o2)=O)C2(CCOC2)C1 26933,N1(C(C2C(C)(C)OC2(C)C)=O)CC2(C1)CN(C(C1CC3(CC3)CO1)=O)CC2CO 26934,C1(NC(c2cc(CC)nn2C)=O)CC2CCC1(CNC(c1cnc(CC)s1)=O)C2 26935,n1(CCc2onc(-c3ccc4ccn(C)c4c3)n2)cnc2ccccc2c1=O 26936,c1(NC2CCCC(NC(=O)CCCc3cccs3)C2)ncnc2c1CCO2 26937,C1(C(=O)OC)(C(=O)NCC(O)CN(C)C(c2cc(O)ncn2)=O)CCCCO1 26938,C(=O)(C(C)(C)CS(C)(=O)=O)NC1CC(C)CN(C(=O)Cn2nc(O)ccc2=O)C1 26939,C(N(C)N1CCC(C)(CC(=O)OC)CC1)c1cccc(OCC)c1 26940,N1(C(CCC2CCC(=O)N2)=O)CCCC(F)(C(=O)NC2CN(CC(F)F)C2)C1 26941,N(C1CCOc2ccc(F)cc21)C(c1ccc(SC(F)(F)F)cc1)C(=O)NC 26942,NS(=O)(=O)c1ccc(C(N2CCC(CCNC(C3CC3c3ccsc3)=O)C2)=O)o1 26943,c1(C(=O)NCC(CCNC(CCCC(C)=O)=O)(C)C)cc2c([nH]1)CCCC2 26944,c1(C(C(=O)NC2CC(F)(F)C2)N(CC(=O)NCC)C)nc(Cl)cc(Cl)c1C 26945,c1(OCCOC)ncccc1C(=O)NC1CCC(NC(=O)C(F)(F)CO)CC1 26946,N1(C(c2cnc(N3CCCC3)s2)=O)CCC2(C(N3CC4CCC3C4)=O)CC2C1 26947,N1(C(COC(CC)C)=O)CCC(CNC(=O)Cc2cnsc2)C(CC)C1 26948,c1(OC)cc(Br)c2c(c1)CCN(C(=O)C(=O)NCC1(OC(C)C)CCOCC1)C2 26949,N1(C(C2N(C(C3C(OC)(OC)CC3)=O)CC(F)(F)C2)=O)CC2CC(C)(C)C2C1 26950,N1(C(c2c(CC)occ2)=O)CC(NC(C23CC(CC)(CO2)C3)=O)C(C(F)(F)F)C1 26951,CCCC(C)(CC)C(=O)NC1CN(C(c2cccc(C3CC3)n2)=O)CC1N=[N+]=[N-] 26952,Cc1cc(N)c(C(=O)NCC#CCNC(=O)C(C)(O)c2ccccc2)cc1C 26953,C(CN(C(=O)Cn1cnnn1)C)(CO)(CO)NC(C(N1C(=O)CCC1=O)CC)=O 26954,N1(C(c2[nH]cc(C#N)c2)=O)CCC(CCNC(=O)CC2OCCCO2)C(F)(F)C1 26955,S(=O)(=O)(c1ccc(Br)cc1NC(CO)CC#CC)NCCC=C=C 26956,C1(CC(C)NC(C2C(OCC)C2C)=O)CCN(C(=O)C(C)OCC)CC1 26957,CC1(C(=O)N2CC(NC(c3sccc3Cl)=O)C3(CCC3)C2)COc2ccccc21 26958,c1(OCCOC)ccccc1NC(N1CCCC1C(=O)NC1CCCCO1)=O 26959,CCCCCCC(CC)NC(C1CCCCCN1C(=O)C=Cc1ccncn1)=O 26960,N1(C(C2N(C)CC(C)(C)C2)=O)CC=C(CC(=O)NCC23CCCC2C3)CC1 26961,N1(C(CC(CC)C2CC2)=O)CCC2C(C1)CN2C(c1csc(Br)n1)=O 26962,C1(CN(C(=O)CSCc2ncc[nH]2)C)CN(C(=O)C=Cc2ccc[nH]2)CCO1 26963,CC1CCC(=CC(=O)N(C(C)(C(=O)NCc2cscn2)C2CC2)C)CC1 26964,CCC(CC(=O)NC(C)CN(C)C(C1CCN(C)C(=O)C1)=O)C(C)C 26965,C1(NC(C2C(C)CCC2)=O)C2CCCN(CCN3CCCC3=O)C2C1(C)C 26966,c1(C2CN2)ccc(N2CCCCC2)cc1.CC1CC(CS(=O)(=O)N(C)C)CN1 26967,N1(C(c2cnsc2)=O)CCCC2CN(C(c3cccn(C4CC4)c3=O)=O)CCC12 26968,N1(C(C(N2CCN(CC(=O)OC)C(=O)C2)CCC=C)=O)CCn2c(C)nnc2C1 26969,C1(C)(NC(C2(C)N(C(CCSCCCC)=O)CC=C2)=O)CCC(C)=C(C)C1 26970,C1(C(=O)NC(C(=O)NC2CC(C(=O)OC)C2)C)CCC2(CCC2)C1 26971,C(=O)(C1CSc2ccccc21)N1C(C)CN(CCC2CCCC2)CC1 26972,C(=O)(C(Cc1cn[nH]c1)NC(c1cc[nH]n1)=O)NCCC(C)SC 26973,C(C)(C(N)CC(=O)N1CCCC1C(=O)Nc1cccs1)SC 26974,N1(C(CCN(CCC)C)=O)CC2(CCC(NC(c3ccnn3CC)=O)CC2)C1 26975,N1(C(C(=O)N(CC(C)NC(CSCC)=O)C)CC)C(=O)c2ccccc2C1=O 26976,c1(NCC(=O)NC(C2N(C(CCCOCC)=O)CCC2)(C)C)ccc(CC)cn1 26977,C(=O)(C1=NOC2COCC12)N(CC(CC)NC(c1cc(C#N)no1)=O)C 26978,CC(C)(O)CC(=O)N1CCC(N(C)C(=O)OC2C(c3ccccc3)C2(F)F)CC1 26979,CC1(C)CC(C#N)(NC(=O)Cc2ccc(NC(=O)OC(C)(C)C)cn2)C1 26980,CS(=O)(=O)c1ccc(C(=O)NC2CCN(C(=O)C(F)C3CNC3)CC2)cc1 26981,C1(CNC(c2scc(C)c2)=O)CN(C(=O)CC2CCCC23CC3)CCO1 26982,c1(CC(N2CCN(C(c3ccnc(C)n3)=O)C(CO)C2)=O)coc2ccccc12 26983,c1(C(=O)NCC(C)(CC)NC(CC=CC=C)=O)cc(OC)cc(OC)c1 26984,CC1(C)CC(CO)(Nc2ccc(Br)c(F)c2)CO1 26985,C(=O)(C1=C(Cl)CCOC1)NC(COCC)C(=O)NC1CC1(C)C(F)F 26986,c1(OCC)ncc(C(=O)NC(C)(C)CCCNC(=O)Cc2ccno2)cc1Cl 26987,N1(C(C2(C(=O)OC)CC2C)=O)CCc2cc(NC(C3CC(OC)C3)=O)ccc2C1 26988,c1(C(N2CC(N(C(CC(C=C)(C)C)=O)C)C(O)C2)=O)ccc(C)c(Br)c1N 26989,c1(C(=O)NCCOC(CNC(C(C(C)O)C)=O)(C)C)cc2n(c1)CCCC2 26990,c1(C(=O)NC(C)CCc2cccn2C)cc2c(cnn2C)nc1C(F)F 26991,c1(NC(C2CCCO2)=O)cccc(OC(F)F)c1.C1(NC(=O)CSC)CCC1 26992,N1(C(CCC(=O)OCC)=O)CCCC(C)(NC(C2CCCC(C)(C)C2)=O)C1 26993,N1(C(CCN(C(CCC(C)OCC)=O)C2CC2)=O)CC2CCC2(OC)C1 26994,n1(CC(=O)NCC(C)CNC(=O)Nc2cc(C3CC3)on2)cc(Br)cn1 26995,c1(CC(=O)NC2CCCC(NC(C(C=C)O)=O)C2)cc(F)ccc1Cl 26996,N1(C(CN(C(C)C)C)=O)CC2CCC1C1CN(C(=O)C(c3cccnc3)C)CC21 26997,c1(CC(=O)NCC(O)CNC(C23CCC(C2)C3)=O)cccc(Cl)c1 26998,C1(C(=O)NC(C#C)CC2CCCC2)C(CC)CCN1C(c1csc(CC)n1)=O 26999,N1(C(c2cnoc2)=O)CCCC(C2CCN(c3cccc(F)c3[N+](=O)[O-])C2)C1 27000,N1(C(CCCOc2ccc(C(C)=O)cc2)=O)CCC(C2(C(=O)O)CC2)CC1 27001,C1(SC)CCC(C(=O)NCCC2(NC(c3ccsn3)=O)CC2)C1 27002,Cn1ccc(=O)cc1C(N1CCOC(C(=O)Nc2nccc(Cl)c2Cl)C1)=O 27003,C1(N(C(C23CC(C)(C2)C3)=O)CC)CCCN(C(c2occc2COC)=O)C1 27004,N1(C(c2nc(C(C)OC)sc2)=O)CCCC(NC(=O)CC2CCC(=O)N2)C1 27005,C1(C(N2C(CNC(=O)C=Cc3ccsc3)CC(O)C2)=O)CC12CCC1(CC1)CC2 27006,c1(C(=O)OCC2CC(C)N2C(=O)OC(C)(C)C)ccnc2c(I)cccc12 27007,C1(C(=O)NCc2cncc(C)n2)COC2(CCN(Cc3cscn3)CC2)C1 27008,C1(C2CC2)(C(=O)NC2CCC(NC(CCC(=O)OC)=O)C2)CCOCC1 27009,C(=O)(C1CCc2nccn21)N1C2(C(N3CC(C(=O)OC)(CC)C3)=O)CC2CC1 27010,c1(OCC)cncc(N2CCCC2Cc2ccc(C)cc2)n1 27011,c1(C(N2CC(CC(=O)Nc3ncncc3Cl)C2)=O)ccc2scnc2c1 27012,c1(C(=O)NCC(c2cccc(C)c2)NC(C2ON=C(C)C2)=O)cc(C)nc(C)c1 27013,C(=O)(C(C)C(=O)OCCC(C)C)NC(CN(C(COC)=O)C)C 27014,c1(CNC2CN(C(=O)OC(C)(C)C)C2(C)C)c(F)cc(Cl)cc1Cl 27015,c1(C(=O)NCCC2CCN(C(c3cnc(C(=O)OC)s3)=O)C2)nnn(C)c1C 27016,N(C(=NCC1(O)CCSC1)NC1CCCCC1)CCN(C(CC)C)C(C)C 27017,N1(C(Cn2ncc(C)c2)=O)CC(C)(CNC(C2(F)CC=CC2)=O)CC1(C)C 27018,C1(C(=O)NCC2(CNC(CN(S(CC)(=O)=O)C)=O)CCC2)OC(C)(C)OC1(C)C 27019,c1(C(=O)NCCCCC(C)NC(CSCC=C)=O)ccc2n[nH]cc2n1 27020,C(=O)(C1=CSCCO1)NC1C(CNC(CC2C(C)=NNC2=O)=O)CCC1 27021,C(=O)C(=O)CC(C)CC.c1(C(=O)NCCC=CCCC)ncoc1C 27022,Cc1c(C(N2CC3C(CN(C(=O)CCCC4CCC4)C)C3C2)=O)cnn1C(C)C 27023,N1(S(CC)(=O)=O)CCCC1C(=O)NCC(c1ccccc1)NC(=O)C1=CCC1 27024,N1(C(CCP(C)(C)=O)=O)C2CCC1CC(NC(C1CCOC3(CCC3)C1)=O)C2 27025,CC1CCC(CO)N(C(C2C3CC4C(C3NC(c3cc(O)nn3C)=O)C24)=O)C1 27026,N(C(=NCCc1ccc(Br)o1)NC1CN(C2CC2)CC1C)CC(=C)C 27027,CC1C2CCC(C2)C1C(=O)N(C)CC1CCC(CNC(=O)Cc2nc[nH]n2)CC1 27028,N=c1nc(O)c(CC(=O)NCCCOCCNC(=O)C(F)=C2CCC2)c[nH]1 27029,CCCS(=O)(=O)C(C)C(=O)NCCCOCCNC(=O)CSc1nccn1C 27030,C1(NC(c2c(C)cns2)=O)CC2CC1CN(C(=O)C(C1CCCCCC1)O)C2 27031,CCC(C)CCC(=O)NCCNC(=O)CC1CC=CCN1C 27032,c1(SCC(=O)NCCC(C)NC(C2C=CC=CC=C2)=O)cccc(F)c1 27033,N1(C(C(c2cccc(F)c2)C)=O)CC(CNC(c2cc(Cl)on2)=O)C(C)C1 27034,N1(C(c2c(OCC)nccc2)=O)CCCN(C(c2ccc(=N)[nH]n2)=O)CC1CO 27035,C(=O)(C1=CC2(CCN(C(C34C=CC(CC3)C4)=O)C2)C1)N(CC(F)Cl)C 27036,C#CC1(C(=O)Nc2cccc(CCO)c2)CCN(C(c2cscc2OC)=O)C1 27037,N1(CC(N2CC(C)(NC(=O)Cc3ccc(C#N)cc3)C2)=O)CCn2ccnc2C1 27038,C=CCCC(C(=O)NCC(CC)C(C)(F)F)NC(C1CCC1COC)=O 27039,c1(C(N2CC(NC(C3(Cl)CC3(C)C)=O)CC(OC)C2)=O)cc(Cl)c2n[nH]cc2c1 27040,Cc1cc(C(=O)NCCC2CC3CCC(C2)N3C(=O)C(C)C2CC2)c(N)c(Cl)n1 27041,c1(NC(=O)C=CC2CC2)cccc(CNC(c2nc(C(F)(F)F)cs2)=O)c1 27042,C1(CN(C)C(c2cn(C)nn2)=O)CCC(NC(=O)CC2CCCC(=O)N2)CC1 27043,c1(C(=O)NCCC(C)NC(C2(CC)CCCO2)=O)ccc(CN2CCCC2)cc1 27044,C1(CCOC)CN(C(c2ccc(C(O)CF)cc2)=O)CCN1C(C1CC1F)=O 27045,c1(C(=O)NC(CC)CN(C(=O)CC2CCOC2)C)ccnn1C(F)F 27046,C(C)(CCCC(=O)N1CCC(CCO)CC1)NC(C(C)OCCCC)=O 27047,C1(C(=O)NC2CON(CC)C2=O)CN(C(c2ccc(C)nc2O)=O)CC1(F)F 27048,N1(C(c2cccc(COC)n2)=O)CC2CCC2(CCNC(C2(C)CCC2)=O)C1 27049,c1(CC)onc(C)c1C(=O)NCCC1(C)CCN(C(C2CCCC2)=O)C1 27050,C=CC1CN(C(=O)C2=CCN(C)C2)CC1NC(c1c[nH]nc1-c1ccoc1)=O 27051,C1(NC(c2n(CC=C)ccc2)=O)CN(C(c2cccc(C)c2)=O)CC(C)(C)C1 27052,CC1CC(C)CC2(C1)NC(=O)N(CC(=O)N(C1CC3(C1)CC(N)C3)C)C2=O 27053,Cn1cc(C(=O)NCC2CCCC(NC(=O)CC3(C4CC4)CC3)C2)ccc1=O 27054,c1(C(=O)NC2C3CCN(C(Cc4nc(=N)[nH][nH]4)=O)CC32)cccc2c[nH]nc12 27055,CN=c1[nH]c(=NCCOCC2CC2)[nH]c(=NCCc2cn(C)c3ccccc23)[nH]1 27056,c1(C(=O)NCC2C(NC(c3cc(CC)oc3C)=O)CCC2)ccc(C)cc1OC 27057,N1(Cc2c(=N)cc[nH]c2)CCCC(C(N2CC3CCCC23)=O)CC1 27058,Cc1cccn2ncc(C(N3CC(O)(CN(C)C(C4CNC(=O)N4C)=O)C3)=O)c12 27059,C1(C(=O)NCC2CC(NC(C(C)OC)=O)C2)CC2CCC1O2 27060,N1(C(CCC#CC)=O)CC(NC(c2ncccc2C)=O)CC2(CC2)C1 27061,C1(CC(=O)NC(CCCNC(CSCC)=O)C)CCC2CC2C1 27062,CN1CC(F)CC1C(=O)NCC1CCC(NC(C2CC2CC(C)(C)C)=O)C1 27063,C1(CNC(CC(C)C#N)=O)CC2(C1)CN(C(=O)Cc1ccoc1)C2 27064,C1(CCNC(C2C(OCC)C2)=O)CCCN1C(=O)CSC(F)F 27065,c1(C(=O)NCC2CC(NC(c3c(C(C)C)ocn3)=O)C2)ccc2c(c1)CCC=C2 27066,C1(CNC(C2CCC(C)(C)CC2)=O)CCC(C)(C)CN1C(C1CC1(C)C)=O 27067,C1(NC(=O)CC2(C(F)(F)F)CC2)COC2(CCN(C(c3ncncc3Cl)=O)C2)C1 27068,c1(C(=O)NC2CC3C2CCN3C(C2(F)CCOCC2)=O)nnn2c1C(=O)NCC2 27069,C(=O)(C1=NOCC1)N1CCC(N(C(CC)C(=O)NCc2ccccc2C)CC)C1 27070,C(C(CC(C)C)C(=O)NCCNC(N)=O)NC(CC(C=C)(C)O)=O 27071,c1(NC)ccc(C(=O)NCc2c[nH]nc2C(=O)N(C)CC2CCOC2C)cc1 27072,C1(C(=O)NC(C)CC2CN(C(=O)CCc3cnoc3)C2)CCc2nncn2C1 27073,C1(C=O)(NC(c2cccnc2C2CC2)=O)CCOCC1.N12CCCC(C1)C2.ClCl 27074,c1(OC)cc(C(N2CCC2(C)C(=O)Nc2cccc(F)n2)=O)cc(O)c1O 27075,C(=O)(C(F)CC(C)(C)C)NCCN(CCC)C(c1ncccc1N)=O 27076,Cn1nc(Br)cc1C(N1CCC(C(C)(C)C)CC1)C(=O)NCC(F)F 27077,N1(C(C(CC)(C)C)=O)CC(C)CN(C(c2ccc(C(F)F)o2)=O)C(C)C1 27078,C12(CNC(C(CC3CC3)NC(=O)CC34CCCC3C4)=O)CCC(CC1)O2 27079,Cc1ccc(C(=O)NC2CC(CC(N3CCOC(C4CC4)C3)=O)C2)c(F)c1 27080,N1(C(C(C=C)CC)=O)CC2(C=C(C(=O)NCC3CC(OC)C3)CO2)C1 27081,N1(C(C(C(=O)NC)(C)C)=O)CC(C(=O)N(C)CCc2nccs2)CCC1(C)C 27082,C(=O)(CC(CC)C(C)(C)C)N(C1CCN(C(=O)COCC)CC1)CCC 27083,C(CC(C)(C)C(=O)NC(C(C)C)C1(NC(=O)C(c2cnns2)OC)CCC1)OC 27084,S(=O)(=O)(c1cc(F)cc(F)c1)N1C2CC(N(CCC#N)C)C(C2)C1 27085,C(=O)(CC1OCCc2ccsc21)N1CC(NC(C(CC#C)CC#C)=O)C(C)(C)C1 27086,C(C1=CCN(C(C2CCC3(CC2)CC3)=O)CC1)NC(C(CC=C)OC)=O 27087,c1(OC)cc(C(=O)N=c2ccn(C3CN(Cc4n[nH]c(C)n4)C3)[nH]2)c(F)c(F)c1F 27088,C12CC(O)CN1OC2=O.C1(CC)CCCN1C(C1CC1C(=O)C1CC1)=O 27089,n1(CC(=O)NCC2COCCN(C(c3csnn3)=O)C2)nc2c(n1)CCCC2 27090,C1(NC(COC)=O)CCCCC1NC(=O)CC1CCC(C)(C)C1 27091,c1(OC)nc(Cl)ncc1Nc1ccnc(OC2CCCC(C)C2)c1 27092,c1(C(N2CC(N(C(=O)CCCn3c(O)nnc3O)C)C(O)C2)=O)n[nH]cc1[N+](=O)[O-] 27093,CN1CC2CCC(C1)N2C(C1CC12CN(C(=O)CC1(O)CCC1)C2)=O 27094,CC1(NC(=O)CNc2ncccn2)CC(NS(C)(=O)=O)C1 27095,N1(C(C(C)O)=O)CCN(C(c2sc(Br)nc2Br)=O)CC1CO 27096,C12CC(F)(F)CN1C(=O)OC2.C(c1ccccc1)=C(CC)C(=O)OC(C)(C)C 27097,N1(C(c2n[nH]c(C)c2O)=O)CCC2CN(C(=O)CCc3nc(C(C)C)no3)C2C1 27098,Cn1c(=O)n(C)c2cc(CS(=O)CC3CC4(CCC(C(=O)O)CC4)C3)ccc12 27099,C(CN=c1cc[nH]cc1S(=O)(=O)NC1CCCSCC1)c1c(C)c(Cl)c(Cl)cc1 27100,c1(CC(N2CC(N(C(=O)CC3=CCCC3)C)C(O)C2)=O)ccc([N+](=O)[O-])cc1 27101,c1(C(c2n(CC)nnn2)NC2CCN(CCF)C2=O)cc(Br)cnc1N(C)CC 27102,N1(C(C2C(C)=CCS2)=O)CCOCCC1C(=O)Nc1cnc(C(C)C)nc1 27103,CCC(F)(F)CC(=O)N1CCC(C)C(NC(c2ccoc2Cl)=O)C1 27104,C(CNC(=O)Cn1cc(N)cn1)(C(C)(C)C)NC(C1(CC=C)CCC1)=O 27105,c1(C(N(C2CCCCN(C(C3CC3C(N)=O)=O)C2)C)=O)cc2cn[nH]c2cn1 27106,C1(NC(C2CCC(CC)O2)=O)CCN(C(c2cc(C)cc(Cl)n2)=O)CCC1CO 27107,C1(CNC(C2(CCCC)CCCC2)=O)CCN(C(=O)CCc2nc[nH]n2)CC1O 27108,N1(C(Cn2cc(C(=O)OCC)nn2)=O)CCN(C(=O)CSCC)C(C(C)(C)C)C1 27109,C(CNC(C1CC1c1cccc(Cl)c1)=O)(C(C)(C)C)NC(C12CC(C)C1C2)=O 27110,C1(CC(C)NC(C2CC2)=O)CN(C(=O)C=CC(=O)NC2CCC2)C1 27111,N1(C(CCn2cc(CNS(CC)(=O)=O)nn2)=O)CCCC(CC(=O)OC)(OC)C1 27112,C1(N(C)C)CCN(C(=O)CCNOCc2ccccc2)C(C)(C)C1 27113,N1(CC#N)CCCC(C2CCN(C(C3CC34CCOCC4)=O)CC2)C1 27114,C1(CC=C)(NC(=O)CC2C(=O)ON=C2C)CCCN(C(C2CCCC23CC3)=O)C1 27115,N1(C(c2c(CN(C)C)cco2)=O)CCOC(CNC(c2cccc(=O)o2)=O)C1 27116,Cc1ccc(C(C)C(=O)N(CC(O)CNC(c2ccc(Cl)cn2)=O)C)cc1 27117,N1(C(CSCCC#N)=O)CC2CC(NC(=O)Cc3csnn3)CC2C1 27118,C(CC(C)(C)C)(C(=O)NCC=CCNC(c1ccc(F)c(CO)c1)=O)OC 27119,O=C1CCN(CC(=O)NCCNC(=O)CC2CC=CCC2)CC1 27120,C(=O)(C(C)C(O)CC)NC(CC=C)C(=O)Nc1ccc(CO)cc1O 27121,C(C(C)C(=O)NOCC1CCOC1)N(C(C(COC)(C)OC)=O)C 27122,CC(=O)CCCC(=O)NCCCN(C(C1CC(C)(C)CCO1)=O)C1CC1 27123,N1(C(c2ccn3c2CCCC3)=O)CC2CCCC(O)C2C1 27124,N1(C(C=CC)=O)CCC(O)(CCNC(C2CCCN2C(N)=O)=O)C1.C(C)(C)(C1CC1)N 27125,c1(C(=O)NC2C3(CC(NC(C4=NOC(C)C4)=O)C3)C2)cc2cc(Cl)ccc2o1 27126,c1(C(=O)NCCCCC2CN(C(C(C)O)=O)C2)c(F)cc(F)c(F)c1F 27127,c1(C(N2CC(F)(CNC(C3OCC(C)(C)C3)=O)C2)=O)cc(N)ccc1[N+](=O)[O-] 27128,C(=O)(C1CCOc2c(F)cccc21)OCCN(CC(C)O)CC1CC(OCC)C1 27129,c1(NC)cnc(C(=O)NC(C)C=CC(=O)NC2CC2(C)C(F)F)cn1 27130,Cc1c(C(=O)NCC2CCCCN2C(C2CCCS2(=O)=O)=O)nn2c1CCCC2 27131,N1(C(C2C(C)C2)=O)CC(NC(=O)C2=CCOC2)CC12CCC2 27132,n1(CC(=O)NCC2CC2CNC(C2CCC(CCO)CC2)=O)ccc(O)nc1=O 27133,N1(C(c2c(C)cc(C)s2)=O)CCC(CO)C(NC(=O)Cc2cccnc2C)C1 27134,C1(C(=O)NC2CC(CNC(C3(C)COC3)=O)OCC2)CCCCN1N=O 27135,c1(C(N(C2CCCN(Cc3ccccc3CO)CC2)C)=O)cccn(C)c1=O 27136,c1(OC)cccc(C(=O)NCC2CC(NC(=O)CCCC(N)=O)C2)c1O 27137,N1(C(CC(CC)C)=O)CCC(CNC(=O)C#CC2(CC)CC2)C12CC2 27138,C1(NC(c2c(F)cccc2F)=O)CC1C1CCCN(C(C2OCCO2)=O)C1 27139,CCC(C(=O)NCC12CC(NC(=O)C(F)OC(F)(F)F)(C1)C2)n1ccnc1 27140,c1(C(=O)NCC2N(C(C(C)(C)c3cnsc3)=O)CC2)cc(OC(F)F)nc(Cl)c1 27141,Cc1cc(C)c(CNCC2COCCN2c2ncc3ccsc3n2)c(C)c1 27142,Cc1ccc(C(=O)NCCC(O)CNC(C2C3CCCCCC23)=O)c(O)c1C 27143,c1(N2CCC(NC(c3scc(OC)c3)=O)C2)nccc(COC)n1 27144,C1(C(N2CC(NC(=O)CCOc3cccc(Cl)c3)(CO)C2)=O)CCCC2(CC2)C1 27145,N1(C(C2C3CN(C(C(CCSC)NC(C)=O)=O)C2C3)=O)CC2CCCCC2C1 27146,c1(C(=O)NCC(CC(C)C)NC(C(c2cccs2)SC)=O)occ2c1CCOC2 27147,N1(CC)CC2(CCCN2C(C23CC2CN(C(c2cc(C(F)(F)F)c[nH]2)=O)C3)=O)C1 27148,C1(CNC(C2CCCC2)=O)CCCN1Cc1ccc(Cl)o1 27149,c1(C(N2CC(NC(C3CCOC3)=O)CC(C)C2)=O)ccc2ccn(C)c2c1 27150,C1(F)(C(N(C(c2onc(C)n2)C)C)=O)CCCN(C(=O)C=C2CCC2)C1 27151,Cc1c(O)ccc(C(N2CCCC(C(C)NC(C3(CF)CCC3)=O)C2)=O)c1C 27152,C1(NC(CCc2cc(C)on2)=O)CC2CCC(C1)N2C(C1COC(=O)O1)=O 27153,C(=O)(C1=CCCCO1)N1CC(n2cc(CNC(C3(COC)CCCO3)=O)nn2)C1 27154,C(=O)(CC1OCc2ccccc21)NCC1C2CN(C(=O)CC(F)(F)Cl)C1C2 27155,C1(C(N2CC3=C(CN(C(CC(=O)OC)=O)C3)C2)=O)C2Cc3c(Cl)cccc3C12 27156,C1(C)(COC)CN(C(=O)Cc2ccc(F)c(Cl)c2F)Cc2ccccc2O1 27157,CC1CN(C(=O)Cc2cccc(F)c2)CCC1C(=O)NC1CC(=O)N(O)C1 27158,CC1CC(NC(C2(C)CSC2)=O)CCN1C(C1CN(C(N)=O)C1)=O 27159,N1(C(C(COC)NC(c2[nH]nnc2C)=O)=O)CCN2CC(F)CC2C1 27160,c1(C(N(C2CN(C(C3CC(CF)C3)=O)CC2F)C)=O)cnc2c(C#N)cnn2c1 27161,CC1(C)CC(C(=O)NC2(C)CCCC2(F)F)CN(C(=O)C(C)(C)C(F)F)C1 27162,Cc1cccc(OC2CN(C(c3ccccc3-c3cncn3C)=O)C2)n1 27163,c1(CN2CC3(C(C(N(CC(O)CO)C(C)C)=O)C3)C2)cc(Br)c(F)cc1Cl 27164,C(=O)(CCS(C)(=O)=O)NC(C=CC(=O)N(CCO)CC)C 27165,c1(C(=O)NCCCCCNC(CC(CC)C2CC2)=O)cc2ccccc2n1CC 27166,C(C(O)C(=O)NCCC1(CN(C(=O)CC(C)N(C)C2CC2)CCO)CC1)OC 27167,c12nnc(n1CC1CCCO1)N(C(C)C)C2.C1(CC(=O)OC)CCC1C(F)(F)F 27168,C1(NC(CCC(=C)Cl)=O)CCCC12CN(C(C1C3CC4C(C3=O)C14)=O)C2 27169,C=CC1CCN(c2nnc(-c3[nH]c(=N)[nH]c3Br)n2C)CC1 27170,N1(C(c2cc(SC)c(C)o2)=O)CCC2CN(C(C3CC(N(C)C)C3)=O)CCC2C1 27171,N1(C(C(CCOC)(C)C)=O)CCCC(C2CN(C(C3(S(C)(=O)=O)CCC3)=O)C2)C1 27172,c1(C(=O)NCC(C(=O)N(C(C=C)C)C)(C)CC)cn2ccccc2n1 27173,C12(CC(=O)NC(COC)CO)CCC1CN(C(c1csc(C)c1)=O)C2 27174,c1(C(=O)NCC(C)N(C(CNS(CCC)(=O)=O)=O)C)cccc2c1OCC2C 27175,C1(C(=O)NCCC(C)(C)NC(c2c(C(C)(C)C)noc2)=O)C2CCCC(F)(F)C12 27176,CCCCCC(O)C(=O)NCC1CN(C(C2COCCN2C)=O)C1 27177,N1(C(C(CCNC(CCN(CCC)C)=O)O)=O)CCCCC(C)(F)C1 27178,c1(C(=O)NCCCN2CCC(NC(c3cc[nH]n3)=O)C2)cc(F)cc([N+](=O)[O-])c1 27179,C12(CNC(c3c(OC)c[nH]n3)=O)CCC1CCN2C(c1cnco1)=O 27180,C1(N(C(CCCN(C(C)C)C)=O)C)CN(CCN2CCN(C)C(=O)C2)CCC1C 27181,CC1COc2c(C(=O)NC3CN(C(=O)CC4CC5(CCC5)C4)CCC3F)cnn2C1 27182,CCC(CNC(C1CC(OC)CN1C(c1ccncc1NC)=O)=O)CC(C)C 27183,N1(C(C2N(C(CC3CC(=C)C3)=O)CCC2CC)=O)CC(C2CCCC2)C1 27184,C(C)(C)(CC(C)NC(=O)C(F)C1CC(NC(=O)CCN2CCCC2=O)C1)OC 27185,c1(C(=O)NCCN(C(C2(CC)CCOC2)=O)C)ccc(C(C)C)nc1O 27186,c1(CNC(C2(C)C(C)(C)C2)=O)nnc2n1CCN(C(c1ccc(Cl)c(N)c1)=O)C2 27187,Cc1sc(C(=O)NCC23CC2CN(C(=O)CN(C)C(C)C)C3)nc1O 27188,c1(C(=O)NCC(C)CNC(C2CCCOCC2)=O)ccc2c(c1)CCCC(=O)N2 27189,C1(CN(C(c2ncccc2Br)c2n(C)nnn2)C2CC2)CCCOC1C1CC1 27190,N1(C(CC=C=C)=O)CCCC(NC(c2coc(Cl)n2)=O)CCC1 27191,Cc1cc(O)cc2c1CN(C1CC3CCC(C1)N3C(=O)Cn1cnnn1)CC2 27192,c1(COC2CC(CC(=O)NCC(CC)OC)C2(C)C)nc2cc(Cl)ccc2s1 27193,n1(CCC)cc(C(=O)NC2CC(N(C(=O)Cc3cccn3C)C)C2)c(C)n1 27194,C1(C#N)(CC)CCN(C(=O)CCN(C)C(c2cc(C3CC3)[nH]n2)=O)CC1 27195,c1(OC)cccc2c1CN(N1CCC(Br)=C(C)C1)CC2 27196,CC(C(CO)NC(c1cnc(C2CC2)[nH]1)=O)NC(=O)C(c1cccn1C)=O 27197,c1(C(N(CCNC(c2n(CC)c(O)nc2)=O)C2CC2)=O)sc(C)c(Br)c1C 27198,Cc1ccc(C(N2CC=CC(NC(c3cccn3C)=O)C2)=O)c(F)c1F 27199,c1(C(=O)NC2CCN(C(C3C(=C)C3)=O)CC2F)c(C)c2cc(O)ccc2oc1=O 27200,c1(CC(=O)NC(CC=C)CNC(=O)Cc2cccc(Cl)c2)ccc(C)cc1Cl 27201,c1(C(=O)NC2CCN(C(c3c(SC)ccs3)=O)C2)cc2c(cn1)OCCC2 27202,C1(NC(c2cn(CCC)nn2)=O)(CO)CCCN(C(C2(F)CC=CC2)=O)C1 27203,CCC(CC)C(C)C(=O)NCCCC(C)(C)NC(C1CCC(C)O1)=O 27204,N12CCC(F)(F)C(C1)C2.Cc1c(CNC(c2ccccc2)C2CC2)c[nH]c1C#N 27205,c1(C(=O)NC2(C)CC(NC(C3(C)N(C)CC(O)C3)=O)C2)cc(F)c(Cl)cc1F 27206,N1(C(C(CSC)C)=O)CCCCCC(NC(c2cc(C)cnc2C)=O)C1 27207,c1(C(=O)NCCNC(Cc2c(C)n[nH]c2C)=O)ccc2c(c1)N(C)C(=O)C(C)O2 27208,Cn1cc(C(=O)Nc2cccc(CN3C(=O)CNC3=O)c2)nc1O 27209,N(C(=NCCc1ccccc1F)NCC1=CCOCC1)Cc1cc(C)on1 27210,C1(C)(CNC(c2c(C)nco2)=O)CCN(C(=O)CSCc2cccnc2)CC1 27211,C(C(C(C)(C)C)NC(C1(O)CC1)=O)NC(c1cc(C(=O)OC)sn1)=O 27212,C1(CNC(C(C)OCC)=O)(OC)CCN(C(C2CN(CC)CCO2)=O)CC1 27213,C(=O)(CC(=O)N(CC(=O)N(C1CC1(C)C)C)CC1CC1)NCC 27214,c1(CC=CCC(=O)NCCCCN(C)C(C2CCC3CC23)=O)ccccc1 27215,C(C(CC(C)C)C(=O)NC(c1ccccc1)CO)NC(c1cnn(C=C)c1N)=O 27216,CCC(CC(=O)NCC1COCCN(C(=O)C(F)C2CCCC2)C1)CC(C)C 27217,CCC(C)(C)CCCC(=O)NCCC1CCN(C(=O)COC(F)(F)F)C(C)C1 27218,Cc1ccc(C2(C(=O)NCC(C)CNC(=O)CC3CCC(C4CC4)O3)CC2)cc1 27219,Cc1cc(C)c(C(=O)NCC(C)C(=O)NCCc2nccs2)s1 27220,C1(CC=C)(NC(=O)C(C)c2ccsc2)CN(C(C2CC(CC(F)(F)F)C2)=O)C1 27221,C1(CNC(CSCC=C)=O)CCCN(C(=O)C(C)Cn2ccc(C)n2)C1 27222,C(=O)(C#CC(C)(C)C)N(C1CCN(C(c2ccccc2-n2cccn2)=O)C1)C 27223,c1(C(N(CC(F)(F)F)CC#C)=O)cn(C2CCCNC2)nn1 27224,C1(C(=O)NC(C(=O)OC)(C)Cc2ccncc2)CNCC12CCOCC2 27225,Cc1ncc(C(=O)NCC2CC(F)CN2C(=O)CC2CCOC2=O)n1C(F)F 27226,c1(N2CCC(OCC)CC2)nc(=NCc2cc[nH]c(=N)c2)[nH]c2c(C)nn(C)c12 27227,CCCCC(F)(F)C(=O)N1CCC1CNC(C1CCC(F)(F)C1)=O 27228,C(CC(C)C(=O)N1CC(c2ocnc2CNC(c2sccc2C)=O)C1)OC 27229,c1(OC)nc(O)ccc1NC(=O)Nc1ccc(NC(=N)N)cc1 27230,C1(c2onc(Cc3n(C)ccn3)n2)CC12CCSCC2 27231,c1(CC)cc(CC)nc(N2CC3C(CNC(=O)C(c4cnn(C)c4)C)C3C2)n1 27232,N1(C(COCCCC)=O)CC2CCC(CNC(C3CC3(C)CC)=O)(C2)C1 27233,C(C(CO)C(C)CC)NC(C1C(CCC)CN(C(=O)C(C)(C)N(C)C)C1)=O 27234,C1(C(C)CNC(C2CCCS2)=O)CCN(C(=O)Cc2cc(Cl)n(C)n2)CC1 27235,C12(C(N3CC(CC(C)NC(c4cccc(N)n4)=O)C3)=O)CC3CC1(CO)CC3C2 27236,C1(C(N)=O)CCN(c2nnnn2-c2nc3c(s2)CCC3)CC1O 27237,c1(C(=O)NC(CCCC)CNC(c2ccc[nH]2)=O)cnc(O)c2ncccc12 27238,C(=O)(CC(C(C)(C)C)NC(c1cc(F)ccc1F)=O)N(CCN=[N+]=[N-])C 27239,N1(C(Cc2nc(C)sc2)=O)CCN(C(c2sc(C3CC3)nc2C)=O)CC1C1CC1 27240,N1(C(C(C)Cn2cccn2)=O)CCCC(CC(N2CCC(CCO)CC2)=O)CC1 27241,Cc1nn(-c2ccncc2)cc1C(=O)N(CCCNC(=O)C(C)(C)CF)C 27242,C(=O)(CCC(=O)NC1CCC1NC(=O)CCCCN1C(=O)CCC1=O)NC 27243,CCCCCC(C)CC(=O)NCc1cc(C(=O)N(c2cccc(C)c2C)C)cs1 27244,C(=O)(CC(CC)CC(C)C)NC(CCC(=O)NCCC(=O)NCC(C)C)C(C)C 27245,N1(c2ccnc(COC)n2)C2CCC1(CNC(c1cccc(F)c1F)=O)CC2 27246,c1(C(=O)NCC(C)N(C(=O)C=CS(C)=O)CC)cc2ccncc2c(O)n1 27247,c1(OC)ccc(C(N2CCN(C(c3c[nH]ccc3=O)=O)C(C)C2)=O)cc1F 27248,CCC(CCC(=O)NCC(O)Cn1cccn1)NC(c1nc(CC)oc1C)=O 27249,C1(NC(C(C)c2ccco2)=O)CN(C(=O)C=CC2(C)COC2)CC1C1CC1 27250,N1(C(CCC(C)(C)C)=O)CCOCC(C)(CNC(C2COCCC2(F)F)=O)C1 27251,Cc1cnc(CCNC(=O)NC2CCN(C(C)C)C2)o1 27252,C12(C=O)CCCCC1CN(C(=O)CCCS(N)(=O)=O)C2.CCC1CC(=O)N1 27253,N1(C(C(C)n2cncn2)=O)CC2CC2(C(=O)NOCCF)C1 27254,CC(c1ccccc1)=CC(=O)NC(CC(=O)N1CCC(C)C1)C(F)F 27255,c1(C(N2C(COC)(CNC(=O)C=C(C)C(C)C)CCC2)=O)cccc(F)c1C#N 27256,C1(CCn2cc(C3N(C(c4c(C)csn4)=O)CCC3)nn2)CCCN(C)C1 27257,c1(C(C(=O)NCC2CCN(C(=O)C=Cc3nccs3)C2)O)cc(Cl)cc(Cl)c1 27258,C1(NC(c2c(C)ncnc2)=O)(CO)CCCN(C(c2ccccc2Br)=O)C1 27259,C=CCCCCCC(=O)N1CCCC(C(C)NC(=O)NC)C1 27260,Cc1sc2ncc(C(N3CC(CC(C)NC(C4(C)CCCC4C)=O)C3)=O)n2c1C 27261,C1(SC)CN(C(C2(OC(C)C)CCCCC2)=O)CC1NC(=O)C=C(C)C 27262,C(=O)(C1=NOC(C)C1C)NC1(CNC(c2c(N)sc(C)c2C)=O)CCOC1 27263,N1(C(CCC(C)(F)F)=O)CCc2sc(CNC(=O)C=C3CCCCC3)nc2C1 27264,C1(C(=O)NCCC2N(C(C3CN(C(N)=O)C3)=O)CCOC2)CS(=O)(=O)CC12CC2 27265,c1(C(N2CCN(C(C(C(C)C)C)=O)CC2C2CC2)=O)cccc2ccnn12 27266,N1(C(CNC(C(C)(C)C2CCCC2)=O)=O)CCN2C(=O)CCC2C1 27267,C#Cc1cncc(CN2CCN(C(=O)CN3CCCCC3)C(CC)C2)c1 27268,N1(C(CCOCC#C)=O)CCC(C)C(NC(c2ccc(NC(C)=O)cc2C)=O)C1 27269,c1(CCC)ccc(C(=O)NCC(C(C)C)NC(=O)C(C)CSC)cc1[N+](=O)[O-] 27270,C1(NC(C(C)OCC)=O)CCCC1(C)CNC(c1cc(Cl)cs1)=O 27271,CC(C)CCCC(C)CNC(C1CC(C)CN(C(c2cncc(F)c2)=O)C1)=O 27272,CC(C)CC(C)CC(=O)NCC1CC(CNC(=O)CC(=O)NCC(F)(F)F)C1 27273,c1(-c2c(C)n[nH]c2)ccc(C2(NC(C3CCC(=O)N3)=O)CC2)c(F)c1 27274,c1(C(=O)NC2C(C)(C)C(CC(=O)NCc3cc(Cl)ccn3)C2)cncc2[nH]ccc12 27275,C(=O)(C(F)(F)c1cncs1)NC(n1cncn1)CNC(C1(C2CCCO2)CCC1)=O 27276,N1(C(C(COC)C)=O)CCCC(O)(CNC(c2ccc(C(F)(F)F)cc2Cl)=O)C1 27277,C(=O)(C(C)C(C)(C)O)NC1CCCN(C(CCSc2c(OC)cccc2)=O)C1 27278,c1(C(=O)NCCCC2N(C(CC(C)SC)=O)CCCC2)cccc2nncn12 27279,c1(C(C)C)n[nH]cc1C(=O)NCC(O)CN(C(=O)CCc1ccsc1Cl)C 27280,C1(NC(c2csc(C)c2C2CC2)=O)CCCC12CN(C(=O)Cn1ccnc1C)C2 27281,c1(NC(C(C2CCN(OC)CC2)N(C)CC2(C)CC2)=O)ccc2c(c1)OCCO2 27282,c1(CN(C(CCNC2CC(=O)C2)=O)Cc2cnccn2)ccccc1 27283,C1(CNC(CCC=CC)=O)CN(C(=O)C(C)Cc2ccncc2)CC2(CCC2)O1 27284,N1(C(CCC#N)=O)CCCC12CCCN(C(c1ccc(S(=O)(=O)CF)cc1)=O)C2 27285,C1(C(N(C2CN(C(=O)CSc3ccn(C)n3)C2)C)=O)CCn2ccnc2C1 27286,N1(C(CC(CC)OC)=O)C(C)CC2CN(C(c3cnnc(C)c3C)=O)CC12 27287,CC(C(CO)NC(=O)CCc1cncn1C)NC(c1cn(C2CCC2)nn1)=O 27288,c1(C(N(c2ccccc2)CCCC)=O)ccc2c(c1)CNC2=O 27289,C1(NC(C(CSC)C)=O)CCSC12CN(C(=O)CCc1ccc(O)c(F)c1)C2 27290,CCCCCC(CC)C(=O)NC1CC(NC(c2ccc(Br)cc2C)=O)C1 27291,c1(C(N2C(C)(C(=O)Nc3cccc(OC)c3)CCC2)=O)cc(Cl)cnc1Cl 27292,C(=O)(C(C)CC(F)F)NCC(CCCC)NC(=O)C(C1CC(F)(F)C1)O 27293,C1(C(=O)NC2CC3CN(C(c4c(C(C)C)scn4)=O)C2C3)CCC2(CCC2)CC1 27294,c1(OC)ccc(C(=O)NC2CC2NC(c2cc(C)cc(F)c2)=O)cc1C1CC1 27295,CC1(CNC(=O)CN2CC=CC2)CC(NC(c2ncsc2Br)=O)C1 27296,Cc1noc(C(C)C)c1C(N1CC(C(C)NC(c2c(C)n[nH]c2C)=O)C1)=O 27297,c1(C(N2CCCC(CN(C)C(C3(Cl)CC3)=O)C2)=O)ccc(Cl)c2occc12 27298,C12(C(N(OCC)CC)=O)CCCC1CCN2C(=O)CCC(C)(C)C#N 27299,C1(C(C(=O)NCc2c(CC)c[nH]n2)C)CCN(C(=O)C(F)OC(F)(F)F)CC1 27300,CC1CN(C(=O)C2=CCCCC2)CC(CCNC(=O)CCc2ccn(C)c2)O1 27301,c1(C(=O)NC2CC2NC(c2noc3c2CCCC3)=O)ccc2cccnc2c1 27302,Cc1nn(Cc2ccccc2Cl)c(Cl)c1C(=O)OCC1C(C)(C)C1(F)F 27303,c1(NC)ccc(C(N2CCC(CC)C2C(N2CC(OC)C2(C)C)=O)=O)cc1 27304,C(=O)(CCCCC(=O)N1CC(O)(C(F)C(=O)N(C)C(C)C2CC2)C1)OC 27305,CC1(F)CCC(C(N2CCC(C(C)(C)NC(=O)C(F)=C3CCC3)C2)=O)CC1 27306,CC(C)C(CC(=O)NCC(C)CNC(c1cnc(C2CCC2)s1)=O)C(C)C 27307,CC#CCCCC(=O)NC1(CCO)CN(C(=O)C(C)SCCC(C)C)C1 27308,c1(C(N2C3C(C(=O)Nc4ccc(F)cc4O)C(C3)C2)=O)cc(O)ccc1[N+](=O)[O-] 27309,C1(C)(CNC(C2(C)C(C)CCC2)=O)CCCN(C(c2ccc(F)s2)=O)C1 27310,C1(C(=O)NCC2N(C(c3cc(C)oc3)=O)CCC2C)CCc2nncn2C1 27311,N1(C(C=CCC(C)NC(C2(O)CCCCC2)=O)=O)CC(CO)CC12CCC2 27312,c1(OC)cccnc1C(=O)NC1(C)CC(NC(=O)CCC2CCCO2)C1 27313,c1(CC)c(C(=O)N(CC(C)NC(=O)CC2(O)CCCC2)CC)cnn1C(C)(C)C 27314,Cc1ccc(C(=O)NC2CC(CNC(=O)CS(C)(=O)=O)C(O)C2)c2c1CCCN2 27315,C(C)(C)(CC=CC(=O)NC1CC(CO)C1)NC(CCOC)=O 27316,C(=O)(C1=COCCO1)NC(CC)CNC(=O)CCC(=O)NCCOc1ccccc1F 27317,C(=O)(C(CO)NC(C1CCCN1CCC)=O)NCC=C 27318,c1(C(=O)NC2CCCC2c2nc(S)n[nH]2)cc(O)nc(C2CC2)n1 27319,C1(CC)CN(C(c2cc(C)oc2C)=O)CCC1NC(c1cnn(CC(F)F)c1)=O 27320,Cc1ncnc(C)c1OCC(=O)N(CC(C)CNC(C12CC(CCO1)C2)=O)C 27321,c1(NCC2(CNC(c3c(F)cccc3Cl)=O)CCCC2)ncnc2ccccc12 27322,c1(NC(C)=O)cccc(C(N2CC(O)(C(C)NC(C3CC34CCCC4)=O)C2)=O)n1 27323,Cc1cc(C)c(C(=O)NC(C)(C)CCCNC(=O)Cn2nnnc2C(C)C)[nH]1 27324,CCCC(C)(C)C(=O)N1CCC(C)(NC(=O)CSCC(N2CC3CCC2C3)=O)C1 27325,C1(C(=O)NCc2ccc(F)nc2F)CC12CCN(C(c1cc[nH]n1)=O)C2 27326,C#Cc1cccc(CNC(=O)C=C(C)CNC(=O)C(C)(C)C(N)=O)c1 27327,C#Cc1cn(C)nc1C(N1CC(NC(C2CC3CC(=O)C2O3)=O)CC(O)C1)=O 27328,C(=O)(CCC(=O)c1ccncc1)N1CC(OCCNC(C2CCNC2=O)=O)C1 27329,C1(C(=O)NCCNC(c2c(OCC)oc(C)n2)=O)CC1C1CC(F)(F)C1 27330,c1(SCCC(=O)NC2CC(C)(NC(C(CCN(C)C)O)=O)C2)cc(F)ccc1F 27331,C1(CC#C)CC(=O)N1.C1(n2cc(-c3ccc(F)cc3)nn2)(CC#C)CCOCC1 27332,C(=O)(CC(O)CC(C)C)NC(C(=O)NC(C#C)C)C1(C)CC1 27333,Cc1ccccc1OCCC(=O)NC(c1nccs1)C1CCC1 27334,Cc1cc(C)c(C(=O)NC2(CNC(C3(CF)CC3(F)F)=O)CCC2)s1 27335,c1(OC)ncccc1-c1cn(C(C)CNC(c2cc[nH]c2C2CCC2)=O)nn1 27336,c1(C(=O)NCC#CCC(=O)NCCC(COC)O)ccc2c(c1)CCC2 27337,C1(C(=O)NCC2CCC(C(=O)NCCCc3nccs3)C2)CCCC(O)C1 27338,c1(C(N(C2C(N(C(C=C(COC)C)=O)C)CCCC2)C)=O)cnc2sccn12 27339,N1(Cc2c(OC)ccs2)CCN(C(c2ccc(C(F)(F)F)[nH]2)=O)C2CC12 27340,CC(C)C(C(=O)Nc1cncc(C#N)c1)C(C)NC(C1CC(O)C1)=O 27341,C1(C(=O)NC2CC3CC(NC(C4=CC(C)(C)C4)=O)CC32)COc2ccccc2O1 27342,C(=O)(C(C)CC(N)=O)NCc1cn(CC2N(C(CSCCOC)=O)CC=C2)nn1 27343,C(=O)(C(C)CN(C(=O)CSCC(N)=O)C)N1CC(C(=O)OC)C1 27344,N1(C(c2ccc(C(C)C)o2)=O)CCOC(C(N)=O)CC1.C1(NC=O)CCC2(CO)CC12 27345,C1(CC(N2CCC(CC=C)C2)=O)CN(C(c2cc(O)n(C)n2)=O)CC1C 27346,Cc1c(C(=O)NCC(C(C)C)NC(=O)COC(F)F)cnn1CCC(C)C 27347,CC(C)CCC(F)C(=O)N1CCC2(CC2C(N2CC3(CCOC3=O)C2)=O)C1 27348,c1(C(N(CC(C)(C)CNC(C2(CC)CCCC2)=O)CC)=O)cc(C)cc(O)c1 27349,c1(C(=O)NC(C)CCCNC(C2CC2(Cl)Cl)=O)ccc(N)cn1 27350,N1(C(c2cn(CC=C)nc2)=O)CC(NC(c2onc(CC)c2C)=O)CC1CO 27351,C=CC(C)C(C)C(=O)NCCCN(C)C(c1cncc(C#N)c1)=O 27352,C1(C)(CNC(C(C=CCCC)O)=O)COCCN(C(c2ccccc2O)=O)C1 27353,CC1(C(=O)NCCn2cnnn2)CC(O)CN1C(=O)Cc1nc[nH]n1 27354,Cc1cccc2c(C(=O)NC3CC4CC3N(C(=O)C3=CCCS3)C4)c[nH]c12 27355,c1(CC(=O)NCCC2CCCCN2C(=O)C=C2CCC2)n[nH]c2ccccc12 27356,c1(-c2nc(C)nn2-c2ccc(F)cc2)ccc2ccccc2n1 27357,C1(C)(CNC(c2ccc(C#C)cn2)=O)CC(F)(F)CN1C(C1COC(=O)O1)=O 27358,c1(OC)ncccc1CC(=O)N(C)CC1(O)CCN(C(=O)CC2(O)CCOC2)C1 27359,C1(N(C)C(C2(C(F)F)CCCO2)=O)CCN(C(c2ccc(CO)nc2)=O)CC1 27360,C1(N(C(=O)CC2CCCC2)C(C)F)CCCN(C(c2oncc2C2CC2)=O)C1 27361,N1(C(CCC=C)=O)CCC(C(N2CCC(N3CCC3)CC2)=O)C(C)(C)C1 27362,C(C)(C)(CN=c1nc(C)cc(C)[nH]1)NC(c1ccc(C#C)cc1)=O 27363,N#Cc1ccc(S(N)(=O)=O)c(N2CC3CC2C2OCCOC32)c1 27364,C1(O)(CNC(CC2(COC)CC2)=O)CCCN(C(C2(N(C)C)CCC2)=O)C1 27365,n1(C(C)C)cnc(C(=O)NCC(C)(C)NC(=O)C(C)NC(c2cccs2)=O)n1 27366,C(C1CCCCCC1)=CC(=O)NCC1N(C(c2c(C)noc2C(F)F)=O)CC1 27367,C1(O)(CNC(CCCN(C)C)=O)CCCN(C(=O)CC2CCC(C)(C)CO2)C1 27368,Cn1cc2c(C(N3CCCC(O)(CNC(C4(C5CC5)CC4)=O)C3)=O)cccc2n1 27369,N1(C(C2(CCC=C)CN(C(=O)C=CC(=O)N(C)C)C2)=O)CCS(=O)C(C)C1 27370,CC1CN(C(C2CCCCN(C(C3CC(F)(F)C3)=O)C2)=O)C2(CC2)C(=O)N1 27371,c1(SC)cccc(OCC2CCCN2CCC(C)NC(=O)COC2CC2)c1 27372,CC1(C)COC(C(=O)NC2CCC(CC(N3CCOCC3CO)=O)C2)C1 27373,C1(NC(C(C)CC2CCCCC2)=O)CCN(CCCN(C)C)CC1C 27374,c1(C(=O)NCC(CO)NC(c2cc(Cl)cnc2O)=O)ccc2c(c1O)CCC2 27375,C=CCC(CC=C)C(=O)N1Cc2[nH]nc(C(=O)NC3CCC3(C)C)c2C1 27376,CC(C)C(CCN(C(=O)CCC1(N(C)C)CCCC1)C)NC(=O)CNC(N)=O 27377,N1(C(C2CC(SC)C2)=O)CCN(C(c2ccnn2C2CCOCC2)=O)CC1 27378,N1(C(C2CCC(=O)N2)=O)CC2(CCCN(C(C3C4CCCC34)=O)C2)C1 27379,N1(C(COC2(C)CCC2)=O)CCOC(C(C)(C)NC(c2ccc(C(N)=O)[nH]2)=O)C1 27380,C1(C)(C(=O)NCc2cn(C(CC)C)nn2)CCC2CC2C1 27381,C1(NC(c2cc(COC)no2)=O)CCN(C(=O)C(F)(F)C(F)(F)F)CC12CCC2 27382,c1(CC(=O)NC2CC(F)(CNC(c3cn[nH]c3)=O)C2)cccc2ccccc12 27383,Cn1nc(-c2nc(-c3cccc4nnsc34)no2)c2c1CNCC2 27384,C(=O)(C1CCCn2cnnc21)N(CCCNC(C1CC2(C1)CC21CCC1)=O)CC 27385,C(=O)(C(O)C(C)(C)CC)NCCCOCCC(NOCC(=C)C)=O 27386,C1CCCC(=O)N1.c1(SC)ccc(C(N2CC(Oc3ccccn3)C2)=O)s1 27387,CC(C)C(C)C(CNC(=O)C=Cc1ccnn1C)NC(c1occ2c1CCC2)=O 27388,C(CC(=O)NC(c1ccccc1C)C)(C(F)(F)F)NC(CC(C=C)C)=O 27389,CC1(C(=O)NCC2C(C(=O)Nc3cnn(CC4CC4)c3)C2(C)C)CNC(=O)C1 27390,C1(CC=C)(C(=O)NCC(F)CNC(C2CCCN2CC)=O)CCCCC1 27391,c1(C(N2C(CNC(CC(CC)C3CC3)=O)C=CC2)=O)ccc(OC)c2ccsc12 27392,c1(C(C(C)N(CCOCCN(CC)CC)C)C)ccc(C)s1 27393,C1(CNC(Cc2c(C)non2)=O)CCCN(C(C2SCCS2)=O)CC1 27394,N1(C(Cc2n[nH]c(=N)s2)=O)CC2CC1CCC2NC(c1cncc(C2CC2)c1)=O 27395,c1(OC)ccc(O)cc1C(=O)NCC(C)CNC(=O)CC(C)=C(C)C 27396,c1(NCC(C2CCCC2)NC(c2ccn(C)n2)=O)ncc2c(ncn2C)n1 27397,c1(N2CCN(C)C(CNC(c3cccc(C(F)F)n3)=O)C2)ncc(C#N)cc1F 27398,c1(CC)ccsc1C(=O)N(C1(CC(=O)NC2CCSC2)CC1)C 27399,c1(CCC(C)NCC(=O)OCc2cc(N3CCCC3)ccn2)ccc(Cl)cc1 27400,c1(C(N2CC(CC(=O)Nc3cnc(Cl)nc3)OCC2)=O)cnn2ccccc12 27401,C1(C(N2CCN(CC(=O)N(CCC)C(C)C)CC2)=O)COCCN1C(=O)NC 27402,C(=O)(C#CC1CCCC1)N1CCN(C)C(C(N2CCC(O)(C(F)F)C2)=O)C1 27403,C1(c2cccc(C)c2)CCCN(N2CCNC(=O)C2C2CCNCC2)C1 27404,N1(C(c2ccc(SC)s2)=O)CC2CCCC2(CNC(=O)CCCC#N)C1 27405,Cc1[nH]c(C)c(C(=O)NCC(C)(C)CNC(=O)CC2CCC(C3CC3)O2)c1C 27406,c1(OC)ccc(CCC(=O)NC2CC(C)(NC(C3CCCC3(C)C)=O)C2)cc1F 27407,C1(NC(C(CC)OC)=O)CC1C1CCCN(C(=O)C(=O)C(F)(F)F)C1 27408,C(=O)(C(C)CCCC(C)=O)NCCn1cc(C(=O)NCC(C(F)(F)F)OC)nn1 27409,N1(C(C23CC(NC(CCC4N(C)CCC4)=O)(C2)C3)=O)CCC2C(C(N)=O)C2C1 27410,Cc1cc(C(N2CCC(NC(c3cc(F)c(Cl)cc3Cl)=O)C2C)=O)cc(F)c1C 27411,c1(C(=O)NCCCN(C(c2nc(Cl)cs2)=O)CC)ccnc(C(C)(F)F)c1 27412,CC1(CF)CN(C(C2(C3CCCN3C(c3cnccn3)=O)CC2)=O)C1 27413,C(CCC(C(=O)NCCC1CC1C)NC(c1cn(C)cn1)=O)OC 27414,N1(C(c2cc(CNC(C3N(C)CCCC3)=O)on2)=O)CC2(CNC(=O)N2)C1 27415,CC1OC2(CNC(C3C(C)OC(C)C3C)=O)CC1(NC(C1CCCOCC1)=O)C2 27416,CCCCCCC(C)NC(=O)C1=CCN(C(=O)CCC2CCCO2)C1 27417,S(=O)(=O)(c1ccc(N2CCn3ncc(Cl)c3C2)nc1)NCC1C(C)COCC1 27418,Cc1ccc(C(N2CCCCC(CNC(c3n[nH]c(C4CC4)n3)=O)C2)=O)nc1O 27419,C(=O)(CCCS(C)(=O)=O)N(C)CC1(CNC(=O)CCCC2CCCC(=O)N2)CC1 27420,C1(CNC(CNC(C(CC)C)=O)=O)CCN(C(=O)CC2CN(C)C2)C1(C)C 27421,c1(C(N2CCOCC(C(N(CCC(=O)NC)CC)=O)C2)=O)cccc2ccoc12 27422,C1(CC(=O)N(CC(O)CNC(=O)C=Cc2cccs2)C)CCC(F)(F)CC1 27423,c1(NC(C(=O)NC(c2c(C)cccc2C)C)=O)ccc2c(c1)CCC2 27424,c1(C(N2CCC(N(C(=O)CC3C=CCC3)CCC)C2)=O)ncc(OC)nc1OC 27425,C1(NC(CNC(N)=O)=O)(CNC(c2ccn(C3CCCCC3)n2)=O)CCOC1 27426,CCCCC(CC)C(=O)NC1(CC(=O)NC2CCOC2C2CC2)CCC1 27427,c1(CN2CC(C)(CC(=O)Nc3ccnc(C(N)=O)c3)C2)ccc(Br)cc1[N+](=O)[O-] 27428,CC1(C)OCCC1C(=O)NCCn1ccc(C(N2CCC3CC23)=O)c1 27429,C1(NC(C=CC)=O)CC=C(C(=O)NCc2cnc(CC)[nH]2)C1 27430,C(=O)(CC(C)(C)C(=O)NC(CN(C(=O)C(C)NS(=O)(=O)CC)C)CC)OCC 27431,c1(NC(C2CCN(S(CC)(=O)=O)CC2)=O)cc(Br)cc(I)c1C 27432,C(CCCC)(CN=c1[nH]c(Cl)ncc1C(C)C)NC(C=CC(=O)NCCCC)=O 27433,c1(C2(CC)CC(NC(c3n(CC(=C)C)nnn3)c3ccsc3C)C2)cccc(Br)c1 27434,C1(NC(CCCOCC)=O)CC(NC(c2cc(CC)ccc2C)=O)C12CCC2 27435,c1(C(=O)NC(CCN(C(COC(C)C)=O)C)C)ccc2c(=O)ccoc2c1 27436,C(=O)(C(C)CC(C)C)N1CCC(C)(CC(=O)NCCNC(=O)OCC)C1 27437,Cc1c(NC(c2oc(CNC(=O)CC3CCC(C)C3)nc2C)=O)cnn1C(C)C 27438,c1(C(C)OC(=O)CCCN(C)C(=O)OC(C)(C)C)ccc(F)c(F)c1 27439,C(=O)(CN=c1cc[nH]cc1)NCCCCCNC(=O)CCC(=O)c1cccnc1 27440,C1(C(N(CCC(=O)OC)C)=O)(C(C)C)CCCN1C(c1ncn(C(C)C)n1)=O 27441,N1(C(=O)Cc2cc(=O)n(-c3ccccn3)[nH]2)CCn2cncc2C1 27442,c1(NC2CC3CC(OC)CC32)nc2c(F)cccc2c(=NCC(C)(C)C(N)=O)[nH]1 27443,C1(NC(CCc2cnn(C)n2)=O)CN(C(=O)C=C(Cl)Cl)CC1N=[N+]=[N-] 27444,Cc1cc(Cl)c(OCC(N2CCC(C)(O)CC2)=O)c(Cl)c1 27445,C1(CC(=O)NCC(C(C)C)OC)CCN(C(=O)CC2CCCC2)CC1 27446,c1(C(N(CCN(C(CSCC#C)=O)C)C)=O)ccc(C)cc1Br 27447,C1(CNC(c2cn(C)nc2)=O)CCCCCN1C(c1ccsn1)=O 27448,c1(CNC(C=CCC2(NC(c3n(C)ncn3)=O)CCC2)=O)cc(=O)cc[nH]1 27449,CC1(C)CN(C(C2(CCNC(c3ccc(=N)[nH]n3)=O)CC2)=O)CCC1O 27450,c1(C(N2CC3C(NC(C4C(CCC)C4)=O)(CC3)C2)=O)cc(S(C)(=O)=O)co1 27451,N1(CC(CCC)(C)C)CCC(O)C(C(=O)NCc2cccc(OC)n2)C1 27452,CCC(C)(CC)C(=O)NCCNC(C1CN(C(C23CCC(C2)OC3C)=O)C1)=O 27453,c1(C(N(C2CCN(C(C34C(=O)C5CC3C4C5)=O)C2)CC)=O)cc(=O)n(C)cn1 27454,CC(C)C(CNC(=O)CCc1cc(Cl)no1)NC(=O)C(C)OCc1ccccc1 27455,c1(OC)cc(C(N2CCC(C(C)NC(c3ccc(C)cc3C)=O)C2)=O)cc(F)n1 27456,C(=O)(C1=C(Cl)CCCC1)N(C(C(=O)NCC(C)N(C)C)CO)C 27457,CCCC(CC)CCC(=O)NC1C=CC(C(N2CCC(O)C2C)=O)C1 27458,C1(C(=O)NCC2(O)CC2)(COC)C=CCN1C(=O)CC1COCCOC1 27459,CCC(CC(=O)NC1CCC(NC(c2cc(F)cc(Cl)c2)=O)CC1)C(F)F 27460,N(C1COc2ccccc21)C(CC1CCN(C(c2cnc(C)n2C)=O)C1)=O 27461,CCCC(C(=O)NC(C(=O)NOCCN1CCCC1=O)C1(O)CCC1)C(C)C 27462,Nc1c(C(=O)NC2CCCCC2NC(C2CC2CF)=O)ccc(F)c1F 27463,c1(CC(C)(CO)N(CC(O)C2CCC2)C)cccc(Br)c1 27464,C#Cc1cc(C(=O)NCCC(C)NC(c2csc(C#N)c2)=O)cc(C(F)(F)F)c1 27465,C12(C(=O)OC)CCC(NCC3=CCS(=O)(=O)C3)(C1)OC2 27466,N1(C(c2cc(COC)cn2C)=O)CCN(C(=O)CN2CCSCC2)CC1CF 27467,c1(NCCCC(C)O)[nH]c(=NC(CC2CC2)c2ccccc2Cl)nc2sccc12 27468,C1(N(C(c2c(OC)csc2)=O)C)CCCC2CN(C(C3CCN(C)C3=O)=O)CC12 27469,C1(C(N)=O)(CC2CC2)CN(C(=O)CCO)C1.c1(CC(=O)NC)cc(C2CCC2)on1 27470,c1(C(=O)NCC(O)CNC(C2(F)CCOC2)=O)ccc2ccccc2n1 27471,C1(CNC(CC(C)OC)=O)CC2(CCC2)CN1C(C1CN(CC(F)(F)F)C1)=O 27472,C1(C(=O)NCCOCCN(C(C2C(C)C2C)=O)C)C(F)(F)C12CCC2 27473,c1(C(=O)NCCC2N(C(C(C)CCO)=O)CCCC2)c([N+](=O)[O-])cnn1C 27474,CC1CCCc2cc(C(=O)NCC3(O)CCCN(C(=O)Cc4ccsc4)C3)nn21 27475,C1(C(=O)NC2COCCN(C(=O)Cc3ccoc3)C2)CC2(C1)CC(F)(F)C2 27476,CC1(C)CN(C(C2CCCOC2)=O)CC(C)(C)C1NC(C1CC1(C)C)=O 27477,c1(C(=O)NC)ccc(C(=O)NC2CN(C(C3COCCO3)=O)CCC2F)cc1F 27478,C1(CNC(C2CCC(CC)O2)=O)CC2(CC2)CN1C(=O)CCCc1cnccn1 27479,C1(NC(=O)C(CO)c2ccccc2)CCCCN(C(C2(CF)CCOCC2)=O)C1 27480,CCC(CO)CN=c1[nH]c(=NCc2cc(F)cc(Cl)c2)c2cc(Cl)ccc2[nH]1 27481,C#CC(C)(C)C(=O)NCCCC1CN(C(c2ccc(CC(N)=O)cc2)=O)CCO1 27482,c1(C(N2CC(C(=O)N(C3CC3)CC3CC3)OCC2)=O)cccc2[nH]ccc12 27483,c1(OCC)cc(C(=O)NCC2(C)CN(C(=O)C=CCN(C)C)CC2C)cc(F)c1 27484,c1(C(=O)OCC)cc(CNC(CC2OCCO2)CO)cc(Cl)c1 27485,c1(C(N2CC(O)(C(C)NC(CC(C)C(F)F)=O)C2)=O)cnc2c(c1)NC(=O)CO2 27486,c1(C(=O)NC2CC(N(CCCCC)C(C3CCCO3)=O)C2)c[nH]c2cc(F)ccc12 27487,Cc1cc(C(=O)NC2CCC(C(=O)NCC34CCC(C3)C4)C2)c(C)o1 27488,Cc1nc2c(o1)CCCC2CC(=O)N1CCN(C(c2ncc(Cl)s2)=O)CC(O)C1 27489,C1(C(N2CCCC(C)(CC)C2)=O)CCCCCCN1C(c1cncc(OC)n1)=O 27490,C(=O)(CCCC(F)(F)F)N(CC(CC)NC(C1(C)CCC(O)CC1)=O)C 27491,CC(CC(=O)NCCC1CN(C(=O)CNC(C2CCC2)=O)C1)C(F)(F)F 27492,C1(CNC(c2cc(C)nc(O)n2)=O)CCCC2(CN(C(=O)C(C)C(C)C)C2)O1 27493,C1(CC)CN(C(=O)CC2CCCCCCC2)CCN1C(C1CC=CCO1)=O 27494,c1(NC)cnc(Cl)cc1C(N1CCC(CCNC(=O)C(C(C)C)NC(N)=O)C1)=O 27495,CC1CC(C(=O)NC2(CF)CCN(C(C3CCN(C4CCSC4)CC3)=O)C2)=NO1 27496,C1(N(CC(=O)NC(C)C(=O)C2CCCC2)C(=O)OC)CCCCC1.C12(C)CCCC1C2 27497,c1(C(N2CCC(NC(c3cccc(OC)c3)=O)(CO)C2)=O)scc2c1OCCO2 27498,C1(NC(CCn2c(C)ccc2C)=O)CC(NC(=O)Cc2ccsc2)C12CCC2 27499,N1(C(C(CSC)OC)=O)CCN(C(=O)C(C(C)(C)C)c2cccc(C)c2)CC1C 27500,N1(C(C2C(CCC)CN(C(=O)C(C)C(O)C(C)C)C2)=O)CCc2oc(C)nc2C1 27501,N1(C(=O)NC2CC(C(N(C)Cc3ccco3)=O)C2)CCn2cnnc2C1 27502,C12(CNC(CC(=C)C)=O)CCC(CC1)N(C(c1ncc([N+](=O)[O-])n1C)=O)C2 27503,N1(C(CNC(CNC(=O)OC)=O)=O)CC=CC1CN(C(C(C1CCC1)OC)=O)C 27504,C(=O)(CCCCN=[N+]=[N-])N1CCCC(C(=O)NC(c2ncn(C)n2)C)C1C 27505,C(=O)(C(O)CC(=O)OC(C)(C)C)N1CCCC(NC(C(CCC)C)=O)C1 27506,N1(C(C2C(C)CC=CC2)=O)CCCCC(CNC(c2cccc(F)c2N)=O)C1 27507,Cc1ccccc1C1(C)CC1C(=O)N(C(=O)CN1CC(C2CCCO2)C1)C 27508,Cc1nc(C(=O)NCC(C)(O)CNC(=O)Cc2nc(=N)[nH][nH]2)c(C)n1C1CC1 27509,CC(CC(=O)NC1CC(CNC(=O)CC2(CO)CC2)CC1O)P(C)(C)=O 27510,N1(C(CC(=C)C)=O)CCc2sc(CNC(=O)CCc3c(F)cccc3Cl)nc2C1 27511,N1(C(C(C(C=C)O)(C)C)=O)CCC2(CCC(CC(N3CCC(O)C3)=O)CC2)CC1 27512,C(C(C(=O)OC)NC(=O)CC(C)NC(=O)CCN1CCOC1=O)OC 27513,C(CCCCC(=O)NCC(c1ccc(F)cc1)NC(c1cccn1CC)=O)=CC 27514,CC(C)CC(C(=O)NC1(C(O)CO)CC1)NC(c1nnc(O)nc1O)=O 27515,Cc1nn2cccnc2c1C(=O)NCC12CC1CN(C(C1CCS1(=O)=O)=O)C2 27516,c1(C(N2C(C(=O)NCCOCC)CC3CC32)=O)c(OC)cccc1Br 27517,C(=O)(C(O)C1=CCCCC1)N1CCOCC(C)(O)C1.CC1(C)CC2CCN1C2=O 27518,C1(NC(c2cc(C)oc2)=O)CCC(C)(C)CC1CNC(=O)CSc1ccncc1 27519,Cc1cc(O)cc(=O)n1CC(=O)NCC1(F)CC(NC(=O)C(CN(C)C)N(C)C)C1 27520,c1(C(N2CCC(NC(C(C(CC)O)(F)F)=O)C(O)C2)=O)cc(S(N)(=O)=O)oc1C 27521,C1(C(=O)NCC2C=CC(NC(C3(CC)CC3)=O)C2)COCCN1C(=O)COC 27522,Cc1cnc(Cl)cc1NC(C1CCCN(C(c2cccnc2C)=O)C1)=O 27523,c1(OC)ccc(F)c(C(=O)NC2CCN(C(=O)CCN(C)C)CC2F)c1F 27524,N1(C(CN(CCC#C)C)=O)CCN(C(=O)CSc2ccccn2)CC(C)(C)C1 27525,c1(OC(C)(C)C(=O)NC2CC(CNC(=O)C3=CCSC3)C2)cccc(N)c1 27526,c1(C(N2CCCCC(NC(c3c(C)c[nH]n3)=O)C2)=O)cccc2nc[nH]c12 27527,c1(C(N(C)CC2CCCN(C(C(C3CCC3)OCC)=O)C2)=O)ncnc(O)c1F 27528,N1(C(C2N(C(C)=O)CSC2)=O)CCCCC(CNC(c2nc(C)nn2C)=O)CC1 27529,c1(N(C)CC2(CC)CCCCC2)nc(N2CCCC(C(C)O)C2)nc2ccsc12 27530,c1(-n2c(C3CCCCN3C(C)=O)nc(CCOC)n2)cccc2ncccc12 27531,C(=O)(C(N)CCC(=O)Nc1cnc2n[nH]c(Br)c2c1)OC 27532,c1(OC)ccc(C(=O)N(CC(C)N(C(=O)Cc2ccoc2C)C)C)nc1 27533,C1(C(=O)NCC(C)S(N)(=O)=O)C(C)OCCN1C(=O)CC1CCOCC1 27534,Cc1nc(NCC2CN(C(C3C=CCC3)=O)CCC2C)ncc1Br 27535,N1(C(COCCCOC)=O)CCCC(NC(c2cc(CO)on2)=O)C1C 27536,C(=O)(C(F)C(C)CNC(C1C=C(C)CS1)=O)NC(C(=O)OC)C 27537,CC1CN(C(c2ccc(-c3ccncc3)s2)=O)CC(C)C1NC(c1cc[nH]c1)=O 27538,C1(CC)NC(=O)N(CC(=O)Nc2cc(C3CCCCC3)no2)C1=O 27539,Cn1c(C(=O)NC2(CNC(=O)CS(N)(=O)=O)CC(F)(F)C2)cc2sccc12 27540,c1(C(N2CC(F)(C(=O)OC)C2)=O)c(-c2cscn2)cncc1F 27541,Cn1ncc([N+](=O)[O-])c1C(=O)NCC12CC(NC(C3CCC(C)(C)C3)=O)(C1)C2 27542,C1(NC(C2CN(C)C2)=O)CC(CNC(c2conc2C(F)(F)F)=O)C1(C)C 27543,N1(C(CCN(CCCCC)C)=O)CCC2CCN(C(C3(C#N)CC3)=O)CC2C1 27544,c1(C(C)C)nc2ccc(NS(=O)(=O)c3cc(Cl)sc3Cl)cc2s1 27545,C1(NC(c2cc(C)n(C)c2)=O)CC(F)CN(C(=O)C(C)NC(c2cccs2)=O)C1 27546,c1(C(N(C)CC2(O)CN(C(c3c(C)nc[nH]3)=O)C2)=O)[nH]c(C)c(S(N)(=O)=O)c1C 27547,C1(NC(C(C)CO)=O)CC2CCC(C1)N2C(=O)CC1=NNC(=O)C1 27548,C12(NC(C(C)=C3CCCC3)=O)CCN(C(c3ccnc4[nH]nnc34)=O)CCC1C2 27549,Cc1c(Br)ccc(F)c1C(=O)NC(C(=O)OC(C)(C)C)C(C)O 27550,c1(C(N2CCC(C)(O)C2)=O)cc(-c2ccco2)cc2[nH]ncc12 27551,C1(C(=O)NCC(CN(C)C(C2(F)CCCCC2)=O)(C)C)CC2C=CC1C2 27552,N1(C(c2c[nH]nc2-c2ccccn2)=O)CC2CC(N=c3ccnc(Cl)[nH]3)C2C1 27553,c1(CC)nc(N2CCN(CCN(C)CCNC(C)=O)CC2)nc2c1cnn2C 27554,C(=O)(C(C(C)CC1CCCC1)N1CCC(F)(C(=O)OC)C1)NCC(=C)C 27555,n1(C(C)C)ccnc1NC(c1ncc(C2CC2)s1)c1nnnn1C(C)(C)C 27556,c1(C(N2C(CNC(c3cc(O)cc(F)c3)=O)CC2)=O)ccc(=O)n2c1CCC2 27557,CC(C)C(CCN(C)C(C1CCCC(=O)N1)=O)NC(=O)C(C1CCCCCC1)C 27558,c1(OC(C)CN(C)C(C2(C)CC=CC2)=O)cccc(N)c1 27559,CC(F)(CNC(=O)C=Cc1ncc[nH]1)CNC(C1CCC1)=O 27560,C1(C(N2C(CNC(c3cc(C)sc3C)=O)CCC2)=O)CCC2CC(C)CN2C1 27561,N1(C(C(CCC2CC2)NC(CN2CCC(C)CC2)=O)=O)CCCC(O)(C(C)C)C1 27562,S(=O)(=O)(c1ccc([N+](=O)[O-])cc1OC)N1CC(C(=O)NC(CC)C)C(O)CC1 27563,N1(C(C(C)NC(=O)N(C)CCS(C)(=O)=O)=O)CCc2ccsc2C1 27564,N1(C(C=CC(=O)OCC)=O)CCC2(COC(CNC(c3ncccc3F)=O)C2)C1 27565,c1(NC(C(C2(O)CCCCC2)NC(C2(CSCC)CC2)=O)=O)c[nH]ccc1=O 27566,N1(C(CSCC(=O)OC)=O)C(C(=O)NCc2conc2C(C)C)CC2CCCC12 27567,c1(C(=O)OCC=CCC)ccc(Oc2ccc(C(=O)O)cc2)cc1 27568,C12(C(=O)OC)CC(NCc3ccccc3)C1C2.C1CO1 27569,N1(C(CC=CC=C)=O)CCN(C(=O)CCc2ccccc2CSCC)CC12CC2 27570,c1(C(=O)NCc2cccnc2Br)n[nH]c2cc(C3=CCCCC3)ccc12 27571,C(C(=O)NCc1ocnc1C(=O)NCC1(F)CC(O)C1)(C(C)C)SC 27572,Cc1cccc(C(=O)NC2CCC(NC(C3CSCN3C(=O)C(C)C)=O)C2)c1F 27573,Cc1nocc1C(=O)NCC(C1CCCC1)NC(=O)C(C)c1ccco1 27574,N1(C(CCSc2n(C)cnn2)=O)CCCC(CCNC(=O)C(=O)NCC2CC2)C1 27575,N1(C(c2ccc(N(C)CC)cc2)=O)C2CCC1C(NC(C1(C)COCCO1)=O)C2 27576,S(=O)(=O)(c1ccc(CCC#N)cc1)N1CCC(C)CC1CCO 27577,CCCCC(F)C(=O)N1CCCCC(C(=O)NCCc2ccc(C)c(C)c2)C1 27578,N1(C(C2C(CC)CCCC2)C(=O)NC(C)C)CCc2ccc(Cl)c(F)c2C1 27579,N1(C(C=CC)=O)CC2CCCC2C1C(=O)N(CCC(C)C)C 27580,C1(NC(CN2C(C)CC2)=O)CCC(C)(NC(c2ccc(Cl)nc2N)=O)CC1 27581,C=CCCC(F)(F)C(=O)NC(CC)CCCC(=O)NC(c1nccn1C)C 27582,c1(C(N2CC3C(NC(C4CCC(C)(CC)O4)=O)C3C2)=O)c(C)nn(C)c1F 27583,CC1CCC(CC(=O)Nc2nn(C)cc2Br)CC1C 27584,N1(C(CNC(=O)NC)=O)CC(CNC(=O)CC(C)C)C(F)(CO)C1 27585,C(=O)(C(O)CC(C)C)NCC1C(NC(C(c2ccc(CCCC)cc2)C)=O)C1 27586,C1(CNC(c2ccc(SCC)nc2)=O)CC12CCN(C(C1CCOCC1)=O)CC2 27587,CCC(C)C(O)C(C)C(=O)NCC(C)(F)CNC(C1CCC(C2CC2)C1)=O 27588,C(C)(C(C(=O)N(C)CC1CCCC1)C(C)C)NC(c1snc(C)c1N)=O 27589,Cn1ncc(C#N)c1C(=O)NCc1ccnc(C(N2CCC(CO)C(O)C2)=O)c1 27590,C1(CC)CC(C(=O)N(C)CCNC(=O)C(F)OC(F)(F)F)CC(=O)N1 27591,NS(=O)(=O)c1csc(C(N2C3CCC2C(CNC(c2cncc(F)c2)=O)C3)=O)c1 27592,c1(CC)cc(C)c(C(=O)NC(C)(CNC(=O)CC2CCCOCC2)C2CCC2)o1 27593,c1(C(=O)NCCOCCNC(C(C2CCC2)OCC)=O)cc(CCO)on1 27594,N1(C(C(CCC)OC)=O)CCN(C(c2cnc(O)o2)=O)CC(CO)C1 27595,c1(C(=O)NCCN(CCOC)C(C2CCNC2=O)=O)cc(COC)c[nH]1 27596,c1(CC(N2CCC(NC(COC(CC)C)=O)C2)=O)ccc(F)cc1 27597,c1(OC)ccc(NC(C2(C)CCCN(Cc3ccc(F)cc3C)C2)=O)c(F)c1 27598,C1(CC)CCN(C(C)=O)C1C(=O)N(CCNC(c1scnc1C)=O)CC 27599,N1(C(c2cccnc2NCCO)=O)CCN(Cc2ncccc2Cl)CC12CC2 27600,c1(C(N2CC(CCC)C(C(=O)NC3CCSC3)C2)=O)ccc(=O)n(C)n1 27601,c1(C(N(CCCNC(C(C)OCC)=O)CCO)=O)cccc(CS(C)=O)c1 27602,c1(C(=O)NCCC2N(C(C3CC=C(C)CC3)=O)CCOC2)cc(C)c(C)cc1C 27603,CCCC(C(=O)NC(C)(CNC(=O)C(N1CCOC1=O)C)C1CC1)OCC 27604,CC1CC(C(=O)N2CCC(N(C(C3(C)CC(O)CN3C)=O)CC3CC3)CC2)=NO1 27605,N1(C(C=COCC)=O)CC(C)CN(C(=O)COc2cccc([N+](=O)[O-])c2)C(C)C1 27606,c1(C(N(C2CN(C(C3C(c4cccc(C)c4)C3)=O)C2)C)=O)[nH]c(C)c(C)c1C 27607,C(=O)(C1=CCCCO1)C(=O)Cn1ccc(C(F)(F)F)n1.C(CN)(N(C)C=O)C1CC1 27608,Cc1cccc(CNC(=O)CC2CCN2C(=O)CSC(C)(C)C)c1F 27609,CC1CCN(C(c2cncc(O)c2)=O)CC1CNC(=O)CSc1nncn1C 27610,C(C(C(=O)N(C(C)C(C)(C)C)C)C(C)(C)C)NC(c1n(C=C)ncc1)=O 27611,C(=O)(C1=COCCC1)NCC1(NC(=O)Cc2ccccc2F)CC(O)C1 27612,CC1CN(C(c2nnn(C)c2N)=O)CCN1C(c1cccc(OC(F)(F)F)n1)=O 27613,C(=O)(C1CCc2c(Cl)cccc21)NCC(CCCC)NC(=O)CS(=O)(=O)C1CC1 27614,C#Cc1cc(C(=O)NCC2(O)CC(NC(=O)CC3CCC3(C)C)C2)ccc1C 27615,N1(C(CCc2cnc(C)o2)=O)CC2CC1(c1cn(Cc3ccno3)nn1)C2 27616,N1(Cc2c(C)nc(Br)s2)CC2(CCN2C(=O)Cc2cncnc2)C1 27617,c1(C(=O)NC2CN(C(C#CC(C)C)=O)CC2O)ccc2[nH]c3c(c2c1)CCCC3 27618,C(=O)(C1=NOC(c2ccc(F)cc2)C1)NCCOCc1onc(CC)n1 27619,c1(CC2N(C(=O)NC3(COC)COC3)CC2)nc(C)c(C)s1 27620,N1(C(C(CCC)C#N)=O)CCCC(C)(C)C1C(=O)NCC1CC(SC)C1 27621,C1(CN2CCC(OCCN=[N+]=[N-])C2)CC(=O)N(C2CCCCCC2)C1 27622,N#CCCCC(=O)N1CCCC1C1CCN(C(C2(C(=O)NC3CC3)CCC2)=O)CC1 27623,Cc1cc(C)n(CCNC(C2CN(C(C)C(=O)NCC3CCCO3)CCO2)=O)n1 27624,c1(C(=O)NCC(C)NC(c2ccc(NCC)cc2Cl)=O)ccc2nonc2c1 27625,C12(CNC(c3cc(C)oc3)=O)CCC(CNC(=O)C=Cc3cnc[nH]3)(CC1)CO2 27626,N1(C(CC(COC)C)=O)CC2C3CCC(C2C1)N(C(c1cc(Br)co1)=O)C3 27627,c1(CNC(CCC=CC)=O)nc(CNC(=O)C(C)=C2CCCC2)cc(O)n1 27628,c1(CNC(N(CCNC)CCN2CCCC2)=O)cncc(OC)c1C 27629,N1(C(=O)NCC2CCCC3(CCC3)O2)CCC2(C1)OCCO2 27630,c1(CCC)c(C(=O)NC2CC2NC(C2(CO)CCCO2)=O)nnn1C(=O)OCC 27631,C1(C(=O)NC2C(NC(c3ccon3)=O)COC2)CC2(C1)CC(F)(F)C2 27632,c1(C(=O)NC2CCCCN(C(C3(COC)C=CCC3)=O)C2)cc(N)c(C)cc1C 27633,c1(CC)ccc(C(=O)NCCOCC2CCCC2)c(O)n1.C1CCNC(=O)CS1 27634,C12(C(=O)NCC(C)F)CCC(CC1NC(=O)CC1(O)CCC1)C2 27635,N(C1CCCn2ccnc21)C(C1CCN(C(c2cc(CC)ncc2)=O)C1C)=O 27636,C1(NC(c2cc(C#N)[nH]c2)=O)CC2CCC1(NC(=O)Cn1cc(Cl)cn1)C2 27637,CC(C)CC(CNC(=NCc1ccsc1C(F)(F)F)NCc1cncnc1)N(C)C 27638,CCCC(O)C(=O)N1CC(CNC(=O)C(C)OCCC(C)C)C1 27639,C1(C)(COC)CC(NC(=O)CCC(C)(C)F)CN1C(=O)C=C(Cl)Cl 27640,c1(C(N2CCC(NC(c3c(CC)non3)=O)C2CC)=O)cc(S(N)(=O)=O)co1 27641,c1(NCC(C)(C)n2ccnc2)[nH]c(=NCC2CCC(CO)O2)nc2scnc12 27642,N1(C(=O)NC(c2c(C)cccc2)C)CCCCC1(CO)CO 27643,C(CCN=C(NCc1csnn1)NCc1ccccc1)CC.Cc1cc(Cl)ccc1O 27644,C1(C(=O)OC)CCC1S(=O)(=O)N1CCCSCC1C1CC1 27645,Cc1ccc(Cl)cc1-n1nc(-c2cccnc2)nc1COC1CN2CCC1CC2 27646,C12(NC(CCCCCN(C)C)=O)CCCC1N(C(C1CCC(=O)C1)=O)CC2 27647,Cc1nn(C)c(C)c1CC(C)C(=O)OCC(=O)NCCCN1CCCC1=O 27648,N1(C(C2(CNC(=O)CCC(C)C)CC(=C)C2)=O)CC(=O)NC(CC)C1 27649,N1(C(C(C(C)C)SC)=O)Cc2ccnn2CC(NC(=O)Cc2cc(C)cs2)C1 27650,Cc1c(C)c(C)c(C(=O)NC2CCN(Cc3cn(CCCO)nn3)C2)c(C)c1C 27651,C1(COC2CCC2)CC(N(C)C)C1.C12(CC1)CC(=O)N(SC)C2 27652,C1(NC(CCSC)=O)CS(=O)(=O)N(C)C12CCN(C(=O)C1=CCCC1C)CC2 27653,CC1CN(C(=O)CC2(O)CCCCCC2)CCN1C(C1COC(=O)O1)=O 27654,C1(N(C(=O)CSSC(F)F)CC)CCN(C(C2CC2c2ccccc2)=O)C1 27655,C1(C(=O)NCCC2CCN(C(C(C)=C3CC3)=O)C2)C2CCC1(C)C2(C)C 27656,N1(C(C=NOC)=O)CCOC(C(C)NC(c2csc(C(F)F)n2)=O)C1 27657,c1(CC(=O)N(CCNC(C2CC(C#N)C2)=O)C2CC2)ccc(-c2nc[nH]n2)cc1 27658,c1(C(=O)NC(CC)CNC(c2cc(C)on2)=O)cc(O)nc2ccc(F)cc12 27659,c1(CC)ccc(C(=O)NC(Cn2ccnn2)C(=O)NC(C)(C)CSC)cc1 27660,c1(C(N2CC(F)(c3cn(C4CCOCC4O)nn3)C2)=O)c(O)cccc1Br 27661,C1(NC(=O)CCc2cccs2)CC2CCC1C(NC(c1ccsn1)=O)C2 27662,C1(C(C(=O)Nc2ccc(OC)cc2)N(CC(=O)NC)C(C)C)CC2C=CC1CC2 27663,N1(C(c2c(C)c(=O)cc[nH]2)=O)CCC12CCOC(C)(C)C2 27664,Cc1nnccc1Sc1ccc(Cl)cc1.C1(c2nnnn2C)C(C)(C)N1 27665,N1(C(C(=O)NCCOC)=O)CC(NC(C2CC23CC(F)(F)C3)=O)CC(C)(C)C1 27666,C(C(C(=O)N1CCC(SC)C1)C(C)(C)C)NC(C(CCOC)(C)C)=O 27667,N1(C(=O)CCN2CCC(F)C2)CCC2C(CCN2C(=O)CO)C1 27668,C1(CNC(Cn2ccc(C)n2)=O)CC(NC(c2cnc(CC(C)C)s2)=O)CC1O 27669,C12(NC(c3cc(C)c(F)cc3)=O)CCCC1N(C(c1cc(O)nn1C)=O)CCC2 27670,N1(C(CCNC(CC(C)C)=O)=O)CC(C(=O)NC2COCC2N(C)C)CC1(C)C 27671,CC(C)CC(C(=O)NCC(C)(C)C(N)=O)N(C(=O)CN1CCNC1=O)C 27672,N1(C(c2ccsc2Cl)C(=O)NCC2CC2)CC(OCC(F)(F)F)CC(OC)C1 27673,N1(C(C(C)CF)=O)CC(C2CCN(C(=O)C(C3CC3)C3CC3)CC2)C1 27674,C(=O)(CC(C)CCC(=O)N1CCOCC1CCNC(c1ncc(C)cn1)=O)OC 27675,c1(C(N(CC(CC)NC(C(CC=CC)C)=O)CC)=O)ccc2nc(C)nn2c1 27676,c1(C(C)C)cc(C(N2CCC(C(C)(C)NC(c3c[nH]ccc3=O)=O)C2)=O)nn1C 27677,c1(C(N2CCC3(NC(=O)C(F)=CC4CC4)C(C2)C3)=O)ccc2nnc(S)n2c1 27678,C(=O)(C#CC1CCOCC1)N1CCC(NC(C(C=CC)O)=O)C1 27679,C1(NC(c2c(OC)n[nH]c2)=O)CC1C1CCN(C(=O)CCC2CCOCC2)CC1 27680,C1(COC(C2CCS(=O)(=O)C2)=O)CC(=O)N(C(c2ccc(Cl)nc2)=O)C1 27681,c1(OC)ccc(NC(=O)CN2CCOCC2c2ccc(O)cc2)c([N+](=O)[O-])c1 27682,n1(CC(=O)NC(CCNC(CC(C=C)CC)=O)C)ccc(=O)n(C)c1=O 27683,N1(C(c2cc(OC)n(C)n2)=O)CC(C(=O)NC23CC(F)(C2)C3)C2(CCC2)C1 27684,N1(CC(=O)OC)CCC(C)C(NC(C2CCCCC2c2nc(S)n[nH]2)=O)C1 27685,Cc1ccc(C(=O)NC(CC(N)=O)C2CCOCC2)nn1 27686,c1(C(=O)Nc2nc(SCC)nc(Cl)c2)cnc2[nH]cnc2c1 27687,N1(C(CC)=O)CCOCC(CNC(=O)CC2CCCN2C(C)=O)C1 27688,c1(OC)cc(OC)c(-c2c(C)n[nH]c2C)cc1CN1CC2COC(=O)C2C1 27689,C1(C(F)(F)F)CCNC(=O)C(C)N1.c1(C(=O)NC(C)(C)C)cccc(F)c1 27690,C1(NC(Cc2nnc(C)o2)=O)CCCN(C(c2cc(C)oc2C(F)(F)F)=O)C1 27691,C(=O)(C1COc2ccc(F)cc21)N1CC2(CCN(C(C(CC=C)CC)=O)C2)C1 27692,C1(CN(C)C(C2(C#N)CCCO2)=O)COCCN1C(=O)Cn1nnnc1C1CC1 27693,C1(CNC(C2C3CCCOC23)=O)CN(C(=O)C=Cc2cc[nH]n2)CCO1 27694,Cc1cnc2n1CCCC2C(=O)NC1CCCC1NC(c1cncn(C)c1=O)=O 27695,c1(CCCC)nc(C)c(C(=O)NCc2ncoc2CCNC(=O)COC)s1.C1(CC)CC1 27696,C1(OCC)CCN(C(=O)CC2(C)CCN2C(=O)CC2CC(OC)C2)CC1 27697,c1(OC)ccc(C(=O)NC2(C)CCCN(C(C3(CCN(C)C)CC3)=O)C2)cc1Cl 27698,N1(C(C(F)OC)=O)CCN(C(=O)C2=CCCC2)C(C)C1 27699,N1(C(C2CC3C=CC2C3)=O)CCC2(CCC2)C(NC(C2(C3CCC3)CC2)=O)C1 27700,N1(C(C2N(C(C(CC)N(C)C)=O)CCC2CC)=O)CCC2C(O)CC12 27701,c1(C(=O)NCC2CCC(C(N3CC4(CCOC4)C3)=O)CC2)nccc2cc[nH]c12 27702,c1(C(=O)NCCC2CCCN(C(=O)C(O)C3CC3)CC2)c[nH]c2cccc(Cl)c12 27703,C12(NC(Cc3cnc(C)[nH]3)=O)CCOCC1CN(C(C1SCCCS1)=O)C2 27704,CC(C)(C)CC(=O)N1CC(O)CC1C(=O)NC(Cc1ccco1)CO 27705,C(=O)(C(C)S(C)(=O)=O)N1C(C(C)NC(=O)C=Cc2cc(C(N)=O)co2)CCC1 27706,c1(C(=O)NC2CC(N(C(=O)CC3CCCO3)C)C2)cnc2c(c1)CCOC2 27707,C(=O)(C(C)CC(C)(C)C)NCc1ccc(CN(C(c2onc(C)c2C)=O)C)cc1 27708,c1(C(C)C(=O)NC(C)(C)CNC(C2(C(C)(F)F)CC2)=O)cncc(F)c1 27709,C1(O)(CN(C)C(c2ccc(Cl)cn2)=O)CCN(C(C2CCC(CCO)CC2)=O)C1 27710,N1(c2ncnc3n[nH]c(C)c32)CCC2CC(CNC(=O)C=CI)CCC2C1 27711,Cc1cncc(CC(=O)NC2(CC(=O)NC3CCSCC3)CCCCC2)c1 27712,c1(C(N2CC3(CN(C(Cc4cc(C)on4)=O)C3)C2)=O)cccc2c1COC2(C)C 27713,C1(C(N2CCC(C(=O)NCC3C(C)(C)COC3)CC2)=O)CCC2(CCC2)C1 27714,C(=O)(CC1=CCOCC1)N(CCCC(=O)NC1CCNC1=O)C 27715,C(CC)(C(=O)NCC(O)CNC(C1(n2cccn2)CCC1)=O)OCC 27716,c1(SC)cc(C(=O)NC(C)CN(C)C(C2(c3ccccc3)CCCC2)=O)c(C)o1 27717,N1(C(c2scc(C)n2)=O)CCC(F)(CNC(C2CC2(Cl)Cl)=O)CC1 27718,CC1CN(C(=O)CC2CC2)CCN1C(C1CCCCC1)=O.c1(OCC)cnn(C)c1 27719,C=CCCC(C(=O)NCC)NC(=O)C=CCN(C(CCO)C(F)F)C 27720,c1(C(=O)NCCC2N(C(Cc3nnc(C)o3)=O)CCSC2)cnn2cnnc2c1 27721,c1(C(=O)NC(C(C)NC(C2CNC(=O)N2)=O)CO)cnc2nccn2c1 27722,c1(C(=O)NCCNC(c2ccc(F)cc2CC2CC2)=O)cc(F)c(O)c(Cl)c1 27723,C12(NC(C3Cc4ccc(F)cc4C3)=O)COCCC1CN(C(c1ccsc1)=O)C2 27724,c1(C(=O)NC(CN(C(=O)C(C)C2CC2)CC)C)cc2c(C)c(C)ccc2[nH]1 27725,c1(C(N(CCNC(=O)CC2CCCO2)CC)=O)ccc2c(=O)n(C)c(C)cc2n1 27726,C1(NC(c2cc(C)[nH]n2)=O)CCCC(N(C(=O)C(F)=CC2CC2)C)C1 27727,C1(NC(c2noc(CC)c2C)=O)CN(C(c2c(C)noc2N)=O)CC1S(C)(=O)=O 27728,C(=O)(C1CSc2ccccc21)N(C)CC1CCN(C(c2ccnn(C)c2=O)=O)C1 27729,Cc1cc(NC(C2CCCN(C(=O)CCCF)CC2)=O)cc(Cl)c1 27730,c1(C(=O)NCC2(F)CC(CNC(CCn3ccc(C)n3)=O)C2)cccc(=O)n1C 27731,N1(c2nc(=N)nc(N(C)Cc3ccccc3Cl)[nH]2)Cc2[nH][nH]c(=N)c2C1 27732,N1(C(c2c(CCNC(C(CN(C)C)O)=O)n[nH]c2)=O)CC(C2CCCCC2)C1 27733,C1(CNC(C(C(C)C)n2cnnc2)=O)CC2COCC2N1C(=O)Cc1nncs1 27734,c1(CCNC(C)=O)ccc(OC(C2CCCN(C(=O)C(C)=O)C2)=O)cc1 27735,c1(CC)c(C(=O)NC(C)CCNC(C2CCOC2)=O)nnn1CC 27736,C1(C(=O)NCc2cc(C(=O)NCC(C)C3CC3)no2)(CC)CCCCC1 27737,c12cc3n(n1)CC1(CCN(CC1)CC2=O)OC3.c1(CC(N)=O)nccc(O)n1 27738,C1(N(C(COC)=O)C)CCCN(C(C2CCCS2(=O)=O)=O)CC1 27739,c1(C(=O)NC2CN(C(C3(C)CC3(F)Cl)=O)C2)cccc(NC(N)=O)c1 27740,C1(CC(C)NC(c2cccnn2)=O)CCN(C(C2CNC(=O)C2)=O)CC1 27741,C(C)(C)(C(C)(C)O)NC(C1C(CNC(c2c(OC)scc2)=O)C1(C)C)=O 27742,C1(C(=O)NC2CC3CN(C(c4ccc(C)o4)=O)C2C3)CCn2nncc2C1 27743,C[Si](C)(C)CCCNC(=O)CNC(=O)CC1(O)CCOC1 27744,C1(C(=O)OCC)(NC(=O)NC2CC2(c2ccc(Br)cc2)C)CCOCC1 27745,N1(CC(=O)NC2CN(C(C(C)OCCC(C)C)=O)C(C)C2)CCc2ccccc21 27746,c1(C(c2ncc[nH]2)NCCC2(C)COC2)nnnn1CCN1CCOCC1 27747,C1(C(N(CC#C)CCOC)=O)(NC(=O)Cc2ccccn2)CC1(C)C 27748,N1(C(c2n(C(C)C)ccn2)=O)CCN(C(C2CC3CCCCC23)=O)C(CO)C1 27749,C1(CC(=O)NCCN2CC=CC2)CSCCN1C(=O)C(=O)Nc1ncc[nH]1 27750,c1(C(=O)NCCN(CCC)C(c2scnc2Cl)=O)cn(CC)nn1 27751,N1(C(C(CCC)(C)CCC)=O)CCC2(CC1)CC(NC(C1CC(C)C1)=O)CCO2 27752,C(=O)(C(CC=C)CC(C)C)NC(CC#C)CC(=O)NCC1(OC)CN(C)C1 27753,CC1(C)CC(CNC(=O)CC2CNC(=O)C2)N(C(=O)C=Cc2cccc(Cl)c2)C1 27754,C1(NC(C2=NOC(C)C2)=O)CC1C1CCCN(C(C23CC(C2)C3)=O)C1 27755,N1(C(C2(OC)CCSC2)=O)CC(C)CN(C(c2cccc(=O)n2O)=O)C(C)C1 27756,N1(C(=O)CCC2CCOC2)CC2CC1CN2C(C1C2(CC2)C12CC2)=O 27757,c1(C(N2CCC(N(C(C(CC=C)C)=O)C)C2)=O)c(C)ccc2ncccc12 27758,C1(CC(=O)NC(C2CCCCC2)CNC(CC2(C)CCCC2)=O)CCS(=O)(=O)C1 27759,c1(C(N2CC3CC(NC(c4c(O)cc(C)nn4)=O)C3C2)=O)ccc(C#N)nc1C 27760,C1(CC)CCC(C)CN1C(=O)C(C)C(C)NC(=O)C(CSC)OC 27761,N1(C(c2c(OC)c(F)ccc2)=O)CCC2CN(C(=O)CCCN(C)C)CC12 27762,c1(C(N(C)Cc2ncoc2C2CC2)=O)ccc(C(F)(F)F)c(Br)c1 27763,C1(C2CCN(C(=O)C(N)=O)CC2)(NC(c2c(N)cccc2[N+](=O)[O-])=O)CC1 27764,C(=O)(C1=C(Cl)CCC1)NC(C(=O)N(C)CCc1cccs1)CCF 27765,c1(OCC)cc(F)c(F)cc1C(=O)NC1CC(NCc2c(F)ccc(C)c2F)C1 27766,N1(C(C(C(=O)OC)OC)=O)CC(F)(F)CC1CCNC(C1CCCN1C(C)C)=O 27767,C#CC1CN(C(=O)CC2C(CC)C2(F)F)CCN1C(c1cc(Cl)cs1)=O 27768,C1(C(=O)NCC(CNC(C2(CC3CC3)CCC2)=O)O)CCNC1=O 27769,C(=O)(C(C)(C)C(C)O)NC.c12cccc(c1)-n1cc(nn1)C1CC21 27770,C(=O)(C(C(C)NC(c1cccn1C)=O)C(C)C)Nc1c(C)noc1 27771,c1(CNC(C2CNCCN2Cc2ccc(Br)c(Cl)n2)=O)ccc(O)c(O)c1O 27772,CN1C(=O)NC2(CCC(C(=O)N(c3ccncc3)C)CC2)C1=O 27773,C(=O)(C(CC)CC(F)(F)F)NCC(C1CC1)NC(c1c(C=C)cnn1C)=O 27774,c1(OC)ccc(C)nc1C(=O)NCC(C)(CO)NC(=O)C(C)C(C)(C)O 27775,c1(C(N2CC(CNC(C3C(CCC)C3)=O)(COC)C2)=O)nc(O)c(C)s1 27776,CC1CC(F)(F)CCN1C(=O)CC1CCC(NC(C2(C(N)=O)CCC2)=O)C1 27777,c1(NCc2c(C)cccn2)ncc(S(=O)(=O)NCC2CC2C)cc1Cl 27778,CC1(C)CC(=O)OC1CNC(C1CCCN1C(=O)C1=CCCSC1)=O 27779,Cc1nccc(C(=O)NCC(=O)Nc2c(C3CC3)cccc2F)c1N 27780,C1(C(=O)NCC2(O)CC2)(CNC(=O)CC2CC3CC3C2)CC12CCC2 27781,Cc1[nH]c2ccccc2c1CC(=O)NCC1(O)CCN(C(c2coc(O)n2)=O)C1 27782,c1(OC)c(F)cc(C(N2CCCN(C(=O)CCc3nc[nH]n3)CC2)=O)cc1F 27783,c1(COCC)nc(-c2cc(C3CCC3)on2)n(-c2cnc(C)s2)n1 27784,C1(CSCC(=O)NC(C)CC2CN(C(C3CC(F)C3)=O)C2)CCCCO1 27785,c1(C(N(CCOCCNC(C(C=CC)O)=O)C)=O)cc(OC)c(Br)s1 27786,C1(C(N(CC(C)O)CCNC(C2(OC)CCCC2)=O)=O)CCC12CCC2 27787,Cc1[nH]nc(CO)c1C(=O)NC(C(C1CCN(C(C2CC(C#N)C2)=O)C1)C)=O 27788,c1(CC)nn(C)c(CC(=O)NCCCC(C)NC(=O)C(C)C(F)(F)F)c1Cl 27789,Cc1cc(NC(=O)NCC2CCSC2(C)C)cc(C(F)(F)F)c1 27790,n1(CC)c(N2CCC(N3CCOC3=O)C2)nnc1CS(=O)(=O)Cc1ccccc1 27791,Cc1c(C(N2CCC(NC(c3cnoc3C3CC3)=O)C2)=O)oc2c(C)cccc12 27792,CON1CCC(C(=O)NC2CCC(C)N(C(=O)CCc3ccc(Cl)s3)C2)CC1 27793,CCCC(C)C(=O)NC1CC(C)(NC(=O)CCc2ccccn2)C1 27794,C1(O)(C(N(C)CC2(O)CN(C(CCc3cnc(C)o3)=O)C2)=O)CCCC(C)CC1 27795,c1(-n2cc(CC(C(=O)O)NC(C3(C4CCCO4)CCC3)=O)nn2)ccc(CO)cc1 27796,C1(C(=O)NCCCCNC(C(C(=O)OC)C)=O)CCc2nc(C)ncc2C1 27797,C(=O)(C(=O)C(C)(C)C)N1CC(C(N(C2CCC2O)C)=O)C(F)C1 27798,C1(O)(CN(C)C)CN(C(=O)CCNC(c2ccsn2)=O)C1 27799,C1(C(=O)NC2CCC(NC(C(OC)OC)=O)CC2)CC(F)(F)CCC1(C)C 27800,N1(C(C(COCC)C)=O)CC(CC(=O)NCCn2cc(C)cn2)CC1(C)C 27801,c1(C(N(C2CCN(C(C(COC)(C)OC)=O)C2)CCO)=O)cncc(F)c1Cl 27802,c1(C(N2CC(CC)N(C(=O)CCn3cc(Cl)cn3)CC2)=O)ccnc2ccsc12 27803,c1(C(N2CCCC(Cn3cc(C(C)(C)OC)nn3)C2)=O)cncc(F)c1C 27804,c1(C(=O)NCC23C(CN(C(CCC#N)=O)C2)C3)csc2ccccc12 27805,c1(CC(=O)NC2CN(C(C(C)(C)NC(=O)OC)=O)C2)ccc(Cl)nc1 27806,Cc1cc(Cl)c(C(=O)NCC(C2CC2)NC(=O)CC2COC(C)(C)CO2)cc1F 27807,Cc1cc(CC(=O)NC2CC2NC(C2CCN(C(=O)CCC3CCCC3)C2)=O)cs1 27808,C(=O)(C#CC1CC1)NC(CC)CN(C(C1CCCN(C(C)C)C1)=O)CC 27809,c1(OC)cnc(C(=O)NCCCN(C(C2(C)CCCCC2C)=O)C2CC2)c(Cl)c1 27810,c1(-c2cn(CC(CNC(c3ccc(CC)[nH]3)=O)OC)nn2)c(F)cccc1F 27811,C#CCCC(C(=O)NC1(C)CN(C(=O)OCC)C1)NC(=O)CC1OCCCO1 27812,C1(NC(c2cn(C(C)C)nc2)=O)C=CCC(C(N2CCCC(CN(C)C)C2)=O)C1 27813,c1(C(=O)NCC(CN(C(C(C)C(F)(F)F)=O)C)O)cccc2c1N(C)C(=O)CO2 27814,O=[N+]([O-])c1ccc(CS(=O)(=O)NC2CC2c2c(F)cccc2Cl)cc1 27815,CC(C)C#CC(=O)N(CC(C)NC(c1cnn(C)c1C1CC1)=O)C 27816,CC1(C)CN(C(=O)CCCNC(C2(C)CCC(=O)NC2)=O)CC1O 27817,C(CN=[N+]=[N-])(C(=O)N(C12CCC(CC1)CC2)C)NC(CC=C)=O 27818,OC1CCCCC(c2cn(CCCCF)nn2)CCNC1 27819,N1(C(c2cn(CC)nc2)=O)CCCCC1C(C)ONC(C1CS(=O)(=O)C1)=O 27820,C1(C2CCN(c3ncnc4c3COC4)CC2)(NC(c2cccc(F)c2Cl)=O)CC1 27821,N1(C(COCC#C)=O)CCCC1CN(C(C1(C#C)CC1)=O)C1CC1 27822,CC1CCC(C)(C(N2CC3CC2(C(=O)NCC(O)CN(C)C)C3)=O)CC1 27823,c1(C(N(CCC)CCNC(C2CCOC(C)C2)=O)=O)cncc(OC)c1C 27824,CC1(C)C(C(=O)NCC(C)(F)CNC(=O)CCNC(=O)CO)CC1(F)F 27825,CC1=NC(C)(CNC(c2coc(C(C)NC(c3cnc(C)o3)=O)n2)=O)CS1 27826,C(=O)(CC(C(F)(F)F)NC(c1cccn1C1CC1)=O)NC1C(OC)CCOC1 27827,C(=O)(C(CC(=O)OC)N(C)C)NC(C(C)NC(C=CC=CCC)=O)(C)C.C1CC1 27828,c1(OC)cc(F)cnc1NC(=O)NC(c1cccc(C(F)(F)F)n1)C 27829,C1(NC(c2c(CC)c[nH]c2)=O)CN(C(=O)C(c2cnn(C)c2)O)CCC12CCC2 27830,C1(C(=O)NC2CC3CN(C(CP(C)(C)=O)=O)C(C2)C3)CCC(S(N)(=O)=O)CC1 27831,n1(CCC(N2CC(O)(CNC(C3CC(=O)NC3)=O)C2)=O)cccnc1=O 27832,CCC(C)C(C(=O)N(C1CC2CCC1O2)C)NC(C1C2CCC(C2)C1C)=O 27833,c1(SC)ncc(C#N)c(N2CCN(c3nc(C)cc(C)n3)CC2C)n1 27834,c1(C(N2CCCN(C(C=CCCC)=O)CC2CO)=O)cccc2c1OCC2C 27835,N1(C(c2n(CC)ncn2)=O)CCCN(C(c2cc(C#N)oc2C)=O)CC1CO 27836,c1(C(=O)NCC2CCCC(NC(CC(=O)NC)=O)C2)cc(N)ccc1Br 27837,C(F)(C(=O)NN1CCCC1C(=O)NC(C1CCCOC1)(C)C)=C(C)C 27838,CCC(C)CCCCC(=O)N1CCC(NC(C2(CO)CCC2)=O)CC1 27839,S(=O)(=O)(c1ccc(CN2CCCCC2)cc1)NC1CCC(OC)C1 27840,N1(CC)CCC1C(=O)NC1(CC(=O)NC2(c3cc[nH]n3)CC2)CC1 27841,c1(C(N(C)CC2N(C(C(C)=C3CCCC3)=O)CCC2)=O)cn2c(n1)C(C)CCC2 27842,C1(NC(C2CC2c2ccncc2Cl)=O)CCCN(C(C2(F)CC=CC2)=O)CC1 27843,C=CCC(C)C(=O)NCC(=C)CCNC(C1CN(C)CC1c1cccnc1)=O 27844,C1(C(=O)NCC2(NC(c3ccc(CC)o3)=O)CCCC2)CCOC1(C)C 27845,c1(OC)ccc2c(c1)CCN2C(C1CCCC(c2nn[nH]n2)C1)=O 27846,C(CNC(=O)C(C)N1CCCC1)(CCNC(c1cnc(C)s1)=O)OC 27847,Cc1nc2c([nH]1)CC(C(N1CC3(CC(NC(c4nnn(C)c4N)=O)C3)C1)=O)CC2 27848,Nc1cc(O)c([N+](=O)[O-])cc1C(N1CCC2(CC1)CC2NC(=O)C=CC(N)=O)=O 27849,CCS(=O)(=O)CC(=O)N1CC(C(N2C3CCCC2CC3)=O)CC1(C)C 27850,c1(C(=O)NCCOCCN(C(=O)Cc2ccoc2)C)c(Cl)ccc(F)c1N 27851,C1(C(N2CCC(O)(CNC(Cc3cnc(C)o3)=O)C2)=O)CC(C)(C)CN1C 27852,Cc1ccc(N(C(c2ccc(C(c3cc(Br)ccn3)=O)cc2)=O)CC2CC2)cc1 27853,C1(NCc2cn(C3(C(=O)OC)CC3)nn2)C2CN(C(c3cncc(Cl)n3)=O)CC12 27854,CCC(CC(=O)N1C2CCC1CC(CNC(=O)CCCS(N)(=O)=O)C2)C(C)C 27855,N1(C(c2nc(C(C)OC)sc2)=O)CC2(CC(NC(c3cc(C)sc3C)=O)C2)C1 27856,N1(C(C(CC)(C)C)=O)CCC2(CC1)CC2NC(c1ccsc1COC)=O 27857,CC(CS(C)=O)C(=O)NCCCCN1CCCN(C(=O)CCN(C)CCO)CC1 27858,c1(C(=O)NC2CC(CC(=O)N(CCCCCC)CC)C2)cccc(C)c1N 27859,C1(C)(C(N(C2CCN(CC)C2)CC)=O)CCCN1C(=O)CCN1CCCCC1C 27860,N1(C(c2ccc(CNC(C(CCC=C)(C)C)=O)cn2)=O)CCc2c(O)noc2C1 27861,Cc1ccc(O)cc1C(=O)NC(CNC(=O)CSc1ccccc1O)CO 27862,C(CC(C)(C)C(=O)NC(C1CN(C(C2CCC(C)CC2)=O)C1)C)SC 27863,C(C(=O)NCCc1c[nH]nc1O)(C(C)(C)O)NC(c1c(CC)n(C)cc1)=O 27864,C1(C(N(c2c(C)csc2)C)=O)CC12CC2(F)F 27865,C1(OC)CC(CNC(c2ncc(F)cn2)=O)N(C(c2cnc(C(C)(C)C)o2)=O)C1 27866,C1(NC(=O)CCCCN2CCCC2)CC2CCC1N(C(=O)Cc1ccccc1)C2 27867,C1(C(=O)NC(C)C2CC2)CC12CCN(Cc1noc(C(F)(F)F)n1)CC2 27868,N1(C(C(CC)(C)OC)=O)Cc2cccc(CNC(c3ccn(C4CC4)n3)=O)c2C1 27869,C(CC(C)C(=O)N(CC(C)NC(=O)C(c1cnn(C)c1)=O)CC)=CCC 27870,Cc1nc(Cc2ccc(F)cc2)oc1C(=O)NCCC(C)N(C)C(C1CSC1)=O 27871,S(=O)(=O)(c1ccc(OC)c(-c2ccc(C=CC(=O)O)cc2)c1OC)N(CC)CC 27872,N1(C(c2ccn(CC)n2)=O)CCC(C)C(NC(=O)CCc2ccon2)C1 27873,C1(N(C(CCOCCC)=O)C)CN(C(=O)Cn2c(C)c(C)sc2=O)CC1(C)C 27874,C1(C(N2CC(C(C(=O)NC(C3C(C(=O)OC)C3)C)O)C2)=O)CCNC(=O)C1 27875,C1(NC(c2cc(CC)n(C)n2)=O)CN(C(C23CC(CO2)C3)=O)CC(C)(C)C1 27876,c1(CC)ccc(S(C)(=O)=O)cc1C(=O)NC1C2CC3CN(C(=O)C4CC4)C1C3C2 27877,c1(OCC(=O)NC(C2CCCN2C(=O)COc2ccon2)C)cc(F)cc(F)c1 27878,C1(OC)(NC2CCC(n3cc(CCC(C)(C)CO)nn3)CC2)CC(C)(C)C1 27879,c1(CNC(c2cccc(CN3CCCC3=O)c2)=O)ccc2c(c1F)OCCO2 27880,c1(N2CCC(CCCCCSC)CC2)ncnc2scc(Br)c12.C1(N)CC1.NC 27881,N1(CCC(=O)NCC#C)CCC2(CCCCC2)CC1 27882,C(=O)(CCCCN1CCCC1)N(C1CN(C(c2cncc(O)c2)=O)C1)C 27883,c1(C(N(C2CN(C(c3cccn3C)=O)CC2F)C)=O)ccc2cc(F)ccc2n1 27884,N1(C(C2C(CC)OCC2)=O)CC2(CC(C(=O)NC(C(=O)NC)C3CC3)C2)C1 27885,C1(C(=O)OC)(CO)CCCN1C(=O)CCCC1CCOCC1 27886,c1(NCC2CCC(NC(c3c(CCC)nco3)=O)C2)ncccc1C#N 27887,C1(C(=O)NCC(CC)NC(CSCC=C)=O)CC2(C1)CC1(CCC1)C2 27888,Cc1nsc(C(N2CC(C)CC2C(=O)NC2CCC(CO)CC2)=O)c1N 27889,c1(C(=O)NCCC2(OC)CN(C(C3CCCC3C)=O)C2)c(C)nn(C(C)C)c1C 27890,C1(NC(C2CCCCC2O)=O)CCN(C(c2ncc(Cl)cc2F)=O)C12CC2 27891,C1(NC(CCc2cnc(C)s2)=O)CCN(CCC2CCOC2)CC1(C)C 27892,c1(C(=O)NC2(C)CCN(C(C(c3cnn(C)c3)C)=O)C2)ccc(N)c(Cl)n1 27893,C1(F)(CNC(c2c(CCC)nco2)=O)CCC(NC(=O)C=Cc2cscn2)C1 27894,C1(O)(CNC(C2(OC)CC(C)C2)=O)CCCN(C(c2cnc(C3CC3)s2)=O)C1 27895,c1(C(=O)NCC(CNC(c2[nH]nnc2-c2ccnn2C)=O)OC)cocc1C 27896,c1(SCC)nccnc1C(N1CC(OC)CC1CCNC(c1ncoc1C)=O)=O 27897,O=C1CCc2cc(C(=O)NCCCOCCNC(=O)CC3CC3)c(F)cc2N1 27898,c1(OC)ccnc(C(=O)NC2CC(C(N)=O)(N(C)C)C2)c1C 27899,C(C(=O)N1CC(N2CCOC2=O)C1)(C(C)(C)C)NC(c1c(C)ccnc1)=O 27900,C1(CC(=O)NCC(CC(C)C)(C)NC(=O)CCF)C2CC3CC(C2)CC1C3 27901,N1(Cc2c(C#N)c(F)ccc2)CCC2(CC1)CCN2C(c1cc[n+]([O-])cc1)=O 27902,c1(CCC)[nH]nc(C(=O)NCC2CCN(C(C3CC3C)=O)C2(C)C)c1[N+](=O)[O-] 27903,N1(C(C2=CC(C)(C)C2)=O)CC2CCC(C(=O)NCC(c3ccsc3)O)(C2)C1 27904,C=CCCCC(=O)NCCCC1CN(C(=O)CCSCC(C)C)CCO1 27905,N#Cc1cc(CNC(C2CC2NC(c2ccncc2Cl)=O)=O)cc(F)c1 27906,N1(C(C2(C#C)CN(C(c3cn(CC)cn3)=O)C2)=O)CCOC(CC)CC1 27907,O=C(CC(F)(F)F)NC(C1CCOC1)CNC(c1csc(C2CCCCC2)c1)=O 27908,N1(CCN2CCC(CC(=O)NC3(CC)CCCCC3)C2)CCC(F)(F)CC1 27909,C1(NC(CCC)=O)CCCC(NC(=O)C(C)Sc2ccc(Cl)cc2)C1 27910,C1(C(=O)NCC(CN(C(C(C)S(C)(=O)=O)=O)C)(C)C)CN(C)CCN(C)C1 27911,N1(C(C2CCC(CCCCC)O2)=O)CCN(C(c2ccc(C)cc2)=O)C(C)C1 27912,C1(NC(c2c[nH]nc2Br)=O)COC2CN(C(=O)CC3CCCNC3=O)CC12 27913,C1(CNC(C2(CC)CC(C)(C)C2)=O)CCN(C(=O)CCOCC(F)F)C12CC2 27914,Cc1ccc(F)c(C(=O)NCC2CC(C(=O)NCC(c3cnn(C)c3)C)=NO2)n1 27915,C1(C(=O)NC2C(CNC(c3cnn(CC)c3C)=O)CCC2)CC12CCCCCC2 27916,N1(C(C2CCCC2O)C(=O)NCCNC(=O)OC)CC(N(C)C)Cc2ccccc21 27917,N#Cc1ccc(CC(=O)NC2CCN(C(=O)CSc3nncs3)CC2F)cc1 27918,c1(C(CNS(C)(=O)=O)OC(=O)C#CC2(C)COC2)nc2ccccc2[nH]c1=O 27919,CC1(C)CCN(CC(=O)NCC(C)(O)CNC(c2cc(C#N)c[nH]2)=O)C1 27920,Cc1ccc(C(F)CC(CC(=O)NC(C)C(C)C)c2ccccc2)cc1C 27921,C1(CCC(=O)NC2(CNC(c3cc(C(C)=O)sc3)=O)CC2)CCCCN1C 27922,C1(NC(CCc2c(C)ncs2)=O)C2CC(NC(C3(C)CCCC3C)=O)CC12 27923,Oc1nc(C2CCC2)oc1-c1nc(-c2cscn2)nn1C1CCCCC1 27924,N1(C(CN(C(C2CCN(CC)C2)=O)C)=O)CCN(C(c2sccc2OC)=O)CC1 27925,C#CCCCCC(=O)NCCC12CC1CN(C(c1ccc(C)cc1)=O)C2 27926,c1(C(C)C)ccc(C(=O)NC2CCCN(C(=O)C#CC3CC3)C2C)c(F)c1 27927,CC(C)(C)C(C#N)C(=O)N1CCC(O)(CNC(c2cccc3nc[nH]c23)=O)CC1 27928,C1(C)(COC)CC(NC(c2n[nH]c3c2COC3)=O)CN1C(c1cc(Cl)cn1C)=O 27929,C(=O)(C(C(C)(C)O)NC(c1nonc1N)=O)NC(c1nnc(C)s1)C 27930,C1(NC(C2N(C(=O)OCC)CCC2)=O)CC2CCC(C1)N2C(=O)C(=O)NC1CC1 27931,c1(C(N2CCC(C(C)(C)NC(C3OCCCO3)=O)C2)=O)cn2c(n1)CCC2 27932,c1(CC)cc(C(=O)NCC2(COC)CCCN2C(c2ccoc2Br)=O)cc(Cl)n1 27933,c1(C(N(CC(C)O)CCNC(c2cccc[n+]2[O-])=O)=O)cnc2ncccc2c1 27934,C(=O)(C1CCc2snnc21)N1C2CN(C(CN(S(C)(=O)=O)C)=O)CC1CC2 27935,O=C1CCCC(C(=O)NCCCCNC(C2(c3ccncc3)CC2)=O)O1 27936,Cc1ccc(C(=O)NC(C)CCC(=O)N(C(C)CO)C2CC2)c(O)c1 27937,CCCCCCNC(=O)C(Cc1cnc[nH]1)NC(=O)CSc1cn[nH]c1 27938,c1(C(N2CCC(C3CCCN3C(=O)CSC(F)F)C2)=O)ccc2ncnn2n1 27939,N1(C(c2c(OCC)nccc2)=O)C2CCC1CN(C(c1noc(C)c1C)=O)C2 27940,Cc1cnc(Cl)c(C(N2CCC(CC(C)NC(c3ccc(F)nc3)=O)CC2)=O)c1 27941,c1(C(=O)NCC2OCCN(C(CS(CC)(=O)=O)=O)C2)ccc(OC)c([N+](=O)[O-])c1 27942,C(N=c1[nH]c(C)c(C(=O)NC(CCO)C(C)C)s1)c1c(F)ccc(OC)c1 27943,Cc1cc(NC(=O)C(=O)N(C)Cc2ccnc(Cl)c2)cnc1C 27944,c1(C(N2CCC(Cn3cc(C(CC)O)nn3)C2)=O)csc(C)c1Br 27945,Cc1cc(C(F)F)oc1C(=O)NC(C)CC(C)NC(c1ccncn1)=O 27946,Cc1ccc(C(=O)NCC2CN(C(c3nncn3C)=O)CC2C)c2ccccc12 27947,c1(C(C)=O)ccc(OCC(N2CCC(C)C2CNC(c2ccon2)=O)=O)cc1 27948,N1(C(CCn2ncn(C)c2=O)=O)CC2CC(NC(c3cnccc3Cl)=O)C2C1 27949,C1(NC(CCC=CC)=O)CC2CC(NC(c3cc(OC)cnc3F)=O)CC2C1 27950,N1(C(C(C2CCCC2)SC)=O)CC(F)(C(=O)NOCCOc2ccncc2)C1 27951,c1(C(N2CC(COC)(CNC(=O)C(C)(Cl)Cl)C2)=O)ccnc(S(N)(=O)=O)c1 27952,C12(CNC(c3c(CC)cccc3)=O)CN(C(=O)CN=S(C)(C)=O)CC1CCO2 27953,CC1CN(C(C2C3CC4C(C3=O)C24)=O)CCC1C(=O)N(CC(O)CF)C 27954,N1(C(C(C(C)C)C2CCC2)=O)CCC2(C=C(C(=O)NC34CCN(CC3)C4)C2)C1 27955,C1(CN(CCC(CC)C)CCOC)COc2ccccc2O1 27956,c1(N(C)C)cccc(NC2(CO)CCN(C(=O)C(C)(CC)OC)CC2)c1[N+](=O)[O-] 27957,Cc1ccc(-c2cn(CC(C)NC(c3nccn3-c3ccccc3)=O)nn2)cn1 27958,C1(NC(c2ccc(C#C)o2)=O)CCN(C(=O)C(C)(C)c2ccnn2C)CC1C 27959,N1(C(C(CSC)(C)C)=O)CCOC2(C1)CN(C(=O)CCc1cccnc1)C2 27960,C1(C(=O)NCCc2cn(CC(=O)O)nn2)COc2ccc(F)cc2C1 27961,Cc1nnc(N(CCCNC(c2nc(Cl)sc2Cl)=O)C2CC2)nc1C 27962,N1(C(CCCC(C)=O)=O)CCC2OCCN(C(c3ccsc3Cl)=O)C2C1 27963,C1(C=O)CN(C(c2c(C)nc(-c3ccccc3)s2)=O)CC(F)(F)C1.C(C)C1CC1 27964,N1(C(C(=O)NCc2cc(OC)c(C)cc2)=O)CC2CCC(C1)C(=O)N2 27965,c1(C(N(C2CCS(=O)(=O)C2)CCCNCC)=O)c(-n2cccn2)cccc1F 27966,c1(C(N2C(CCNC(c3scc(C)c3)=O)CCC2)=O)ccc(C#N)c(C)c1 27967,C1(NC(CCC2CCCN(C(CSC)=O)C2)=O)CCOC(C)(C)C1 27968,c1(CC(=O)NCCCCCCN(C(CCC(=C)C)=O)C)ccc(S(C)=O)cc1 27969,C1(C(N(C(CO)C2CC2)C)=O)CCCCC1CNC(=O)Cc1c[nH]nc1C 27970,N1(CC(=O)NC(CC)C)CC2C(C(=O)NCC(C3CC3)ON3CCOCC3)C2C1 27971,N1(C(C(C)N(C)C)=O)CCC(C(=O)NCCc2cc(C3CCCN3)no2)C1 27972,C1(Cc2cn(CCN(C(CCOC)=O)C)nn2)(CO)CCOCC1 27973,N1(C(c2ccc(CC)nc2C)=O)CC(C)N(C(C2CC2(Cl)Cl)=O)CC1C 27974,C1(CNC(C(CC)CC)=O)CN(C(=O)C(C)(C)n2ccc(C)n2)CCCO1 27975,Cc1oc([N+](=O)[O-])cc1C(N1CCC(O)(CNC(=O)C(F)C2CC2)C1)=O 27976,c1(C(=O)N(CC(CO)NC(C2CC2C(F)F)=O)C2CC2)ccc2ccccc2n1 27977,Cc1occc1C(=O)NC1CCC1C(=O)NCCNC(=O)N(C)C 27978,N1(C(C(CCC)O)=O)CC(NC(c2cncc(C)n2)=O)CC12CCCCC2 27979,CC(C)(CCC(=O)NC1CCCC(F)(F)C1)NC(=O)Cc1ccsc1 27980,CC1CCN(C(=O)CCSC2CCCC2)C(C(=O)NC2CC3CC4C(C3)C24)C1 27981,C1(C(=O)NC2CCC(CCNC(C3(C#N)CC3)=O)C2)CCS(=O)(=O)CC1 27982,c1(C(N(CCC(C)NC(C2CCCC2(C)C)=O)C)=O)cnc(N)c(Br)c1 27983,O=C(C(O)C(F)(F)F)N1CCN(C2CN(C(C3(Cl)CC3(F)F)=O)C2)CC1 27984,N1(C(C(CCC)OC)=O)CCCC(F)(C(=O)NC2CC2CC(C)(C)C)C1 27985,C(=O)(C(CCSC)NC(c1cnn(C(C)C)c1)=O)N(CC(C)C#N)CC 27986,C1(CC#C)(C(=O)NCc2ccc(Cl)cn2)CCN(C(=O)CCSC)C1 27987,c1(C(C)=O)cccc(C(=O)NCC(F)CNC(C2(c3ccc(F)cc3)CC2)=O)c1 27988,c1(SC)nc2ncnc(NCC3(F)CCN(C(=O)C(C)C4CCCO4)CC3)c2s1 27989,C1(NC(COCCOCCOC)=O)CC(CO)CCN1C(=O)CC(C)F.C(C)(C)(C)O 27990,c1(OC)ccc(OC)c(C=CC(=O)NC2CC(NC(c3c(F)cccc3F)=O)C2)c1 27991,Cc1ccc(C(=O)NC2CCOCC2NC(=O)CCc2ccoc2)cc1N 27992,C1(C(=O)NC(CCOC)C(C)C)CCCCC1(C)NC(c1c[nH]c(=N)c(C)c1)=O 27993,c1(NC2CC(OCC)C2)ccc2c(c1)CN(C1CCC(=O)NC1=O)C2=O 27994,N1(CCC)CCN(C(C2CC(OC)CN2C(=O)Cn2cccn2)=O)CC1 27995,C1(CC2CN(C(C(=O)NCC(C3CCCS3(=O)=O)(C)C)=O)C2)CC2COCC2C1 27996,CCCS(=O)(=O)C(C)C(=O)N(C(C)CCNC(c1cc2sccc2n1C)=O)C 27997,N(C1CCc2c(Br)cccc21)c1cc(NC(CC(C)(C)OC)C)nc(C(C)C)n1 27998,c1(NC(=O)NC(CC)C)ccc(NCC(F)(F)C(C)C)c(C)c1 27999,c1(C(=O)NC(CN(C(CC(=C)C)=O)CC)CC)cc(OC)c(OC(C)C)c(Cl)c1 28000,c1(C(c2nnnn2CC(F)F)NCCC(C)CO)ccc(Cl)c(F)c1 28001,N1(C(c2c(CC)sc(=N)[nH]2)=O)CCCOC(CNC(=O)C2=C(Cl)CC2)C1 28002,CN1C(CN=C(NCC2CCCSC2)NC2CC2)CCS1(=O)=O 28003,c1(OCC(N2C(CNC(=O)C3=COCC3)CCC2)=O)ccc(F)cc1Cl 28004,N1(C(CN(C)Cc2ccccc2)=O)CC(CNC(c2cc[nH]n2)=O)C(O)C1 28005,CN1c2ccc(C(=O)NCCCNC(c3coc(Cl)c3)=O)cc2C(C)(C)S1(=O)=O 28006,C1(NC(C2CCC2C(F)F)=O)CCN(C(=O)CCc2cnc[nH]2)C1C1CC1 28007,N1(C(CSCC(N)=O)=O)CC2(CCC2NC(=O)C=CCF)C1 28008,c1(CC(C(=O)OC)NC(c2ncc(C)cn2)C)ccc(OC)cc1Cl 28009,c1(CNC(CN(CCOC)C(C2CC2c2ccoc2)=O)=O)cc(C)cc(C#N)c1 28010,CN=c1[nH]cc(C(=O)NC2CCN(C(=O)C(C)n3ccnc3)C2C)s1 28011,c1(C(=O)NCC(CN(C(C2(COC)CC2)=O)C)(C)C)[nH]c(C)c([N+](=O)[O-])c1C 28012,N1(C(CC2(C=C)CCCCC2)=O)CC2(C1)CN(C(=O)C(C)NC(=O)NC)CCO2 28013,c1(CCCC)ccc(CC(=O)NC(CNC(=O)CCCCOCC)C2CC2)cc1 28014,c1(C(C)NC(C2C(C#N)C2(C)C)=O)ccc2nc(O)[nH]c2c1 28015,C(=O)(CC1=CCN(C)CC1)NCC(C#C)OC.O1NC(=O)C2CC2C1C 28016,c1(C(N2CCN(C(CSCCCC)=O)CC2C(C)C)=O)cccc2cncn12 28017,CC1CCCCC1CN(c1ccccc1)C(C1CCCCC1)=O.C1(=O)CN1 28018,N1(C(c2nc(OC)oc2)=O)CCC2(CCN(C(=O)Cn3cc(CO)nn3)C2)C1 28019,C1(CNC(c2c(CC)n(C3CCCC3)nc2)=O)CC2(CC2)CN1C(C1CC1C)=O 28020,N1(C(c2c(O)ccc(C#N)c2)=O)CCC2(CCCC2NC(=O)CC(F)(F)F)CC1 28021,c1(CC)cc(C(c2nnnn2C)NCC(C)F)on1.N1(Cc2cccs2)CCOCC1 28022,c1(OC)ccc(C)nc1C(N1CC(OC)C(NC(=O)COc2cc(C)on2)C1)=O 28023,C(=O)(C(C(C)(C)C)n1ccnn1)N(CC(CC)NC(c1csc(=NC)[nH]1)=O)C 28024,Cc1[nH]nc2c1CCC(C(=O)NC1CCCN(S(=O)(=O)c3ccc(Br)cc3)C1)C2 28025,C1(O)(C(CNC(C=C(CC)C)=O)C)CCN(C(=O)Cc2ccccc2SC)C1 28026,c1(NC(=O)C(N2CCN(c3ccnnc3)CC2)=O)ccccc1-n1ccnn1 28027,C1(OC)CC(C(=O)NCC2CN(C(c3cnn(C)n3)=O)C2)C12CCC2 28028,c1(C(=O)NC2CC(NC(c3n(C)ccc3)=O)C23CCC3)cc(N=S(C)(C)=O)ccn1 28029,N1(c2cc(C#N)ncn2)CCCC2C1CCN2C(c1ccc2c(c1)CC(=O)N2)=O 28030,C1(OC)CN(C(=O)Cc2nccn2C)CC1NC(C1CCOCC1)=O 28031,CCCCS(=O)(=O)C(N(CC(CC)NC(CC(=O)C(=Cc1cccnc1)C)=O)C)=O 28032,C(=O)(CC1=CCCCC1)N1CC(NC(c2cc(N)c(Cl)nc2)=O)C(C(F)(F)F)C1 28033,c1(OC)ccc(C(=O)NCC2CC(O)CN2C(=O)C(F)=CCCF)nc1OC 28034,S(=O)(=O)(c1[nH]c(=NCCCCCN(C)C)ccc1Br)N1C(C)c2cccn2CC1 28035,Cc1cn2ccc(C(=O)NC(C3CN(C(c4cnns4)=O)C3)C)cc2n1 28036,N1(C(C(C)(C)N2CCCCC2)=O)CCOCC(C(=O)NCc2conc2Br)C1 28037,Cc1ccc(NC(c2nnnn2C(C)C)(C)CC2CCCOC2)cc1C 28038,C=CC1CN(C(=O)CCN(C(=O)CCCCCC)CC)CCO1 28039,CCC(C)(C)CCCC(=O)N1CC(NC(=O)COc2ccccc2)CC1(C)CC 28040,Cc1cc(Br)oc1C(=O)NCC1COC(CNC(=O)C=Cc2cocn2)C1 28041,C1(C2CCN(CC)C2)CCCCCN1Cc1cc(C(=O)O)c(C(F)F)o1 28042,c1(C(=O)NCC(CNC(c2c(N)nc(Cl)cc2)=O)CO)ccc2nonc2c1 28043,CCC(C)C(O)C(C)C(=O)NC1CCCC1CC(=O)NC12CCCN(CC1)C2 28044,C1(C(N(C)CC2CN(C(c3cn(C4CC4)nn3)=O)CCO2)=O)CCC=CCCC1 28045,C1(CCC(=O)NCC(CC)(C)NC(c2cc(Cl)ccn2)=O)NC(=O)NC1=O 28046,CC1CN(C(=O)C2=CCSC2)CC2(CCN(c3nnc(C(N)=O)s3)C2)O1 28047,C(CN=c1nn[nH]n1-c1ccccc1)N(C(=O)CC1CCC(C(F)(F)F)O1)C 28048,C1(C(=O)NCC2CCN(C(CCC(C)C)=O)CC2)COC(C)(C)CO1 28049,N1(C(CCC(CC)CC)=O)CC(C2CCCCN(C(C3CCSC3)=O)C2)C1 28050,c1(CN2CCC(C(=O)NC3CCS(=O)(=O)C3)C(O)C2)cc2ncccc2[nH]1 28051,C12(NC(COC3(C)CCC3)=O)CC(CNC(c3ccc(=O)oc3)=O)(C1)OC2(C)C 28052,C12(CNC(c3[nH]c(CC)c(Cl)n3)=O)CCC(C1)N(C(C1CCC(OC)CC1)=O)C2 28053,C1(NC(c2c(NC(C)=O)cccc2)=O)CCN(Cc2ccc(O)c(O)c2)CC1F 28054,N1(C(c2c(CC)noc2)=O)CCC(C(=O)NCCN(C2CC2)CC)C(C)C1 28055,C12(C(N(C(CN(C(CNC(CCC)=O)=O)C)C)C)=O)CC1COC2(C)C 28056,C1(NC(CN2CCN(C(C3(SC)CC3)=O)CC2)=O)CCC(F)(F)C1O 28057,C1(CN(C(C2OCCOC2C)=O)CC)CCCN(C(c2ccnc(O)c2)=O)C1 28058,C(C(C)(C(=O)Nc1conc1C)NC(c1ccc(C#N)o1)=O)SC 28059,C(C[Si](C)(C)C)NC(CN(CC#C)C(c1cc(Cl)cs1)=O)=O 28060,C(CC(N)=O)(C(=O)N1CC(C(=O)NC2CC2)C1)NC(c1nccc(CC)c1)=O 28061,c1(C(=O)NCC2CN(C(CCSCC)=O)CC2O)cc(CC)cnc1O 28062,C1(NC(CCOCCOCC)=O)CN(C(=O)C(C)CF)CC1F 28063,N1(C(CCC(=O)N(C)C)=O)CCC(C2CCN(C(c3ccc(F)cc3Cl)=O)C2)C1 28064,c1(CCC(=O)NC2C(NC(Cc3c(C)scc3)=O)COC2)cccc(N(C)C)c1 28065,c1(C(N(c2n(CC)nc(C)c2)C2CC3CNC2C3)=O)cc(F)ncc1NC(C)=O 28066,N1(C(CC)=O)CCC(C(=O)NCC(CC)NC(=O)CC(O)c2ccccc2)C1 28067,c1(NC(C2(C)N(C(c3cncc(OC)c3)=O)CC2)=O)ccc2ncc(Br)cc2c1 28068,N1(C(C(C2CC(F)(F)C2)OC)=O)CCC(NC(c2ccns2)=O)CC1C 28069,N1(C(c2cc(CC)on2)=O)CCN(C(c2c[nH]c(=NC)o2)=O)C(C2CC2)C1 28070,C1(C(N2CCC(C3(C)N=N3)CC2)=O)CN(C(c2ccccc2Cl)=O)CC1(F)F 28071,CCCCCCC(C)(c1nnnn1C(C)(C)CC)NCC(=C1CCSCC1)F 28072,C=CC(C)(O)CC(=O)NC1CCCCN(C(c2nc(OC)cc(OCC)n2)=O)C1 28073,c1(NCC2CN(C(C3C(OC)CCC3)=O)C(C)C2)nnc(C)c(C)c1C#N 28074,C=C(C)C(C)(C)C(=O)NCCNC(c1ccnc(C(C)(C)O)c1)=O 28075,N1(C(c2cccc(C)c2F)=O)CCC2(C1)CN(C(=O)C#CC1(C(F)F)CC1)CCO2 28076,c1(CNC(NCc2ccc(C#N)nc2)=NCCCF)ccc2c(c1)OCCCO2 28077,N1(C(CCCCCNC(Cc2c(C)n(C)cn2)=O)=O)Cc2cccc(F)c2C1 28078,N12CC3CCCC(C3)(C1)C(=O)NCC2=O.N=c1[nH]c(CSCC2CCCO2)cs1 28079,N1(C(C=C(C)C(F)F)=O)CCC(F)(C(N2CCCC2C2(C)CC2)=O)CC1 28080,C#CCCCC(C(=O)Nc1ccc2c(c1)CCC2)N(C1CCCS(=O)(=O)C1)C 28081,c1(-c2onc(C(C3CCS(=O)(=O)CC3)C)n2)ccnc2c(I)cnn12 28082,Cc1c(C(=O)NCC2CCN(C(=O)C(F)=CCCF)C2)cnn1CC1CCCC1 28083,c1(OC)c(C(N2CC(C3CCCN(CCN(C)CCO)C3)C2)=O)cccc1Cl 28084,CC1CN(C(c2cnn3c2SCC3)=O)CC(C)N(C(c2cncs2)=O)C1 28085,C(=O)(C(F)C(C)CNC(c1ccc(C)o1)=O)N(C(CC)C(=O)OC)C 28086,N1(C(C2(C)C(C)C2)=O)CCC2(CC1)CN(C(c1c(F)cncc1F)=O)CCC2O 28087,c1(C(=O)NC(C(C(C)C)NC(Cc2c(C)ocn2)=O)C)ccsc1S(C)(=O)=O 28088,N1(c2c(C#N)cnc(C)n2)Cc2ccc(NC(=O)C(c3ccccc3)O)cc2C1 28089,Cc1ccc(N)c(C)c1C(=O)N(CC(O)CN(C(=O)CC(C)C1CC1)C)C 28090,CCC(CC(=O)N(CC(C)C(=O)NC(C)CC1CC1)C)CC(C)C 28091,C1(NC(C=C2CCN(C(C3(COC)COC3)=O)CC2)=O)CC(=O)N(C)C1=O 28092,C1(CNC(C(CCCC)C)(C)c2nnnn2CC(F)F)Cc2ccccc2CO1 28093,c1(C(=O)NC(c2cc(F)cc(Cl)c2)CNC(C2CC(O)C2)=O)n[nH]cc1[N+](=O)[O-] 28094,N1(C(c2c(C)ncc(N)c2)=O)CC(NC(C2(C)CCCCC2)=O)CC(C)(C)C1 28095,CON1CC(C(=O)NCCC2CC(NC(=O)C=Cc3ccoc3)C2)CC1=O 28096,C(=O)(C1=CC2C=CC1C2)N1CCCC(C(=O)Nc2c(C(C)C)nccc2)CC1 28097,C12(CNC(CC=CC=C)=O)CCCCC1CN(C(c1ccc(CO)c(Cl)c1)=O)C2 28098,C1(N(C(c2c(C(C)NC(CCC=C)=O)noc2)=O)C)COC(C)(C)C1 28099,C#Cc1cccc(CNC(C2(CCNC(=O)C(c3cnccn3)C)CCC2)=O)c1 28100,N1(C(c2cnco2)=O)CC2CCN(C(c3ccc(-n4cnnn4)cc3)=O)C(C2)C1 28101,CC1(C)CC1(C#N)C(N1CC2C(NC(=O)Cc3cn[nH]c3)C2C1)=O 28102,c1(C(=O)NCC2C(C)CN(C(c3nnc(C(C)(C)C)s3)=O)C2)cc(C#N)cn1C 28103,c1(C(=O)NC2C(C)(C)CCN(C(C3(C)COC3)=O)C2)cc2nn[nH]c2cc1F 28104,C(=O)(C1=CCCC(C)(C)C1)N(C1CCN(C(C2(S(C)(=O)=O)CCCC2)=O)C1)C 28105,CC(C)(C)C(CNC(C1CCC(F)(F)C1)=O)NC(c1cnc(-c2ccco2)s1)=O 28106,N1(C(c2cnn(C)n2)=O)CCCC(C2CCCCN2C(=O)C(=O)NCC2CC2)C1 28107,c1(C(=O)OC)ccc(NC(=O)CC2CC(NCc3ccc(O)cn3)C2)cn1 28108,CN(S(=O)(=O)N1CC(O)C(O)(CSCC(C)(C)C)C1)C1CCC1 28109,Cc1csc2nc(CC(=O)N(C3CN(C(=O)CC4CC(C)C4)CC3O)C)cn12 28110,C12(CNC(=NC)NC3CCCSC3)CCC(F)(CN(C(=O)OC(C)(C)C)C1)C2 28111,C(=O)(C(O)CCc1ccccc1)NC(C(C)NC(c1coc(CC2CC2)n1)=O)(C)C 28112,C1(OC)(CNC(=O)C(=Cc2cccs2)C)CCN(C(C2C3CCCCC23)=O)C1 28113,N1(C(CCc2ccn(C)n2)=O)CCC2(NC(=O)C=CC(c3cccnc3)=O)CC2C1 28114,C(=O)(CS(=O)(=O)CC(F)(F)F)NCC1(C(F)F)CCN(C(C(CC)(C)O)=O)C1 28115,c1(C(N(CC(C)NC(C2CCCO2)=O)C)=O)ccc(N)c(C(F)(F)F)c1 28116,C1(C(=O)NC(C(C)C)(C)CNC(=O)C(C)(C)N(C)C)CCCC(=O)N1C 28117,n1(CCCC)ccc(C(=O)NC2(CNC(=O)Cc3c[nH]nc3C)CCCC2)n1 28118,c1(C(N2CC(O)(C(=O)NC3CCN(C(=O)OCC)C3)C2)=O)ccc(O)nn1 28119,c1(C(=O)NC2CCCC(CNC(=O)CCF)C2)ccc2c(n1)CCC2 28120,Cn1ncc2ccnc(C(=O)NCC3(O)CCN(C(=O)Cc4ccc(Cl)s4)C3)c12 28121,c1(NC(C2N(Cc3c(C)c(O)ccc3)CCOC2)=O)cnn2ccc(Cl)nc12 28122,Cc1nc(O)sc1C(=O)NC(C)(CSC)C(=O)N(C)C.C1CCN(C(N)=O)CC1 28123,N1(C(COC2(C)CCC2)=O)CCCC2(NC(=O)C(C)(C)C3CC3)CCCC12 28124,CC(C)C(C(=O)NCC1CN(C(=O)Cc2ccccc2F)CC(C)(C)O1)C(C)C 28125,C(=O)(C(CCSC)NC(=O)C(C)NC(=O)CC)NC(CC=C)C1CCC1 28126,C1(NC(c2cscc2Br)=O)CN(Cc2cncnc2)CC1(F)F 28127,c1(C(=O)NCC2C(NC(c3cc(OCC)n[nH]3)=O)C2)ccccc1CC(C)(C)C 28128,c1(NC(C(C)NC(c2c(COC)cco2)=O)C(C)C)ncc(Cl)c(C)c1C#N 28129,c1(C(N2C3(CN(C(C4CN(CCC)C(=O)C4)=O)C3)CC2)=O)cc(F)cc(F)c1F 28130,N1(C(C2=CC(C)CC2)=O)CCC2(CC1)CCN(C(c1c[nH]nc1C1CC1)=O)CC2 28131,c1(C(N2CC(C)C(NC(c3cscc3S(C)(=O)=O)=O)C2)=O)ccn2ccnc2c1 28132,C(c1csc2ccccc12)=CC(=O)NC1CCCCN(CC)C1=O 28133,c1(C(=O)NCC2(F)CN(C(C3CC(C)OC3=O)=O)C2)cccc2ncn(C)c12 28134,CC(C)CCCCCC(=O)NC(C1(CNC(=O)Cn2cc(C(F)F)cn2)CC1)C 28135,c1(CC(=O)NCC(C)NC(c2c[nH]nc2-c2ccccc2)=O)cc(F)cc(F)c1 28136,c1(CNC(N2CC(c3ccn(C)n3)OCC2)=O)ccc(I)c(Br)c1 28137,C1(OC)CC(CNC(=O)C(=O)NC(C)Cc2cccnc2)C1(C)C 28138,C1(CC)CN(C(=O)CC2CCCCC2)CCN1C(=O)CN1CCCCCC1=O 28139,N1(C(C(CC2CCCC2)NC(c2c(C)nc(O)s2)=O)=O)Cc2n[nH]cc2C1CO 28140,C1(CNC(C(CC=CC)NC(=O)OC(C)(C)C)=O)CC(c2ccc(C)cc2)=NO1 28141,N1(C(Cc2cc(C)sc2C)=O)CCC2CN(C(C3CC3c3cccs3)=O)C2C1 28142,Cc1c(C(N2CCC(CCNC(C3CC(=O)N(CC4CC4)C3)=O)C2)=O)ncn1C 28143,N1(C(CS(N)(=O)=O)=O)CCOCC(NC(=O)C(F)Cc2ccccc2)C1 28144,Cc1nc(Cl)ccc1CC(=O)NCC(O)CN(C)C(c1ccn(C)c1)=O 28145,Cc1ccc(CNC(N2CCC(NC(C34CC(CO3)C4)=O)C2)=O)cc1 28146,c1(OC)ccc(C(N2CC(O)CC2C(=O)NCc2ccc(Br)c(Br)c2)=O)cc1I 28147,C1(C(=O)NC2CCC(NC(CC3C(C)(C)CCO3)=O)CC2)CCOC(=O)CC1 28148,c1(C(N(CCNC(Cc2cnc(C)[nH]2)=O)CC2CC2)=O)ccc(OC(F)F)nc1 28149,C12(CC(N3CCC(n4ccnn4)C3)=O)CCC1CN(C(=O)C=C1CCCCC1)C2 28150,C1(NC(=O)Cn2cccc2)CCCN(C(c2cc(Cl)sc2Cl)=O)CC1 28151,C1(CCC(N2CC(N(CC(=O)N(C(C)C)C)C)C2)=O)CCCCO1.C(C)(C)O 28152,c1(C(=O)NC2C(C)N(C(C3(F)CCCCC3)=O)CC2)ccc2c(O)n[nH]c2c1 28153,N1(C(c2c(C)cncc2C)=O)CCC2C(CCCN2C(=O)C(F)CC(C)C)C1 28154,c1(NC(c2c(CNC(c3ncc(F)cc3F)=O)ccs2)=O)ccc(Cl)c(O)c1 28155,C1(NC(C2CC(=O)NCC2)=O)C2CC(O)C1N(C(=O)CC1(C(F)(F)F)CC1)C2 28156,CC1CCCCC1(CNC(=O)Cc1sc(O)nc1O)NC(=O)CC1CCCCC1C 28157,N1(C(c2nc(OCC)sn2)=O)CCC(C2(NC(c3cc(CC)[nH]n3)=O)CC2)CC1 28158,CCCCCS(=O)(=O)CC(=O)N1CCC(NC(c2cc(OC)c(O)c(N)c2)=O)C1 28159,C1(NC(c2n(CCOC)ncc2)=O)CC(C)N(C(c2nn(C)cc2SC)=O)C1 28160,N1(C(COCC)=O)CCC(C2CCN(C(c3cc(-c4cccn4C)[nH]n3)=O)C2)C1 28161,c1(C(N(CC(C)O)CCNC(c2cncc(C=C)c2)=O)=O)cnc2scc(C)n12 28162,S(=O)(=O)(c1c[nH]ccc1=NCC1(S(=O)(=O)CC)CC1)NCCCC 28163,N1(C(c2ccc(CC)o2)=O)CCC(CNC(c2cccc(CO)c2C)=O)C1(C)C 28164,c1(C(N2CCC3(C(NC(=O)CCBr)C3)CC2)=O)cnc2cc(Cl)ccc2c1 28165,c1(CC(N2CC(OC)C(NC(=O)C(C)S(N)(=O)=O)C2)=O)ccc2c(c1)NC(=O)C2 28166,N1(C(C(CC)SC)=O)CCC2(CC1)CCN(C(=O)C=C(C)c1ccco1)CC2C 28167,CC1=C(C(=O)NC23CCN(C(=O)CC(C)(C)C)CC2C3)CCC1 28168,N1(C(c2c(CC)csc2)=O)CCC(CNC(=O)Cn2nc(C)oc2=O)C(C)C1 28169,C(=O)(CC1OCCc2ccsc21)N1CC(NC(CCCCC(C)C)=O)CC1(C)C 28170,c1(C(=O)NCC(C2CC2)NC(C(N2CC(C)C2)C)=O)cc2cc[nH]c2cn1 28171,C(=O)(CCCCCN(C(C1CCC1C)=O)C1CC1)N(CC(F)F)CC 28172,C(C)(C)(CC(F)C(=O)NCCc1cccnc1)NC(c1scc(C)c1)=O 28173,c1(C(N2CCCC(NC(C(C)n3cccc3)=O)C2)=O)ccc2c(c1)COC2 28174,C(CC(=O)N1CC(CC(C)(C)C)C1)N(C(=O)C=CC(F)(F)F)CC 28175,C(C(C)(C(C)C)NC(c1csc(N2CCCCC2)n1)=O)NC(C(C)OCC#C)=O 28176,C1(NC(C(C#C)(C)C)=O)CCC(C)(CNC(c2conc2C(C)(C)C)=O)CC1 28177,c1(C(=O)NC2C=CC(CNC(C(C)CN(C)C)=O)C2)ccc(=O)n(CCF)n1 28178,CC1CCC(C)(NC(c2conc2CNC(C2C3CCC(=O)C23)=O)=O)C1 28179,c1(-c2cn(CC)nn2)ccn(C)c(=O)c1.Cc1c(Cl)cnn1CC(=O)N(C1CC1)C 28180,C1(C(=O)NCCC2CCCN2C(=O)CC2CCCC23CC3)(OC)CCS(=O)(=O)C1 28181,C1(NC(C(C)NC=O)=O)CCN(C(c2ccnn2CC#N)=O)CC1(C)C 28182,CC1CCCCC1C(=O)NC(C)(C)C=CC(=O)NCC(F)Cl 28183,c1(C(N)=O)ccc(CC(N2CCOCC2CNC(=O)CCC2CCCO2)=O)cc1 28184,C1(CNC(C(C(CC)C)O)=O)CCCC2(CN(C(=O)Cc3cccc(Cl)c3)C2)O1 28185,Cc1c(C(=O)NCC2CN(C(=O)C(F)C3CCC3)CCCO2)nn(C)c1N 28186,Cc1cccc2c(C(N3CCCC(N(CCF)C(C4CC4(F)F)=O)C3)=O)coc12 28187,N1(C(Cc2ccc(CC)cc2)=O)CC(NC(c2cccn2CC)=O)CC1(C)CC 28188,N1(C(C(C(C)C)SC)=O)CCN(C(=O)Cn2ccccc2=O)CC12CC2 28189,Cc1cccc(C(=O)NCC(F)CNC(c2cnc(CC(C)C)[nH]2)=O)c1C 28190,c1(C(=O)NC2CCNC2=O)cc2c(s1)CCN(Cc1cc(Cl)ccc1Cl)C2 28191,C(=O)(C(F)(F)CO)N(C1C(C(NOCc2scc(C)c2)=O)CCC1)C 28192,c1(C(=O)OCC)ccc(NC(=O)Cn2cc(CCCNC(C)C)nn2)cc1C 28193,CC1(C)CC(CNC(=O)CCOCCCNC(=O)Cn2cccn2)CO1 28194,N1(C(C=C(C)C(C)(C)C)=O)CC2CCCCC2(CNC(=O)Cc2ccsn2)C1 28195,C#Cc1ccc(C(=O)NC2(COC)CCN(C(=O)CC(C)CCC)C2)cc1C 28196,CP1(=O)CCN(NC(=O)CC2CS(=O)(=O)C2)CC1 28197,C#CC1CN(C(C2CCC2C#N)=O)CCN1C(c1cnc2[nH]nnc2c1)=O 28198,C(=O)(CCCCCCNC(=O)COCC1CC1)N(C(C1CCOCC1)C)C 28199,N1(CCN(CCOCC)C2CC2)CC(OC(=O)C(=O)NCC)CCC1=O 28200,c1(OC)ccc(CCC(=O)NCCCCN(C)C(c2nn(C)cc2Cl)=O)c(C)c1 28201,C#CCC(C)(C(=O)NCC(C)S(N)(=O)=O)NC(c1cccnc1NC)=O 28202,Cc1c(F)ccc(CN2CCC(F)(C(=O)NC(c3cccnc3)C)C2)c1Cl 28203,CCCC(CCC)C(=O)NCCN(C1CCCCC1)C(C1CC1CCOC)=O 28204,c1(C(=O)NC(CNC(c2cc(SC)oc2)=O)(C)CO)ccc([N+](=O)[O-])s1 28205,n1(CCC(N2CCC(C(C)NC(c3ccc(CC)[nH]3)=O)C2)=O)ccc(O)nc1=O 28206,CCCC(C(=O)OC)C(=O)N1CCC(C)(C)C1C(=O)NCc1cnc(O)nc1O 28207,C1(Cl)(C(N(C(C)CNC(=O)COC)CC)=O)CC1.C1CCC1 28208,C(=O)(CCN(OC)C(=O)C(N1CCOCC1)C1CC1)Nc1cc(SCC)ncc1 28209,c1(N2CC(C)(NC(C(C)OCC3CC3)=O)C2)ncnc2sc(C(F)(F)F)nc12 28210,C(=O)(C1=NOC(C)(C)C1)NC1CCC(NC(CC(CN(C)C)O)=O)C1 28211,N1(C(c2cnn(C3CCOC3)n2)=O)CCN(C(c2csnc2Br)=O)CC1 28212,c1(C(=O)OC)cc(CCNC(=O)C(F)C2CC(NC(c3ccc[nH]3)=O)C2)on1 28213,C(=O)(C(C)(C)C(F)F)N1CCCC(CCNC(C2C(C)(C)C2(F)F)=O)C1 28214,N1(C(CN(C)CC)=O)CCCC12CCN(C(C1CCC(C)=C(C)C1)=O)C2 28215,N1(C(c2c(CC)ncs2)=O)CCCC(C(C)NC(c2c(C)nnn2C)=O)C1 28216,C(CCCCCNC(=O)Cc1ccnc(C)c1)N(C(Cc1c(CC)con1)=O)C 28217,c1(C(=O)NCC#CCNC(=O)C=CC2CCCO2)cc2ccccn2n1 28218,c1(C(=O)NC(CC(C)NC(=O)Cn2cc(Cl)cn2)C)ccc2c(c1)CCC2(F)F 28219,S(=O)(=O)(c1ccc2c(c1)COCC2)NCc1c2c(ccc1)OC(C)(C)C2 28220,C1(C(=O)NC2CCCC(NC(=O)CSCC(F)(F)F)C2)(CC)CCC(O)CC1 28221,c1(C(=O)NC(CN(CCC)CC2CC2)C)cnn2c(-c3ccccc3)ccnc12 28222,C[Si](C)(C)CCNC(=O)C(CO)NC(=O)Cc1cc[nH]n1 28223,Cc1ccccc1CC(C)C(=O)NCCC1(NC(=O)CCSCC(N)=O)CC1 28224,CS(=O)(=NC(=O)CC1CCCCS1(=O)=O)c1ccccc1 28225,c1(C(N(C)CC2CCCN(C(CCC3CCC(C)O3)=O)C2)=O)c[nH]cc(F)c1=O 28226,C12(NC(CC(CC)C(C)C)=O)CCCC(CN(C(c3cccn3C)=O)C1)C2 28227,N1(C(CCC(C)(C)F)=O)CC2CCC(C1)N2C(C1(C)CSC1)=O 28228,c1(NC(N(CCCNC)C)=O)cccc(C(N)=O)c1.C1(=O)CN1 28229,Cc1nnc2n1CCN(C(=O)NCc1ccc(C3CCC3)nc1)C2 28230,N1(C(C2CC(CCC)OCC2)=O)C2CCCC1CN(C(c1cccc(CO)n1)=O)C2 28231,C1(NC(C(C)(C)C)=O)CC2CC(NC(C3CCCN(c4nccs4)C3)=O)C1C2 28232,C(=O)(C(CCCOC)NC(C1CC=CCC1)=O)NCCSCC#C 28233,CCC(CC)CC(F)C(=O)N(C(C)CNC(=O)C(C)(C)C1CCOC1)C 28234,N1(Cc2cccc(CC)c2)CC2CC(NC(=O)CS(=O)(=O)C(C)C)CC1C2 28235,CCC(CC(=O)N1CCC(C(C)O)CC1)NC(=O)C(=CC1CCCC1)C 28236,NS(=O)(=O)CCC(=O)N1CC(Cn2cc(C3(O)CCOC3)nn2)C1 28237,Cc1nc(C(C)C)ccc1CNC(=O)C=CC(C)NC(C1CC1(C)C)=O 28238,N1(C(C2(CCOC)CC2)=O)CCC2C(C1)CN2C(=O)CC1(C(F)(F)F)CC1 28239,C#CC1CN(C(=O)CCOCCN(C(=O)C(C)CC(C)C)C)CCN1C 28240,N1(C(CC(CC2CC2)NC(C2(C=C)CCCC2)=O)=O)CCCC(C)(OC)CC1 28241,Cc1ccc(CN2C(C(=O)NCC3CCC(O)CC3)CC3CC23)c(Cl)c1Cl 28242,C1(C(=O)NCc2ccc(CNC(C3C(C)N(C)CC3)=O)cc2)CC2CCC1CC2 28243,N(C1CC(C)n2ccnc21)C(CCC(Cn1cc(CNC(CC)=O)nn1)(F)F)=O 28244,C1(CNC(C2CN3CCC2CC3)=O)CCN(C(=O)Cc2ccccc2Cl)C12CC2 28245,C(=O)(C1Cc2ccc(Cl)cc21)NC1C2CN(C(C3(C)COC3)=O)CC1COC2 28246,C1(CC(=O)NCC(N2CCN(C(c3ncccc3F)=O)CC2)C)CC2(CCC2)C1 28247,C1(C(C(=O)NCc2ccco2)N(CC(C)C)Cc2ccccc2)CCOC(C)C1 28248,N1(C(C2(CNC(C3COCC(C)O3)=O)CCCCC2)=O)CCCN2CCCC2C1 28249,C(=O)(C(C)(C)C(F)(F)F)NCCC1CCC(NC(CCC(=O)NCC)=O)C1 28250,CCCCCCCC(=O)N1CC(CNC(=O)C(c2ccc(Cl)cc2Cl)O)C(C)C1 28251,C12CCCCC1C(=O)N2.C1(N(C)C)CC(C)(NC(=O)CCC2CC2(C)C)C1 28252,C1(NC(CCCCOCCC=C)=O)CC2C1CCN2C(=O)CC(CC)C1CCC1 28253,N1(C(C(C(C)C)OCC)=O)CCC2(CCCN(Cc3ccc(Cl)c(F)c3)C2)C1 28254,N1(C(C(CC)C#N)=O)CCCC(C(=O)NC2COCC2CO)CC1 28255,N1(C(c2cccc(OC)c2N)=O)CC23CCCC2(C1)CN(C(c1ccc[nH]1)=O)C3 28256,Cc1ccccc1CC(N1CCCC(CCNC(c2cncn2C(C)C)=O)C1)=O 28257,c1(OCC#C)cncc(CN2CCC(SC)CC2)n1 28258,C(CC(C)(C)CC(=O)NCC1CC(C)CCN1C(c1ccc(=O)n(C)n1)=O)OC 28259,c1(C(=O)NC2(CC=C)CCN(C(=O)CSCCC(C)C)C2)cnc(C)c(C)c1 28260,CC1C2CCC(C2)C1C(N1CCC(C)(C(N2CCOCC2C(C)O)=O)C1)=O 28261,c1(C(N2CC3(N(C(C(O)NC(=O)OCC)=O)CC3)C2)=O)csc2ccc(Cl)cc12 28262,c1(-n2c(-c3cnc(OCC)nc3)nc(C(C)O)n2)ccc(Cl)c(F)c1 28263,c1(C(=O)NC(CC=C)CNC(=O)CCCC2CCCCC2)ccc(CO)cn1 28264,c1(C(=O)OC)cncc(C(=O)NC23CC(NC(C4CCCNC4=O)=O)(C2)C3)c1 28265,C(C(CNC(c1cc(F)n(C)n1)=O)S(C)(=O)=O)NC(c1cc(CC)sn1)=O 28266,C(C(CC1CCCC1)C(=O)NC1CCC(C)CC1)NC(COC(C)=O)=O 28267,CC(C)(C)COCC(=O)NC(C(=O)NCCOC(F)(F)F)C1(C)CC1 28268,N1(C(C2C(COC)CC2)=O)CCN(C(c2ccccc2Cl)=O)CC(O)C1 28269,CCC(C(=O)OC)C(=O)NC1(CNC(c2cccc(SC(F)(F)F)c2)=O)CCC1 28270,c1(C(N(CC(=O)Nc2cn(CC)nc2)C2CCC2)=O)cnnc(C)c1 28271,c1(-c2nc(CCN(C)C)nn2Cc2cccc(O)c2F)cc(F)c(CO)c(F)c1 28272,N1(c2cc(CC)nc(C)n2)CCOC2(CCCN(C(=O)CC3CCC(C)C3)C2)C1 28273,C1(N(C(CCC#CC)=O)C)CN(C(c2cncn(C)c2=O)=O)CC12CC2 28274,C1(NC(CCC(C)c2ccccc2)=O)CC=C(C(=O)N2CCSCC2)C1 28275,C(C(C)C(=O)NC(C)(CNC(=O)COCCCC(C)C)CC)OCC 28276,N1(C(C2CCC(=O)OCC2)=O)CCN(C(c2ccc(F)s2)=O)C2CCC12 28277,C(=O)(CS(=O)(=O)N(C)C)NC(C1CN(C(c2cn(C(F)F)cn2)=O)CCO1)C 28278,N1(C(C2C3(CN(C(c4cc(OCC)c(Br)cc4)=O)C3)C2)=O)CCC(C)C(F)(F)C1 28279,N1(C(c2c(CNC(C3(C)CCCN(C)C3)=O)occ2)=O)CC2(CNC(=O)N2)C1 28280,N1(C(C(C)CS(C)(=O)=O)=O)CCN(C(C2(C)CCN(C)C2=O)=O)CC(C)(C)C1 28281,N1(C2c3cc(sc3)C(C)NC2=O)CC(C)(C)C1C(=O)OC.C1(NC(=O)NC)CCC1 28282,C1(C(=O)NCCN(C(C=C2CCC(C)C2)=O)C2CC2)(CO)CC(C)(C)C1 28283,C=CCC(CC(F)F)NC(=O)C(CCC1CC1)NC(c1ccncc1CC)=O 28284,C1(C(=O)NCC(C)NC(C2CC23CCCC3)=O)CC2(CCO1)CC2 28285,C1(NC(C(c2ccc(Cl)cc2)(C)C)=O)CN(C(C2CC(C)(C)C2)=O)CC(F)(F)C1 28286,CCS(=O)CC(=O)NCCN(CCOC)C(c1cccnc1OCCO)=O 28287,n1(CC(=O)NC2CC(NC(c3cocn3)=O)C(O)C2)ccc2ccccc2c1=O 28288,CC1=C(C(=O)N2CCC(CO)(NC(c3ccc(CC(C)C)nc3)=O)C2)CCO1 28289,O(NC(=O)CN=c1[nH]c(=NCC2(OC)CCCC2)c2cc(F)cc(F)c2[nH]1)CC 28290,c1(C(N(C)CC2CCCN2C(c2coc(Cl)c2)=O)=O)ccc(F)c(O)c1 28291,c1(C(=O)NCCCC(C)NC(C2(CO)CCCO2)=O)cc2cccnc2nc1O 28292,c1(OC)ccc(C(=O)NC2CCC(NC(c3c(Br)cncc3Br)=O)C2)cc1OC 28293,C1(C2(O)CCN(C(C3(C)CC3(Cl)Cl)=O)CC2)(NC(c2c(CC)occ2)=O)CC1 28294,C(=O)(C(C)(C)CCC(=O)OC)NCC1CCCN(C(C2(C(=O)OCC)CC(=C)C2)=O)C1 28295,C1(C(N(C2CC(CO)C2)C)=O)CCOC1C(=O)NC1CCCC1F 28296,C1(COCC)CCCN(C(=O)C(Cn2cccn2)NC(c2ccc(C#N)o2)=O)C1 28297,C(=O)(Nn1nnc2c1CCCC2)C1C2(CC(NC(C(C)(C)OCC)=O)C2)C1 28298,C(=O)(C1=CC2(CCN(C(=O)Cn3c(O)nnc3O)C2)C1)NCc1cc(C)oc1 28299,c1(CO)cccc(Br)c1NC1CCCC(n2ccnc2)C1 28300,c1(C(=O)NC2C3CN(C(CC(CC)SC)=O)CC32)cccc2c(C)coc12 28301,c1(C(=O)NCCC(CNC(C2COCC2(C)C)=O)OC)cc2nccnc2[nH]1 28302,C(=O)(CS(=O)C(F)(F)F)NCC(C1CCCC1)NC(CNC(CC(C)(C)C)=O)=O 28303,C(CCC(C)(C)C(=O)Nn1nnc(C)c1C)NC(C(CC#C)O)=O 28304,N1(C(C2C(CC)OCCC2)=O)CCN(C(=O)C(F)(F)c2ccccn2)CC(O)C1 28305,CCC(C)C(O)C(C)C(=O)N1C2CCC1C(NC(=O)CCNC(C)=O)C2 28306,N1(C(C2N(C(c3scc(OC)c3)=O)CCC2)=O)CCC2(CCOC2)CC1 28307,C1(NC(C(CC=CCC)C)=O)C2CCC1CN(C(=O)CC1CC(F)C1)C2 28308,N1(C(C)CSc2cncn2C)CCC(O)(Cn2cc(-c3cncc(F)c3)nn2)C1 28309,c1(CNCC(=C)Cl)csc(C2OCCO2)c1 28310,C1(C(=O)Nc2c(C)nsc2C)CCN(C(c2cncc(C#N)c2)=O)C(C)(C)C1 28311,c1(C(N2C(CC)C(NC(c3cccnc3)=O)CC2)=O)ccc(OC)c(Cl)c1F 28312,CC1(CNC(C2CC23CCCC3)=O)COCCN(C(=O)C=CC=C(Cl)Cl)C1 28313,C1(C(=O)NCCC(C)N(C)C(c2ccc(C3CC3)o2)=O)C2CC(F)(F)CC12 28314,Cn1nnc(Cn2nnnc2C(C2(C(F)F)CCC2)NCC2CC2)n1 28315,Cc1nc(N2CCCC(NC(c3cc(C)c(F)cc3C)=O)C2)c2c(n1)CCC2 28316,CCC(C#N)(CC)C(=O)N1CCC(C(C)NC(c2csc(F)c2)=O)CC1 28317,c1(COC(C)C)ccc(F)c(C(=O)N(CC(C)N(C(=O)CC2(CO)CC2)C)C)c1 28318,N1(CC(=O)N(C2CCN(C(=O)Cn3ncn(C)c3=O)CC2)CC)CCCCCC1 28319,c1(CC)cc(CC)cc(S(=O)(=O)N2CC(CO)OC3(CCC3)C2)c1 28320,C=CCC(C)(C)C(=O)NCC1(O)CC(NC(c2nnn(C)n2)=O)C1 28321,C1(CNC(C2(CC)CC2(F)F)=O)CCCN(C(C2(C(C)(C)C)CCC2)=O)C1 28322,C1(C(N2CCC(C(C)NC(=O)CCn3cc(Cl)cn3)CC2)=O)CCCCC(=O)C1 28323,N1(C(C(CCC)(C)O)=O)CC(C)(C)OC2(C1)CN(C(=O)C(C)C(O)CC)C2 28324,N1(C(C=C(CCN(C)C)Cl)=O)CCC2(CCN(C(c3ncccc3N)=O)C2)C1 28325,C1(C(N2CCN(C(c3ccc(C(C)=O)nn3)=O)CC2)=O)CCc2ncncc2C1 28326,c1(C(=O)NC2CCC(CNC(CC)=O)C2)ccc(CCC(N)=O)cc1 28327,c1(C(=O)NCC2N(C(c3cc(C(C)=O)oc3)=O)CC2)c(Br)ncn1C 28328,C(=O)(C1=NOC(CNC(=O)CC2C=CCC2)C1)N(C(CCO)C(F)F)C 28329,c1(C(=O)NC23CCN(C(c4ccc(C)c(O)c4)=O)CC2C3)nccn2cnnc12 28330,C1(C(N2CCN(C(c3cnc(Cl)s3)=O)C3C2C3)=O)CCc2ccccc2CC1 28331,c1(NCC)ccc(Nc2cn(C)nc2C(=O)N(C)C)cc1OC 28332,N1(C(C(C)(C)OC)=O)CCN(C(=O)CC2(c3ccccc3)CCOCC2)CC1 28333,N1(C(C=CCCC)=O)C2CCC1C1CC1(NC(C1CCCC(F)(F)CC1)=O)C2 28334,c1(OC)cc(CNC(=O)C(=O)NC(C2CC3CCC2CC3)C)c(F)cc1F 28335,C(CCC(=O)N(C)CC1CN(C(c2occc2Br)=O)C1)N(C(C)=O)C 28336,Cc1nc(C)c(C(=O)NCCN2CCC(NC(=O)CS(N)(=O)=O)CC2)[nH]1 28337,Cc1ccc2c(C(N3CC(NC(C4(N(C)C)CCC4)=O)CC3C)=O)csc2c1 28338,C1(C(=O)NCCC2CC(NC(c3nc(CC)sc3)=O)C2)CN2CCN1CC2C 28339,Cc1ncn(C)c(=O)c1C(=O)NCC#CCNC(=O)CSCC(=O)OC(C)(C)C 28340,N1(C(C(C)=C(C)C)=O)CCN(C(c2cc(C#N)ccc2C)=O)C2CCC12 28341,N1(C(c2c(COC)n(C3CC3)nc2)=O)CCN(C(=O)CSCCN(C)C)C(C)C1 28342,C1(OC)CC2(C1)CC(NC(c1cnn(CCNC(=O)CC3CCC3)c1)=O)C2 28343,C1(N(C)C)(C(=O)NCC2C=CC(NC(c3cccnc3S)=O)C2)CCCCC1 28344,N1(C(c2cn(CCC(C)C)nn2)=O)CCC(NC(=O)CCC(C)(C)O)C(C)C1 28345,N1(C(CNC(C)=O)=O)CCCC(N(C)C(C2COCC(=O)N2C(C)C)=O)CC1 28346,C1(N(C(C)C(F)F)C(=O)CCNC(c2cncnc2)=O)CCC(C#N)CC1 28347,c1(CCC)nc(C)c(C(=O)NCCN(C(=O)CSCC)C2CC2)s1 28348,c1(C(N2CC3C(NC(c4c(CC)nco4)=O)(CC3)C2)=O)cc(N)c(C)cc1Cl 28349,c1(C(N2CC(NC(CN(C)CC)=O)C3(C2)CC3)=O)cc(C)c(C)cc1C 28350,c1(NCC(CC)N(C)C)ccc(S(=O)(=O)NCC(N2CCOCC2)C)cc1Br 28351,c1(NC2C(C)(CC)C2)ncnc(NCc2cc(C(C)C)on2)c1C 28352,C(=O)(CS(=O)(=O)CC1CCCO1)NC1(CNC(C(C)n2cncn2)=O)CCC1 28353,c1(C(N2CC(NC(c3ccc(C)s3)=O)C(F)C2)=O)ccc(F)c(C(F)F)c1 28354,N1(C(c2c(C)nc(-c3c(C)cnc(F)c3)s2)=O)CC2CC(C1)c1ccccc12 28355,c1(NC(=O)NC(C2CCC(F)(F)C2)C(=O)OC(C)(C)C)cc2ccsc2n1C 28356,C1(C(=O)NCCC2CN(C(C3(C)CC4CC4C3)=O)C2)CCC2(CCCO2)CC1 28357,n1(CC(=O)NC(C2CCN(C(=O)Cn3cc(CO)nn3)C2)C)ccsc1=N 28358,CC1CC2(CC(C(=O)NCC3CCCCC3NC(C3CC(C)CC(=O)N3)=O)C2)C1 28359,C1(CNC(CCC2(NC(CSC)=O)CCCC2)=O)CCCCC1(C)C 28360,C1(N(C(C(CSC)C)=O)C)CN(C(c2c(O)cccc2F)=O)CC12CC2 28361,CCC(c1ccc(C)cc1)=CC(N1CCN(C(=O)COCCF)CC1C(C)C)=O 28362,c1(CCC(N2C(C(=O)NC3(CC)CCOC3)CCCC2)=O)ccc(OC)c(F)c1 28363,N1(C(C2CC(NC(C3CC3Br)=O)C2)=O)CC(O)(c2cnn[nH]2)C1 28364,C1(NC(c2cn(CCC)nc2)=O)CCCCCC1NC(=O)C(F)(F)c1cncs1 28365,C(=O)(CC(F)(F)C(F)F)NC1CCCC(CNC(c2c(C)nc(C)s2)=O)C1 28366,N1(C(CC2CCC(=O)NC2=O)=O)CCC(NC(=O)C=CC2CC2)C(CO)CC1 28367,C(=O)(C(CC(C)C)N(C)C(c1ccc(O)nn1)=O)NC(CC#C)C(N)=O 28368,c1(C(=O)OC)cc(CS(N2CC3CC2CN3C(=O)C(F)(F)F)(=O)=O)oc(=O)c1 28369,N1(C(c2ccc(C)c(Cl)c2)=O)CCC2(CC1)CC2NC(C1(C)CCSCC1)=O 28370,C1(CNC(C(C(C)C)NC(C)=O)=O)CN(C)CCN1c1cnc(C#N)cn1 28371,C1(C(C)NC(c2cc(Cl)c[nH]2)=O)CCCCN1C(=O)CCc1cccs1 28372,N1(c2cc(C)nc(Cl)n2)CCC(NC(C2CCC3CCCCN23)=O)C(C)(C)C1 28373,CC1COCCC1NC(C1CC12CC(NC(C1(c3cc[nH]n3)CC1)=O)C2)=O 28374,N1(Cc2c(O)ccc(OC)c2)CCC2(CC1)CC(C(=O)Nc1cn(C)cn1)CO2 28375,c12cscc1OC2.CC(C)C=CC(=O)N(CCC(C)(C)C)C(C)C 28376,c1(OC)ccccc1OCC(=O)NCC(O)CN(C(=O)C1=CCSC1)C 28377,C1(NC(CCSCC)=O)COCCC1C(=O)NC1CC=CCC1C 28378,N1(C(C2C(C)CC2)=O)CCOC(CC(=O)N(C2CCCCC2)CCO)C1 28379,N1(C(C=C2CCN(C)C2)=O)CCC2CN(C(C3CC(N4CCOCC4)C3)=O)CC12 28380,Cc1cc(NC(C2C3CCC(C3)N2C(=O)COc2cnc(Cl)cn2)=O)cc(F)c1 28381,N1(CCCC2C(C)C2)CC2(CO)CC2(C)C1 28382,c1(CNC(CC(COC)OC)c2nnnn2CC(F)F)cnc2cc(Br)ccn12 28383,c1(NC(C2C3(CC(NC(c4ccn(CC)c4C)=O)C3)C2)=O)cccc2occc12 28384,C1(CC(=O)NC2CC(CCOC)C2)C2CC(C2)N1C(c1cc(C)oc1C)=O 28385,Cc1cc(C(N2CCCC(C(N3CC(C(C)(C)C)C3)=O)CC2)=O)cc(O)c1 28386,c1(NC(C2(C)CN(Cc3cccc(C=O)c3Br)C2)=O)csc2nccnc12 28387,N1(C(C(C=C)(C)C)=O)CCN(C(c2ccc(CO)nc2)=O)C(c2cnn(C)c2)C1 28388,c1(C(N(C2CCCN(C(C3CCC(=O)NC3)=O)C2)CCF)=O)nnc2ccccn12 28389,C1(NC(C2N(C(c3c(C)cc(CC)o3)=O)CCC2)=O)C(=O)NCCC1C 28390,C#CCC(C(=O)NOCC1CCCOC1)NCc1cn(C(C)(C)C)nn1 28391,c1(OCCC)ccc(C(=O)NCc2ccc(CO)c(F)c2)cc1C 28392,c1(CC(=O)NC(C)CN(C(=O)CNC(c2cn[nH]c2)=O)C)csc(NC2CC2)n1 28393,C1(NC(C2CN(CC)C(=O)CC2)=O)CN(C(=O)CSC(C)C)CC2(CC2)C1 28394,c1(C(=O)NCCC(C)N(C)C(c2cccnn2)=O)csc2ccc(F)cc12 28395,c1(C(N2C(C#N)CCC2)C(=O)NC2CC2)ccc2c(c1)CCC2 28396,C(C1=NOC2CN(C(=O)C#CC3CCOCC3)CC12)NC(c1c(C)scc1)=O 28397,c1(C(=O)NCC2(O)CCN(C(C3(C#N)CCC3)=O)C2)ccc2ncnn2c1 28398,C1(C)(NC(CNC(CNC(c2cnc(C(C)C)o2)=O)=O)=O)CCCC1(C)C 28399,CCCCC(C)CCC(=O)NC1COCC1(C)NC(=O)OC(C)(C)C 28400,N1(C(c2cc(C)sc2C)=O)CC(C)OC2(CCN(C(C3CC3C(C)C)=O)CC2)C1 28401,c1(N2CC(C(=C)C)OCC2)nc(=NCCc2ccoc2)[nH]c2c1cnn2C 28402,C(=O)(C1CCCc2c1ncn2C)NCC(C)(CO)NC(c1cc(C)on1)=O 28403,N1(C(C(OC)OC)=O)CCC(NC(C2(c3ccc(C(F)(F)F)cc3)CC2)=O)C1C 28404,c1(Cn2cc(C3CC(NC(C4(CC)CCCC4)=O)C3)nn2)cc2n(n1)CCCO2 28405,c1(OC)cc(C(=O)NC2CCC(N(C)C(c3cccc(=O)n3C)=O)C2)c(F)cn1 28406,C1(CC(=O)NCCNC(C)=O)CC2(C1)CN(C(c1cc(C)cs1)=O)C2 28407,C1(NC(C2CC(OC)C2)=O)CC2(C(=O)NCC(C)CN(C)C)COC1C2 28408,C1(C(N(CCN(C(C)C)C(c2ncc(Cl)n2C)=O)C)=O)CCC2CC2CC1 28409,N1(c2c(C(=O)OC)cncc2)CCC(C)(CNC(c2ccc(F)c(C)c2)=O)CC1 28410,N1(C(C2CC(CC)N(C(=O)Cc3cn(C)cn3)CC2)=O)CCC(F)(F)C(O)C1 28411,CCCCC(C)(F)C(=O)N(C)CC1(O)CCN(C(=O)C=Cc2cccc(F)c2)C1 28412,c1(CC)ccc(C(C)NC(C)CC2CCNCC2)cc1 28413,C1(CN(C2CCN(C(c3ccc(-c4ccco4)s3)=O)C2)C2CC2)CCCOCC1 28414,N1(C(c2c(OC)cnnc2)=O)CCC2(CCN(C(=O)C(N=[N+]=[N-])C(C)C)C2)C1 28415,C12(CCS(=O)(=O)CC1)C(=O)N2.c1(CC(C(=O)NCC2CCC2)N)ccc(Cl)cc1Cl 28416,n1(CC)cnc2c(NC(c3cc(F)c(F)c(F)c3)C)[nH]c(=NC(C)CF)nc12 28417,c1(C(C)(C)C)cc(CNC(=O)C(c2ccc(-c3nn[nH]n3)cc2)O)cc(F)c1 28418,c1(C(=O)NCC(CN(C(c2ccc(C(F)(F)F)o2)=O)CC)(C)C)cnnc(C)c1 28419,C#CCCCCC(C(=O)NC(C)CC)N1CCC2CCC(C1)N2C 28420,C1(NC(C=CC)=O)CN(C(c2ccc(C(=O)OC)cn2)=O)C2CC12 28421,C(CNCCO)(N=c1ccc(Br)c(C(=O)N(C)C)[nH]1)c1c(OCC)cccc1 28422,C1(CNC(COC)=O)CCCC2CN(C(c3cnc(CC(C)C)s3)=O)CC12 28423,C(=O)(C1=C(Cl)CCC(C)C1)N(CCN(C(CC(C)P(C)(C)=O)=O)C)C 28424,C(=O)(CS(=O)(=O)CC(C)C)N1CCN(C(CC2(CC=C)CCCC2)=O)C(CO)C1 28425,Cc1ccccc1-n1cc(C(N2CC(NC(C3CC3C(=O)O)=O)C2)=O)nn1 28426,CCN=C(NCc1ccc2c(c1)OCO2)N1CCC(O)CC(C)(C)C1 28427,N1(C(C23C(CN(Cc4cccc(N(C)C)c4)C2)C3)=O)CC2CCCC2C1 28428,c1(CC(=O)N(CCC(C)NC(=O)CCCCN(C)CCO)C)ccc2c(c1)CCO2 28429,C1(NC(C23OC(C)(C)C(C2)C3)=O)CCCC1C1CCCC1 28430,c1(C(=O)NCC2CCC(NC(CCCOC(C)C)=O)C2)ccc(C(O)CF)cc1 28431,N1(C(c2c(C)n(C)nc2)=O)CCCC2(CCN(C(c3cc(N)cc(O)c3)=O)C2)C1 28432,C1(NC(c2n(CC)nnc2)=O)CC2CN(C(c3cccc4c[nH]nc34)=O)CC2C1 28433,C1(CC(=O)NCCC2(O)CN(C(COCCSC)=O)C2)CCCCC1C 28434,C1(NC(C2C(=C)C2C(=O)OC)=O)CC(CO)N(C(=O)C(C)CC2CCCC2)C1 28435,N1(C(Cc2cn(CC)nc2)=O)CC(OC)CC1(C)CNC(c1ccc(C)nn1)=O 28436,N1(C(C(N2CCP(C)(=O)CC2)C)=O)CC2CCC1C(NC(=O)CS(C)(=O)=O)C2 28437,C1(NC(=O)CN2CC=CC2)CS(=O)(=O)C2CN(C(C3CC4CC4C3)=O)CC12 28438,C(=O)(C(CO)C(C)(C)C)NCCCN(C(c1cnn(CC)c1C)=O)CC 28439,c1(COC)nc(N2CCC(C(C)NC(C3CC3C)=O)C2)cc(O)n1 28440,C1(N(C(C(C)c2cccs2)=O)C)CN(C(C2CC(=O)C23CCC3)=O)CCC1O 28441,CCCC(O)C(CO)NC(=O)C(CCC1CCC1)NC(=O)Cc1cccn1C 28442,CC1=CCCN(C(C2CC(=O)CN2C(C2CC(O)C(F)C2)=O)=O)C1 28443,N1(C(C(COC(C)C)NC(C)=O)=O)CCC(C(=O)NC2(C(C)O)CCC2)C(O)C1 28444,c1(CCC(=O)NC(C2(O)CCN(C(C3C4COCC34)=O)CC2)C)cc(F)cc(F)c1 28445,N1(C(=O)NC(C)CNCCn2cc(NC(=O)OC(C)(C)C)cn2)CCCC(O)C1 28446,c1(C(=O)NCC(C2CCCC2)NC(c2cnn(C)c2Cl)=O)c(F)cc(Cl)cc1F 28447,N1(C(C(CC=CC)C)=O)CCN(C(c2cnn(C(F)F)c2)=O)CC1CC(F)(F)F 28448,O=C1NCC2(CO1)CN(C(C1(CNC(c3ccc(CO)cn3)=O)CCCO1)=O)C2 28449,C1(CC)CCCCCCN1C(C1CCCC1NC(c1ccncc1)=O)=O 28450,CCCC(CC)C(=O)NCC1(F)CCCN(C(c2cc(O)ccc2Br)=O)C1 28451,N1(C(CCOC)=O)CCC(C(F)F)(CNC(=O)C(C)Oc2ccccc2F)C1 28452,N1(CCC(=O)NC2(C)CN(C(C3CCCC34CCC4)=O)C2)C(=O)NC(C)(C)C1=O 28453,N1(CCNC(C(C)CC2CC2)=O)CCC(NC(C2CCOC2(C)C)=O)CC1 28454,Cc1nn(C)cc1C1CCCN1C(C1CCCCN1C(=O)Nc1ccccc1)=O 28455,c1(C(C(=O)NC2CCOC2)N(C2CC2)CC2CC2)ccc(Br)cc1 28456,C(C(C)(C)CN=C(NCC(c1ccco1)N1CCCC1)NC1CCCC1)OC(C)(C)C 28457,C(C)(C(C)C(=O)NCc1noc(C)n1)NC(CSCCOC)=O 28458,C1(COC)CC(CNC(=O)C(C)Cc2ccnn2C)N(C(c2cccn2C)=O)C1 28459,Cc1ccc(CN2CCC(CNC(c3ccn(C4CCCCC4)n3)=O)C2)o1 28460,c1(C(=O)NC2(CNC(C(C3CCCOC3)OCC)=O)CC2)coc(Br)c1 28461,CC(C)CC(C(=O)NC(CC1CC1)C(=O)NCCC(C)N1CCC1)C(N)=O 28462,C12(C(N(C)CC)=O)CC(CN(C(c3cnn4c3CCC4)=O)C1)C2 28463,CCCC(C)(CC)C(=O)NC(C)CCNC(=O)C1=CSCS1 28464,c1(C(=O)NCC2N(C(c3cnn(CC)c3Br)=O)CC2)cc2c(s1)CCCC2 28465,C12(CC(N3C(COC)(CNC(c4ccn(C)c4)=O)CCC3)=O)CCC(CC1)OC2 28466,C(CC(=O)N1CCN(C(c2ccc(O)nn2)=O)C(CF)C1)(C(F)(F)F)OC 28467,C1(CC)(CC)CC(C(=O)NC(C)CC(C)NC(=O)CN(C)C(C)=O)C1 28468,C1(NC(c2c(OC)ccs2)=O)CN(C(C2(C)CCNC2=O)=O)CCC12CCC2 28469,CCCC(C)CCCC(=O)NC1CN(C(=O)Cc2nnc(S)n2C)CC1C1CC1 28470,C(C)(C)(CN=c1[nH]c2ccccc2o1)NC(C(C(CC)C)O)=O 28471,c1(C(C#C)O)ccc(C#N)cc1.C1(COC(=O)OC(C)(C)C)CCCN1C(=O)NC 28472,c1(C(N(C(C)CN(C)C(C2CC(CCO)C2)=O)C)=O)cccc(C2(C)CC2)c1 28473,Cc1cncnc1C(N1CCCCC1CNC(=O)CC1CC(=O)NC1=O)=O 28474,N1(C(CN(C)CC)=O)CCC2(C=C(C(=O)NC3CC(CSC4CC4)C3)C2)C1 28475,CCCC(CNC(C1CCCC1O)=O)C(=O)NCCC1CC1C 28476,N1(C(c2c(C)n(C)nc2)=O)CCC(C2CC(NC(C3(C)CCCS3)=O)C2)CC1 28477,CC1CC(CCNC(=O)CCOC2CC2)CCN1C(=O)CC(Cl)Cl 28478,Cc1cc(C(=O)NCC2(C(=O)NCCCN3CCCC3C)CC=CC2)ncc1F 28479,CC(C)CC(F)(F)C(=O)NC1CCCCC1NC(C1(NC(N)=O)CCCCC1)=O 28480,C1(NC(C(CCCCC)O)=O)CCN(C(c2ncc(C)cn2)=O)CC12CCC2 28481,C1(CNC(c2coc(CO)c2)=O)OCCC1NC(=O)CSC1CCOC1=O 28482,CC1CCC(CCNC(=O)CC(C2CC2)NC(c2ccnn2C2CC2)=O)C1 28483,c1(OC)ccnc2c(NC(=O)Cc3csc(=NCc4cocn4)[nH]3)cccc12 28484,C(=O)(C(C)(O)C(F)(F)F)NCC(CC(C)C)(C)NC(=O)CCn1cnnn1 28485,N1(C(C(C=C=C)C)=O)CCN(C(=O)Cn2nc(C)c(Cl)c2C)CC1C(F)F 28486,CC(C)C(CNC(c1cc(Cl)on1)=O)NC(C1(C)CCCS1)=O 28487,Cc1ccc(N)c(C(=O)N(C)CC2CCCN2C(=O)C(C)(C)N2CCCCC2)c1 28488,C(CNC(=O)Cn1cc(C)cn1)(CC(=O)NCCn1nncc1C)OC 28489,c1(C(=O)NC2(C)CC(NC(C3(n4cnnn4)CC3)=O)C2)ccc2oncc2c1 28490,c1(OC(CC)C)cc(C(N2CCC(CF)CC2)C(=O)NC)ccn1 28491,N1(C(C=CCN(C(C2(OC(C)C)CCC2)=O)C2CC2)=O)CCC12CCCC2 28492,N1(C(=O)OC(C)(C)C)CCCC(C(N2CCC(COC3CC3)C2)=O)CC1 28493,c1(C(=O)NCC(CCOC)NC(=O)Cn2cccc2)ccn(C(C)C)c1C 28494,Cc1cccc(C(O)C(=O)NC2CC2NC(=O)CCC2(C)CC2)c1 28495,C1(C(=O)NCC2(CO)C(C)(C)C2)CN(C(C2C3CCCCC23)=O)CC1(F)F 28496,C(=O)(C(C)(C)C(C)O)N(CC(=O)NCc1ccnn1C(C)C)CCOC 28497,CCC(N=c1[nH]c(N2CCC(C(F)F)CC2)nc2ccc(OC)cc12)c1nccs1 28498,Cc1csc(=O)n1CC(=O)NCC1CC(C)N(C(=O)C=CC(C)(C)C)C1 28499,CCC(C)CC(=O)C(=O)N1CCC2(CC(C(N3CCOC(C)C3C)=O)C2)C1 28500,c1(NC(CN(C2CCCN(C(C(C)C)=O)C2)C)=O)ccc([N+](=O)[O-])cc1.C(C)(C)O 28501,C1(C)(C(=O)NCC(CNC(c2c[nH]c(=NCC)s2)=O)OC)COC(C)(C)CO1 28502,Cc1n[nH]cc1CNC(C1OCCC1CNC(C1(C)CCC1)=O)=O 28503,n1(CC)nnc2cc(C(=O)NCC(O)CNC(C3COC3)=O)ccc12 28504,C1(CC)CN(C(C2CCC(C)CC2)=O)CCN1C(c1ccc([N+](=O)[O-])s1)=O 28505,C(=O)(C1=CCCOC1)NC1CCCC(C(=O)NCCCSCC)C1 28506,C=CCCC(F)(F)C(=O)NCC1CN(C(c2cnn(CCC)c2CC)=O)CCO1 28507,c1(C(=O)NCC2C(NC(c3c(OCC)cccn3)=O)C2)cc2cc(O)ccc2[nH]1 28508,c1(C(N(C2CCN(C(=O)CSC3CC3)C2)CC#C)=O)cc(Cl)n(C)n1 28509,N1(c2nc(CC)nc(Cl)c2CC)CC(NC(=O)C(O)C(C)C)C2(CCOCC2)C1 28510,C1(C(N2CCC(c3cccc(F)c3)CC2)=O)CC2CC2N1C(C1CC1F)=O 28511,Cc1nn(C)c2ncc(NC(=O)NCCCOc3c(F)cccc3F)cc12 28512,c1(CC(=O)N(C)C)ccc(C(=O)NC2COCCC2NC(c2ccns2)=O)cc1 28513,C1(O)(CCNC(C(COC)OC)=O)CCCN(C(=O)CCC(C)(C)OC)C1 28514,c1(C(=O)NC(C2CCCC2)CNC(C(CC=C)CC)=O)cccn2nccc12 28515,C1(C(C(=O)NCCC(C)N(C(=O)CC2(C)CC2)C)OCC)CC(F)(F)C1 28516,C1(C(N)=O)CC(=O)N1.C1(NC(=O)CC2(N3CCCC3)CC2)CCCN(C(C)=O)C1 28517,c1(OC)cnc(Cl)c(NC(C2CCN2Cc2ccc(C(C)(C)C)cc2)=O)n1 28518,c1(CN2C(C(=O)NC3(C(=O)OC)CCC3)C=CC2)cc(O)c(Br)cc1O 28519,c1(NC(C2(CNCc3c(C)cccc3)CC2)=O)cccc2nscc12 28520,C(=O)(CC(F)(F)F)NCC(=O)NC1(CNC(=O)COC2CCCOC2)CCOC1 28521,c1(C(=O)NC2CC(CCNC(C(CCC)C)=O)C2)cncc(N)c1C 28522,c1(OC)cc(C(=O)NC(CNC(C2CC(=C3CC3)C2)=O)C2CC2)c2occc2c1 28523,C(=O)(CC(O)c1ccccc1)NCC(C)N(C)C(C1(C)CCCC1)=O 28524,CCC(C)(C)CCCC(=O)NC1(CCNC(c2ccc(CO)cc2)=O)CCCC1 28525,c1(C(N2C3C(NC(CSCC#C)=O)CC(C3)C2)=O)cccc2nccnc12 28526,c1(C(=O)Nc2c(C(N3CC4CC4C3)=O)ccs2)n[nH]cc1[N+](=O)[O-] 28527,C(=O)(C(F)(F)F)N.CC(C(=O)NCCCN(C1COC1)C1CC1)N(C(C)=O)C 28528,CCC(C(=O)NCC1CN(C(c2ccc(C)c(CO)c2)=O)CC1(F)F)C(C)C 28529,c1(NC(C)=O)c(C(N2CCC(NC(=O)Cn3cccc3)C2C)=O)cccc1C 28530,C#CC1CN(C(=O)CCn2cccn2)CCN1C(c1cnc(O)o1)=O 28531,CN1CCC(C(=O)N2CC(CO)(NC(=O)C3=CCCC3(C)C)C2)c2ccccc21 28532,c12ccc(F)c(c1)C2N(C1C2CN(C(C3(N(C)C)CC3)=O)CC21)C.COC 28533,C1(CC)(NC(c2ccc(CNC(C34CC(OC)(C3)C4)=O)cn2)=O)CCN(C)CC1 28534,N1(C(CN(c2ccccc2)C(C)=O)=O)CCOCC(NC(C2CCCO2)=O)C1 28535,C1(CNC(CC2CC(C(=O)OC)C2)=O)CCCCN1C(=O)COCP(C)(C)=O 28536,N1(C(CCC=CC)=O)CCOC2(C1)CN(C(=O)C(C)OCCc1ccccc1)C2 28537,CC1CCC(C)(C(N2CC3(CC(NC(c4[nH]cc5c4CCC5)=O)C3)C2)=O)CC1 28538,Cc1ccnc(O)c1C(=O)NCCC1CC(N)C1 28539,n1(NCC2(CC#N)CCN(C)C2)c(=O)c(F)cn(-c2ccccc2)c1=O 28540,S(=O)(=O)(c1ccc(C)c(C)c1)NCC(N1CCC(C#CC)C1)=O 28541,C12C3CC4C1C4C3C(=O)N2.c1(CC2N(C(C3CC(O)C3)=O)CC2)ccc(Cl)o1 28542,CC1CN(C(c2cncnc2)=O)CC1NC(c1ccc(SC(F)(F)F)o1)=O 28543,Cc1ccc(O)c(C(N2CCN(C(c3nc(O)sc3C)=O)C(C(C)(C)C)C2)=O)c1 28544,CC1CCCCCN1C(=O)CSCCNC(c1cncc(F)c1)=O 28545,N1(C(c2cccc(C(C)(C)O)c2)=O)CC2(C(=O)O)CCC2(C(=O)O)C1 28546,c1(C(=O)NCC2(CNC(C(c3cncnc3)C)=O)CCC2)ncc(Cl)cc1F 28547,C1(C(N(C)CCNC(C2CCC(C(F)(F)F)CC2)=O)=O)CCc2nnc(O)n2C1 28548,C1(NC(CSC(C)C)=O)CC2CN(C(=O)CN3CC(=O)NC3=O)CC2C1 28549,C1(C(=O)NCCC2CN(C(=O)CCC3CCCCO3)C2)CC2COCC2C1 28550,CCC(CCCO)NC(=O)C(CO)NC(=O)CC(C)=C(C)C 28551,c1(CC(=O)NC(CC2CN(C(c3cc(C)oc3)=O)C2)C)cnc(Cl)cc1C 28552,C1(O)(CC(=O)N(C(C)CNC(=O)C(c2ccc(Cl)s2)C)C)CCCCCC1 28553,CC1=C(C(=O)N2C3CCC(C3)C2C(N2CC(F)(F)CC2CO)=O)CCC1 28554,c1(C(=O)NC2CC(C)(C)CN(C(c3cncs3)=O)C2)cc(F)cc2nn[nH]c12 28555,C1(NC(c2nnc(C)s2)=O)C2CC1CN(C(C1CC1C1CCCC1)=O)C2 28556,C(=O)(C(C)(C)CS(N)(=O)=O)NC1(CCNC(C2(C)CC2c2ccccc2)=O)CC1 28557,C1(O)(CCNC(c2csc(O)n2)=O)CN(C(c2ncoc2Br)=O)C1 28558,c1(C(N(CCNC(CCCC#C)=O)C)=O)cc(C)n(CC(=O)OC(C)=O)c1C 28559,CC1(C(=O)N2CCC(NC(=O)COc3cn[nH]c3)C2)COc2ccccc21 28560,C(=O)(CCS(=O)(=O)CC(C)C)N1CC(NC(Cc2cc(C)on2)=O)C(CO)CC1 28561,c1(C(=O)NCC(CC)NC(c2cnc(C3CC3)nc2O)=O)cc2n(n1)CCC2 28562,CC(Cc1cccn1C)N=c1ccnc(NC2CCC(=O)NC2)[nH]1 28563,N1(C(C(=O)C2CC2)=O)CCC(O)C2(CCN(C(c3ccn4ccnc4c3)=O)CC2)C1 28564,c1(C(=O)NC2C(CNC(c3ccn(CC)n3)=O)CC2)ccc(=O)n(CCOC)c1 28565,CC(=NO)C1CC(C(N2CC(NC(=O)CSCc3ncc[nH]3)C2)=O)C1(C)C 28566,Cc1cccnc1C(N1CC(CC(C)NC(c2cncc(C(C)(F)F)c2)=O)C1)=O 28567,N1(C(c2c(CNC(CC=CC=C)=O)n[nH]c2)=O)CCc2ccncc21 28568,Cn1nc(C(=O)NC2CC(CNC(C3(C#N)CCCO3)=O)C2)cc1Br 28569,c1(CC)ccc(Cl)c(NC(N2CCN(C(c3nocc3C)=O)CC2)=O)c1 28570,c1(C(=O)N(C(CN(C)C)(C)C)CCC(=O)NC2CC2)ccccn1 28571,C1(C(N(CC(C)O)CCNC(=O)C(C)(C)C)=O)CCn2nccc2C1 28572,c1(SC)ccncc1C(=O)NC1COCCC1NC(C12CSCC1C2)=O 28573,c1(C(=O)NCC23C(CN(C(CC=CCC)=O)C2)C3)ccc(F)c(C(F)(F)F)c1 28574,C1(CNC(C(C)c2cccs2)=O)CC(C(F)(F)F)CN1C(N)=O.n12cc(nn1)C2 28575,c1(C(=O)NCC2N(C(CC(C)C)=O)CC(C)CC2)cccc2cc[nH]c12 28576,C(CC(=O)NCC1CC2(CC2)C(=O)O1)(C(F)F)NC(CNC(C(CC)C)=O)=O 28577,c1(-n2ccc(C)n2)ccccc1C(=O)NCC(F)CNC(C1CCOCC1)=O 28578,C1(C(=O)NCC2C(NC(c3cc(C(F)(F)F)ccn3)=O)CC2)CC2(CCCC2)C1 28579,N1(C(CC(CC)C)=O)CC(F)(F)CC1CNC(=O)C(=O)Nc1nc(C)ccc1C 28580,c1(C(N(CCN(C)CC2CCC(C)(C)CC2)C)=O)occ2c1CCC2 28581,N1(C(C2C(CCC)C2)=O)CC(NC(=O)C=C2CCCCC2(C)C)C2CCCC12 28582,c1(C(=O)NC2CC(NC(C3C(C)(C)COCC3)=O)C2)ccc2cc[nH]c2n1 28583,O=C1CC(C(=O)N2CC(CNC(C3(O)CC3)=O)OC3COCC23)c2ccccc21 28584,C(C(=O)N(CC(C)(O)C1CC1)C)(C(C)OC)NC(CC1(CSC)CC1)=O 28585,CC1(NC(c2csc(Cl)n2)=O)CCN(C(C2CCCC2)=O)C1.C12CSCN1C2=O 28586,c1(OC)snc(C)c1NC(=O)NCC1CCN(C(C2CCCN2C)=O)C1 28587,C1(CC)CCC(C(=O)N(C2(C(N3CC(C(F)(F)F)C3)=O)CC2)C)CC1 28588,C1(CNC(COCC(=O)NC)=O)CN(C(=O)CCc2ccc(NC)cc2)CCO1 28589,c1(C(N(CCN(C(C(C(=O)OC)OC)=O)C)C)=O)ccc(C(F)F)c(C)c1 28590,C1(C(=O)OC(C)(C)C)CCC(C(N)=O)CC1.n12cc(nn1)CNC1CC2C1 28591,n1(SC)ncc2cc(-c3ccc(NCC(N4CCOCC4)(C)C)cn3)cnc12 28592,CCC(C(=O)NCC1CCC(NC(=O)Cc2ccc(C)o2)C1)OC1CCCCC1 28593,C#CCCCCC(=O)NC1CCN(CCNC(=O)CC2CCCS(=O)(=O)C2)CC1 28594,N1(C(C2(OCC)CCC2)=O)CCCCC1CNC(=O)C(c1cccc(F)c1)O 28595,Cc1cn2cc(C(=O)N(C3CCN(C(=O)C4=COCCC4)C3)C)sc2n1 28596,C1(C(=O)NC(C=C)CO)CCCCN1C(c1cncn1C1CC1)=O 28597,c1(C(=O)NCC(CN(C(C(C)N(C(C)=O)C)=O)C)(C)C)cccc(CS(C)=O)c1 28598,C1(CC(=O)OCC)CN(C(CC2CC2)C(=O)NC2CCC2)CC(C)O1 28599,CC1(C)CC1(S(C)(=O)=O)C(=O)NC1CC(S(C)(=O)=O)C1 28600,Cc1cnc2cc(C(N3C4CCC3CC(CNC(=O)COC(C)C)C4)=O)ccn12 28601,c1(C(=O)NCC(c2ccc(OC)cc2)O)c[nH]c2cc(-c3nn[nH]n3)cnc12 28602,C(=O)(CC(C(F)F)C(C)(C)C)NCCCN(C(c1cccc(OC)c1)C)CC 28603,c1(C(=O)NC2(CCCNC(CCOCC)=O)CC2)c[nH]ccc1=O 28604,C1(C(=O)NC2(CO)CC(CO)C2)(CNC(C2C(OC)CCC2)=O)CC12CCC2 28605,C1(C(=O)NC(C)(C)CNC(c2[nH]ccc2-c2ccccc2)=O)CCC2(CCC2)O1 28606,C(C)(C(=O)N(C(C)CO)C)N(C(=O)C=CCC1CCC1)CC 28607,c1(C(=O)NCC2(O)CCCN(C(C(C)n3ccnn3)=O)C2)ccc(N)c(Cl)c1O 28608,c1(C(=O)NC(C)CC(F)(F)F)cc(NCC=CCO)ccc1Cl 28609,C(=O)(CC(CC)CC(F)(F)F)NCC1CCCCN(C(CC(=C)C)=O)C1 28610,N1(C(C=COCC)=O)CCCC2(CCC(NC(c3cc(C)c(C)nc3O)=O)C2)C1 28611,n1(CC)nccc1C(C(=O)NC1CCOCC1)N(C)C(C1CCCC1)C 28612,c1(C(=O)NC2CC3(C(NC(CCCC4C(C)C4)=O)C3)C2)cccc2c1C(=O)NC2 28613,Cc1cc2[nH]c(C(=O)NCC(C3CC3)N(C)C(C34CC(C3)C4)=O)cc2s1 28614,C1(NC(c2c(CC)ccs2)=O)CC2CC(NC(c3cnc(O)s3)=O)CC2C1 28615,c1(NC(C2C(NCc3c(C)noc3C)CCC2)=O)nc(Cl)ccc1I 28616,C12(CC(=O)NCC3C(CNC(CCCCCSC)=O)C3)CCC(CC1)C2(C)C 28617,N1(C(c2n[nH]c(C)c2O)=O)CCc2cc(CNC(c3csc(O)n3)=O)ccc2C1 28618,N1(C(Cc2c(C)ccc(C)c2)=O)CC2CCC(C1)C2CC(N1CCC(C)C1)=O 28619,c1(C(=O)NCC2(C)C(C)CN(C(=O)C=Cc3cocn3)C2)nnn2c1CCCC2 28620,CC1CN(C(c2nc(C3CC3)cs2)=O)CC(CCNC(=O)COCC(F)F)O1 28621,C1(C(N2CCOC(CCCNC(C3CC3C(F)F)=O)C2)=O)(OC)CCC(C)CC1 28622,Cc1ccc2c(c1)CC(C(=O)NCC(C)N(C(=O)CCSc1nccn1C)C)S2 28623,N1(C(C2C3(CC(NC(CC(CC(C)C)C)=O)C3)C2)=O)CC2C(=O)NC(=O)C2C1 28624,Cc1sc(C(N2CCC(OCCNC(=O)C(CO)OC)C2)=O)c(C)c1C 28625,N1(C(CCC=CC)=O)CCOC(C)C1C(=O)NC(C)C(=O)N(C)CC 28626,C(=O)(CCCCC(C(F)(F)F)NC1CC(SC)C1)OC 28627,C=C(C)C(CC(=O)N1CCC(CN(C)C(c2cnc(C)cc2Cl)=O)CC1)OCC 28628,N1(C(Cn2c(C)c(Cl)cn2)=O)CCC2(CC1)CC2NC(=O)C(C)CC(C)C 28629,N1(C(c2cc(Br)co2)=O)CCC2(CO)CN(C(c3ccnc(O)c3)=O)CC2C1 28630,CCC(CC(=O)NC(C)(C)C(C)CC(=O)N1CC(CC)(CC)C1)C(F)F 28631,c1(C(=O)NC(CCCC)CNC(=O)CNS(=O)(=O)NC)coc2c1C(=O)NCC2 28632,N1(C(CCC=CC)=O)CCN(C(=O)C(C)(C)CCF)CC1c1ncc[nH]1 28633,C1(C(=O)NC2(CNC(C(=Cc3ccccc3)OC)=O)CC2)CCOC2(CCC2)C1 28634,C(C)(CNC(c1nnsc1C)=O)(CC(C)C)NC(CCCC)=O 28635,Cc1c(C(=O)NC(C)(CNC(=O)CCC2CC2(C)C)CO)nnn1C(C)C 28636,c1(C(=O)OC)ccc(CNCC2CCCC2N)cc1Cl 28637,c1(C(=O)NC(C)(Cc2ccccc2)C(F)(F)F)ccc([N+](=O)[O-])cn1 28638,C1(C(=O)NC2C(COC)(CO)C2)CN(CO)CC12CCC2.C1(C=O)CC(CO)(CO)C1 28639,N1(C(=O)NC2CC(c3ccc(Br)cc3)C2)CCC12CC1CCC2C1 28640,C1(C)(C(N2CCC(NC(CCC(CC)OC)=O)CC2)=O)CC2CCC(C1)S2(=O)=O 28641,c1(C(=O)NC2(CNC(c3c[nH]c(=NC)s3)=O)CC2)ccc2c(c1)C(=O)N(C)C2 28642,C(=O)(CCCC(=O)OC(C)(C)C)NC1CCCC(NC(C=CSC)=O)C1 28643,c1(C(C)C)ccc(CC(=O)NCC(C2CC2)N(C(=O)CC2CCCCO2)C)cc1 28644,C1(NC(c2cc(C)c(C)[nH]2)=O)CS(=O)(=O)C12CCN(C(=O)C(C)(Cl)CCl)CC2 28645,c1(C(=O)NC2CC(OC)CN(C(c3c(Cl)n[nH]c3C)=O)C2)c(C)cc(C)nc1O 28646,c1(-c2ccc(C(=O)NCCC)s2)ccc2c(C(=O)NCC3CCO3)cnn2c1 28647,c1(C(C(=O)NCCCC)NC(C2CCN2C(C)(C)C)=O)cccnc1 28648,C(=O)(CC(CC)OC)NC1(C(=O)NCC(C=C)(C)C)CSC1 28649,C1(NC(C(CCC)O)=O)CCN(C(c2cc(NC(C)=O)ccc2C)=O)C12CC2 28650,c1(OCC(=O)NCC2(C)CC(NC(C3(CC#C)CC3)=O)C2)ccc(O)cc1 28651,CCCCC(CC)C(=O)NCC(O)CC(N1CCC2(CSC2)C1)=O 28652,C1(C)(CNC(c2c(C)sc(Br)c2)=O)CCCN(C(=O)CC2CCC2)C1 28653,N1(CCC)C(=O)CCC1C(=O)NCC(C)(C)CN(C(=O)Cn1nc(C)nc1C)C 28654,c1(CN(CC=C)CC=C)cn(CCC2CN(C(c3cc(C)cs3)=O)C2)nn1 28655,Cc1c(CS(N2CCCC(OC3CCC3)C2)(=O)=O)cccc1Br 28656,CC1CN(C(c2ccn(C)c(=O)c2)=O)C(C)CN1C(C1CCNC1=O)=O 28657,C1(CCC#C)CCCN(C(c2ncoc2CNC(C2CCOC2=O)=O)=O)C1 28658,C1(CC)(NC(=O)C(F)F)CCN(C(=O)C(C)(C)C)CC1 28659,c1(C(N2C(C(C)C)CN(C(=O)C(C)n3ccnc3)CC2)=O)ccc([N+](=O)[O-])cn1 28660,CCC(CC)CC(F)C(=O)N1CC(C(N2CC3CCC=CC23)=O)(SC)C1 28661,c1(N2CC(CNC(c3cn(CCOC)nc3C)=O)(OCC)C2)ncnc(C)c1F 28662,c1(C(=O)NC2C(F)CCN(C(c3cnn(CC)c3C)=O)C2)sc2cncn2c1C 28663,c1(C(=O)NC2CCN(C(C=NOC)=O)C23CC3)cccc2[nH]ncc12 28664,c1(COC(c2cccc(C(F)C(F)(F)F)n2)=O)cc(Cl)ccc1F 28665,CC1(C)C2CCC(NC(=O)NC(C3CCCCC3)Cc3ccccc3)C1C2 28666,C(=O)(C1=CCC2CCC1N2C(=O)COC)N(C(CC)COC)C 28667,n1(CC(=O)N(CC(C)NC(C2CCCCC2O)=O)CC)nc(C)c([N+](=O)[O-])c1C 28668,C1(NC(c2c(OCC=C)cccn2)=O)CN(C(c2cc[nH]c2C)=O)CC2(CC2)C1 28669,N1(C(c2c(C)nn[nH]2)=O)CCC(C)(O)C1C(=O)N(C)Cc1ccsc1 28670,c1(C(=O)NCC(C)CN(C(=O)C(C)Oc2ccc(Cl)cc2)C)cccc(CO)n1 28671,CC(C)CC(F)C(=O)NC1CCC(F)(CNC(c2ccc(Br)cc2)=O)C1 28672,N1(C(c2cccc(C)c2F)=O)CCCC(C2CCN(C(C3CCOCC3)=O)C2)C1 28673,C1(NC(COCCC#C)=O)CC(NC(C2CC(c3cccc(Cl)c3)C2)=O)CC1O 28674,C1(C(=O)OC)CC(F)(F)CN1C(c1cc(C)c(C)s1)C(=O)NC(C)C 28675,C1(CNC(C(CC)(C)C)=O)C2CCCC1N(C(c1cc(C#N)no1)=O)C2 28676,C1(NC(CC(CC=C)(C)C)=O)CC2(CCC(CNC(C3C4COCC34)=O)CC2)C1 28677,n1(-c2cn(C)nc2)cc(C#N)cc1Sc1cc(Cl)cc(Br)c1 28678,CCCC(C)(C)CC(=O)C1CCC1O.c1(C(C)N)cn(CCOC)nn1 28679,N1(C(C(C)OCC2CC2)=O)CC(CNC(C2(C)CCN(C)C2=O)=O)CC(C)C1 28680,C(=O)(C(O)CC(C)(C)C)NCC(C)C(=O)NC(c1nncs1)C 28681,c1(C(N(C2CCN(C(c3cnsn3)=O)C2)CCC)=O)cc(Cl)cc(Cl)c1F 28682,c1(OC)nccc2c(C(N3CC4C(NC(c5cc(C)oc5C)=O)C4C3)=O)c[nH]c12 28683,N1(C(CCc2ncc(C)[nH]2)=O)CCCCC(NC(c2n[nH]c(C)c2F)=O)C1 28684,C12(C(CO)NC(=O)NC(C(C)C)C3CC3)CC3CC(CC(C3)C1)C2 28685,c1(C(C(=O)NC(CNC(Cc2cc(CC)no2)=O)C)O)ccccc1F 28686,CC1(CC(N2CC(CO)(NC(c3coc(Br)c3)=O)C2)=O)CCS(=O)(=O)N1 28687,C(C1CCCN1C)=CC(N1CC(CC(C)NC(C2(c3ccccn3)CC2)=O)C1)=O 28688,CC(C)(C(=O)N1CCC(NC(c2cc(Br)sn2)=O)C1)c1cc[nH]n1 28689,C12(NC(CCOC3(C)CC3)=O)CCC(CNC(=O)C=Cc3ccncn3)(C1)OC2 28690,c1(C(N2CC(C)C(CNC(C3COC3)=O)C2)=O)ccc2c(Br)cncc2c1 28691,c1(C(=O)NCC2N(C(CSCCOC)=O)CCCC2)cccn2nncc12 28692,N1(C(C=CCCC)=O)CCCC(C(=O)NCc2conc2C)CC1 28693,c1(C(=O)NC2CN(C(c3cc(Cl)cnc3Cl)=O)CC2F)ccc2nonc2c1 28694,C1(NC(=O)Cc2nc(C3CC3)cs2)CN(C(c2cc(Cl)ns2)=O)CC12CCC2 28695,C(=O)(CCCC=C)N(C)C.C1CCCCN(CC#C)CCC(=O)N1C 28696,c1(C(=O)NC(CC)CNC(=O)CC2CCC(=O)N2)cc(C)c(F)cc1O 28697,Cc1ccc(C(=O)NC(C)(CNC(=O)C(F)F)C(C)C)c(=O)n1C 28698,c1(SCC(=O)NCC2CCN(C(c3c(C(C)(C)C)csc3)=O)C2)ccccc1F 28699,c1(C(=O)NC2CC(NC(C(c3scc(C)n3)C)=O)C2)cc2nccnc2cc1C 28700,c1(OC)ccccc1C(C)C(=O)NC(C)CC(C)NC(c1nocc1C)=O 28701,c1(CC(=O)N(CC(CC)NC(=O)CN2CCC(C)(O)C2)CC)ccc(F)cc1 28702,c1(CN(C(c2ccc(Cl)cc2)CCSCC)C)nnc2n1CCC2 28703,c1(C(=O)NCCCNC(c2ccc(OC(F)F)cc2)=O)cc(F)c(F)c(Cl)c1F 28704,c1(OC)ccc(CNC2CC(Oc3ccccc3)C2)c(OC(F)(F)F)c1 28705,C1CC2CCCCCC12.n1(CC(C)(C)NC(CCN(C(C)=O)CC)=O)ccc(C)n1 28706,C1(CNC(c2cc(Br)cs2)=O)COCCN1C(C1C2CCCOC12)=O 28707,N1(C(Cn2ncc(CC)c2)=O)CC(NC(C2(CC)CCCC2O)=O)C(CO)C1 28708,c1(OC)ccc(C(C)CNC(C2CCC2(C)C)=O)cc1 28709,c1(C(N2CCC(NC(CSCCCC)=O)C2C)=O)cc2cccnc2cc1F 28710,c1(C(N(CC(C)NC(=O)COCC2(F)CC2)CC)=O)c(F)cc(OC)cc1F 28711,c1(C(NOCC2(C)CC2)=O)cccnc1NC(=O)CC1CC(O)C1(C)C 28712,CC1CCC(C(=O)N(CCNC(c2cncc(CO)c2)=O)C2CC2)CC1 28713,C1(C(F)(F)F)(OC)CC(NC(=O)N(C2CS(=O)(=O)C2)C)C1 28714,Cc1csc(=O)n1COC(c1ccc(CC2CCC3CC23)cc1)=O 28715,C1(CCOC)CN(C(=O)CCc2ccc(OC(C)C)cc2)CCN1CC#N 28716,N12CCN(C(CCl)C1)Cc1cccnc1C2=O.C1(CN)CCC(=O)N1 28717,CC(C)CCC(=O)NC(c1ccccc1F)CNC(c1ccco1)=O 28718,N1(C(c2cc(C)nn2C)=O)CCC2CC1CN(C(c1cnc(C)s1)=O)C2 28719,Cc1cc(O)c(C(=O)NC(C2(O)CCN(C(=O)CN3CCC(C)C3)CC2)C)nn1 28720,CCC(CCC(=O)NCC1(C)CC1(C)C)NC(C1(Cl)CC1C(C)=O)=O 28721,C1(C(N2C(CC(=O)NC(CSCC)CO)CC(O)C2)=O)CCC(O)CN1C 28722,C1(N(C)C)CC2(CCC(CNC(C3CCC4CCCCN4C3)=O)CC2)C1 28723,N1(C(C2OCC(C)C2)=O)CCC(C)C(NC(c2ccn(CCF)n2)=O)C1C 28724,c1(C(N(CCNC(C(C)OC)=O)C2CC2)=O)csc2ccc(F)cc12 28725,N1(C(C2=CC(C)(CC)C2)=O)CCN(C(=O)CCCC(C)=O)CC2(CC2)C1 28726,n1(CC)nc(C(C)C)cc1C(=O)N(CC(C)NC(c1cc(C)c(Cl)s1)=O)C 28727,c1(C(=O)NCC(CNC(C(c2ccccc2Cl)OC)=O)O)nccc2nn[nH]c12 28728,CCCC(F)C(=O)NC(COC)CC(=O)NCC1(CN(C)C)CCC1 28729,Cc1nnc(O)c(C(N2CC(NC(=O)CCCN=[N+]=[N-])C(C)C2)=O)c1C 28730,N1(C(C(C=CC)O)=O)CCC(CO)(CNC(C2(OC)CCC(C)(C)C2)=O)CC1 28731,C=CCCCC(=O)NCCOCCN(C)C(c1cnc(SC)n1C)=O 28732,c1(C(N(C2CCN(C(=O)CC3CCCO3)C2)C)=O)cnc2n1CCCC2 28733,c1(C(=O)NCC(CNC(c2cc(C)no2)=O)S(C)(=O)=O)ccn2ncnc2c1 28734,C(=O)(C(O)C(C)CC)NCc1cc(C(N2CCC(C(CC)C)CC2)=O)on1 28735,C#CCS(=O)(=O)CCNC(=O)C(=O)NC1(C)CC=CCO1 28736,C(=O)(C(=O)C(C)(C)C)NCC1(OC)CCN(C(=O)CCn2ccccc2=O)C1 28737,C1(CNC(C2C(C)N(C)CC2)=O)CN(C(c2cc(C(F)(F)F)ns2)=O)CC1(C)C 28738,c1(NC(C2CC(NC(CNC(CCC)=O)=O)C2(C)C)=O)n[nH]c2ccccc12 28739,c1(OC)nn(C)cc1C(=O)NCC12CC(CN1C(c1csnn1)=O)C2 28740,C(=O)(C(O)(C(C)C)C(F)(F)F)NC1CN(C(CC(=C)Br)=O)C(C)(C)C1 28741,CCC(CNC(=O)C(=O)Nc1ccn(C)n1)CC(F)(F)F 28742,N1(C(c2cc(CCC)[nH]n2)=O)CC(C)(CNC(=O)CS(=O)CC)CC1(C)C 28743,c1(CN2C(NC3(c4ccccc4)CC3)CCCC2)ccc2[nH]nc(Cl)c2c1 28744,N1(C(COCC(=O)N(C)C2CC2)=O)CC2CC(O)C1C2NC(=O)CN1CCCCC1 28745,N1(C(CN2CCN(C)C(=O)C2)=O)CCCC2(CCN(C(=O)C(F)(F)C(F)F)C2)C1 28746,C(=O)(C1=CCCCO1)NC1C(C)(C)C(CC(=O)Nc2ccc(C3CC3)nc2)C1 28747,c1(C(=O)NC2C(NC(C3(C(=O)OCC)CC3)=O)C2)occc1C 28748,N1(C(C2C3COCC23)=O)CCCC(C(=O)NC(c2ccccc2F)CO)(CO)C1 28749,C(=O)(CCC(C)S(C)(=O)=O)N(C1C2CN(C(c3cc(C)c(C)s3)=O)CC21)C 28750,C1(COC)(CNC(c2cnn[nH]2)=O)CCN(C(c2nc(C(F)(F)F)ns2)=O)CC1 28751,c1(OCC)ccc(OCC(=O)NCCN(C(=O)C(C)=CC2CC2)C)cc1 28752,C(=O)(C(CC(C)CC)NC(c1cc(OC)no1)=O)Nc1cnc(CCC)nc1 28753,N1(C(C2C3CN(S(=O)(=O)C4CCOCC4)CC23)=O)CCc2ccc(F)cc2C1 28754,C(=O)(C(C(C)(C)C)c1ccccc1)NC1CC(NC(c2cn(COC)nc2)=O)C1 28755,C(=O)(CC(C)C(C)(C)C)N1CC=C(C(=O)N2CCCC(CC=C)C2)C1 28756,Cc1nc2ncc(C(N3CC4C(NC(C5CC(C)(C)CO5)=O)C4C3)=O)cc2o1 28757,C12CC(O)C1NC2=O.O=C(COC1CC1)OCC1(O)CC1 28758,c1(C(=O)NC2C=CCN(C(=O)CCCN3CCOCC3)C2)csc2ccccc12 28759,N1(C(c2c(C(=O)OC)coc2)=O)CCN(C(c2n[nH]c3c2CCC3)=O)C2CC12 28760,CC(C)CS(=O)(=O)CC(=O)N1CC=CC1CNC(c1ccccc1)=O 28761,C(=O)(CCC(c1ccccc1)N(C)C)NC(C1CCN(C(=O)C(C)(C)F)CC1)C 28762,CC1(C)CC(C(=O)NC2CC(NC(c3ccc(O)nc3Cl)=O)C(O)C2)CCO1 28763,N1(C(=O)NCCCC#C)Cc2nnc(C)n2CC1C(=O)OC 28764,c1(C(=O)NCCN(CCC)C(c2cccc(CF)c2)=O)nn(C)c2c1CCC2 28765,N1(C(CSSC)=O)CCN(c2cc(CNC(=O)CCC(F)F)ccn2)CC1 28766,n1(CCNC(=O)C(O)Cc2cnc[nH]2)cc2ccccc2n1 28767,c1(OC)ccc(C)c(NC(C2COCCN2C(c2ccncc2Cl)=O)=O)c1 28768,C12(CNC(C=CC(C)(C)C)=O)CN(C(=O)C=CSc3nc[nH]n3)CC(F)(C1)C2 28769,CC(C)CC(C(=O)NCCC(O)CO)NC(C1C2CCC(F)C12)=O 28770,C1(C(N(CCCNC(C2CCN(C)C2)=O)CC)=O)CC12CC(C)(C)C2 28771,C1(NC(C(CSC)OC)=O)CCN(C(=O)CC2(C#N)CC2)C1(C)C 28772,N1(C(C2C(NC(c3c(C)nc(O)cc3)=O)CCOC2)=O)CC(C)C12CCOCC2 28773,c1(NC(CC2CCN(Cc3c(C)n[nH]c3)C2)=O)ccc(C(C)C)cc1 28774,N1(C(c2c(OC)nsc2)C(=O)NC2CC2)CCCC(C)(O)CC1 28775,CC(Cl)(Cl)C(=O)NCC(C1CCOC1)NC(=O)C=Cc1cc[nH]n1 28776,C1(CNC(C(COCC)C)=O)CN(C(=O)Cc2cccnc2Cl)CC1O 28777,c1(CC)nc(C)c(C(N2CC(OC)C(Cn3cc(COCC(=O)O)nn3)C2)=O)s1 28778,CCCC(C(=O)NCc1cc(C(N2CCC23CC(C)(CO)C3)=O)ccn1)C(C)C 28779,c1(C(=O)NC(CN(C(c2cc(C)[nH]c2)=O)C)C)cc(C#N)ccc1C 28780,c1(CNC(C=C)(C)CC)cc(C)c(-c2ccccc2OC)s1 28781,c1(C(N2CC(CC(C)NC(CCCNC(C)=O)=O)C2)=O)ccc(C(N)=O)cn1 28782,C1(NC(CSCC#C)=O)C(CNC(c2cc3ccncc3s2)=O)CCC12CCC2 28783,c1(C(C(=O)NCC(C)N(C(Cc2cnc(C)[nH]2)=O)C)O)ccc(Cl)c(F)c1 28784,N1(C(CC=CC(C)(C)C)=O)CC(NC(c2cc(C3CC3)no2)=O)CC(O)C1 28785,C1(C2CCC2)(C(=O)NCC2N(C(=O)Cc3ccccc3F)CC2)CC1(F)F 28786,c1(C(=O)NCc2nnc(SC)s2)ccc2c(c1Cl)OC(F)(F)O2 28787,N1(C(c2[nH]cc(CC)c2)=O)CC(CC(=O)NCC2C(C)(C)C2(C)C)C2(CC2)C1 28788,C1(c2nnnn2C(C)(C)C)(NCC2(SC)CCCC2)CCCC2CC12 28789,C(=O)(C(F)C(C)CNC(c1cc(C)cc(O)c1)=O)NC(CCOC)(C)C 28790,CCC(C(=O)NCC1(F)CC(NC(C2(C)COC2)=O)C1)Nc1ccccc1 28791,Cc1cc(F)cc(C)c1C(=O)NC1CC(N(C)C(C2CC(C)(C(C)(C)C)C2)=O)C1 28792,C=CCCCCCN(C(=O)CC1CCCN1C(=O)C(O)C1CCC1)C 28793,C(CCCCC(=O)N(CCCCN(C)C(C1CCCN(C(C)C)C1)=O)C)OC 28794,C1(NC(C(CCSC)O)=O)CCC2(CCN(C(C3(CCN(C)C)CC3)=O)C2)C1 28795,Cc1cccc(C(=O)NC2CCCCC2NC(=O)COc2ccsc2)c1F 28796,C1(O)(CC(=O)N(C2CCN(C(CC(C)OC)=O)CC2)CC2CC2)COC(C)(C)C1 28797,O=C(C1=CCCO1)NCCN(C(=O)C(F)(F)c1cnccn1)C1CC1 28798,c1(-c2nnc(N3CC(C)(C)SCC3)n2Cc2ccccn2)ccc2ccoc2c1 28799,N1(C(CCc2n(C)ccn2)=O)C(C(=O)NC2CCOC2)CC2CCCC12 28800,c1(C(C(=O)NC2CN(C(C)=O)C2)C)cccc(Cl)c1.C12C(C1C)C(=O)N2 28801,C1(NC(C=C(C)C)=O)CCC(N(C)C(c2cc(-c3cccs3)[nH]n2)=O)CC1 28802,c1(OC)cc(C(=O)NC2CCCC2NC(C2(F)CC2)=O)cnc1O 28803,C(=O)(CCCCCNC(C1(C(=O)NC2CC2)CC1)=O)N(CC(CN(C)C)O)C 28804,c1(C(N2CCCCC(N(C(=O)COCCF)C)C2)=O)cncc2sccc12 28805,c1(OC)c(C(=O)N(C(C)CC2CN(C(C3CCC3OC)=O)C2)CC)cccc1Br 28806,C1(C=O)CCC(O)CN1C(c1sccc1C#N)=O.CCCCC1(CO)CC1 28807,C(=O)(N=c1[nH]oc2c1CC(N(c1cccnn1)C(C)(C)C)CC2)c1nn(C)nc1Br 28808,C(CCCCC(=O)Nc1ccc(Cl)nc1C)N(C(c1c(C#C)c[nH]n1)=O)C 28809,C12(NC(CC(CC)O)=O)CCCCCC1N(C(=O)CC(C)(O)COC)CC2 28810,N1(c2nnc(C#N)s2)CCC2(NC(c3ncc(Cl)s3)=O)CCCC12 28811,Cc1cc(C(N2CC3CC(CNC(c4cnc(O)o4)=O)C3C2)=O)n2nccc2n1 28812,c1(NC(C2N(Cc3cccc(OC)c3Cl)CCC2)=O)nc(Cl)c(C)c(Cl)n1 28813,N1(C(C(CCSC)NC(C2CCCCCN2C)=O)=O)CC2CCCCC12C 28814,C1(c2n(CC)nnn2)(NC(c2ccc(SC)nc2)C)CCCC2(CCCCC2)C1 28815,C(C(=O)NCC1CCC(F)(F)C1)(C(C)(C)C)NC(c1c(CC)cno1)=O 28816,C1(C(=O)NC2(CO)CCCNC2)CC12CCOc1ccccc12 28817,N1(C(=O)CCc2ccc(O)cc2)CCC2CCCC12CNC(C1(F)CCCC1)=O 28818,C1(NC(CC2N(C)CCCC2)=O)C2CC1CN(C(=O)C=CC(=O)NC1CC1)C2 28819,C1(O)(CN(C(c2c(CC)occ2C)=O)C)CCCN(C(=O)C(F)(F)C(F)F)C1 28820,N1(C(C2CC(SC)C2)=O)CCC2CN(C(c3cnc4ccccn34)=O)C2C1 28821,c1(C(=O)NC2CC(CCNC(COC)=O)C2)cnoc1-c1ccccc1 28822,c1(C(N(C2(CNC(C3CC(C(F)(F)F)CO3)=O)CC2)C)=O)ccnc2c1ccn2C 28823,c1(CNC(CC(=O)NCCCC)Cc2cccs2)cccc(F)c1I 28824,C1(CC=C)(NC(=O)CS(=O)(=O)CCO)CC2CCC(C1)N2C(=O)C(C)CF 28825,C1(OCC)CC(NC(C2CC23CCC(F)(F)CC3)=O)C12CCCCC2 28826,C(=O)(C1=CC2(CCOCC2)C1)NCC(C(C(C)C)C)NC(c1c[nH]ccc1=O)=O 28827,N1(C(C2SCCS2)=O)CCN(C(c2ccnc3c2CCO3)=O)C2CCCCC2C1 28828,N1(C(CC(=O)OC(C)(C)C)=O)CC(C(=O)NCC(F)CO)CC12CCC2 28829,C1(O)(CCNC(c2c(CC)c[nH]n2)=O)CCCN(C(C2CCCC2CC)=O)C1 28830,CCCCC(C(=O)N1CC(O)(C2CC2)C1)NC(C1CC(O)C1)=O 28831,c1(C(N(C2CCC(NC(CCC(=O)N(C)C)=O)C2)C)=O)oc2ccccc2c1Cl 28832,c1(OC)nn(C)cc1C(N1CC(CNC(=O)Cn2nc(C)oc2=O)CC1C)=O 28833,C#CCC(C(=O)N1CCCC(CN(C)C(c2cnn(C3CCCC3)c2)=O)C1)C1CC1 28834,C12(C(=O)NC3C(C)(NC(C4C(CC)CCO4)=O)CCC3)CC=CCN1CCC2 28835,N#Cc1cccc(-c2cn(CCCCNC(=O)Cc3nc[nH]n3)nn2)c1 28836,C1(CC(=O)NC(CCCNC(c2c(CC)nco2)=O)C)CCC(F)(F)CC1 28837,C(=O)(CCCC(F)(F)F)NCC(C)NC(C(c1ccc(OC)cc1)C)=O 28838,C(=O)(C1CCCc2nn(C)cc21)NCC(C)NC(=O)CCc1c(F)cccc1Cl 28839,C1(F)(C(N2CCN(CCCCCNC(C=C(C)Cl)=O)CC2)=O)C2CCCCC12 28840,Cc1cc(C(=O)N(C2CN(C(=O)C(N3CCCC3)C3CC3)C2)C)cc(NC2CC2)n1 28841,c1(C(C(=O)NC(C2(CNCC3CC3)CC2)C)C)cn(C)c2ccccc12 28842,N1(C(C(C)OCC)=O)CC2CC(NC(c3cc(C(C)C)[nH]n3)=O)CC2C1 28843,Cc1cc(N)cnc1C(N1CCOC(C(C)NC(=O)C=Cc2ccsc2)C1)=O 28844,N1(C(C2(C#C)CC2)=O)CC2(CC(NC(=O)C(CC)N(C)C)C2)C1 28845,C(CNC(=O)CNC(C)=O)(C(C)(C)C)NC(C1(COC)COC1)=O 28846,C1(C(=O)Nc2cc(CCC)n[nH]2)COCC1(C)C 28847,CC1CCN(C(c2ccc(Cl)cc2N)=O)CC1NC(=O)CSc1ccccc1 28848,C=CC1(CNC(=O)NCCN(C)C(C)C)CCC1 28849,C12(CNC(C(C)CC(N)=O)=O)CCC(CN(C(c3cc4cccnc4[nH]3)=O)C1)C2 28850,N1(C2CCN(CCC)CC2)CCN(C(c2cccnc2)=O)C(=O)C1 28851,C=CCC(CC)C(=O)NC(C(=O)NC1CNC(=O)C1)c1ccoc1 28852,N1(C(CC2OCC(C(N)=O)OC2)=O)CCC2(CCN(C(=O)CNC=O)CC2)C1 28853,C(CCOCCO)(C(=O)NCC(C)C#N)NC(CSCC#C)=O 28854,N1(C(c2cn(C)nc2)=O)CC2CC(NC(C3CC4(CCCO4)C3)=O)C1C2 28855,Cc1nccc(C(=O)NC2C3CN(C(c4c(Cl)nsc4Cl)=O)CC23)c1O 28856,C#Cc1ccc(C(N2CCN(C(=O)Cc3ccoc3C)C3CC23)=O)cc1F 28857,CC1=NOC(=O)C1CC(=O)NCC1(CNC(C2(O)CC(F)(F)C2)=O)CC1 28858,N1(C(c2c(CNC(c3cc(CC)n(C)n3)=O)c[nH]n2)=O)CC2CC1CN2C(C)C 28859,C(=O)(C#CC1CCOCC1)NC(C1CCCCC1)C(=O)NC1C(C)C1C 28860,c1(C(N2CC(C(C)NC(c3ccc[nH]3)=O)C2)C(N)=O)ccc(Br)cc1 28861,N1(C(C(N2CCCC(O)C2)C)=O)C2CCCC1CN(C(c1ccno1)=O)C2 28862,C1(N(N2CCC(C=O)CC2)C)CS(=O)(=O)CC1O.n1(CC)cc(CCC(C)(C)O)nn1 28863,C#Cc1cccc(C(=O)NC(CCC)CCCNC(C2CC(C)(C)CN2C)=O)c1Cl 28864,N1(C(=O)N(C2CCC(O)C2)C(c2ncc(Br)cn2)C)CCC2(CO)CCCC12 28865,c1(NC(c2n(CCC)nnn2)c2ccc(Cl)s2)ccc(-c2ncco2)cc1OC 28866,Cc1cccc(C(N2CC(NC(=O)C(C(C)(C)C)NC(N)=O)C(C)C2)=O)c1N 28867,c1(C(=O)NC(C#C)C2CC2)cccc(CNC(C2CC3(CC3)CO2)=O)n1 28868,N1(CC(CCC)O)CCOc2cccc(OC)c21 28869,C1(CC(=O)NC2COCC2C(=O)NCCc2ccccc2)CCC=CCC1 28870,C=C(C)CC(C(=O)N1CC(OCCF)C1)NC(=O)Cc1nocc1C 28871,C(=O)(CC(CC)c1cn[nH]c1)N(CCN(C(C(=O)NCC)=O)C)C(C)C 28872,C1(NCC(C)C2CC2)CC2CCCCC2C1 28873,CN1CCC(O)(CNC(c2cc(CNC(C3(C)CC3(C)C)=O)cs2)=O)C1 28874,N1(C(C2(C)CCCC(=O)C2)=O)CCC(C)(C)C(NC(c2ccc(F)s2)=O)C1 28875,C12CN(CCCO1)CC2.Cc1ccc(C)n1C(=O)NCC1CC[Si](C)(C)C1 28876,c1(CCC)cc(C(=O)N(CC(O)CNC(=O)C=Cc2cnsc2)C)c(C)o1 28877,c1(C(N(CC2N(CC)CCC2)CC2(c3ccccc3)CCC2)=O)sc(Br)c(C)c1C 28878,Cc1cnc(NCC2(C)CCN(C(=O)CCC(C)(C)C)C2)c([N+](=O)[O-])c1 28879,c1(OC)ccc(Cl)c(C(=O)NC2CN(C(c3cc4n(n3)CCC4)=O)C3CC23)c1 28880,C1(N(C(=O)Cc2cn(C)cn2)CC)CCCN(C(c2cnn(C)c2Cl)=O)C1 28881,N1(CC)CC(NC(=O)N(CC(O)C2CCC2)C2CC2)C(C)C1 28882,c1(NC(C(CC2CC2)NC(c2cn(C3CC3)nn2)=O)=O)ccc(CO)nc1 28883,C1(CNC(c2c(C)nns2)=O)CC(C)N(C(C2CCC(NC(N)=O)CC2)=O)C1 28884,C1(C(=O)NCC2C(CNC(CCCC(N)=O)=O)C2)C2C3CC4C1C1C2CC3C41 28885,c1(CC)ccccc1C(=O)NCCNC(C1CCN(C(C2CCCC2)=O)CC1)=O 28886,CC1(C)CCC(C(N2CCOCC2CCNC(C2COCCN2C=O)=O)=O)CC1 28887,C(=O)(CCCC(=O)N1CC(NC(=O)CCCCCNC(C)=O)C(C)C1)NCC 28888,N1(C(c2nc(CC(C)C)sc2)=O)CC2CC(NC(=O)CCN3CCCC3=O)C2C1 28889,N1(C(=O)NCc2ccc(C)c(C)c2)CCc2cc(-c3cccc(F)n3)ccc2C1 28890,C(=O)(CCC(C)S(C)(=O)=O)N(CCn1cc(CN(C)CCO)nn1)CC 28891,CCC(C(=O)NCC1(OC)CN(C(=O)CC(C)F)C1)N(C)C 28892,Cc1sc(NC(=O)C2CC2)c(C(=O)N(C(C2CCCN2C(=O)CC#N)C)CO)c1C 28893,c1(-c2cn(C(C(=O)N(C3CC3c3cncnc3)C(C)=O)C)nn2)cc(C)ccn1 28894,C1(C(=O)NCC2CCCC(CNC(c3ccc(Cl)o3)=O)C2)CC12CCOCC2 28895,CS(=O)(=O)CC(=O)NC1CCC1CNC(=O)CC1COCCO1 28896,c1(C(=O)NC(CCOC)CNC(C2CC2C(C)(F)F)=O)cnc(C)cc1C 28897,Cc1cc(C(=O)NCCCN(CCCCNC(C2CC=CCO2)=O)C)sc1C 28898,C1(N(C(CS(=O)(=O)NC)=O)C)CN(C(C2CC(F)(F)C2)=O)CCC1O 28899,C1(NC(COCCC=C)=O)CC(C2CCN(C(=O)C=Cc3cccc(C)c3)C2)C1 28900,c1(C(C)N(C)CC2CCN(C(=O)OC(C)(C)C)C2)nccn1C(F)F 28901,c1(C(=O)NCCC2(C(N(C(C#C)C)C)=O)CC2)ccc(F)s1 28902,c1(C(N(CCCN(C)C(C2CSCCS2)=O)C)=O)ccc(-n2cccn2)nc1 28903,N1(C(Cc2cncc(OC)c2)=O)CCC(NC(=O)CCc2nc[nH]n2)C(O)C1 28904,C1(n2ncc(C(N(C3CCCN(C(=O)C(C)(F)F)C3)CC)=O)c2)CCC(C)CC1 28905,c1(CC)ccc(C(C)=CC(=O)NCC(C)(C)NC(C2COC(C)(C)CO2)=O)cc1 28906,C(=O)(C1=CCCN(C(=O)CC23CCCC2C3)C1)N(c1ccc(C2CC2)cc1)C 28907,CCC(CC(C)CO)NCc1cn(Cc2occc2C(=O)O)nn1 28908,C=C(Cl)C(C)(C)C(=O)N1CC(O)(C(C)(C)CNC(C2CC23CCSCC3)=O)C1 28909,O=C(C1=CCS(=O)(=O)C1)N1CCC2(C1)CN(C(c1cc(F)cc(F)c1)=O)C2 28910,C1(NC(C(C)Oc2ccccn2)=O)CCCN(CCn2cc(Cl)cn2)CC1 28911,Cc1ccc(F)c(C(N2CC(NC(c3cc(Cl)ncc3Br)=O)C(F)C2)=O)c1 28912,C(CCS(C)=O)(C(=O)N1CCC(OCc2ccc(Cl)c(F)c2)C1)N(C)C 28913,C(=O)(C1=CCC(C)CC1)N1CC2CC(C(=O)NC(CCCCC)C)(C1)C2 28914,C(=O)(CCCCC(=O)OC)N(C)CC1N(C(CNC(=O)NC)=O)CCCC1 28915,C1(CC)(NC(=O)Cc2cc(COC)on2)CCN(C(c2cccc(Cl)n2)=O)CC1 28916,c1(SCCC(=O)N(C2CC(NC(CCOCCC)=O)C2)C)ncnc2[nH]cnc12 28917,C1(CNC(C2CC(C)(C)O2)=O)CCC2(CCN(C(=O)CC3CCC3)CC2)CO1 28918,C1(C(=O)NCCc2c(C)noc2C)CC(O)CCN1C(c1cnc(O)o1)=O 28919,N1(C(c2c(C)nn(C3CCC3)c2)=O)CCN(C(C2(C)CC3CC3C2)=O)CC1C 28920,CC(CCCO)(N=c1ccn(Cc2ccc(F)cc2)[nH]1)c1ccccc1 28921,C1(CC(=O)NC(c2c(C)nccc2)C)C2CCCC2N1C(=O)C(C#N)C(C)C 28922,C1(CNC(c2ccco2)=O)(CNC(c2cc(O)cs2)=O)CC12CCC2 28923,C(c1cccc(F)c1Cl)=CC(=O)NCCC1(CNC(CCN(C)CCO)=O)CC1 28924,c1(C(=O)N(C2CCOC2)CCCNC(C(C2CC2)OC)=O)ccccc1 28925,c1(OC)cccc(NC2CCCCC2OC(C)C)c1.C1(=O)NNC(=O)NC12CC2 28926,C1(C(=O)NC2(COC)CCN(C(=O)CCCC(F)(F)F)C2)CC2C=CC1CCC2 28927,c1(NC)cc2c(cc1Br)CCC2.c1(C2C(C)C2)cc(C)[nH]c(=NCc2ccnc(Br)c2)n1 28928,c1(CCC(=O)N(CC(CC)NC(=O)C(C)CN2CCOCC2)C)cn(C)nn1 28929,c1(NC(=O)CCNC(c2ccc(Cl)o2)CO)ccc(Cl)cc1F 28930,CC(C)CC(CCO)NC(C1OCCC1CNC(C1(n2cccn2)CC1)=O)=O 28931,c1(C(=O)OC)cc(C)cnc1N(C1CCCN(C(C2CC(=O)NC(=O)N2)=O)C1)C 28932,Nc1cc(C(=O)NC2(CNC(=O)CSc3nncs3)CC2)cc(O)c1 28933,c1(COC)cccc(C(=O)NC(C)CN(C(=O)CCSCC(C)C)C)n1 28934,N1(CC=C)C(=O)NC(c2csc(-c3ccsc3)n2)C2=C1CN(C(C)(C)C)C2=O 28935,S(=O)(=O)(c1ccc(N2CCCC(OCC(F)F)C2)cc1Br)NCC1(C)CSC1 28936,C#Cc1ccc(Cl)c(C(=O)NCCCCNC(=O)Cn2cc(C3CC3)cn2)c1 28937,c1(OCC2OCCO2)ccccc1CN(C1CCCC1)C(C1CNC(=O)O1)=O 28938,C1(CNC(C2CCC(C)C2)=O)CCCN(Cc2sncc2Br)C1 28939,c1(OCc2c(-c3c(F)cccc3)nccc2)cccc2c(Br)cccc12 28940,C1(C(N(OCC(=O)OC)C)=O)(c2cccs2)CCOCC1 28941,C(N=c1[nH]c(=NCC2CN(C3CCC3)C2)[nH]c2ccsc12)c1c(C)cccc1Cl 28942,c1(C(=O)NC2C(CNC(C(C)(C)c3cnc[nH]3)=O)C2)cccc(-n2ccnc2)c1 28943,N1(C(Cc2c(OC)nccc2)=O)CC2CC(NC(C3CCC3C(F)F)=O)CC1C2 28944,C(=O)(C1CCCc2nncn21)N1CC2CN(C(c3cc(Cl)cc(Cl)c3)=O)CC2C1 28945,N1(C(C2N(C)CCC2)=O)CCN(C(=O)C(O)C2CC2)C(CO)C1 28946,c1(C(C(=O)NC(C)C)N(C(CC(C)C)C)C)ccc(SCC(F)(F)F)cc1 28947,c1(C(N(C)CC2N(C(CCCC#C)=O)CCC2)=O)cc(OC)c(N)c([N+](=O)[O-])c1 28948,C1(CC(=O)N(C(C)CCN2CCOCC2)C2CC2)CCC(C)(C)CN1 28949,C1(CC(=O)NC(C2CCOC2)CO)(NC(C(CO)N(C)C)=O)CCCCC1 28950,CC1(C)C=C(C(=O)Nc2cccc(NC(C3CC3c3ccnc(Cl)c3F)=O)c2)C1 28951,c1(C(N2C(C)CC(CNC(=O)CC3CCOCC3)C2)=O)cncc(C#N)c1 28952,c1(C(N2CCC(NC(COCCCC)=O)C2(C)C)=O)cc(F)cc(Cl)c1N 28953,c1(C(=O)NCC2(F)CN(C(=O)C=C3CCC3)C2)cc2cccc(Br)n2c1 28954,c1(C(=O)OCC)cccc(C#CCSc2noc3c2COCC3)c1 28955,C(c1nc2cc(Br)cnc2s1)=C(C)C 28956,CC1(CNC(c2ccc(CNC(c3cccc(F)c3F)=O)o2)=O)CCCCC1O 28957,c1(CCNC(N2CCCC(Nc3cc(Cl)c(Br)cn3)C2)=O)ccccc1[N+](=O)[O-] 28958,C(=O)(C1=C(Cl)CCOC1)N1CCC(C(N2CC(CC)NC(=O)C2)=O)C1 28959,C(CN=c1nc(N2CC=C(Br)CC2)c2c([nH]1)CCS2)N1CC(C)OC(C)C1 28960,N1(C(CNC(CNC(CC(C)SC)=O)=O)=O)CCCC2OCCC12 28961,c1(CC)cn2c(n1)CC(C(=O)NCC(C)N(C)C(c1cc(C)cc(O)c1)=O)CC2 28962,N1(C(c2cn[nH]c2)=O)CC2CC2(NC(C2(Oc3ccccc3)CC2)=O)C1 28963,c1(CC)ccc(F)c(C(N2CC3CCOC3(CNC(=O)CC(=O)NC)C2)=O)c1F 28964,n1(CCC(N2C(CNC(C(C)OC)=O)CCC2)=O)ccc2ccccc12 28965,C1(C(N2CCCC2CCNC(C2(CF)CC2)=O)=O)CC12CCC(F)(F)CC2 28966,CCCCC(C)CCC(=O)N1CCC1CNC(c1sccc1CC#N)=O 28967,C(=O)(C1=C(C)OCCS1)N1CC(OCC)C(CNC(C2CCC(C)(C)OC2)=O)C1 28968,N1(C(c2ccc(SC(F)F)cc2)=O)CC2CN(C(C3CC3(F)F)=O)CC2C1 28969,N1(C(C2=CC(C)(CC)C2)=O)CC2CC(C1)CN(C(c1cc(Br)c[nH]1)=O)C2 28970,c1(OCC)ccc(C(=O)NCCN(C(=O)C2CC2)C(C)C)c(Cl)c1 28971,N#CC1CCN(C(=O)CC2CN(C(=O)CC3CCCOCC3)CC23CC3)CC1 28972,c1(C(N2CCCC(O)(CNC(C(C)(C)OC)=O)CC2)=O)cc(F)c2c(c1)CCC2 28973,c12ccnc(c1F)OCCCNC(=O)C21CC1.C(=O)(C(C)(C)OC(F)F)NC 28974,C(=O)(C1=CCOCC1)NC(COC)C(=O)NCC1CCN(C)C1=O 28975,CN1N=C(C(=O)Nc2cccnc2C(N2CCCC(NC(N)=O)C2)=O)CCC1=O 28976,c1(C(N2C(C)C(NC(=O)CCc3csc(=N)[nH]3)CC2)=O)csc2c(F)cccc12 28977,c1(CCCC)ccc(C(N2CCN(C(C)C(=O)NC3(C(N)=O)CC3)CC2)=O)cc1 28978,c1(OC)nc(C)ccc1C(=O)NCC1(C)CN(C(c2c[nH]nc2F)=O)CCO1 28979,c1(C(N2CC(CC)N(C(=O)CCC(=O)OC)CC2)=O)cc2c(C)nn(C)c2s1 28980,c1(SCCC)cccc(C(=O)NCC(C)(C)NC(C2CCOC2=O)=O)c1 28981,CC1CC2CN(C(=O)C(CO)C(F)(F)F)CC2N1C(=O)CCC(C)(C)N(C)C 28982,c1(CC)cc(C(N2CC(C(F)(F)F)(C(C)(C)O)C2)=O)no1.C12CC1(C)CNC2=O 28983,Cc1noc(C)c1C(C)CC(=O)NCC1(CNC(C2(C)CNC(=O)C2)=O)CC1 28984,n1(CC)nc(C(=O)NC2C(C(c3ccccc3)=O)CC2O)c2cccc(O)c12 28985,c1(C(=O)NC2C(SC)CN(C(C3CCCC3(C)C)=O)C2)cc2c(cn1)OCCC2 28986,Cc1cc(C)n(CCNC(=O)CC(C2CC2)NC(=O)CC2CC(C)(C)CO2)n1 28987,c1(OC)cc(C(=O)N(C2CC(NC(=O)C(C)(C)CO)C2)C)cnc1OCC 28988,c1(C(=O)NCCC2(CNC(C(C)OCC=C)=O)CC2)scnc1C(F)(F)F 28989,CCCC(C)(C)CC(=O)NC1C(C)(C)C(NC(C2CSCCS2)=O)C1(C)C 28990,Cn1cccc(C(=O)NCC2C3CN(C(C4(CCF)CC4)=O)CC23)c1=O 28991,C1(NC(CSS(C)(=O)=O)=O)CCN(C(=O)CCN2CCCC2=O)CC1C(N)=O 28992,c1(COC)nc(Cl)cc(=NC(C)CCNC(c2nc3cccnc3s2)=O)[nH]1 28993,C1(NC(C)=O)CN(C(=O)C(Cc2cccc(Cl)c2)NC=O)CC2(CCOCC2)C1 28994,C1(C2CCN(C(C3COC(=O)N3)=O)C2)(NC(CC2(C)CC2)=O)CC1 28995,C12(NC(Cn3c(C(C)C)ncc3)=O)CCN(C(=O)COCCN(C)C)CCC1C2 28996,c1(C(=O)NC2CCC(CNC(=O)CCn3cccc3)C2)cc2c(=O)[nH]ccn2n1 28997,N1(C(CCN(C(=O)CCCCN(C)C)CC=C)=O)CCCOC(CC)C1 28998,C1(CC(=O)NC(CC(C)NC(c2n(C(C)C)ccn2)=O)C)COCC(C)(C)O1 28999,c1(CNC(C(COC)C)=O)ccccc1CNC(C)=O 29000,C(C(C(=O)N1OC2CCC1C2)NC(=O)C(=O)NCC)SCC 29001,C1(CC)CCN(C(=O)C=CC2CCOCC2)C1CNC(=O)Cc1ccsc1 29002,N1(C(COCCCC)=O)CCCC1(C)C(=O)NC1C=CCCCC1 29003,C1(NC(COCC=C)=O)CCN(C(c2ccc(OC)cc2N)=O)CC1F 29004,c1(C(=O)NCC(=C2CN(C(c3nc(OCC)oc3)=O)C2)F)cccc(C(C)C)c1 29005,C(=O)(CCC(=O)NCCC1(O)CN(C(c2cc(C(C)C)on2)=O)C1)NCC 29006,Cc1[nH]c(C)c(C(=O)NCCCNC(c2cccc(N(C)C)c2)=O)c1C 29007,c1(C(N2C(C)(OC)CC2)=O)cccc(Cc2cn(CC(=O)O)nn2)c1 29008,c1(C(=O)NCC2(O)CCN(C(C3(CC4CC4)CC3)=O)C2)csc2ccc(F)cc12 29009,C1(NC(C(C)SCC)=O)CC(C(=O)N2CC=CC2(C)CO)=CC1O 29010,c1(C(N2CC(OC)C(NC(=O)C=Cc3cnc[nH]3)C2)=O)sc([N+](=O)[O-])cc1Cl 29011,CC1CCN(C(=O)C=Cc2ccccc2)CC1NC(=O)CC1CC(=O)NC1=O 29012,C1(NC(c2c(CC)ocn2)=O)C(C)CN(C(=O)C2=C(C)CCCC2)CC1C 29013,C1(CC(C)NC(c2cc(OC)ns2)=O)CCN(C(=O)CC2CCS(=O)(=O)C2)CC1 29014,N12CCN(CC1C#N)Cc1ccc(s1)C2=O.c1(NC(C)=O)cnccc1C 29015,c1(C(N2CC(CC)N(C(=O)Cc3ccsn3)CC2)=O)ccc(C)c(OC)c1F 29016,C1(C(N(CC(C)NC(c2cnc(O)s2)=O)CC)=O)CCC(NC(C)=O)CC1 29017,c1(CC)ncc(C(=O)NC(C)C(C)(C)NC(C2CC(n3ccnn3)C2)=O)s1 29018,CCCCC(O)C(=O)NCC(CNC(C1(c2cc(C)on2)CCC1)=O)C(F)(F)F 29019,C1(NC(CC(C)C)=O)CCCCCN(C(C23CC(CC(F)F)(C2)C3)=O)C1 29020,c1(C(=O)NCCCCC(C)NC(C(CC)OCC)=O)ccc([N+](=O)[O-])cc1C 29021,c1(C(N2CC(F)(C(=O)NCC(CNC)O)C2)=O)ccccc1Oc1ccncc1 29022,C(CC(C(=O)NC(C(C)(C)O)C1CC1)NC(=O)CCc1ccc(C)o1)=CC 29023,N1(C(c2c(OC)n[nH]c2)=O)CCC(CF)(NC(C2CSCCS2)=O)C1 29024,Cc1sc(-c2ccccc2)nc1C(=O)NC1CN(C(C2CCCO2)=O)C1 29025,C1(C(=O)NCC(CN(C(c2c(C)occ2)=O)C)C)C2CCC1(c1nccs1)C2 29026,C1(NC(C2CCC(C#C)CC2)=O)C(C)(C)C(NC(=O)C(C)=C(C)C)C1(C)C 29027,N1(C(c2cncc(NC(c3ccncc3Cl)=O)c2)=O)C2COCC1CC(F)C2 29028,C(=O)(C1COc2ccccc21)NCC1(C)CCN(C(c2cc(F)ccc2N)=O)C1 29029,C1(C=O)CCCC(=O)C1.C1(COC)(NC(=O)CC2(N(C)NC)CC2)CCOC1 29030,C1(NC(C2(CCC)CCNC2=O)=O)CCCCN(C(c2cc[nH]c2)=O)CC1 29031,CCCCC(=O)C(=O)NC(C)(C)CC(=O)N1CCCC1C1(C)CC1 29032,C=CC(F)(F)C(=O)N(CCCNC(=O)CC1COC(C)(C)C1)C 29033,c1(NC23C(CN(C(c4cccc(C)c4C)=O)C2)CCC3)nc2c(C)cccc2o1 29034,C12(NC(C3CC3F)=O)CC(CO)(C1)OC21CN(C(=O)C2CCCc3ncnn32)C1 29035,C1(C(N2CC(CNC(CN(C3CCC3)C)=O)C2)=O)OCCOC1c1ccccc1 29036,c1(NC(CNC(C2N(C(C)C)CCC2)=O)(C)C)nc2cc(Cl)cc(Cl)c2o1 29037,c1(C(=O)NCC(CN(C)C(c2ccccc2C(C)(C)C)=O)(C)C)nc(=N)cc[nH]1 29038,c1(CC)nc(Cl)nc(N2CCCCC(CNC(C3(C(N)=O)CCC3)=O)C2)c1C#N 29039,C12(C(=O)NCC3CCN(C(C(=O)NCC)=O)C3)C=CC(CC1)C2 29040,C1(NC(C2CC(C#C)(O)C2)=O)CCCC(C(=O)N(C)Cc2occc2C)CC1 29041,CC(C)(F)CCC(=O)NCC1CC2CCC1N2C(=O)CCCc1ccccn1 29042,CC1(C)CCCC1(O)CNC(=O)CC1(NC(C2OC3CCC2C3)=O)CC1 29043,CCCCC(O)CCC(=O)NC1CC(C)N(C(=O)Cc2cnn(C)c2C)C1 29044,Cc1noc(Cl)c1CC(=O)NC(C)(C)CCCNC(=O)C(n1cnc(C#N)n1)C 29045,c1(C(N2C(C)CC(NC(c3nccn3C)=O)C2)=O)ccccc1S(=O)(=O)C(F)F 29046,C1(NC(C2N(C(C)C)C(=O)CC2)=O)CCCCN(C(=O)C(F)C2CCC2)C1 29047,Cc1cccc(C(=O)NCCC(O)C(=O)NC2CC3CCC(C2)C3O)c1C#N 29048,CCCC(CCCNC(=O)Cc1ccc(Br)cn1)NC(c1c[nH]ccc1=O)=O 29049,CC1(C(=O)NCc2nocc2C(=O)N(C2CC2)CC2CC2)COCCO1 29050,C(=O)(C1=C(Cl)CCC1)NC(CCCCNC(C(CC)(C)C)=O)C 29051,n1(CC)nccc1C=CC(=O)NCCCCNC(C1CCCC(C(F)(F)F)O1)=O 29052,CC(C)CCCCCCNC(=O)C(CCC1CCC1)NC(=O)CC1CCC(=O)C1 29053,C1(CNC(C2(OC)CCSC2)=O)CN(C(c2c[nH]c(=O)cn2)=O)CCC1(F)F 29054,CC1CC=C(C(=O)NCc2cncc(C(=O)NC(c3nnc(O)n3C)C)c2)CC1 29055,C(=O)(CC(C)(C)C(=O)N(CCCN(C(=O)C(=Cc1cccnc1)C)C)C)OCC 29056,C(CCCCC(=O)NC1CC(NC(=O)CC2CC(F)C2)C12CCC2)OCC 29057,c1(C(C)=O)ccc(CC(=O)NC2CC(C)(NC(C3(C4CCCO4)CC3)=O)C2)cc1 29058,N1(C(=O)OC(C)(C)C)CCC2(C1)CN(N1CCc3nc(Cl)ccc3C1)C2 29059,c1(N(C)C)cc(F)c(NC(C2CCN(c3ccc(Cl)cc3)C2=O)=O)cc1[N+](=O)[O-] 29060,c1(CNC(N(c2ccc(F)cc2F)CC)=O)cccc(Cl)c1OCCO.C1CO1 29061,C1(CCC(=O)NCC2CC(NC(C(C#N)C3CC3)=O)C2)NC(=O)NC1=O 29062,C1(NC(C(CC)(C)C#N)=O)CC2(C1)CC1(CC(NC(=O)C3=C(Cl)CC3)C1)C2 29063,N1(C(C2C(C(=O)OC)CC2)=O)CC(NC(c2n[nH]cc2Br)=O)C2(CC2)C1 29064,c1(C(=O)NCCN(C(c2cnn(C(F)F)c2)=O)CC)cc(N)c(Cl)c(O)n1 29065,C(CN=C(NC1CCC1)N1CCCC2(CC2)C1)SCC.N(CC)CC 29066,c1(C(=O)NCC2CCN(C(C(OC)OC)=O)CC2C)cc2c(C)ccc(F)c2o1 29067,C(c1ccco1)=C(C)C(N1CCC(C(F)C(=O)NCCCc2ncc[nH]2)C1)=O 29068,CCC(C)(O)C(=O)N1CC(C(C)NC(C2(O)CCC2)=O)C1 29069,N1(C(C(=O)N(C)C)=O)CC(C)(C)OCC1CNC(C12CCC(CO)(CC1)CC2)=O 29070,C1(C)(C(=O)Nc2cc(C)sc2)CCCN1C(c1ccc(C(N)=O)[nH]1)=O 29071,C#Cc1ccc(CNC(=O)C(CC2CCOCC2)NC(=O)C(CC)OC)cc1 29072,C1(NC(=O)COCc2cscn2)CC2CCC(C1)N2C(=O)CCOCC(F)F 29073,CC1CN(C(=O)C=Cc2cncc(F)c2)CC1(C)CNC(c1ncncc1F)=O 29074,N1(C(CCCC)=O)CCCC2(C1)CN(C(c1cc3cnccc3o1)=O)CCO2 29075,Cc1cc(C(=O)N(CCNC(c2ccn(C(F)F)n2)=O)CCOCCO)sc1C 29076,CC1(C)CC2(CC(C(N3CCC(CNC(=O)CCS(N)(=O)=O)C3(C)C)=O)C2)C1 29077,CCCCC(O)CC(=O)N1CC2C(C(=O)N(CC(=O)N(C)C)C3CC3)C2C1 29078,N1(C(c2ccc(COC)o2)=O)CCCCC(CNC(=O)C(CBr)=CC2CC2)C1 29079,c1(C(=O)NCC(CC(C)C)NC(C2NC(=O)C3CC23)=O)cn2c(n1)CCC2 29080,C(=O)(C(C)C(F)(F)F)NCc1c(CNC(c2n(CCCC)ncc2)=O)nccc1 29081,C1(C(N2CCC(CNC(C3CC4CCC3CC4)=O)C2)=O)CCC2CCC1O2 29082,C(c1cccc([N+](=O)[O-])c1)=CC(=O)NC1C(C(N2CC(C)(O)C2)=O)C1 29083,c1(OC)ccc(NC(C2CCCN2C(C2CCC2)=O)=O)cn1 29084,Cc1c(CC(=O)NC2CCCCC2Sc2ccccn2)nc(Br)n1C 29085,C#CC1(O)CC(C(=O)NC2CC(C)(C(N3CCCC3CC(C)(C)C)=O)C2)C1 29086,c1(CC(=O)NC2CN(C(CC(C)C)=O)CC2C)c[nH]c2c(Br)cccc12 29087,Cn1nc(C(=O)NC2CCC(CNC(C3(C)COC3)=O)CC2)cc1Br 29088,C1(CNC(C2(CC3CC3)CCCO2)=O)NCC12CCC2 29089,N1(C(C2C(C=C)C2)=O)CCC(NC(=O)Cc2sc(O)nc2O)CC1c1ccccc1 29090,c1(SC)ccc(C(N2CC(C)(NC(C3CC4CC4C3)=O)C2)=O)cc1Br 29091,c1(C(=O)NCCOCCN(C(C(CCCC)O)=O)C)ccc(Cl)c(S(N)(=O)=O)c1 29092,n1(CC(=O)NC2C(CNC(c3c(CC)cco3)=O)C2)c(C)nc2ccccc12 29093,c1(CC)ccccc1CC(N1CC(CNC(=O)C=C(C)c2ccco2)(OC)C1)=O 29094,Cc1nccc(CCC(N2CC(NC(C3CCN(C(C)C)CC3)=O)CC2C)=O)n1 29095,C1(O)(CC)CCN(C(c2ncccc2OCC(F)(F)F)=O)C1 29096,c1(C(N2CC3CCN(C(CC(C)C(F)(F)F)=O)C3C2)=O)cnn(C)c1S(N)(=O)=O 29097,C1(CC)(CC)CNC(=O)[NH+]1[O-].c1(CN(C)Cc2ccccc2)ccc(C)cc1 29098,C1(C)(C(C)(C)C)CC(C(=O)NCC(CO)NC(=O)CC2CSCCO2)C1 29099,N1(C(c2cn(C)nc2CC(C)(C)C)=O)CCOCC12CCS(=O)(=O)C2 29100,N1(C(C(N2CC(C(C)NC(C(CCC)C)=O)C2)=O)C)C(=O)NC2(CCCC2)C1=O 29101,C1(NC(c2n(C=C)ncc2)=O)CC2CC1CN(C(=O)CCc1cccnc1Cl)C2 29102,N1(C(c2c(C)ncc(Cl)c2)=O)CCN(C(=O)C=Cc2nc[nH]n2)C2(CC2)C1 29103,O=S(=O)(c1cc2sc(=NCCCCO)[nH]c2cc1Cl)NC1C2CCC(F)(F)C12 29104,N1(C(C)(C)C)CCC(CNc2cn(C3CCCC3)nn2)CC1 29105,Cc1cc(=NC(Cc2ccccc2C)C(C)C)[nH]c(=NCC(C)(C)C(F)(F)F)[nH]1 29106,c1(C(C)OC(=O)C(C)Sc2ccccc2)cccc(OC(F)(F)F)c1 29107,C1(C(=O)NC(c2cccc(F)c2)C)CCN(C(=O)C2=CC(C)(C)C2)CC1C 29108,C(=O)(C(CC(C)C)NC(=O)OC)NC1CCN(C(CNS(CC)(=O)=O)=O)C1 29109,CC1=C(C(=O)N2CC(NC(c3cc(Cl)cn3C)=O)CC2CO)CCCC1 29110,c1(NCC(CNC(c2cnc(CC)nc2O)=O)O)ncc2c(Br)cccc2n1 29111,c1(C(N(CCC)CCNC(=O)CN(C)C(N)=O)=O)cc(F)ccc1OC 29112,O=C(CCCCN1CCCC1)NCC12CC1CN(C(C1(O)CCSC1)=O)C2 29113,Cc1c(C(=O)NC(C2CCN(C(=O)CSC3CCOC3=O)CC2)C)c(Cl)nn1C 29114,c1(CCC(=O)NC(C(C)C)CNC(C2(CC(F)F)CC2)=O)ccc(F)cc1F 29115,Cc1ccn(C)c1C(=O)NCc1nocc1C(=O)NC(c1ncccn1)C 29116,C1(C)(CNC(C(CCC)C)=O)COCCN(C(c2ccc(CO)cc2F)=O)C1 29117,c1(C(=O)OCC)sc2ncn(-n3cnnc3-c3ccccc3F)c(=O)c2c1C 29118,c1(OC)ncnc(C(=O)NCc2ccc(C#N)cc2)c1F.C12(O)CCN(C1)C2=O 29119,N1(C(CCC=C=C)=O)CCN(C(=O)C(C)(C)COC)CC1C(C)C 29120,c1(C(=O)NC2CC(CNC(Cc3nc(C)sc3)=O)C2(C)C)ccc(CO)c(Cl)c1 29121,Clc1ccc2c(c1Br)CN(c1ccn3nccc3n1)CC2 29122,O=C1NCCC2C(C(N3CCCC3c3ccsc3)=O)C12 29123,c1(CC(N2CCCN(C(C(C)N(C(C)=O)C)=O)CC2)=O)noc2ccccc12 29124,c1(NC)ccc(C(=O)NCC23COC(CF)(C2)C3)cc1.C12CC(C)N(C1)C(=O)C2 29125,Cc1nc(S)sc1CC(N1CCC(F)(CNC(c2cncc(F)c2)=O)C1)=O 29126,C1(N(C)CC)CN(C(c2ccc(C3CCC3)cn2)C(=O)NC)CC12CCC2 29127,C1(NC(c2cc(CN(C)C)on2)=O)CCCCC1CNC(=O)C(C)(C)C1CCC1 29128,Cn1ccc2cc(-c3nc(-c4ccnc(Cl)c4)nn3Cc3ccccn3)ccc12 29129,c1(C(C(=O)NC(CC)C)N(C)CCc2cccc(Cl)c2Cl)scc2c1OCCO2 29130,c1(C(N2C(C)CC(NC(C(CCC)(C)O)=O)C2)=O)c(F)cc(F)cc1F 29131,c1(CC(=O)N(CC(C)O)CCNC(CCc2cnc(C)s2)=O)ccccc1C 29132,C1(C(C)NC(c2c(CC)noc2)=O)CCCCN1C(c1cccc(C(N)=O)n1)=O 29133,N1(C(c2c(CC)c[nH]c2)=O)CCOC(CNC(=O)C(C)(CO)OC)C1 29134,CCCCC(C)(F)C(=O)N(CC(C)NC(c1cc(N(C)C)ccn1)=O)C 29135,N1(C(CC(C)(C)NC(C2CC3C=CC2O3)=O)=O)CCC2C(C1)C2(F)F 29136,C12CCCCN1C(=O)C1(CC1)C(=O)NC(C)C(=O)NC2.C1(NC)CC2CCC1O2.CO 29137,N1(C2CCN(C(=O)CCC3CCCC3)CC2)C2CCC1CN(C(C1(F)CC1)=O)C2 29138,C(C(F)(F)C(=O)NC1CCC1CNC(c1cc(-c2ccccc2F)no1)=O)OC 29139,c1(C(=O)NC(C2CCOC2)CNC(C2(C)CC2(F)F)=O)cc2nc(F)ccc2o1 29140,C=CCCC(c1nnnn1CCCSCC)NC(C)CNc1cnc(SC)s1 29141,O(C1CCOc2ccc(Br)cc21)Cc1cn(-c2cc(F)c(C(=O)O)c(F)c2)nn1 29142,C=C(Cl)CCC(=O)N1CC=CC1CNC(=O)CCC1CCCCO1 29143,C(=O)(C1=C(Cl)CCC1)N1C(CCNC(CSCC)=O)CCC1 29144,N1(C(c2ccc(C(C)=O)c(O)c2)=O)CC2CCC1CN2C(c1c(C)csc1Cl)=O 29145,c1(CC(=O)NC2(CO)C(C)C2)csc(-c2cccnc2)n1 29146,C1(CC(=O)NC(C2CCN(C(=O)C(F)CC3CCOC3)CC2)(C)C)SC(=N)NC1=O 29147,C1(NC(c2c(SC)cn(C)n2)=O)C2COCC1CN(C(C1CCCO1)=O)C2 29148,c1(C(=O)NC(CCNC(C2N(CC)C(=O)CC2)=O)(C)C)ccc2c(c1O)CCC2 29149,C1(CNC(C(C)C2CCCC2)=O)CCCCN1C(=O)C(c1csc(=N)[nH]1)=O 29150,CC(C)C(C(C)NC(c1nocc1Cl)=O)NC(=O)CCNC(N)=O 29151,n1(CC)nc(C)cc1C(=O)N(C)CC1CCCC1NC(C1(C)CC1C)=O 29152,c1(CCC(=O)N(CC(C)NC(CCOC)=O)C)ccc(Br)cc1 29153,c1(C(N2CC(COC)N(C(C)=O)CC2)=O)cc2c(cc1Br)OCCO2 29154,c1(CNC(N(C)Cc2ncc(C)o2)=O)cc(Cl)c(Cl)c(Cl)c1 29155,C1(C(=O)NC(C2N(C(c3n(CC)ncc3)=O)CCC2)C)CCCC(C)(C)CC1 29156,c1(C(=O)NCC(F)CNC(C2(CO)CC2)=O)cc2sc(Br)cc2[nH]1 29157,Cn1c(C(=O)N(CCNC(C2CC2F)=O)CC2CC2)cc2occc12 29158,Cc1nc(O)[nH]c1C(N1CC(NC(c2cscc2C#N)=O)C1)=O 29159,N1(C(C(C)SCC=C)=O)CC2CC(C(N3CC(C(=O)NC)C3)=O)(C2)C1 29160,C1(C(N2CCN(C(=O)Cc3cccnc3)CC2)=O)CC12CCCOC2 29161,c1(CC(N2CCC(C(=O)OC)CC2(C)C)=O)cccc2c1CCCC2 29162,C(c1ccc(Cl)cc1F)=CC(=O)NC1CCC(CNC(c2n(CC)ncn2)=O)C1 29163,C(C)(CCC(=O)N(C)CCN(C(=O)CCc1ccc(OC(F)F)cc1)C)OCC.CC 29164,c1(C(=O)NCCN(CCC)C(C2CC23CCOC3)=O)ccc(C)c(C(C)=O)c1 29165,c1(OC(C)C)ccc(C(c2nc(-c3ccc(C(=O)C(C)C)cc3)no2)C)cc1 29166,c1(C(=O)NCCN(C)C(c2nocc2Cl)=O)cncc2c1CCC2 29167,c1(NCc2nc3ccc(C)cn3c2)cc(=NCCS(=O)(=O)N(C)C)[nH]c(C)n1 29168,c1(C(N2CC(C(C)NC(CC(COC)C)=O)C2)=O)ccc2c(c1)CCO2 29169,N1(CCC(=O)NC(C2CCCN(C(=O)CCF)C2)C)CCCCC1=O 29170,c1(OC)ccc(C(=O)NCCCCCCNC(C2CCCCN2C)=O)nc1N 29171,Cc1cccc2c1ccn2CC(=O)NC(C)CNC(C1CC(=O)NC(C)C1)=O 29172,C1(COC)COCCN1C(=O)CC1CCN(C(c2ccncc2Cl)=O)C1 29173,Cc1nccn1CC(N1CCCC1C(=O)NCC1(C)CSC1)=O 29174,N1(C(C(N2CCCC(COC(C)(C)C)C2)=O)=O)CC(S(C)(=O)=O)C1 29175,C1(NC(C2(NC(CSCCCC)=O)CCC(C)(C)C2)=O)CC(C2CCCC2)C1 29176,CC1(C(=O)NCc2cc(C(F)(F)F)ccc2O)CCCN(C2CCCSC2)C1 29177,N(C1CN(C(c2cc[nH]n2)=O)Cc2ccccc21)c1nc(C)nc(Cl)c1C 29178,CC1(C)CCC2CC(NC3CCCOC3)c3cccc1c32 29179,c1(NC(C(CC2CC2)NC(C2CCC(=O)C2)=O)=O)cnc(F)nc1 29180,N1(C(CC(C)N(C)C)=O)CCCC2CN(C(c3cncc(C#N)c3)=O)CCC12 29181,c1(CN(C(c2ncc(Cl)n2C)C(=O)NCCCC)C)noc2ccccc12 29182,C(C(=O)NCC1CCN(C(c2csc(C)n2)=O)C1(C)C)(C(C)(C)C)NC(=O)OC 29183,c1(CC=O)cccnc1.C(C(C)(C)CO)NC(CN(CC)CC)C 29184,c1(C(N2CCCC2NCc2nc(CO)cs2)C(=O)NC)csc2ccccc12 29185,Cc1cc2c(C(=O)NC(C)CC(C)NC(c3cnc(O)nc3O)=O)cccc2o1 29186,c1(C(N2C(C(=O)NCCc3c(C)nn(C)c3)CC2)=O)cc(C#N)cn1C 29187,Cc1ccc2c(c1)CC(C(N1CCCCC13CN(C(C1CC1[N+](=O)[O-])=O)C3)=O)S2 29188,C12(CNC(=O)CC3OCCO3)CCCC1CCN2C(=O)Cc1cnc[nH]1 29189,C=CCCCC(=O)NCCC1(NC(=O)C(C)NC(C2CCCC2)=O)CCCC1 29190,C1(NC(CC2CCCC(CC)C2)=O)CC12CCN(C(c1ccc[nH]1)=O)CC2 29191,C=Cc1cnn(C)c1C(=O)NCC(C1CC1)NC(c1ccc(Cl)c(OC)c1)=O 29192,CCCCN=C(NCC(c1ccnn1C)O)NC1CCN(C(=O)CCOC)C1 29193,c1(C(=O)NCCCCC2CCCN(C(=O)CO)C2)cc(Cl)c2c(c1)OCCCO2 29194,CC(C)CC(CNC(=O)CSCC(C)C)NC(=O)CSc1cccs1 29195,c1(Cn2nnc(C(C)(C)C)n2)cncc2ccccc12.N1CCc2ncncc2C1 29196,C#CCC(C(=O)NCC(O)COCC)NC(=O)C(C)NC=O 29197,c1(C(N(C2CC3CNC2C3)C(CC)CO)=O)ccc(C(N)=O)cc1 29198,N1(C(C=Cc2cn(C)nn2)=O)C2CCC(C2)C1C(=O)NCc1ncn(C)n1 29199,c1(C(N2CCOC(CNC(=O)C(F)(F)C(O)C3CC3)C2)=O)ccc2nsnc2c1 29200,N1(C(CC2CCC(C)CC2)=O)CC2CCC1C1CN(C(=O)CSCC(N)=O)CC21 29201,N1(C(C(=O)OC)C)CCC(C(N2CCCCC2CO)=O)(OC)CC1 29202,C1(C(=O)NCCSCC(=O)NCC2CN(C)C2)CCCCCCC1 29203,C=C=CC(C)C(=O)N1CC(O)(C(C)NC(=O)CCOCC2CCC2)C1 29204,c1(C(=O)NCC(=C)CCNc2cc(=O)n(C)cn2)ccc2c(c1)COCC2 29205,N1(C(C2N(C(C(=O)OC)C)CC2)=O)CCC(C2CCC2)(C(=O)OC)C1 29206,CCS(=O)(=O)c1ccc(F)c(C(=O)N(CCC(C)NC(=O)Cc2ccco2)C)c1 29207,C12(NC(CC(C)O)=O)CCC(CC1)N(C(=O)Cn1cnc([N+](=O)[O-])n1)C2 29208,C#CCC(C)(C(=O)N(C1CC(C(=O)NC)C1)C)NC(C1CC(=O)CS1)=O 29209,C1(NC(C(CN(C)C)NC(C2CC3(C2)CC32CC2)=O)=O)CCCCCC1(C)C 29210,C(C(C)(O)CCC)NC(C=C(CNC(C(C)OCC=C)=O)C)=O 29211,N1(C(C2C(OC)CC2)=O)CC2C(C(=O)NOCCN3CCCC3=O)C2C1 29212,c1(CN(C(=O)NC2C(C)(C(=O)OCC)C2)C)cc(C(F)(F)F)cc(C)c1 29213,N1(C(COCCCCC)=O)CCCCC1C(=O)NCc1cnc[nH]1 29214,c1(C(N2C(C)(CNC(=O)C3=C(Cl)CC3)CCC2)=O)cc(=O)n2ccccc2n1 29215,N1(C(c2cnc(C(C)OC)s2)=O)CCCC(N(C)C(c2c(C)nsc2C)=O)CC1 29216,N1(C(c2ccc(CC)cc2O)=O)CC2CC(NC(c3nnsc3C)=O)CC2C1 29217,N1(C(CC2CC(C)(C)OCC2)=O)CCC2(CCCN2C(=O)C(O)C2CCC2)C1 29218,c1(C(=O)NC2(C(=O)OC)CC2)cn2cc(-c3cnc4c(c3)NCCO4)ccc2n1 29219,S(=O)(=O)(c1c[nH]ccc1=NC1CC1C1CCCC1)NCc1cc(CC)on1 29220,C=C(C)CC(C(=O)NCCCCNC(N)=O)NC(c1ccsc1)=O 29221,C1(C)(C(N2CCC(NC(c3ccn(C)c3)=O)C(CO)C2)=O)CC(C2CC2)=NO1 29222,Cc1cccc(CC(=O)OCC(=O)NCC2(CCC#N)CC3CC3C2)c1I 29223,Cn1cc(-c2cc(C(=O)NC3(C)CN(C(C4(c5nccs5)CC4)=O)C3)no2)cn1 29224,C1(C#CC(=O)N2CCC(OCCNC(C3CC3F)=O)C2)(CC)COC1 29225,C1(C)(NC(C=CC)=O)CCN(C(c2oc(-c3ccccc3)nc2C)=O)C1 29226,C1(CNC(CC(CC)SC)=O)CCCCCN1C(=O)COc1cc(C)ccc1C 29227,n1(CC)nnc2c(N3CC4CC(NC(=O)Cc5ccc(Cl)cn5)C4C3)ncnc12 29228,N1(C(CNS(CCCC)(=O)=O)=O)CC2CCCN(C(=O)C(C)C(F)F)C2C1 29229,S(=O)(=O)(c1ccc(=NCc2ccc(S(C)=O)cc2)[nH]c1)N1CC(N(C)C)C(O)C1 29230,C1(OC(C(CCC)(C)C)=O)CCCN(C2CCCc3ccccc32)C1=O 29231,Cc1oc(C(=O)NCCNC(C2CCCCN2C2CCCC2)=O)cc1S(N)(=O)=O 29232,C(=O)(C(C(=O)NCC(C)(C(C)C)NC(=O)C1=CCC1)c1ccccc1)OCC 29233,C(=O)(CCC(C)(C)NC(c1cc[nH]c(=N)n1)=O)NC1CCN(CC)C1 29234,c1(CCNC(C2CCN(c3ncc(I)cn3)CC2O)=O)c[nH]c2ccc(Br)cc12 29235,c1(C(=O)NCC2CCCC(NC(CCCSC)=O)C2)coc2c(F)cc(Cl)cc12 29236,c1(C(N2CC(CNC(COCCC)=O)C3C2C3)=O)cc(N)c(Cl)c(O)c1 29237,N1(C(C(c2cccc(O)c2)C)=O)CC(NC(=O)COC2CCOCC2)C(C)C1 29238,c1(OCC)ncccc1C(=O)NCC(COC)NC(=O)C=C=C(C)C 29239,N1(C(C(n2ncc(C)c2)C)=O)CCCCC1CC(N1CC(F)(CF)C1)=O 29240,C(c1cnc2ccccc2n1)=CC(=O)NC1CC2CC1N(C(c1cocn1)=O)C2 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29258,Cc1ncc(Br)c(N(c2ncc(Br)c(O)n2)CC2CNC2)n1 29259,CC1CC(=O)NC(C(=O)N(C(C)CNC(c2ccc(CO)cn2)=O)C)C1 29260,C1(NC(CCC#CC)=O)CC(O)CN(C(=O)CCC2CC2)C1 29261,c1(C(=O)NCCC(C)NC(C2N(C(C)=O)CC(O)C2)=O)ccc(=O)n(C)c1 29262,C(=O)(C1=CCCOC1)NCC1CCC(NC(c2ccc(OC)s2)=O)CC1 29263,c1(CNC(c2nnnn2CCC2CC2)(CSC)C)cccc(OC(C)=O)c1Cl 29264,c1(C(N2CC(C)(CC(=O)NCC3(C)N=C(C)SC3)C2)=O)cc(C)c(F)cc1Br 29265,c1(N(C(C)C)CC)ccc(C(=O)NC2(C)CCN(C(=O)C(F)=CCCF)C2)cn1 29266,N1(C(C)=O)CCN(C(c2cccc([N+](=O)[O-])c2C)=O)CC12CCCCC2 29267,N1(C(CC(C)C)=O)CCCCC1C(N1CCC(C)C1C)=O 29268,C#Cc1ccc(C(N2CCN(C(C3C4CCCC34)=O)CC2CC(F)F)=O)nc1.O 29269,C(=O)(C(C)CCC(C)(C)C)NC1C2CN(C(c3cc(C)c(O)c(C)c3)=O)CC21 29270,C1(N2CCC2=O)CCC(C)N(CCCC2CCOCC2)C1.C(=O)(C(F)(F)F)OC 29271,C12(NC(=O)CC3CCCO3)CC(CNC(=O)CC3CCCCC3)(C1)C2 29272,c1(C(N2CC(OC)C(NC(=O)C(C)(C)CC#N)C2)=O)ccnc2nc(C)nn12 29273,c1(NC(C(N2CCOCC2)C)=O)cc(CNC(c2csnc2C2CC2)=O)[nH]n1 29274,CCCC(C(=O)OC)NC(C1CCC(SCc2ccc(F)cc2)O1)=O 29275,N1(C(c2c(CNC(C(c3cn(C)nc3)O)=O)cc[nH]2)=O)CC(N=[N+]=[N-])C1 29276,c1(C(=O)NCCN(C(C(C)C)=O)C2CCCC2)cc(CN(C)C)ccc1O 29277,c1(CC)cc(Cl)ccc1Oc1ccccc1.n12cc(nn1)C(C)NC(=O)C2 29278,C1(CNC(C2(C(C)(F)F)CC2)=O)CN(C(=O)CCCOc2ccccc2)CCN1C 29279,C(=O)(C(O)CSC)NCCOCC(=O)NCC(=C)Cl 29280,C1(=O)CCCCC(=O)N1.CCCC(C(=O)NCC(C)(C)OCC)NC(N)=O 29281,C12(NC(COCCC(C)C)=O)COC(C1)C(NC(c1cccc(CC#N)c1)=O)C2 29282,C1(C(=O)NC(c2nc(C(C)(C)C)no2)CC)CCC(=O)NC1 29283,C1(C(=O)NC(C)CN(C)C(C2(C#N)CCCC2)=O)(COC)CC=CCC1 29284,C1(NC(=O)CN2CCCCC2)CN(C(=O)C=CC2CCCO2)Cc2nccn2C1 29285,N1(CC(N2CCCC(CNC(=O)Cc3cnoc3)CC2)=O)CCCCC(O)C1=O 29286,c1(OC)ncccc1CC(=O)NCC1C2CC1N(C(=O)CN1CCCC1C)C2 29287,N1(Cc2c(OCC)nn(C)c2)CCC(O)CC1C1CC1 29288,CC1CCc2[nH]nc(C(=O)NCCC3CCCN3C(=O)C(C)c3cccs3)c2C1 29289,N1(C(Cc2ccc(C(=O)NC)cc2)=O)CC2CCC(N(C)C)CC2C1 29290,C(=O)(C(C)N=c1cc[nH]cc1)NCC(CNC(CCOCCOCCCC#C)=O)C 29291,c1(NC(NC2CCc3ccc(Br)cc32)=O)nc(O)c2ccc(Cl)cc2n1 29292,c1(N2CC(NC(C)=O)C2)nc(NCC2COCCN2C)c2ncn(C(C)C)c2n1 29293,C1(C(=O)NC(CC)(C)O)CC(O)CN1c1ccncn1 29294,C1(C(N(CCC(=O)NC)C)=O)C2CC3C(C2NC(=O)CC2CCCCCC2)C13 29295,C(=O)(CCCC(=O)OCC(=O)Nc1cccs1)OC(CC(C)C)c1nn[nH]n1 29296,Cc1cccc(CC2(SCC(=O)NCC3CCCC(C(=O)NC4CC4)C3)CC2)c1 29297,C(=O)(C1=C(CCC(=O)NCC(CNC(=O)C(C)(F)F)CO)NC(=O)NC1C)OCC 29298,c1(C(=O)NC2C(NC(c3[nH]c(=N)sc3)=O)C2)cnc2cccnn12 29299,C1(C(=O)NCCN(C(C(C)OC)=O)Cc2ccccc2)CC2CCC1CC2 29300,c1(C(=O)NC2CCC(NC(CC=C(C)C)=O)CC2)[nH]nc([N+](=O)[O-])c1Cl 29301,N1(C(c2c(C)nns2)=O)C2CCC1CN(C(c1cccc(C(F)F)n1)=O)C2 29302,C1(OC)CN(C(C2(CO)CCC2)=O)CC1CNC(=O)COCc1nc[nH]n1 29303,c1(C(N2CCCC2C2CCOC2)C(=O)N(C(CC)(C)C)CC)ccc(C)c(C)n1 29304,C(=O)(CCCC(=O)N1CC(CNC(C2(F)CCOC2C)=O)CC1C)NC(C)C 29305,C(C#Cc1cc(Cl)cnc1F)NC(N1CCC(O)(C(C)O)CC1)=O 29306,C1(NC(C(C)OC2COC2)=O)CCC2CN(C(c3ccnn3CCO)=O)CCC2C1 29307,N1(C(C2CCC(C)O2)=O)CC2CCCC1(CNC(c1ccc3c(c1)CCO3)=O)C2 29308,c1(C(N2CC(NC(c3cc(CC)n(C)n3)=O)C(O)CC2)=O)cc2n(c1)CCSC2 29309,c1(C(C)=O)cc(NC(C2CC2C(=O)Nc2ccc(Br)c(F)c2)=O)cc(C#N)c1 29310,N1(C(C)C(C)(C)O)CCOCC(C(=O)NCC2CC3CCN2CC3)C1 29311,CC1(C)C2CN(C(C3CC3F)=O)C(C(N3CCCC(O)C3)=O)C12 29312,C#CC1(C(=O)N(C)CC2CN(C(=O)Cc3csc(C)n3)CCO2)CCOCC1 29313,CCCC(C)CC(C(=O)NCC(C)C)N1CCCC1(CCC)CO 29314,C1(NC(CC(COC)C)=O)(CO)CCCN(C(=O)Cc2conc2C)C1 29315,c1(CCN(C(=O)Cc2ccsc2Cl)CC)cn(C2(CN3CCOCC3)CC2)nn1 29316,N(C1CC(F)(F)c2cc(Br)ccc21)C(N1CCC(O)(c2cccc(F)c2)C1)=O 29317,c1(SCC(=O)NCC(C)(CO)NC(=O)CCCCCC2CC2)c(F)cccc1F 29318,C1(CNC(c2cc(Br)n[nH]2)=O)CCCC12CCN(c1nc3ccccc3o1)CC2 29319,C1(CC)CCN(C(=O)CCOC)C1C(=O)Nc1ccnc(C(=O)OC)c1 29320,S(=O)(=O)(c1ccc(OCC23CC(N)(C2)C3)cc1)NC(c1cccc(COC)c1)C 29321,C1(C(N2C(C(C)NC(c3c(C)occ3)=O)CCC2)=O)CSC(c2ccccc2)=N1 29322,c1(C(C(=O)NC2C(CNC(CN(C)C)=O)C2)O)ccnn1C 29323,c1(C(N2CCC(CCNC(C(C)=CC)=O)CC2C)=O)cccc2c1ccn2C 29324,C1(NC(Cc2ncc(CC)[nH]2)=O)CCCN(C(=O)CSCC2CCCCO2)C1 29325,n1(CC)ncc(C(=O)N(CCCNC(=O)COCP(C)(C)=O)C2CC2)c1Cl 29326,C1(CNC(C2C(C(=O)OC)C2)=O)CCCC(CNC(c2ccc(C)cc2)=O)C1 29327,C1(C(N2CCC(c3cn(-c4ccncc4)nn3)C2)=O)(SC)CC(=O)C1 29328,CC1CN(C(=O)Oc2ccccc2Cl)CCC1N(C1CC2OC(=O)OC2C1)C 29329,c1(C(C)C)ccc(C(=O)NCC2(C)CCCN(C(c3csc(S)n3)=O)C2)c(O)c1 29330,C1(CCC)(NC(=O)COCC(F)F)CCCN(C(=O)CCCn2cncn2)C1 29331,N1(C(c2c(CCNC(CCOCCC)=O)n[nH]c2)=O)CCOCC(O)C1 29332,C1(NC(C(CC2CCOCC2)NC(C2CCCO2)=O)=O)CC2CC1CC2CO 29333,O=S(=O)(c1cnc(C(F)F)s1)NCCCCCCCC1CC1 29334,Cc1ccc2c(N3CCSCC3C(=O)NCC(F)F)ncnc2c1 29335,c1(C(C(=O)Nc2ccccc2)N(C)Cc2snc(C)n2)ccnc(Cl)c1 29336,c1(COC)ccc(CNC23CC(C(=O)NC(C)CC(=O)OC)(C2)C3)cc1 29337,N1(C(C(c2ccccc2F)C)=O)CCCC(CO)(NC(c2cccn2C)=O)C1 29338,CC(C)(O)C(F)C(=O)NCCC1CC(F)CN1C(=O)C1CC1 29339,C(C(C(C)(C)C)NC(=O)CCc1nc(C(C)OC)no1)NC(C1C(CC)C1)=O 29340,c1(C(C(=O)NC(C)CC(=O)N2CCCC2)(C)C)ccc(Cl)nc1 29341,c1(N2CCN(C(C(=O)NC)C)CC2)nccc(=NC(C)c2nc(C(C)C)cs2)[nH]1 29342,N1(C(C(C)(CO)NC(=O)CC2C=CCCC2)=O)CCOC2(CCC2)CC1 29343,c1(NC(C2CN(S(CC)(=O)=O)C2)=O)cc(C2CCCC2)nn1C 29344,CC1CCN(C(=O)CN2CCS(=O)CC2)CCN1C(=O)CC1CCCC(C)(C)C1 29345,C1(C(=O)NCC2(CC)CCCC2)CCN(C(=O)C(C)(C)COC(C)C)CC1C 29346,N1(C(C(C=C)(C)O)=O)CCc2nc(CNC(C3CC(C)CC(C)(C)C3)=O)sc2C1 29347,c1(CC)nn(C)cc1C(N1CCCC(NC(c2cc(C(=O)OC)c[nH]2)=O)C1)=O 29348,CCCCCC(C(=O)Nc1ccccc1Cl)N1CC2CCOC2C1 29349,C(CN=c1ccc(C(=O)NCc2nc(CNC(=O)CCS(C)=O)cs2)c[nH]1)OC 29350,N1(C(C(CC)=CCCC)=O)CCN(C(=O)CCc2nncnc2O)C(CO)C1 29351,N1(C(=O)COC2CCCC2O)CC2CCCC(C1)N2C(C1CC(F)(F)C1)=O 29352,C(C(CC1CCCC1)C(=O)Nc1ccc(SC)cc1)NC(CC(=O)NCC#C)=O 29353,c1(C(N2C(CNC(CCCN(C(C)=O)C)=O)C=CC2)=O)cnc(N)c(N)c1 29354,c1(C(=O)NC2C(N(C(c3cn(C(C)C)nn3)=O)C)CCCC2)cc(N)cc(O)c1 29355,CC(C)C(C(=O)NCCCCCN(C)C(C1(CO)CC1)=O)NS(N)(=O)=O 29356,C(C1c2ccccc2CCN1C(c1conc1C)=O)NC(C1(COC)CC1)=O 29357,N1(C(c2c(C)c(N)n(C)n2)=O)CCCC(C2CN(C(=O)C(C)OCC(C)C)C2)C1 29358,c1(NC(=O)NCCC2=CCCC2)ccc([N+](=O)[O-])cc1 29359,c1(CN2CCC3(C(C(=O)NCCc4ccc(F)nc4)C3)C2)cc(Cl)cc(Cl)c1O 29360,C1(CN(C(=O)Cc2cn(C)cn2)C)CCN(C(c2csc(C#N)c2)=O)CC1 29361,C(=O)(CCCCCNC(N)=O)NC(C)CCCCNC(C12CCC1C2)=O 29362,C1(CC)CC(C(=O)NCC(c2ccsc2)O)CCN1C(c1csc(C)n1)=O 29363,C12(CC(N3CC(C4N(C(=O)COCCF)CCC4)(O)C3)=O)CCC(CC1)C2 29364,N1(C(C(C)=C(C)C)=O)CCN(C(c2nn[nH]c2C(F)(F)F)=O)C2(CCC2)C1 29365,Cc1cc(C(=O)NCc2ocnc2C(=O)NC2CC3CCC2C3)c(C)o1 29366,C1(C(N2CC(OC)CC(C(=O)NCC3(COC)CC3)C2)=O)CCCCC(C)(C)C1 29367,Cc1nn(C)c(Cl)c1CC(N1CCC(CNC(=O)C(C2CCC(=O)N2)C)CC1)=O 29368,C1(NC(c2ccnc(C)n2)=O)CCCCCN(C(c2ccc(C3CC3)cc2)=O)C1 29369,c1(NCCNC(c2nc(C(F)(F)C(=O)O)cs2)=O)ccc(F)cc1 29370,c1(C(=O)NCCC2N(C(C(CC=C)C)=O)CCC2)ccc(C)c(OC)c1 29371,C1(C(=O)NCC2N(C(C(CC)N3CCCC3=O)=O)CC=C2)CC2(C1)CC(C)(C)C2 29372,C(=O)(C1=CCCN(C(C2CCCC2C(C)C)=O)C1)NC1C=C(C)CCC1 29373,C1(NC(N(CC(O)COCc2ccccc2)C)=O)CC12CCCC2 29374,N1(C(C(=O)NC(c2ccnc(C(F)(F)F)c2)C)=O)CC2CC1c1ccccc12 29375,C(C(CCC(F)(F)F)NC(c1cnn(C)c1F)=O)OC 29376,C(=O)(C1=NOC(C)(C)C1)NCC1C(N(C)C)CN(C(CC2CCCN(C)C2)=O)C1 29377,C(CC(CC)C(=O)NCC1CN(C(=O)CN2CCN(C)C(=O)C2)CC1(C)C)=CC 29378,C1(NCC(C)Cn2cccn2)CCCC1NC1CN(C(=O)OC(C)(C)C)C1 29379,C1(C(N2C(C)(C(=O)OC(C)(C)C)CC2)=O)CCn2c(Br)cnc2C1 29380,c1(N2CC(N(C)C(c3cnn4c3CCCC4)=O)C2)ncnc2cc(I)sc12 29381,C(=O)(C1CCCc2nc[nH]c21)NC(C)(CNC(c1snc(O)c1Cl)=O)C1CC1 29382,CC(C)C(C(F)F)NC(=O)NC1CCN(CCCF)CC1 29383,c1(C(N2CCC(C(C)NC(CCSC)=O)CC2)=O)c(C)nn(C(C)C)c1C 29384,N1(C(CC=CCC)=O)CCOC(CNC(c2sc(-c3ncccn3)nc2C)=O)C1 29385,C(=O)(C1=C(C#N)CCC1)NCC(CC=C)NC(c1cccc2[nH]ncc12)=O 29386,CCC(CC)(C(=O)NCCC1CN(C(C2(COC)CC2)=O)CC(C)O1)OC 29387,C12(NC(C=CC(=O)N(C)C)=O)CCCN(C(=O)CCOCC(F)(F)F)CC1C2 29388,CC1CN(C(C2(C)CCC(=O)C2)=O)CC(C)N1C(c1ccoc1Cl)=O 29389,C(=O)(CN=c1cc[nH]cc1)NC1CC(NC(c2cc(CC)no2)=O)C12CCC2 29390,C(=O)(CCC(C)(C)C)N1CC(NC(C(CC)C)=O)C(C)C1 29391,C1(C(N2CC(O)(C(CNC(C(C=CC)O)=O)(C)C)C2)=O)COc2ccccc2O1 29392,c1(OC)cc(C(=O)NC2CCCCC2NC(c2ncccc2N)=O)cc(F)c1F 29393,Cc1nc(C)c(C(=O)NC(C2CCN(C(C3CC3(C)C)=O)CC2)C(C)C)[nH]1 29394,c1(C(N2CC(C)(CC(=O)NCc3cc(F)ccc3Cl)C2)=O)cc(F)ccc1C#N 29395,c1(CC(=O)NC2(CCNC(CCCSC)=O)CC2)ccc(O)c(F)c1 29396,C1(NC(C2(CC#C)CCCC2)=O)CC2CC1CN(C(c1ncc(C(F)F)s1)=O)C2 29397,C1(C(N2CCC(O)(CC)C2)=O)Cc2nnsc2S1 29398,C12(CNC(c3cc(C(C)C)nn3C)=O)CN(C(=O)C=CC3CC3)CC1CCO2 29399,C1(NC(C2CCOCC2)=O)CS(=O)(=O)C2CN(C(c3ncccc3Cl)=O)CC12 29400,C1(CC)CCN(C(C2CSC2)=O)C1CNC(c1ccc(C(=O)NC)nc1)=O 29401,c1(NC(=O)NC(c2cccc(Cl)c2)c2onc(C)n2)cc(F)ccc1O 29402,C1(F)(CNC(=O)Cn2c(O)nnc2O)CCCN(C(C2C3CC4C(C3)C24)=O)C1 29403,N1(C(c2nn[nH]c2Cl)=O)CCN(C(=O)C=CBr)C2CCCCC2C1 29404,C(=O)(CC(CNC(=O)CC1CSCCO1)OC)N(CCCCC)C 29405,O=CN1CCCN(C(=O)CC2CC=CCC2)CC1 29406,C#CC1(O)CCN(C(=O)C(CC(=C)C)NC(c2ccccc2C#N)=O)C1 29407,N1(c2nnc(Cc3ccc(C)o3)n2CC2CCCO2)CCc2nc(Cl)ccc2C1 29408,c1(C(=O)NCCN(C(c2cn(C3CCC3)nn2)=O)CC)coc2c(F)cc(Cl)cc12 29409,Cc1oc(C(=O)NCCCN(C(C2(C#N)CC2C)=O)C2CC2)cc1S(N)(=O)=O 29410,CN1C(=O)CCC1CC(N1CCCCC1CCNC(c1csc(Cl)n1)=O)=O 29411,c1(NC(CC2CCN(Cc3ccc(OCC)c(Cl)c3)C2)=O)cc(Br)c(Cl)cc1F 29412,O=C(C1=NN2CCCN=C2N1)NCC1CC1NC(C1(Oc2ccc(F)cc2)CC1)=O 29413,C1(C)(NC(C2CCN(C(=O)NC)C2)=O)CCN(C(=O)CCCCN2CCCC2)C1 29414,c1(C(=O)NC(C(C)(C)C)CNC(=O)Cn2cnc(=N)[nH]2)ccc(S(C)(=O)=O)s1 29415,C1(C(=O)NC(c2ccc(F)cc2Cl)c2n(C)ccn2)CCN2CCOCC12 29416,C(=O)(C(CO)C(C)(C)C)NC(CNC(c1ccc(C#C)o1)=O)CC(C)C 29417,C1(CNC(c2c(CC)onc2)=O)CN(C)CCN1C(=O)CC(C)F 29418,N=c1[nH]c2cc(C(=O)NCC3C4CN(C(=O)CSc5nncs5)CC34)ccc2o1 29419,c1(C(=O)OC)cc(Br)c(C(=O)O)cc1NC(C1CC1c1ccccc1Cl)=O 29420,N1(C(C(C)NC(=O)CC(C)(C)C)=O)CCC(C)C(CNC(=O)CCCC2CC2)C1 29421,C1(CC(=O)NC(C(c2ccccc2)NC(C(C)=C2CCCC2)=O)C)CCC2CC2C1 29422,c1(C(N2C(C(=O)Nc3ccc(C#N)cc3)CC(F)C2)=O)c(Br)cc(F)c(Cl)c1F 29423,c1(C(=O)NC2C(CNC(C(C)(C)c3ccc(Cl)s3)=O)CCC2)cc2n(n1)CCO2 29424,N1(CCNC(=O)CC(F)(F)F)C(=O)CCN(CC2CCCc3nc[nH]c32)C1=O 29425,O=S(=O)(c1cc(Br)c(F)cc1F)NCC1CCN(Cc2cc(I)c[nH]2)C1 29426,C(=O)(C(C)CCCC(C)C)N1CC(CC=C)(NC(=O)CNC(=O)C(F)(F)F)C1 29427,CONC(=O)C(=O)NCCC1CN(C(=O)CC=C(Cl)Cl)CC1C 29428,C(=O)(C(C)(C)CCCNC(=O)C1=COCCC1)N1CC(C)C(CO)C1 29429,n1(CC)c(S(=O)(=O)NCC2COC(C)(C)C2)cnc1C 29430,Cc1cc(C(=O)NCCC(C)NC(c2c(C)ccnc2C)=O)c2c(c1)CCCN2 29431,CCC(CC(=O)N1CCOCC1CN(C(=O)C=Cc1nccn1CC)C)C(F)F 29432,CC(C)(C)C1=NOC(C(=O)NCC2CCN2C(=O)C=C2CCCCC2)C1 29433,C1(CCC)(NC(=O)CC2(OC)CN(C(C3(CSC)CC3)=O)C2)CCNC1=O 29434,C(CC(=O)NC1(C(=O)OC)CC1(C)C)(CC(C)C)NC(CN(C(=O)OC)C)=O 29435,N1(C(CCCC#C)=O)CC2CCCC2C1C(=O)NC(C)CC(=O)NC 29436,Cc1cc(C(F)(F)F)c[nH]c1=NCCC(=O)Nc1cccc(Br)c1 29437,C1(COC)(NC(c2cc(C(F)F)nn2C)=O)CCN(C(C2(F)CCCC2)=O)C1 29438,c1(NC)ccc(C(=O)NCCCCC(C)NC(c2ccc(F)o2)=O)cc1 29439,C(C(F)(C(=O)NCC1CC2CCC(C1)C2)C(C)C)NC(CCC(CC)=O)=O 29440,C=CCCCC(C(=O)N(CC(O)COCC)C(C)C)NC(=O)Cc1ccc(C)nc1 29441,c1(CC)cc(C(N2CCC(N(C(=O)CC3CCCC(O)C3)C)C2)=O)c(C)o1 29442,C(=O)(C1(C)CCn2c(C)nnc21)N1CC(O)(CNC(C(CC)O)=O)C1 29443,C(=O)(C1CCCn2ncnc21)NCCNC(c1nccc(OC)c1C)=O 29444,c1(OC)cc(C)c(C(=O)NC2CN(Cc3ccncc3Cl)CC2F)c(C)c1 29445,N1(C(c2[nH]cc(CC)c2)=O)CCN(C(c2sc(C(C)(C)C)nc2C)=O)CC1C 29446,C1(C(=O)NCC(CC)NC(c2cnc(C)cc2Cl)=O)CCc2ccnn2C1 29447,C1(C(N(CC(C)NC(c2nn(CC)c(C3CC3)c2)=O)C)=O)CCc2nccn2C1 29448,Cc1nc(C2CC2)nc(C)c1C(N1CC(NC(C2CC(C)OC2=O)=O)C1)=O 29449,C(=O)(C(O)Cc1cnn(C)c1)NCCN(C(C(c1ccc(Cl)s1)C)=O)C1CC1 29450,C1(C(N(CCCN(C)C)CC)=O)C(CC)CCN1C(C1OCCC1(C)C)=O 29451,c1(C(N2C(C)CC(NC(C3CC(C#C)(O)C3)=O)C2)=O)cccc2c(C)[nH]nc12 29452,N1(C(C(C)N(c2n(CC)cnc2)CCC)=O)CC(OC)C2(CC2)C1 29453,c1(CCC(N2CCC(N(C(C=NOC)=O)C)C2)=O)ccc([N+](=O)[O-])cc1 29454,N1(C(c2cc(OC)c(C)cc2)=O)CCC2CN(C(c3cnn(C)c3Br)=O)CC12 29455,c1(C(COC)N(C)C(c2nnsc2C)=O)ccc(Cl)cc1 29456,c1(OC)c(F)ccc(C(N2CC(NC(c3ccc(Cl)o3)=O)CC2C)=O)c1F 29457,CC(CCCNC(=O)CCc1cnoc1)NC(=O)C(C)(C)C1(O)CCOC1 29458,c1(C(=O)OCC)nc(C(=O)NC(C)CNC(=O)C(C)(C)c2csc(C)c2)c(C)s1 29459,O(NC(=O)C(CNC(c1ccsc1)=O)CC1CCCC1)CC(C)(C)C 29460,C1(CC(C)C)CC1N=c1[nH]c(N2CCCC(c3cccnc3)C2)nc2c1CCC2 29461,NS(=O)(=O)C1CC(C(=O)NCc2cccc(CNC(C3CC3CF)=O)c2)C1 29462,c1(C(=O)NC2C(NC(CCOCCC)=O)CC2)csnc1C 29463,C#CCC(C(=O)NC)NC(C1CC(NC(=O)C(C)OCC2CC2)C(O)C1)=O 29464,C12(F)CCN(C1)C2=O.c1(CC)conc1C(=O)NC1(C(=O)OC(C)(C)C)CC1 29465,c1(C(N(C)CCNC(=O)CCOC2CCC2)=O)c[nH]c2cccc(F)c12 29466,c1(C(N2C(c3ncc(-c4ccc(OC)cc4)[nH]3)CCC2)=O)c(Cl)cc(Br)cc1Cl 29467,c1(C(C)C(N2CCCC3CC23)=O)cc2ccccc2o1 29468,C(=O)(CC1=NN(C)C(=O)C1)N1CCC(C)C(CNC(c2cnn(CCF)c2)=O)C1 29469,C(CC(C(C)(C)C)NC(=O)CN1CC=CC1)N(C(C(CO)OC)=O)C 29470,C1(N(C)C(C2CCNC2=O)=O)CN(C(c2cc(C(C)(C)C)ccn2)=O)CC1(C)C 29471,N1(C(c2ccc(OC)cc2)=O)CC(C)(C(=O)NCC(C)C(C)(C)C)CC1(C)C 29472,C1(NC(Cc2cc(COC)on2)=O)CN(C(=O)CP(C)(C)=O)CCC1C 29473,C(C(N=c1cc(C)nc(NC2CC3(C2)CC(O)C3)[nH]1)C1CC1)OC 29474,c1(CCO)ccc(C(c2nnnn2C2CC2)NCc2ccc(Br)cc2)cc1 29475,Cc1nc(Br)c(C(=O)NCCC(C)(O)C2CC2)s1 29476,N1(C(C2CCOCC2OC(F)(F)F)=O)CCC2CCN(C(=O)C=CCO)C2C1 29477,C1(C(N2CC(NC(CC=CC=C)=O)(CO)C2)=O)CCCC2(CCC2)O1 29478,C(=O)(CC(C)(C)CC(=O)NCC1CC1CNC(C1CC2(CCC2)C1)=O)OC 29479,C(CC(C)C)(C(=O)NCC(CNC(=O)CCc1cnoc1)CO)OC 29480,CN=c1nc(C(=O)NC2CC2NC(=O)CCn2cnnn2)cc(C)[nH]1 29481,C1(CNC(C(CC(C)C)C)=O)CC2CCC(C1)N2C(c1nn(C)cc1N)=O 29482,C=CCCC(C(=O)N(C)Cc1cn(C)cn1)NC(=O)CC1CCCCN1C 29483,c1(CC(=O)NC23CC(NC(CCc4ccn(C)n4)=O)(C2)C3)cccnc1Br 29484,C1(CNC(C2CC(CC)C2)=O)CC(C(=O)N(CC(C)(C)O)C)=NO1 29485,C(N=c1[nH]c(=NCc2cnc(Br)n2C)c2[nH]ccc2[nH]1)C1CC(C(C)C)OCC1 29486,c1(C(N2CCC(C3(C(F)(F)F)N=N3)C2)=O)cc2ccsc2s1 29487,c1(CCC)ccc(C(=O)NC2COCC2NC(c2nnc(O)nc2O)=O)cc1N 29488,N1(C(=O)Cc2ccc(Br)cn2)CC2CCC(C1)C2NCc1c(F)cccc1Cl 29489,N1(C(CC(C)C2CCCCC2)=O)CCC2(CC1)CN(C(=O)C=CI)CCO2 29490,c1(C(C(C)SC)N(C(=O)CCn2cc(CC(C)(C)C)nn2)C)cccnc1.CO 29491,c1(C(=O)NC2CC(O)(CNC(CS(CC)=O)=O)C2)cc(Cl)n[nH]c1=N 29492,N1(C(C2(CC)CC(F)(F)C2)=O)CCOc2cccc(C(=O)O)c2C1 29493,C1(O)(CC(N2CC(O)(CN(C)C(c3ccc(NC=O)cc3)=O)C2)=O)CCCCC1 29494,N1(C(C2OCCN(C)C2=O)=O)CC(NC(C2CCC(F)(F)CC2)=O)CC2(CC2)C1 29495,C1(CNC(C2(N(C)C)CC2)=O)COCCN1C(c1ccc(Br)s1)=O 29496,C(C(C)C(C)C(=O)N(CCC(=O)N(C(CO)CC(C)C)C)CC1CC1)OC 29497,C(C)(CO)(C(=O)N1CC(C)(C)C1C(C)C)NC(c1c(OC)nsc1)=O 29498,N1(C(c2c(C)sc(O)n2)=O)CC(C)C(NC(c2cc[n+]([O-])cc2)=O)C(C)C1 29499,c1(C(N2CCC(C)(CNC(C3CC4(CC(=C)C4)C3)=O)C2)=O)cc(C)c(F)cc1N 29500,C1(N(C)C)CCCCC1CNC(=O)C1=C(Cl)CC1.C12CCCC1C(=O)N2 29501,c1(C(C(=O)NCCCSCCOC)N(CC(CC)N(C)C)C)csc(Cl)n1 29502,c1(CNS(C)(=O)=O)cccc(C(=O)NCC2CC(NC(C3(C)CCC3)=O)C2)c1 29503,c1(C(N(CC(C)O)CCNC(Cc2ccc(C)s2)=O)=O)ccc(Cl)cc1F 29504,Cc1ncc(F)c(=NCC2CN(C(=O)CC3CCC(C)C3)C2)[nH]1 29505,N(C(=NCC(C)Oc1ccccc1F)NC(C)C1CC1)Cc1cnc(C)o1 29506,C1(NC(C2(OC)CC(CO)C2)=O)CCC(C(=O)NCCCO)CC1 29507,c1(CC(=O)NC(C)CCNC(=O)CC2(C)OCCO2)ccc(C#N)nc1 29508,N1(C(COC(C)=O)=O)CCN(C(C2CC(Oc3ccc(CO)cc3)C2)=O)C2CC12 29509,Cc1ccccc1CC(C)C(=O)NCC(C(C)C)NC(=O)CN(C(=O)C(C)C)C 29510,C1(CNC(C2(N(C)C)CCCC2)=O)C2CC1N(C(C1CCS(=O)CC1)=O)C2 29511,C(c1ccc(C)c(Cl)c1)=CC(=O)N(CCCNC(CSc1ccc(C)cc1)=O)C 29512,c1(C(C(=O)NC(CC=C)CNC(C2(CC)CCC2)=O)CC)c(C)noc1C 29513,C1(C(=O)OC)COCCC1NC(=O)CC1CSCCS1 29514,N1(C(c2c(C)cncc2C)=O)CC2CC(NC(C3CCCCS3)=O)CC1C2 29515,c1(CC(=O)NCC2CCN(C(c3ccoc3Br)=O)C2)c[nH]c2cnccc12 29516,N1(CC=C(C)C)CCC(NC(=O)Nc2ccc(C(N)=O)cc2)C1c1ccccc1 29517,C1(C(C)CNC(=O)C=CCO)CCN(C(C2CCC23CCC3)=O)CC1 29518,n1(CC)ccc(=NC(=O)C2(CNC(c3cc[nH]c3)=O)CCCCC2)[nH]1 29519,Cc1cnc(N2CCSCC2C)c(S(=O)(=O)N2CCOC(c3ccsc3)C2)c1 29520,C1(C)(CNC(CC(C)(O)c2ccccc2)=O)CCCN(C(C2(CF)CCC2)=O)C1 29521,C(=O)(C1=CCC(NC(c2ccc(C#N)n2C)=O)C1)NC1C(C=C)COC1 29522,C12(C(F)F)CCN(C1)C2=O.c1(CNC(C(=O)NC(C)C)=O)cnc(Cl)s1 29523,C1(C(=O)NCCCN(CCCNC(=O)Cc2cccn2C)C)COC(C)(C)CO1 29524,Cc1coc(C2CC2)c1C(=O)NCC1(O)CC(CNC(C2CC(C)(F)C2)=O)C1 29525,C(=O)(CCS(N)(=O)=O)NCCN1CCC(NC(C2(C)CS(=O)(=O)C2)=O)CC1 29526,N1(C(C(CC=C)CC)=O)CCC2(CCCN2C(=O)CCCOCCC)C1 29527,CCCCC(CNC(c1ccc(OC(C)CC)cc1)=O)NC(C1CCCCO1)=O 29528,c1(CC(N2C3CC(NC(CC(CC)O)=O)CC2CC3)=O)ccc2c(c1)NC(=O)C2 29529,CC1(C)CN(C(=O)CC2CC(=O)NC2=O)CC1Nc1nccc(CO)n1 29530,C1(C(=O)NC(C)C(C)(C)CO)(COC)C=CCN1C(c1ccc(F)cc1)=O 29531,C1(C(N2CCC(NC(c3c(OC)oc(C)n3)=O)C2)=O)CC(c2cnn(C)c2)=NO1 29532,C1(NC(CC2(COC)CCCC2)=O)CC(C)N(C(c2ncncc2Cl)=O)C1 29533,C1(C(=O)OCC)CC(O)CN1C(c1ccc(-c2ccc(C(F)(F)F)cc2)o1)=O 29534,C(=O)(C1=CS(=O)CCC1)N1CCC(NC(C(C)NC(=O)CC(C)(C)C)=O)C1C 29535,N1(OC)CCSC2CCCCC12.C1(N2C3(CC3)CCOCC2=O)CC=CC1 29536,C=C1CC2(C1)CC(C(N1CC(OCCNC(C3CCOC(CCC)C3)=O)C1)=O)C2 29537,C(=O)(CCCNC(c1cc(Cl)c[nH]1)=O)NC1(C(=O)OCC)CCC1 29538,N1(C(C(C)(C)Oc2ccccc2)=O)CCN(C(C2CC(F)(F)C2)=O)CC(O)C1 29539,N1(C(CN2C(C)CC2)=O)CCC2(CCC2)C(NC(c2csc(S)n2)=O)C1 29540,N1(C(c2c(COC)nc(=N)[nH]c2)=O)CC2CC1CN(C(=O)CS(N)(=O)=O)C2 29541,CC(CC(=O)N1CCCC1CN(C(=O)C(C)(C)c1ccns1)C)P(C)(C)=O 29542,N1(C(C2C(=C)CC2)=O)CCC2(CCC2)C(CNC(c2ccc(N)cn2)=O)C1 29543,O=S(=O)(c1ccc2c(c1)OCCCO2)NCC1(CF)CC2(CCC2)C1 29544,CCC(C)C(C(=O)NCCC(C(C)C)NC(c1ccnn1CC(C)C)=O)OC 29545,N1(C(=O)NCC2(CCC(=O)OC)CC2(F)F)CC(C)(C)C12CCOCC2 29546,c1(C(=O)NC2CC(C(N(CC(F)(F)CO)C)=O)C2(C)C)cnn(C)c1C#N 29547,N1(C(CC2CC(OC)C2)=O)CCCC(O)(CNC(=O)C=Cc2ccc(C)o2)CC1 29548,Cc1noc(CCC(=O)NC(C2CCN(Cc3nc(CC4CC4)no3)C2)C)n1 29549,N1(C(C2CCC(=C)CC2)=O)CCCC2(CCSCC2)C1 29550,C1(C(=O)NC2CC(O)(CNC(C3(CC(C)C)CC3)=O)C2)CCS(=O)(=O)N1 29551,CC1(NC(C2CCC(NC(C3CCCC3F)=O)CC2)=O)CC(F)(F)C1 29552,c1(C(=O)NCC2CCN(C(c3cc(C(C)=O)oc3)=O)C2)cnn(C)c1C 29553,c1(C(=O)NCC(C)NC(c2c(CC)nco2)=O)ccc(OCC(C)C)cc1 29554,c1(C(=O)NCC2C(NC(CC=C(C)C)=O)COC2)cnn2c1C(C)CCC2 29555,c1(C(=O)NC2CC(O)(CNC(CC3CCN(C)C3)=O)C2)cccc(C(F)F)c1Cl 29556,c1(OC)ccc(C(C)=CC(N2CC(OC)CC(NC(C3(O)CCC3)=O)C2)=O)cc1 29557,c1(C(=O)OCC)c(C)[nH][nH]c1=NC(=O)c1csc(-c2cc(NCC)cc(F)c2)n1 29558,Cc1ccncc1C=CC(=O)NCC(CC(C)C)NC(c1ccnc(C)c1C)=O 29559,C12(NC(CCC#CC)=O)CCOCC1CN(C(c1cc3sccc3s1)=O)C2 29560,c1(N2CC(CCOC)OCC2)nc(NC(c2cccc(F)c2)C)c2ncsc2n1 29561,S(=O)(=O)(CCCCCS(N)(=O)=O)N(CC(C)(C)C(F)F)C(CC)(C)C 29562,N1(C(CC(CC)(F)F)=O)CCCC12CCN(C(c1cnc3ncc(Cl)cn13)=O)C2 29563,C1(C)(CNC(Cc2n(C)nnc2)=O)COCCN(C(C2CCC3CCC2O3)=O)C1 29564,N1(C(CC(COC)NC(c2cc(CC)no2)=O)=O)CCC(O)C(C)(C)C1 29565,Cc1cccc(C)c1C1CCCN1C(C1CCN(CC2(C)CCN(C)CC2)C1)=O 29566,C12(NC(C3C4CN(C(C5OCC(C)(C)C5)=O)C3C4)=O)CCC(CC1)OC2 29567,CC1(OCC(=O)NCCC(O)CO)CN(CCSCCNC2(C)CC(F)C2)C1 29568,C1(NC(C2CC2CF)=O)CN(C(=O)CC2CCS(=O)(=O)CC2)CC12CCC2 29569,C1(CNC(C2(NC(C)=O)CCC2)=O)CC2CCC1N2C(=O)Cn1cc(CO)nn1 29570,CC1CCCCC1(C)C(N1CCC(CF)(NC(c2ccc(C(N)=O)[nH]2)=O)C1)=O 29571,N1(C(=O)Cn2cccnc2=O)CC2CCC1CN2C(c1nc(Cl)ccc1Cl)=O 29572,c1(C(=O)NC(CC)CN(C(c2nccnc2C)=O)CC)ccc(S(=O)(=O)NC)o1 29573,C(CCS(N)(=O)=O)NC(C=C(C)CNC(C1CC1(Cl)Cl)=O)=O 29574,C1(C(N(CCC=C)CC)=O)(NC(C2(C(N)=O)CC2C)=O)CC(CO)C1 29575,N1(C(c2c(C)cncn2)=O)CCC2(CCC(NC(c3scnc3C)=O)C2)C1 29576,Cc1c[nH]c(CC(N)=O)c1C(=O)NCC1CCC(O)CC1 29577,N1(C(c2cc(OC)c(Cl)cc2OC(C)=O)=O)CCC2(CC1)CCN(C(=O)CO)CC2 29578,c1(C(N2C(C)CC(CNC(CCc3cc(C)no3)=O)C2)=O)ccc(N)c(O)c1 29579,C1(NC(CCCCOC)=O)CC2CCC(C1F)N2C(C1CN(CC(F)(F)F)C1)=O 29580,c1(OC)cccc(C(=O)NC2CC(CO)N(C(C3(C4CC4)CCCO3)=O)C2)n1 29581,C#CC1CN(C(c2ccc(OC)c(F)c2)C(=O)NCC=C)CCO1 29582,C1(C(=O)NCC(C)CC2CCCC2)CCCN(C(c2ccc(C(F)F)o2)=O)C1 29583,N1(C(CCC(N)=O)=O)CC2CC1CC2NC(=O)C#CC1CCC1 29584,C1(c2scc(C)n2)CCCN(C(=O)C(C)C)C1.C1(=O)CCCn2ccc(n2)N1 29585,C1(C2(O)CCN(C(C3CCCO3)=O)CC2)(NC(c2[nH]cc(C(C)(C)C)c2)=O)CC1 29586,C#CCCC(=O)NC(C)C(CO)NC(=O)C(CO)NC(=O)OCc1ccccc1 29587,Cc1ccc(C(O)C(=O)NC2CC(NC(c3cnc(O)n3C)=O)C2)cc1 29588,Cc1nn(CC(N2CC3CCC3(NC(=O)CCCNC(N)=O)C2)=O)c(C)c1Br 29589,CC(C)CC(CNC=O)CC(=O)NC1CCC1NC(c1ccc(CO)cc1)=O 29590,C(=O)(CCCCN1CCCCC1)NCCOC1CN(C(C2CC(OC)C2)=O)C1 29591,CCCC(CC(=O)NCC(C)(C)N(C)C)NC(c1ccc(CO)nc1)=O 29592,C1(CNC(CC(=O)NCC)=O)CC2(CO1)CN(C(=O)CN1CCC(C)C1)C2 29593,CCS(=O)(=O)CC(=O)NC1CCC(C)(CNC(=O)CS(=O)(=O)N(C)C)C1 29594,C(=O)(C1=CCC(C(F)(F)F)OC1)NC1C(NC(C=CCN(C)CC)=O)CCC1 29595,CC1CC(CCNC(c2ccc(C(N)=O)[nH]2)=O)CCN1C(c1ccoc1)=O 29596,N1(C(c2c(OC)noc2C)=O)CCCN(C(=O)CN2CC(=O)NC2=O)CCC1 29597,C1(NC(CC=C)=O)(CC)CCN(C(c2cccc(C(C)(F)F)n2)=O)CC1 29598,c1(C(=O)NCC=CCNC(C2C(CC)CCC2)=O)ccc2c(c1F)CCC2 29599,C1(N(C(COC(C2C(c3n(CC)ccn3)OCC2)=O)=O)C)CC2CCC1O2 29600,c1(OC)ccc(N(C)C(c2ccn(C)c(=O)c2)=O)cc1F 29601,C1(C(=O)NCC2CCC(NC(c3c[nH]c(=O)cn3)=O)C2)C2CCC1(c1ccco1)C2 29602,Cc1ccc2c(c1)C(NCCCC(N)=O)C(C)C2 29603,C1(NC(COCCCCCCCC)=O)CCN(C(=O)C(C2CC2)SC)CC1(C)C 29604,N1(C(C2C3(CC(NC(C(CC=C)(C)C)=O)C3)C2)=O)CC(O)C2(CCCC2)C1 29605,N1(C(C(C)CN(C)C(C2CCCOCC2)=O)=O)CCc2sccc2C1 29606,N1(C(CCC)=O)CC2C3CN(C(C4Cc5cccc(OC)c5O4)=O)CC3C2C1 29607,N1(C(C(C(C)(C)C)SC)=O)CCC2(CC1)CCN(C(C13CC(C1)C(C)O3)=O)C2 29608,c1(C(C)C)cccc(CC(=O)N(C)CCn2cc(-c3ncccn3)nn2)c1 29609,C(C(C)(O)C(=O)N1CC(C(C(=O)NCC2CCCN(CC)C2)OC(C)=O)C1)OC 29610,c1(N(C2CCCCC2S(C)(=O)=O)C)ccc2c(n1)CCCC2=O 29611,Cc1sc(O)nc1C(=O)NC(C)C(C)NC(=O)C(C)(C)CN1CCOCC1 29612,N1(C(C2N(CC)CCC2)=O)CCC(NC(c2ccc(C(C)C)c(C)c2)=O)C1(C)C 29613,CC(CC(C)(C)C)C(=O)NC1CC(O)CN(C(c2cscc2C2CC2)=O)C1 29614,N1(C(CC(CC)O)=O)CCC2(CC1)CC2NC(=O)CSc1nnc(C)n1C1CC1 29615,C(C)(C)(CC(=O)N1CCCCC1CNC(=O)C(c1ccc(C)s1)C)SC 29616,O(NC(=O)C(CO)NC(c1ccnn1CCF)=O)CCN(C)C 29617,CC1CC1N=c1nc2c(ncn2C)c(N(C)CCSc2ccc(F)cc2)[nH]1 29618,c1(C(N2CCN(C(=O)NC)CC2)=O)cccc(P(C)(C)=O)c1 29619,Cc1ccc(O)cc1C(=O)NCC1CC1NC(c1cn(C(C)(C)C)cn1)=O 29620,C1(C(=O)NCCC2(CNC(C3CCCN(CC)C3)=O)CC2)CN2CCN1CC2C 29621,Cc1cccc(OCCCC(=O)NCCCCCNC(c2cc(C)[nH]n2)=O)c1 29622,C(CC(N)=O)(C(=O)N1C(CO)CC1CO)NC(CC1(CSC)CC1)=O 29623,c1(C(=O)NC(CCNC(c2cc(CC)[nH]n2)=O)C)cccnc1SC(F)F 29624,n1(CC)nnc(C(=O)NCCCCC(=O)NCC2(F)CCN(C)C2)c1C 29625,C12(C(N3C(CNC(C=CC(CC)=CC)=O)CC3)=O)CCOC1CCOC2 29626,c1(CC)cc(C(=O)N(C)CC2CCCN(C(=O)C(=O)N(C)C)C2)oc1CC 29627,N1(C(C2N(C)CC2)=O)CCC2(NC(c3cn4ccc(F)cc4n3)=O)CCCCC12 29628,c1(CC(=O)NCC2(NC(=O)CC3CCCCO3)CCC2)cccc(Cl)c1 29629,C1(CNC(=O)CCC2CC2(Cl)Cl)CC2(CCC2)CN1c1nc2ccccc2o1 29630,Cc1cncc(-c2cn(CC3CCN(C(c4oc(C5CC5)nc4C)=O)C3)nn2)n1 29631,CC1CCc2nnc(C(N3CCN(C(C)C(=O)N(C)C)CC3)=O)n2C1 29632,C1(NC(c2n(C)ncc2)=O)CC2CCC1(NC(c1cc(C(N)=O)co1)=O)C2 29633,N1(C(CSC)=O)CC2CCC(CNC(C34CC(C3)C(C)O4)=O)(C2)C1 29634,C1(NC(c2cn(CC)nc2C)=O)CC12CCN(C(=O)CCc1ccc(F)nc1)C2 29635,S(=O)(=O)(c1cc(Cl)ccc1Cl)NCC1(F)CCCN(C(C(CC)O)=O)C1 29636,c1(OC)ccc(CC(C)C(=O)NC(C)CCNC(=O)Cc2sccc2C)cc1F 29637,C1(NC(C2CN(CC)C(=O)C2)=O)CC2CCC(C1C)N2C(c1cc(C)c(C)o1)=O 29638,C1(C(=O)NCCCC2(NC(C3CCC(CC)O3)=O)CC2)C2CCC3C(C2)CC13 29639,C(C)(C)(CC(F)C(=O)NC(C)C(C)SC)NC(CC(COC)COC)=O 29640,C(CC1=CCN(C2CCNC2=O)CC1)NC(C(F)(F)C1(CC)CCC1)=O 29641,c1(C(N2CC(N(C(c3c(C)cccn3)=O)C)C(F)C2)=O)cncc(Cl)c1Cl 29642,N1(C(C=CSC)=O)CC2C3CCC(C2C1)N(C(=O)Cc1n[nH]c(C)n1)C3 29643,c1(OCCC)cccc(CC(=O)NC(C)C(C(C)C)NC(c2cncnc2)=O)c1 29644,N1(C(=O)NC2C(C(=O)OC)CCCN2)CCCC(C(=O)O)C1C 29645,C(=O)(C1CCCn2nccc21)N1CCC(CCc2cn(C(C)CO)nn2)CC1 29646,Cc1cc2c(COC(c3ccnc(SCC(F)(F)F)c3)=O)csc2s1 29647,N1(C(c2ccc(C)s2)=O)CCC(CNC(=O)CNc2cccc(Cl)c2)C12CC2 29648,n1(CC(=O)NC2CC(C(N(C(CF)CF)C)=O)C2)cnc(C#N)n1 29649,c1(C(N2CC(CCNC(c3cc(C)c(N)cn3)=O)C2)=O)ccc2c(n1)OCCO2 29650,C(CC(Cc1ccccc1)NC(C1(Br)CC1)=O)NC(c1cnns1)=O 29651,c1(C(=O)NC(C2CCCC2)CNC(C2CC=C(C)CC2)=O)cccc2nc[nH]c12 29652,C1(NC(CNS(CCCOC)(=O)=O)=O)CN(C(=O)Cn2cccn2)CC2(CC2)C1 29653,C1(OC)CC2CC1CN(C(C1(F)CCN(C(c3ccc(O)nc3)=O)CC1)=O)C2 29654,C(=O)(C(CCC(C)C)NC(c1cnn(C)c1Cl)=O)N(CCCSC)C 29655,c1(C(=O)NCCC(C)N(C(CC)=O)C)cccc2c(I)n[nH]c12 29656,C(c1ccc2c(c1)OCCO2)=CC(N1CCCC(N(C(C(CC)CC)=O)C)C1)=O 29657,C#CCCCCCC(=O)N1CC2(CC(C(=O)NC3CC(=O)N(C)C3)CO2)C1 29658,c1(C(N)=O)cc(C(=O)NCC2CCCC2NC(=O)CCOC2CCCC2)ccn1 29659,Cc1nnc2cnc(C(=O)NC3CC(CNC(c4ccc(Cl)c(Cl)c4)=O)C3)cn12 29660,c1(NC(C2N(Cc3cccc(CC)c3)CCNC2)=O)ccc(I)c(Br)c1 29661,C1(C(=O)NC2C(C(=O)NC(c3c(C)nns3)C)CC2)CCC(C)CC1 29662,c1(C(C)C)conc1C(=O)NC(C)CC(=O)NC1COCC1CN(C)C 29663,C(=O)(C(CC1CCCC1)NC(c1cc(F)c[nH]1)=O)N(C)CCOCC1CC1 29664,n1(CC(=O)NCCN(C(c2ncncc2C#N)=O)CC)cc(C)ccc1=O 29665,C1(NC(=O)OC(C)(C)C)CN(C(=O)NC2CC3CCCC3C2)C2CCCC12 29666,C(=O)(CCCCC(N)=O)N1C(C)CC(C(=O)NCCOC(F)F)CC1 29667,c1(CNC(C(C)C#N)=O)cccc(CNC(=O)CC(C2CC2)C2CC2)c1 29668,C1(C2CC2)(NC(C2CCC(NC(Cc3c(C)ccs3)=O)C2)=O)CCCC1 29669,CC1(C)CN(C(=O)Cc2cccnc2)CC1NC(c1ccccc1C(=O)N)=O 29670,Clc1ccccc1Cn1nnnc1N1CCN(CCSc2ccccc2)CC1 29671,C(=O)(CCN=[N+]=[N-])NC1(CCC(=O)NC(c2ncc[nH]2)C)CCCC1 29672,C1(NC(c2nc(C)sc2C)=O)CCN(C(=O)C(F)C(C)C)CC1CO 29673,C1(CNC(c2cc(O)cc(O)c2)=O)CCN(Cc2c(F)cncc2F)CC1(F)F 29674,c1(C(N(CC(C)C)CC(=O)NCC2CC(=C3CCC3)C2)=O)ncccc1N 29675,N1(C(=O)Nc2ccc(NC3CCN(c4ccccc4)C3)nc2)CC2CC=CC1C2 29676,CC(CC(=O)NCC1CC12CCC2)C(C)(C)NC(C1CC=CC1)=O 29677,C(=O)(C#CC1CC1)NCc1c(C2CN(C(CC(C)c3ccncc3)=O)C2)ocn1 29678,CCC(CNC(=O)CC(C)SC)(CC)NC(=O)C(C)CC1CC1 29679,Cc1nn(C)c(C(=O)NCC2CN(C(=O)COC(F)F)CCCO2)c1Cl 29680,S(=O)(=O)(c1ccc(OC(F)(F)F)cc1)N(C(=O)C(=O)NC1(C2CC(N)C2)CC1)C 29681,C=CC1OCCC1C(N1CCN(CC2(NC(=O)Cn3ccnc3C)CC2)CC1)=O 29682,c1(C(=O)OCC)ccc(C(c2nnnn2CCSC)NCCc2nncs2)o1 29683,C1(C(=O)NC2(CO)CN(C(CN(c3ccc(Cl)nn3)C)=O)C2)COC2(CCC2)C1 29684,c1(C(=O)NCC2N(C(C3=C(C)OCC3)=O)CCOC2)ccc([N+](=O)[O-])c(F)c1 29685,C1(NC)CCN(C(=O)C=O)C(C)C1.n1(CC)nc(NCC2CC2)cc1C1CC1 29686,C=CCC(CC=C)C(=O)N1CC(NC(c2ccc(OCC)cn2)=O)CCC(O)C1 29687,C(=O)(C(C)(C)C(F)F)N(C)CC1CN(C(C(C)SC)=O)C1 29688,CCC(C)(CNC(C1CC(C)(C)C1)=O)NC(c1snnc1C1CC1)=O 29689,c1(CNC(C2CC(NC(COCCOC)=O)C2(C)C)=O)ccc(O)c(C)c1 29690,c1(C(C)=O)ccc(C(N2CCCC(C)C2)=O)cc1F.C1(=O)C(=O)NCCN1.C(C#N)S 29691,c1(NC(CC(C=CC)OC)=O)ccc(S(=O)(=O)CCNC(=O)OC(C)(C)C)cc1 29692,C1(COC)CN(C(c2cc(F)c[nH]2)=O)CCN1C(=O)CCCc1ccc(O)cc1 29693,N1(C(C2CC(SC)C2)=O)CC2CC(NC(=O)CC3(O)CCCC3)CC(C2)C1 29694,c1(C2CCN(CC3CCN(Cc4c(Cl)c[nH]n4)CC3)C2)cccc2c1OCO2 29695,c12ccc(cc1CN1CCCC1CCC(=O)OC)o2.N1(CC)CCCC(C)C1 29696,c12sc(C)cc1NC2=O.N1(CCN(C(CNC(=O)OCC)=O)C)CCC(C)C1 29697,Cc1cc2ccc(C(N3CCC(NC(c4[nH]c(O)nc4C)=O)CC3C)=O)cn2c1 29698,N1(C(C2N=C(C)SC2)=O)CCOCC(CNC(=O)Cc2cccc(N)c2)C1 29699,C1(C(N2CC=CC(C(=O)NCCC3CC(F)(F)C3)C2)=O)C2CCC(F)(F)C12 29700,C(=O)(C(C)CC(F)(F)F)NCCN(CC(C)O)C(c1ccn(C(C)C)n1)=O 29701,c1(C(=O)NC(C(C)NC(c2c(C)cc(F)cn2)=O)CO)cnc2c(c1)COCC2 29702,C1(C(=O)NCCOCCCNC(=O)Cn2cccc2)CC(=O)N(c2cn[nH]c2)C1 29703,c1(CC(=O)NC2C(CNC(CN(S(CC)(=O)=O)C)=O)C2)ncc(C)s1 29704,c1(NC(=O)Nc2cc(C)c(Br)cn2)cc(C(F)(F)F)cc(S(C)(=O)=O)c1 29705,C1(C)(C(=O)NCC(C)(CO)NC(CC2CC(=C)C2)=O)CC(=O)N(C)C1 29706,c1(C(N(CCCNC(C(CC)C)=O)Cc2ccccc2)=O)nc(C)ccc1F 29707,c1(C(N2CC(c3cn(CC(C)(C)O)nn3)C2)=O)snc(-c2ccccc2)c1Cl 29708,CCCCC(O)C(C)C(=O)NCCCC(=O)N(CC(C)OC)C 29709,N1(C(c2c(CNC(COCCOC)=O)c[nH]n2)=O)CC2C(NC(C)=O)C2C1 29710,C1(C)(CC)NC(=O)N(CC(=O)NC(C)C(C)NC(c2c(Cl)n[nH]c2CC)=O)C1=O 29711,C(=O)(C(C(C)C1CCC1)N1CCC2CC12C)NC(C(=O)OC)Cc1ccccc1 29712,CC(C)C(F)(CNC(C1CCCCCN1C)=O)C(=O)NCC1CCC1(F)F 29713,C#Cc1ccccc1CC(=O)NC(C)CN(C(=O)C(O)C=CC(C)C)C 29714,Cc1cc(C)n2nc(C(N3CCC3CNC(=O)C3=CCCCO3)=O)cc2n1 29715,C1(CNC(c2scc(C)c2C)=O)CN(C(c2ccc(C(F)F)o2)=O)CCC1C 29716,N1(C(=O)NC(c2cnn(C)c2)C(C)C)CCOC(C)(CO)C1 29717,c1(C(=O)NC(CC#N)CO)cc(I)c(F)cc1F 29718,C1(NC(CCC(=O)OC(C)(C)C)=O)CC2CC1CN2C(c1cnc(C(N)=O)s1)=O 29719,CC(O)C(C(=O)NCC1(CO)CC1)NC(C1CC(F)(F)C1)=O 29720,c1(-c2nc(COC)nn2-c2cccc(OC(F)(F)F)c2)cnn2ccc(O)nc12 29721,N1(C(CC)=O)CCCC2(CCN(C(C3CCn4nccc4C3)=O)C2)C1 29722,C=CC1(CNC(C2C(CC)CCCN2C(c2sccc2F)=O)=O)CCOCC1 29723,C1(NC(C2C(OC)CCC2)=O)CN(C(C2CCCCO2)=O)CCC1C(F)(F)F 29724,CCCCCCC(=O)NCC(C)(C)CN(C)C(C1CCCSC1C)=O 29725,c1(NCC23N(C(=O)OC)CC(C2)OC3)nc2ccccc2nc1C 29726,c1(C(=O)NCCCC2N(C(C(CCCC)O)=O)CCC2)c(C)nc2sc(C)cn12 29727,C(CCC(C)C(=O)NCC12CC(CO1)N(C(=O)CCc1nc(O)n[nH]1)C2)OC 29728,c1(C(=O)NCCCCNC(=O)Cc2cccnc2)cc(O)c2sccc2c1 29729,C1(CNC(CC(C)n2ccnc2)=O)C(C)CCCN1C(=O)CC1(O)CCCOC1 29730,c1(NC(C2CSCCN2C(c2ccc(Br)s2)=O)=O)cccc(O)c1F 29731,c1(C(N2CC(O)(CNC(c3c(C)cc(F)s3)=O)C2)=O)cc2ccc(Cl)cc2o1 29732,N1(C(C2(CC)CC2)=O)CCCC2CN(C(=O)C(=O)Nc3ccc(C)cc3)CC12 29733,C(C(CC1CC1)C(=O)NCC(C)(C)OC)NC(C(C1CCCC1)OC)=O 29734,n1(CCS(N)(=O)=O)nc(-c2ccc(Cl)nc2)nc1C1CCC(=O)N1C1CCCC1 29735,N1(C(C(CNC(c2ccc(C)nc2O)=O)O)=O)CC2OCC(C)C2C1 29736,c1(C(=O)NC2CN(C(c3c(C#C)cn(C)n3)=O)C2)ccc2c(O)nc(C)nc2c1 29737,CCC(C#N)(CC)C(=O)NCC(O)CNC(C1(OC)CC1)=O 29738,C(=O)(CCCCCCNC(C1CCOC1(C)C)=O)NCC(C(C)O)C 29739,c1(C(=O)NCC(CC)NC(C2(O)CCCCC2)=O)cn(C)nc1C(C)(F)F 29740,N1(C(C2CC(NC(CCC3(C#N)CCC3)=O)C23CCC3)=O)CCOC2COCC12 29741,C1(COC)(CNC(c2csc(C)c2N)=O)CCN(C(=O)C(C)c2ccsc2)CC1 29742,N1(C(C(C2(C)CC2)NC(C(COC)C)=O)=O)CC2(CC(C)CO2)C1 29743,C1(OC)CC2CCC1CC2C(N1CCC(N(C)C(c2ccc(C)c(C)c2)=O)C1)=O 29744,c1(C(=O)NC2C(NC(C3(C=C)CC3)=O)CCCC2)cc(C)nc(O)c1 29745,N1(C(C2COCCO2)=O)CC2C(NC(C3(C(F)(F)F)CC(F)(F)C3)=O)C2C1 29746,C(N=c1cc(CC2CC2)nc[nH]1)C1(F)CC(NC(CC(C(C)C)O)=O)C1 29747,c1(C(=O)NC(C)CN(C(=O)C(c2ccc(C#N)cc2)C)C)sccc1S(C)(=O)=O 29748,c1(OC)ccnc(C(=O)NCC2CCCCN(C(=O)C(C)n3ccnc3)C2)c1F 29749,c1(C(=O)NCC(C)CN(C)C(c2cc3nc[nH]c3cn2)=O)cncc2sccc12 29750,N1(C(=O)OC(C)(C)C)CCCC(Nc2ccccc2)C1.N1(C(=O)O)CCCC1(C)C 29751,C1(C(N2C(C=C)CC2)=O)(NC(=O)CCOC(C)=O)CCCC1C 29752,CN1CCN(C(=O)CCC2NC(=O)NC2=O)C(CNC(=O)C(C2CC2)C2CC2)C1 29753,c1(N2CCC(CCNC(=O)C(c3ccccc3)O)CC2)ncc2cccnc2n1 29754,N(C(=NCCNC(C)=O)N1CCCC2(CC2)C1)Cc1c(CC)oc2ccccc21 29755,C1(NC(c2nccc(C)c2)=O)CC(CNC(=O)C=Cc2cnc[nH]2)C12CCC2 29756,C(=O)(CC(C(F)(F)F)OC)NC1C(CNC(c2cc(OC)nc(Cl)c2)=O)CC1 29757,c12ccc(cn1)NC(=O)N2c1cccc(-c2nn[nH]n2)c1.c1(OCC)cnsc1 29758,C1(C)(CN(C(=O)NCC(c2ccc(Br)cc2F)C)C)C(C)(C)C1(C)C 29759,C1(NC(C=C(C)C(C)C)=O)C2CC1N(C(=O)CC(c1ccccc1)NC(N)=O)C2 29760,C(N=c1[nH]c(N(C)CCc2nccs2)nc2c1SCC2)c1n(CCC)ccn1 29761,CCCC(C#N)C(=O)NCC1(F)CC(NC(=O)CCc2cncn2C)C1 29762,C(=O)(CC(F)(F)CC)NC(CCC)C(=O)NCCCSCCO 29763,N1(C(c2ccc(CC)nc2)=O)C(C(=O)NCC(CC2CC2)OC)CCC12CC2 29764,c1(OC)ncnc(N2CCC3(CC3C(=O)Nc3ccc(O)cc3C(N)=O)C2)c1C 29765,N1(C(C(CC#C)(C)C)=O)CCC(C2CCCN(C(C3(CC)CCC3)=O)C2)CC1 29766,N1(C(c2cc(C(C)C)ncc2)=O)CC2CCC(C1)N2C(=O)Cc1cnn(C)c1 29767,C1(C(N2CCC(NC(c3cnn(C)c3Cl)=O)C2)=O)Cc2ccccc2CO1 29768,Cc1nn(C)cc1C(=O)N(C)CCNC(=O)CN1CCCCC1=O 29769,CCC(C)C(C(=O)NCCc1nc(C)no1)NC(=O)CC(C)n1cccc1 29770,CC(C)CCCC(C)C(=O)NC1C2CC3C(C2)C13C(=O)N(C(CO)C1CC1)C 29771,c1(C(N(C2CCN(C(C(=CC3CCCC3)C)=O)C2)C)=O)nc(Cl)c(Cl)s1 29772,C1(NC(C(C)Cc2ccccc2)=O)COCCN(C(c2cnc(S)n2C)=O)C1 29773,CCCCC(=O)C(=O)NCC=CC(N1CC(S(C)=O)C1)=O 29774,C1(C(=O)NCc2ccc(N3CCCCC3)nc2)CCC2(CCC2)NC1 29775,N1(C(CCSCC)=O)CC(NC(c2cc(C)n(CC(F)F)c2C)=O)CC1(C)CC 29776,C(=O)(CS(=O)(=O)C(C)(C)C)NCC12CC(NC(CC(CC)C)=O)(C1)C2 29777,CCCC(CC)C(=O)N1CCC(CNC(c2csc(CC)n2)=O)C12CC2 29778,C(=O)(CCC(F)(F)C(=O)N1CCCCC1CNC(C1(C)CNC(=O)C1)=O)OCC 29779,N1(CCNC(C=CC2(C)COC2)=O)CCC(NC(C2CC=CCC2)=O)CC1 29780,Cc1nc(C(C)(C)C)sc1C(=O)NCC1(NC(C2CCCC2)=O)CCCC1 29781,C(=O)(CC(O)CC(C)(C)C)N1CCC(N(C(c2cncc(C)c2)=O)CC2CC2)C1 29782,c1(C(N2C(C)CC(NC(=O)C3=COCCO3)C2)=O)cccc2c3c([nH]c12)CCC3 29783,C(CO)(CCF)NC(C(C)N(C(=O)C=C1CCC1)C1CC1)=O 29784,Cc1cccc2c1c(C(c1nnnn1C)NC(C)CC(F)(F)F)cn2C 29785,c1(C2(C(=O)NC(C)CN(C)C(C3(C)CC3Br)=O)CC2)ccccc1 29786,Cc1oc(C#N)cc1C(=O)NC1CCC(NC(=O)CCC2(C)NC(=O)NC2=O)C1 29787,CCC(CC(=O)N1CCCC1(C)CNC(=O)CC1(C)CCOCC1)C(C)(C)C 29788,CC1(C)OCCC1CC(=O)NC1CCCC1NC(c1ncccc1O)=O 29789,N1(C(c2c(C)n(C)cc2)=O)CCCCC(NC(c2ccc(CO)s2)=O)C1 29790,Cc1ccc(O)nc1CNCC1CCCN(CC2CC2)C1 29791,N1(c2cc(=NC)[nH]cc2)CCC2(CC1)COC(C(=O)NCCN(C)C)C2 29792,N1(C(CC(=O)OCC)=O)CCC(NC(=O)Cn2nnc(C)n2)CC(C)(C)C1 29793,N1(C(c2c(C)nn(C(C)(C)C)c2)=O)CC2CCC1C2NC(=O)COC(C)C 29794,C1(C(=O)NC2CN(C(c3c(C)onc3)=O)CC2(C)C)Cc2ccccc2S1 29795,C(C1=NOC2CCCC12)NC(C(=O)N(C(COc1ccc(C)cc1)C)C)=O 29796,C(=O)(CC(F)(F)C(F)F)NC(CN(C(C1CC(C)(C)C(C)(C)C1)=O)CC)C 29797,c1(C(=O)NC(CCCCNC(COCCC=C)=O)C)ccnc(Cl)c1OC 29798,CCCC(CC)C(=O)NCC1CCC1NC(=O)COC1CC=CC1 29799,C12(C(=O)NCC(CC)(C)OC)CC(CN1C(=O)CCOCC(C)(C)C)C2 29800,C(=O)(CC(C)P(C)(C)=O)NCC(CNC(CCCC(=O)NCCC)=O)(C)F 29801,Cc1cc(=NCCC2C(C)CCCN2C(c2cn(C3CC3)cn2)=O)[nH]c(CO)n1 29802,N1(C(C#C)C)CCCN(C(c2cscc2Br)C(=O)NC2(C)CC2)CC1 29803,N1(C(C(c2ccc(C)cc2)C)=O)CC2=C(C1)CN(C(c1c[nH]cc1C)=O)C2 29804,C12(C(=O)NC3(C(=O)OCC)CC3)CCC(CN(C(=O)C3=NOCC3)C1)C2 29805,CCCC(C)(CCC)C(=O)NC1CN(C(=O)CCN(C)C(C)=O)CC1C1CC1 29806,C(CC1=CCN(C(c2cc(C#N)c[nH]2)=O)CC1)NC(C(C1CC(F)(F)C1)OC)=O 29807,c1(C(N2C(CNC(C3CC(=O)N3)=O)CC(C)(C)C2)=O)cnc(O)c2ncccc12 29808,Cc1nc2ccnn2c(C)c1C(N1CCN(C(c2cnc(O)n2C)=O)C(C)C1)=O 29809,Cn1cnc(C(O)CNC(=O)CC2(NC(C3CC(F)(F)C3)=O)CC2)c1 29810,Cc1ccc(C(=O)NC2(CNC(=O)Cn3nnc(=N)[nH]3)CC2)cc1C(C)(C)C 29811,N1(C(c2cc(SC)oc2)=O)CCN(CC(C)NC(=O)CCCCN(C)C)CC1 29812,C1(CNC(c2c(C)cco2)=O)CN(C(=O)CCCCN(C)C)CC12CCC2 29813,c1(C(N2CC(NC(CCS(C)=O)=O)C(O)C2)=O)cn2c(Br)cccc2n1 29814,C1(CNC(C2(C)N(Cc3n(C)cc(Br)n3)CC2)=O)CCC(F)(F)CC1 29815,C1(CC(=O)NCC=CCNC(CCCc2n(C)cnn2)=O)(N(C)C)CCOCC1 29816,c1(C(N2C3CC(C(N(CC(C)C)CCC)=O)C2CC3)=O)ccc2cc[nH]c2c1 29817,CC1OC2(C(=O)NCCC(C)(C)NC(c3cnn(C)c3Br)=O)CCC1C2 29818,N1(C(C#CC2(OC)CC2)=O)CCN(C(=O)CSC2Cc3ccccc3O2)CCC1C 29819,C1(C(=O)NCCCCC(C)NC(c2c(SC)ccs2)=O)C2CCC3C(C2)CC13 29820,Cc1c(Br)c(C(N2CCC(CNC(=O)C(C)N(C)C)C23CC3)=O)nn1C 29821,C1(C(=O)NCC2CCC(NC(Cn3c(C)c(Cl)cn3)=O)C2)CCC2(CCC2)CC1 29822,C(=O)(C1=CCOCC1)N1CC(C2CN(C(CCC3(C)CC3)=O)C2)OCC1 29823,C1(CC(=O)NC(C(C)C)CNC(=O)CCN2CCCC2=O)CCCS(=O)(=O)C1 29824,c1(C(=O)NCCCCNC(CSCCOC)=O)cc(C)ccc1C1CC1 29825,c1(CC)cccnc1C(=O)NCCCN(C(=O)C(=Cc1ccccc1)C)C1CC1 29826,Cc1ccc(C(N2CCCCC2CC(=O)Nc2ccnc(F)c2F)=O)c(I)c1 29827,N1(C(Cc2cccc(CC)c2)=O)CCC(NC(C2CC(=O)N(C)C2)=O)C(O)C1 29828,C(=O)(CC(C)(C)C#N)N1CCCC(C(C)NC(CCC(=C)C)=O)C1 29829,C1(CNC(C=Cc2c(C)nn(C)c2Cl)=O)CCC2(CC1)OCCO2 29830,n1(CC)ncc2c(NC3CCCC(CNC(=O)C(F)(F)CC(C)C)C3)ncnc12 29831,C12(C(=O)NCc3c(C)nccc3)COCC1CN(C(=O)C1CC1)C2 29832,C12(C(=O)NCCc3cncc(C)n3)CC(CN(C(C3(C)CCOC3)=O)C1)C2 29833,CCCCCC(C)(C)C(=O)NCCC1(C)CCN(C(=O)CC2CCCO2)CC1 29834,Cc1c(C(=O)NC2CCN(C(=O)C(F)(F)C(C)(C)O)CC2O)nn2c1CCCC2 29835,c1(OC)ccc(C2CCN(C(=O)NCCNC3COCCC3O)CC2)cc1 29836,N1(C(c2nn(CC)nc2C)=O)CCC(NC(c2cc(Cl)sc2Cl)=O)C(CO)C1 29837,N(C(=NCCCC(=O)OC(C)C)N1CCCc2ccccc2CC1)C(C=C)C 29838,CC1(C)CC2(CC2C(=O)NCCCNC(c2cnc(Cl)[nH]2)=O)C1 29839,C1(CNC(C2CCN2Cc2ccccc2)=O)CC(O)CN1C(C1CCC(O)C1)=O 29840,c1(OC)c(C(=O)NC(C2CCCN2C(=O)CC2(OC)CCCC2)C)ccnc1F 29841,C1(C)(C(=O)NCC(CNC(CCOc2c(C)cccc2)=O)C)CCS(=O)(=O)CC1 29842,c1(C(=O)NC(CC(C)C)CNC(=O)C(F)=CCCF)cc(Cl)ccc1C(C)C 29843,C(CCC)(C(=O)NC1CCN(C2CN(C(=O)C=Cc3cccs3)C2)CC1)=CCC 29844,Cc1cc(CO)ccc1-c1cn(C(C)CNC(=O)C(c2ccccc2Br)O)nn1 29845,C1(C2CC2)(CNC(CCOc2ccn(C)n2)=O)CCN(C(C2CC(F)C2)=O)C1 29846,C1(C2CCN(C(=O)C(F)C(C)C)CC2)(NC(c2ccnc(OC)n2)=O)CCC1 29847,C1(NC(=O)Cn2cc(C3CCC3)nn2)CN(C(=O)C2CC2)C2(CCCC2)C1 29848,N1(C(c2cnc(C(C)=O)s2)=O)CC2(CC(NC(C3COCCC3(F)F)=O)C2)C1 29849,C#CC1CCCN(C(=O)C(C)(C)NC(C2CC3(CCC3)C2)=O)CC1 29850,C1(C(N2CC(CC=C)(NC(C3CNC(=O)N3)=O)C2)=O)CC(C)(C)CO1 29851,c1(C(=O)NCCC(C)NC(=O)C=Cc2ccc(F)cc2)cc2c(Cl)cccc2[nH]1 29852,N1(C(COC(CC)C)=O)Cc2[nH]nc(C(=O)NCc3cc(C)sc3C)c2C1 29853,c1(CC(=O)N(C2CCN(C(=O)C3=COCC3)C2)CC)cc(C)ccc1F 29854,Cc1cc(C(=O)NC2(C(=O)NCCC(C)(C)C)CCC2)c[nH]1 29855,CC1CC(c2ccccc2)(C(=O)N(CCCN(C(=O)CC2CCCO2)C)C)C1 29856,C(=O)(C(CC=C)CC=C)NC(C(=O)N1CC(OCC#C)C1)CCF 29857,c1(CCC)[nH]nc(C(=O)NC2CN(C(C3CCN(C(=O)NC)C3)=O)C2)c1[N+](=O)[O-] 29858,CC1CCCN(C(=O)CC2CCCC2C)C1CNC(c1cnc(C#N)s1)=O 29859,N1(C(C(=C(C)C2CC2)F)=O)CCC2(CC1)CC2NC(c1ccc(CO)c(Cl)c1)=O 29860,C1(N(C(C2C3COCC23)=O)CC)CCCN(C(c2cocc2C)=O)CC1 29861,c1(C(C2CC2)C2CC2)ccc(C)o1.C1(C(COC)NC(=O)N)CCCOC1 29862,C1(C(=O)NC2C(NC(C3(CCCC)CCC3)=O)CC2)CCSCC1 29863,N1(C(C=CC(C)Sc2cccnc2)=O)CCC(C(=O)O)CC1 29864,c1(C(N2C(C(C)NC(=O)CCc3cncnc3)CCC2)=O)c[nH]c2ncccc12 29865,Cc1cc(=NC2CCC(=O)N(C)C2)[nH]c(N2CCC(C(F)(F)F)C(CO)C2)n1 29866,C1(C(=O)NC(CCNC(CC(CC)OC)=O)(C)C)CC12CCS(=O)(=O)CC2 29867,C1(C(=O)NC)C=CC(NC(CCSc2nnnn2C2CC2)C2CCCO2)C1 29868,C1(CNC(C(CC(=C)C)NC(C)=O)=O)CN(C(=O)C2=NOCC2)CC2(CCC2)O1 29869,C1(CCNC(c2c(C)cc[nH]2)=O)CN(C(c2ccnn2C(F)F)=O)CC1C 29870,C(CCCC(=O)N1CCCC1(C)CNC(=O)C(=Cc1cnc[nH]1)C)OCCC=C 29871,C1(NC(c2ccc(CO)cc2)=O)CCC(NC(=O)C(F)Cc2ccccc2)CC1 29872,C1(c2nnnn2CCOC)(Nc2cn(CCCC)nn2)CC2CCCCCC2C1 29873,c1(C(N2CC3C(CNC(CC)=O)C3C2)=O)oc2ccccc2c1CS(C)(=O)=O 29874,C1(C(=O)NC(C(=O)N(CC(C)OC)C)Cc2ccco2)CCCCN1C 29875,c1(C(=O)NCCC(C)NC(Cc2ccn(CC)n2)=O)cc(C(C)=O)c(C)nc1C 29876,C12(C(N(CCNC(C(CN(C)C)O)=O)C3CC3)=O)C3CCC(CC13)C2(F)F 29877,CC1CCC(CNC(c2cnc(N(C)C)cn2)=O)CN1C(=O)C=CC1CC1 29878,C1(NC(C(CC#C)(C)NC(C2CC(N=[N+]=[N-])C2)=O)=O)CCCCN(C)C1=O 29879,C(CC(C)(C)C)(C(=O)N1CC(CC(=O)NC2(COC)CC=CC2)C2(CC2)C1)OC 29880,C12(CCOCC1)C(=O)NC(C)C(=O)NCCO2.C(CCNC1CCC1)SC 29881,Cc1ocnc1C(=O)NC1CC(F)(CNC(C2CC(O)(c3cccnc3)C2)=O)C1 29882,c1(C(N(CC(C)NC(=O)C=C(C)C)CC)=O)ccc(OC)cn1 29883,C#Cc1cccc(C(N2CCC(CN(C)C(C3CC(=O)NC3(C)C)=O)C2)=O)c1F 29884,Cc1noc2nc(C(=O)NC(C)Cn3cc(C4CCCO4)nn3)ccc12 29885,N1(C(=O)OC(C)(C)C)CCCC(C(F)(F)F)(CCn2nc(Br)cc2Br)C1 29886,c1(CN2CCC(CC(=O)N(C)CCO)CC2)cccc2nonc12 29887,CCCC(CC(C)C)C(=O)NC1CC(NC(=O)CCCC(F)(F)F)CC1O 29888,C(=O)(CCCC(=O)Nc1ccccc1)N1CCC(CNC(C2C(OCC)C2)=O)C1 29889,N1(C(C(CC=C)C)=O)CCC2C(C1)CN2C(C12CC(c3ccccc3)(C1)C2)=O 29890,CCCCCC(C)CC(=O)NC1C2CCC1N(C(=O)C1=NNC(=O)CC1)C2 29891,Cc1noc(N)c1C(N1CC2CC2(CO)C1)=O.c12cn(nn1)CC(=O)NC2 29892,C(CNC(=O)C(O)CN(C)C)(CC(=O)Nc1ccccc1Cl)OC 29893,C(=O)(C(CC)C(=O)NC(C)Cn1cccn1)OCC 29894,CC1CN(C(=O)CCn2ncn(C)c2=O)CC1CNC(=O)C(C)OCC(F)(F)F 29895,Cc1cc2ccc(C(=O)NCC3(O)CCN(C(=O)Cc4ccoc4)CC3)cc2o1 29896,N1(C(c2c(C)snn2)=O)CCC(CCCNC(C2(P(C)(C)=O)CC2)=O)CC1 29897,N1(C(c2c(C)cns2)=O)CCC2CCN(C(c3cc4n(n3)CC(F)C4)=O)CC12 29898,c1(C(=O)NCCOCCNC(=O)Cc2cccc(Cl)c2Cl)cccc2ncnn12 29899,c1(C(N2CCN(C(C(=O)NCC3CC3)=O)CC2C2CC2)=O)nccn2ccnc12 29900,C1(NC(CCCC(C)C)=O)CC(NC(c2csc(=N)[nH]2)=O)C12CCOCC2 29901,C1(C(=O)NC2CCC(NC(CCC(N)=O)=O)CC2)CCN2CCC1C2 29902,C1(C2CC2)(CNC(COCCCC)=O)CCN(C(c2cnn3c2OCCC3)=O)C1 29903,C=C(C(=O)OCC=CC)C(C)(C)C.c12ccc(cc1)CCC(=O)N2 29904,CC1(C)CNC(=O)c2c(C(=O)NCC3CC(NC(=O)CC4CC4)C3)coc2C1 29905,Cc1ccc(-n2nc(-c3ccoc3)nc2CC2CC(C)C2)cc1Cl 29906,O(S(=O)(=O)C=Cc1ccccc1)C1CCCN(C(=O)OC(C)(C)C)C1 29907,c1(N2CC(NC(C3(C(F)(F)F)CCC3)=O)C(F)CC2)ncnn2ccc(Br)c12 29908,C(=O)(C(C(C)C)c1ccncc1)N(CCCNC(C(c1ccnn1C)OC)=O)C 29909,C(CCNC(c1ccc(C(C)C)s1)=O)(C(C)C)NC(C1(CC)CCCO1)=O 29910,c1(OC)cc(CC(N2CC(O)(CN(C)C(c3cnc(CC(C)C)s3)=O)C2)=O)on1 29911,N1(C(c2cc(C(C)=O)on2)=O)CCC(F)(CNC(C2(CF)CC2(F)F)=O)C1 29912,c1(C(C(=O)NCCCN(C(CCC(=C)Br)=O)CC)O)ccc(C#N)cc1 29913,C1(C(N(CC(C)NC(CS(=O)(=O)NCC)=O)CC)=O)CCCC2(CCOCC2)O1 29914,c1(C2(C)CC2)ccc(OCC(N2CC(CO)(NC(C3CCCN3C)=O)C2)=O)cc1 29915,C(=O)(CC1=CCOCC1)N(CCCNC(=O)Cc1cccnc1O)C(C)C 29916,C(=O)(C1c2c[nH]nc2CN1C(c1ccc(C(N)=O)o1)=O)N(C1C(C)COCC1)C 29917,C1(C#N)(C(=O)OC)CCN(C(=O)CSC2CCOC2=O)C1 29918,CCC(CC(=O)NC1CCC(NC(=O)Cc2ccc(C#N)cc2F)CC1)C(F)F 29919,C(=O)(CC(O)CNC(C1CC1C(F)(F)F)=O)N(CC(CC)CC)C1CC1 29920,c1(OC)ccc(F)cc1C(=O)C(=O)NCC1CC(OC(C)(C)C)C1 29921,c1(NC(C2C(NC(C3CC3C3CCCCC3)=O)C2)=O)ccc2ncoc2c1 29922,C(=O)(C(F)CC1CC1)N(C(C)CN(C(=O)CCOC1CC1)C)C 29923,Cc1cnc(C(=O)NC2CCCCC2CNc2nccc(CC#N)n2)cn1 29924,C1(C)(CNC(C2C(C(=O)OCC)C2)=O)CN(C(c2ccc(F)c(F)c2)=O)CC1C 29925,C(CC1=CCN(C(=O)C(F)(F)C(F)(F)F)CC1)NC(c1ccc(Cl)cc1)CC 29926,N1(C(C(C(C)C)n2cccc2)=O)CCCC(NC(C2CC2F)=O)CCC1 29927,N1(C(CCSC)=O)CCc2c(C(=O)Nc3cccc(C(F)(F)F)c3F)n[nH]c2C1 29928,CC1CCCN(C(c2cnc(C(F)F)s2)=O)C1CCNC(=O)CCNC(N)=O 29929,c1(CC)ccc(F)c(C(=O)NCC(O)CNC(c2c[nH]c(=N)o2)=O)c1 29930,C1(CN(C)C(c2[nH]nnc2C2CC2)=O)C=CC(NC(=O)CC2CCCC2)C1 29931,c1(NCCC2CCN(C(C3(COC)COC3)=O)C2)ncnc2scc(C)c12 29932,C(C(CNC(C1SCCS1)=O)S(C)(=O)=O)NC(CCNC(=O)NC)=O 29933,CC1CCCCC1OCC(=O)NCC(=O)N(CCCNC(c1csc(Cl)c1)=O)C 29934,N1(C(C(C=C)(F)F)=O)CCCN(C(C2CC3CCC(C2)C3O)=O)C(C)C1 29935,CCCC(C)(CC)C(=O)N(CCCCC(=O)NC1(C(=O)OC)CC1C)C 29936,c1(C(=O)Nc2ccc(OC(C)C)cc2Cl)cccc2oc(O)nc12 29937,c1(C(N2CC3CNC(=O)C3C2)=O)c(F)c(F)c(Cl)c(F)c1F 29938,c1(OC)ccc(F)cc1C(=O)NCCC(C(C)C)NC(=O)C1=CCSC1 29939,c1(C(N(CC(CNC(C2(COC)CCC2)=O)C)C)=O)cccc2c1CC(=O)N2 29940,C12(C(=O)NC(CC=C)C)CC(C)(CN1C(c1c[nH]c(=N)c(C)c1)=O)C2 29941,C1(OC)(CN(C)C)CCN(C(=O)C(CCSC)NC(=O)C(C)OC(C)=O)C1 29942,N1(C(Cc2c(F)ccc(OC)c2)=O)CC2CCCC2(NC(=O)CC(O)C(C)C)C1 29943,CC(=O)CCN=C(NCCC1(CO)CCC1)N1CCN(c2cccc(F)n2)CC1 29944,c1(CC(CNC(C(=O)N(CC)Cc2cccnc2O)=O)CO)ccc(Br)c(F)c1 29945,c1(NC2(C(=O)NCCCC3(OC)CC3)CCCC2)ccc(F)cc1N 29946,OCCC(N=c1[nH]c(=NC2CCCCC2F)[nH]c2ccsc12)C1CCOCC1 29947,C#Cc1ccc(C(=O)NCC2(COC)CCCN2C(C2CC2CC)=O)c(C)c1 29948,C(=O)(C(O)CC(C)C)N(CCOC)CCNC(=O)CCCc1cnn[nH]1 29949,Cc1nc(C(c2nnnn2-c2ccccc2)NCC2CCN2C(C)(C)C)sc1C 29950,c1(OCC=C)ccc(Cl)c(C(N2CC(F)(F)CC2CNC(=O)CC(C)(C)O)=O)n1 29951,N1(C(CCCCCNC(C(C)C#N)=O)=O)CCc2c(C#N)cccc21 29952,C1(C(C(=O)NC2(CNC(C3(COC)CC=CC3)=O)CC2)C)CCC(C)(O)CC1 29953,N1(C(c2c(OC)nn(C)c2)=O)CCC2(NC(=O)CCc3cnn[nH]3)CC2C1 29954,n1(CC)cc(CC(=O)NCC(C)(C)NC(C2(C)CCCO2)=O)cn1 29955,c1(C(=O)NCC2(C(C)NC(CNC(CCC)=O)=O)CC2)cn(C(C)(C)C)cn1 29956,C1(O)(CN(C(C(=O)NCC)=O)CC)CCN(C(=O)CCOCC(C)C)C1 29957,C(=O)(CCCCC(N)=O)N1CCCC(CCCCNC(C(CN(C)C)O)=O)C1 29958,c1(C(N2CC(NC(c3c(CC)con3)=O)C(O)C2)=O)cnc2ccc(C#N)cn12 29959,c1(N2CCC(OCC)CC2)[nH]c(=NCc2ccc3ccsc3c2)nc2scnc12 29960,Cn1cnc2c(N3CC(CNC(c4cn(CC5CCOC5)nn4)=O)C3)ncnc12 29961,C(CCCC(C)(C)C(=O)NNC(=O)CCCCC(C)C)OC(C(=C)C)CC(=O)OC 29962,N1(C(C2CCN(C(CC3CCCC(C)O3)=O)C2)=O)CC(C)CCC12CC2 29963,N1(C(Cn2c(C)nnn2)=O)CCCCC(CNC(=O)Cc2ccc(Cl)nc2)C1 29964,c1(C(=O)NCC(C(C)C)NC(=O)C(C)(C)c2ccccc2)nn(C)cc1Cl 29965,c1(C(=O)NC2CN(C(C(CC)Sc3ccccc3)=O)CC2O)cc(F)cnc1O 29966,c1(C(C)(C)C)cncc(C(=O)NCC(=O)NCCCOCC(F)F)c1 29967,N1(C(C2(C)CCN(Cc3c[nH]ccc3=N)C2)=O)CCc2ccc(C#N)cc2C1 29968,C(C(C(=O)NCC1CCCO1)N(C)Cc1cocn1)(C1CCCC1)OC 29969,C(c1ccccc1)=CC(=O)NCC(CN(C(c1cc(CCC)[nH]n1)=O)C)O 29970,Cc1cc(C(N2CCCC(C)(NC(C3CC(CF)C3)=O)C2)=O)cc(N)c1Cl 29971,C1(NC(=O)CC2CC(C)(C)CN2C(=O)CC2CC2(C)C)CC(C)(C)C12CCC2 29972,c1(C(c2n(CC=C)nnn2)NCc2ccc(CO)o2)ncccc1Br 29973,c1(C(=O)NCC2(F)CCC(CNC(C3C(C)C3)=O)C2)n[nH]c2c1CS(=O)(=O)CC2 29974,CCC(C(=O)NCCC(C1CN(C(=O)CC2(C)CCCC2)C1)C)NC(N)=O 29975,N1(C(C2C(CCC)C2)=O)CCC(C(=O)NC2C=CCCC2CO)CC1(C)C 29976,c1(C(C(=O)NCC(C)N(C(=O)C(O)P(C)(C)=O)C)=O)cc(Cl)cc(Cl)c1 29977,c1(N(C)CC)cccc(S(=O)(=O)N(CC(C)(C)S(C)(=O)=O)CC)n1 29978,CC(C)CCC(O)C(=O)NC1CCC(CC(=O)NCC(O)CNC(N)=O)CC1 29979,C(=O)(CCC(C)(C)OC)NCC(CNC(C(CC)OC)=O)(C)C 29980,c1(C(=O)NC2C3CN(C(c4ccc(OC)o4)=O)CC32)cc(OC)cnc1C 29981,C(CCCCNC(c1cc(C2CCOC2)[nH]n1)=O)N(C(C(C)C1CCC1)=O)C 29982,C(CCCC(=O)NC(COC)CC(=O)NC(C)Cc1nc[nH]n1)OCC 29983,c1(C(=O)NCCN(C2CCCC2)C(c2c(COC)cc[nH]2)=O)ccn(C)c(=O)c1 29984,CCCCC(O)C(=O)N1CC(NC(=O)CCc2ccc(F)cc2)C2(CC2)C1 29985,CC1C(C(=O)NCCN(C)C(c2cc(CF)on2)=O)CCN1C(=O)OC(C)(C)C 29986,C1(F)(CNC(c2nc(CC)oc2)=O)CCC(NC(C2CNC(=O)C2)=O)C1 29987,C1(NC(C(C)(C)C)=O)CCCCN(C(c2cnc(Br)c(N)n2)=O)C1 29988,N1(C(CCNc2ccc(C)cc2)=O)CC(CNC(c2cc(C)on2)=O)CCC1C 29989,C(c1cc(F)c(F)c(F)c1)=CC(N1CCN(C(CC(C)SC)=O)CC1CF)=O 29990,c1(OCC)ncccc1C(=O)NCCOCCCNC(=O)C(CC)n1ccnc1 29991,O=C1CN(C(C2CCSC2)=O)C(C(=O)NCc2nccc(O)n2)CN1 29992,Cn1ccc(-n2cnc(C(=O)NCCCn3cc(CC(O)C4CC4)nn3)c2)n1 29993,C1(CNC(CNC(=O)NC)=O)CC2(CCC2)CN1c1cc(Cl)nc(COC)n1 29994,c1(C(N(CC(CNC(C2(CC#C)CCCC2)=O)C)C)=O)[nH]nc2ncccc12 29995,c1(-n2cc(C3CN(C(C4CCS(=O)CC4)=O)C3)nn2)cc(F)ccc1Br 29996,N1(C(C(CCC)N(C)C)=O)CCN(C(C2(C)CCC2)=O)CC1C 29997,C1(CNC2(CC(N)=O)CCC2)CC1(Br)Br 29998,CC(O)(CNC(c1cc(CNC(C2CSC2)=O)on1)=O)CO 29999,CCN=c1ccc(C(=O)NC2CC(OC)CN(C(=O)CCCN(C)C)C2)c[nH]1 30000,C1(NC(C2C(OC)C2)=O)CC(NC(c2ccc(C3CC3)cc2)=O)C(O)C1 30001,c1(C(N2CCN(C(c3sccc3Cl)=O)C(C(F)F)C2)=O)cc2cnccc2o1 30002,C1(C(=O)NCCC(C)N(C(c2ccc(C)o2)=O)C)CC=CCC1C 30003,c1(C(=O)NC2C(NC(c3nc(COC)sc3)=O)CCC2)cnc2sc(C)c(C)n12 30004,c1(C(=O)NCCOCCOCCNC(C2C(=C)CC2)=O)cc(C)c(F)c(C)c1 30005,C1(C)(CN(C(COCCC=C)=O)C)CCCC1NC(c1sccc1SC)=O 30006,CC(C)(C)CCC(=O)NC12CCC(NC(C3CCC(C)(C)CC3)=O)(CC1)C2 30007,N1(C(c2ccc(CC)[nH]2)=O)CCC2(CC1)CC(CNC(c1cc(O)n(C)n1)=O)C2 30008,N1(C(c2ccsc2Cl)C(=O)NCC(C)C)CC(C)CC2CCCCC12 30009,Cc1ccc(C(N2CCC(CCC(=O)NC(C3CCCC3)CO)C2)=O)cc1 30010,n1(CC(C)C)nc(C)c(C(N2CCC(CC(N3CCCCC3CO)=O)C2)=O)c1C 30011,N(C(=NCCS(=O)(=O)N1CCOCC1)NCC1(C)CCOC1)C(COC)C 30012,c1(C(=O)OCC)c(C)n(CCCNC(=O)NC2(CO)CC(COC)C2)c(=O)n1C 30013,C1(C(=O)NCCN(C(=O)CC2C=CCC2)C)(OC(C)=O)CC(C)C1 30014,CC1CC(NC(C2CN(C(=O)CC3(O)CCOC3)CCO2)=O)C(=O)O1 30015,c1(C(N2C(C(=O)NCc3ccccc3)CC(OC)C2)=O)cc2cc(O)ccc2[nH]1 30016,C1(CC(=O)N(C)CCOCCCNC(=O)CC2COC(=O)C2)OCCC1(C)C 30017,N1(C(CCCc2n(C)cnn2)=O)CC2CC1CCC2NC(=O)Cc1ccnn1C 30018,Cc1ccc2nc(C)c(C)c(C(N3CC(C4CNCCO4)C3)=O)c2c1 30019,N1(CCCC)CCc2nc(C(=O)NCC3CCCN(C(=O)OC)C3)cn2CC1 30020,CC(=O)n1cc(-c2nc(NC(c3ccn(C(F)F)n3)=O)cs2)cn1 30021,CN1CC(C)(C)CC1C(N1CCC(C(=O)NCCCN2CCCC2)C1)=O 30022,CCC(N=c1[nH]c2c(c(=NC(C)c3nccnc3C)[nH]1)COC2)c1ccccc1 30023,Cn1cc(CNCC2CCCN2C(c2cccc3[nH]ccc23)=O)c2ccccc12 30024,CCC(CC)C(F)C(=O)N1CC(F)CC1CC(=O)NCc1ccc(F)c(C)c1 30025,n1(CC(=O)NCC(CNC(Cc2c(C)nsc2)=O)CO)ccc(=O)cc1C 30026,CCC(CC)CC(F)C(=O)NC1(CCNC(=O)CC(C)C(F)(F)F)CCCC1 30027,c1(C(N2C(C(=O)Nc3nc(C)ccc3O)CC(=C)C2)=O)ccc2c(c1)CCC2 30028,c1(OC)ccc(F)c(Cc2nc(C(C)SC3CC3)nn2-c2cccnc2C)c1 30029,CCCCC(O)C(C)C(=O)NC1CCCC1C(=O)NC1(C)CC(C)(C)OC1=O 30030,C(=O)(C=C1SCC(=O)N1C)N1CCCC(CNC(c2c(N)cc(C)c(C)c2)=O)C1 30031,c1(C(N2CC(NC(C(C)OCC)=O)(CO)C2)=O)c(C)nc(O)nc1S 30032,C12(CNC(=O)CC3CCC=CCC3)CCCC1N(C(c1sc(O)nc1O)=O)CC2 30033,Cc1ccc(C(=O)NC(C(=O)NOC2CC3CCC2C3)c2cccnc2)nc1C 30034,Nc1c(C(N2CC(F)(F)CC2CNC(=O)CCF)=O)cccc1[N+](=O)[O-] 30035,C1(OC)CC2CC1CN(C(C1CC(O)CN1C(c1sncc1C)=O)=O)C2 30036,c1(C(=O)NC2(CNC(CN(C3CCC3)C)=O)CCCC2)ccnc(N(C)C)c1 30037,c1(C(C(N2CC(CN(C)C(C3CCCOC3)=O)C2)=O)O)ccc(Cl)cc1 30038,CP(C)(=O)C(O)C(=O)NC1CCC(NC(=O)CN2CCC(O)CC2)CC1 30039,c1(C(CNC(C2CCC2F)=O)NC(COCCC=C)=O)ccccc1 30040,CC(CC(=O)N1CCN(C(c2cnn(CC3CCC3)c2)=O)C(CF)C1)C(F)F 30041,N1(C(C(C)OCC=C)=O)C2CCC(C2)C1CNC(c1cncc(F)c1)=O 30042,C1(C(N2C(COC)CC2)=O)(NC(C2CNC(=O)N2)=O)CCCC1 30043,C1(NC(=O)CC2CCOC2)C2CC1N(C(=O)C=CCO)C2 30044,Cc1cc(C(=O)N(C(C)CNC(c2ncn(C(C)C)n2)=O)C)c(Br)s1 30045,C1(NC(=O)Cc2cnc[nH]2)CN(C(=O)C2=CCOC2)CC2(CCC2)C1 30046,N1(c2nccc(C(N3CCNC(c4cccc(Br)c4)C3)=O)c2)CCc2ccccc21 30047,C(=O)(CC(O)CN(C)C)NCC(C)(Cn1cccn1)NC(Cc1nc(C)sc1)=O 30048,N=c1nc[nH]c(=NCCOC2CCN(C(=O)C=C3CCC3)CC2)[nH]1 30049,N1(C(C2(C#N)CCOC2)=O)CC(O)C(C#N)C1 30050,n1(CC(=O)NCCN(C)C(C2CCSC2)=O)cc(C2CC2)cn1 30051,c1(C(=O)NCC(C)(C2CCC2)NC(CSCC)=O)ccnc2ccncc12 30052,c1(CC)ccc(F)cc1C(N1CC2CC1CN2C(C1(C(C)(C)O)CCC1)=O)=O 30053,c1(C(=O)NCC(n2cc(-c3c(COC)nns3)nn2)C)cc2n(n1)CCCO2 30054,O=S(=O)(c1sccc1I)NCCOCC1CC1 30055,Cc1nc(=N)[nH]cc1CNC(=O)NC1CCN(CC2CC2)CC1 30056,C(CC(CNC(=O)C(CO)N(CC(F)(F)F)C)NC(=O)CO)OC 30057,N1(C(=O)CNC(C2(CO)COC2)=O)CCC(c2nncs2)C1 30058,c1(C(=O)NCC(CO)NC(=O)CSc2ccncc2)cc(Br)c(Cl)s1 30059,C(=O)(CCCCCc1csc(CC)n1)N(C1CC1(F)F)C(N1CCC(C)CC1)=O 30060,CCC(C)C(=O)C(=O)N1CC(C)C(C)(C(N2CC(C)C(C)C2C)=O)C1 30061,N1(C(C(CO)NC(C2N(CCC)CCC2)=O)=O)CCC2(CCN(C)C2)C1 30062,C12(C(N(OC)C)=O)CC1CN(c1ccnc(NCC3CCCCO3)n1)C2 30063,c1(C(N2C(C)CC(CNC(c3ccc(F)nc3)=O)C2)=O)ccc(F)c(N)c1 30064,c1(C(=O)NC2(CNC(CCn3ccc(C)n3)=O)CC2)cn2ccc(Br)cc2n1 30065,N1(C(CCc2c[nH]c(=N)[nH]2)=O)CCC2(CC1)CC2C(N1CCC(CF)CC1)=O 30066,C=CC(C)(CC)NC(c1cc(CNC(c2cocn2)=O)[nH]n1)=O 30067,N1(C(C)CNC(c2cc(C(N)=O)c[nH]2)=O)CCN(C(=O)CN2CCOC2=O)CC1 30068,CC(C(C)C(=O)NCCOCC(C)(C)O)NC(C1SCCS1)=O 30069,CC1CN(C(=O)C(Cl)=CCl)CC(C)C1Nc1ncnc(Cl)c1C#N 30070,Cc1nncc(C(N2CCC(C)(C)C2C(=O)NC2CCCC2C#N)=O)c1C 30071,N(C(=NCCOC1CCCCC1)NCc1ccnn1C)Cc1cccc(C)c1 30072,c1(C(N2CCN(C(C3(C)C=CCC3)=O)CC2C2CC2)=O)ccc2ccccc2c1 30073,Cc1nc(C(C)(C)CNC(=O)NCCc2ccoc2)n[nH]1 30074,C(=O)(CCCS(N)(=O)=O)NCCCN(C(C(C)NC(COC)=O)=O)CCO 30075,C1(NC(C=CC(C)(C)SC)=O)CN(C(c2cn(C)c(=O)cn2)=O)CC2(CC2)C1 30076,c1(C(=O)NCC2(O)CCN(C(CCCCC)=O)C2)cc(OC)c(O)c(N)c1 30077,C(C)(CCC(=O)NC1CN(C(=O)CC)CC1SC)OCC 30078,c1(CC(=O)NCC2CC(NC(c3cccc(C(F)(F)F)n3)=O)C2)ccc(O)cc1 30079,C1(N(C(C(N2C(=O)CCC2=O)C)=O)C)CCCN(C(=O)Cn2cnnc2O)CC1 30080,Cc1ccncc1C=CC(=O)NC1(CO)CCCN(C(=O)CCc2cc[nH]n2)C1 30081,Cc1cnc(C(N2CC(CCNC(=O)C(c3ccc(F)c(F)c3)O)C2)=O)cc1Cl 30082,CC1CC(=O)NC(C(=O)NCC2(F)CCN(C(c3cnc4sccn34)=O)C2)C1 30083,CCCC(O)(CCC)CC(=O)NC1CC2CC(C1)N(C(c1c[nH]c(Br)c1)=O)C2 30084,C1(O)(CNC(CCC)=O)CCN(C(=O)C(O)c2ccsc2)C1 30085,N1(C(c2ncc(C)nc2)=O)CCC2(C=C(C(=O)N3CC(CO)C(O)C3)C2)C1 30086,N1(C(c2cc(C)ncc2)=O)CCC2CCN(C(=O)COCC(F)F)CC12 30087,n1(NC(=O)CC23CC4CC(CC(C4)C2)C3)ccc(=NC(=O)C#CC2CC2)nc1O 30088,Cc1cnn(CCC(=O)NCCOC2CN(C(C3CCCN3C)=O)C2)c1 30089,C(=O)(C(CC(C)C)NC(C)=O)N(CC(CC)NC(=O)CSc1cccs1)C 30090,c1(CC)onc(C)c1NC(C1CC(CNC(=O)C=Cc2ccn(C)c2)C1)=O 30091,c1(C(=O)NCC2C(NC(CN(C)CCO)=O)COC2)cc(CC2CC2)nn1C 30092,C(=O)(C(C)(C)C#N)NCC(C)(C)CC1CN(C(c2ccsn2)=O)C1 30093,C(C(O)C(=O)N(CC(C)C(=O)NCC1CSCCO1)C)SC 30094,C(C(=O)NC(CO)C(CC)NC(C1(CC)CNC(=O)C1)=O)(C(C)C)SCC 30095,S(=O)(=O)(c1cccc(C(=O)N=c2cc[nH]cc2Cl)c1)NC(COC)COC 30096,N1(c2ccnc(C)n2)CC23CCCCC2(CN(C(C2(CC4CC4)CC2)=O)C3)C1 30097,NS(=O)(=O)C1(C(=O)NCC2(F)CCC(CNC(=O)CC3CC=CC3)CC2)CCC1 30098,c1(C(=O)NC2CCC(CCNC(Cc3c(C)non3)=O)C2)cc2n(c1)CCOC2 30099,C=C1CCN(C(=O)CC=CCC)C(C(N2CCC(CF)CC2)=O)C1 30100,c1(CCNC(C(CC)N(C)C(c2cc(C3CC3)no2)=O)=O)noc(=O)n1C 30101,C1(CC(=O)NCCC2(NC(C(C(C)C)C)=O)CCCC2)COC(C)(C)CO1 30102,c1(C(=O)NCCC2(O)CCN(C(=O)C3=CCSC3)CC2)cc2c(nn1)CCC2 30103,C1(C(=O)NC2CCCC2CNC(=O)CC(=O)NCC2CC2)(CC)CCOC1.C1CC1 30104,C(=O)(C(C)S(=O)(=O)CCC)NCC1(COC)CN(C(C(C)=CC)=O)C1 30105,CCC(C)C(=O)C(=O)N(C)CC1(O)CCCN(C(c2sccc2CO)=O)C1 30106,c1(C(=O)NCC2CCCC(CNC(C3(N(C)C)CC3)=O)C2)cc(F)cc(F)c1 30107,N1(C(C(C)Cn2ccnc2)=O)CCCC(CC(=O)NCC2CC(=C3CC3)C2)CC1 30108,C1(C(N2C(CCCNC(COCCC#C)=O)CCCC2)=O)CCOCC1(C)C 30109,N1(C(C=Cc2c(C)nccc2)=O)CC(C2CCCCN(C(=O)CSC(F)F)C2)C1 30110,C(C1=NOC2OCCC12)OC(C1CCC=CC1O)=O 30111,C1(C(=O)NC(CC#C)CCOC)CCN(C(=O)c2csc(C)c2)O1 30112,N1(C(C(C)OCC)C)CCC(O)(NCCCN(C)C)CC1 30113,N1(C(c2c(OC)ccc(C)c2)=O)CCCCC(N2CCCC(C(F)F)C2)C1=O 30114,C1(OCC)CCCC1NC(=O)C(c1ccnn1C)C 30115,CCCC(CC(=O)N1CCC1CC1CC1)c1ccccc1.n12nnnc1CC2=O 30116,C(=O)(CCC(=O)N1CCOC(CNC(C2(n3cccn3)CC2)=O)C1)NCC 30117,c1(C(=O)NCCCN2CCN(C(C3(O)CC3)=O)CC2)cc([N+](=O)[O-])ccc1Br 30118,N1(C(=O)C2=COCCO2)CCCN(C(c2cc[nH]c3nccc2-3)=O)C(CO)C1 30119,Cc1ccc2nc(C(C)C)cc(C(N3CCCC3CN(C(=O)C(F)F)C)=O)c2c1 30120,N1(C(c2cccnc2S)=O)CCC2(CCCN2C(c2ccc[n+]([O-])c2)=O)C1 30121,c1(C(=O)NCCCC(C)NC(C2(OCC)CCC2)=O)c(C)nn(CC(F)F)c1C 30122,C1(C(=O)Nc2cnc[nH]2)CN(Cc2ccc(Br)cc2)CCC1O 30123,N1(C(C2C(NC(CCCN=[N+]=[N-])=O)C=CCC2)=O)CCC12CCCCC2 30124,c1(C(N2C(CO)CC(NC(C=C(C)C)=O)C2)=O)cc2c(Br)coc2cn1 30125,N1(C(c2c(CC)nn[nH]2)=O)CCC2(CCCN2C(=O)CCCC2CCCO2)C1 30126,c1(C(N2CCC(O)(CNC(C(n3c(C)ncc3)C)=O)C2)=O)nnn2c1CCCC2 30127,Cc1cccc(N2CCC(N(C)Cc3ccn(-c4ccccc4)n3)C2=O)c1 30128,C(=O)(CCCCCN(C)C)N(CC(CC)NC(=O)CSc1n[nH]c(C)n1)C 30129,C1(NC(CN(C)C(N)=O)=O)CCC(NC(c2ccc(=O)oc2)=O)CC1 30130,Cc1cc(C(N2CC3CCC2C(NC(C2CCC2)=O)C3)=O)c(N)c(F)c1 30131,C1(NC(Cc2c(C)ccs2)=O)CN(C(=O)CN(C(=O)C2CC2)CCC)CC1C1CC1 30132,CC(C)CC(C)C(=O)N(CC(O)CN(C(=O)COc1ccc(CO)cc1)C)C 30133,c1(C(=O)NC(C2CCCC2)CNC(C23CCN(CC2)C3)=O)ccc([N+](=O)[O-])[nH]1 30134,c1(C(N2CC(OCCNC(Cn3ncc(C#C)c3)=O)C2)=O)cc(Cl)c(F)cc1F 30135,C(CC1=CCN(C(c2cnc(C(C)(C)C)[nH]2)=O)CC1)NC(c1cc(C)c(Cl)s1)=O 30136,N1(CC(N2CC(NC(C3CCS(=O)CC3)=O)CC(C)C2)=O)CCc2ccccc21 30137,N1(C(c2c(C)coc2)=O)CC(NC(c2[nH]nnc2-c2ccnn2C)=O)CC1C 30138,C#CCCCC(=O)NC(Cc1ccoc1)C(N1CC2C=CC2C1)=O 30139,C1(NC(CCC=C=C)=O)CC=C(C(=O)N2CCC(OC(C)=O)C2)C1 30140,Cc1cccc(F)c1C(=O)NC1CCC(NC(C2CC23CC3)=O)CC1 30141,N1(C(C(C)(C)c2cccs2)=O)CCCC(O)(CNC(c2ccc(C(F)F)o2)=O)C1 30142,CCC(CC(=O)NOCC(=O)NCc1nccs1)C(C)(C)C 30143,N1(C(CCN(CC)CC)=O)CCC(C(=O)NC(CCO)C2CC2)(CC)CC1 30144,n1(CC(N2C(C)CC(CNC(=O)CC3CS(=O)(=O)C3)C2)=O)nnc2c1CCCC2 30145,c1(C(=O)Nc2ccc(C#N)nc2)cnc2c(-c3ccc(CO)nc3)cccc2c1 30146,CCCCC(CC)C(=O)NCC(C)(C)NC(c1ccn(CC)c(=O)c1)=O 30147,c1(C(N2CC(NC(c3ccccn3)=O)C3C2C3)=O)ccc2cnccc2n1 30148,C1(C)(NC(C2N(CCC)CCC2)=O)CCN(C(c2cc(C)c(C)s2)=O)CC1 30149,N1(CC)CCCCC1C(=O)N(C)CC1(NC(c2cnn(CC(F)(F)F)c2)=O)CC1 30150,N1(C(=O)OC(C)(C)C)C2CCC1CC(CNC1CCC(O)CC1)C2 30151,C(=O)(C(CN(C)C)C(C)C)NCC(N(C(c1cc(C)sc1)=O)C)C1CC1 30152,C1(C(=O)NC(C)C2CC2)C2CCC(C2)C1NC(=O)C=Cc1ccccc1 30153,c1(-c2cccc(OCC)c2)ccc2oc(CO)cc2c1 30154,c1(C(N2C(C)CCC(NC(CNC(=O)OCC=C)=O)C2)=O)cnc(OC)nc1C 30155,C#Cc1ccc(C(=O)NCC(C)(CC)C(=O)N2CCC(O)C2)cc1C 30156,c1(C(=O)NCC(CC)NC(=O)C(CC)Nc2nc(C)cs2)cccc(=O)o1 30157,Cc1c(C(N2CCN(C(=O)CC3C=CCCC3)CC2CO)=O)nn(C)c1Br 30158,CC(F)(F)C(C)(C)CNC(C1(NC(=O)COCC2CCCO2)CSC1)=O 30159,N1(CC)CCCC1CC(=O)N(CC(O)CNC(c1cscn1)=O)C 30160,Cc1cc(C(=O)NC2CC23CCN(C(=O)OC(C)(C)C)CC3)nc2nccn12 30161,CN1CCOC(C(=O)NCC2(F)CCC(CNC(C3SCCS3)=O)C2)C1=O 30162,c1(OC)ccc2c(C(N3CCC(N(c4c([N+](=O)[O-])cnn4C)C)C3)=O)cnn2c1 30163,C1(C(=O)OC)CCCC(C(N2CCCCC2CNC(c2coc(CO)n2)=O)=O)C1 30164,N1(CC(N2CC(O)(CCNC(CCCOCC)=O)C2)=O)OC(C)(C)CC1=O 30165,C#CCCCCCC(=O)N1CCCOC(CNC(=O)C(N2CCC(O)CC2)C)C1 30166,C1(NC(c2cc(O)nc(O)n2)=O)COC2(CCN(C(c3cccnc3Cl)=O)C2)C1 30167,CC1CN(C(=O)CC(C)(C)CCC2OCCO2)CCC(c2cccs2)O1 30168,c1(CN2C3(COC3)C2=O)ncc(C#N)cc1Br.N1(C(C)(C)C)CCCS1(=O)=O 30169,c1(C(=O)NCCCNC(CC2(C)CCCO2)=O)ccc(-c2ccccc2)cc1F 30170,Cc1ccnc(CNc2c[nH]nc2C(=O)Nc2nccnc2C(F)(F)F)c1 30171,C1(CN(C(CCC2(C)N=N2)=O)C2CC2)CCCN1C(=O)C(C1CCOCC1)O 30172,c1(CN2CCC(C)(NC(c3ncn(CC)c3)=O)C2)cc(OC)c2c(c1)CCO2 30173,N1(C(c2n(CC)cnn2)=O)CC=CCC12CCOCC2 30174,N1(C(c2cc(N3CCOCC3)ccn2)=O)Cc2cccc3c2C(CCC3)C1 30175,n1(CC)ncc(C(=O)NCC2CCN2C(c2ccc(C)s2)=O)c1C 30176,CCC(CNC(C1(n2ccnn2)CC1)=O)NC(=O)Cc1cnc[nH]1 30177,c1(C(N(CCNC(C2CCCC2)=O)CCOCCO)=O)cc(C(=O)C2CC2)on1 30178,C=CCC(C)(CO)CN=c1[nH]c(=NCc2nc(CC)ns2)[nH]c2c1COC2 30179,c1(NC(C2CN(C(C3CC3(F)F)=O)CCO2)=O)cc(Br)ccc1I 30180,Cc1ccc(OCC(=O)NC(C)(CNC(c2cn(C)cn2)=O)C2CCC2)cc1C 30181,Cc1c(C(N2CC(C)(NC(C34CC(C(C)C)(CO3)C4)=O)C2)=O)[nH]c2ccccc12 30182,c1(C(C(=O)NC(CSC)CC(C)C)C)c(Cl)cccc1Cl 30183,N1(C(CN2CC(C)(OC)C2)=O)CCN(C(=O)C2=CCCN(C)C2)CC2CCCCC12 30184,S(=O)(=O)(CCC(=O)NCC1CC(C(F)(F)F)CN1C(c1cccc(=O)n1C)=O)NC 30185,c1(C(=O)NC(CC)CNC(=O)CN2CCN(C)CC2)cnc2ccccn12 30186,N1(C(c2c(C)oc(C(C)C)n2)=O)C2CCC1CC(NC(=O)C(C)CC1CC1)C2 30187,C1(C(N(CC(C)NC(C23CCCC(C)(C2)OC3)=O)C)=O)CNC(=O)CC12CCC2 30188,C=CC1OCCC1N=c1[nH]c(N2CCN(CC(F)(F)F)CC2)nc2ccccc12 30189,N1(C(=O)NC2CC3N(C)C(CCC3)C2)CCn2cccc2C1c1ccccc1 30190,C12(C(N(C(CNC(CC(C=C)C)=O)C)CC)=O)C3CC(CC13)C2(F)F 30191,C1(CNC(C(CC)SC)=O)CCN(C(=O)Cc2scnc2C)C12CCC2 30192,N1(C(C(C)NS(CC)(=O)=O)=O)CCCC(C)(CNC(=O)Cc2ccns2)C1 30193,CCC(C)CCC(O)CC(=O)N1CCC(NC(C2CC(=O)C2(C)C)=O)CC1C 30194,CC1CCN(C(C2COC(=O)N2C)=O)CC1NC(=O)C(C)(C)F 30195,O(NC(=O)Cc1nocc1C)C(CCC=C)OC.C1CS(=O)(=O)N1 30196,Cc1cccnc1C(N1CCC(C)C1C(=O)NC1CC(n2ccnn2)C1)=O 30197,C1(CC(=O)Nc2cccc(C3CC3)c2)CCCC12CN(C(c1ccsc1)=O)C2 30198,c1(CN2CC(CC(=O)NC3CCS(=O)(=O)C3)OCC2)cc(F)c(Cl)cc1O 30199,c1(C(=O)NCCCC2(CNC(CC=C=C)=O)CCCC2)c(C)cc(C)nc1O 30200,c1(CC)nn(C)c(CC(C)C)c1C(=O)OCC(=O)Nc1cc(Cl)cnc1O 30201,c1(C(=O)NC(C(CC)C)C(N2CCC3(CC(CO)C3)C2)=O)ccn2nccc2c1 30202,c1(C(N(CC(CN(C(C(C)OCCCC)=O)C)O)C)=O)cc(O)cc(C#N)c1 30203,C1(CNC(C2(C)CCC(=O)C2)=O)CC(C(=O)NC2(CC(N)=O)CC2)=NO1 30204,N1(C(=O)CSC(F)(F)F)CC2CN(C(C3CC3(Cl)Cl)=O)CC2C(F)(F)C1 30205,CCC(CC)C(C)C(=O)NCCC1(C(=O)NOCCCN(C)C)CC1 30206,C1(C(N2C(CNC(c3cn(CC)nn3)=O)CCCC2)=O)CCCCC(F)(F)C1 30207,CCC(C(=O)NCC1CC2(CC(CNC(=O)COCc3nc[nH]n3)C2)C1)C(C)C 30208,N1(C(CC(C)(C)C#N)=O)CCC(O)(C2CCN(C(C3CC(=O)N(O)C3)=O)CC2)C1 30209,C1(C2CC2)(C(N2CC(CC(C)NC(=O)Cc3nccn3C)C2)=O)CCC1 30210,c1(C(N)=O)ncn(CC(=O)NCC2CCC(NC(C3CC4CC4C3)=O)C2)n1 30211,N1(CCCC(=O)NCCN(C(=O)CC(F)F)CCC)C(=O)NC(C)(C)C1=O 30212,c1(C(N2CCCN(C(C34CCC(OC)C3C4)=O)CC2)=O)ccc2c(c1)CCCS2 30213,C1(C)(NC(CN(CCCCCC)C)=O)CCN(C(C2CCC23CCC3)=O)C1 30214,c1(OC)ccc2sc(CNC(C)C(=O)Nc3ccc(C)c(C)c3)c(C)c2c1 30215,Cc1cn(C)nc1C(=O)N(CC(C)CNC(C1CCCN1S(C)(=O)=O)=O)C 30216,c1(NCC(CC)(C)COC)nc2ccccc2nc1N1CCC(OCCO)C1 30217,CC1C(NC(=O)COC2CCOC2)CCN1C(=O)C=CC1CCC1 30218,N1(C(C(n2ncc(C)c2)C)=O)CCC2(CC1)CC(N1CCCC(C)(F)CC1)C2 30219,C=C(C)C(C)(C)C(=O)NC1CCC(N(C)C(c2ccccc2C(C)O)=O)CC1 30220,S(=O)(=O)(c1ccccc1F)NC(C1C(NC(c2cccc(F)n2)=O)C2CCC1C2)=O 30221,N(C(=NCCc1ccco1)NCC1CCC(C)(C)C1)Cc1ccc(OC)cc1 30222,CC1CN(C(=O)COCCF)CCCN1C(=O)CC12CCC(CC1)OC2 30223,CC1OCCC1C(=O)NCC1CCOC1C(=O)NCCc1cnnn1C 30224,C1(CNC(=O)NC)CCN(C(=O)Cn2ccnc2C(C)C)CC1 30225,C(C(C)(C)C(=O)N1CCCCC1Cn1cc(C2(O)CCC2)nn1)OC 30226,Cc1sc(=O)n(CC(N2CCCC2CCNC(c2cc(Cl)c(Cl)n2C)=O)=O)c1C 30227,C(C)(CO)(C(=O)N1CCC(CCC)C1)NC(CC=C)=O 30228,C=C(Cl)CC(C(=O)N=c1cc(C)n(CCO)[nH]1)NC(=O)C1=CC2(CCOC2)C1 30229,C(=O)(C1=NOC2(CCOC2)C1)NCCOCCNC(C1(c2c(C)c[nH]n2)CC1)=O 30230,CC1C(=O)N(CC(=O)NCC2CCC2NC(c2nc(=N)cc[nH]2)=O)C(=O)C1C 30231,C1(C(=O)NCCC2CCN(C(C(C)n3cncn3)=O)CC2)CC(F)(F)C12CCC2 30232,C(C(C)(Cn1cccn1)N=c1[nH]nc(C)o1)N(C1(O)CCSCC1)CC 30233,N1(C(C(CC(C)C)OC)=O)CCC2(CCC(NC(c3ccc(C)c(C)c3)=O)C2)C1 30234,C1(C(=O)NC23CC(NC(C4(CC#C)CC4)=O)(C2)C3)CCC(N(C)C(C)=O)CC1 30235,C1(CNC(C=CCC)=O)CC(CNC(=O)CCOC2CCC2)CO1 30236,C(=O)(C1CCC(=O)c2cccn21)NCCCCC(C)NC(c1cc(OC)ns1)=O 30237,C1(NC(c2cc(CC)ncn2)=O)CN(C(=O)C(=O)C(C)CC)CC(F)(F)C1 30238,C(=O)(C(CCF)NC(C1CCCSC1C)=O)NC1C(SC)COC1 30239,C(CCC(C)C)(C(=O)N1CCC(C)=C(C)C1)NC(C=C(CCC)CCC)=O 30240,C1(CC(=O)NC2(CNC(=O)CC3CCCCC3)CCOC2)CCCS1(=O)=O 30241,C(=O)(C(F)C(C)CNC(=O)C=C1CCCCC1)N(C(C)C(=O)OC)CC 30242,c1(C(=O)NC2CCN(C(C(CNC(C)=O)(C)C)=O)C2)n[nH]c2ccc(F)cc12 30243,N1(C(c2ncn(C)n2)=O)CCOC2CN(C(=O)CC3CCC(C)(C)O3)CC12 30244,c1(C(=O)NCC2(O)CC(C(N(C)Cc3ccncn3)=O)C2)ncccc1N 30245,N1(CCC)CC(C(=O)NCCCCCNC(=O)COCC(C)(C)C)CC1=O 30246,S(=O)(=O)(c1ccc(C#N)c(N2CCC3CC23)c1)N1CCCC(=C)C1 30247,c1(C(C)C)ncc(Cl)c(C(=O)NCCC(C)N(C(=O)Cc2cnns2)C)n1 30248,C1(NC(c2ccc(OC)nc2C)=O)COC2CN(C(=O)CNC(=O)C3CC3)CC12 30249,c1(C(=O)NC(CCN(C(c2c(CC)nn[nH]2)=O)C)C)cccc(Cl)c1F 30250,c1(C(=O)NC2(C)CC(NC(Cn3c(C)nnn3)=O)C2)cccc2c1OCC2(C)C 30251,CC(C)CC(C(=O)NC1CC2CC(NC(=O)CSc3nnnn3C)C1C2)C(N)=O 30252,C(=O)(C(C(=O)OCC1CC1)NC(=O)CCSC(C)CCOC)OCC 30253,C1(CCCC)CCC(NC(N2CCOC(c3cc(C)no3)C2)=O)CC1 30254,N1(C(C(CC(F)F)NC(CCCNC(=O)OC)=O)=O)CC2(CNC(=O)N2C)C1 30255,c1(OC)ccc2nc(N3CCC(NC(=O)Cn4cc(C(C)O)nn4)C3)sc2c1 30256,N1(C(=O)OC(C)(C)C)CC2(CCCN(N3CCCC(CC(F)F)C3)C2)C1 30257,C1(COC)CN(C(=O)Cc2cncc(Br)c2)CCN1C(=O)CC(C)OC 30258,C(C(CC(C)C)C(=O)NC(C)(C)CNC(C1(C)CC1)=O)OC 30259,c1(N2CCC(CC)C2)ncc(C)cc1S(=O)(=O)N1CCC1(C)NC(=O)NC 30260,C(=O)(C1=CC(O)CCC1)N1C(CN(C(=O)CCCC2CCOCC2)C)COCC1 30261,Cc1ccc(C(=O)NCCC(=O)NC(C)CC(C)NC(=O)CCC(C)C)cc1C 30262,N1(C(c2c(C)nsc2C)=O)CC2(CO)CC1(C(N1CCC(CN(C)C)C1)=O)C2 30263,N1(C(c2c(C#N)nc[nH]2)=O)CC2CCC2(CCNC(=O)COCC(F)F)C1 30264,C1(NC(C2CC(C#C)(O)C2)=O)CS(=O)(=O)CC1NC(=O)C=C1CCN(C)CC1 30265,C1(NC(C2(CC=C)CCOCC2)=O)CC2(C1)CN(C(c1csc(CCC)n1)=O)C2 30266,CC(C)CC(O)CC(=O)N1CCC=CC1C(=O)NCC1(C)CCN(C)C1 30267,C1(CNC(=O)Cc2ccc(Cl)cn2)CC2COCC2N1C(=O)CCCN1CCC1 30268,N1(C(C)C)C(=O)CCC1C(=O)NC(C)(CNC(c1c[nH]c(=N)o1)=O)C1CC1 30269,CC1CC2CN(C(=O)CN=S(C)(C)=O)CC2N1C(=O)C(=O)C(C)(C)C 30270,CC1=C(C(=O)NCC2C=CC(NC(=O)CC3CCC3)C2)C(C)n2nnnc2N1C 30271,C(=O)(CC(CC)C(C)(C)C)N(CCC(=O)NCc1nc(C)c(C)[nH]1)CC=C 30272,C(=O)(C1=CCC(C)CC1)NCC(CC=C)NC(c1ncsc1S(N)(=O)=O)=O 30273,c1(C(N2CCC(C(C(=O)Nc3c(CC)cccc3)C)C2)=O)ccc2cncn2c1 30274,C1(CNC(Cn2c(CCC)ncc2)=O)CC(F)CN1C(c1cnncc1OC)=O 30275,C(=O)(CC(F)(F)C(F)F)N1CC(NC(=O)C=Cc2ccsc2)C(F)C1 30276,c1(C(=O)NC2C(OC)COC2)ccnc(CNC(=O)C(C)(C)NC(C)=O)c1 30277,C#CCCCCCC(=O)N1CCC(NC(c2c(C)cccc2Cl)=O)CC1C1CC1 30278,c1(CC(=O)NCCC2CN(C(=O)N(C3CCC3)C3CC3)CCO2)cccc(I)c1 30279,N1(C(c2scc(OC)c2OC)=O)CC(NC(=O)CC(C)(C)OC)CC1(C)C 30280,c1(CC)nn(C)c(CC(=O)NCC2COCCN2C(c2ccnc(O)c2)=O)c1Cl 30281,N1(C(c2cc(C)c(C)s2)=O)CCCC(O)(CN(C)C(C2(C)CC(C)(C)C2)=O)C1 30282,c1(CC(=O)NCC(CC=C)NC(c2ncc(C)cc2C)=O)csc2ccccc12 30283,Cc1cccc2c1c(CN1CCC(C#N)(NC(=O)C(C)n3cccn3)C1)cn2C 30284,C1(C(=O)NCC2CN(C(=O)CC3CCCCO3)C2)(COC)CCCCO1 30285,C1(NC(=O)CC(Cl)Cl)CN(C(=O)C(F)n2ccnc2)CC12CC2 30286,N1(C(C2C(C)=NOC2=O)=O)CCCCC(CNC(=O)C(C)Cc2ccccc2)C1 30287,C1(CCCCNC(c2c(C)c[nH]n2)=O)CCN(C(c2c[nH]ccc2=O)=O)CC1 30288,C=C=CCCC(=O)NC1CC(C(C)NC(=O)Cn2ncccc2=O)C1 30289,CN1CCC2CN(C(C3CC(NC(C4(O)CCC4)=O)C3)=O)CC2C1 30290,N1(C(C2CCC(OC)CC2)=O)C2CC1CN(C(C1(C)CNC(=O)C1)=O)C2 30291,N1(C(C2C=CCN(C(C3CCCC(OC)C3)=O)C2)=O)CCC(C2=NOCC2)C1 30292,C1(NC(CCCOC)=O)CC=C(C(=O)NC2(C(C)O)CC2)C1 30293,C1(C(N(C(C)C(N2CCC(CN=[N+]=[N-])C2)=O)CC)=O)CCOC1(C)C 30294,n1(CCOC)cc(C(=O)NC2CCCC2CNC(=O)CC2CC2(Cl)Cl)nn1 30295,N1(C(=O)NC2CCC(N3CCNCC3)CC2)CCCCC(Cc2ccccc2)C1 30296,N1(C(CCC)C)CC(C(=O)NCCC(C)NC(C2(C(F)F)CCCC2)=O)CC1=O 30297,CC1C(C=CC(N2CCCC2CCCNC(=O)C(=C2CCCCC2)F)=O)C1(Cl)Cl 30298,Cc1cccc2cc(C(=O)NC3CCCC3NC(=O)C#CC3CC3)[nH]c12 30299,N1(C(c2ccc(OC)c(OC)n2)=O)C2CCC1CC(N(C)C(C1OCCO1)=O)C2 30300,c1(C(CC)N)cccc(O)c1.c1cn(-c2ncccn2)nn1 30301,c1(C(=O)NC(CC(C)NC(c2c(C)nncc2)=O)C)ncc(C#N)cc1Cl 30302,CC12COC(C(=O)NCCC3CSCCN3C(=O)CC3CCCCC3O)(C1)C2 30303,c1(NC(N2C(C(C)C)CC(O)C2)=O)cccc(C(F)F)c1Cl 30304,Cc1cc(C(=O)NC2CCC(C(N3CCC(O)C(F)C3)=O)C2)cc(O)n1 30305,Cc1cnc(F)cc1C(N1CC(CNC(=O)C(C)NC(c2ccccc2)=O)C1)=O 30306,N1(C(C(C)c2ccco2)=O)CCC(C)(C(N2CCC(C(C)(C)O)C2)=O)C1 30307,C1(C(=O)NC(CC#C)C(=O)NCCc2nc(CC)no2)CC2(CCO1)CC2 30308,c1(N(C)C)ccccc1NC(C1C=CC(NCc2csc(Br)c2)C1)=O 30309,C(=O)(CCC(=O)NN(C)C)NC(C1C(C(=O)NCC(CCC)C)C1)C 30310,C1(CCOC)(NC(=O)C(C)N(C)C)CCN(C(C23CSC(C2)C3)=O)CC1 30311,n1(C(C)C)nnnc1C(C1C=CCC1)NCCCN(S(C)(=O)=O)C 30312,C1(NC(c2n(C)nc(C3CC3)c2)=O)CCN(C(=O)CC2CC=CC2)CC1(C)C 30313,N1(C(C(C)C2CCCOC2)C(=O)NCC(F)F)CCc2ccc(F)c(F)c2C1 30314,N1(CCNc2ccc(C(=O)OC)o2)CC2CCC1CN2Cc1ccccc1 30315,Cc1ccc(F)cc1C(=O)NC1CCCN(C(=O)Cn2ccc(C(F)(F)F)n2)C1 30316,N1(C(CO)=O)CCCc2ccc(S(C)(=O)=O)cc21.CC(C)(C)O.C1(=O)C(=O)NCCO1 30317,C(=O)(C(C)(C)C(C)O)NCc1cccc(CN(C(CC(C)O)=O)C)c1 30318,N1(C(CN(c2nc3ccccc3s2)CC)=O)CCCC2(CC(NC(=O)CO)C2)C1 30319,CCC(COC)C(=O)N(C(C)CN(C)C(c1cc(Cl)cnn1)=O)C 30320,CCCCCC(O)CC(=O)NCCC1CCCCN1C(=O)C(CC)SC 30321,C1(NC(c2ncnc(=N)[nH]2)=O)CC2CC(NC(c3ccno3)=O)CC12 30322,C1(CO)CCN(c2cc(N3CCOC(c4ccsc4)C3)ncn2)CC1 30323,C#CC1(C)CCCN(C(=O)C(CC(=C)Cl)NC(C23CCC(C2)C3)=O)C1 30324,C1(CNC(Cc2[nH]cc(C)c2)=O)COCCN(C(c2csc(CO)n2)=O)C1 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30343,C1(C(=O)NCC2CC3(CC3)CN2C(c2ccc[nH]2)=O)CCC(C2CC2)CC1 30344,C1(CC)(NC(=O)CCn2cc(CCCCN)nn2)CCCOC1 30345,N1(C(Cn2cc(C(=O)OCC)nn2)=O)CC2(C1)CN(C(C1CC3(C1)CC(O)C3)=O)C2 30346,C1(C(=O)NC(CC=CC)C(=O)N2CCC(CC3CC3)C2)CCC(O)CN1C 30347,N1(C(c2c(C(C)(C)C)ocn2)=O)CCC(F)C(NC(C2(F)CC2(C)C)=O)C1 30348,C1(C(N2C(C)COC(CO)C2)=O)CC2CN(C(=O)C=CC(C)(C)C)CC2C1 30349,C1(NC(C(C)N(CCc2cccs2)C)=O)CN(C(=O)C(N)=O)CCO1 30350,C1(N(C(=O)Cc2nc[nH]n2)CC)CCN(C(=O)Cc2ccsc2C)C1 30351,N1(CCC#C)CCN(C(=O)COCCNC(=O)CC2CCCN2C)CC1 30352,N1(C(C(CC)(C)CC)=O)CCC2CC(CNC(c3ccsn3)=O)CCC2C1 30353,Cc1nc(NC2CC3CN(C(c4ccn(O)c(=O)c4)=O)CC23)c(F)c(C)n1 30354,Cc1ncc([N+](=O)[O-])n1CC(N1CCN(C2CCCC2O)CC1)C 30355,c1(NC)ccc(F)cc1C(N1CCCCC1CNC(c1c(C)cncc1F)=O)=O 30356,C1(NC(C(CC(=C)C)C)=O)CN(C(=O)CN(C)C(N)=O)CC1S(C)(=O)=O 30357,N1(CC(c2c(OC)ccc(OC)c2)=O)C2CCCC1CC(O)C2 30358,c1(-c2ccc(CC)s2)cn(C)nc1C.N12CCCC1C2C(=O)NC(CC)C 30359,CC1C(C(=O)N(C(C)(C)CC(=O)NCC2CCCC23CC3)C)=NOC1C 30360,N1(C(c2ccc(CC)o2)=O)CCN(C(c2cc(Cl)cn2C)=O)CC1CC(F)(F)F 30361,CC1CN=C2NC(C(=O)N3C4CCC3C(CNC(c3cccnn3)=O)C4)=NN2C1 30362,C(C1=CCN(C(C2CCC(CCO)CC2)=O)CC1)NC(c1cn(C)nn1)=O 30363,Cc1cc(C(=O)NCC2C(CNC(c3cc(C)oc3C)=O)C2(F)F)c(C)[nH]1 30364,CC(C)(C(=O)NC1CC(F)(CNC(c2cc(C3(C)CC3)on2)=O)C1)C(N)=O 30365,N1(C(C2(SC)CC2)=O)CCC(C2(NC(=O)C(N3CCCCC3=O)C)CC2)CC1 30366,c1(NC)cnc(C(=O)NCC2(CNC(c3nsc(N(C)C)n3)=O)CC2)cn1 30367,C(=O)(C1=CCCSC1)N1C(C(=O)N(C2CCC3(CC3)C2)CCO)CCC1C1CC1 30368,CC1C(C(N2CCN(C(=O)CN(C)C(=O)Oc3ccccn3)CC2)=O)CCN1C 30369,c1(CC)nc(CC(=O)NCC2CCN(C(=O)CSC3CCCCO3)C2)cs1 30370,C1(C(=O)NCCC2CCC(NC(COCC)=O)C2)CC12CCC1(CC1)CC2 30371,c1(-c2cnc(N(c3n(C)ncc3)C(C3(F)CCOC3)=O)s2)cccc(Cl)c1 30372,c1(C(=O)NC(CNC(CCN(C)CC)=O)(C)C2CC2)ccc(C2(C#N)CC2)cc1 30373,c1(C(N2CC(CNC(COC)=O)N(C)CC2)=O)cc2ccccc2n1CC1CC1 30374,c1(SC2ON=C(C)C2)cccc(CC(=O)N(C)Cc2ccccc2)c1 30375,C1(NC(C(CCC)C)=O)CCC12CN(C(=O)CCCCN1CCCCC1)C2 30376,c1(C(=O)NC(CCC(=O)OC(C)(C)C)C(=O)O)cc2ccc(C(=O)O)cc2o1 30377,C1(=O)C(C)Cc2cn(nn2)CCN1.c1(C2C(C(C)=O)C2)cn(CC(C)(C)O)nn1 30378,CCC(C)C(C(=O)NC1CCCCC1CC(=O)NOCc1ccc(F)nc1)N(C)C 30379,c1(C(N(C2C3CN(C(=O)CC4(C)CC4)CC23)C)=O)ccc(Cl)cc1 30380,C=CCC(CC(=O)NCc1nn(C)c(=O)o1)NC(=O)CSC(F)(F)F 30381,CC(C)(O)C(F)(F)CNC(=O)C(CNC(=O)Cn1cccc1)CC1CCCC1 30382,c1(C(N2CCN(CCN=[N+]=[N-])CC2)=O)cc2c(F)ccc(F)c2s1 30383,c1(C(=O)OC)ccc(C(=O)NC(C)CNC(=O)C(=O)NCC2CC2)nc1C 30384,c1(OC)ccc(SCC(=O)NCC(C2CC2)NC(=O)CCCc2ncco2)cc1 30385,c1(C(=O)NCC2N(C(C(C)=CC3CC3)=O)CCC2C)cnc2c(c1)CCCO2 30386,N1(C(C2CC(C)OCC2)=O)CCCC(C2CCN(C(=O)CSC(F)(F)F)CC2)C1 30387,CN1CCCCC1CC(=O)NC1CC1C(=O)Nc1ccccn1 30388,c1(C(N2C(C(=O)NC3CCC(O)CC3)CCCC2)=O)cn2ncccc2n1 30389,C1(NC(C2CCCOC2)=O)(CO)CCCN(C(c2cnn[nH]2)=O)C1 30390,C#CCC(CC(=O)N1CCC(OCC=C)C1)NC(C1(C#N)CCCC1)=O 30391,C1(NC(CC2(OC)CC2)=O)CCN(C(=O)Cc2csc(Cl)n2)C1C(C)C 30392,C(=O)(C1=CS(=O)CCC1)N1CCC(NC(C2C(F)(F)C23CCC3)=O)(CF)C1 30393,C1(NC(CCOC(C)C)=O)CC(NC(c2cc(O)cc(F)c2)=O)C12CCOCC2 30394,C1(COC)(NC(C2CCN2S(C)(=O)=O)=O)CN(C(=O)CCCN2CCCC2)C1 30395,C1(CNC(C(N2CCN(C)CC2)C)=O)C(C)CCCN1C(C1CC12CC2)=O 30396,c1(C(N2CCC(C)(CNC(COC)=O)CC2)=O)ccc2c(c1)C(C)(C)CO2 30397,C1(C(N2CCC(C)(NC(C(CC)C)=O)C2)=O)C2Cc3ccccc3C12 30398,C1(NC(CCc2nc(C)c(C)o2)=O)CCC2CN(C(=O)OC(C)(C)C)CC2C1 30399,NC(CNC(=O)CN1C(=O)C2CSCN2C1=O)CC1CCc2ccccc21 30400,CC(C)C(C)(O)C(=O)N1CCC(CCC(=O)NC(CN(C)C)CCO)C1 30401,C1(C(N2CCN(C(c3cc(C4CC4)nc(O)c3)=O)CC2)=O)CCc2nncn2C1 30402,c12cc(c3c(c1)OCO3)S2.n1(CC)ccnc1CNC(=NC)N(C)C 30403,O=C(NNc1cccnn1)c1ccc(OC2CCNCC2)cc1 30404,C12CCN(CC1)C2=O.c1(NCCNC(=O)Nc2ccccc2)ccc(I)o1 30405,C1(C)(C(N2CCC(OCCNC(c3c(CC)noc3)=O)C2)=O)CCC(F)(F)C1 30406,C1(NC(c2cnc(C(F)F)s2)=O)CN(C(=O)C2=CCCC2)CCC1F 30407,C1(OC)CCOCC1NC(=O)C(c1ccc(Br)cc1)(C)N 30408,C1(CCC(C)(C)NC(C2CC2(F)F)=O)CCN(C(=O)COC(=O)CO)CC1 30409,C=Cc1ccc(CNC(C23CC2CN(C(C2Cc4ccccc4O2)=O)C3)=O)cc1 30410,C(=O)(C(F)C1CCOC1)N(C)CCOCCCN(C(=O)CNC=O)C 30411,CC1CN(C)CC1C(=O)NC1(CCNC(c2ccc(C3CCOC3)s2)=O)CCC1 30412,c1(C(=O)NC(C)CN(C(=O)C(C)NC(N)=O)C)coc(OCC(F)(F)F)n1 30413,C(=O)(CCCCN=[N+]=[N-])N1C(C)CN(C(=O)Cc2ccc(F)c(F)c2)CC1 30414,CN1CCC(C(=O)N(CCCNC(C2CC2NC(=O)Nc2ccccc2)=O)C)C1 30415,c1(SCC)ccc(COC(=O)C(C)C(C)c2ccccc2Cl)cn1 30416,C1(CNC(C(C=C=C)C)=O)CCN(C(c2cc(OC)ccc2OC)=O)C1(C)C 30417,N1(C(C2CC=CC(NC(C3N(C)CC(O)CC3)=O)C2)=O)CC(O)CC12CCOC2 30418,C#CCCCC(C(=O)O)NC(C1CNCCN1)=O 30419,N1(C(CC(=O)NC)=O)CC2C(CNC(C3(c4ccccc4F)CC4(CC4)C3)=O)C2C1 30420,Nc1ccc(C(N2CC(CC(N3CCC3CO)=O)C3(CC3)C2)=O)nc1F 30421,C1(C(N(CC)Cc2nc[nH]n2)=O)CC(F)CN1C(=O)Cc1ccc(C(C)(C)C)cc1 30422,c1(C(=O)NCCCCCNC(C(N2CCOCC2)C)=O)cc(O)ncc1Br 30423,Cc1cc(=NCc2n[nH]c3c2CCC3)[nH]c(=NCc2ccc(C(F)(F)F)cc2)[nH]1 30424,C=CCC(C(=O)N(C)CC1CCCN1C(c1ccc(OC(F)F)nc1)=O)C(C)C 30425,N1(C(CCC2C(C)(C)C2)=O)C(CC(=O)NCC23CCCC2C3)C2CCCC12 30426,c1(C(N2CC(C)C(CNC(=O)CC3CCCCO3)C2)=O)c[nH]c2c(F)cccc12 30427,c1(OC)ncnc(C(N2CC3C(CN(C)C(C4(C)CCCCC4)=O)C3C2)=O)c1F 30428,C1(C(N2CCN(C)CC2)=O)CCC2(CC2)N1C(=O)CCc1nc(Br)n[nH]1 30429,C1(NC(CC=C)=O)CN(C(=O)Cc2c(Cl)cccc2Cl)CC12COC2 30430,N1(C(c2ccn3cncc3c2)=O)CC2CCN(Cc3cnc(Br)c(F)c3)CC2C1 30431,c1(N2CCCC(CNC(c3cc(CCC)nn3C)=O)C2)cc(S(C)(=O)=O)ncn1 30432,C(=O)(C(C)(C)CC(F)F)NCC(C(C(C)C)C)NC(c1ccsc1Cl)=O 30433,C1(C#N)(C(NNC(c2n(CC)nc(NC(=O)OC(C)(C)C)c2)=O)=O)CCOCC1 30434,N1(C(C2C(C)SCCC2)=O)CC(CC(=O)NC(c2ccon2)(C)C)C2(CC2)C1 30435,Cc1cncc(C(=O)NC2CCC(NC(C3CN(C4COC4)C3)=O)CC2)c1C 30436,CCC(CCO)CN=c1nc(N2CCC(CC#N)C2)c2c(ncn2C)[nH]1 30437,CC1(C)CCC(C(N2CC(C#N)C2)=O)CN1C(=O)CCc1ccncn1 30438,CC(C)C(C)(CN=c1cc(F)nc[nH]1)NC(C1CCN1C1CCCC1)=O 30439,c1(CN2C(C(=O)Nc3ccc(C)nc3)C=CC2)ccc2c(c1)CCCC2 30440,C12(NC(C(C(CC)C)O)=O)CCCCCC1N(C(=O)Cn1ccccc1=O)CC2 30441,c1(C(N2CCC(NC(CS(CC)=O)=O)(CO)C2)=O)[nH]c2cc(F)ccc2c1C 30442,N1(C(C2CCC(=O)C2)=O)CCc2ccccc2C(NC(=O)Cc2ccc(Cl)s2)C1 30443,N1(C(c2c(CNC(C(c3cnn(C)c3)C)=O)occ2)=O)CCCN(C)CC1C 30444,Cc1cc(=NCCC2CCCCN2C(c2ccc(C)c(Cl)c2)=O)[nH]c(CO)n1 30445,C1(C(C)NC(=O)CC2CCCC2)CCCCN1C(=O)CC1(C(F)(F)F)CC1 30446,c1(-c2nc(C(CC)C)nn2C23CC(C2)C3)ccc(Cl)c(S(C)(=O)=O)c1 30447,c1(OC)cc2cc(C(=O)NC(C)CCS(C)=O)[nH]c2cn1 30448,N1(C(C=CS(C)=O)=O)CCN(C(c2ccccc2C(N)=O)=O)CC1c1cn[nH]c1 30449,c1(CCC)cccc(OC(C2CC2c2cccs2)=O)c1 30450,Cc1nn(C2CCS(=O)(=O)C2)c(C)c1CN1CCCC(NC(=O)CC(F)(F)F)C1 30451,N1(C(CC(C)SC)=O)CC(NC(c2cc(C)cc(F)c2)=O)CC(F)C1 30452,c1(C(N(C(C)CNC(=O)C(F)(F)C(F)F)CC)=O)ccc2c(c1)COC2 30453,N1(C(C2(C)ON=C(C)C2)=O)CC(CO)C2(C1)CN(c1nc(C)nc(C)c1F)C2 30454,C(=O)(CC(C)CC(C)(C)C)NCCC(=C)CNC(=O)CS(=O)(=O)N1CCCCC1 30455,c1(C(N2CCC(CC(=O)N(C3CC3)CC)C2)=O)cc(F)cc(F)c1 30456,c1(N2CCC(C(C)C)CC2)[nH]c(=NCC23CC2CN(C)S3(=O)=O)nc2sccc12 30457,C1(C(=O)NCCCCNC(c2oc(C)c(CO)c2)=O)CCOC2(CCC2)C1 30458,N1(CCc2ccc(C)cc2)CCCC(C(=O)NCC(C)C)C1C 30459,c1(C(=O)NC(CNC(CC(CCC)(C)C)=O)CCOC)c(F)ccc2nc[nH]c12 30460,C(=O)(C(F)C(C)C)NC(CCOC)CNC(c1ccc(CN2CCCCC2)s1)=O 30461,c1(C(N2CCC(CC)(NC(c3cnoc3)=O)CC2)=O)ccc2c(c1)nc(O)n2C 30462,C1(CC(=O)N(CC(CN(C)Cc2sccc2Br)O)C)CC(C)(C)CO1 30463,CCC(C)(CNC(C1(C(C)C)CCN(C(=O)CC(C)SC)C1)=O)CO 30464,C1(NC(C2SC3C=CC2CC3)=O)CC2CCC1N2C(=O)C1=C(Cl)CCC1 30465,CC(C)(C(=O)NCC(CNC(C1CN(CC(F)(F)F)C1)=O)CO)n1cccn1 30466,C(=O)(CC(C)C(F)(F)F)NCC1=CCCN(C(C2=CCCC2C)=O)C1 30467,C1(CC=C)(C(=O)N(CC(=C)C)C)CN(C(C2C=C(C)CS2)=O)C1 30468,C(C(CC(F)(F)F)NC(=O)CC(CN(C)C)CC)NC(c1cc(OCC)n[nH]1)=O 30469,C1(C(C)(C)CNC(C2COC(=O)N2)=O)CCN(C(C2CCC23CCC3)=O)CC1 30470,CC(C)(CC(=O)NC1CN(C(=O)CC2CCn3cncc3C2)CC12CC2)C(F)F 30471,C(=O)(C1CCCc2nccn21)NC(CN(C)C(c1nc2ncccn2n1)=O)(C)C 30472,C1(NC(c2ccn(CC)n2)=O)CS(=O)(=O)CC1NC(c1cc(Cl)no1)=O 30473,S(=O)(=O)(c1cc(C)cnc1NCc1csc(C)c1C)N1CCCC(CSC)C1 30474,Cc1cc(=NCC2(CNC(=O)Cc3c(O)ncnc3O)CC2)[nH]c(C2CC2)n1 30475,C(=O)(CCCCCCc1ccccc1)N(C(c1ccccc1OC(F)F)C)CCO 30476,c1(C(N2CC3C(CNC(=O)C=CC4CC4)C3C2)=O)ccc(F)c(F)c1 30477,Cn1ncc(C(=O)NCCNC(C2COC(C)(C)C2)=O)c1C#N 30478,CC1CC(C(N2CCCC(CN=[N+]=[N-])C2)=O)CN(C(=O)CCNC(=O)CO)C1 30479,c1(C(N2CCC(OC)(CNC(=O)C3=CCOC3)C2)=O)c(Cl)cc(Cl)cc1Cl 30480,C1(C(N2CCN(Cc3ccc(Br)cc3)CC2)=O)CC2CC2N1Cc1cnco1 30481,N1(C(c2ccnc(C)n2)=O)CC2C3CCC(C2C1)N(C(C1(N(C)C)CCC1)=O)C3 30482,CC1CCC(C)(C=CC(=O)NCc2ccccc2SC(F)(F)F)C1(C)C 30483,C1(C(=O)NCCC2(OC)CN(C(c3ccccc3C(N)=O)=O)C2)CC(O)C(F)C1 30484,c1(OC)ccc(Cl)c(C(=O)NCCC2(NC(C3CCC(C4CC4)C3)=O)CC2)n1 30485,C(CS(=O)(=O)CC(=O)NC1CCC1CNC(=O)CCc1scnc1C)OC 30486,N1(C(C2CC2NC(=O)COC2CC2)=O)CCC(N2CCC(NC(C)=O)CC2)CC1 30487,c1(NC(C2N(C(CCC=CC)=O)CC=C2)=O)ccc(C(=O)OCC)c(Cl)c1 30488,C1(CNC(C(C)OCC)=O)(CNC(C2CC(F)C2)=O)CC12CCC2 30489,c1(C(N2CCN(C(CCOCC)=O)C(CCO)C2)=O)oc2ccccc2c1CC 30490,C(=O)(C(C)(C)CS(N)(=O)=O)NCC1CN(C(c2c(CC)ncs2)=O)C(C)C1 30491,c1(-c2cn(CC(CNC(c3cc(C)[nH]n3)=O)C)nn2)cncc(C(=O)O)c1 30492,c1(CN2CCCC(CC(=O)Nc3c(C(N)=O)nccn3)C2)ccc2c(c1)CCO2 30493,c1(CS(N2CCCC(C(=O)NC3CC3)C2)(=O)=O)ccc(F)c(I)c1 30494,C1(CNC(CCN(C(C)C)C(c2nccn2C2CC2)=O)=O)CCOC1C 30495,c1(NCCS(=O)(=O)NCC)nc2ccccc2nc1NCc1ccc(Br)cc1C 30496,CC(C)(C(=O)NC(Cc1ccccc1)CCNC(=O)C=CCF)c1ccccn1 30497,C(C(C(=O)NCCN1CC=CCC1)NC(c1ccn(C(F)F)n1)=O)OC 30498,N1(CC(C)(C)NC(C(CC)OC2CCCCC2)=O)CCN(C(C2CC2C)=O)CC1 30499,C1(C)(C(=O)NC2C(N(C(CCOCCC)=O)C)CCCC2)CCCCCCC1 30500,C(C1CCCCCC1)=CC(=O)NCCCC(C)NC(C1CC(C(C)C)C1)=O 30501,N1(C(c2c(CC)[nH]nc2Cl)=O)CCC(NC(=O)CCc2cccc(C)c2)C(C)C1 30502,C(C)(CCCC(=O)NCC1CCC(O)C1)NC(C(C)C)=O 30503,c1(C(=O)NC(C(C)NC(CN(CCC#C)C)=O)C(C)C)sc2nccnc2c1N 30504,C(=O)(CC(C)CC(=O)NC1CCN(C(C2(C3CC3)CCOCC2)=O)C1)OC 30505,C(C(N=c1[nH]nc(C#N)s1)C(C)C(C)C)NC(c1c(F)cc(OC)cc1F)=O 30506,C12(NC(c3c(COC)cc[nH]3)=O)CCC1CN(C(=O)Cc1csc(C)c1)C2 30507,N1(C(C=COCC)=O)CCOC2CCN(C(=O)C=CC(C)C)CC12 30508,N1(C(C=CCNC(C(C)c2cc[nH]n2)=O)=O)CCCC(C)C1CCO 30509,C(=O)(C(C)CC(F)F)NCC(C(C)C)NC(Cc1cnc(C)[nH]1)=O 30510,CC1CCN(CC2CCCC(=O)N2)CC1NC(c1ccsc1-n1cnnn1)=O 30511,C12(C(=O)NCC(CNC(c3nc(OCC)oc3)=O)(C)F)CCCCC1C2 30512,CC1CCC(C(=O)Nc2cncnc2)CN1C(=O)C(=O)N(CCC(N)=O)c1nccs1 30513,c1(NC(C2(NC(CN(C)C(=O)C3CC3)=O)CC2(C)C)=O)ccc2ccoc2c1 30514,C(C(C(=O)NC1COCC1NC(=O)C(C)(C)c1cocn1)OC)OC 30515,N1(C(Cc2cn(CC)nn2)=O)CC(F)CC1C(=O)NCc1cnnn1C 30516,N1(c2nc(OC)nc(C)c2)CCC(F)(F)C(CNC(c2sccc2F)=O)C1 30517,CC1CCN(C(=O)CC2N(C(=O)CN3CCSCC3)CCC2(C)C)CC12CCC2 30518,CC1(C)CCN1CC(=O)NC1CCCC1NC(C1(c2cccnc2)CCCC1)=O 30519,C(CC(C(C)C)NC(=O)CCNC(C)=O)NC(C1CC(C(F)F)(OC)C1)=O 30520,c1(CC(=O)NC(C(C)NC(COCCCCC)=O)CO)ccc(C2CC2)cc1 30521,c1(C(=O)NC2C3(CC(NC(C4(C)CC(=C)C4)=O)C3)C2)cn2c(n1)CCC2 30522,C1(C(=O)NCC2(C(=O)OC)CCC2)C=CC(NC(=O)CC2CC(=O)C2)C1 30523,Cc1cnn2cc(C(N3CC(O)CC3c3ccc(F)cc3)=O)cnc12 30524,CC1CN(C(=O)CN2CCCCCC2)CCCN1C(C1CCCC(C#N)C1)=O 30525,C1(OC)CCCCC1C(=O)NCc1cccc(CNC(=O)COC2CCOC2)c1 30526,C1(CNC(c2c(OCC#C)nccc2)=O)CN(C(c2cnn[nH]2)=O)CC(C)(C)O1 30527,N1(C(C=C(C)C(C)(C)C)=O)CC2(CCC2CNC(C2(C(F)F)CCOCC2)=O)C1 30528,c1(C(C(=O)NCC(=C)C)N(CC(F)C2CCC2)C)ccc(Cl)c(C)c1 30529,O(C1CCCc2ccccc21)CC(=O)NC1CCN(C(c2cnc(C)o2)=O)C1C 30530,C1(CCCNC(CNS(NC)(=O)=O)=O)CN(C(=O)CC2CSC2)CCO1 30531,C1(COC(c2cc(Cl)c(Br)cc2F)=O)CC2CCC(C1)S2(=O)=O 30532,N1(C(c2ccc(CNC(C(CC)COC)=O)cn2)=O)CC(O)CC1(C)C 30533,c1(C(=O)NCC(N(C(CC(CCC)C)=O)C)C2CC2)cnc2scc(C)n2c1=O 30534,N1(C(CCN(CCC)C)=O)CC(NC(c2ccc(=NC)[nH]c2)=O)CC(C)(C)C1 30535,C(C(C(=O)NC(c1cn[nH]c1)C)C(C)C)NC(C1CC(CCC)C1)=O 30536,C(N=c1cc(CC(C)C)nc[nH]1)C1CN(C(C(C=C)c2ccccc2)=O)CC1C 30537,c1(C(=O)NC(C2N(C(C(C)c3cncs3)=O)CCC2)C)n[nH]c2ccc(Cl)cc12 30538,Cc1cnnc(O)c1C(=O)NCCCCCNC(=O)CC(C1CC1)NC(N)=O 30539,c1(C(N(CCCCNC(c2cn(C)cn2)=O)C)=O)cc(OC(F)F)n(C)n1 30540,C(=O)(C1=NOC2(CCC2)C1)N1CC(=C(CNC(=O)C2=CCCCC2)F)C1 30541,N1(C(C(c2ccc(C)o2)C)=O)CCN(C(=O)C(O)CC(C)C)CC12CCC2 30542,CC1(C)CCC(C(=O)NCC2(C)CCCN(C(c3coc(C(F)F)c3)=O)C2)OC1 30543,c1(C(=O)NCC2CCC(NC(=O)COCC3CC3)C2)ncccc1Cl 30544,c1(OCCCC(=O)NCC2CCN(C(C(CSC)C)=O)C2)cccc([N+](=O)[O-])c1 30545,Cc1cc(C(N2CCCC(CC(=O)NC3CN(C)CCC3O)CC2)=O)cnc1O 30546,N1(C(C2(CO)CCN(C(c3c(OC)ccnc3)=O)C2)=O)CC2COCC2(CO)C1 30547,c1(NCCN2C(=O)CCCC2)nccc(=NCC2(CF)CC(F)(F)C2)[nH]1 30548,C12(C(N3CC(NC(C4(OC)CCOCC4)=O)C3)=O)CCOC1CS(=O)(=O)C2 30549,c1(CN(c2nnc(CC3CC3)n2Cc2cc(Br)cs2)C)c(F)cccc1Cl 30550,c1(NC(c2cccc(C(F)(F)F)c2F)C)ccc(-n2cncn2)c(F)c1 30551,C(=O)(C(F)C(C)CNC(c1ccsn1)=O)N(C(C)C)CCN(C)C 30552,c1(C(N(C2CC(C(=O)NC3CC3(F)F)C2)C)=O)ccccc1S(C)(=O)=O 30553,C=CCC(C(=O)NC(C)CCN(C)C(c1cnn(C)c1OC)=O)C(C)C 30554,c1(OC)ccc(C(N2CCC(CNC(c3c[nH]nc3OC)=O)C(C)C2)=O)c(O)c1 30555,C1(NC(COCCSC)=O)CC12CCN(C(c1csc3cncn13)=O)CC2 30556,c1(C(=O)NCC(CCNC(CN(c2ccccc2)C(C)=O)=O)O)c(C)n[nH]c1C 30557,C1(C(N(CC(CC)OC)C)=O)CCC(C)(C)N(C(=O)CC2(O)CCCCC2)C1 30558,c1(C(=O)NCC2(C)N(C(=O)C=CCO)CC(OC)C2)cc2cnn(C)c2s1 30559,N1(C(C2CCN(C(C)=O)CC2)=O)CCC(CNC(C2CC(OC)C2)=O)C(O)C1 30560,N1(C(=O)CCF)CCCC(C2CCCN(C(c3ccc4nncn4c3)=O)C2)C1 30561,C(CCCCCNC(c1cccc(C(OC)OC)c1)=O)N(C(CSC)=O)C 30562,Cc1[nH]nc(C(=O)N(C)CCOCCCN(C(=O)Cc2ccnn2C)C)c1Cl 30563,N1(C(c2c(C)c(Br)cnc2)=O)CCCN(C(=O)C(C(C)C)N(C)C)CC1C 30564,Cc1noc(C)c1.C1(C(=O)NCC)CC(O)CN1C(c1ccc(OC(F)F)nc1)=O 30565,n1(C(C(=O)N(CCNC(c2c(C)ccnn2)=O)C2CC2)C)cnc2ccccc12 30566,CC1=C(C(=O)N2C3CCC(C3)C2CC(N2CCCCC2C(F)F)=O)CCC1 30567,c1(C(=O)OCC)cc(CN(C)CC2CCCOC2c2ccccc2)nn1C 30568,c1(CCC(=O)NCC(C2CCCC2)NC(COC(C)C)=O)cnn(C)c1 30569,n1(C(C)C)cnnc1CC(N1CC(CCCCNC(C2CC2C)=O)C1)=O 30570,C1(NC(Cc2cnc(C)s2)=O)CC2CC1CN(C(C1(Br)CC1)=O)C2 30571,C1(CNC(C2(CSC)CC2)=O)CCN(C(=O)Cc2cccc(C)c2)C12CCC2 30572,C1(NC(C2CN(C)C(=O)C2)=O)CC12CCN(C(c1conc1C(C)(C)C)=O)CC2 30573,CCC(=O)CCC(=O)N(CCCCN(C)C(c1cocc1C(N)=O)=O)C 30574,N1(C(C(C)SCCCC)=O)CC(C2CC2)(C(=O)NCc2csc(C)c2C)C1 30575,C1(NC(C=NOC)=O)CCC2(CCN(C(=O)CCc3ncc(F)cn3)C2)C1 30576,c1(C(=O)OC)cncc(CNC(=O)C(=O)NCCCCN(C)C)c1 30577,N1(C(C2N(CCC)CCC2)=O)CCc2ccccc2C1CNC(c1ccns1)=O 30578,c1(SC)ccc(N(C(=O)Cc2nn[nH]n2)Cc2cccc(-c3nn[nH]n3)c2)cc1 30579,C1(NC(C2CCN(C)C2)=O)CCC12CN(C(=O)C=CCF)C2 30580,N1(C(C(CCC)OCC)=O)CC2CCC(N(C)C(c3ccc(Cl)cn3)=O)C2C1 30581,Cc1snnc1C(=O)NCC(=O)N(C1CN(C(=O)C(C)NC(=O)C(C)(C)C)C1)C 30582,N1(C(C(CC)C)=O)Cc2nnn(CC)c2C(C(=O)Nc2ccncc2O)C1 30583,N1(C(CCC(=O)NC)=O)CC(NC(C2(C(F)F)CCCCC2)=O)CCC1C 30584,Cc1cccc(C)c1NC(=O)CNC1CCC(Nc2ncccn2)CC1 30585,CCC(F)(F)C(=O)N1CCC(C(C)CNC(=O)CCC2CC(F)(F)C2)CC1 30586,N1(c2n(CCS(=O)(=O)N(C(C)C)CC)c(CO)nn2)CCOC2(CCSC2)CC1 30587,N1(C(C2C3N(C(c4cc(C)c(O)nn4)=O)C(CC3)C2)=O)CC2CCC1C(CO)C2 30588,S(=O)(=O)(c1ccc(N(CC(c2ccccc2)F)C)nc1)N(C(CC)CSC)C 30589,N1(C(c2c(OC)csc2)=O)CC(CNC(C2CC(=C3CCC3)C2)=O)C(O)C1 30590,c1(C(=O)NCCN(C(c2ccc(F)c(OC)c2F)=O)CC)cccc2ccnn12 30591,c1(C(N2C(C(C)NC(CNC(CC)=O)=O)CCCC2)=O)cc(C)n(C(C)C)c1C 30592,C(=O)(C#CC1CCOCC1)N1CC(CCCCNC(c2n(CC)c(O)nc2)=O)C1 30593,C(=O)(CCC(=O)C(C)(C)C)N1CCC(C)C1CNC(=O)C(c1ccccn1)O 30594,N1(C(c2c(COC)noc2)=O)CC2CCN(C(c3cc(N)ccc3C)=O)C2C1 30595,CC(C)C(C)C(CNC(=O)COC(F)F)NC(c1cc(N)ccc1F)=O 30596,C(=O)(C(C)(F)C(F)(F)F)NC(C1CCN(C(C2(C(=O)NC)CC2)=O)CC1)C 30597,S(=O)(=O)(c1cccc(C(=O)NC23CC(NC(=O)Cc4conc4C)(C2)C3)c1)NC 30598,Cc1cc(CCNC(=O)CN(C(=O)CC2CC(C)C2)C(C)C)nn1C 30599,c1(CC(=O)NCC(CC)NC(C(CCC)NC(N)=O)=O)cc(Cl)cc2c1OCC2 30600,Cn1[nH]nnc1=NC1CS(=O)(=O)CC1NC(C1CC(c2ccccc2)=NO1)=O 30601,N1(C(C(C(C)(C)C)O)=O)CC2(C(=O)NCCn3ccnc3)CCC1CC2 30602,C1(C(=O)NCC2CC(CN=[N+]=[N-])C2)C2CCN(C(C3(CO)CC=CC3)=O)CC12 30603,c1(CC(=O)NC(C2CCCO2)COC)cccc(NCc2ccccc2Cl)c1 30604,C1(NC(c2n[nH]c(C)c2C)=O)CC2CC(NC(=O)CCn3cccc3)CC2C1 30605,Cc1nc(C(C)C)ccc1C(=O)N(C)CC1(O)CN(C(=O)COc2ccon2)C1 30606,c1(C(=O)NCC(C)N(C)C(c2cnco2)=O)c(F)ccc(N)c1Br 30607,CCC(F)(F)CC(=O)N(C1CN(C(c2n[nH]cc2C(F)(F)F)=O)CC1(C)C)C 30608,N1(CCCNC(c2cscn2)=O)CCN(C(c2cnn[nH]2)=O)CC1 30609,c1(CC)cc(C)c(C(=O)NCCC2(C(=O)N(CCN3C(=O)CCC3=O)CC)CC2)o1 30610,N1(C(CCOCC(C)C)=O)CCC(CN(C(=O)C(F)(F)c2ccncc2)C)CC1 30611,C1(F)(CNC(C=C(C)C(C)C)=O)COCCN(C(=O)CC2(CS(C)(=O)=O)CC2)C1 30612,S(=O)(=O)(c1cccnc1)NCCC(=O)NCC1C(CNC(=O)C2=CCC2)C1 30613,Cc1cncc(N)c1.c1(CCC(NOC(=O)C(F)(F)F)=O)ccc(O)nn1 30614,C(=O)(CCCCN(C(=O)C(C)(C)C1(O)CCC1)C)NCC(C)CCO 30615,S(=O)(=O)(c1ccc(=NCCCC(F)(F)F)[nH]c1)N1C(c2cccnc2)CC(C)C1 30616,c1(C(N(C2CCCN(C(C3CCCC34CC4)=O)C2)CC)=O)ccc(C)cc1C 30617,CC(C)C(C(=O)N1CCC(C(CO)NC(C2CC2C(F)F)=O)CC1)NC=O 30618,C1(NC(C2CCCN(C(C(N3CCNC3=O)C)=O)C2)=O)CC2(C1)CC(O)C2 30619,c1(OC)ncccc1CC(=O)NC1CN(C(c2cnccc2C)=O)CC1O 30620,N1(c2ccnc(NC3CC(C)(C#N)C3)n2)CCC2CCC12C 30621,c1(C(=O)NCC2C(NC(c3cnc(OCC)nc3)=O)C2)c(F)ccc2nc[nH]c12 30622,C(=O)(C(CCC(N)=O)n1cc(C2(F)COC2)nn1)N(C)Cc1cn(C)c(=O)n1C 30623,N1(C(c2nc(C(C)C)oc2)=O)CCN(C(c2cncc(O)c2)=O)C2(CC2)C1 30624,c1(NC)ccc(C=CC(=O)NCC(C)(C2CCC2)NC(=O)C(C)CF)cc1 30625,Cc1c(C(=O)NC2C=CCCC2CNC(=O)COCC2CCCO2)nnn1C 30626,c1(C(=O)NCC2CCN(C(C(C)(CO)OC)=O)C2)cc(Cl)c(F)cc1N 30627,CCCCC(=O)C(=O)NCC1CN(C(C2CC23CCOCC3)=O)CCO1 30628,c1(C(=O)NC2CCCN(C(C(=Cc3cnc[nH]3)C)=O)C2C)cnc2ccsc2c1 30629,c1(-c2ccc(CC)cc2)ccc2[nH]cc(C(N3CCCC(C(=O)OC)C3)=O)c2c1 30630,C1(C(=O)NCC(=O)N(C)C)CCN(c2ncccn2)C1 30631,C=CC1(C(=O)NC(C)CCc2cn[nH]c2)CCN(C(=O)CCc2ccn(C)c2)C1 30632,c1(C(=O)NCC(CC)(CC)NC(C2C=CCC2)=O)ccc(N)cc1Cl 30633,N1(C(C2CC(SC)C2)=O)CC(NC(c2ccccc2SC(F)F)=O)C(F)C1 30634,O(NC(=O)C(CCF)NC(c1ccco1)=O)CCCC(=O)OC 30635,c1(C(=O)NCCC2(CN3CCN(C(=O)C4CC4)CC3)CC2)ccc2nncn2c1 30636,Cc1nc(C)c(C(=O)NC(C2CCN(C(c3cc(C(F)(F)F)no3)=O)CC2)C)[nH]1 30637,N1(C(=O)N(CC2CCCO2)CC2CCCO2)CCCN(Cc2cccnc2)CC1 30638,c1(CNC2CCC(NC(C(CC)N(C(C)=O)C3CC3)=O)C2)cc(F)c(F)cc1Br 30639,c1(C(N(C2CCC(NC(c3cc(=O)cc[nH]3)=O)C2)C)=O)ccc(CO)nc1 30640,C(=O)(CC(O)CC(C)(C)C)N1C2C(N(C(CCCCCCC)=O)C)CC(C2)C1 30641,C1(C(=O)NCC(C)N(C(=O)C(=O)NCC2CC2)C)CC2CSCC(C1)C2 30642,C1(NC(C2(CC(C)C)CC2)=O)CN(C(=O)CC2OCCO2)C2(CCC2)C1 30643,C(C(C)(CO)NC(=O)CCCSC(F)(F)F)NC(C1C(COC)C1)=O 30644,C1(C(N(CCC(C(C)C)NC(=O)C(C)c2ccco2)C)=O)CN2CCCN1CC2 30645,Cc1cc(C(=O)NC2CCCC(C(=O)Nc3ncc(C#N)s3)C2)n(C(F)F)n1 30646,C#Cc1ccc(C(=O)N(C)Cc2ccc(C(=O)NCC(O)COC)s2)c(C)c1 30647,Cc1c(-c2nc(-c3cccnc3O)nn2CC2CCOC2)cnn1CCO 30648,C12(CNC(C3C(C=C)C3)=O)CC3CC(CC(NC(=O)C(O)C(F)(F)F)(C3)C1)C2 30649,N1(C(C(CC)(CC)OC)=O)CCN(C(C2CCCCN2C)=O)C2(CC2)C1 30650,CC1CN(C(C2CCC3(CCC3)OC2)=O)CCCN1C(=O)CC1CC(C2CC2)C1 30651,C12(C(N(CCN=[N+]=[N-])CC)=O)CC1CCN2C(=O)CC1CC2CC2C1 30652,n1(CCS(CC)(=O)=O)c(=NCCc2sc(N(C)C)nc2C)[nH]c2cc(Cl)ccc12 30653,C1(C(C)CO)CCN(C(=O)C(c2ccnn2C)NC(=O)CCN(C)C)CC1 30654,N1(CC2C(C)(C)CCN(CC3CC4CNC3C4)C2)C(=O)C2CC=CCC2C1=O 30655,COn1cnc(C)c1C(=O)NC1CC1CNC(c1cc(C)ccc1C1CC1)=O 30656,C1(CCNC(c2ccc(Cl)s2)=O)CCN(C(=O)COc2cccc(O)c2)CC1 30657,C(C(=O)NCC(CO)OC)(C1CCC1)NC(COCCC=C)=O 30658,c1(C(=O)NCCCCNC(c2ccnc(C)n2)=O)cccc2c1COC2 30659,c1(C(=O)NCCN(C(=O)C(F)CC2CCC2)CC)ncncc1Cl 30660,CC1Cc2ccccc2N1C(C1CC2CCCC2N1)=O 30661,N1(C(C(CC)NC(N)=O)=O)CCN(C(c2n[nH]c(O)n2)=O)CC1c1cnn(C)c1 30662,n1(CC)cc(CN2CCC(CC(N3CCCC(CN(C)C)C3)=O)C2)c(C)n1 30663,c1(C(C)(N(n2cccn2)C)C2CC2)nc(-c2ccccc2)nn1-c1cnn(C)c1 30664,c1(OC)ccc2nc(C)c(C(=O)NCC3CCC3NC(c3ccsn3)=O)n2n1 30665,C1(NC(c2c(COC)cccc2)=O)CN(C(=O)Cc2ncccc2C)CCC1C 30666,C1(C(=O)NCC2C(NC(=O)Cc3ccc(Cl)cc3)C2)CN2CCC1CC2 30667,Cc1cnc(C(=O)NC2CCN(C(=O)C(=CC3CCCCC3)F)C2(C)C)cc1C 30668,Cc1ncc(C(=O)NC2(C)CCCN(C(c3c[nH]c(Br)c3)=O)C2)c(=N)[nH]1 30669,c1(C(=O)NC(C2CCCCN2C(=O)COc2cccnc2)C)cccc(N)c1O 30670,N1(C(Cc2nc(C)[nH]n2)=O)CCCC12CCN(C(=O)CCc1nncn1C)CC2 30671,C(=O)(CC(O)(C(F)(F)F)c1ccc(C)o1)NC(CNC(C=C(CC)CC)=O)C 30672,C1(C)(C2CCCN(C(C(=O)NCCCOC)c3cccs3)C2)NC(=O)NC1=O 30673,C1(NC(=NCCSC)NCCc2cccc(O)c2)CCOC2(CCSC2)C1 30674,N1(C(c2cc(CC)[nH]n2)=O)CCC=C(C(=O)N2CC3CCC2C(O)C3)C1 30675,n1(CCC)ncc(CN2CC(CC(=O)NC3CSC3)C2)c1C 30676,c1(C(N2CCCCC(NC(C(CCC)C#N)=O)C2)=O)noc2ncccc12 30677,c1(C(N2C(C)C(NC(c3sccc3F)=O)CC2)=O)cc2c[nH]cnc-2n1 30678,C(=O)(CC(O)CC(C)(C)C)N1CC(CC)C(NC(c2ccncc2)=O)C1 30679,C1(C(=O)O)C=CCN(Cc2ccc(N3CCCC3)nn2)C1 30680,c1(C(C(=O)N2CC(N(C(Cc3cnc(C)[nH]3)=O)C)C2)(F)F)cccc(F)c1F 30681,C1(C(=O)NCc2ccc(C#N)o2)(NC(CC=CCCCCC)=O)CCCCC1 30682,c1(C(N2CCCC2)=O)ccc(Cl)c(S(=O)(=O)N2C3CCCC2CC(O)C3)c1 30683,C1(CN)C2CC3CC(C2)CC1(CNC1CCCc2c[nH]nc21)C3 30684,C1(OC)(CNC(C2(C)CCCCCC2)=O)CCN(C(c2[nH]c(O)nc2C)=O)CC1 30685,CC1(C#CC(=O)N2CCC3C(NC(=O)CSCC(F)(F)F)C3C2)COC1 30686,C1(NC(C(CC)C)=O)CN(C(C2(C(F)(F)F)CCCC2)=O)CC1n1cccn1 30687,C1(NC(c2ccnc(Cl)c2)=O)CCCCN(C(c2c(O)ncnc2O)=O)C1 30688,C1(C(=O)NCC2C=CC(NC(C3(OC)CC3)=O)C2)CS(=O)(=O)CC(=O)N1 30689,C(C)(CC(=O)N1C(CNC(C2CCCCC2)=O)CC2CC12)(C(F)(F)F)N(C)C 30690,c1(COC)cccc(CNC(C2COCCN2C)=O)c1 30691,c1(C(=O)NC(CNC(c2nccc(C#C)c2)=O)C(C)C)ccc(F)c(C#N)c1 30692,c1(CC(=O)NCC2Cc3cc(Br)ccc3O2)ccc2c(n1)OCCO2 30693,C#Cc1cn(C)nc1C(=O)NCC(O)CC(=O)N1CC(OCCO)C1 30694,C1(C(F)(F)F)(OC)CCCN(C(=NCc2ccc(C)cc2C)NC(C)C)C1 30695,C(=O)(CCCS(C)(=O)=O)N1CCCN(C(c2c(C)ncn2C)=O)CC1 30696,CCC(O)(C(=O)NCC1CC2CC2N1C(=O)C(C)=C1CCCC1)c1ccccc1 30697,C1(NC(c2cc(C)no2)=O)CCC2CN(C(c3cncc(C(N)=O)c3)=O)CC2C1 30698,CC1CCCCN1CC(N1CCC(C(C)C(=O)NCCC(O)C2CCC2)CC1)=O 30699,c1(C(N(CC(CNC(Cc2cc(C)on2)=O)O)C)=O)sc(C)nc1C 30700,C1(SCC)CCC(NC(c2c[nH]nc2-c2ccccc2Cl)=O)CC1 30701,c1(C(C)NCC(c2ccc(OC)cc2)(C)O)nc(O)c2c(C)c(C)sc2n1 30702,N1(C(C2C(OCC)C2)=O)CCC(CCC(=O)NC(C)CC2(O)CCC2)C1 30703,c1(C(N2CC3(C(=O)OCC)C(C(F)(F)F)(C2)C3)=O)cc(C)c2nc(C)cn2n1 30704,c1(C(=O)NCC(C(C)C)(C)NC(C2CC3(C2)CC3F)=O)cnc(C2CC2)[nH]c1=N 30705,c1(C(C)=O)ccc(NC(c2cccc(I)n2)=O)cc1.c12ccc(nc1)[nH]c2=O 30706,N1(C(C(c2ccc(C)cc2)C)=O)CC2CC(NC(=O)CC3CCOCC3)CC1C2 30707,N1(CCNC(=O)CSC2CC2)CCN(C(C2(C(F)F)CCC2)=O)CC1 30708,C12(NC(C3C(C)(C)C(OC)C3)=O)CC(CNc3ncnc4sccc34)(C1)OC2(C)C 30709,C1(C(=O)NC2CCN(CC)C2)CCC(CNC(C2C3COCC23)=O)CC1 30710,C1(OC)(OC)CC(C)(C(=O)NC(C)CNC(=O)C=C(C)C)C1.C(C(C)(C)C)O 30711,c1(C(=O)NC2(C3N(C(c4nncc(OC)c4)=O)CCC3)CC2)c(Cl)cccc1Cl 30712,c1(SC)cc(C(=O)NCC(c2ccccc2F)NC(=O)CC2CC2(C)C)c(C)o1 30713,c1(CCCC(=O)N(C2CCN(C(CC=C(C)C)=O)C2)C)ccccc1Cl 30714,CCC(CC(C)C)C(=O)N1CCC(CO)C(NC(=O)CC2CCCC(C)C2)C1 30715,c1(C(N2CC3C(CNC(C(CCN(C)C)O)=O)(C3)C2)=O)c(Cl)cncc1Cl 30716,Cc1cc(NC(c2cc(CNC(c3cc(CO)ccn3)=O)on2)=O)c(=O)n(C)c1 30717,N1(C(C(CCCC)O)=O)CC(CNC(=O)C(=C2CCCCC2)F)OC2(CCC2)C1 30718,N1(C(C2CCN(CC)C2)=O)CCC(O)(C(=O)NCC2(O)CC(CO)C2)C1 30719,c1(NC2CCN(CC=C)CC2)ncc(S(=O)(=O)N2CCCC(C)C2)cc1Cl 30720,CCC(CCOC)C(=O)N(CC)CC1CCCN1C(c1nccc(OC)c1O)=O 30721,C1(C(=O)NC(CC)C2CCC2)C2CC2CN1C(=O)CC1(C)CC1 30722,C(CC#CC(C)(C)C)NC(CC(CC)N(C(=O)CCC1(C#N)CCC1)C)=O 30723,Cc1cc(C(=O)NC2CCN(C(=O)COCCCF)CC2F)cc2nc[nH]c12 30724,c1(CC(N2CCC(C(C)(C)NC(=O)CC34CCCC3C4)C2)=O)cccnc1Cl 30725,Cc1cc(Cl)cc(C)c1OCC(=O)NCC(C)N(c1ncnc(NC(C)C)n1)C 30726,c1(NCC(C)S(N)(=O)=O)ncccc1S(=O)(=O)NC(CC(N)=O)C1CC1 30727,c1(CCCN2C(=O)CCC2)nnc(N(c2ccccn2)C)n1CC1CC1 30728,Cc1ccc(C(N2CC3(CCC3NC(=O)CC3CC4(CCC4)C3)C2)=O)cc1C#N 30729,CN1CCCC(F)(C(=O)NCCOC2CCN(C(C3(C)CCC3)=O)CC2)C1 30730,c1(C(=O)NCc2c(CNC(CC=C)=O)nccc2)cc2ccc(C)cc2o1 30731,C1(C)(CNC(COC(CC)(C)C)=O)CCN(C(=O)CSCCN(C)C)CC1 30732,C1(C(N2CCC(N3CCN(C(=O)Cc4cnco4)CC3)C2)=O)CCCCC1(F)F 30733,C(=O)(C(C)CC(F)F)NC1CC(C(C)NC(c2ccn(CCC)n2)=O)C1 30734,CCC(C)C(=O)N(C(CNC(C1CC2CC2C1)=O)C1CC1)C 30735,c1(-c2cccc(C3C(C(=O)NC(CC(C)=O)C)C3)c2)ccc(S(=O)(=O)N(C)C)cc1 30736,C1(NC(c2n(CC)ccn2)=O)CCCN(Cc2nnc(C3CC3)s2)C1 30737,C(=O)(N=c1nc[nH]n2cccc12)C1N(C(c2cccc(OC(C)=O)c2)=O)CCC1 30738,C(=O)(C(C)=NOCC#N)NCC1C(C(=O)NCC(COCC)C)C1(C)C 30739,CCC1=C(C(=O)NCC2CCN2C(C2CCc3n[nH]c(C)c3C2)=O)CCCO1 30740,C1(NC(c2c(C)cccn2)=O)C2COCC1CC(NC(=O)C1=NOC(C)C1)C2 30741,N1(C(C(C)NC(C)(C)C)=O)CC(C2CN(C(=O)CSC3CCCCO3)C2)C1 30742,C1(COC)(NC(=O)C(F)CC2CCCC2)CN(C(=O)Cn2cc(Cl)cn2)C1 30743,CCC(CCC(=O)NCC1(C)CC(NC(=O)CSc2ccc(C)cc2C)C1)OC 30744,Cc1c(O)ccc(C(=O)NC2CC2CNC(=O)CCC(=O)NC2CCCC2)c1C 30745,C1(C)(C(=O)NC2CC(CNC(C(C)OC3CCCC3)=O)C2)CCC(F)(F)CC1 30746,c1(C(=O)NC(CCCCNC(C2(C)ON=C(C)C2)=O)C)c(C)nc(O)nc1C 30747,c1(OC)cc(CN2CC3(CC(C(=O)Nc4cccc(C)c4Cl)C3)C2)cc(F)c1 30748,C(CCCCCC(=O)NCC(O)C1CCC1)NC(C(COC)(F)F)=O 30749,C(CC(=O)NCC1C(C)CCN1C(=O)CN(C)CCOC)(C(F)(F)F)OC 30750,CCCC(C(=O)N1CCCCC(N(C(=O)CCOCCCOC)C)C1)C(C)C 30751,O=C(CC1=CCOCC1)N1CCCN(C(=O)C(c2ccccc2F)O)CCC1 30752,N1(C(C2C(C(=O)O)CC2)=O)CCN(Cc2ccc(CC(F)(F)F)cc2)CC1 30753,CC1(C(=O)NCCOCCNC(C2CCCCNC2=O)=O)CCCNC1=O 30754,C1(CNC(CCCOCCOC)=O)Cc2ccccc2CN1C(c1cc[nH]c1)=O 30755,C(=O)(CCCCCCCC=C)NCC(C)N(C(COCCC#C)=O)C 30756,c1(CC)cc(C(N2CC(F)(c3ccccn3)C2)=O)no1 30757,C(=O)(C1=NNC(C(F)(F)F)C1)NC1(C)CCN(C(CCc2n(C)ncn2)=O)C1 30758,c1(NC(CNC(=O)OCC)=O)ccc2c(N)ncn2c1.c1ccccc1 30759,C(=O)(C1c2ccccc2CN1C(c1cnc(O)c(Cl)c1)=O)NC1CC(=O)OC1 30760,Cc1nc(C(N2CCC(CC(N3CCC(C(C)(C)O)C3)=O)C2)=O)c(C)s1 30761,C1(N(C)C(=O)C2CC2)CCN(C(=O)C#N)CCC1COCCO 30762,c1(C(=O)NCC#CC(=O)NCc2onc(COC)n2)cnnc(C)c1C 30763,c1(C(=O)NCC(CNC(CC(CC)CC)=O)OC)ccc(F)c2ccoc12 30764,CCCC(C#N)N(C(c1ccc(CCCC)o1)C(=O)NC)CC 30765,C1(C(N2CC(C)CC(CC)C2)=O)(CC)CCCN(C(=O)CC#N)C1 30766,C1(C(=O)Nc2ccc(OC)c(N3CCOC3=O)c2)CCC(C2CC2)CC1 30767,N1(C(CN2CCC(C)(C)C2)=O)CCC(NC(c2cc(C3CC3)no2)=O)C(OC)C1 30768,N1(C(C(C(C)C)SCC)=O)CC(NC(c2cnnn2C(C)C)=O)CC1(C)C 30769,c1(C(N2CC(C)(C)C(NC(=O)C(F)=CCCF)C2)=O)cc(F)c(O)c(F)c1 30770,c1(C(=O)NCC(C)CNC(c2ccnc3ccnn23)=O)cc2c(s1)CCCCC2 30771,c1(NCC2OCC(CNC(CSc3cn(C)nc3)=O)C2)ccnc2ncnn12 30772,C(CC(F)F)(C(=O)NC1CC2(CCCC2)C1)N(C(c1c(CC)con1)=O)C 30773,c1(C(C)C)[nH]nc2cncc(C(N3CCC(C)(NC(=O)C=CCO)C3)=O)c12 30774,c1(OC)cccc(C(N2CCCC(F)(F)C2)C(=O)NCc2cccc(Cl)c2)c1C 30775,c1(NCCC2(O)CN(C(C(CC)SC)=O)C2)ncc(Br)cc1[N+](=O)[O-] 30776,C1(C)(C(=O)NCCCN(C(=O)CC2(C#N)CC2)C)CCC(=O)N1 30777,CC1(C2CC2C(=O)N(CCNC(c2ccc(C(F)(F)F)nc2)=O)C2CC2)COC1 30778,NS(=O)(=O)N1CC(C(=O)NC2(C3CN(C(=O)CCCCCF)C3)CC2)C1 30779,NS(=O)(=O)c1ccc(O)c(C(=O)NC2CC(NC(c3ccc(O)nn3)=O)C2)c1 30780,C1(NC(CCC(=O)NCCC)=O)CN(CCOCC)CCC1C 30781,C1(CC(=O)NCc2cn(CCNC(C=CSC)=O)nn2)CC2(CC2)CO1 30782,C1(C(N(CCCSC)C)=O)CCN(C(=O)C(C)c2cccs2)C1C(C)C 30783,C(c1ccc(F)cc1)=CCNCc1nccc(CC(=O)O)n1 30784,S(=O)(=O)(c1cnccc1N1CC(OC)CC(C)C1)NCc1nnc(COC)s1 30785,CC1(C)CC(C(=O)N(C2CCCC2)CCCNC(C2CC3CC2CC3O)=O)=NO1 30786,C(CC(C)(C)C(=O)N1CCN(CC(N)=O)CC1)NC(C(c1ccc(C)o1)C)=O 30787,CCC(C(=O)N(C1(C(N2CCC3CCC23)=O)CCC1)C1CC1)C(F)(F)F 30788,N1(CCCNC(C(CC)C)=O)CCN(C(=O)C=CC(N2CCC(C)CC2)=O)CC1 30789,Cc1[nH]c2ncnc(N3CCC(C)(NC(C4C5CCCC45)=O)C3)c2c1C 30790,C1(C)(CC)CCCN(C(C2CCC(O)CN2C(=O)CC2CCOC2=O)=O)C1 30791,N(C(=NCCC1CC=CCO1)NCc1cnccn1)CCOC(C)(C)C 30792,C(=O)(CS(=O)(=O)C1CCCC1)N(C1(c2nn[nH]n2)CC1)C 30793,c1(C(N2CCOC(CCNC(C3CC(C(F)F)C3)=O)C2)=O)ccc2nnnn2c1 30794,C1(NC(C=CCCC)=O)CN(C(=O)C(c2cccc(C)c2)(C)C)CC1O 30795,C1(CNC(C(CC)OCC)=O)CC(NC(=O)Cc2cscn2)C(O)C1 30796,C=CC1(CO)CCN(C(=O)C(C)(CSC)NC(=O)COc2cccnc2)CC1 30797,Cn1cc(CC(O)C(=O)NCCCOCCNC(=O)C=Cc2cnc[nH]2)cn1 30798,C1(C(=O)NCCC(CC)C)CC12CC(NC(c1cnccc1C)=O)C2 30799,c1(C(=O)NC2C(C)N(C(c3cc[n+]([O-])cc3)=O)CCC2)ccc(N)cc1[N+](=O)[O-] 30800,c1nnn2c1CN(CCCNCCCNC1C3COCC13)CC2 30801,C(=O)(N=c1nc2ncc(Cl)cn2[nH]1)CCc1ncc(C(C)(C)C)o1 30802,n1(CC)nc(C)c(CC(N2CCC(O)(C(C)NC(=O)CCCC(N)=O)C2)=O)c1C 30803,N1(CCCC=C)CCC2C(CCCN2C(=O)C(c2cnn(C)c2)C)C1 30804,Cn1c(=O)oc2c(C(=O)NCC(CNC(c3ccnc(O)c3)=O)CO)cccc12 30805,OCC1CN(CC2CC3(CCC3O)C2)Cc2ccccc21 30806,N1(C(C(C)n2cccc2)=O)CC(CNC(=O)CC2(C(F)F)CC2)CC(C)(C)C1 30807,N1(C(C(COCC)C)=O)CC2(CCN(C(=O)C(C)(C)c3cccs3)CC2)CC1C 30808,c1(C(=O)NC(CNC(c2cc(CC)c(CC)o2)=O)CO)ccn2cncc2c1 30809,N12CCC(CC1)c1n[nH]cc1C2.C(=O)(C(C)C(C)C)N(c1c(C)cns1)CC1CC1 30810,c1(C(N(C2CCC(CNC(=O)CSC(F)F)CC2)C)=O)cccc(F)c1C(F)F 30811,N1(C(c2cc(CCC)on2)=O)CCC(O)(CN(C)C(C2CCN(C)C2C)=O)C1 30812,C1(NC(=O)CN2CC3CC3C2)COC2CN(C(=O)CCSC3CCCC3)CC12 30813,N1(c2n(CC)c(-c3nc(C(F)(F)F)c[nH]3)nn2)CCCN(CC(F)(F)F)CC1 30814,S(=O)(=O)(C(F)(F)F)N1CCC(C(=O)NCC2C=CCN2C(=O)Cc2cnc[nH]2)C1 30815,N1(C(CC(C)n2ccnc2)=O)CCC2(CC1)CC2NC(C1CSC1)=O 30816,c1(C(N2CC(O)(CNC(C3(C)C(CC)CCC3)=O)C2)=O)ccc2oc(=N)[nH]c2c1 30817,C12(NC(Cc3cc(CC)no3)=O)CCCCCC1N(C(c1nnsc1N)=O)CC2 30818,CC#CCCC(=O)N1CCC(C(N2CCCC2COC(C)=O)=O)O1 30819,N1(C(=O)CCN(C(c2ccco2)=O)C2CC2)CC2(CCC2O)C1 30820,n1(CCCC)nnnc1C(c1csnc1OC)NCC(n1cccn1)C 30821,CCCCCCC(=O)N1CCCC(C(N2CCC3CC2CO3)=O)C1 30822,c1(-c2ccccn2)cc(-c2noc(C3CCC(=O)O3)n2)ncn1 30823,C(=O)(CCS(N)(=O)=O)NCC(C(C)(C)C)NC(CCC(C)SC)=O 30824,c1(CC(C(=O)N(CCNC(=O)Cc2cc(C)[nH]n2)CC)O)ccccc1Cl 30825,C(C(=O)NC(C)CCOC)(C(C)C)NC(CCOCCC)=O 30826,C1(CNC(C(C)(C)CCl)c2n(CCOC)nnn2)COc2ccccc2C1 30827,C1(C(C#C)NC(=O)N(CCCN(C)C)C)CC(F)(F)C1 30828,S(=O)(=O)(c1cc(F)ccc1F)NC(C1CC(NCc2c(OC)nc(Cl)cc2)C1)=O 30829,C1(CNC(c2ccoc2Br)=O)CCCCC1NC(C1(C2CCCO2)CCC1)=O 30830,c1(N2CCC(Nc3c(C(=O)OC)c(C)sc3)C2=O)cc2ccccc2o1 30831,Cc1ccn(C)c1C(=O)NCC1CCCN(C(C2CCC(=O)N2C)=O)C1 30832,N1(C(c2ccnnc2C(F)F)=O)CCCS(=O)(=O)CC1C1CC1 30833,C(=O)(C(O)C(C(C)C)OC)NCCC(CNC(C(F)=CCC)=O)(C)C 30834,c1(NC(N2CCC(NC(COCC)=O)C2c2cccnc2)=O)cc(Cl)c(F)c(Cl)c1 30835,c1(OC)ccc2c(c1)C(C(=O)N1CCC3CC1CN3c1nccc(Br)n1)CC2 30836,C1(C(=O)NCC2(C)CCN(C(C=COCC)=O)C2)CCC12CCOCC2 30837,N1(C(c2cn(CCCOC)nc2)=O)CC(NC(c2ccoc2Br)=O)C(O)C1 30838,c1(C(=O)NC2C(C)CN(C(c3nn(C)cc3Cl)=O)CC2)cc2c(cc1O)OCO2 30839,N1(C(C(C#C)(C)C)=O)CC2CC(NC(=O)Cc3cnccc3C(F)(F)F)C(C2)C1 30840,c1(NC(C(COCC)NC(=O)CC2CC2(C)C)=O)ccn2nccc2c1 30841,c1(C(=O)NC(CCN(C(c2ccc(SC)o2)=O)C)C(C)C)c(C)ccc(C)c1N 30842,C1(C(=O)NC(C2(C(N3CCC3CC(N)=O)=O)CC2)C)CC=CC(O)C1 30843,C12(CNC(c3cc(CO)ccc3Cl)=O)CCC(CC1)CN2C(=O)C(F)F 30844,CC1CCN(C(C2(C(F)F)CC2)=O)CCN1c1ncc(I)cn1 30845,Cc1nn(-c2cccc(F)c2)cc1C(N1CCCC(NCC(F)F)C1)=O 30846,c1(C(=O)NC2CC(C)N(C(=O)C3=CCOCC3)C2)c[nH]c(=N)nc1O 30847,Cc1cnncc1C(=O)NC1(C)CC(NC(C2CCCSC2)=O)C1 30848,N1(C(C(C)OCCCCCC)=O)CC(NC(c2ccnnc2C)=O)CC(C)(C)C1 30849,N1(C(C=C(CCC)C)=O)CC(O)(C2(CNC(c3cccc(Cl)c3Cl)=O)CC2)C1 30850,C1(CNC(C(CN(C)C)(F)F)=O)CC2CCC1N2C(C1SCCCS1)=O 30851,CCCCCC(O)C(=O)NCC1CN(C(c2cnc(NC)cn2)=O)CC12CCC2 30852,n1(CCOC)ccc(C(=O)N(CCCN(C(=O)Cc2nonc2C)CCCC)C2CC2)n1 30853,C1(CNC(C(CC)=CCCC)=O)CN(C(=O)COC)CCN1C 30854,N1(C(CC(C)C(F)F)=O)CCOC2(C1)CN(C(C1(C#N)CC3(CC3)C1)=O)C2 30855,C=CCCC(CO)NC(=O)CC1(Cn2cc(C(=O)N)nn2)CC1.C1(CC2CC2)CC1 30856,c1(NC(CC2(C)CN(Cc3cc(Cl)ccc3Br)C2)=O)ccc(Cl)c(C#N)c1Cl 30857,n1(CC)cc(CC(N2CCCCC2CCCNC(=O)CCS(C)=O)=O)c(C)n1 30858,C(c1ccncc1)=C(C(=O)NC(CCN(C(C(CC)F)=O)C)C)C 30859,c1(CNC(c2ccc(-c3ccc(SC(C)C)cc3)cn2)=O)c(O)ccc(F)c1F 30860,C1(=O)C(CO)N1.c1(C(N)=O)[nH]ccc1C(=O)N.C12(C(=O)NC)CC(CO)(C1)C2 30861,C1(NC(C)=O)CCN(C(=NCC2CCCN2Cc2cccs2)NC2CCC2)C1 30862,c1(C(C(C(=O)N(C)CCOc2ccc(C(F)(F)F)cc2)N)=O)ccc(F)cc1F 30863,C1(C(=O)N(CCN=[N+]=[N-])C)(NC(CC2(OC(C)C)CC2)=O)CC(CO)C1 30864,c1(OC)cc(C)c(Br)cc1C(N1CCC2(CC2C(=O)Nc2cc(O)ncn2)C1)=O 30865,N1(C(C2N(CC)CCC2)=O)CCN(C(=O)CSc2cccc(C)c2)C2(CCC2)C1 30866,CON(CCC(=O)NC1C2CCCCCC12)C(=O)C1CC(C#N)(OC)C1 30867,C12(NC(c3c(COC)scc3)=O)CCC1CN(C(C1CC3(CC3)CO1)=O)C2 30868,N1(C(C2C(CC)CCC2)=O)CCC(CO)(CNC(C2CCC(=O)N2)=O)CC1 30869,c1(-c2cncc(COCC)c2)ccn2nc(C(=O)Nc3nc(C#N)cs3)cc2c1 30870,C=C1CCN(C(=O)C(C)OCCC(C)C)C(C(=O)NCC(C2CC(C)(C)C2)O)C1 30871,Cc1nc2c(s1)CCCC2C(=O)NC1CCN(C(c2c[nH]c3cccnc23)=O)C1 30872,c1(C(=O)NCC(CC)NC(=O)CCC2CCN(C)CC2)oc(C)cc1C 30873,C1(C(N(C)Cc2cccnc2Br)=O)CC12CCOc1ccc(F)cc12 30874,N1(c2ccnc(N3CCC(Cc4ccn(C)n4)C3)n2)CCCC2(CCCCCC2)C1 30875,C(CCC1CCC1)(C(=O)NCc1cnn(C)c1O)NC(c1c(C)ocn1)=O 30876,c1(C(=O)NCC(C)CNC(=O)CC2CCCCC2)ccc2nnnn2c1 30877,c1(C(=O)NC2CC(N(C(CCC(=O)NC)=O)C)C2)cc(N)nc(Br)c1 30878,C(C(=O)N(CC)OC)NC(C(CNC(C1(CC#C)CC1)=O)C)=O 30879,N1(C(c2c(C)nsc2N)=O)CC(C2CN(C(=O)CCC3CCCOC3)C2)C1 30880,N1(C(C2CNC(=O)N2)=O)CCCC2(CCN(C(c3cocc3C(N)=O)=O)C2)C1 30881,C(=O)(C1CCc2c(Cl)cccc21)N(C)CCNC(C1(C(F)F)CC(F)(F)C1)=O 30882,C=C1CCN(C(C2CCC23CCC3)=O)C(C(=O)OC(C)(C)C)C1 30883,CCC(C)CCCCC(=O)NCC1CC(F)(F)CN1C(=O)CC1=CCN(C)CC1 30884,N1(C(c2ccn(CCC)n2)=O)CC2CCC(C1)N2C(c1cnc(C2CC2)s1)=O 30885,c1(C(=O)NC2CCC(CCNC(C(C(C)C)C)=O)C2)nn(C)c(Cl)c1Br 30886,N1(C(C(CC)OCC)=O)CC(OC)CC(NC(C2CC(C)CC2)=O)C1.OCC 30887,C(=O)(C(COC)COC)N1CC(N)(CS)C1.C(=O)(C(C)OCC(C)C)SCC 30888,C(=O)(C(CC(C)C)NC(N)=O)Nc1nc(-c2c(C)occ2)nn1-c1cccc(F)c1 30889,C1(CN(C(=O)CN(C)C(C2(C)COCCO2)=O)C)CCCCCC1 30890,c1(C(=O)NCC(C2CCCCC2)NC(C(C(C)C)F)=O)csc([N+](=O)[O-])c1 30891,C1(NC(C(c2cn(C(CC)CC)nn2)(C)C)=O)CCN(C(=O)C(F)CC)CC1 30892,C(C(=O)NCC)(C(C)(O)C(F)F)NC(CCC(=C)C)=O 30893,N(C(=NCCc1cnc(C)cn1)N1CCC(CS(C)(=O)=O)C1)CC(=C)C 30894,C1(NC(COCCN(C)C)=O)CN(C(C2CCCC23CC3)=O)CC12CCOCC2 30895,N1(C(c2cccc(O)c2OC)C(=O)NCC=C)CCOc2cccc(Br)c2C1 30896,C(=O)(C(C)(CC)CC)NC(CNC(Cc1c(SCC)cccc1)=O)CCOC 30897,c1(NC2CCC(C(=O)Nc3cnc(C)nc3Cl)CC2)nccc(S(C)(=O)=O)n1 30898,c1(N2CC(C)C(NC(c3cnsn3)=O)C2)ncc([N+](=O)[O-])cc1Cl 30899,c1(CN2CCN(Cc3n(C)cc(F)c3)CC2)cccc2c1SCCC2 30900,N1(C(=O)NCc2cc[nH]n2)CCCC1(C(C)C)CO.C1(CC)CCC1C(=O)NC 30901,c1(N(C(=O)CCc2nc[nH]n2)C)ccc(Br)cc1CC#N 30902,N1(C(C(CC)c2ccccc2)=O)CCN(C(c2n[nH]c(C)c2F)=O)C2(CCC2)C1 30903,N1(C(C2CCC(CC)CC2)=O)CCc2cc(NC(=O)OC)ccc2C1C 30904,CC1CCC(NC(c2c[nH]ccc2=N)=O)CN1C(c1csc(-c2cccs2)n1)=O 30905,C1(C(=O)NC(CNC(C(CC)(C)O)=O)(C)C)CCC(=O)N(CC(F)(F)F)C1 30906,CC1CN(Cc2cn(CC34COC(C3)C(O)C4)nn2)C(C)CC(C)O1 30907,c1(C(N2CCC(NC(Cc3c(C)con3)=O)(CO)C2)=O)c(C)cccc1[N+](=O)[O-] 30908,C(=O)(C1CCCc2nn[nH]c21)N1C(C)CC2CN(C(c3c(C)coc3C)=O)CC21 30909,N1(C(CCCC(C)=O)=O)CC2CCCN(C(C3OCCN(C)C3=O)=O)C2C1 30910,N1(C(c2c(OC)nsc2)=O)CC(CC(=O)NCC2CC2C(C)C)C2(CC2)C1 30911,c1(CC)cc(C(=O)NC2C=CC(Cn3cc(C4CCN(C)C4)nn3)C2)c(C)nn1 30912,C1(NC(C(F)=CCC)=O)CCN(C)C12CCCN(C(=O)CCC1CCCN1C)C2 30913,c1(C(=O)NC2CN(C(c3cc(OC)cc(F)c3)=O)CC2F)cc(Cl)c(F)cc1F 30914,n1(CC)cc(C(=O)NCC2CCC(NC(C3CNC(=O)N3)=O)C2)c2ccccc12 30915,N1(C(C(CC#C)C)=O)CCc2ccccc2C(NC(=O)C(C)(C)C(F)F)C1 30916,N1(C(c2c(SCC)nccc2)=O)CC2(CCN(C(C3CC(C)CO3)=O)CC2)C1 30917,c1(NC(CNC(c2c(C)cccn2)=O)C(C)C)ncc(C#N)cc1Br 30918,C(=O)(CCN(OC)C(=O)CSC1CC1)NC(C)CO 30919,c1(OC)cc(C(=O)NCC2CCCCN2C(c2nccn2C)=O)ccc1O 30920,C1(C)(CNC(C2(N(C(C(CN(C)C)O)=O)C)CC2)=O)CC2(CC2)C1 30921,C(CC(=O)NCC(C)(C1CC1)NC(=O)CN(C)C(=O)OC(C)(C)C)C1(C)CC1 30922,Cc1ccc(F)c(NC(=O)Cc2cccc(NC(c3cc(C)cc(Cl)c3)=O)c2)c1 30923,N1(C(CN(C)CC)=O)CCC2C(CCCN2C(c2cc3nc[nH]c3cn2)=O)C1 30924,N1(C(CC(C)(C)OC)=O)C2CCC1CN(C(c1cncc([N+](=O)[O-])c1)=O)C2 30925,c1(C(=O)NCCC(C)(C)NC(=O)Cc2nc([N+](=O)[O-])n[nH]2)c(F)ccc(F)c1N 30926,C1(CNC(c2c(C)n[nH]c2C)=O)CN(C(c2cc(CC3CC3)on2)=O)CCCO1 30927,C1(CNC(C=CCCC)=O)CCCC1NC(c1snnc1CC)=O 30928,N1(C(C(C)(C)C2CCC2)=O)CCC(NC(=O)CC=CC(=O)O)CC1 30929,CCC(CC(=O)NCCC(C)(C)NC(c1ccc(C(F)(F)F)[nH]1)=O)SC 30930,c1(C(N2CCCC(N(C(CCN(CC)CC)=O)CCF)C2)=O)ccc(O)cc1C 30931,c1(SC)cccc(C(=O)NC2CCCN(C(=O)C(C)(C)CC(F)F)C2)c1[N+](=O)[O-] 30932,N1(C(CCOCC)=O)CCC2(CC1)CC2(CO)NC(=O)CNC(c1cccs1)=O 30933,CC1(C)CC(CNC(c2cncc(Cl)n2)=O)N(C(=O)CCC2COC(C)(C)O2)C1 30934,c1(C(=O)NC(C2CCCCN2C(=O)Cc2conn2)C)nn(C)c2c1COCC2 30935,C(=O)(C(C)(F)C(=O)NC1CC(CNC(c2cc(Cl)cc(Cl)c2)=O)C1)OC 30936,N1(C(CNC=O)=O)CCN(C(C2CCCC23CCC3)=O)C2CCC12 30937,C(C1=CCN(C(=O)CC2CCC3CC3C2)CC1)NC(c1ccnn1C1CC1)=O 30938,C1(NC(c2ccsc2Cl)=O)CN(C(=O)C(F)=CC2CC2)CC12CCOCC2 30939,N1(C(c2c(OC)ccs2)=O)CCN(C(C23CCCC2C3(F)F)=O)C2(CC2)C1 30940,C1(CNC(C(N)=O)=O)CC(NC(=O)Cc2cccc(OCC(F)F)c2)C12CCC2 30941,c1(C(N2C3(CNC(CC(CC)O)=O)CC(C2)C3)=O)cc2cc(C)cc(C)c2[nH]1 30942,C(CS(=O)(=O)CC(=O)NC1CC1CNC(c1nc(C)c(C)nc1C)=O)OC 30943,c1(CC)cc(C(N2CCC(C(C)NC(=O)C(C(C)C)C3CCC3)CC2)=O)c(C)o1 30944,c1(C(=O)NC2C(NC(C(CC(C)C)NC(C)=O)=O)CC2)cc2ncccc2s1 30945,Cc1c(N)ccc(C(N2CCC(NC(=O)C3=CCC(C)CC3)C2(C)C)=O)c1Cl 30946,N1(C(c2cc(C)cc(F)c2)=O)CC(C)CN(C(C2COC3COCC23)=O)CC1C 30947,CC1CCCCCC1NC(C1(CCC(=O)O)CCCC1)=O 30948,N1(C(C(CC=CC)NC(=O)C=CC(C)(C)SC)=O)CCC2(C=CCO2)CC1 30949,C=C(Cl)C(C)(C)C(=O)N1CC(NC(c2cnccc2Cl)=O)C(SC)C1 30950,C12(CC(=O)NCCNC(c3c(CCC)onc3C)=O)CC3CC(CC(C3)C1)C2 30951,Cc1ccc(C(=O)NC(C)(C)CNC(=O)CC2CC(O)C2(C)C)c(F)c1Br 30952,CC1CC(NC(C2CN(Cc3nccs3)CCC2O)=O)C(=O)N1c1ccccc1 30953,C#Cc1cc(C(=O)NCC2CCC2NC(=O)Cc2sc(C)cc2C)cc(N)c1 30954,N1(C(c2cccc(OC)c2O)=O)CCC2CN(C(C3CCCC(C)C3)=O)CC2C1 30955,c1(SC)ncc(C(=O)NCCOC2CCN(C(C3C4COCC34)=O)C2)n1C 30956,c1(C(N(CC=CC(=O)N(C2(COC)CC2)C)C)=O)ccc([N+](=O)[O-])o1 30957,C(C)(C)(C(=O)NCCC(C)(C)NC(=O)C(C)Sc1nnnn1C1CC1)OC(C)=O 30958,c1(C(N2CC(C)C(NC(=O)C(c3ccc(F)c(F)c3)O)C2)=O)nc(Cl)ccc1N 30959,O=C(C1CCCc2nccn21)NC12CCOCC1CN(C(c1c[nH]nc1F)=O)C2 30960,c1(CC(=O)NC(C2CCN(C(C3CC3C#N)=O)CC2)C)c[nH]ccc1=O 30961,N1(C(C(CC=C)N(C)C)=O)CCC(C2CC2)C1CNC(=O)Cc1ccc(F)cc1 30962,c1(NC)c(C(=O)NC2CCC2CCNC(=O)C(C)C(C)(F)F)cccc1F 30963,c1(C(N2CC3(CCN(C(C4C(OC)C4)=O)C3)C2)=O)cc2n(n1)CC(C)NC2=O 30964,CC1CN(C(C2C3(CC3)C23CC3)=O)CC2(CCN(C(=O)CC3OCCO3)C2)O1 30965,N1(C(CSCC#C)=O)CCC2(CC1)CN(C(=O)Cc1nonc1C)C2 30966,C12(NC(N3CCCC(C(C)C)C3)=O)CCC(C(F)(F)F)(C1)OC2 30967,C12(NC(c3ncn(-c4cn(C)nc4)c3)=O)CCC(CC1NC(=O)COCCF)C2 30968,N1(C(C2CC(=O)NC2)=O)CCC2(C=C(C(=O)NOCCCCF)C2)C1 30969,CCCC(C)=CC(=O)NC(C(=O)NCC1(OCC)CCC1)c1cccs1 30970,c1(C(=O)Nc2ncc(F)cc2F)nc(=NCc2ccccc2)[nH]cc1Cl 30971,C1(NC(C2(Br)C(C)(C)C2)=O)CCCN(C(c2ccc(F)o2)=O)CC1 30972,c1(C(=O)NCCCC(CO)NC(CCc2cnc(C)s2)=O)cccc2nccn12 30973,Cc1cc(C(=O)NCC(C)NC(=O)COc2cccc(O)c2)ccc1F 30974,C(CCCCCCC)NC(C(=O)N(CC(C)O)CCNC(C(C=C)(C)O)=O)=O 30975,c1(CNC(C(c2cnccn2)C)=O)ocnc1-c1cn(Cc2nncs2)nn1 30976,C(=O)(C(=O)CCC(C)C)NC1CCN(C(C(=O)Nc2c(CC)cc(C)cc2)C)C1 30977,N1(C(c2cc(CC)on2)=O)CC(NC(c2coc(Cl)n2)=O)Cc2ccccc21 30978,N1(C(c2cnc(OCC)s2)=O)CC(C)CN(C(c2oc(C)nc2C)=O)C(C)C1 30979,c1(CCNC(=O)C(=O)NCC2(F)CC3(CNC3)C2)ccc(Br)cc1Cl 30980,N1(C(CC(C)SC)=O)CCCCC1C(=O)NCCCC1(C)CC1 30981,CC1(C)CC(NC(=O)COCCF)CN1C(=O)Cc1nc[nH]n1 30982,C(c1cc(C(F)(F)F)ccc1Cl)=CC(=O)NCC1CN(C(=O)CO)CCCO1 30983,C#Cc1cn(C)nc1C(=O)NC1(CNC(=O)CC(C)C(C)C)CCOC1 30984,CC12CCN(c3ccncc3C#N)CC1C2(Cl)Cl 30985,C1(NC(C(C2CCN(C(CC3CC(=C)C3)=O)C2)F)=O)CCCCC1(C)O 30986,n1(CC)nc(C(=O)NC(C)CC(C)NC(=O)C(=O)Cc2ccc(F)cc2)c(C)n1 30987,C1(C(=O)NC2CC(C)(CNC(Cc3c(C)ocn3)=O)C2)CC(=O)NC(C)C1 30988,Cc1cc2[nH]c(=O)c(C(=O)NCCC3CN(C(C4(Cl)CC4)=O)CC3C)cn2n1 30989,Cn1c(N(CCN)CC2CCCCO2)nnc1-c1ccccc1F 30990,N1(C(c2cccc(CCC)c2)=O)CCCC(F)(C(=O)NCc2cnsc2)C1 30991,O(NC(=O)C(F)(CNC(=O)CCC(F)(F)F)C(C)C)CC#C 30992,C(C(=O)N=c1cc(C)o[nH]1)SCC(=O)NCCCC(CO)NC(CCCC=C)=O 30993,N1(C(C(C)OCCC(C)C)=O)CC(NC(c2cncc(Br)c2)=O)C(C)C1 30994,CCCC(C(O)c1ccccc1)NC(c1sccc1Cl)COC 30995,C(C(CNC(c1ccc[n+]([O-])c1)=O)C(F)(F)F)NC(c1c(CCC)nsc1N)=O 30996,C1(C)(C(N2CCN(CCCNC(c3c(C)ncnc3)=O)CC2)=O)CCCCC1C 30997,c1(CNC(c2c(C)cco2)=O)ncccc1CNC(=O)CN1CCC(C)C1 30998,Cc1ccc(S(=O)(=O)NC2CN(C(c3cccc(C)c3Cl)=O)CC2F)c(F)c1 30999,c1(C2C(NC(=O)NCCc3cc(OC)ncc3)C2)cc(C)cc(Br)c1 31000,CCCC(C)CCCC(=O)NC(CNC(c1ncc(OC)cn1)=O)C(C)(C)C 31001,S(=O)(=O)(CCC(=O)NC1CCC(CNC(=O)COC2CCCOC2)C1)N(C)C 31002,C1(C)(CC)CC(CC(=O)Nc2cnc(C(C)NC(=O)OC(C)(C)C)s2)CC1 31003,N1(C(c2c(OC)nn(C)c2)=O)CCCC(NC(c2ccc(O)nn2)=O)CC1 31004,N1(C(c2c(C)nn(C)c2Cl)=O)CC2(CCN(C(=O)CCc3cncc(O)c3)C2)C1 31005,C1(CSC)COCCN1C(=O)C(n1cc(COC(=N)O)nn1)C 31006,c1(C(N(C2CCCN(C(=O)C(C)=C3CC3)CC2)CC)=O)ncc(OC)cc1F 31007,O=C(N=c1c(Cl)c[nH]cc1I)C1CC12CCN(C(c1ccccc1Br)=O)CC2 31008,N1(c2cc(C)nc(Cl)n2)CCCC(C2CCN(C(=O)C(C)(C)S(C)(=O)=O)CC2)C1 31009,CC(CC(=O)N1CCN(C(=O)CCc2ccc[nH]2)C(CCO)C1)C(F)(F)F 31010,c1(C(N2CCOC(CCOC)C2)C(=O)NCCC(=O)OCC)cc(C)nc(C)n1 31011,CC1C(NC(c2cc(F)ccc2F)=O)CCCN1C(=O)CCCn1cccc1 31012,N1(C(c2ncn(C)n2)=O)CCCN(C(c2cccc(=O)n2C)=O)C(CO)C1 31013,c1(C(N2C(CN(C(CSCCC(C)C)=O)C)CCC2)=O)ccccc1CC(C)C 31014,C(=O)(CCCC(=O)N1CCC(CNC(c2ncoc2C)=O)C1)OCC 31015,N1(C(C(CC)CC)=O)CCCC(NC(C23CCN(CC2)CC3)=O)CC1 31016,c1(C(N(CC(CC)NC(c2cc(N)ccc2O)=O)CC)=O)cnn2cnnc2c1 31017,N1(C(C2CC(C(F)F)(OC)C2)=O)CC(OC)CC(NC(=O)CN(C2CC2)CC)C1 31018,C12(N)CCC(n3ccnn3)(CC1)C2.Cc1nnn(CC(N2CC(SC(F)F)C2)=O)n1 31019,c1(OC)c(C(N2CC(CO)(NC(c3ccc(=O)oc3)=O)C2)=O)cnn1C 31020,Cc1c(C(=O)NC2(CNC(C3CC4(C3)CC4(F)F)=O)CCCCC2)cncc1F 31021,n1(CC(=O)NC)ccc2ccc(NC(=O)C(N3CCC(CO)(CO)C3)=O)cc12 31022,n1(CCNC(=O)CNC(C2CCCC2)=O)cc(-c2nccs2)nn1 31023,CN1CCN2CCN(C(C3CCCN(C4CCC(C)(C)C4)C3)=O)CC2C1 31024,N1(C(CCC2C(C)C2)=O)CCCC1CCc1cccs1 31025,C(CN=c1ccc(S(=O)(=O)NC(c2nnc(C)s2)C)c[nH]1)SC 31026,CC1(C)CCN(C(C2CC2(C)C)=O)C(C(=O)Nc2ccc(F)c(O)c2)C1 31027,c1(CC(=O)NC(CN(C(CC2C(CC)C2)=O)CC)C)ccc(OC)c([N+](=O)[O-])c1 31028,C1(NC(C2CC(N(C(CCN(C)CC)=O)C)C2)=O)CCSCC1 31029,c1(C(C(=O)NC(CC)C)N(C2CC2)C(c2ccccc2)c2ccco2)ncc(C)s1 31030,CC(CCCNC(C1(C2CCCO2)CCCC1)=O)NC(c1ccon1)=O 31031,CC1CN(C(c2sccc2F)=O)CC(C)CN1C(c1cnn(C)c1C(F)(F)F)=O 31032,C1(NC(C(C)NC(CC)=O)=O)CC(OC)C(OC)C1.C12(CC1)CCCN2 31033,N1(C(c2c(C#C)c[nH]n2)=O)CCCC(COC)(NC(C2CCCN2C2CC2)=O)C1 31034,C(=O)(C(O)CC(N)=O)NC(C(N1CCCC(CCC#C)C1)=O)(C)CO 31035,C1(NC(CCNC(CC(C)C)=O)=O)CCC(C)N(C(=O)C=C2CCOCC2)C1 31036,C1(CNC(c2n(C(C)(C)C)ncc2)=O)CCCC(NC(C2C3CCCC23)=O)C1 31037,C1(CNC(C(COC)O)=O)CCN(C(C2CC(c3cccc(F)c3)C2)=O)C1(C)C 31038,N1(C(C2CCN(C(c3c(OC)ccs3)=O)C2)=O)CCc2c(O)noc2C1 31039,c1(C(=O)NC(C(=O)NC(CN(C(CCOC(C)C)=O)C)C)C)ccccc1Cl 31040,C(=O)(C1CCc2c(Cl)cccc21)NCC1CCC(C)(C)CN1C(C1(CO)CC1)=O 31041,CC1=NOC(=O)C1CC(N1CCOC(CN(C)C(C2CN(C)CCO2)=O)C1)=O 31042,c1(C(=O)OC)ccc(CNC(=O)C(N2CCN(c3ncc(C)s3)CC2)=O)cc1C 31043,Cc1ccc2c(C(=O)NCCC3(NC(=O)CC(C)(O)C(F)(F)F)CC3)onc2c1 31044,N1(C(=O)CCc2ccon2)CCC2CN(C(=O)CCc3ccc(CO)cc3)C2C1 31045,C(C)(C(=O)NCC(C)N(C(=O)CNS(=O)(=O)N(C)C)C)(C(C)C)OC 31046,N1(C(CNC(C)=O)=O)CCC(C)(NCc2cccc(OC(C)C)c2)C1 31047,c1(CC(=O)N(C)CC2CCCN(C(=O)CS(C)(=O)=O)C2)cnc2cccnn12 31048,C#CCC(C)(C(=O)NC1CN(C)NC1=O)NC(C1CCCCN1C)=O 31049,C1(C)(C(=O)NC(CNC(Cc2nc(C(C)C)sc2)=O)C)COC(=O)C1 31050,Cc1ccc(N)c(C(N2CCCC2C(C)NC(=O)CCCC2CCCC2)=O)c1 31051,C1(CCC(=O)NC)CN(C(=O)N(C)CCOCCOC)CCC1C 31052,n1(CC)ncc(C(=O)NC2CC(OCC(=O)NC3(C)CCSC3)C2)c1C 31053,c1(C(=O)NCc2scc(CNC(c3cc(C)ns3)=O)n2)cc(O)nc(C2CC2)n1 31054,CC(C)C(O)C(C)C(=O)NCC1(F)CN(C(c2ncn3c2CCC3)=O)C1 31055,c1(C(N(CC(C)NC(C(C2CC(F)(F)C2)OC)=O)C)=O)coc(C#N)c1 31056,c1(CC(=O)NCC(C)CN(C)C(C2CC2c2ccccc2)=O)c[nH]c(=N)nc1O 31057,c12ccccc1C(=O)OCC2=O.C1(OCC)(OC)CC1C(=O)OC 31058,c1(CCC(=O)NC(CN(C)C(c2ccc(Cl)s2)=O)(C)C)ncc(F)cn1 31059,c1(OC)ccc(C(N2CCCC(N(C(=O)C=CC(F)(F)F)C)CC2)=O)c(N)c1F 31060,N1(C(Cc2ccc(OC)cc2F)=O)CCN(C(C2(C)CCOC2)=O)CC2(CC2)C1 31061,c1(C(N2CCN(C(c3cnn(CC)n3)=O)CC2C(F)F)=O)cc(C)[nH]c(=NC)n1 31062,c1(C(=O)NCC2(C)CC(NC(c3ccn(COC)n3)=O)C2)ccc(C)c(F)c1 31063,C(=O)(C1CCc2nccn21)N1C(C)(C)CC(NC(C2(CC3CC3)CC2)=O)C1 31064,c1(NCC2CCN(C(=O)CSc3ccc(F)cc3)C2)ccc2c(c1)CCN2 31065,CC1=C(C(=O)N2CCCC2CCNC(c2ccc(F)c(F)c2F)=O)CCS1(=O)=O 31066,CC(CNC(C1CC1(C)C(F)F)=O)C(F)C(=O)NCC1CSC1 31067,C#Cc1ccc(C(=O)NC2(C(N3CCC(CO)C3(C)C)=O)CC(O)C2)nc1 31068,N1(C(c2c(C)cnn2C)=O)CC(CNC(C2Cc3nncn3C2)=O)C2(CCC2)C1 31069,C(=O)(C(F)CC(C)(C)N(C)C1CC1)N1C(CC)(CC)COCC1 31070,C1(C)(C(NOC2CCCN(CC)C2)=O)CC(O)CN1C(=O)CCc1cscn1 31071,C1(CNC(C2C(CCC)C2)=O)(CO)CC12CCN(C(c1cnnn1C)=O)CC2 31072,CC1(C)CC(C(N2CCOC(C#N)C2)=O)CN1C(C1CC2CC(=O)C1C2)=O 31073,c1(CNC(c2cc(F)ncc2NC(=O)C(Cl)(Cl)Cl)=O)ccc(F)c(C2CC2)c1 31074,[N-]=[N+]=NC1CN(C(c2ccc3cc[nH]c3c2)=O)CC1NC(C1CC2CCC2C1)=O 31075,C1(C)(C(N2CC(N(C(c3c(SC)cn(C)n3)=O)C)C2)=O)CCCS1(=O)=O 31076,N1(C(Cc2nnc(C)o2)=O)CCC(C2CC2)(NC(c2ccc(C)c(F)c2F)=O)C1 31077,N1(CCC2CN(C(C=C(CC)C)=O)C2)CCN(C(C23CCCCC2C3)=O)CC1 31078,C(=O)(CCC(C)(C)F)N1CCCC(CN(C(c2nncn2C2CC2)=O)CC)C1 31079,C(CN=c1[nH]c(=NCCc2cccn2C)[nH]c2cc(C)ccc12)NC(C)=O 31080,C=CC(CC)CC(=O)NCC1CN(C(C2CC3(CCC3)CO2)=O)CCN1C 31081,c1(C(N2CCC(C(C)NC(C3(F)CCC3)=O)C2)=O)ccnc(NC2CCC2)c1 31082,C(C1(C)OCCc2ccccc21)NC(=NCC)NCCc1ccc2c(c1)OCO2 31083,C1(C)(CNC(CSCC#C)=O)CN(C(c2cccc(O)c2C)=O)C(C)(C)C1 31084,C1(NC(CC=CCC)=O)CCN(C(c2cncc(S(C)(=O)=O)c2)=O)CC12CCC2 31085,N1(C(C(C)c2cccs2)=O)CCCC(CCNC(=O)COc2ccccc2)C1 31086,N1(C(Cc2n(C)cnn2)=O)CC2CC(NC(c3cncnc3)=O)CC1C2 31087,N1(C(C2C(C)(Br)C2)=O)CCC2(CCN(C(c3cn(CC4CC4)nn3)=O)C2)C1 31088,Cc1nc(C(=O)NC2C3CN(C(=O)C=CC4CCC4)CC23)c(=O)[nH]c1C 31089,c1(C(=O)NC2CCCN(C(C(=Cc3ccco3)C)=O)C2)c(N)cc(F)cc1Cl 31090,C1(C(=O)OC)CCCC1C(=O)NCCNC(C1CC(Cl)(Cl)C1)=O 31091,C(=O)(CS(=O)(=O)CC(C)C)N1C2CC(CC(NC(CC3C(C)=NOC3=O)=O)C2)C1 31092,c1(C(=O)NC(CC)(C)CNC(C2(C)CCOCC2)=O)nc2ccccc2cc1C 31093,C1(C(N2C(CN(C(c3occc3C)=O)CC)CCC2)=O)Cc2ccccc2S1 31094,C1(C(=O)Nc2cc(Cl)ccc2Br)COC2(CCN(Cc3ccc(Br)cn3)CC2)C1 31095,c1(C(=O)NC2(COC)CN(C(C3CCC(CN(C)C)O3)=O)C2)c(Cl)nn(C)c1Cl 31096,C1(NC(c2cc(OC)n[nH]2)=O)CC2CCC(C1)N2C(C1CCCC1C(C)C)=O 31097,N1(C(c2nc(OCC)oc2)=O)CC2(NC(=O)C(C)OC)CCCC2(F)C1 31098,C1(NC(C(C)(C)C2CCCO2)=O)CN(C(C2CCC3(C2)N=N3)=O)CCC12CCC2 31099,CCCCCC(O)CC(=O)N1CCC(NC(c2c(Cl)ccc(F)c2F)=O)C(F)C1 31100,c1(C(C(=O)NCC2(C(=O)NC(c3cccs3)C)CC2)C)ccccc1 31101,C(C(F)(F)CCC(=O)NNC(=O)c1cnccn1)n1cc(CCOC)nn1 31102,c1(CC(N2CC(C(C)NC(CCOCC(C)C)=O)C2)=O)nc(OC(C)(C)C)n[nH]1 31103,C12(CNC(C(C)(C)C)=O)CCCCC1CN(C(c1ccc(O)nc1Cl)=O)C2 31104,N1(C(CC=C)=O)CCCCC1CN(C)C(C1(n2cccn2)CCOCC1)=O 31105,C1(CNC(c2n[nH]c(C)c2C)=O)CN(C(C2CS(=O)(=O)C2)=O)CC1(F)CO 31106,C1(F)(C(N(CCCNC(c2ccc(COC)s2)=O)C2CC2)=O)C2CCCCC12 31107,c12ccc(cn1)c(=O)n2C1CNC(=O)CO1.Cn1nccc1COc1ccccc1 31108,C1(C(N(CC(CNC(CCCOC)=O)C)C)=O)CC(C(=O)OC(C)(C)C)=NO1 31109,N1(C(CN(CCC#C)C)=O)CCC2(COC(CNC(=O)CC3OCCCO3)C2)C1 31110,c1(CC(N2C(C(=O)OCC)C3C=CC2C3)C(=O)NC)cc2ccccc2o1 31111,N1(C(CC2N(C)CCOC2)=O)CC2(CC(NC(C3CC(F)(F)C3)=O)C2)C1 31112,N1(C(C(C)(C)CF)=O)CCC2(CC1)CCN(C(=O)CC1(c3ccon3)CCC1)C2 31113,n1(CCC)cc(C(=O)NC2CCCC2(C)CN(C)C(c2csc(O)n2)=O)c(C)n1 31114,O=C(COCc1ccccc1)N1CCC(S(=O)(=O)Nc2ccccc2)C1 31115,C(=O)(C(C)(C)CC(F)(F)Br)NC1CC(n2cc(C(N3CCCC3)C)nn2)C1 31116,C1(C(=O)NC(CNC(c2c(C)ncn2C)=O)C(C)C)CCCCN(C)C1=O 31117,N1(C(c2cc(C#N)sc2)=O)CCC(C2CCN(C(=O)CCCCCF)CC2)C1 31118,C(=O)(CC(C)CC(=O)NC(CNC(=O)CCn1cc(C)cn1)CO)OC 31119,N1(C(CONC(C2CC(=C)C2)=O)=O)CC(CO)CCC1C 31120,C1(NC2COC2)CCN(C(=O)CNC(CNC(N)=O)=O)C1 31121,C(CN=c1[nH]c(Cl)nc2ccccc12)NC(C(C(C)C)NC(C)=O)=O 31122,C(C(C(C)(C)C)NC(C1(C)COC(=O)N1)=O)NC(C(c1cn(C)nc1)=O)=O 31123,c1(C(N(C)CC2CCC(NC(CC3C(OC)CC3)=O)CC2)=O)cc([N+](=O)[O-])c[nH]1 31124,C1(CCC)(NC(=O)C(COC)N(C)C)CCCN(C(=O)C(c2ccc(Cl)s2)=O)C1 31125,c1(C(C)C)cncc(C(=O)NCC2CC(NC(=O)CCc3cccn3C)C2)c1 31126,c1(C(N(CC(CC)NC(c2cccnc2)=O)C)=O)c(C)oc(C)c1C 31127,N1(C(C2(c3cccnc3)CCC2)=O)CCC2(CCCN2C(=O)CN(CCO)CCO)C1 31128,c1(C(N(CC(C)O)CCNC(C2(C)CC=CC2)=O)=O)ccc(-c2cnn[nH]2)cc1 31129,C1(C(=O)NCCS(=O)(=O)NC)CC2CC1CN(C(=O)CCc1cscn1)C2 31130,C(=O)(C(F)(F)C(F)(F)C(F)(F)C(F)F)NC1C(C)(C)C(C(=O)O)C1 31131,c1(C(C(=O)NCC2CC(NC(c3cnc(Cl)s3)=O)C2)(F)F)ccc(F)cc1F 31132,N1(C(Cc2c(C)ncs2)=O)CC2CC1C2NC(C1CC(n2cccn2)C1)=O 31133,C1(NC(c2ccc(C)[nH]2)=O)CCN(C(=O)CCC=Cc2ccccc2)CC1C 31134,N1(C(CNC(CC)=O)=O)CC2CCC(C1)CC(NC(C13CCC(OC)C1C3)=O)C2 31135,c1(C(N(CC(CC)NC(=O)Cc2ccns2)C)=O)c(NC(N)=O)cccc1F 31136,CC(CNC(=O)COC(F)(F)F)CNC(=O)C(F)C1CCCC1 31137,C1(NC(C(C)C2CC2)=O)CN(C(c2n[nH]cc2Br)=O)CC1C(F)F 31138,N1(C(C2C(c3ccc(-c4cc(SC)n[nH]4)nc3)C2)=O)CC(CO)CC1(C)C 31139,c1(C(N2C(CNC(C3CCCCCC3)=O)C3CCC2C3)=O)ccc2n[nH]cc2n1 31140,c1(C(=O)NC(CN(C(C2(COC)CC=CCC2)=O)C)C)ccc2ccccc2c1 31141,C1(NC(CCSCC)=O)CC2CCC1N(C(c1cc(C(N)=O)cs1)=O)C2 31142,O=C(C#CC1CCCCO1)NCC1(NC(C2CCC(=O)NC2)=O)CCCCC1 31143,C1(CNC(C(C)=C(CC)C)=O)CCC(C(=O)NC(c2noc(CC)n2)C)C1 31144,Cc1nc(Cl)nc(N2CC3CN(C(C4CCS(=O)(=O)C4)=O)CC3C2)c1C#N 31145,C(C(C(=O)NCCC1(O)CCN(C(=O)C=CCO)C1)C(C)(C)C)OCC=C 31146,C1(NC(CCOCCOC)=O)CN(C(c2ccsc2)=O)CC1C 31147,CC(C)CC(C)(C)C(=O)NCC1CC(C)CN(C(=O)C(Cl)=CCl)C1 31148,C1(C(N(C)Cc2nnnn2C)=O)CC(=O)CN1C(=O)CSC1CC1 31149,C1(C(N2CC(CNC(Cc3c(OC)nccc3)=O)C2)=O)CCc2ncncc2C1 31150,C1(C2CC2)(CNC(C(CC)C(C)O)=O)CCN(C(c2nncs2)=O)C1 31151,N1(C(c2cc(OC)c(O)nc2)=O)CC2(CCN(C(c3nc(C)n(C)n3)=O)C2)C1 31152,CCCCCC(O)CC(=O)NC12CC1CN(C(=O)CC(N1CCCCC1=O)C)C2 31153,c1(CC(C)C)nccc(C(=O)NC(C)CC2CN(C(c3ccccc3F)=O)C2)n1 31154,N1(C(c2sc(C)c(Br)c2)=O)CCC2(CCOC2=O)CC1 31155,C1(C(C)NC(=O)C(CN(C)C)N(C)C)CCCCN1C(c1ccc(C(F)F)s1)=O 31156,C1(C(N2CC(C)(C)C2c2cccnc2)=O)(COC)CCCNC1 31157,C1(C(=O)NCCC(CNC(=O)CNC(=O)C2CC2)O)CC(c2ccccn2)=NO1 31158,C(N=c1[nH]c(=NC(C)CCc2ccccc2)[nH]c2c1CCC2)C1(CC)CC1 31159,C(CCCCC(=O)NCCC(O)C1CCCC1)N(C(C=CC(=O)OCC)=O)C 31160,CCCC(CNC(C1CCC(=O)N1C)=O)CCO 31161,c1(CC)c(C(=O)NC(C)CNC(c2cccc(-n3ccnc3O)c2)=O)nnn1C 31162,C(=O)(C(O)CC(F)(F)F)N(CCNC(c1c(Cl)n[nH]c1C1CC1)=O)CC 31163,c1(-c2scc(C(N(CCCNC(C(CC)SC)=O)CC)=O)n2)cccc(C#N)c1 31164,c1(CC)cnc(O)c(C(=O)NCC(C)(C)NC(c2cc(C3CC3)ccc2Cl)=O)c1 31165,C(CO)(CCC(C)C)NC(CSCCNC(Cc1scc(C)c1)=O)=O 31166,c1(C(=O)NC2(C#N)CC2)ccc2c(c1)CCN(C(c1ccc3ncnn3c1)=O)C2 31167,c1(CC)ccc(C(C)C(=O)N2CC(CCNC(c3cccnc3O)=O)C2)cc1 31168,C1(O)(C(C)NC(CC)=O)CCN(C(c2cccc(-n3cncn3)n2)=O)CC1 31169,C1(NC(CCCC#C)=O)CCCC12CCN(C(c1cc(N)nc(Br)c1)=O)C2 31170,c1(C(N2CC(OC)(CNC(=O)C(C#N)C(C)C)C2)=O)cc(S(C)(=O)=O)co1 31171,N1(C(COCCCOC)=O)CCCN(C(=O)CN2CCC(C)CC2)CC1C(C)C 31172,CC1(C)C(CC(=O)NC(C2CCCCC2)C(=O)NCc2ccc(O)cc2)C1(C)C 31173,CC1CC(NC(c2nncs2)=O)CCN1C(=O)CCN1CCOCC1 31174,N1(c2nnc(COC)s2)CCC2(CCC2)C(NC(=O)C2Cc3ccccc32)C1 31175,CC(C)C(C)C(CNC(C1(Br)CC1)=O)NC(C1(C(F)(F)F)CC1)=O 31176,C(=O)(C(=O)C(F)(F)F)N(CC(C)NC(C1(C)CCCO1)=O)C 31177,N1(C(CCC(=O)NCC)=O)CCCCC(C2CN(C(c3coc(Br)n3)=O)C2)C1 31178,N1(C(Cc2c(C)non2)=O)CCC(C2CCCCN2C(=O)CSCC(=O)O)CC1 31179,Cc1cc(Br)cc(C)c1OCC(=O)NC1CC1NC(=O)C1=CCOCC1 31180,Cc1cc(CN2CCOC(C(N3CCC(CO)C(O)C3)=O)C2)c(C)cc1Br 31181,N1(C(c2cccn(C)c2=O)=O)CCCC(NC(=O)CCc2cnn[nH]2)C(F)C1 31182,N1(C(CC=C)=O)CCOCC12COCCN(C(=O)CCCCC(C)CC)C2 31183,c1(C(N2CC(C)(c3cn(-c4ccc(Cl)nc4)nn3)C2)=O)nccc2cccnc12 31184,C(=O)(CCCCCNC(=O)CC1CC1(C)C)NC(c1nccs1)(C)C 31185,c1(COC)ncc(NC(C23CC(CN2C(=O)CC(=O)OC)C3)=O)cn1 31186,c1(C(N(C)CCOCCNC(C2CCS(=O)(=O)N2)=O)=O)cc(Cl)n[nH]c1=N 31187,c1(C(N2C(CC(N3CC(=C)C3)=O)COCC2)=O)cccc(C)c1C#N 31188,C(=O)(C1=C(C)CCOC1)NCCN(CC(C)O)C(c1cnc(CC)[nH]1)=O 31189,C1(C(=O)N(C2CN(C(=O)C(=CC3CCCC3)C)C2)C)(OC)CCCOC1 31190,CS(=O)(=O)c1cc(NC2CC(F)(CNC(C3CC4C=CCC(C3)C4)=O)C2)ncn1 31191,C(=O)(C1=CCC(F)(F)CC1)NCC1(C)CCC(NC(CC(CC)C)=O)CC1 31192,N1(C(c2c(C)scn2)=O)CC2C3CCC(C2C1)N(C(c1cccnc1O)=O)C3 31193,C(CCCC(=O)N1CC(OCC(=O)N(CCCC(O)CO)C)C1)N(C)C 31194,N1(C(c2ccn(CCCC)n2)=O)CCC2CN(C(C3(n4cnnn4)CC3)=O)CC12 31195,c1(C(N(C(C)CCNC(C2(O)CCOC2)=O)C)=O)cccc(Cn2cccn2)c1 31196,c1(CC)cc(C(N2CCC2C(=O)N(C)C)=O)ns1 31197,c1(C(=O)NCC2COCCN(C(C3(C#N)CC3)=O)C2)cc2c(Cl)cncc2o1 31198,c1(OC)cc(N)c(F)cc1C(=O)NCc1cc(O)nc(CNC(=O)C(C)OC)n1 31199,C#Cc1ccc(C(N2CCC(O)(C(C)CNC(c3ccc(Cl)s3)=O)C2)=O)cc1F 31200,C1(S(=O)(=O)NC2CC2)(CNC(C2(c3cccnn3)CC2)=O)CCC1 31201,C1(C(N2CC(C(C(=O)NCC3(c4ccno4)CCC3)O)C2)=O)COCCC1(F)F 31202,c1(C(=O)NC2CCN(C(C3N(C(C)C)CCC3)=O)C(C)C2)nnc2n1CCCC2 31203,C12(NC(C3CCC4(CCC4)O3)=O)CCCC1N(C(c1cnccc1Cl)=O)CCC2 31204,N1(c2cc(NCC3OCC(C)C3)ncn2)C2CCC1CN(C)C2 31205,CC1CC(C(=O)NCC2(C(=O)NCC(F)Cl)CC2)=NO1 31206,C1(NC(C2(C)COC(=O)N2)=O)CC2(NC(=O)C(=C3CCCCC3)F)COC1C2 31207,C(C)(CCCCO)NC(C(CNC(C(CC1CC1)OC)=O)OC)=O 31208,c1(OC)ccccc1CN1CCC(CNC(c2cc(C#N)cs2)=O)C1 31209,c1(C(CC(=O)N(C2CN(C(Cn3nc(C)c(Cl)c3)=O)C2)C)C)ccc(F)c(F)c1 31210,c1(C(N(c2cc(I)ccn2)C)=O)cccc(Oc2ccccc2)c1 31211,C1(NC(C2(CC)CC2)=O)CC=CCC1C(=O)N(CC(F)(F)Cl)C 31212,C1(NC(c2cc(Br)cs2)=O)CCCN(Cc2ccc(I)c(O)c2)CC1 31213,c1(CC(=O)NCC(C2CCCCC2)NC(C2N(C)CC(O)C2)=O)ccc(F)c(Cl)c1 31214,N1(C(c2ncn(CC)c2)=O)CCC(C)C1CNC(=O)C=Cc1ncco1 31215,c1(C(=O)NC(CC(C)NC(c2cccc(C(C)=O)c2)=O)C)cc(C)c(C)nn1 31216,C1(NC(C2CCC3(CN(S(=O)(=O)CCCl)C3)O2)=O)CCc2ccccc2O1 31217,c1(N(C(C(C)CCCc2ccccc2)=O)C2CCCC2)cccc(S(C)(=O)=O)c1 31218,CC(F)(C(=O)N1C2CCC1CN(C(c1ccc3cnnn3c1)=O)C2)C(F)(F)F 31219,c1(C(N2CCC(C)C(NC(=O)CCF)C2)=O)c(Cl)oc2ccccc12 31220,N1(C(CCN2C(=O)C=CC2)=O)CCCCCC1.C(C)(CCC=C(C)C)SC 31221,C1(NC(c2c(C)cc(F)nc2)=O)CCC2CC1CN2c1nc(Cl)ncc1Cl 31222,C(=O)(C(CO)N(C)C)N(CC(=O)NC1(CC(=O)OCC)CC1)C(C)C 31223,C(CCCC(CO)NC(=O)COC(F)F)NC(Cc1cccc(OC)c1)=O 31224,C1(COC(C2C(C)C(=O)C2)=O)(CF)CCOCC1 31225,C1(c2n(CCC)nnn2)(Nc2cccc([N+](=O)[O-])c2C)CC2(COC(C)C2)C1 31226,c1(CC(N2CCC(CCOC)(NC(=O)CC3CC3)C2)=O)ccc(Cl)c(C)c1F 31227,C1(C(=O)NC2(CC)CCCN(C(=O)C(C)=C3CCC3)C2)CC(C(C)=NO)C1(C)C 31228,N1(C(C)=O)CC2CCC(NC(c3ccnc(C(N)=O)c3)=O)(C2)C1 31229,c1(C(N2CC(CNC(CC3CCN(C)C3=O)=O)C2)=O)ccnc2ncnn12 31230,c1(C(=O)NCCN(C(CC(C)O)=O)CC(C)O)cnc2c(c1)NCC2 31231,c1(CC)nc(C)c(C(=O)NC(C)CNC(c2nnsc2SC)=O)o1 31232,c1(C(N2CC(CNC(=O)C(n3cc(Br)cn3)O)C2)=O)c(F)ccc(F)c1F 31233,C1(OC)CC2(C1)CC(NC(C1(C)CCN(C(C3CCC(=O)C(C)C3)=O)C1)=O)C2 31234,N1(C(C(CC=C)C(C)(C)C)=O)CCC2C(CCCN2C(c2cn[nH]c2)=O)C1 31235,c1(C(N2CC3(C(=O)NC4CCCC4(F)F)CC2CO3)=O)ccc2[nH]ccc2n1 31236,C12(C(N3CCCC(N(C(=O)C4=CSCS4)C)C3)=O)CC3CC(C(=O)N1)C2C3 31237,c1(C(N2CCN(c3nc[nH]n3)CC2)C(=O)NCC=C)cnc2c(c1)COC2 31238,c1(C(N2CCCC(C(=O)Nc3ccc(Cl)cc3CO)C2)=O)cc2ccoc2cn1 31239,c1(OC)cnc(C(=O)NCC2(CNC(=O)Cc3ccon3)CC23CCC3)c(Cl)c1 31240,CCC(COC)C(=O)N(CCNC(=O)C(c1ccc(Cl)cc1)C)C1CC1 31241,c1(SC)cc(C)c(C(=O)NC23CC(C2)N(C(=O)COC2CCCCC2)C3)o1 31242,C1(C(=O)NC(C2CCC(C(=O)NCC(F)(F)C(N)=O)O2)C)CC(O)C(F)C1 31243,C=CC1(c2ccccc2)COCCN1C(=O)C=CC(=O)Nc1ccc(Br)o1 31244,N1(C(c2ccc(OCOC)cc2)=O)CC(NC(=O)CC2C(C)C2(F)F)CC(F)C1 31245,C1(C)(CNC(C2C(C)(C)C2)=O)CCN(C(c2cnn(C3CC3(F)F)c2)=O)C1 31246,c1(C(=O)NC2CCC(C)(NC(COC)=O)CC2)ccc2ncccc2c1F 31247,C1(C(=O)NC2CCCC2CF)COC2(C1)CN(C(=O)Cn1ncnn1)C2 31248,CCCC(=O)N(CCN(C(=O)Cn1cccc1)CC)CC 31249,C1(C(=O)NCC(C)(O)CN(C)C)(CC)CCNC1 31250,Cc1cc(NC(C2CCN2C(=O)Cc2ccc(Cl)s2)=O)cc(Br)c1 31251,Cc1ccc(F)c(C(N2CC3CCN(C(=O)Cc4c(C)noc4C)C3C2)=O)c1Cl 31252,c1(C(CC)C)nc(C)cc(=NC(C)CC(C)NC(=O)C(C)(C(C)C)OC)[nH]1 31253,N1(C(CCC(=C)Cl)=O)CCN(C(=O)CC2CCC(F)(F)CC2)CC(O)C1 31254,N1(C(Cc2c(C)cccc2C)=O)CCN(C(c2cncnc2C)=O)CC(CO)C1 31255,c1(C(=O)NCC2CC(NC(COCC)=O)C2)ccccc1SC(C)C 31256,CCCCCCCC(F)C(=O)N1CCOCC12CCCC2 31257,C(=O)(CCN=C(NCC(C1CCCCO1)(C)C)NC1CC=CC1)N(C)C 31258,CC1(C)CN(C(=O)Nc2cc(OCc3ccccc3)ccc2Cl)CCC1CO 31259,Cc1scc(C(=O)NCC(C)(O)CNC(c2cccn2C2CCCC2)=O)c1N 31260,C(=O)(C(CC(C)C)N(C)C(C)=O)NCC(CC)(C)NC(c1ccccc1OC)=O 31261,C(=O)(C(C)(O)C(C)C)NCCCN(C(c1ncc(OC)nc1)=O)C 31262,Cc1occ(C(F)(F)F)c1C(=O)NCC1CCC(NC(=O)Cc2n[nH]c(=N)s2)C1 31263,c1(C(N(C)CC2(NC(c3coc(N(C)C)n3)=O)CC2)=O)ccc(CCC(N)=O)cc1 31264,C1(C(=O)NC2CCN(C(=O)CCc3ncco3)C2C2CC2)CCCS(=O)(=O)C1 31265,C1(NC(c2n(CC)cnn2)=O)CC2CN(C(=O)Cn3c(C)csc3=O)CC2C1 31266,CCC(C)(C(=O)NCC1(F)CC(NC(C2CCCC(C)(C)C2)=O)C1)C(N)=O 31267,C1(C(=O)NCCC2CN(C(C(C)OCCC#C)=O)C2)CC2CCC1O2 31268,c1(C(=O)NC(C(=O)NCCSCC)C2CC2)ccc2c[nH]nc2c1 31269,Cc1ccc(N)cc1C(N1CCCC(CO)(NC(=O)Cn2nnnc2C)C1)=O 31270,N1(C(C2CC(Cn3cc(CSC)nn3)C2)=O)C2CCCC1C(C(=O)OC)C2OC 31271,CCC(C(=O)N1CCC(NC(=O)CN2CCN(C)C(=O)C2)C1C(C)C)C(F)(F)F 31272,c1(C(=O)NC(CC(CC)C)C(=O)NCCOC)noc2ccc(Br)cc12 31273,C1(CN(c2csc(-c3ccco3)n2)CCNC(CCCC)=O)CCCCCC1 31274,C(C)(C(=O)N1CC(C(O)C(=O)NCCn2ccnc2)C1)OCC=C 31275,C(=O)(C(O)CC(N)=O)N1CCC(C(=O)Nc2cn(CC#C)nc2)(OC)C1 31276,N#Cc1c[nH]c(C(N2CCC(CN3CCN(c4cc(N)ncn4)CC3)CC2)=O)c1 31277,C1(NC(CC2(C=C)CCC2)=O)CCCN(C(c2cccnc2C(F)F)=O)CC1F 31278,N1(C(C(c2cnn(C)c2)NC)=O)CCc2ncc(C(F)(F)F)cc2C1 31279,c1(C(=O)NC2C3CC(NC(C)=O)C(C3)C2)noc2c1CC(F)(F)CC2 31280,CCCC(O)C(=O)NCC12CC(CN1C(C1(c3ccccc3)CC(C)C1)=O)C2 31281,C1(C(C)(C)C)(CNC(CN(S(CC)(=O)=O)C)=O)CCN(C(=O)C(F)C2CC2)C1 31282,c1(NC(c2ncc(-c3c(OC)ccnc3)cn2)=O)cc(Br)c(O)cc1Br 31283,CCC(CCC(=O)N1CCC(C)C1NC(=O)C=CC(=O)NC1CC1)OC 31284,C1(N(C(c2c(C)nsc2)=O)C)CCCCC1NC(C1(C)CCC1)=O 31285,N1(C(c2c(C)cco2)=O)CCC(C2CCN(C(=O)CC3COC(C)(C)C3)C2)CC1 31286,C1(C(=O)NC(C)C(N)=O)C2CCC1CN(C(c1cc3ccoc3s1)=O)C2 31287,c1(OCC(=O)NC2C(NC(c3c(C)cno3)=O)C2)cccc(Br)c1C#N 31288,C(C(C)(C)CC(=O)N1CC(NC(=O)CCc2c(C)noc2Cl)C(C)C1)OC 31289,c1(CCC)c(C(=O)N(C2CCCN(C(=O)C(F)=C(C)C)C2)C)nnn1CC 31290,c1(NC(C(C)SCCCC)=O)nc(Cl)ncc1NC 31291,CC1(c2cn(-c3ccc(C(=O)O)cc3)nn2)CCCN1C(C1CCOCC1)=O 31292,Cc1ccc2c(C(=O)NC3CCC4CCN(C(c5cccnc5)=O)C34)n[nH]c2c1 31293,N1(C(C(C)C)=O)CCCCC1C(C)NC(=O)CCCc1nccs1 31294,C(=O)(C(CC)CC(F)F)N(CC(CNC(CCOCCOCC)=O)(C)C)C 31295,N1(C(c2nc(=N)[nH]cc2)=O)CC(F)(F)CC1C(=O)NC1C(O)C2CCOC12 31296,C1(C2C(NC(CN(c3ccccc3)C)=O)C2)CCCN1C(=O)CSCC(C)(C)C 31297,C1(C)(CNC(CC2N(C(Cc3c(C)con3)=O)CCC2)=O)CCCCO1 31298,N1(C(CCCC#C)=O)CCC(NC(=O)C=Cc2ccc(C(N)=O)cc2)CC1C 31299,C1(CC)(NC(=O)CSCC(C)C)CCCN(C(c2ccnn2CC(F)(F)F)=O)C1 31300,CC1(C)CN(C(=O)C(C)(C)C2CC2)CC1NC(=O)Cc1ccccc1Br 31301,c1(NC(CCCC=C)C)ncc(S(=O)(=O)N(CC)CC2CCOCC2)cc1Cl 31302,c1(CC(C)NC(c2c(C)nc(COC)s2)=O)cc(F)c(F)cc1Br 31303,C(=O)(C#CC1(C)CCCO1)NC1CCC(NC(c2cc(C)cc(Cl)c2N)=O)CC1 31304,C1(COC)CN(N2CC(c3ncc(C(C)C)[nH]3)C2)CC1OC.c12ccc(cc1)NC2 31305,Cc1cc2ccccc2nc1C(N1CC(CNC(c2ccc(F)c(O)c2)=O)C1)=O 31306,C1(NC(c2cc(CC)c(CC)o2)=O)CC(C)CN(C(=O)CC(=O)NC2CC2)C1 31307,C(=O)(C1=CCC(C)CC1)N(CCN(C(C1CC1CC(C)(C)C)=O)CC)CC 31308,N1(C(C)C)CCCCC(N=c2[nH]c(=NC3CC(OC(F)F)C3)[nH]c3c2CCC3)C1 31309,C(=O)(C1=CCS(=O)(=O)C1)N1CCC(NC(C(C(=C)Cl)(C)C)=O)C(F)C1 31310,C(C)(CSC)(C(=O)NCCCC(F)(F)F)NC(c1cn(CCC)nc1)=O 31311,N1(CC(=O)NCCCCCF)CCN(C(c2cnco2)=O)CC1 31312,C1(C#N)(C(=O)NCCC(C)NC(c2c(C)cc(O)nc2)=O)CC12CCOCC2 31313,N1(C(CC(C)(C)n2cnnn2)=O)CCN(C(C2C3CN(CC(F)(F)F)CC23)=O)C(C2CC2)C1 31314,C1(CC)CN(C(=O)CCNS(=O)(=O)C(F)F)CCC1NC(C1(CCOC)CC1)=O 31315,N1(C(=O)NC2CC(O)C23CCOCC3)CC2CC3CCCN3C2C1 31316,c1(CC(C(=O)NC(CN(C(COC(CC)C)=O)C)(C)C)O)ccncc1Br 31317,CC1(C)COC(CC(=O)NC(C(=O)N2CC(CC(N)=O)C2)c2cccs2)C1 31318,C1(CN(C(c2cc(C(C)(C)C)on2)=O)CC)CCCN1C(=O)CC1(N2CCCC2)CC1 31319,C1(N(CC(C2CC2)NC2(C(=O)OC)CCC2)C2CC2)C2CCCCC12 31320,N1(C(C2NC(=O)C(F)C2)=O)CCCC2(CC(NC(c3cnco3)=O)C2)C1 31321,n1(CCC)cc(C(=O)NC2CC23CC(NC(=O)CS(=O)(=O)NCC)C3)c(C)n1 31322,C1(NC(c2c(C)n[nH]c2)=O)COC2CN(C(c3ocnc3C)=O)CC12 31323,c1(CCC)ncc(NC(=O)C(C)(C)CN(C(=O)C=CC2CCOC2)C)cn1 31324,c1(CCCC)nc(C(N2CC(CO)(NC(c3nc(C(C)(C)C)no3)=O)C2)=O)cs1 31325,C#Cc1ccc(C(N2CC3CC(NC(C45CCCC4CCC5)=O)C3C2)=O)nc1 31326,n1(CCNC(=O)CCC2CC(C(c3cn(C4(C)CC4)nn3)=O)CO2)cnc(=N)[nH]1 31327,N1(C(C(C)N(C(C)=O)C)=O)CC(F)(F)CC1CNC(c1cccc(C)n1)=O 31328,C12=CNC=CC1=NCC1(F)CC(C1)NC2=O.c1(OCC)scc(OCC)c1OC 31329,c1(-c2cc(C)no2)cccc(CNC23CC(C(=O)NC(C#N)C(N)=O)(C2)C3)c1 31330,S(=O)(=O)(c1ccc(Br)cc1NCC1OCC1(C)C)N1CCCC(CCC)C1 31331,c1(SCC)nccnc1C(=O)NCC(C(C)C)NC(C1(CC)CCC1)=O 31332,CC1C(NC(C2CCC2)=O)CC2CCC1N2C(=O)CC1CC(F)(F)C1 31333,C1(C(=O)NCCCCNC(c2c(C)n(C3CCOC3)nn2)=O)CCCS(=O)(=O)C1 31334,c1(C(C)NC(c2ccnnc2)c2nnnn2CCF)cccnc1 31335,c1(C(=O)NCC2(F)CCC(NC(C3CCS(=O)(=O)N3)=O)C2)ccc2nn[nH]c2c1 31336,Cc1ccncc1CC(=O)NC1CN(C(c2ncc(Cl)s2)=O)CC1C 31337,c1(C(N2C(CNC(C3C(COC)C3)=O)CCC2)=O)ccc2ncc(=O)[nH]c2c1 31338,C1(c2cn(CCCN(C)C(c3cncc(OCC#N)c3)=O)nn2)COCC1(C)C 31339,C1(CNC(C2CCN(C(C)=O)C2)=O)CCCN(C(c2n[nH]cc2C(C)(C)C)=O)C1 31340,C(=O)(CCC(C)OC(c1ccc(C2CCC2(C)C)cc1)=O)OCC 31341,CCCCC(C(=O)N1CC(S(C)=O)C1)NC(=O)CC=CC(C)(C)C 31342,c1(C(=O)NCC(O)CNC(C2CC3CC3C2)=O)ccc(S(=O)(=O)C(F)(F)F)cc1 31343,C1(CNC(CN2CC(C)C2)=O)CC2CN(C(C3(C(C)(C)C)CCCCC3)=O)CC12 31344,c1(C(N2C(C(=O)NCC3CCCO3)COCC2)=O)ccc(O)c(F)c1 31345,CC1SCCC1NC(C1(CCNC(C2CC3(CC3)C2)=O)CCCC1)=O 31346,c1(OC)ccccc1CC(=O)NCCNC(c1cc(O)cs1)=O 31347,c1(CN(C)C(C2N(C(CC3C(CC)C3(F)F)=O)CCC2)=O)nnn(C)c1N 31348,C1(F)(CNC(=O)Cn2cnnn2)CCCN(C(=O)CCCc2ccncc2)CC1 31349,CCC1=NOC(C(=O)NCCN(C(=O)CCc2ccncc2Br)C)C1 31350,C(C)(CCC(=O)NC(CSC)C(=O)NCc1nc(CSC)no1)OC 31351,C1(C(CNC(CC(C)F)=O)(C)C)CCN(C(c2cnn(C)c2C(F)(F)F)=O)CC1 31352,C1(CNC(CCSCCC)=O)CCCCN(C(C2(C)CSC2)=O)C1 31353,C(CC(=O)NC)C(C1CN(C(C2CC2c2nc[nH]n2)=O)C1)C.c1(C(=O)N)cnco1 31354,N1(C(c2cncc(COC)c2)=O)CC(NC(=O)Cc2cc(OC)no2)CC(O)C1 31355,N1(C(C2C(C)(C)CC(=O)NC2)=O)CC23CCCC2(C1)CN(c1ncc(F)cn1)C3 31356,N1(C(c2c(C)ncc(N)c2)=O)CC2CCCC(C1)N2C(=O)C(F)(F)C1CCCC1 31357,C(=O)(C1=CS(=O)CCC1)NC(C1(O)CN(C(C2(OC)CCCCC2)=O)C1)C 31358,Cc1cc(C)c(C#N)c(NC(C2CCCN(C(c3ccc(Cl)nc3)=O)C2)C)n1 31359,c1(OC)ccc(C=CC(=O)NC2CCN(C(C3(C)CC3(F)F)=O)CC2O)cc1Cl 31360,c1(C(=O)NC2C(NC(COCCC)=O)COC2)sc([N+](=O)[O-])cc1Cl 31361,c1(C(=O)OC)cc(C(=O)NC2CN(C(=O)CSCCC(C)C)CC2C)n(C)n1 31362,c1(OC)cnc(F)cc1C(=O)NC1COCC1NC(=O)C=CC1CCCC1 31363,Cc1c(CNC(c2nn(-c3ccccc3)nc2C)C)nnn1C 31364,N1(C(C2CCC(C)(CC)O2)=O)CCC2CCN(C(=O)C(CC)(CC)OC)CC12 31365,c1(C(N2CCN(C(C)CNC(C3(CC4CC4)CC3)=O)CC2)=O)nccn2nccc12 31366,c1(C(N2C3CN(C(C4(O)CC(C)(C)C4)=O)C(C3)C2)=O)cc2n(n1)CCC2 31367,C1(N(C(=O)C(O)CC2CC2)C)CCCN(C(c2ccc(OC(F)F)cc2)=O)CC1 31368,c1(C(N2C(CNC(=O)COCC3CCOC3)C=CC2)=O)nccc2cc[nH]c12 31369,c1(CC(=O)NC(C2(O)CN(C(=O)C=Cc3cccs3)C2)C)sccc1Br 31370,c1(NC(c2c(OC)ccc(C(F)F)c2)=O)cc2cncn2c(O)n1 31371,N1(C(Cc2c(OC)nccc2)=O)CC2(CCCCN2C(C2OCCOC2C)=O)C1 31372,C12(NC(COC)=O)CC(CNC(C3(Cl)CC3(F)F)=O)(C1)OC21CCC1 31373,C1(NC(CC2(NC(c3cc(SC)oc3)=O)CC2)=O)CCCCC1CCO 31374,c1(OC)c(C(N2CCC(CNC(C3CC3C(=O)NCCO)=O)C2)=O)ccnc1Cl 31375,C1(C(=O)NCC(CC)NC(=O)CC2CCCO2)(OC)CCS(=O)(=O)C1 31376,N1(C(=O)NC(C2CCC3(CC3)N2C(=O)OC(C)(C)C)C)CCCc2ccccc21 31377,c1(C(N2CCC(N3CCN(C(C)=O)CC3)C2)=O)ccc2c(n1)OCCO2 31378,c1(C(=O)OC)nn(C)c(NC(C2CN(C(C3CN(C)C3)=O)CCS2)=O)c1Cl 31379,CCCCN=C(NCCC1(NC(=O)OC(C)(C)C)COC1)NC1CCS(=O)(=O)C1 31380,N1(C(Cc2nn(C)c(Cl)c2)=O)CCC2C(C1)CN2C(C1CCCNS1(=O)=O)=O 31381,C1(C(N2CCOC(c3cn[nH]c3)C2)C(=O)NCC(F)F)CCOC2(CCC2)C1 31382,Fc1cc2nc(-n3nc(C4CC4)nc3CCC(F)(F)F)[nH]c2cc1F 31383,C1(C(=O)NCC(C)(C(C)C)NC(c2c(OC)n(C)nc2)=O)CCN(C)C(=O)C1 31384,N1(C(C2(C)CCSCC2)=O)CCC(F)C(NC(C2(n3cccn3)CCC2)=O)C1 31385,C(=O)(C(C)CC(C)C)N1C(C2CCN(Cc3nc(CC)on3)C2)CCC1 31386,N1(C(c2ccc(NC)c(F)c2)=O)CCC2CCN(C(C3CC=CC3)=O)CC12 31387,c1(C(N2C(C(N3CCC(CN(C)CC)C3)=O)C=CC2)=O)ncccc1Cl 31388,N1(C(=O)NC)CCC(C(=O)NCC(O)CNC(c2sccc2-n2cnnn2)=O)C1 31389,CCC(CCOC)C(=O)N1CC2CC(C1)C2NC(=O)CC1C(=O)NN=C1C 31390,c1(NC(C)=O)cccnc1C(N1CCOC(C(C)NC(=O)CCNC(N)=O)C1)=O 31391,C(=O)(CC1=CCN(C)CC1)NC(CCC)C(O)C(=O)NCC1CCOC1=O 31392,C1(CN(C(=O)Nc2cnco2)CC)CCCN(C(=O)OC(C)(C)C)C1 31393,Cc1nc(C)c(C(=O)NCC2CCOC2C(=O)Nc2ccc(C(C)C)nc2)s1 31394,CC(CC1CCCO1)C(=O)N(CCCOCCNC(c1csc(O)n1)=O)C 31395,C1(NC(C2CCC(O)(c3cccc(F)c3)CC2)=O)CCCC(F)(F)C(=O)N1 31396,C1(C(=O)NCCCN(C)C(C)C)CC(C(F)F)(NC(C(C)=C2CCC2)=O)C1 31397,C1(CC)CCN(C(c2cc(C)oc2C)=O)C1CNC(=O)C=CC1CCOC1 31398,C(=O)(C(C)(C)C(F)F)NC1CCC(F)(CNC(C2N(C(C)=O)CCC2)=O)C1 31399,C1(C(=O)NCC2(O)CCN(C(CCCN=[N+]=[N-])=O)C2)CCCCCC1(F)F 31400,c1(C(N(CCNC(CC)=O)CCOC)=O)ccc2c(c1)CCCCN2 31401,O=C(CCC(F)(F)F)NCC12CC1CN(C(c1cncc(O)c1)=O)C2 31402,CCC(CNC(C1CCOC(C)C1)=O)(CC)NC(=O)Cc1ccnnc1O 31403,C1(C(N2CCC(CCN(C(=O)Cc3ccc(Cl)s3)C)CC2)=O)(CC)CNC(=O)C1 31404,CN1CC(F)CC1C(N1CC(OCCNC(C2CC2[N+](=O)[O-])=O)C1)=O 31405,C1(COC)(CNC(C2C(C)C2C)=O)CCN(C(=O)Cc2cnc(C)[nH]2)CC1 31406,C1(CNC(C(CC)(C)COC)=O)CC2CCC(C1)N2C(=O)C1=NOC(C)(C)C1 31407,C1(O)(CNC(c2c(CC)occ2)=O)CCCN(C(=O)C(C)(C)C2(C)CC2(F)F)C1 31408,C1(C(=O)NC(CC)CNC(C2C3(CC3)C23CC3)=O)CCc2c(ncn2C)C1 31409,C1(NC(c2ccnc(C(C)C)n2)=O)CC2CC1N(C(=O)Cc1nc[nH]n1)C2 31410,N1(Cc2ccc(OC)nc2OC)Cc2[nH][nH]c(=NC(=O)c3cccc(O)n3)c2C1 31411,c1(C(=O)NC2C(NC(C(C3CCC3)OCC)=O)CCCC2)cc2c(o1)CCCC2 31412,Cc1c(C(=O)NC2CN(C(C3CC4(CC4)CO3)=O)C(C)(C)C2)cccc1C#N 31413,C1(CN(C(c2[nH]nc(CO)n2)=O)CC)CC(C(F)(F)F)CO1 31414,C1(C(=O)N(C)CC2(C)CCC2)(CC)CN(C(=O)C(C)NC(=O)C2CC2)C1 31415,Cc1sc(Cl)nc1C(=O)NC1CCCC1NC(=O)C(F)=C1CCC1 31416,C#Cc1cncc(C(=O)NCC(CCNC(c2cc(C)sn2)=O)OC)c1 31417,N1(C(C(CCC)NC(CC(C=C)CCC)=O)=O)CCC2(CCC(OC)C2)C1 31418,c1(C(=O)NC(CCNC(C(C2CCCCC2)OC)=O)C)cccc(C(F)F)c1 31419,C(C1CN(C(c2ccccc2F)=O)CC1C(=O)Nc1cnc(CO)nc1C)=CC 31420,c1(COC(C)=O)ccc(C(=O)NC(C)(C)CCCNC(=O)CC2CCOCC2)cc1 31421,N1(C(c2c(C)nccc2Cl)=O)CCC(C2CCN(C(C3CC4(CCC4)C3)=O)C2)C1 31422,c1(OCC)ccc(N)c(C(=O)NC2C3CN(C(C4CC(=O)NC(C)C4)=O)CC23)c1 31423,N1(C(C(CSC)O)=O)CC(NC(=O)C(N2CCC(C)CC2)=O)CCC1C 31424,CC1CCN(C(c2ccnc(Cl)c2F)=O)CC1NC(c1cc(F)cnc1Cl)=O 31425,Cc1cc(C(=O)NC2CCC(NC(=O)C(C)OC3CCCCC3)C2)cc(N)c1O 31426,C(CC(CC)C(=O)N1CCCC1C(C)(C)NC(=O)CCCC1CCOCC1)=CC 31427,C12(CNC(Cc3n[nH]c(=N)s3)=O)CCC(CN(C(=O)C3=COCC3)C1)C2 31428,c1(C(=O)OC)ccccc1C(=O)N(CC(C)N(C(=O)C(C)Cc1ccco1)C)C 31429,N1(C(C(CC#C)NC(C)=O)=O)CC(C2CN(C(c3ccc(N)c(OC)c3)=O)C2)C1 31430,C1(OC)CN(C(C2C=CCCC2)=O)CC1NC(=O)C(F)(F)c1nccs1 31431,C(=O)(CCCC(C)C)NCC1C(CNC(c2c(SCC=C)cccc2)=O)C1 31432,C(=O)(C(F)CC(C)C)N(C(CCNC(C1(CC=C)COC1)=O)C)C 31433,CC(O)C(O)CNC(=O)CCC1CCC(NC(C2CCO2)=O)C1 31434,c1(OC)cccc2c1ccn2CC(C1CC1)OC1CCCN(C(=O)NC)C1 31435,C1(C)(CC)C=C(C(=O)NCC(C)N(C)C(c2ncc(Cl)cc2F)=O)C1 31436,C(=O)(C=CS(C)=O)NCC1C(NC(C=CC=CC)=O)COC1 31437,C1(C)(C(N2CC(CNC(c3ccc(C(C)=O)nc3)=O)C(O)C2)=O)CCCS1(=O)=O 31438,N1(C(C(C2CCCC2)OC)=O)CC(CNC(=O)C=CC(F)F)CC1(C)C 31439,C(=O)(C1Cc2ccccc21)N1CC2CN(C(=O)C=CC3CCOC3)CC2C1 31440,c1(C2(NC(=O)NCC(C(C)O)O)CCC2)ccc(Cl)nc1O 31441,C(=O)(CS(=O)(=O)CCOC)N(C(C)CNC(c1cc(CS(C)(=O)=O)on1)=O)CC 31442,CC(C)CCCC(=O)NCC1(F)CCC(NC(C2CCC(C)(C)OC2)=O)C1 31443,N1(CC)CCC(C(=O)NCCCCN(C)C(c2c[nH]nc2-c2cnn(C)c2)=O)C1 31444,CC(C)C(C)(CNC(=O)CN1CC2CCC1C2)NC(=O)CN1C(=O)CNC1=O 31445,c1(CN2C(CNC(c3c(C)cc[nH]3)=O)CCC2)ccc(C(F)(F)F)cc1Br 31446,c1(C(=O)NC(CNC(C2CC(C3CCC3)C2)=O)C2CCC2)noc2c1COCC2 31447,c1(C(N(CC(C)NC(=O)C(O)CN(C)C)CC)=O)cccc(NC(C)=O)c1 31448,C(C(C(=O)NC1(CC)CCN(C(=O)C(CCC)CC)CC1)C(C)(C)C)OCC=C 31449,C(=O)(CCCC(N)=O)NCC(C1CCN(C(c2cccc(N)c2)=O)CC1)C 31450,CC(CCC(C)(C)C)C(=O)OCCC1(C(F)(F)F)CCC1 31451,c1(OCCNC(=O)Cc2cc(O)nnc2O)cc(F)c(F)cc1Br 31452,c1(C(N2CCC(C)(NC(=O)Cc3nnc(O)s3)C2)=O)ccc(Cl)c2cccnc12 31453,CC(CCCNC(c1cc(Cl)c[nH]1)=O)NC(=O)CCOc1ccccc1 31454,Cn1nc(C(F)F)cc1S(=O)(=O)NCCc1cccc(Cl)c1 31455,C(C(=O)NCC(Br)=C(C)C)(C1CCOC1)NC(C1(OCC)CC1)=O 31456,C1(C(=O)NCCN2CCOCC2)(CNC(CN(C2CCSC2)C)=O)CCCC1 31457,C(=O)(CCC(F)(F)F)N1CC(NC(=O)CSC2CCC2)C(C(F)F)C1 31458,C(=O)(C(C)(C)C(C)(C)O)N(C(C)C(=O)N(C)C)C1CC1.C12C=CC(C1)N2 31459,Cc1nc2ccccc2cc1C(=O)NC1CC2CC1N(C(=O)C(C)(C)C)C2 31460,c1(C(=O)NCC(CN(C(C2CC(O)(CC#C)C2)=O)C)O)nc(OC)c(C)s1 31461,O=C1CCC(NC(c2conc2CNC(=O)CCCN2CCCC2)=O)C(=O)N1 31462,C(=O)(CC1OCCc2ccsc21)NCC1CCN(C(C2C(C)(C)C2(C)C)=O)C1 31463,C1(C(=O)NCC(C)(CC(C)C)NC(CCC(=C)Cl)=O)CCOC2(CCOCC2)C1 31464,C1(C(=O)NCC2(CC)CCCC2)CCN(C(=O)C(C)(C)C2CCCO2)C(C)(C)C1 31465,c1(CN(C2C3CNC2C3)CC(=O)NCCCC)ccc(OC)cc1 31466,Cc1[nH]nc(C(N2CC3C(NC(=O)C(C)(C)n4cc(Cl)cn4)C3C2)=O)c1F 31467,C1(COC)(CNC(c2ccc(C(N)=O)o2)=O)CCN(C(=O)C=C(C)Cl)C1 31468,c1(CC)ncc(CNC(C2(CCNC(=O)C=C3CCC3)CC2)=O)[nH]1 31469,c1(OCC(=O)NCC(CC)(CC)NC(CCC#CC)=O)ccc(C(C)C)c(C)c1 31470,C#Cc1ccc(C(=O)NCC2(C)CCC(NC(c3cc(OC)nn3C)=O)C2)cc1 31471,c1(C(=O)NCC2CC2NC(C2CCC3(CC3)C2)=O)cc(=O)c2ccncc2o1 31472,c1(OC)ncc(C(C2N(C(c3cnn(C)c3)=O)CCC2)=O)c(C)c1Br 31473,CC1(C)CN(C(c2cccc3cc[nH]c23)C(=O)NC2CCC2)c2cccc(Cl)c21 31474,N1(C(c2cc(C3(C)CC3)n[nH]2)=O)CCCCC1CN(C(C1CCOC1=O)=O)C1CC1 31475,c1(CC)nnsc1C(=O)NCC1(C(N2CC=CC2)=O)CCCO1 31476,N1(C(C2(CSC)CC2)=O)CC(C2(NC(c3cnc(S)n3C)=O)CC2)C1 31477,Cc1cccn2cc(C(=O)NCC3C(O)C(O)CN3C(c3cscc3Cl)=O)nc12 31478,c1(CCC(=O)NCC(C)N(C(c2ccnc(OC)n2)=O)C)ccc(C#N)cc1F 31479,N1(C(C2N(Cc3c(OCC)cc(F)cc3)CC(F)C2)=O)CCC2(CC1)OCCO2 31480,Cc1nc(C#N)c(NCCC(N2CCN(C(=O)C(C)(C)C(N)=O)C3CC23)=O)o1 31481,C1(C(N2CCC(C(C)(C)NC(C(C)=CC)=O)C2)=O)CCc2[nH]nc(O)c2C1 31482,N#CC1CCCC(C(=O)NC(Cc2ccco2)C(N2CC(F)CC2CO)=O)C1 31483,c1(C(=O)NC2CC(CNC(C(CC=C)C)=O)C2)ccc(Cl)cc1-c1ccccc1 31484,Cc1ccc(CC(=O)N(CCCNC(=O)C(C)OCCN(C)C)CCO)c(Cl)c1 31485,C1(OC)CCC(C(=O)NCCC2(SC)CCC2)C1.c12csc(n1)C(C)NC(=O)C2 31486,O=C1OC2CC(C(=O)NCC3CCC3NC(c3cncc(C(F)F)c3)=O)CC2O1 31487,C(C)(CCCC(=O)NOCC(=O)NC1CC1)NC(C(CCCC)=O)=O 31488,Cc1cc(NC(C2CC(CF)C2)=O)ccc1NC(C1C2CCCC12)=O 31489,c1(C(C)C)nc(NCC2CNC(=O)CO2)cc(=NC2CC3COCC(C3)C2)[nH]1 31490,N1(C(C2(CNC(COCCCOC)=O)CC23CCC3)=O)CCCC2(CCC2)C1 31491,c1(OC)cccc(CC(=O)NCCOC2CCCCC2NC(c2cscn2)=O)c1 31492,CCC(C(=O)NCC(O)CCNC(=O)Cc1csc(C(C)C)n1)NC(C)=O 31493,n1(CC)nc(C(N2CCOC(CNC(=O)C(C)CCOC)C2)=O)cc1C(F)(F)F 31494,C12(NC(c3ccc(C)c(F)c3)=O)CCOCC1CN(C(=O)C1CC1)C2 31495,C(=O)(C#CC(C)(C)C)NCC(C(=O)NC1CC2CC(O)C1C2)N(C)C 31496,c1(C(N(CC(=O)NC(C)CN=[N+]=[N-])C)=O)ccncc1F 31497,Cc1ccc(F)c(C(N2CC(NC(c3c(C)nc(C)nc3C)=O)C(C)C2)=O)c1Cl 31498,c1(C(N2C(C(=O)Nc3ccc(Cl)c(O)c3)CC2)=O)cnc2c(Br)cccc2c1 31499,c1(C(N2CCC(CNC(C(CCC#C)O)=O)C2(C)C)=O)ccc2occc2c1 31500,n1(C(C)(C)C)cc(C(=O)NCC2(Cc3cc(C(=O)NC4CCC4)sc3)CC2)nn1 31501,c1(OC)ccc(C)cc1N1CCC(Nc2nnc(C3CC3)n2C2CCCC2)C1=O 31502,c1(C(N(C2CCN(C(c3cncn3C)=O)C2)CC)=O)c2c(nn1C)CCC2 31503,c1(CN2C(C(=O)NCCCOCC)CCC2)cc(C(C)C)ccc1C 31504,C=CC(C)(C)CCNC(=O)C(C)N(C(c1ccnc(CO)c1)=O)C1CC1 31505,C1(CC(=O)NC(C2(O)CCCCC2)C(=O)N(C2CC(F)(F)C2)C)CC2CCC1C2 31506,n1(CC)nc(C(=O)NCC23CC2CN(C(=O)C=CC(=O)NC2CC2)C3)ccc1=O 31507,c1(C(N(CC(CC)NC(=O)C=CC2CCOCC2)C)=O)cn(C)nc1C 31508,CCC(C)CC(=O)C(=O)N1CC(C(=O)NCCCCCCF)C(C(C)C)C1 31509,c1(OC)ncc(C(=O)NOCc2cn(CCCN3CCOCC3=O)nn2)cn1 31510,c1(N(C)C)ccc(NCc2c(Cl)ccc(F)c2F)cc1C#N 31511,c1(CC)c(C(=O)N(CC(C)NC(=O)C(c2ccc(Cl)s2)=O)C)cnn1CC 31512,N1(C(C(CO)NC(CN2CCC(C)CC2)=O)=O)CC(C)OC2(CCC2)C1 31513,c1(CCN(CCOC)C(CC(C)C)=O)ccc(OCC(F)(F)F)cc1OC 31514,Cc1cccc(CC(N2CCN(CC(C)O)C(C)C2)=O)c1Br 31515,C=C(C)CCCNC(c1[nH]ccc1CNC(=O)C(c1cnn(C)c1)O)=O 31516,C(N=c1[nH]c(=NCc2ccc(F)cc2)[nH]c2cc[nH]c12)c1cc(CC)[nH]n1 31517,CC1CN(C(C2CC(n3ccnc3)C2)=O)CCC1NC(c1ccc(O)nc1)=O 31518,C(=O)(C(F)CC1CC1)NCCC(C)NC(COCCOCCOC)=O 31519,N1(C(CCCCSC)=O)CC2CCCN(C(=O)CCc3cc(C)[nH]n3)C2C1 31520,C=CCCCCCNC(c1csc(CNC(=O)C(C)C2CCCO2)c1)=O 31521,c1(C(=O)NCC2N(C(c3cncc(CC)c3)=O)CCOC2)cc(Cl)c(F)cc1F 31522,C1(CC)(CNC(C2(CNC(=O)CC3OCCCO3)CC(C)(C)C2)=O)CCC(=O)N1 31523,C(N=c1[nH]c2cc(F)ccc2o1)C1CCN(C(c2cccc(OCC)c2)=O)C1 31524,Cc1cc2[nH]c(C(N3CCC(CN(C)C(C4CCC5(CCC5)C4)=O)C3)=O)cc2s1 31525,C1(CC=C)(C(=O)NS(=O)(=O)C2CC3(CC3)C2)CCS(=O)(=O)CC1 31526,N1(C(C(C)OCC)=O)CCC2CN(C(c3cc(OC)nc(OC)c3)=O)CC2CC1 31527,C(=O)(C(F)(CNC(=O)Cn1ccnc1)C(C)C)NC(C#C)C(C)OC 31528,CC(CN=c1[nH]c2cccc(F)c2s1)(C1CC1)NC(=O)CCc1cc(Cl)cs1 31529,Cc1nn(C)c(NC(=O)C(C)C(C)(C)c2ccccc2)c1Br 31530,N1(CCC)CC(C(N2CCCC2CN(C)C(c2csc(Cl)c2Cl)=O)=O)CC1=O 31531,C1(C(=O)NCC)Cc2nccnc2CN1C(c1ccc(F)cc1CC)=O 31532,CCC(C)C(O)C(C)C(=O)N1CCC(CCC(=O)NCCSCCOC)C1 31533,c1(C(=O)NCC2CCN(C(C(C)OC)=O)C23CC3)ccnc2[nH]c(C)nc12 31534,C12(NC(C(C=C)O)=O)CCC(CC1)N(C(=O)Cc1sccc1C)C2 31535,C(=O)(CC(F)(F)C(F)F)NC1C(NC(CC(n2c(C)cc(C)n2)C)=O)COC1 31536,C(=O)(C(C(C)(C)C)N(C)C)NC1C(NC(c2cc(CC(C)C)[nH]n2)=O)CC1 31537,C(=O)(C(C)(F)C(=O)NCCCOCCNC(C1(C)CCC1)=O)OC 31538,C1(O)(CN(C(=O)C2=COCCO2)C)CCCN(C(=O)CC2CCCC2(F)F)C1 31539,c1(CC)noc(C)c1C(=O)OC.c12ccc(nc1)CNC(=O)Cn1cc-2nn1 31540,C(=O)(CCCCNS(C)(=O)=O)NCC(CC)N(C)C(C1CN(S(C)(=O)=O)C1)=O 31541,C=CC1CN(C(=O)C(CC(C)C)OC)CC1NC(=O)CCN1CCC(O)CC1 31542,Cc1cccc(C(C)C)c1C(=O)NC1(C2CN(C(=O)C=CCCC(C)C)C2)CC1 31543,N1(C(COC(CC)(C)C)=O)CC(C)CCC1CNC(c1cccc(F)c1F)=O 31544,c1(C(=O)NCC(CCOC)NC(c2cnc(CC(C)C)s2)=O)ccn(C)c(=O)c1 31545,c1(CC)noc2ncc(C(N3CCC4C(NC(=O)C(C)=CC(C)(C)C)C34)=O)cc12 31546,c1(C(C(=O)NCCC2CC2)N(C(C)COC)CCOC)ncn(C)n1 31547,c1(NS(CC)(=O)=O)ccc(C(=O)NCC(C)(C)CNC(=O)CC(=O)OC)cc1 31548,C1(CC)C=CCCN1C(=O)CCC1(C)CCCN1C(=O)COCCCOC 31549,c1(OC)cc(C(=O)NCC2CCCN2C(=O)C=C(C)C(F)F)c2ccccc2n1 31550,c1(CC)cc(C(=O)NC2CN(C(C3OCCO3)=O)C3CC23)n(C)n1 31551,c1(NC(=O)NCCC(O)c2cccs2)ccccc1CCC(F)(F)F.O 31552,C1(C(=O)NCCC(N)=O)COC2CN(C(c3ccc(F)c(F)c3Br)=O)CC12 31553,C(=O)(CC1=CCN(C(c2cnc(NC)cn2)=O)CC1)NC1(C)CC(C(=O)OC)C1 31554,C1(CC)CCC(NC(C2(F)CCN(C(=O)C(C)C(=O)OC)C2)=O)CC1 31555,CCCCC(C(=O)NC1(C(=O)NC)CC=CC1)NC(=O)C(O)CC(C)C 31556,N1(C(c2c(C)cns2)=O)CC=CC(NC(=O)CCCOCCN(C)C)C1 31557,C1(CNC(C(C)=C2CCC2)=O)(NC(=O)CC2CCCCCC2)CC2CCC1CC2 31558,C1(C(N(CCC#C)CCO)=O)CCN(C(c2occc2CC)=O)C(CC)C1 31559,c1(CN=C(NCC(O)CF)NC2CCC2)ccc2c(c1)CCO2 31560,c1(COC)cccc(C(=O)NCC2CCC(F)(CNC(=O)CC3CCCO3)C2)c1 31561,N1(C(C2CN(C(c3c(C)nn(C)c3C)=O)CC(C)C2)=O)CCOC2(CCC2)C1 31562,c1(C(=O)NC2C(CNC(=O)COC(F)F)C2)cc2ccc(Br)cn2n1 31563,c1(COCC(=O)NC2CCCO2)ccccn1.N12CC(O)(C1)CCNC(=O)C2=O 31564,c1(NC(=O)C(N2CCCC2C2COCCC2O)=O)cnc2c(c1)CCC2 31565,N1(C(CCSCC(C)C)=O)CCCC(C)(NC(=O)Cc2ccc(Cl)cc2)C1 31566,Cc1cc(CC(CO)NC(=O)Nc2cccc(N3CCCC3)c2)ccc1Br 31567,C1(NC(COC(CC)C)=O)C(C(=O)NCC(C)(O)COC)C1(C)C 31568,C=CCCN=C(NCC12CC3CC1C2C3)NC1CCCC(OC(F)F)C1 31569,N1(C(=O)CSc2cncc(N3CCCC3)n2)CCc2[nH]nc(CO)c2C1 31570,c1(C(C)(C)C)ccc(C(=O)NC2(CNC(C3CCCOC3)=O)CCC2)[nH]1 31571,N1(C(c2cccc(NC(C3C(N)C3)=O)c2)=O)Cc2ccccc2CC1C(=O)N(C)C 31572,c1(C(=O)NC2C(NC(c3cscc3F)=O)C2)ccc(-c2ccco2)[nH]1 31573,c1(C(=O)NCCOC2CC(NC(CC(C)C(F)F)=O)C2)cc(N)cc2ccccc12 31574,N1(C(c2ccc(C)cn2)=O)CC2CCN(C(=O)CC34CCCC3C4)C(C2)C1 31575,c1(C(N(C)CC2CCCN2C(C2OCC2(C)C)=O)=O)c(C(F)(F)F)cnn1C 31576,CC(C)CC(CNC(c1cnn[nH]1)=O)NC(=O)CSc1nnnn1C 31577,CC1(C)CC(CNC(c2ccco2)=O)CN1C(c1ccccc1C1CCCC1)=O 31578,C1(NC(C2CC(NC(COCC(C)C)=O)C2(C)C)=O)CCN(C)C1(C)C 31579,c1(OCC)ccccc1C=CC(=O)NC(C)CC(C)NC(=O)CCSCC(C)C 31580,C(=O)(C(CNC(=O)CC1CCC(=O)NC1)C(C)(C)C)N1CC(CN(C)C)C1 31581,N1(C(CC2CCCN(C)C2)=O)CCN(C(=O)C(F)=CC2CC2)C(CC(F)(F)F)C1 31582,C1(C(=O)NC23C(CN(C(C4C=CCC4)=O)C2)C3)CCC(F)(F)CC1 31583,c1(C(C)=O)ccc(C(N2CCCC2C(C)NC(=O)CCF)=O)o1 31584,N1(C(c2cnccn2)C(=O)NCCSC)Cc2cc(Cl)c(Cl)cc2C1 31585,c1(C(=O)Nc2scc(CC(N3CCC(C(F)(F)F)C3)=O)n2)nc2ccccn2n1 31586,CC(C)CC(C(=O)NCC(C)N(C)C)N(C(=O)CC1(O)CCCCC1)C 31587,N1(C(CN(C)S(N)(=O)=O)=O)CCn2nc(CNC(C3(F)CCC3)=O)cc2C1 31588,C1(NC(C2CCCC2c2nc[nH]n2)=O)(Cc2ccc(Cl)cc2)CCCCC1 31589,N1(C(N)=O)CCCCC1C(=O)NC1C=CCN(C(C2CCC2)=O)C1 31590,c1(NC(C2C(CNC(c3c(C)occ3)=O)OCC2)=O)cccnc1OC(F)F 31591,C(CCC(O)C(=O)NCC(C)(C)C)NC(c1n(C)cc(Cl)c1)=O 31592,C1(C(N2CCOC(CNC(=O)CN3CCCNC3=O)C2)=O)(COC)CC=CCC1 31593,C1(C(N(CC(C)O)CC)=O)C2CCC(C2)C1NC(=O)CCCn1ccnc1 31594,Cc1c(C(=O)NCC2(C)CCN(C(c3cnc(Cl)cc3Cl)=O)C2)cc(O)cc1N 31595,CC(C)CC(C(=O)NCCCNC(=O)C(C)(C)C1CCCO1)NC(=O)NC1CC1 31596,N1(C(CSCC=C)=O)CCC2(CC1)CN(C(C1C3CCC(C3)S1(=O)=O)=O)C2 31597,c1(COC(Cc2c(C)cc(O)cc2)=O)cc(=O)oc2cc(O)c(Cl)cc12 31598,c1(OCC#C)ccc(-c2cccc(C(N3CCCC3CCCOC)=O)c2)cc1 31599,c1(C(=O)NCC(CC=C)NC(c2cnn3cnnc3c2)=O)ncc2[nH]ncc2n1 31600,C1(NC(Cc2ccc(C)o2)=O)CC12CC(NC(C1(CF)CC(F)(F)C1)=O)C2 31601,CC1(F)CCCN(C(C2CCOCCN2C(=O)Cc2ccc3c(c2)CC3)=O)C1 31602,C(=O)(C(C#N)C(C)(C)C)NCCc1c(C(N2CCC(CC#C)C2)=O)c[nH]n1 31603,C1(C(=O)NC2C(C)(C)C2)CCOCC1NC(=O)C(C)(F)c1ccon1 31604,Cn1cnc2cc(C(=O)NCC3(CO)CC3c3ccccc3)ccc2c1=O 31605,Cc1[nH]nc(C(N2CC3CCC3(CNC(=O)C(C)(O)C3CCC3)C2)=O)c1[N+](=O)[O-] 31606,Cc1nc(C(C)NC(=O)CC2(C)CCN2C(=O)Cc2cccs2)c(C)o1 31607,N1(C(CCC(=O)OC)=O)CCC(CNC(=O)C(=Cc2ccccc2Cl)C)CC1C 31608,c1(CNC(=O)Cc2cnco2)cccc(NC(=O)CC2CCSC2)c1 31609,C1(C#N)(COCC(=O)NCC(C)CNC(C2CCOC2)=O)CC12CCOCC2 31610,c1(CC)[nH]c(C(N2CCC3(NC(=O)CS(C)(=O)=O)CC3C2)=O)c(C)c1C(=O)OC 31611,N1(C(CCCc2cc(C)no2)=O)CCC2(CCCN(C(C3CCC(=O)N3)=O)C2)C1 31612,c1(C(N(CCOC)CCNC(c2cc3sccc3s2)=O)=O)c2ccccc2nn1C 31613,C=C(CNC(=O)C(F)C(C)CNC(=O)C=Cc1ccco1)C1CCOCC1 31614,c1(C(=O)NC2C(CNC(CC3N(C)CCC3)=O)C2)ccc2c(O)nc(S)nc2c1 31615,C1(NC(C(C)OCC(C)C)=O)CCCCCN(C(=O)CCCC2CCCCC2)C1 31616,c1(-c2cn(C(C(N3CC(COC)OCC3)=O)C)nn2)ccnc(F)c1OC 31617,N1(C(C2CCCN(CC)C2)=O)CCC(NC(=O)CC(F)(F)F)CC1C 31618,c1(OC)cc(C(N2CCN(Cc3ccc(C)s3)CC2)C(=O)NC(C)C)ccn1 31619,N1(c2cc(C(=O)OCC)ncn2)CCC2C(CCN2Cc2ccc(OC)nn2)C1 31620,CN1CC2CC1CN2C(=O)CCC(=O)Nc1ccccc1.C12=CC=C(C=C1)C2NC 31621,C(=O)(C1OCCn2ccnc21)NC1C(NC(c2cc(CO)on2)=O)C1 31622,N1(C(C(CC)OCC)=O)CCC(NC(c2nn(CC)cc2Cl)=O)C(F)C1 31623,C1(CNC(C2CC(=C)C2)=O)CCC2CN(C(c3ncoc3C3CC3)=O)CCC2C1 31624,c1(C(=O)NCCc2c(CNC(C(C(C=C)C)C)=O)nco2)cn2cc(C)sc2n1 31625,Cc1cnc(F)cc1C(N1CCN(C(=O)CCC[N+](=O)[O-])C(C)C1)=O 31626,C1(C(=O)O)CCC2(CC2)N1C(C1(C(F)(F)F)CC1)=O.CCCCN(CC1CC1)C 31627,c1(C(N2C(C(C)(C)NC(c3cnn(C)n3)=O)CCC2)=O)ccccc1O 31628,C(=O)(C(C(C)C)NC(=O)CC1CCCCO1)N(CCC#C)CCOC 31629,C(CNCc1ccccc1)(C(=O)NC1CN(C(N)=O)C1)N(C)C 31630,C1(C(N(CC(CN(C(C(CC)C)=O)C)O)C)=O)CCC2CCCCC2C1 31631,Cc1ccc(F)c(C(=O)N(CCCCN(C)C(C2(C)C=CCCC2)=O)C)c1Cl 31632,N1(C(CCCNC(C)=O)=O)CCCCC1CNC(C1CNC(=O)N1)=O 31633,c1(C(=O)NC(C2(O)CN(C(CC(C)OC)=O)C2)C)ccnc(C2CC2)n1 31634,C(=O)(C1CCCc2cc(O)ccc21)N(C1CCN(C(C2(C)CCCC2)=O)C1)CC 31635,c1(Cn2cc(CC3CN(C(C4CC4N4CCCCC4)=O)C3)nn2)ccc(Br)cc1 31636,C1(C(=O)NCCC2CCC2)CCCCCN1C(=O)CN1CCN(CCO)CC1 31637,C(=O)(CC1=CCCCC1)NC1CCCN(c2ccc(SC)nc2Cl)C1 31638,O=C(C1CCCc2nn[nH]c21)N1CCC(OC2CN(CCC3CC3)C2)CC1 31639,C=CC1(C(=O)NCCC2CCOC2)CCN(C(=O)Cc2ccc(C)s2)C1 31640,C12(CC(=O)N(C3CN(C(=O)CN4C(=O)CCC4=O)C3)C)CCC(C)(C1)OC2 31641,C1(O)(C(=O)NCC(C)(C2CC2)NC(=O)CCN2CCC(O)CC2)CCCCCC1 31642,C1(NC(C2NC(=O)OCC2)=O)CCCN(C(c2ncsc2Br)=O)CC1 31643,O=C(CC(O)COC1(CNC(c2cc(C3CC3)[nH]n2)=O)CCC1)OCCO 31644,C(=O)(C(C)(O)C(F)(F)F)NC(CONC(C1(C)CCC1)=O)C1CCC1 31645,C(CC(=O)Nc1cc(C)cnc1C)(CC(C)C)NC(CC(COC)(C)C)=O 31646,N1(C(Cc2cc(C)sc2C)=O)CCCC(CO)(CNC(C2OCCC2(C)C)=O)C1 31647,Cc1ccc(F)c(CC(=O)NC2CC2NC(=O)CCCC2CC2)c1 31648,N1(C(C2C(=O)NCC2)=O)CCCC2(CCN(C(=O)CN3CCn4nccc43)C2)C1 31649,C(=O)(CS(=O)(=O)CCO)N1C2C(NC(COCc3ccc(C)cc3)=O)CC(C2)C1 31650,C1(NC(C(CCOCC)NC(C2CCCCS2)=O)=O)CCCC2(CC1)CC2 31651,c1(C(N2C3CC(N(C(C(CC)O)=O)C)CC2CC3)=O)c2ccccc2nn1C 31652,N1(C(=O)NCCCO)CC(C(=O)Nc2ncccc2Cl)CC(F)C1 31653,C1(CCO)(NC(=O)C#CC2CC2)CCCCC1.C12CC1C(=O)NC(=O)N2 31654,c1(C(=O)NCC(C(C)C(=O)OC(C)(C)C)O)cn(C)c2cc(Cl)ccc12 31655,N1(C(CC(C=C)(C)O)=O)CC(C2CN(C(C3CCC(C)(C)OC3)=O)C2)C1 31656,C1(NC(c2cc(C)nn2C)=O)CCSC12CN(C(c1ccc(N)cc1O)=O)C2 31657,C1(NC(c2c(OC)nn(C)c2)=O)CN(C(c2cn(C3CCC3)nn2)=O)CC1(C)C 31658,C1(N(C(=O)Cc2csc(C(C)OC)n2)CC#C)CCN(CC23CC(C2)C3)CC1 31659,N(C(=NCCC1CCOC1)NCc1ccc(Br)o1)Cc1n(CCCC)nnn1 31660,c1(CC(=O)NC2(CO)CN(C(CC(CC)C3CCC3)=O)C2)cnc2ncccn12 31661,C1(C(=O)NCC=CCNC(C(c2cccnc2)C)=O)CCc2nnc(O)cc2C1 31662,c1(-n2cc(C3N(C(C(COC)NC(C)=O)=O)CCC3C)nn2)cccc(O)c1Cl 31663,C1(C(N2CC3C(NC(C4C=CCC4)=O)C(C3)C2)=O)COc2ccccc2O1 31664,N1(C(C2CC(CC)C2)=O)CCN(C(=O)C(C2CCOCC2)O)CC1CC(F)(F)F 31665,N1(C(CC#C)COC)CCN(C(=O)OCc2cnn(CCC(C)C)c2C)CC1 31666,CCC(CN(C)C)CC(=O)NCCN(C(C1COCC2(CC2)O1)=O)C1CC1 31667,C1(C(=O)NC2CCC(CNC(=O)CC3(C)CCCO3)CC2)(OCC)CCCCC1 31668,N1(C(C(CC)C#N)=O)CC(C(=O)NCC2(O)CCN(C)C2)CC(C)C1 31669,c1(C(N2CC(C)N(C(c3cccnc3)=O)CC2)=O)cc2c(F)c(Cl)ccc2[nH]1 31670,C1(C(=O)NC(CC)C(C)O)CC(F)CN(C(c2ccc(C(F)(F)F)cc2)=O)C1 31671,C1(CNC(CSSC)=O)CCN(C(=O)C(C)Sc2ccc(N)cc2)C1(C)C 31672,c1(C(=O)Nc2nc(C3CCC(F)(F)CC3)cs2)ccc2c(c1)NS(=O)(=O)C2 31673,c1(C(=O)NC2CCCC(N(C(CCC(=C)C)=O)C)C2)cnc(O)c(OC)c1 31674,C1(NC(C2CC(N(C(CN(CCC)C(C)=O)=O)C)C2)=O)C(C)C1C 31675,N1(Cc2cc(C(=O)OCC)on2)CC(NC(C2(CC)CC2)=O)CCC1C 31676,CCC(O)C(C)C(=O)N(C1CCCCC1NC(=O)CC(C)SC)C 31677,c1(C(=O)OC(c2ncc(Br)cn2)C)cc(Cl)c(N)c([N+](=O)[O-])c1 31678,c1(C(=O)NCC2N(C(C(C)n3ccnc3)=O)CC=C2)nn(C)c(Cl)c1Cl 31679,N1(C(C2(C)CCCCO2)=O)CCOC2(C1)CN(C(=O)Cn1ccnn1)C2 31680,C1(CCC(=O)N(CC(C)NC(C2CSC2)=O)C)CC(C)(C)CO1 31681,C(C)(CNC(=O)C(C)(C)n1cccn1)(C(C)C)NC(c1cnc(CC)s1)=O 31682,C1(NC(C2(CNC(C3CN4CCN3CC4)=O)CCCO2)=O)CC1C1CCCCC1 31683,Cc1oc(-c2ccccc2)nc1C(=O)NC1CC(NC(C2CC(C)OC2=O)=O)C1 31684,Cn1nccc1COCC(=O)NCC1CCC1NC(c1csc(Cl)n1)=O 31685,N1(C(C(C)C)=O)CC=CC1CNC(=O)CCC1(OCc2ccccc2)CCC1 31686,Cn1cc(CC(=O)NC2COCC2NC(c2cnns2)=O)cn1 31687,CC1CN(C(C2CC23CC(C)(C)C3)=O)CC2(CCN(c3ncnc(Cl)c3Cl)C2)O1 31688,C(=O)(C(F)C(F)(F)F)NCC1(NC(c2c(NC)nccc2)=O)CC1 31689,C12(NC(=O)CSCc3ccccc3)CCCC1N(C(=O)COc1cn[nH]c1)CC2 31690,C(CC1=CCCCCC1)NC(C(C)NC(C(C)NC(=O)C1CC1)=O)=O 31691,C(CCCC(=O)N(C(C)CCC(C)C)C)NC(C(COCC)C)=O 31692,c1(OC)c(C(=O)NC2CCN(C(c3cc(C(C)(C)C)[nH]c3C)=O)C2)ncnc1C 31693,c1(C(=O)NCC2CCC(NC(C3(CCCC)CC3)=O)C2)[nH]nc2ncnc(O)c12 31694,C12(NC(C=CC)=O)CCCC1N(C(=O)CC1CC1)CC2.c12ccc(C)cc1NC2 31695,N1(C(Cc2n(C)ccn2)=O)CCCC(C2CN(C(c3cc(Cl)ncc3F)=O)C2)C1 31696,Cc1ccc(C(=O)NC2CC(NC(=O)C(C(C)C)N3CCCS3(=O)=O)C2)cc1 31697,C=C(C)C1CC(=O)N(C2CC2)C(C)C(=O)NO1.c1(C(N)=O)c[nH]ccc1=O 31698,c1(C(=O)NC(C(C)NC(CCCc2scc(C)n2)=O)C)c(C)c(Cl)cc(C)c1N 31699,C1(NC(=O)CSc2nc[nH]n2)CCC(CC(N2CCOC(CC3CC3)C2)=O)CC1 31700,C(C(=O)NCCC(=O)NC(N)=O)(C(C)C)N(C(C(CC)C)=O)CC 31701,c1(C(=O)NC(CC=C)CNC(c2c(C)ncn2O)=O)cc(Cl)ccc1OC 31702,C(=O)(CC(C)N(C)C(C1CC(O)C1)=O)NC(CN(CCCC)C)C 31703,C1(C(=O)NC2(CO)CN(C(CN(CCCCCC)C)=O)C2)CC=CCC1C 31704,N1(C(Cc2cnc(C)o2)=O)CC2CC(NC(c3c[nH]cc3Br)=O)CC1C2 31705,CC1CCCn2ncc(C(N3CCC(NC(c4cc5ncccn5n4)=O)C3)=O)c21 31706,Cc1cccn2c(C(=O)NC3(C)CC(NC(=O)C(F)CC4CC4)C3)cnc12 31707,C12(C(N3CC(CNC(c4ccc(C)cc4F)=O)OCC3)=O)CCOC1CCOC2 31708,C1(CNC(c2cc(OC)n(C)n2)=O)CC2(CC2)CN1C(=O)CCCc1cncs1 31709,Cc1oc2ccccc2c1C(N1CCCOC(CCNC(=O)C2=CCOC2)C1)=O 31710,N1(C(CC)=O)CCN(CCNC(=O)CC2(O)CCCOC2)CC1 31711,C(CN=C(NCCC(C)(C)O)NCCc1cccs1)n1ncc(C)c1 31712,N1(C(c2csc(C)n2)C(=O)NC(C(=O)OC)C)CCN(c2ccccc2O)CC1 31713,c1(C(=O)NC(C2CN(C(c3c(Cl)cc(C)s3)=O)C2)C)c(C)nc(C2CC2)nc1O 31714,c1(CC)[nH]c(=N)sc1C(=O)NC1CCCN(C(=O)CC2CCC23CCC3)C1 31715,CC1CN(C(C2CC23CC3)=O)CC(C)N(C(=O)C(C)Cc2ccccc2)C1 31716,C1(CNC(CCC=C(C)C)=O)CN(C(=O)CCC2CCN(C)C2)CC12CCC2 31717,C1(C(N2CCSCC2)=O)(CC)CCCN1C(=O)Cn1cnnc1O 31718,c1(C(=O)OC)cc(Br)cc(NC(C2CN(Cc3cncc(O)c3)CCO2)=O)c1Cl 31719,Cc1c(C(N2CCC(C)(N3CCCC3)C2)C(=O)NCC2CCCO2)cccc1Cl 31720,CC12CCOC(C(=O)NCC3CC(C(=O)NCC(=O)OCCO)CO3)(C1)C2 31721,C1(CNC(c2ccnn2CC(F)(F)F)=O)CN(C(=O)CCOCC(F)F)CC1O 31722,c1(C(=O)OC)cn(C)nc1OCCCOC1C=CCN(C(=O)OC(C)(C)C)C1 31723,c1(N(C(C(N)=O)C2CCCO2)C)ccc2nc(O)[nH]c2c1 31724,c1(OC)ccc(NC(=O)CC2CC(NC(=O)OC(C)(C)C)C2(C)C)c(O)c1 31725,c1(C(C)=O)cccc(OCC(N2CC(N(C(=O)Cc3ncc(C)s3)CCO)C2)=O)c1 31726,C(=O)(CC(O)CC(C)(C)C)NCC(CNC(CCCc1ccc(C)c(C)c1)=O)O 31727,c1(C(N(C)Cc2c(CNC(C3C(C)CCO3)=O)cccc2)=O)c(Cl)cncc1Cl 31728,c1(C(N(C)CCOCCNC(=O)CC2(C)CCCC2)=O)c(F)ccc2n[nH]cc12 31729,C1(C(=O)NC2C(CNC(=O)CSC(F)F)CCCC2)CCCCC(F)(F)C1 31730,Cc1cc([N+](=O)[O-])cnc1N1CC2CCN(C(=O)Oc3ccccc3)CC2C1 31731,C1(N(C(C(C2CCCC2)NC(C)=O)=O)C)CCN(C(c2ccc(C(C)=O)[nH]2)=O)C1 31732,c1(CC(N2CC(CC=C)(NC(=O)CC3CCC(O)C3)C2)=O)sc(C)cc1C 31733,Cc1cc(C#N)cnc1C(=O)NC1(C)CCCN(C(c2nc(Cl)cs2)=O)C1 31734,C12(C(=O)NC(CNC(c3ccnc(C)c3C)=O)(C)C)CCOC1CCOC2 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31752,CCC(C)(C(=O)NCC1CCN(C(C23CCC(O)(CC2)CC3)=O)C1)C(N)=O 31753,Cc1ccc(C(=O)NC2C(Cl)(Cl)C23CC3)cc1Br 31754,N1(C(C(C)CC2CCCCC2)=O)CCC(O)C(NC(=O)C=CC2CC2)C1 31755,C(C(C)(F)CNC(=O)C=CC(c1ccccc1)=O)NC(COCC(C)C)=O 31756,C12(NC(COCCCCOCC#C)=O)CCC(CN(C(c3cc(C)cs3)=O)C1)C2 31757,C1(CC(=O)NCC(=O)NCC)N(C(c2cc(C)[nH]c2C)=O)CCC1(C)C 31758,Cc1cnc(F)cc1C(=O)COC(C1CC(C(=O)O)C1)=O 31759,c1(C(=O)NC(C2CCOC2)CNC(c2ccc(C)nc2)=O)c[nH]cc(F)c1=O 31760,C(=O)(CC1CCOc2ccccc21)N1CC(O)(CCNC(CC(COC)C)=O)C1 31761,c1(C(N2CC(CC(N3C(C#N)CCC3)=O)C3(C2)CC3)=O)c[nH]c2ncccc12 31762,c1(C(N(C(CNC(Cc2c(C)ccc(F)c2)=O)C)C)=O)cccc(S(C)=O)c1 31763,CCC(C(=O)N(CCNC(=O)CC(c1ccc(Cl)cc1)O)C(C)C)C(C)(C)CC 31764,Cc1ncc(N)cc1C(N1CC(C2(NC(=O)Cn3cc(Cl)cn3)CC2)C1)=O 31765,C1(C(N2CC(C)C2c2ccccc2)=O)N(C(=O)C2=CCCCC2)CCC1(C)C 31766,CCC(CC)CC(=O)NC1CC(C(F)C(=O)Nc2c[nH]ccc2=O)C1 31767,Cc1cc(CNC(C2(C3CC3)CN(C(C3CCOC3(C)C)=O)C2)=O)ccc1O 31768,C1(NS(CC)(=O)=O)CCCN(c2nnc(-c3nn(C)cc3Br)n2C2CC2C)C1 31769,c1(OC)cccc(NC(C2(O)CCN(C(c3ccc(O)c(F)c3)=O)C2)=O)c1C 31770,N1(C(C23CC(NC(c4c(CCC)nco4)=O)(C2)C3)=O)CCC(O)CC12CC2 31771,CCC(O)CC(=O)N1CCCCC1Cn1cc(C2C3CCCCC23)nn1 31772,N1(C(CC2(C(=O)OC)CC2)=O)CCN(C(C2CSCCS2)=O)CC(C)(C)C1 31773,c1(CCC(=O)NC23CC(C2)N(C(c2ccncc2)=O)C3)cc(F)cc(F)c1 31774,N1(C(c2c(CC)[nH]c(=N)s2)=O)CC(F)(F)CC1CCNC(C12CC(CO1)C2)=O 31775,C1(CCN(C(=O)COC(c2ccccn2)=O)C)CCCCN1C(=O)C(C)(C)C 31776,CCC(CC)C(=O)NCC(=O)NCC1(C(=O)NC(C)Cn2cnnc2)CC(C)(C)C1 31777,N1(C(C(C2CCCC2)NC(c2ccn(C)c2)=O)=O)CCC(N2CCC2)CC1 31778,c1(CCC)nc(C)c(CN2CCC(N(C)C(C3CCOC(C)C3)=O)C2)o1 31779,c1(CC)ccc(C(=O)Cc2ccccc2)cc1C.C12CN(CC(OC)C1)C(=O)N2 31780,N1(C(C(F)OC)=O)CCC(O)(CNC(c2scnc2Cc2nccn2C)=O)CC1 31781,C(=O)(C(F)C(C)(F)F)N(CCCNC(CCC(=O)NCCCN(C)C)=O)CCO 31782,N1(C(CN2CC(C)C2)=O)CC(CNC(c2cnn(C3CCCC3)c2)=O)C(C)C1 31783,C1(NC(CSc2c(C)cno2)=O)CC2CN(C(=O)CN3CC(=O)NC3=O)CC12 31784,C1(N(C(C)C)CCN(C(=O)CCCNC(=O)C2CC2)C)CCCC(C)C1 31785,C1(NC(C(CCO)N(C)C)=O)CN(C(C2CCC=CCCC2)=O)C2(CCC2)C1 31786,c1(OCC)cc(C(=O)N(CC(O)CN(C(=O)CCc2cc[nH]n2)C)C)on1 31787,N1(C(CCCCC#C)=O)CC(C)CN(c2cc(=O)n(C)c(O)n2)C(C)C1 31788,C1(NC(C(C)OCC#C)=O)CCN(C(c2cnc(C(C)(C)C)nc2)=O)C1C(C)C 31789,c1(C(=O)NCC2CCN(C(CN3CC(CC)C3)=O)CC2C)csc(=NC2CC2)[nH]1 31790,C1(C(C)C#N)CCN(C(c2cc(CNC(c3nonc3N)=O)[nH]n2)=O)CC1 31791,N1(C(C=CCC)=O)CCC(C2CC2)(CNC(c2ccc(Cl)s2)=O)C1 31792,Cc1ccn(C)c1C(=O)NC1CC1NC(C1(C2CCCCC2)CCOCC1)=O 31793,Cc1cccnc1CN1C(CNC(c2cncc(NS(C)(=O)=O)c2)=O)COCC1 31794,N1(c2nc(SC)c(C)cn2)CCC2(CCN(C(=O)CCC3CCC3)C2)C1 31795,C(=O)(C1CCc2c(Cl)cccc21)NC(C)CNC(c1ccc([N+](=O)[O-])cc1F)=O 31796,c1(C(C)(C)C)ccoc1NC(C1(NC(=O)CSC2CCCCO2)CCCC1)=O 31797,C1(NC(Cc2ccc(CC)cc2)=O)CC2(C1)CC2N=c1[nH]c2cccc(C)c2o1 31798,C1(CC)CN(CC)CCN1C(c1cccc(CNC(=O)C#CC(C)(C)O)n1)=O 31799,CCCCC(C(=O)NC1CC(CCO)C1)NC(=O)C=CCCC(C)C 31800,C1(NC(C2CC2CF)=O)CC2CC1N(C(=O)Cn1ccccc1=O)C2 31801,CC1N(C(c2cc(CNC(c3ccnn3C)=O)[nH]n2)=O)CCOC1(C)C 31802,c1(C(=O)NCCC(C)NC(=O)C(CO)N(C)C)cc(Cl)ccc1[N+](=O)[O-] 31803,C1(CNC(N2CCC(N(C(C)C)CC#N)CC2)=O)CCCC1S(C)(=O)=O 31804,C1(C(=O)NC(C(=O)NC)C(C)C)CC12CCN(C(=O)C(O)C(F)(F)F)C2 31805,N1(C(C(CSC)OC)=O)CC2CC(C(N3CCC(CSC(C)C)C3)=O)C(C2)C1 31806,CCC(C#N)CNC(=O)COCCNC(=O)COCC1CCOC1 31807,N1(C(CCC=CCC=C)=O)CC(F)(F)CC1C(=O)NC(c1ccc(C)s1)C 31808,c1(C(N2CCC(C)(CNC(C(CCSC)O)=O)C2)=O)sc2nnc(S)n2c1C 31809,c1(NC(=O)NCC2CC2Nc2ccc(C(F)F)cn2)ccc(Br)cn1 31810,C(C)(C(CC(=O)NCc1ccc(C#N)s1)NC(C1CCC(C)(C)C1)=O)OC 31811,C(=O)(C(F)(F)CCn1ccnn1)NCCC(C(C)C)NC(c1ncccc1O)=O 31812,n1(CC)cc(C(N2CCN(CCO)C(C)C2)=O)c(=O)c2cc(Br)ccc12 31813,c1(C(=O)NC2(C)CCCC2C)ncccc1CNC(COC(C)=O)=O 31814,c1(OCC(=O)NCC(CNC(=O)CC2CCC(O)C2)OC)ccc(C)c(C)c1 31815,CC(C)CC(F)(F)C(=O)NCC12CC(NC(=O)CCCN3C(=O)CCC3=O)(C1)C2 31816,C(CCCCC(=O)N(CCC(=O)NCCc1cnccc1C)C)NC(C)=O 31817,C1(NC(CCCC#CC)=O)CCN(C(=O)CC2CCCCO2)C12CCC2 31818,c1(CCCC(=O)NC2CC(NC(C3CCCCC3O)=O)C2)ccc(O)cc1 31819,CC1CCN(C(c2ccnc(-n3cccc3)c2)=O)C1CNC(=O)C(C)CO 31820,C(CC(C(=O)NCc1ncc(C(N2CCOC(C(C)C)C2)=O)cn1)OC)OC 31821,C(CC(=O)NCCCCCNC(C1CS(=O)(=O)C1)=O)(C1CC1)NC(=O)OC(C)(C)C 31822,Cc1ccncc1CC(=O)NCC1(C)CCC(NC(=O)CCc2cccs2)C1 31823,N1(C(=O)CN2CCC(F)CC2)CCC2(CCN(C(=O)C3=CC4C=CC3C4)C2)C1 31824,C1(NC(C2CCC(NC(=O)OC)CC2)=O)CN(C(=O)CC2CCCC2)CC2CC12 31825,N1(C(C(C)C2CCCC2)=O)CC(CC(=O)NC2CCCCCC2F)CC1(C)C 31826,c1(C(=O)NC(C2(CNC(CCOCCOC)=O)CC2)C)cnc(C)s1 31827,c1(OC)ncc(-c2cncc(C(=O)NCC3CCCC3CO)c2)c(SC)n1 31828,c1(CC(=O)NCC2CCCN(C(=O)C(c3ccc(F)cc3)O)C2)cccnc1Cl 31829,O=S(=O)(C1CCCCC1)NC1CN(c2ccccc2)C1.C12CCCN1CC2 31830,CC(C)CC(O)CC(=O)N1CCCCCC1C(N1CC(N(C)C)C1)=O 31831,c1(C(=O)NCC(=C)CCNC(C2CCS2(=O)=O)=O)cccc2c1NC(=O)CC2 31832,C1(NC(C=CC(=O)OCC)=O)CCCCCC1C(=O)Nc1cc(C)ccc1OC 31833,C(=O)(C1OC(=O)c2ccccc21)N1CCC2(C(NC(c3c(C)occ3)=O)C2)CC1 31834,C1(CC(N2CCC(C(C)NC(C3CC(=O)C3)=O)CC2)=O)CCCC(F)(F)C1 31835,CC(C)CC(C(=O)NOC(c1ncccn1)C)ONC(C1CCCC1)=O 31836,CC(C)C(O)C(=O)NC1(CF)CCN(C(=O)CCc2csc(Br)c2)C1 31837,C1(CCCCCNC(C2CC2F)=O)CCN(C(C2CCC(F)C2)=O)CC1 31838,CS(=O)(=O)c1ccc(C(=O)NC2CC23CCN(C(=O)C2=COCC2)CC3)s1 31839,c1(C(=O)NC2CCCN(C(C3CC(SC)C3)=O)C2)n[nH]c2cc(C)ccc12 31840,c1(C(=O)NCC(CC)NC(=O)CSc2nnnn2C)cccc(N2CCCC2)n1 31841,CCC(CCCC(=O)NCc1nc(C)c(C)[nH]1)NC(=O)CN(C1CC1)CC 31842,CC1CNC(=O)CN1C(C1CC12CCN(C(=O)CN1CC3CC3C1)C2)=O 31843,N1(C(CC(COC)(C)C)=O)CC2CC(O)C1C2NC(=O)CCC1CCCO1 31844,N1(C(c2cnccn2)=O)CCC(C2(NC(C3CN(C4CCOC4)C3)=O)CC2)CC1 31845,Cc1nsc(N2CC(F)(F)CC2CNC(c2cn(C3CCC3)nc2C)=O)c1C#N 31846,c1(COC(N2CCN(C(CC(C)C)=O)CC2)=O)cccc2c1OCCC2CCO 31847,N1(C(CC(C(=O)OC)C)=O)CCC2C(C1)CN2C(=O)Cn1cc([N+](=O)[O-])c(C)n1 31848,C=C(Cl)C(C)(C)C(=O)NCC1(NC(=O)C(C)OCC(C)C)CCCCCC1 31849,C1(C(N(C)Cc2ncnn2C)=O)CCN(C(=O)C2=CCCSC2)CCO1 31850,C1(C(=O)NCC(C)CNC(=O)CNCc2cccnc2)C2COCC12 31851,c1(CCC)cnnc(C(=O)NC2CCC2NC(=O)CCC(C)C)c1 31852,c1(C(=O)NC(CNC)C(C)(C)C)cc2cccnn2c1 31853,N1(C(C(C(CC)C)O)=O)CCCC12CCCN(C(=O)CCN(C)C)CC2 31854,C1(CC(N)=O)(NC(=O)CCN2CCC(F)(F)C2)CCCN(C(=O)CC2CCC2)C1 31855,C12(CNC(c3cc(Cl)no3)=O)CCCC1CN(C(C13CCC(CF)(C1)OC3)=O)C2 31856,C1(CNC(=O)COCC2CC2)CC(NC(C2(C(F)F)CCC2)=O)C1 31857,CCC(C)(CC)CN=c1nc(N2CCC(n3cncn3)C2)c2[nH]ccc2[nH]1 31858,N1(C(CN2CCN(C(=O)Cc3cc(Cl)c[nH]3)CC2)=O)CC(CO)OC(C2CC2)C1 31859,C(C(F)(C(=O)NCCC(O)C(C)C)C(C)C)NC(C(=Cc1ccccc1)C)=O 31860,C(=O)(C(O)CCCNC(=O)CC1(N(C)C)CCC1)NC1C(CCC)C1 31861,C(=O)(C1COc2ccccc21)NCC1CN(C(CCCC)=O)C2C(O1)CCC2 31862,N1(C(C2C(C)(C)C(NC(=O)CCCC3CCC3)C2)=O)CCC2(CC1)CC2C#N 31863,N1(C(C=C(C)Cl)=O)CCC(C2CC2)(CNC(=O)C(C2CCOCC2)O)C1 31864,C1(C)(C(=O)NC2(CNC(C(COC)(C)C)=O)CCCCCC2)CC(C)OC(C)C1 31865,C1(NC(c2ccc(F)s2)=O)CC(O)CN(C(=O)C2=CCCS2)C1 31866,CCC(C)C(C)C(=O)NCCCN(C(c1ncc(C)cn1)=O)C1CC1 31867,c1(CC)cc(NC(C2(F)CCN(C(c3cc(Br)ccc3F)=O)CC2)=O)ccc1F 31868,C(C1CN(C(=O)C(C)C2CCC2)CC1C(=O)NC(C)C(F)(F)F)=CC 31869,c1(N(C)Cc2ccns2)nc(N2CCCC(CCO)CC2)c2c(n1)CSC2.C1CC1 31870,C(=O)(C(CCC1CCC1)NC(c1cnc(C2CC2)o1)=O)Nc1c(C)csc1 31871,N1(c2nc(C)cc(OCC)n2)Cc2nccn2CC(NC(c2coc(C)c2)=O)C1 31872,Cc1ccc(O)c(C(=O)NC2CC(OCC(N3CCCC(F)(F)C3)=O)C2)c1 31873,c1(C(=O)NC(CNC(c2c(C)ccnc2)=O)(C)C(C)C)onc2c1CCCC2 31874,CC(C)(C)C(O)CNC(=O)NCC(COC(=O)Nc1ccccc1)(C)F 31875,S(=O)(=O)(c1ccc(Br)cc1NC(C)CCSC)NC(C=C)COC 31876,CC1CC(NC(=O)CCCN2CCCCC2)CN(C(c2coc(C#N)c2)=O)C1 31877,C(=O)(C=C1SCC(=O)N1C)NCC12C(CN(C(c3c(C)c(Cl)ccn3)=O)C1)CC2 31878,Cc1nc2cc(C(=O)NCC3CC3NC(=O)CC3(CO)CC3)cc(Br)c2o1 31879,Cc1noc(C(=O)OCC(=O)NC2CCC(C)(C)C2)c1I 31880,Cc1cc(C(N2CCN(CC(=O)NCC3CNC(=O)C3)CC2)=O)oc1C 31881,N1(C(c2c(C)cc(CC)o2)=O)CC2(CCN(C(c3c(C)cnn3C(C)C)=O)C2)C1 31882,CCC(C)(C(=O)NCC1CN(C(=O)CCc2cc(Cl)no2)CCC1(F)F)C(F)F 31883,C(=O)(C(C)(CNC(=O)CC(CC)C1CCC1)CC)NC(CCCC)C 31884,C(=O)(C(C(C)CC)c1ccco1)N1CC(CNC(CCC)=O)(NC(C)=O)C1 31885,C1(NC(c2sc(CCC)c(CC)c2)=O)CCC(C)N(CCc2ccc(C)s2)C1 31886,C1(C(C)NC(Cc2c(C)cco2)=O)CCCN(C(=O)CCc2c(C)noc2Cl)C1 31887,N1(C(Cc2c(C#C)cccc2)=O)CCN(C(=O)CC2CC(=C)C2)C(C)C1C 31888,CCC(CCCC(=O)NCCCc1nncs1)NC(C1CCC(O)C1)=O 31889,c1(C(=O)NCCCN(C(=O)CC2CCN(C)C2=O)CC)cc(OC)c(Cl)s1 31890,N1(C(C2Cc3ccncc3C2)=O)CC2CCN(C(c3ncccn3)=O)C2C1 31891,CC1(C)COCCC1C(=O)NC(Cn1cncn1)C(N1CC2CC=CC1C2)=O 31892,c1(C(N2C(CNC(CCOCC(C)C)=O)CC3(CC3)C2)=O)nsc2ccccc12 31893,c1(CC)ccc(N)c(C(=O)NC(CNC(c2cc(O)n(CC)n2)=O)CCC)c1 31894,n1(CC)nncc1C(=O)NC12CC(CNC(=O)C(C3(O)CCCC3)F)(C1)C2 31895,C1(CC)CCC(NC(=O)C(Cn2ccnn2)NC(=O)C(C2CCOCC2)C)CC1 31896,c1(C(N2CCN(C(c3n(C)nc(C)c3F)=O)CC2)=O)ccc(C#N)nc1O 31897,c1(C(=O)NC(CNC(C(CC#C)C2CC2)=O)C(C)C)cc(F)cnc1OC 31898,c1(NC(C2C(NC(C3C(C)(C)OC(=O)C3)=O)C3CCC2C3)=O)cc[nH]c2nccc1-2 31899,Cc1cccnc1C(=O)NCC1(C(=O)NCC(c2nccs2)C)CC2(CC2)C1 31900,n1(C(C)C)ncc(F)c1C(=O)NC1CCCC1CNC(=O)C(c1ccccc1)C 31901,C1(NC(c2ccc(F)cn2)=O)CN(C(c2cccc[n+]2[O-])=O)CC1O 31902,N1(C(C2(SCC)CCC2)=O)CCC(N(C(=O)Cc2cccc(CO)c2)CC)CC1 31903,Cc1cnc2n1CCC(C(=O)NCCN(C(=O)C1=CCCS1)C)C2 31904,N1(C(C23OCC(C)(C2)C3)=O)CC=C(CNC(=O)Cc2cccnc2)CC1 31905,N1(C(c2ccnc3c2CCC3)=O)CCN(C(C2CCC(O)C2)=O)C2(CCC2)C1 31906,C1(NC(COCCCC)=O)CC2CCC(C1C)N2C(C12CC(CO1)C2)=O 31907,c1(NCC2CN(C(C3CCc4nccn4C3)=O)C2)ncc([N+](=O)[O-])cc1F 31908,CC1CCN(C(=O)CN2CCCCCC2)CC1NC(=O)CC1CC=CCC1 31909,CC(CC(=O)N(C)CC1CCCN(C(C23CCC(C2)C3(C)C)=O)C1)CC(C)(C)C 31910,c1(CC(=O)N(C(CCNC(C(COC)COC)=O)C)C)cnn2ccccc12 31911,C1(OCCCNC(C(C)c2ccco2)=O)CCN(C(c2c[nH]ccc2=O)=O)CC1 31912,CCCC(C)(O)C(=O)NCC(C)(C)CNC(c1ccnc(SC2CCCC2)c1)=O 31913,N1(C(C2CCC(=O)CC2)=O)CCC2CCCC12C(=O)NOCC1CCOC1 31914,C(=O)(C(C)(C)C(N)=O)N1CCC(CC(C)NC(c2nc(=O)n(C)[nH]2)=O)CC1 31915,C1(CC(N2CC(C)(NC(=O)CCCn3cncn3)C2)=O)CCCCC1O 31916,N1(C(c2cc(N)cc(F)c2)=O)CCC(C2CC2)(CNC(c2ccc(CO)nc2)=O)C1 31917,CC(C)CCCC(C)C(=O)N(C1CCN(C(=O)C=CCO)CC1)CC1CCCO1 31918,c1(C(=O)NC2CN(c3ncc4sccc4n3)CC2F)cc(Br)cc2[nH]ccc12 31919,Cc1ncccc1CC(=O)NC1CC(NC(=O)CC2COC(C)(C)C2)C1 31920,C1(OCC(N2CCN(C3CC(C)OC3=O)CC2)=O)CCC(F)(F)CC1 31921,C(CC(CC)C(=O)N1CCN(C(=O)Cc2ccco2)CC1)=CC 31922,c1(NCCN2CCN(c3cc(COC)ncn3)CC2)ccccc1S(=O)CCC 31923,c1(C(=O)NC2(C(F)F)CC(NC(c3ccc[n+]([O-])c3)=O)C2)cnc2n1CCCC2 31924,c1(C(N2CC3CN(C(c4scc(OC)c4)=O)C3CC2)=O)[nH]cc2c1CCS2(=O)=O 31925,CC(=O)C(C)(C)CC(=O)N1CCC(C(=O)NCC2CCOC2C(C)C)C1(C)C 31926,N1(C(C2(SC)CC2)=O)CC2CC1CC2NC(=O)Cc1c[nH]nc1C 31927,c1(NC(N(CCCC#C)Cc2cccc(Br)c2)=O)ccc(C#N)c(C)n1 31928,c1(C(=O)NCC(CNC(C=Cc2ccc(C)s2)=O)C)ccn2cnc(C)c2c1 31929,C1(NC(C(C)OCC=C)=O)C2CCN(C(c3sc(Br)cc3C)=O)C12 31930,c1(CC(=O)NCC2N(C(C(CCOC)C)=O)CC=C2)cn2c(C)csc2n1 31931,N1(C(CNS(C)(=O)=O)=O)CCCC1CC(=O)NCCOCCN(C)C 31932,Cc1ccnc(C(=O)NCC(C)(C)CCNC(=O)CN2CCOCC2)c1 31933,N1(C(c2c(CC)scn2)=O)CCC(C(C)(O)CNC(C2CCCO2)=O)CC1 31934,c1(C(N2C(CNC(Cc3ccc(C)cc3)=O)CC(F)C2)=O)cc(N)ccc1C 31935,N1(C(C2CC(=C)C2)=O)CCC(C2CCN(C(C3CC4CCC3O4)=O)CC2)CC1 31936,c1(NC(CC2N(C(C(CC)=O)=O)CCOC2)=O)nc(O)ccc1[N+](=O)[O-] 31937,C1(CCC(=O)N(CCN(C(=O)C(C)c2ncco2)C(C)C)C)CCC(=O)N1 31938,C1(C(C)C)(CNC(=O)C(Cc2ccoc2)NC(=O)CSCCC#N)CCCC1 31939,C(CC(C(=O)NC1CCCSCC1)NC(=O)C(C1CCOCC1)=O)OC 31940,c1(CS(C)(=O)=O)ccc(C(=O)NCCNC(C2CCOC2c2ccccc2)=O)o1 31941,N1(C(C(C)OCOC)=O)CC2CN(C(=O)C(C3CCCCC3)O)CC2(C)C1 31942,CC1CC(CNC(C2(C(F)F)CC2(F)F)=O)=NO1 31943,c1(N2C3(CNC(N4CCC5(CCOC5)C4)=O)CC3CC2)ncnn2ccc(Br)c12 31944,CC(Cc1nncn1C)N=c1[nH]c2c(c(=NCC3C4CCCCC34)[nH]1)CSC2 31945,c1(C(=O)NCC(C)N(C(c2cc(C)c(C)nn2)=O)C)ccc2ccccc2c1O 31946,Cc1cn2c(n1)CC(C(N1CC(NC(c3cc(N)cc(O)c3)=O)CC1C)=O)CC2 31947,C(=O)(C(O)CNC=O)NCC1(CCOC)CC1.n1(CC(=O)N)cnnn1 31948,c1(C(C)C)ccc(C(CNC(C2CC(C)(C)C2)=O)NC(=O)Cn2ccnn2)cc1 31949,C1(C(=O)Nc2cnc(OCC)c(Cl)c2)COCCC1C1CCNCC1 31950,C(=O)(C(C)S(=O)(=O)C(C)C)N1CCC(NC(c2cc(C)c(OC(F)F)cc2)=O)C1 31951,Cc1cc(C(=O)NCCOc2ccc(F)c(F)c2)c2ccc(Br)cc2n1 31952,C(=O)(CCCCn1ccnn1)NCC(C1CCOC1)NC(=O)C=CC(F)(F)F 31953,c1(C(=O)NC2(CO)CN(C(C(C)SCC)=O)C2)cc(OC)cc2c1OCC2 31954,C(=O)(CC(F)(F)C(F)F)NCC(CC=C)C(=O)N1CC2CC2C1 31955,C1(CCNC(C2CC(C)(F)C2)=O)CCN(C(c2ncoc2-c2ccco2)=O)CC1 31956,C(=O)(C(C)CC(F)(F)F)NCCCC(C)NC(C1(N2CCOCC2)CCCC1)=O 31957,N1(CCOC)C(=O)CC(CNCCCc2cccnc2)C1c1cnn(C)c1 31958,C#Cc1cncc(C(=O)NC23CC2CN(C(c2ccc(C)nc2C(C)C)=O)C3)c1 31959,C1(C(=O)NCCN(C(=O)C(O)c2cnc[nH]2)C2CC2)CCC(OC(F)(F)F)CC1 31960,C1(CNC(C(c2ccc(Cl)cc2)N(C)C)=O)COCCN(C(=O)CC(F)(F)F)C1 31961,C1(C(N(CCCCCNC(=O)CCCn2ccnc2)C)=O)CC2CCC1C2 31962,C1(NC(CC2CN(C)C2)=O)COC2(C1)CN(C(C1(F)CCOC1)=O)C2 31963,N1(C(C2(OCC)CC2)=O)CCC=C(C(=O)NCCSCC(C)C)C1 31964,c1(C(=O)NC(C(C)NC(C(COC)C)=O)CO)c(C)ccc(Cl)c1N 31965,c1(C(C(=O)NCCC#N)N(CCSCC)C)ccc(C(C)C)cc1F 31966,C1(CC(=O)NCC(C)CN(C)C(c2cc(Cl)c(Cl)[nH]2)=O)CCCC(F)(F)C1 31967,CCC1=NOC(CNC(C2C3CC2N(C(=O)CC(C)c2ccco2)C3)=O)C1 31968,c1(N(C)C)cccc(N2CCN(CN3CC(C)OCC3)CC2)c1.C(C)(C)(C)S 31969,N1(C(C(CC)C#N)=O)CC(C2CCCN(C(c3cc(OC)ns3)=O)C2)C1 31970,CCC(CC(C)C)C(=O)NC(C)CN(C)C(c1cn(-c2ccccc2)nn1)=O 31971,C1(C(N2CC(C(N3CCC(C(F)F)C3)=O)(COC)C2)=O)COCC(C)O1 31972,c1(C(=O)NC2C3CN(C(C4C(C)=CCS4)=O)CC2C3)cc2cccc(C)c2o1 31973,c1(NC(C2CCC(CNC(C3(O)CCC3)=O)O2)=O)cncc(F)c1 31974,C(CCCCNC(=O)CCC1CC1)N(C)C(C1SCCS1)=O 31975,CC1(C)CCC(C(=O)NCc2ncoc2CNC(=O)CC2CC3CCC2C3)CC1 31976,C=CCN=C(NCc1nnc(-c2ccccc2)s1)N1CCC(OC)C1 31977,C(=O)(C1=CCS(=O)(=O)C1)NC(C(C)C)CCOC(F)(F)F 31978,n1(CCC(N2C3(CC)CC(NC(=O)OC(C)(C)C)(C2)C3)=O)cc(Br)c(O)nc1=O 31979,n1(CC)nc(C(N2CC(F)(C(=O)NC(C)CCC(C)C)C2)=O)cc1C 31980,Cc1oc(C(C)C)nc1C(=O)N(CC(O)CN(C(=O)C=Cc1ccncn1)C)C 31981,c1(C(N2CCSCC2CCO)=O)cnc2c[nH]nc2c1 31982,C1(NC(c2ccon2)=O)CCC2CCN(C(=O)C#CC3CCCCO3)C1C2 31983,N1(C(C(COC)C)=O)CC(C)C(C)(C(=O)N(C(C(N)=O)C2CC2)C)C1 31984,C(=O)(C1CCCc2scnc21)NCC1CN(C(CCCCC(=O)NC)=O)CC1C 31985,CCCCCC(C)CC(=O)NC1(CO)CN(C(C2(C)CCOC23CC3(F)F)=O)C1 31986,c1(C(C2CC2)OC)ccc(Cl)c(Cl)c1C.c12nc(no1)CS2 31987,C(=O)(CC(C)C(=O)NC1C=CC(CNC(C2CC2C(F)F)=O)C1)OC 31988,C1(C(=O)OCC)CC2(CCN2C(c2nc(Br)cs2)C(=O)NCC(F)F)C1(C)C 31989,C1(CNC(c2ncc(OC)cn2)=O)CC(C(F)(F)F)CCN1C(=O)C(C)O 31990,N1(C(C(CC(C)C)F)=O)CC2CCN(C(=O)Cc3cc(C4CC4)nn3C)CC12 31991,c1(CN(C(CNC(C2C(C)C2)=O)C)C(c2cccc(CF)c2)=O)cccc(Cl)c1 31992,C1(C(=O)NC(C(C)C)(C)CNC(=O)Cc2cnsc2)CCc2nncn2CC1 31993,C1(C(=O)NCCC)C(C(=O)N(CCCN(C)C(C23CC(C)C2C3)=O)C)C1(C)C 31994,CC1CN(C(=O)C(O)Cc2cnc[nH]2)CC1P(C)(C)=O 31995,c1(CC(=O)NCCC(=O)NCCC(C)C)ccc(F)cc1F 31996,C(=O)(CCC(=O)C1CC1)NC1CCN(C(CSCC(N)=O)=O)C1.C1CS1 31997,N1(C(C(C)OC(C)(C)C)=O)CCN(C(c2cccnc2)=O)C(CC(F)(F)F)C1 31998,N1(C(c2ncc(C)cn2)=O)CC2CCC1C(CNC(c1ccc(F)c(Cl)c1)=O)C2 31999,N1(C(CC(C)OC)=O)CC2(C1)CN(C(C1CCn3nncc3C1)=O)CCO2 32000,C(=O)(C(C)CC(C)C)NC(CNC(c1cccc(C(=O)NC)n1)=O)C 32001,CN1C(=O)CC(N2CC(CNC(=O)NCCS(C)(=O)=O)C2)C1=O 32002,c1(C(N2CC(O)CC(NC(=O)C(F)F)C2)=O)ccc2c(c1)CCO2 32003,C=CCCCCCC(=O)N1CCCC1(C(=O)NCC1CN2CCC1C2)COC 32004,c1(NC(N2C(C)CCC(C(=O)NCCOCCO)C2)=O)ccc(S(C)(=O)=O)cc1 32005,c1(COC(C)C(N2CCCC2CN(C(=O)Cn2cc(Cl)cn2)C)=O)ccccc1 32006,C1(=O)CCCCCNC2C(C)CN1C2.c1(NC(=O)CC2CC(F)C2)ccccc1 32007,N1(C(CC(C)F)=O)Cc2ccccc2CC1CNC(C1(CCN(C)C)CC1)=O 32008,c1(CC)ccc(Cl)cc1NC(C1CCCN(C(C2CC2c2ccccc2)=O)C1)=O 32009,c1(N(c2ccccc2)CC)ncccc1S(=O)(=O)N(C1CNC1)C.C(CS)OC 32010,Cc1ccn(CC(=O)NC(C)(C)C(C)NC(=O)CNC(=O)CN(C)C)n1 32011,CC1CCc2[nH]nc(C(=O)NC34CCCC3CN(C(=O)CCCC(N)=O)C4)c2C1 32012,N1(C(c2c(CC)c[nH]n2)=O)CC=CC(NC(=O)COC)C1 32013,c1(Nc2cccc(-c3c[nH]c(=NCc4ccc(Br)cc4)s3)n2)ccc2c(n1)CCC2 32014,C1(NC(Cn2c(C)nc(C)n2)=O)CC2(C1)CC(C(=O)NC1CCC(N(C)C)C1)C2 32015,c1(OC)ccc(F)c(F)c1CN1CCOC(C(=O)Nc2ccc(C#N)cc2O)C1 32016,C1(C(N2CCCC(CNc3ncc([N+](=O)[O-])cn3)CC2)=O)CCC2CCCCN12 32017,c1(C(=O)NC2(C(=O)NCCOc3ccc(C)cc3)CC(=C)C2)ccc(C#N)cc1 32018,Cc1cc(C(N2CCCC(C(N3CCCCC(CO)C3)=O)CC2)=O)c(O)nn1 32019,C(c1ccncc1)=C(C)C(=O)N(CCCNC(C1CCCCC1C)=O)C 32020,c1(CN2CCCC(CNC(c3ccc(C#C)cc3)=O)C2)ncnc2c1ccn2C 32021,C1(CNC(c2c(CC)cccc2)=O)CCN(C(C2CC(F)CN2C)=O)C12CC2 32022,N1(C(c2c(C)ocn2)=O)CC2C(CN(C(=O)CC3CC4CC4C3)C)C2C1 32023,CC1CN(C(C2(N(C)C)CCC2)=O)CC1CNC(=O)CN1CCC(F)CC1 32024,Cc1csc2nc(CC(N3CC(NC(C4(C(N)=O)CC4)=O)CCC3C)=O)cn12 32025,C1(C(=O)NC2CC(CNC(C(c3ccncc3)C)=O)C2)COCCN1C 32026,c1(OC)ccc2nc(CNC(C)(C)CCc3ccccn3)ccc2c1Br 32027,N1(C(Cn2c(C)nnn2)=O)CC(NC(c2cc(O)nc(Cl)c2)=O)CC(F)C1 32028,c1(C(=O)NC(CC)CN(C(=O)C(C)CF)C)ccc(OCCO)cc1 32029,C1(C(=O)NCC2(C)CN(C(=O)Cc3ccc(F)cc3)C2)C2CCC(F)C12 32030,c1(NC(C2N(CC)CCCCC2)=O)[nH]c2ccccc2c1C(=O)OC 32031,C(=O)(C1=CC2C=CC1C2)N(CCCCCNC(=O)CCC1CCCOC1)C 32032,N1(C(c2ccc(C(N)=O)o2)=O)CC2(CC(NC(=O)CCc3csnn3)C2)C1 32033,C12(C(=O)NCc3ccc(C)cc3C)C3CCC(CC13)C2(F)F 32034,c1(C(=O)NCCCC(C)NC(c2c(OC)noc2C)=O)ccc2ncsc2c1 32035,c1(SCC)ccc(NC(=O)NCC2(OCC)CCOC2)o1 32036,C1(C)(CC)C=C(C(=O)N2CC3CC3(C(N3CCC(N4CC=CC4)C3)=O)C2)C1 32037,C(CCC(C)C)C(=O)NOCCCCC.C=C=CC(C)C=O 32038,C1(C(N(C)CC2N(C(Cc3cccc(C)c3)=O)CCOC2)=O)CC(C(C)C)=NO1 32039,CCCCCS(=O)(=O)CC(=O)NCC(C)NC(=O)C#CC1CCCCC1 32040,c1(C(=O)OC)ncc[nH]c1=NC1CCCC(NC(C2CCOCC2)=O)C1 32041,C1(NC(C(CC(C)C)O)=O)COC2(C1)CN(C(=O)Cc1c(F)cccc1C#N)C2 32042,C(=O)(C(CNC(=O)CC1CSC1)CC(C)C)NC(C#C)(C)C1CCC1 32043,CC1(CNC(=O)CCC2NC(=O)NC2=O)CCN(C(=O)COC(F)F)C1 32044,N1(C(c2nc(OC)c(C)s2)C(=O)NCC2CCOC2)CCCC2CCC(C)CC12 32045,C(C(CC(F)(F)F)NC(c1cnc(O)o1)=O)NC(CCC1CCC(=O)NC1)=O 32046,N1(C(CCN(C(c2ccoc2C(F)(F)F)=O)CC)=O)CCCC(CN(C)C)C1 32047,c1(CC)c(C(=O)NCCC2(NC(c3cc(N)ccc3C)=O)CC2)cccc1C 32048,N1(CC(N2CCCC2)=O)CCCCC1=O.N12CCCC(C1)NC(C)(C)C2 32049,c1(C(=O)NCC2(NC(c3c(CC)nccc3)=O)CC2)cc(O)ccc1C 32050,N1(C(C2=C(C)CCC2)=O)CC(NC(=O)COCCCF)C(C2CC2)C1 32051,c1(C(N2CC(NC(C3(C#C)CCC3)=O)C(O)C2)=O)cc(F)ncc1OC 32052,c1(C(=O)NCC(C)C#N)cnc(CNC(C2CC2(Cl)Cl)=O)nc1 32053,c1(CC(=O)NCC2(C)N(C(C(CC#C)C)=O)CCC2)ccc(Br)cc1CC 32054,CC1(C)OCCOC1C(=O)NCCC1CCN(C(=O)CN(C2CCCC2)C)CC1 32055,CCC(C)(C)CCCC(=O)NCC1(C(=O)NOC2CCCC2)CC12CCC2 32056,CC(C)(CCCNC(=O)C(O)CC1CCCC1)C(=O)NCC1(C2(O)CCC2)CC1 32057,C(CN=S(C)(C)=O)N(C)C(c1csc(C(=O)OC(C)(C)C)n1)=O 32058,CN1CCC(C2(C(N3CC(CNC(c4ccc(Cl)o4)=O)C3)=O)CC2)CC1 32059,C1(C(N2C(CC(=O)OC)CCC2)=O)CCCN(C(C2CC2(Cl)Cl)=O)C1C 32060,C#Cc1cccc(C(N2CCSCC2C(=O)N(C)C(C)C2CC2)=O)c1 32061,C(=O)(C1=C(C)NC2=NCCCC2=C1)NCC1N(C(COCCCCC)=O)CC1 32062,CC1CC(NC(C2(c3ccccc3)CCC2)=O)CCN1C(=O)CSC1CC1 32063,N1(C(C2CN(C(C3N(C)C(=O)CC3)=O)CC(F)(F)C2)=O)CCN2CCOCC2C1 32064,c1(CC(=O)N(C2CN(C(c3nonc3N)=O)CC2F)C)cncnc1O 32065,C(=O)(CC(O)CC1CC1)NC(CNC(CCSCCC)=O)C(C)C 32066,c1(CC)ccc(C(=O)N(C2CN(C(=O)COC)CC2F)C)cn1 32067,c1(N2CCC(C)(CO)C2)ccc(S(=O)(=O)NC2(CO)CCC2)cc1Br 32068,C1(C(=O)NCC23CC2CN(C(=O)CCC2CCCCC2)C3)C2CCCCCC12 32069,c1(C(=O)NC(CNC(C(C)=CC)=O)(C)C2CC2)cc(C)c(-c2ccc(Cl)cc2)s1 32070,C1(CC#C)(C(=O)N(C(=O)CCC=C=C)CCCCC)CCCCO1 32071,n1(CC)ccc(=NC(=O)C2COC(C)(C)CN2)[nH]1 32072,c1(C(=O)NCC(C)N(C)C(C(C)C(N2CCCCC2)=O)=O)[nH]ccc1C1CC1 32073,c1(C(C(=O)NCCCCNC(C(SC)SC)=O)F)ccccc1 32074,CC(=O)CCCC(C)C(=O)N1CC(C)CC1C(N1CCC(N(C)CCO)C1)=O 32075,C(=O)(C(C(C)C)n1cncn1)N(CC(CNC(C(CC)n1cncn1)=O)(C)C)C 32076,C(=O)(C(O)CC(F)F)NC(CCNC(CCc1cnc(C)o1)=O)C 32077,c1(NC(C2CN(C(c3ccccc3O)=O)CCC2O)=O)ccc(F)c(Br)c1F 32078,C1(CNC(=O)NC(c2ccc(SC)cc2)C)CCCCC(F)(F)C1 32079,N1(C(c2cc(CCC)[nH]n2)=O)CCC(C)C(NC(c2ncc(N(C)C)cn2)=O)C1 32080,C1(O)(CC(=O)N(C2C(OC)CN(C(CN(C(=O)OC)C)=O)C2)C2CC2)COC(C)(C)C1 32081,C1(C(=O)NC2CCN(c3ccc([N+](=O)[O-])cc3)C2)CCCC2(C1)CC2(F)F 32082,CC(C)C(C(=O)NC1CCOC1C(=O)N(C)Cc1ccnn1C)n1cccc1 32083,C(C(C)(C)CNC(C1(Cl)CC1(F)F)=O)N(C(=O)CCCc1cccs1)C 32084,c1(C(N2CC(C)(NC(C(C=C=C)C)=O)C2)=O)ccc(C(=O)N(C)C)nc1C 32085,c1(C(C)NC(=O)NCC(C)(C)C(F)F)ccc(-n2cccn2)c(F)c1 32086,C(C)(CCCNC(=O)C(F)(F)c1nccs1)NC(C(C)NC(C)=O)=O 32087,C12(C(=O)NC(CCCCC)C)CCC(CN(C(c3n[nH]c(C)c3O)=O)C1)C2 32088,Cc1c(C=CC(=O)NC2CC(C)(NC(c3ccc(Br)cc3O)=O)C2)cnn1C 32089,Nc1ccc(-c2cn(C3CC(NC(=O)CCc4nc(Cl)n[nH]4)C3)nn2)nc1 32090,C1(CNC(c2coc(O)n2)=O)CC(O)CN1C(=O)Cc1ccsn1 32091,C(=O)(CCC(=O)N(C)CCN(C(=O)C(C)(F)CC1CC1)C)N(C(C)C)C 32092,CCC(CC)(CC)C(=O)NC1CC2CC1N(C(C1CC1c1ccccc1Cl)=O)C2 32093,c1(OCCC)c(Cl)cc(NC(c2cnc(OC)c(F)c2)=O)cc1Cl 32094,Cc1c(NS(C)(=O)=O)cccc1N=c1cc(N)nc(-c2ccccc2)[nH]1 32095,CC(C)S(=O)(=O)CC(=O)NCC1(CNC(C2CCCO2)=O)CCC1 32096,c1(C(=O)NCCCC(C)NC(=O)C(F)OC(F)(F)F)cncc(C2CC2)c1 32097,C1(CNC(CCCC=C)=O)CC2CCC1N(C(=O)Cc1cc(C)cs1)C2 32098,C1(CNC(C2CC(C)OC2C)=O)(CO)CCN(C(C2(CO)CCC2)=O)CC1 32099,C1(CNC(=O)CCN(C(c2cn(C3CC3)cn2)=O)CC2CC2)CCOC1=O 32100,c1(CN2CCC(NC(=O)Cc3cc(Cl)ccc3Cl)C(O)C2)cncc2ccccc12 32101,C1(NC(C(CC(C)C)N(C)C)=O)COC2(C1)CN(C(=O)Cc1ccncc1Cl)C2 32102,CC1(C)CC(NC(=O)C(O)C(C)(C)C)CCN(C(=O)CSC(C)(C)C)C1 32103,C1(CCNC(=O)Cn2cccc2)CCCN(C(c2sc(Cl)cc2Cl)=O)C1 32104,c1(C(N2CC(CC(C#C)C)C2)=O)cc(F)c(C)cc1Cl 32105,N(C1CCc2ccccc21)C(C12CC(Nc3nccc(Br)n3)(C1)C2)=O 32106,C1(C(C)C)CCC(C(=O)NC(C)CCNC(=O)CCC(C)N(C)C)CC1 32107,C(=O)(C(F)(F)C(C)O)NC(CNC(c1c(C(=O)OC)nn(C)n1)=O)C(C)(C)C 32108,Cc1cn2cc(C(=O)NCC3(NC(=O)C(C)N(C)C)CCOCC3)ccc2n1 32109,c1(C(=O)NC23C(CN(C(C(C=C)(C)CC)=O)C2)C3)ccc([N+](=O)[O-])c(N)n1 32110,N1(C(c2ccc(C)cc2)=O)CCCN(C(=O)C(CO)c2ccccc2)C(CO)C1 32111,C1(COC)CN(C(=O)C=C(C)C(F)F)CCN1C(C1CCC12CCC2)=O 32112,C1(C(N2CC(=C)C2)=O)CC(=O)CN1C(=O)CCc1cccn1C 32113,C1(NC(CC(CCC)(C)C)=O)CC(C2CCN(C(=O)C(C)c3ccco3)CC2)C1 32114,C1(N(C(CN(C)CC)=O)C)CCC2CN(C(c3ocnc3C3CC3)=O)CC12 32115,C(CC(=O)NCC(CO)NC(=O)CC1CC(OC)C1)OCC#C 32116,Cc1csc2c(CC(N3CC(C4(NC(=O)C(C)CN(C)C)CC4)C3)=O)cccc12 32117,c1(N2CC(NC(c3cc(I)c(O)c(I)c3)=O)C2)ncnc2ncc(Br)cc12 32118,c1(C(N(CC(C)CNC(=O)CCn2cnccc2=O)C)=O)ccc(N)c(Cl)c1O 32119,CCC(C)CCCC(=O)N1CC(NC(C2CN3CCC2CC3)=O)C(C)C1 32120,Cc1c(C(=O)NC(C)C(CO)NC(=O)C2=NOC(C)(C)C2)nc2sccn12 32121,c1(SC)ccc([N+](=O)[O-])cc1C(=O)NC1CC(NC(=O)C#CC2(C)CC2)C(O)C1 32122,CC1(C)c2[nH]nc(NC(c3ccc(Cl)c(Cl)c3Cl)=O)c2CN1C(=O)C=CC1CC1 32123,C1(c2ccccc2)(CC(=O)NCC2CCN2C(=O)Nc2ccccn2)CCCO1 32124,c1(C(=O)NCC(CC)NC(c2cnccn2)=O)nonc1N 32125,Cc1nc2c([nH]1)CC(C(=O)N(C)CCNC(c1ccc(C(C)C)o1)=O)CC2 32126,Cc1ncc(C(N2CCCC2CC(=O)NCc2cnn(C(C)C)c2)=O)c(=N)[nH]1 32127,Cc1ncc(NC(C2C3CC2N(C(c2cnc(N(C)C)o2)=O)C3)=O)cc1Br 32128,Cc1cc(N2CCC(NC(C3CCCC3(C)C)=O)C(F)C2)nc(S(C)(=O)=O)n1 32129,c1(C(=O)NC2CC(CNC(C(C)(O)C3CCC3)=O)C2)cc(Cl)nc(Cl)c1 32130,C=C(C)CC(C(=O)NC1CN(C(C2CC(C)(C)CN2C)=O)C1)OC 32131,c1(C(=O)NCC2CCCN(C(C(C)(C)CC#N)=O)C2)cc(F)cc2nc[nH]c12 32132,C(=O)(C1CCCc2cncn21)NCCCCNC(C(C)N1CCC1)=O 32133,Cc1nc(C(N2CCC(C(=O)NC(C(=O)OC)C3CC3)C2C)=O)c(C)s1 32134,C#CCC(C)(C(=O)NCC(CNC(=O)C=CC(=O)OC)OCCCC)NC(C)=O 32135,c1(C(=O)NC(C2CCCC2)CNC(C(F)OC)=O)c[nH]nc1Cc1ccccc1 32136,C1(NC(CC)=O)CCCC(NC(c2cc(-c3ccc(C)s3)[nH]n2)=O)CC1 32137,N1(C(C(C=C)O)=O)CC(C(N2C(C(=O)OC)CC2C)=O)CC(C)C1 32138,Cc1coc(C(=O)NC(C)(C)C(=O)NCC2C=CCC2)c1 32139,C1(C(N2CC(NC(C(c3cccc(Cl)c3)CC)=O)C2)=O)CCC2CC2C1 32140,CCCCCCCCCCC(=O)NC(C)CN(C(=O)C(c1ccc(Cl)cc1)O)C 32141,c1(C(N2CCC3CCC(C2)N3C(C2CCCO2)=O)=O)cc2cccc(F)c2o1 32142,c1(C(N2CC(N(C(C=CC(C)C)=O)C)C(F)C2)=O)cc2nccn2c(O)n1 32143,C1(CNC(CCC(C)C)=O)CC2CCC(C1)N2C(=O)COCc1cccnc1 32144,c1(C(C(=O)NC2(C=C)CNC2)(F)F)ccccc1Br 32145,c1(C(N2C(C#C)CCC2)C(=O)NC2CC(F)(F)C2)cccc2[nH]ncc12 32146,c1(C(N2CC(SC)C(NC(=O)C(C(C)C)N(C)C)C2)=O)cnn2ccn(C)c12 32147,CC1(CNC(c2[nH]ccc2CNC(C2OC3CCC2C3)=O)=O)CCCCO1 32148,CCCCC(CNC(C1CC(OC)(OC)C1)=O)NC(=O)CC1CCC(=O)N1C 32149,C1(CNC(=O)CCC2CCC(=O)N2)CN(C(C2CC2F)=O)CCC12CCC2 32150,C1(NC(CCCOCC)=O)C2CC(O)C1N(C(=O)C(C(C)C)c1cc(C)no1)C2 32151,c1(CC(=O)NC(C2CN(C(C(C)c3cc[nH]n3)=O)C2)C)cccc2cn[nH]c12 32152,CC1(C)C(C(=O)NCC(P(C)(C)=O)c2ccccc2)(CO)C1(C)C 32153,C(=O)(C(F)(F)CC(C)C)N1CCC(CCN(C(c2c(C)ncc(N)c2)=O)C)CC1 32154,C1(CNC(CC(C)n2ccnc2)=O)CCN(C(=O)C(C)(C)N(C)C)CC1 32155,c1(NCCCC2CN(C(=O)OC(C)(C)C)C2)ncnc2c1ccn2CC(=O)O 32156,c1(-c2cc(C)cc(OC)c2F)cccc2[nH]nc(C(=O)Nc3conc3C)c12 32157,Cn1ccc(S(=O)(=O)NC2(CNCc3cnc(Cl)cc3F)COC2)n1 32158,C#CCCCC(C)C(=O)N(C1CC(C#N)C1)CC(=O)NCC1CCC(=O)NC1 32159,N1(C(C2C3CN(C)CC32)=O)CCC2C(CCN2C(c2ccc(F)cc2Cl)=O)C1 32160,C1(NC(C(C)OC)=O)CCN(C(c2cnc(-c3ccccn3)nc2)=O)CC1O 32161,N1(C(C(c2n(C)cnc2)O)=O)CCN(C(c2cocn2)=O)C(CO)C1 32162,c1(OC)cc(C)cc(C(=O)NCC2CC(OC)CN2C(=O)CC(F)F)c1C 32163,c1(C(=O)NCC2CC(F)(CNC(C(CC#C)C)=O)C2)cc(C)c(C)c(C)c1 32164,c1(C(=O)NC2C(NC(CC=C)=O)CCC2)sc(O)nc1C 32165,c1(OC)nccc(C(=O)NC2(CO)CN(C(=O)C(CCSC)NC(=O)C3CC3)C2)n1 32166,C1(C(=O)NCCNC(C2(C(=O)OC(C)(C)C)CC2)=O)CC2(C1)C(F)(F)C21CCC1 32167,Cc1c(CN(C)C(=O)NCCC2COCCO2)cccc1F 32168,N1(C(C(CNC(=O)COC2CCOCC2)O)=O)CCC2(CC1)CSC2 32169,C12(NC(CCN(C(CCC)C)C)=O)CC(C(=O)OC)C(C1)C2 32170,c1(CNC(CN(CC)CC)=O)nc(CNC(C2(C)CCCN2C)=O)cc(O)n1 32171,C1(OC)CC2CC(C(=O)NCC3CCC3)CC12.c1(C(=O)NCCO)ccco1 32172,C1(CNC(c2ccc(OC)cc2)=O)(OC)CCN(C(C2CN(C)CC2C)=O)CC1 32173,Cc1nc(NCC2CCCC2)cc(N2CCOC(CN3CC4CC4C3)C2)n1 32174,C(=O)(C1=C(C(=O)C2CC2)C(c2cn3c(Br)cccc3n2)N(C)C(=O)N1C)OC 32175,N1(C(C2CCCC(C(=O)OC)C2)=O)CC2(CCCCN(C(c3ccsc3)=O)C2)C1 32176,c1(C(=O)OCc2cc(CC(=O)OC)no2)sc(C)c(Br)c1C 32177,c1(OC)cnc(NC(C2CC23CN(Cc2cc(C)[nH]n2)C3)=O)c(F)c1 32178,N1(C(C2(COC)CCOCC2)=O)CCN(C(=O)C(C)n2ccnc2)CC12CC2 32179,C(=O)(C1=NOC2COCC12)N1C2C(C(N3CCCC(F)C3)=O)C(C2)C1 32180,C(CC(=O)N1CCN(C2CCC2)CC1)(C(C)OC)NC(C(COC)COC)=O 32181,N1(C(C2C(C=C)C2)=O)CCC(O)C(NC(=O)Cc2csc(-c3ncccn3)n2)C1 32182,CC(CC(N)=O)C(=O)NC12CC(C(=O)NCC(C)(C)CC(C)O)(C1)C2 32183,Cc1cc(F)sc1C(=O)NC1(c2ccccc2)CCN(C(c2nonc2N)=O)C1 32184,N1(C(C(C)CNC(=O)CC2CCC(=O)C2)=O)Cc2ccnn2CC1C 32185,Cc1ccc(N(CCCNC(=O)C2=CC3CCCC23)C(C)C)c([N+](=O)[O-])c1 32186,CN1CCC(C)(C(=O)NCCC2(CNC(=O)C(F)CC3CCCCC3)CC2)C1 32187,C=C(C)CC(C(=O)N(C(CC)C(=O)NC1(C)CCC(C)C1)C)NC(C)=O 32188,c1(CC(=O)NCC2CCCCN2C(c2cccc(F)c2O)=O)cc(Cl)ccc1Cl 32189,CC1CN(c2nc(C3CCOCC3)ns2)CCC1NC(c1ccnc(O)c1)=O 32190,c1(C(=O)NC(C2CCN(C(C3C(CC)C3)=O)C2)C)ccc(Cl)nc1 32191,C1(C(=O)NCC2C(C)(C)C(NC(c3ccc(Cl)o3)=O)C2)CCc2[nH]nc(O)c2C1 32192,C1(CNC(C(C)OCCCC)=O)CCCCN(C(=O)CC2(CSC)CC2)C1 32193,N1(C(C2N(C)CCOC2)=O)CC2(CCN(C(C34COC(C3)C4)=O)CC2)C1 32194,CCC(C(=O)NCC(COC)NC(c1cccc(C)c1F)=O)C(C)(F)F 32195,C1(C(=O)NCC(C)NC(=O)CC2(CO)CC2)CC2C(C1)C2(C)C.C(C)(C)(C)OC(=O)N 32196,C1(NC(CN(CCOC)C)=O)CN(C(=O)C(c2ccc(Cl)cc2)C)CC12CC2 32197,N1(C(=O)Cc2cn[nH]c2)CCCC(C2CN(C(C3COCCC3(F)F)=O)C2)C1 32198,C(CC(C)C)(C(=O)N1CC(N2CC(NC(=O)CC3(CSC)CC3)CC2=O)C1)OC 32199,c1(C(N2C(C)CC(NC(C3CCCC3(C)C)=O)CC2)=O)cncc(N=[N+]=[N-])c1 32200,N1(C(CNS(N(c2ccc(N)cc2)C)(=O)=O)=O)C2CCC1CN(C(=O)N(C)C)CC2 32201,C(=O)(N=c1[nH]nc(Br)s1)NC1CCCN(C(c2nc(CN(C)C)no2)C)C1 32202,C1(CCNC(CCN(C)CC)=O)CCCCN1C(c1ocnc1C1CC1)=O 32203,c1(C(=O)NC2C(NC(CC3OCC(C)(C)OC3)=O)C2)ccc(Cl)c(Cl)c1O 32204,c1(C(N2CCCC(N(C(c3cnc(O)s3)=O)CC)C2)=O)cnn2cccc(Cl)c12 32205,c1(C(=O)NCC2(NC(C(CC)NC(N)=O)=O)CCCCC2)cn2cnnc2cn1 32206,n1(CC(=O)NC(CNC(C2(C)CCOC2)=O)(C)C2CC2)cnc2sccc2c1=O 32207,C#CC1CC1C(=O)NC1CC(N(C(=O)CC2CCN2C(=O)OC(C)(C)C)C)C1 32208,N1(C(c2c(C)nsc2)=O)CC2(CC(C(=O)NCC(C)(O)C3(C)CC3)CO2)C1 32209,c1(CNC(=NCCC2(C)CC2)NCC2CC2)nc(O)c2ccc(C(F)(F)F)cc2n1 32210,CC(C)(C)CC(F)C(=O)N1CC(CNC(=O)CSCC(F)F)C(F)(F)C1 32211,CC1(C(N2CC(C3CCCO3)C2)=O)CN(C(C2CCC(=O)C2)=O)C1 32212,Cc1cc(C2CC2)ccc1C(=O)NC1C2CC1N(C(C1CC1c1ccsc1)=O)C2 32213,N1(C(c2cnn(CC)n2)C(=O)NCCOCC)CCC2CCN(C)CC12 32214,c1(CC(=O)NC2CC(NC(c3ccnnc3O)=O)C2)cc(F)cc(F)c1Br 32215,N1(C(CC(C=C)(C)C)=O)C(C)CC2CN(C(=O)CC3COCC(C)(C)O3)CC12 32216,C1C(F)(F)CCC(=O)N2CCC(CC2)c2cn1nn2.C(CO)(CC(C)(C)C)SC 32217,Cc1c(S(N)(=O)=O)cnc(N2CCC(OC3CCC3)CC2)c1Br 32218,c1(C(=O)NC(CCCC)CNC(c2cc(OC)cnn2)=O)c(F)cc(F)cc1Cl 32219,c1(C(=O)NCC(C)CNC(=O)C(C)NS(C)(=O)=O)cccc2cncn12 32220,C1(C(=O)NC(C#C)(C)C2CC2)C2CC3C(C2NC(=O)CCCCN(C)C)C13 32221,c1(CC(C(=O)OC)Nn2cc(C3CC=CCC3)nn2)ccc(OC(F)(F)F)cc1 32222,c1(CN2CC(NC(c3c(C)ccc(Br)c3)=O)C(C#N)C2)ccc2nc[nH]c2c1 32223,C(C(=O)Nc1cncnc1C)(C(C)(C)C)NC(CCSCCCC)=O 32224,N1(C(COc2cccc(OC)c2)=O)CC2CC(NC(=O)C(C#N)C(C)C)C(C2)C1 32225,c1(C(N(CC(CC)NC(c2c(CC)cc[nH]2)=O)C)=O)nccc2ccn(C)c12 32226,C1(NC(C=C(C)C)=O)CN(C(c2snnc2C(C)C)=O)CC1C 32227,C1(CC)CN(C(C2C(C)C2C)=O)CC1C(=O)N(C(C)C(=O)OC)CC 32228,N1(C(C(CCCC)O)=O)CCN(C(C2CC(OC)C2)=O)C2(CCC2)C1 32229,C1(C)(C(=O)NCC(=C2CN(C(CCCOC(C)C)=O)C2)F)CCCS1(=O)=O 32230,C1(C(=O)NC2CC(C)(NC(C3CC3(Cl)Cl)=O)C2)COCCN1CC(F)F 32231,c1(C(N2CCC(CC(=O)N(CCC)Cc3cnccc3C)C2)=O)cnc(C)nc1 32232,CC1CC2CC1CN(Cc1ccc(OCCC(N)=O)cc1)C2 32233,N1(C(C2OCCN(C(C)=O)C2)=O)CC2(CCN2C(=O)C2=CCOCC2)C1 32234,C1(C(=O)NC2CCC(CNC(C(C)C#N)=O)C2)CC2(CC(=O)N2)C1 32235,O=C1C=C2CN(C(C3CC3Nc3ncc4[nH]ccc4n3)=O)CCC2S1 32236,C1(CNC(=O)CCCc2ccsc2)CC(F)(F)CN1C(C1CC(F)C1)=O 32237,c1(C(C(=O)N(CCNC(C(C)n2cccn2)=O)C2CC2)C)ccnn1C 32238,C(c1cnc2ccccc2n1)=CC(N1CCC(CC)(NC(C2CC2C)=O)CC1)=O 32239,S(=O)(=O)(c1ccc(NC2CCOC(CC)C2)cc1Br)NCC(C)(C)OCC 32240,c1(C(N2CCCC(CN(C(C(C(=C)Cl)(C)C)=O)C)C2)=O)cn2cc(C)ccc2n1 32241,C1(CCNC(C2C(OC)CC2)=O)CCCCN1C(c1cccnn1)=O 32242,c1(C(=O)Nc2n[nH]cc2C(F)F)ccc(-c2ccccc2)c(F)c1 32243,C1(CNC(CC=C(C)C)=O)CC2(CCN(C(c3cn(C(C)C)cc3C)=O)C2)CO1 32244,CCC(C(C)(C)O)NC(c1cnn(CCNC(C2CCC(=O)C2)=O)c1)=O 32245,C(=O)(CCCCC(N)=O)NC(CC(=O)NC1CCCN(C)C1=O)C(F)F 32246,C(N=c1[nH]c(=NCCN(C)C2CC2)[nH]c2cc[nH]c12)C1N(CC)CCCC1 32247,C#Cc1ccnc(C(N2CCN(C(=O)C(CC)CC=C)C(C(C)(C)C)C2)=O)c1 32248,C1(F)(CNC(C(CCCC)C)=O)CCCN(C(=O)Cc2ccc3occc3c2)CC1 32249,CC1(C)CC(C(N2CC3C(NC(c4cccc(F)n4)=O)C3C2)=O)CCO1 32250,C(=O)(CCC(C)S(C)(=O)=O)NC(CNC(c1c(C)nn(C2CC2)c1Cl)=O)C1CC1 32251,CCC(C)C(C(=O)NCC1(C(N2CCC(O)CC2)=O)CCCO1)N(C)C 32252,c1(C(N2CC(O)(CCNC(CC(=C=C)C)=O)C2)=O)cnc2scc(C)n2c1=O 32253,CC(c1ccccc1Cl)=CC(=O)NC1CC(CNC(c2cc(C)nc(C)n2)=O)C1 32254,Cc1ccc(O)c(C(=O)NCC(C)NC(c2ccn(C)n2)=O)n1 32255,c1(C(N2CC(=O)NC2)=O)cc2n(n1)CCCN(Cc1cc(F)ccc1[N+](=O)[O-])C2 32256,N1(C(C(C)OCC=C)=O)CC(COC)(NC(=O)CC(C)OC)C1 32257,c1(C(C(=O)NC(C)C)N(CCC(=O)OCC)CCC)nn(CC)cc1Cl 32258,N1(C(c2ccc(CCC)[nH]2)=O)CC(NC(c2cccc(N)c2)=O)CC1(C)COC 32259,C1(C(=O)OC)C2CC1N(C(=O)C(C1CCN(C(=O)C(C)(C)Cl)C1)F)C2 32260,c1(NCC(CC)CO)nc(N2CC(N)CC(O)C2)nc2c1ncn2C(C)C 32261,N1(CC)CC(C(=O)NC2CN(C(c3ccnc(NC4CCC4)c3)=O)C2)NC1=O 32262,C(CCCCCC(=O)NC1COC(c2nn[nH]n2)C1)n1cc(-c2c(C)ncs2)nn1 32263,N1(C(c2cnc(C(C)=O)s2)=O)CCCC2(NC(=O)CNC=O)CC2C1 32264,C(CC(=O)NOCC=CCl)(C(C)(C)C)NC(C(C(=O)OCC)OC)=O 32265,c1(C(N2CCC(C)(NC(c3nc(C)c(C)[nH]3)=O)CC2)=O)cnc(O)c2ccsc12 32266,C(CC(C(=O)NC1(CO)CCC1)NC(=O)Cc1ccc(C)s1)=CC 32267,c1(C(=O)NCC2=CCN(C(C3CC=CC(O)C3)=O)CC2)cccc2ccoc12 32268,C(CNC(c1cc(OC)cs1)=O)(CCC)NC(C(C)=C(CC)C)=O 32269,C12(C(N(CCN(C)C(C3(n4ccnn4)CC3)=O)C)=O)CC(C1)C(C)(C)O2 32270,C1(F)(C(=O)NCC2CC(NC(CSc3n(C(C)(C)C)cnn3)=O)C2)CCCCC1 32271,N1(N2CC(N3CCN(C(C4CCC(C)(C)C4)=O)CC3)C2)CC2(CCOCC2)C1 32272,O=S(=O)(c1ccc(NCCCCCF)c(Br)c1)NC1C=CCCCC1 32273,N1(C(C=CC(=O)OCCCC)=O)CCC(C2CCCN(C(c3coc(Cl)c3)=O)C2)C1 32274,Cc1cnc(N(C23CC(N)(C2)C3)C(C23CCC(CC2)CC3)=O)nc1C 32275,C(=O)(CCCCCF)NC(C1CCCC(C(=O)NCC2C(C)CCC2)C1)=O 32276,C1(CCN)CCCN1N(C)CCCC1CCC1 32277,N1(C(c2cc(CCC)[nH]n2)=O)CCCC(N2CCN(C(C3CCOC3)=O)CC2)C1 32278,Cc1ccnc(C(C)(C)C(=O)NC(C)CN(C(=O)C(F)OC(F)(F)F)C)c1 32279,N1(C(c2c(C)c(F)ccc2)=O)CCCC2CN(C(=O)C3=CCCCC3)CCCC12 32280,C#CCCCCC(=O)NC1CC1CNC(c1ccc[n+]([O-])c1)=O 32281,c1(CN(C(=O)C=CC2CC2)C)cccc(O)c1 32282,N1(C(C(OCC)OCC)=O)CCC(C(=O)NC2CCC2C(F)(F)F)C(O)C1 32283,C(=O)(CCC(C)(C)Nc1c(-n2nnc(C3CN(c4ncco4)C3)c2)nnn1C)OC.C(=O)NC 32284,C1(C(N)=O)CCCN1C(=O)CN(C(=O)CCN1CCCC1=O)C1CC1 32285,c1(C(N2C(C)CC(NC(=O)COc3ccsc3)C2)=O)cc(F)cc2nc[nH]c12 32286,CN1CC(CC(=O)NC2(C)CCC(CC(=O)O)CC2)c2ccccc21 32287,c1(-n2c(C(c3ccccn3)NC3CSC3)nnn2)ccc2c(c1)CCC2 32288,C1(NC(CN(C)S(N)(=O)=O)=O)CC12CCN(C(c1csc3cncn13)=O)CC2 32289,C1(CNC(c2c(CC)noc2C)=O)CN(C(=O)C(C)(C)C(N)=O)CC(C)(C)O1 32290,N1(C(C(Cn2ccnn2)NC(CCCOC)=O)=O)CC2C(C1)C2(C)C 32291,c1(C(=O)NC2C(CNC(COCCC=C)=O)CCC2)cc(C)nc2ccnn12 32292,N1(C(c2nc(OC)c(C)s2)=O)CC(C2CN(C(C3CCC(C(N)=O)CC3)=O)C2)C1 32293,C12(C(N(CC#C)CC3CCCO3)=O)CC1CN(C(=O)C(C)=NOCC#N)C2 32294,c1(C(N2CCCC(N(C(=O)C(F)C(F)(F)F)CC)C2)=O)cc(C)nc(Cl)c1N 32295,C1(CC#C)CCCCN1C(=O)C(C)N(C)C(c1ncccc1F)=O 32296,C1(C)(CN(C(=O)CNC(=O)COC2CCOCC2)C)CCOC1 32297,C(C(O)C(=O)NC1CCC1NC(=O)COCCSC)=CC 32298,Clc1ccc(CN2CCC2COc2ccccc2)cc1Cl 32299,C(CC(=O)NOC(C)(C)C)C1CC(NC(C2C(C)C2)=O)C1 32300,C1(O)(CNC(CCc2onc(CC)n2)=O)CCN(C(c2snnc2C2CC2)=O)C1 32301,N1(C(C2C(N(CCOC)C(C3CCCCC3)=O)CCC2)=O)CCCCCC1 32302,CCCCC(C)C(=O)N1CCN(C(c2cc(CC)no2)=O)C(C(C)C)C1 32303,N1(C(C(C)(C)OC)=O)CC2(C(=O)NCC(CC3CC3)CO)CC1CO2 32304,c1(SC)nc(N2CCC(NC(c3ccn(C)c3)=O)C(F)C2)cc(C(F)F)n1 32305,C(=O)(C1=COCCC1)N(C)CC1CCN(C(c2c(C)n[nH]c2)=O)C1 32306,N1(C(CN(C)C(C2CCN(c3ccncc3)CC2)=O)=O)CC(N(C)C)C(O)C1 32307,C1(NC(CN(C(C(C)OCCCC)=O)C)=O)CCC(C(C)O)CC1 32308,Cc1cnc(C)c(C(=O)NCC2CCCN2C(=O)CCCNS(C)(=O)=O)c1 32309,c1(-c2nc(-c3scc(C)n3)nn2C2CCOC2)cc(Cl)ncc1Cl 32310,C1(CNC(CC(CCC)CC)=O)CCCC2(CN(C(c3ccnnc3)=O)C2)O1 32311,c1(OC)ccoc1CNC1CC(C(N2CCCC2CO)=O)C1 32312,Cc1c(C(N2CC(NC(=O)CP(C)(C)=O)CCC2C)=O)cc(Br)cc1N 32313,S(=O)(=O)(C1COC(C)(C)C1)NC(C(NOCC)=O)C1CN(C(=O)OC(C)(C)C)C1 32314,CCN=C(NCc1ccccc1SC)NC1CCC(C(=O)OC)C1 32315,C12(NC(CSCC(=O)NC)=O)CC1CN(C(=O)C(C)OCCc1ccccc1)C2 32316,O=C(N=c1cc(C2CC2)[nH][nH]1)C1CCOCN1C(=O)CC(F)(F)F 32317,N1(C(C(=O)NCC)=O)CC(CNC(C2CCC(N(C)C)CC2)=O)C(O)C1 32318,C12(C(=O)NC(CC(N)=O)c3cn(CC4CCOC4)nn3)CCCCC1C2 32319,Cc1cc(C(=O)N(CCNC(=O)C(C)CF)CC2CC2)sc1C 32320,C1(N(C)C(c2cncc(C(F)(F)F)c2)=O)CC2CC1N(C(C1CS(=O)(=O)C1)=O)C2 32321,c1(OCCN(C2CCC2)CCOC)ccccc1Cl 32322,N1(C(c2ccc(C(N)=O)nc2)=O)CCN(C(=O)C2=CCSC2)C2CCCCC12 32323,N1(C(C2N(C(c3c(C)oc(Cl)n3)=O)CC(=O)NC2)=O)CCOC2(CCC2)C1 32324,C#Cc1ccc(C(=O)NC(C)C(C(C)C)NC(=O)CN(C)CCC)c(F)c1Cl 32325,C1(CNC(C2(COC)CCC2)=O)CCC(C)(C)CN1C(c1ccc(C)nc1)=O 32326,C(C1=NOC2CC12)NCC1(O)CC(NC(=O)OC(C)(C)C)C1 32327,C(=O)(C1Cc2ccccc21)N1C(CN(C)C(c2csc3nnsc23)=O)CCCC1 32328,Nc1[nH]c(=O)c(Cl)nc1C(=O)NC1(CCNC(C2CC(O)C(F)C2)=O)CC1 32329,Cc1nc(C(=O)NC2(CCNC(C3(N(C)C)CC3)=O)CCCC2)c2n1CCCC2 32330,N1(C(C(C2CN(C(C3CC=C(C)CC3)=O)C2)O)=O)CCC(C)(O)C(O)C1 32331,N#Cc1cnccc1CN1CC2C(C1)N2C(c1c(Br)cccc1Br)=O 32332,CC(CF)CC(=O)NCc1cn(C2CCN(C(=O)COCC3CC3)C2)nn1 32333,n1(CC)ccnc1C(=O)NCCCC1CCCN1C(=O)CN(S(C)(=O)=O)C 32334,C1(CC(C)C)C(=O)N1.C1(NC(C(C)C)=O)CN(Cc2ccccc2)CC1C#N 32335,N1(CC(=O)Nc2ccc(-c3nccc(C)n3)cc2)Cc2c(F)cccc2C(C)(C)C1 32336,C12(NC(=O)CC3COCCOC3)CCCC1CN(C(c1cc(O)nc(O)n1)=O)C2 32337,CC1CCCCN1CC(N1CCN(C(=O)Nc2nccs2)CC1)C 32338,C=CCC(CC)C(=O)N1CCNCC1.C1CC(C2CC2)CN1 32339,Cc1cc(C(N2CCC(C)(CNC(C3CC4CC3CC4O)=O)CC2)=O)ccc1O 32340,C12(C(N3CCC(O)(C(C)NC(C(=C(C)C4CC4)F)=O)C3)=O)CC3CC1C2C3O 32341,c1(CNC(CN(C(C2CC2C2(C)COC2)=O)CC)=O)nc(C)cc(C)n1 32342,c1(CC(=O)NCC(C(C)C)NC(c2cnc(C(C)(C)C)[nH]2)=O)cc(F)cc(F)c1 32343,N1(C(CCCC=C)=O)CCCN(C(=O)C2=CCOCC2)CCC1 32344,c1(C(=O)NCC#CCNC(=O)COCC2CCC2)cn2ccnc2cn1 32345,N1(C(C(C)OC)=O)CCCC(N(C)C(c2ccc(-n3cncn3)cc2)=O)C1 32346,c1(C2C(NC(C3CC(=O)NCC3)=O)C2)ccc2c(c1)CN(C(=O)COC1CCC1)C2 32347,c1(C(=O)NCC(CNC(C(C2CCCOC2)OC)=O)C)c(F)ccc(F)c1F 32348,c1(C(=O)NC2(C)CN(C(c3c(O)cc(C)nn3)=O)C2)cc(F)cc2nccnc12 32349,C1(NC(c2c(C)cc(C)s2)=O)CCN(C(=O)C(c2cccc(Cl)c2)(C)C)CC1O 32350,C1(C)(CC)CCN(C(C2CCC(NC(=O)C(O)CCN(C)C)CC2)=O)C1 32351,C1(N(CCCC#C)C(=O)Cc2ccc3occc3c2)CCCC12CCNCC2 32352,c1(C(N2CC(COC)(CNC(C3CCC(C)S3)=O)C2)=O)nc(C)ccc1OC 32353,C1(NC(CC2CC(C)C2)=O)C2CC3C1C3C2C(=O)NC1Cc2ccccc2C1 32354,C(=O)(C(Cc1ccc(O)cc1)C(F)(F)F)NCC1C(NC(CCC=C)=O)CC1 32355,C(=O)(C1=CCCOC1)NC(C1CC(NC(C2CC(OCC)C2)=O)C1)C 32356,Cc1cc(CNC(c2c(Cl)cnn2C)c2nnnn2CC2CCCO2)cnc1O 32357,CC1C(C(=O)NC2CCN(C(=O)C=Cc3cnc[nH]3)C2)OC2CCCCC12 32358,CC(=O)CCCC(=O)NC12CCC(C1)N(C(=O)C(C(C)(C)C)OC(C)(C)C)C2 32359,C1(C(N2C(CNC(=O)C(=O)NCC(F)F)C(O)C(O)C2)=O)CCCC(F)(F)CC1 32360,CCC(F)(F)C(C)(C)C(=O)N1CCC(C(C)NC(C2(C#N)CC3CC3C2)=O)C1 32361,c1(C(N2C3CCC(NC(c4cnc(Cl)s4)=O)C(C3)C2)=O)cnc(O)c([N+](=O)[O-])c1 32362,C(=O)(CCNC(c1cnsc1)=O)NC1C(C)C1 32363,c1(NC(C(CCCC)NC(=O)C(F)CC2CCOC2)=O)ccc2c(c1)CCC2 32364,CC(C)CC(C)(CNC(=O)CCOC1CN(C(=O)CCc2ccoc2)C1)N(C)C 32365,Cc1cc(NC(=O)CC2CCN(C(c3cc(Cl)ccc3O)=O)C2)nc(Cl)c1 32366,N1(C(C(C)CCO)=O)CC(NC(c2ccc3nc(O)[nH]c3n2)=O)C(S(C)(=O)=O)C1 32367,c1(OC)ccc(C(C(=O)NCC(C2CCC2)NC(c2cc(Cl)no2)=O)OC)cc1 32368,c1(C(=O)NC2CN(C(C3(OC)CCCCCC3)=O)C2)cc2c(C)c(F)ccc2[nH]1 32369,Cc1cn2ccc(C(=O)NCCOCCN(C(=O)CC(C)CN(C)C)C)cc2n1 32370,N1(C(C2CCN(C(C)=O)CC2)=O)CCC2(CCN(C(c3nc(C)sc3C)=O)C2)C1 32371,N1(C(C(C)(C)n2ccnn2)=O)CCCCC1CCNC(=O)Cc1cnns1 32372,c1(OC)cc(NC(C2CC2NCc2ccnc(-c3ccccc3)c2)=O)c(C)cn1 32373,N1(C(C)(C)C(=O)NCCc2nnc3n2CCNC3)C(=O)c2ccccc2C1=O 32374,c1(OC)ccc2c(c1)C(=O)CCN2C(=O)Cc1c(C)nc(C)nc1O 32375,N1(C(c2c(CC)non2)=O)C2CCCC1CC(NC(c1cnnc(O)c1)=O)C2 32376,C1(C(C)C)CN(C(C2CCC2(C)C)=O)CCN1C(=O)C1=CCCS1 32377,C(=O)(CN=c1[nH]c(C)cs1)NCC1CN(C(C(C)OC)=O)CC1C 32378,c1(C(N2CC(O)(CCNC(C3(F)CCOC3)=O)C2)=O)cc(F)ccc1Br 32379,C1(CNC(CC2(OC)CCC2)=O)C(C)CCCN1C(=O)CCC(C)C 32380,N1(C(c2c(C)cc(CNC(C3CC34CCCC4)=O)o2)=O)CCCC2C(=O)NCC12 32381,N12CCCN(CCC1)C(=O)C2.C(C(=O)OC(C)(C)C)OCCOCCOCC#C 32382,C1(c2c(CN3CCCC(c4scc(CC)n4)C3)c[nH]n2)CCC2CC1CO2 32383,C1(CC(=O)N(CCC)CCNC(=O)C2=C(Cl)CC2)CSc2ccccc2O1 32384,C1(NC(CC(C)C(F)F)=O)COC2(C1)CN(C(C1CC=CC1)=O)C2 32385,N1(C(CC2(OC)CC2)=O)CC(NC(=O)CCc2ccc(N(C)C)nc2)C(C)(C)C1 32386,c1(CC)nc(Cl)nc(N2CCC(NC(C3CCC(NC(C)=O)CC3)=O)CC2)c1Cl 32387,N1(C(CCOC)=O)CCC(C)C1C(N1CCN(C2CC2)CC1)=O 32388,c1(C(=O)NCC2(CC(=O)Nc3cncc(CO)c3)CC2)c[nH]ccc1=O 32389,CC(C)CC(C)(CNC(C1CC12CCCC2)=O)NC(=O)C=C(Br)Br 32390,n1(CC)nc(C)c(C(=O)OC)c1C.n1(CCCC)nnnc1C(CC(C)SC)N 32391,O=S(=O)(c1ccc(F)c(Br)c1)Nc1nccn2c(Br)ccc12 32392,C#CCC(CO)NC(C1(CNC(=O)CCOC2CC2)CCC1)=O 32393,C1(CC(=O)NC2CCN(C(C)C)CC2)CC2(C1)CN(C(C1CC(C)(F)C1)=O)C2 32394,C(CC(O)C(=O)NCC1CCN(C(=O)CSc2cccc(F)c2)C1)SC 32395,C1(NC(c2ccc(C(C)C)cc2O)=O)CN(C(=O)CCS(C)=O)C2(CCC2)C1 32396,c1(OC)cc(C(=O)N(C2CC3CNC2C3)CC2CNC(=O)CO2)cc(Cl)c1 32397,c1(C(N2CCC(C3N(C(C(CCCC)F)=O)CCC3)CC2)=O)cc(F)c(O)c(F)c1 32398,C12(CNC(C(CC=C)NC(C)=O)=O)CCC(CC1)N2C(=O)C(F)(F)COC 32399,c1(C(C(=O)Nc2ccc(OC)cc2)N(C2CCOCC2C)C)cc(C)ccc1Br 32400,c1(OCC(=O)NC2CC(N(C(C3(O)CN(C)C3)=O)C)C2)cccc(NC(N)=O)c1 32401,CC(C)C(C)CC(=O)N1CC(NC(C2CCC(C)(C)C2)=O)C1 32402,N1(c2n(Cc3ccc(OC(=O)OC(C)(C)C)cc3)nnn2)CCCc2sccc2C1 32403,c1(C(N2CCCC(CC(=O)OC)C2)C2CC2)cccc(C(F)(F)F)c1F 32404,CC1=C(C)CC(C(N2CCC(C(=O)NC3CNC(=O)C34CC4)C2C(C)C)=O)CC1 32405,NS(=O)(=O)c1ccsc1C(N1CC(O)(CNC(=O)CCc2cc(Cl)no2)C1)=O 32406,c1(C(=O)NC(C(=O)NCC2(OC)CC2)C)c[nH]c(=N)c(C)c1 32407,CCC(C)(C)C(O)C(=O)N1CC(C2(NC(=O)C(C)CSC)CC2)C1 32408,CCC(CC(=O)N1CCC(C)(NC(=O)CCCNC(=O)OC)C1)OC 32409,C1(C(C)NC(C2CCN2S(C)(=O)=O)=O)CCN(C(C2(O)CC2)=O)C1 32410,C(=O)(C(C)(C)CCC)N.C(=O)(CNCCCN(C(=O)CSC(C)(C)C)C1CC1)OCC 32411,N1(C(C2(C)CN(Cc3ccc(C)nc3)C2)=O)CCC2SC(=O)C=C2C1 32412,c1(C(N2C(C)CC(NC(c3cc(CO)n(C)n3)=O)C2)=O)cccc2c1CCO2 32413,Cc1cc(S(N)(=O)=O)cc(C(=O)N(C(C)CNC(=O)CCCCC#N)C)c1C 32414,N1(C(c2c(N(C)C)cccc2)=O)Cc2ccc(C(=O)NCC(C)(C)F)cc2C1 32415,Cc1ccc(C2(C(N3CCCC(N(C(=O)C(C)N4CCC4)C)C3)=O)CCC2)cc1 32416,C(=O)(N=c1[nH]sc2c(Br)cccc12)NCCCC(=O)N(C)C 32417,CCC(F)(F)CC(=O)N1CCCC(NC(=O)CCCn2cccn2)C1C 32418,c1(-c2[nH]c(=N)sc2)ccc(C(=O)NC2CC(NC(C3CCOC3C3CC3)=O)C2)cc1 32419,c1(CC(N2C(C(=O)Nc3onc(C)c3Br)CCCC2)=O)cc(F)ccc1[N+](=O)[O-] 32420,CCN=c1ccc(C(=O)NC2CC2NC(c2ccc(C(F)(F)F)s2)=O)c[nH]1 32421,N1(C(C2CCN(C(c3cc(OCC)c(Cl)nc3)=O)CC2)=O)CCCC(F)(F)CC1 32422,C(C(=O)N=c1cc[nH]c(C)c1F)C1C2CN(Cc3c(NC)nc(F)cc3)CC21 32423,C1(C(=O)NC)CC2(CC(OCC)C2)C1.C12CCCCN1C2=O 32424,C(=O)(C(C)S(N)(=O)=O)N1CC(N(C)C(c2ccc(N3CCNC(=O)C3)cc2)=O)C1 32425,C=CCC(CC(F)F)C(=O)N1CCN(C(=O)CCC(CC)CC)C(CC(F)F)C1 32426,N1(C(c2cccnc2)=O)CCC2(CCN(C(c3cnc(Cl)cn3)=O)CC2)C1 32427,c1(C(=O)NCC(CNC(c2csnn2)=O)CO)ccc(-n2cncn2)cn1 32428,N1(C(c2ncn(C)n2)C(=O)NC2CC2)CCC(CC2CCOC2)CC1 32429,N1(C(C=CC(C)=O)=O)CCC(CC(C)(C)NC(=O)Cc2nccn2C)CC1 32430,CC1CN(C(=O)CSCC=O)CC1CNC(=O)C(F)(F)c1ccncc1.CC#N 32431,c1(C(=O)OCC)cc(C(=O)NC(C)CC(C)NC(C2(C(C)(F)F)CC2)=O)[nH]n1 32432,c1(C(=O)NCC(CC)NC(C2CCN(C)C2)=O)nncc2ccccc12 32433,Cc1ccc(O)c(C(=O)NC(c2cnn(C)c2)C(N2CCC3CC23)=O)c1 32434,c1(N2CCC(CNC(C=C(CC)CC)=O)C2)ncnc(C(F)(F)F)c1C(=O)OC 32435,Cc1ccc2ncc(C(N3CCC(C)C3CNC(=O)C(C)(C)CC(F)F)=O)n2c1 32436,C1(NC(c2c(C)nn(C)c2F)=O)COC2(CCN(C(=O)CS(=O)(=O)N(C)C)C2)C1 32437,CCCC(CCNC(C1CCC1CNC(C1(OC)CCOC1)=O)=O)CCC 32438,CCCC(CCC)CC(=O)NC(c1cn(C)nn1)C(N1CCC(O)CC1)=O 32439,C(CCCCCC(=O)NC(C(=O)OC)C1CCC1)NC(c1n(CCC)ccc1)=O 32440,c1(N2CCC=C(C(=O)NCc3cc(C)c(O)c(C)c3)C2)ccnc(S(C)(=O)=O)n1 32441,C1(CCC)(NC(c2cccc(N(C)C)n2)=O)CCCN(C(=O)C(C)C(F)F)C1 32442,c1(C(=O)NCC23CC(NC(C4CC(=C)C4)=O)(C2)C3)cc(OC)c2occc2c1 32443,N1(C(Cc2c(C)nc[nH]2)=O)CC(NC(=O)C2=CCOCC2)CC12CCOCC2 32444,n1(CC(N2CCC(CNC(CCC(=C)C)=O)(OC)C2)=O)ccc2c(C)cccc12 32445,c1(C(=O)NC2C(CNC(C(C)c3ccsc3)=O)C2)ccc(Cl)c(F)c1O 32446,C1(C)(NC(CN(C2CCC2)C(C2C(C(C)C)CCC2)=O)=O)CN2CCC1CC2 32447,Cc1cnccc1C(C)C(=O)NCCN1CCC(NC(=O)C(N)=O)CC1 32448,c1(COC)cccc(C(=O)NC(C)C(C)NC(C2(C(F)(F)F)CC2)=O)c1 32449,N1(C(C2(C(C)NC(=O)CC3C=CCC3)CC2)=O)CCCC(CC2CC2)CC1 32450,c1(C(=O)NCCOCCCNC(C2(C(=O)NC3CC3)CC2)=O)csc(Cl)c1 32451,C1(C(N(CC(CC)NC(=O)CSCC(C)C)C)=O)CCOC1C(C)C 32452,C1(O)(C(N2CC(C)OCC2C)=O)CCCC(C)CC1 32453,C(=O)(C(C)(C)C(=O)NC1CN(C(=O)CC(=O)OC(C)(C)C)CC1C)OC 32454,CC1=CCSC1C(=O)NC(C)(C)C=CC(=O)NCC1(S(C)=O)CC1 32455,Cc1c(C(=O)NC2CCCC(NC(c3occc3F)=O)C2)ccn1C(C)C 32456,Cc1cccc2c1CC(C(=O)N(CC(C)CNC(=O)C(O)C1CCC1)C)N2 32457,c1(CNC(c2cc(C(=O)OC)n(C)c2)=O)ccc([N+](=O)[O-])cn1 32458,c1(C(=O)NCC2CN(C(=O)CC=C(Cl)Cl)C3(CCC3)C2)cnc2ncccc2c1 32459,c1(C(N(CC(C)NC(=O)CC(F)F)CC)=O)cc(O)nc2cc(OC)ccc12 32460,N1(C(c2cc(C)n(C)n2)=O)CC(N(C(=O)CSCc2ccccn2)C)C(C)(C)C1 32461,N1(C(CCCC)=O)CC2CC1CN(C(=O)C(C(C)C)NS(=O)(=O)c1cnn(C)c1)C2 32462,C1(CCC)CN(C(c2cc(Br)c(Br)o2)C(=O)NCc2nnn(C)n2)CCO1 32463,N1(C(C2CC(=C)C2)=O)CC(CNC(=O)C=Cc2cc(Cl)sc2Cl)OC(C)(C)C1 32464,C1(NC(CCC(=C)Cl)=O)CC12CCC(NC(c1ccsc1)=O)CC2 32465,CC1CC(=O)NCC1C(=O)NCC1CN(C(C2SCCCS2)=O)CCCO1 32466,N1(CCC=CCCC)CCCC(CNC(=O)C(c2cccc(C(F)(F)F)n2)C)C1 32467,C(=O)(CCC(=O)NC(CNC(c1sc(N(C)C)nc1Cl)=O)C1CCC1)OC 32468,C1(CNC(C2CCCC(C(N)=O)C2)=O)(NC(c2cc(F)n[nH]2)=O)CCCCCC1 32469,C1(NC(C#CC(C)C)=O)CCCC2CN(C(c3coc(C(C)(C)C)n3)=O)CC12 32470,C1(C(N2CC(C)(CNC(=O)C(O)C3CC3)OCC2)=O)OCC2CCCC1C2 32471,CC1CC(NS(=O)(=O)c2cccnc2NCC2(CO)CCC2)c2nccn21 32472,N1(C(C2(CC#C)CCCCO2)=O)CCCCCC(NC(c2ccoc2Cl)=O)C1 32473,C(CC(C)N=c1nc(N2CCC(N(C)CCO)CC2)c2cccc(F)c2[nH]1)SC 32474,c1(C(=O)NC23CC2CN(C(=O)CCCn2cncn2)C3)ccn2ccsc12 32475,N1(C(Cn2ccc(C)n2)=O)CCC(NC(=O)Cc2ccccc2Cl)C(C)C1 32476,N1(C(C(CC)C)=O)CCN(C(=O)CCCCCF)C(CC(=O)NC)C1 32477,Cc1cnc(NCCCCO)c(S(=O)(=O)N(C)C(c2csc3ccccc23)C)c1 32478,N1(C(C(C2CCCO2)NC(CCS(N)(=O)=O)=O)=O)CCC2(COC(=O)N2)C1 32479,c1(CCC(=O)NCC2N(C(c3cc(C)nn3C)=O)CC=C2)ccccc1[N+](=O)[O-] 32480,C1(NC(=O)CCn2ccnn2)CCN(C(c2cnn(C3CCOC3)n2)=O)C1 32481,C1(CCC(=O)NCC(CC)NC(C2CSCN2C(C)=O)=O)CCC(=O)N1 32482,CC(C)=C=CC(=O)NCCC1(C(=O)N(C(C)CC(F)(F)F)C)CC1 32483,C(c1ccnc2ccccc12)=CC(=O)NC1CCCC1NC(C1CC2CC2C1)=O 32484,S(=O)(=O)(c1cncc(Br)c1)NC(C(=O)OC)Cc1ccc(F)cn1 32485,N1(C(CCc2ccc(C)o2)=O)CC=CCC1C(=O)NCc1nnc(O)o1 32486,c1(C(N2CC(CCNC(CS(CC)=O)=O)C(C)C2)=O)ccc(C)cc1C 32487,c1(CCC(=O)N(C)CCOCCN(C(=O)CCC2CCOC2)C)cccnc1 32488,CC1CCC(C(=O)NC2(CCNC(=O)CCNC(=O)C(C)(C)C)CCC2)S1 32489,c1(OC)ccc(S(=O)(=O)N2CC3CN(Cc4ccc(C)c(F)c4)CC3C2)cc1 32490,C1(C(N(C(CCNC(C(C)(C)SC)=O)C)C)=O)CCCN(C(=O)OC(C)(C)C)C1 32491,N1(C(c2c(CC)nns2)=O)CCC(C)(C)C1C(=O)NCCc1ccc(C)cc1 32492,c1(C(=O)NC2C(CNC(C(C)OCCC=C)=O)C2)ccc(F)c2[nH]ccc12 32493,c1(C(=O)NC2(C)CC(NC(c3c(C)ncnc3O)=O)C2)cc(F)cc(Cl)c1N 32494,CC1CN(C(=O)CCC(C)N(C)C)CC(C)N(C(=O)C2=NNC(=O)CC2)C1 32495,C1(C2C(N(C(CCc3ccsc3)C(=O)NC(C)(C)C)C)CCC2)CCCN(C)C1=O 32496,c1(C(C)C)ncccc1CN(C(C)C(F)F)CCO 32497,Cc1ccc(CC(=O)NCCC2CN(C(=O)C=Cc3cccs3)CCO2)cc1 32498,N1(C(c2c(C#C)c[nH]n2)=O)CC(F)(F)CC1(C)CNC(c1c[nH]cc1C1CC1)=O 32499,C=C=CC(C)C(=O)N(CC(=O)N(C)CC1COC(=O)N1)C1CC1 32500,Nc1cc(C(=O)NCC2(NC(c3nc(C4CC4)cs3)=O)CCC2)cc(F)c1 32501,c1(OC)cc(C(=O)NCC2CCN(C(C3CCC=CCC3)=O)C2)cc(C2CC2)c1 32502,Cc1c(C(=O)NCC23CC(NC(=O)Cn4cc(Cl)cn4)(C2)C3)cccc1Cl 32503,c1(CC)nn[nH]c1C(=O)N(CCCNC(c1ccc(CN(C)C)s1)=O)CCO 32504,N12CCc3cc(ccc31)C2C(=O)NC1CC1.N1(NC(CC)=O)CCC2CCC12 32505,N(C1Cc2ccc(F)cc21)C(=O)C=Cc1ccc(Cl)c(Cl)c1 32506,C1(n2c(C(c3nnnn3CC)NCc3cnc(CC)[nH]3)nnn2)CCCCCC1 32507,C12(CNC(c3n(CC)ncc3)=O)CC(CO1)N(C(=O)C(C)OCC(F)(F)F)C2 32508,C1(C)(CNC(c2c(OC)nsc2OC)=O)CN(C(=O)CCC#N)C(C)(C)C1 32509,C(CN=c1cc[nH]cc1S(=O)(=O)NCC1(CO)COC1)OC 32510,C(=O)(C(=O)C(C)(C)CC)N(CC(=O)NOCC1CCCO1)CC#C 32511,Cc1cc(C(N2CC(F)CC2C(=O)NCC2CC(=C3CC3)C2)=O)nc(O)n1 32512,C(=O)(C(C(C)(C)C)c1cc[nH]n1)N1CCCC(CNC(CSCCC)=O)C1 32513,C1(C2CCCO2)(C(=O)Nc2cccc(C(C)(C)C#N)c2)CCCO1 32514,N1(C(C(CCCC)NC(=O)Cc2cn(C)nc2C)=O)CC2(CCOCC2)C1 32515,C1(C(=O)NC)CC(F)(F)CN1C(C(=O)NCc1cccs1)C1CC1(C)Br 32516,C(=O)(CC1=NNC(=O)C1)NC(C)(CNC(C1CC(CC2CC2)C1)=O)C1CC1 32517,C1(C2(C)CC2)(C(=O)NC(C2C(C(N(CC#C)CC#C)=O)C2)C)CC1 32518,c1(N(C)Cc2c(C)cccc2F)cccc(S(=O)(=O)N2CCC(C(C)C)C2)n1 32519,CCC(CC(=O)NCC(C)(C)NC(c1ccc(CC)cc1C)=O)C(F)F 32520,c1(C(=O)NC(C(CO)NC(c2c(C=C)cnn2C)=O)C)c(F)cc(F)cc1Cl 32521,c1(C(=O)NCC(c2ccccc2)(C)C)cnn2c1OCC1(COC1)C2 32522,N1(C(Cc2ccn(C)n2)=O)CCOCC1CNS(=O)(=O)CC1CCCO1 32523,C1(CCC)C(=O)NCCN1C(=O)C(C)(CSC)NC(C1CN2CCC1C2)=O 32524,c1(OC)ccc(C(N)=O)cc1NC(C1CC(c2ccccc2OC(F)(F)F)C1)=O 32525,N1(C(C(c2cc(C)c(F)cc2)=O)=O)CC2CN(C(=O)C(O)O)CC2C1 32526,Cc1ccc2c(c1)C(C(=O)N1CCN(C(=O)CC3CCC(C)(C)C3)C(C)C1)CC2 32527,c1(OC)ccc2cc(C(N3CCN(C(=O)C(F)=CCCF)CC3C)=O)ncc2c1 32528,C1(CNC(C(C)CNC(=O)Cc2ccc[nH]2)=O)CC12CCOCC2 32529,c1(C(C(=O)NCC(C)CNC(=O)CCC(C)(C)C)C)c(F)cccc1F 32530,c1(C(=O)NCC2(CN(C(CC(C=C)CC)=O)C)CC2)ccc(Cl)c(OC)c1F 32531,CCC(C(=O)N(C)CCOCCN(C(=O)C(C)C1CCC1)C)C(C)C 32532,Cc1ccc(CN(CCCS(C)(=O)=O)C(C2CC(F)(CN)C2)=O)c(O)n1 32533,N1(C(C2CC(SC)C2)=O)CCCC(C2CC2NC(c2cccc3cc[nH]c23)=O)C1 32534,c1(NC(C2C(C(N(C(c3cccnc3)(C)C)C)=O)C2)=O)cc(Br)cc2[nH]ncc12 32535,c1(C(=O)NCC2(NC(CN3CC(C)(OC)C3)=O)CC2)ccc(F)c2c1CCC2 32536,CC1(CO)CCCN(C(=O)C(C2CCN(C(=O)C=CCOC(C)(C)C)C2)F)C1 32537,C1(C(=O)NCCN(C(c2ccc(F)cc2NC)=O)CC)Cc2cccnc2C1 32538,Cc1cc(C(=O)N(CCN(C(=O)C(CO)N(C)C)C)C2CC2)nc(C)c1 32539,C1(C(=O)Nc2c(CC)nc[nH]2)CC2CCC1(N=c1[nH]nc(-c3ccccc3)o1)C2 32540,C1(NC(C2(C)CCNC2=O)=O)CCCN(C(C2CC(F)(F)CS2)=O)CC1 32541,c1(C(N(C)Cc2cn(CCSCC(=O)NC3CC3)nn2)=O)cccc(Br)c1[N+](=O)[O-] 32542,N1(C(C(CNC(C(CC)(C)OC)=O)CC2CC2)=O)CCC(C)=C(F)C1 32543,C1(CNC(CC(C)(C)C)=O)CC(C)(C)CN1C(C1CCC(C(F)F)CC1)=O 32544,Cn1ncc2c(NCCCn3cccn3)[nH]c(=NCC3CC34CCC4)nc12 32545,C1(C(=O)NC(C(=O)OC)C)CC12CC(NC(=O)Cc1cn[nH]c1)C2 32546,C1(C)(C(=O)NCc2c(C(N3CC(c4c(C)nn[nH]4)C3)=O)cco2)CCN(C)C1 32547,c1(N2CCN(C(C(=O)N(CC#C)CC=C)C)CC2)ncnc2sc(C)nc12 32548,c1(C(C(=O)NC(C(C)C)CNC(C2CC3CC3C2)=O)(C)F)ccccc1F 32549,c1(Nc2c(C(=O)O)cn(C)n2)cccc2c1CNC(=O)O2 32550,C(=O)(CC(Cl)Cl)NC1(C(=O)NCCC2(COC)CC2)CSC1 32551,O=S(=O)(c1cc2sc(=NCC3(CCO)CC3)[nH]c2cc1Cl)N1CC(O)C(F)C1 32552,c1(C(=O)NC2(CNC(C(CC#C)O)=O)CCCCC2)ccc(F)c(O)c1F 32553,CC(C)(C)CC(F)C(=O)N1CCC(CCNC(c2ccnn2C2CC2)=O)CC1 32554,c1(OC)ncc(CN2CCC(Cc3cccc(N4CCC(O)C4)n3)C2)cc1Cl 32555,N1(C(C2(C(=O)NC3CC(N(C)C)C3)CC2)=O)C(C(=O)OC(C)(C)C)CCC1(C)C 32556,Cc1nc2ccc(C(N3CC(NC(C4CCC(=O)O4)=O)C3)=O)cc2n1C 32557,c1(-n2c(C(CC)CC(C)C)nc(C3CCCS(=O)(=O)C3)n2)nc2cc(Cl)ccc2s1 32558,n1(CCC)ccc(C(N2CC(NC(=O)CCC3CC3(F)F)C2)=O)n1 32559,N1(C(c2sc3cc(C)sc3c2)=O)CCC(C2CCN(C(=O)CC#N)CC2)C1 32560,C1(O)(CNC(C2(C(C)C)CC2)=O)CCCN(C(c2ccc(O)cc2Cl)=O)CC1 32561,C1(NC(=O)OC2CCCCC2O)CNCCC1c1cccc(F)c1 32562,N1(Cc2c(OCC)cccc2)CC2CN(C(=O)CC3CC4CCC3C4)CC12 32563,C1(C(=O)NC(CCOC2CC2)C(=O)O)C2CN(C(c3ccc(F)cc3)=O)CC12 32564,n1(C2CN(C(C3(Cl)C(C(C)=O)C3)=O)C2)cc(C(c2ccccc2)NC=O)nn1 32565,CCC(F)(F)CC(=O)N1CCC(C2N(C(C3CCCN3CC)=O)CC2(C)C)CC1 32566,N1(C(C2C(C)(C(F)F)C2)=O)CCN(C(=O)CCC2CC2)CC12CC2 32567,c1(-c2onc(CC)n2)cccc(CNC(=O)CC2(NC(C)=O)CCCC2)c1 32568,N#Cc1cccc(Cl)c1NC(C1CN(Cc2nc(Cl)ccc2Cl)CCO1)=O 32569,Cc1cnn(C)c1C(N1CC(C)(NC(=O)C(C)C2CCCC2)C1)=O 32570,Cc1ncnc(C)c1C(=O)NCC(C1CCOC1)NC(c1c(C)cc[nH]c1=N)=O 32571,C=C(Cl)CCC(=O)N1CC(CCNC(C2CC3CCC2C3)=O)(OC)C1 32572,C1(C)(C(=O)NCC2N(C(CCC(C)C#N)=O)CC2)CCCCNC1=O 32573,c1(CNC(C)=O)ccc(C(N2CC(O)(CCNC(=O)CC3CC=CC3)C2)=O)cc1 32574,c1(C(N2CCN(C(c3cn4c(n3)CCC4)=O)C3CC23)=O)ccc(F)c(Br)c1 32575,C(=O)(C1=CC(C)(C)C1)NC(C(c1c(OC)cccc1)NC(C1(SC)CC1)=O)C 32576,C1(CNC(CNS(NC)(=O)=O)=O)CCN(C(=O)C2=CCOC2)CC1C 32577,c1(C(N2CC(O)CC(NC(CN=S(C)(C)=O)=O)C2)=O)cnc2ncnn2c1O 32578,C=CC(CC)CC(=O)N1CCN(C(=O)CN2CCCCC(=O)C2=O)C(CCO)C1 32579,c1(CC)nn(C)c(CC)c1C(=O)NCC=C1CCN(C(=O)C(C)S(C)(=O)=O)CC1 32580,c1(NCC(N2CCCC(CS)C2)=O)ccc[n+]([O-])c1 32581,N1(C(C=CC(CC)C)=O)CCN(C(c2cnncc2O)=O)C(C)C1C 32582,C1(C2=CCCCCC2)(C(N(CCCNC(c2c(C)onc2CO)=O)C)=O)CC1 32583,C1(N(C(CCN(C(=O)CC=C(C)C)CC=C)=O)C)CCCC(O)C1 32584,c1(C(=O)NC(CNC(C(CN(C)C)O)=O)CO)cc(C#N)no1 32585,N1(C(Cc2cc(C)sc2C)=O)CCC12CN(C(=O)Cc1cncs1)C2 32586,N1(C(C2=CCC(NC(C(C(C)C)=O)=O)C2)=O)CCn2ccnc2C1 32587,N1(C(C(C(=O)OCC)OC)=O)CCC(O)(CC(=O)NC2CCN(C(C)=O)C2)CC1 32588,c1(CC(=O)N(CC(=O)NCCCc2ncn(C)n2)CC#C)cccc(C)n1 32589,Cc1c[nH]c(C(=O)NCCOCCC(=O)NCC(C)CCCO)c1C 32590,c1(OC)cc(O)ccc1-c1nc(C)c(NC(c2cnc(SC)nc2Cl)=O)s1 32591,c1(CC(N2CC(N(C(C(C=C)O)=O)C)C(C)(C)C2)=O)cnc2ccccc2c1 32592,C1(C(=O)NC2C=CCN(C(c3ccccc3Br)=O)C2)CC2CC(O)C(C1)C2 32593,C=CCCCCCCC(=O)NCC1CCC1C(=O)NC1CC(C)(CC)C1 32594,N1(C(C(CC)(C)COC)=O)CC2C1CCCN2C(c1cc2ccsc2n1C)=O 32595,C1(NC(C(C)C2CCC2)=O)(CNC(c2c[nH]nc2[N+](=O)[O-])=O)CC2CCC1CC2 32596,C1(C(=O)NCC(=C2CN(c3ncc(Cl)cn3)C2)F)CCc2ccccc2C1 32597,C12(CNC(C3(COC)CCCC3)=O)CCC1CN(C(=O)C1=CCCCC1)C2 32598,c1(C(N2CC3CC3(NC(C3(CF)CC3)=O)C2)=O)ccc(Cl)cc1Br 32599,c1(C(=O)NC(CC)CN(C(=O)Cc2ccoc2C)C)occ(C)c1C(=O)OC 32600,C(=O)(CC(C)n1ccnc1)N(CCC(C)NC(=O)CCc1ccncc1)C 32601,N1(C(CC2CCN(C)CC2)=O)CC2(NC(C3COC(=O)N3C)=O)CCCC2(F)C1 32602,c1(OC)cc(OC)c(C(N2CC(NC(=O)C(C)CF)C(O)C2)=O)c(N)c1 32603,Cc1cc(Br)c2ncnc(N3CCCC(c4n[nH]c(C)n4)C3)c2c1 32604,Cn1cc(Cl)cc1C(c1nnnn1CCN1CCOCC1)NCC1CC(C)(C)CO1 32605,c1(C(=O)OC)cc(C(=O)NCc2cccc(-c3ncc(C)o3)c2)c(C)s1 32606,N1(C(c2ccc(CSC)o2)=O)CC2CCC(C1)N2C(=O)CCC1CCCO1 32607,n1(CC)nc(C(N2CCC(C(C)NC(C3CCCC3C(C)C)=O)C2)=O)c(C)n1 32608,C1(CCNC(CCN(C(COC(C)C)=O)CCCO)=O)CC=CCC1 32609,CC1CC(NC(c2ccc(=O)n(C)c2)=O)CN(C(c2cc(Cl)sc2Cl)=O)C1 32610,N1(C(C(C=C)(C)C)=O)CCC(NC(c2ccc(OC)cc2OC)=O)C(C(C)C)C1 32611,C(=O)(C(F)(F)CCn1cc(C(C)O)nn1)NCc1c(OCCC)cccc1 32612,C1(NC(C(=Cc2ccncc2)C)=O)CCN(C(C2CC2C(F)F)=O)C1(C)C 32613,C1(CNC(c2c(C)cnnc2)=O)CN(C(=O)CC(C)N2CCCC2=O)CC1(C)C 32614,Cc1cccc(-c2cc(C(=O)N(C(C)CNC(C3(C(C)(F)F)CC3)=O)C)on2)c1 32615,C12(C(=O)NCC3CC4(CCC4)CO3)CC(CN(C(c3nn[nH]n3)=O)C1)C2 32616,n1(CC)nc(C)c(C(N2CC(NC(C3(O)CCSC3)=O)C(SC)C2)=O)c1Cl 32617,C1(N2CCOCC2)(C(N(CCN(CC)CC)CCC2CC2)=O)CCCC1 32618,C(C)(CO)(C(=O)NCCC(O)CO)N(C)C(C1CC1c1ccoc1)=O 32619,C1(CNC(=O)C=Cc2ccoc2)CC2CCC1N2C(=O)CCc1cccc(F)c1 32620,c1(CCC(N2C(CNC(C(C)CN(C)C)=O)C3CC3C2)=O)cnc2ncccn12 32621,N1(C(CSCC#C)=O)CC(C)(C)OCC1CNC(c1ccc(N(C)CC)nc1)=O 32622,Cc1ncnc(O)c1CC(N1CCC1CNC(C1(O)CC(F)(F)C1)=O)=O 32623,C1(C(=O)NC(C)CCNC(C2(C#N)CC2)=O)OCC2COCCC12 32624,C12(C(N3C(CCCNC(c4occ(C)c4C)=O)CCC3)=O)CCOC1CCOC2 32625,Cc1c(C(N2CC(O)(CCNC(C3CCN(C(N)=O)C3)=O)C2)=O)c(Cl)nn1C 32626,N1(C(c2cc(C)[nH]c2)=O)CCC2(COCCN2C(=O)C=CC2CCCN2C)C1 32627,C1(C(=O)N(C2(CC(=O)OC)CC2)C)CC(NC(=O)COC2CCC2)C1 32628,n1(C(C)C)ccc(CC(N2CC(NC(c3ccsc3Br)=O)C2)=O)n1 32629,Cn1cc(C(=O)NCCC2(CNC(=O)Cn3ccc(Br)n3)CC2)nn1 32630,CCC(C)N(OC)C(=O)C1CC(NC(=O)C(C)CC#N)C1 32631,N1(C(C(CCF)NC(=O)CC2CCC(O)C2)=O)CCOC2(CCC2)C1 32632,N1(C(CC2N(C(=O)CCc3cnco3)CCCC2)=O)CC(C2CC2(F)F)C1 32633,c1(CNC(=O)NCC(C2CCCO2)O)cncc([N+](=O)[O-])c1 32634,c1(C(=O)NCC2(NC(c3c(CC)onc3)=O)CCC2)cc2cccn2cn1 32635,N1(C(C(CC)NC(N)=O)=O)CC(CNC(c2cncc(C(F)(F)F)c2)=O)C(C)C1 32636,c1(CC(=O)NCC2CN(C(c3c(Cl)ccc(N)c3)=O)C2)noc2ccc(F)cc12 32637,C(CC(C)C)(C(=O)OC(C)C)Oc1c(CNC2C(OC)CC2)ccnc1 32638,C(=O)(CCC(C(C)C)NC(c1cc(C(C)C)[nH]n1)=O)NC(C(=O)NCC(C)C)C 32639,C(=O)(C#CC1CCCOC1)NC1CC2CN(C(Cc3n(C(C)C)cnn3)=O)CC21 32640,c1(CC(=O)NCC2CCN(C(=O)CSC3CCCCO3)C2)ccc(Cl)nc1F 32641,c1(C(C)C(N2CC(O)(CNC(c3cnco3)=O)C2)=O)ccc(F)c(F)c1 32642,C1(NC(CCOCCC)=O)CN(C(c2cnc(S)n2C2CC2)=O)CC1OC 32643,C(C(C(=O)NC(c1cscn1)C)C(C)C)NC(c1ncc(C)nc1)=O 32644,c1(C(=O)NCc2c(CC)cns2)cc(-c2cccnc2)ncn1 32645,C1(C(=O)NCCC(C)NC(C2CC(=O)N(C)C2)=O)CC(C)(C)C1C(F)(F)F 32646,N1(c2c(C)cncn2)CCOC2(CCCN(C(=O)C(F)C(C)(C)O)C2)C1 32647,CC(O)C(C)(C)C(=O)N1CCC(OCC(=O)Nc2cnn(C)c2C2CC2)C1 32648,C1(CCC(N2CC3C(c4cn(C(C)(C)C(N)=O)nn4)C3C2)=O)CC2(CCC2=O)C1 32649,N1(C(CC2CCC(OC)CC2)=O)CC(C2CN(C(=O)C(C)(CO)OC)C2)C1 32650,N1(C(c2cnc(-n3cncn3)nc2)=O)CC2(CC(C(F)F)C2)C1 32651,N1(C(C(C(C)C)C)=O)CC2(CC(CNC(C3CC3c3cnn(C(C)C)c3)=O)C2)C1 32652,c1(C(=O)NCC(CNC(C(C)CN2CCCCC2)=O)CO)cccc(N)c1F 32653,N1(C(C(C)NC=O)=O)CCN(C(C2CCCC2)=O)CC1c1ccnn1C 32654,C=CCC(C(=O)NCCCN1CCC1)NC(C1OCCOC1C)=O 32655,c1(CC)c(C(=O)NC2(CO)CN(C(=O)C3=CCCCC3)C2)sc2ccccc12 32656,CC(C)CC(C)CC(=O)N1CC(C)N(C(=O)CC2CC(C)(C)CO2)CC1C 32657,Cc1ncc(Cl)c(C(N2CCC(O)(CNC(C3CC4COCC4C3)=O)C2)=O)n1 32658,Cc1cc(C(=O)NC2CCC2CNC(C2(N=[N+]=[N-])CC2)=O)cnc1C(F)F 32659,c1(C(=O)NCC2C3(CN(C(c4nc(C)oc4)=O)C3)CC2)cc2n(n1)CCCC2O 32660,c1(C(=O)NCC2CCN(Cc3c[nH]c4cccnc34)C2)ccc2c[nH]nc2c1 32661,c1(C(=O)NC2(C(=O)NCCC(O)C3CC3)CCCC2)cccc2[nH]ccc12 32662,c1(OC)nccc(C(N2CC(NC(=O)C(C)C)C(C)C2)=O)n1 32663,CC1CCC(C)(C)N1C(C1CCN(c2ccncn2)CC1)=O 32664,c1(CCC(=O)OC)ccc(NC(=O)C(=O)NC(C2CCC(C)C2)C2CC2)cc1 32665,CC1CCN(C(C2CC(O)(C#N)C2)=O)C(C)C1NC(C1CN(C(N)=O)C1)=O 32666,c1(C(N2CC(NC(c3cc(OC(C)C)ncc3)=O)C2)=O)nc2cc(F)ccc2s1 32667,C1(C(C(C)NC(=O)N(C)C(c2ccco2)C)(C)C)Cc2ccccc2O1 32668,CC(C)(O)C(F)C(=O)NCC1CN(C(C2CC(=O)N2)=O)C1 32669,c1(C(N2CCN(c3nc(C)cc(SC)n3)CC2C)=O)ccnc2c1OCO2 32670,c1(CC)ccccc1-c1cn(CC2CCCC2NC(c2cnnn2C)=O)nn1 32671,c1(C(=O)NC(CNC(c2ccc(C)nn2)=O)C2CCC2)c(C)nn(C(C)C)c1C 32672,c1(CN(C(CCC)=O)C)cnn2c1CN(C(=O)C(C)SC)CC2 32673,CC1CCC(NC(c2cccnc2O)=O)CN1C(=O)CC1(NC(C)=O)CC1 32674,CC(CN=c1[nH]c(=NCC2CCC3(CCC3)O2)[nH]c2c1CCCC2)C1CCCC1 32675,C1(OC)CCC(C(N2CC3CC3(NC(=O)C=C(C)C(F)F)C2)=O)CC1 32676,C1(CNC(C2CCCCCC2)=O)CCC2(CO1)CC(NC(C1CCSC1)=O)C2 32677,C1(CC(=O)NCC(CN(C(C(c2ccc(C)cc2)O)=O)C)O)CCC(C)(C)CC1 32678,N1(C(c2nc(C(C)OC)sc2)=O)CCCC1(C)CNC(c1ccnn1C)=O 32679,CC1(C)CC(C(N2CCN(C(=O)C=Cc3ncc[nH]3)C(CO)C2)=O)C(C)(C)O1 32680,C12CCCC(C1)NC2=O.C1(CC#N)CN(C(=O)CO)C1 32681,C1(n2cc(CNC(CCSC)=O)nn2)CCN(C(=O)OC(C)(C)C)CC1 32682,c1(C(=O)NCC2C(NC(c3c(N)n(CCO)nc3)=O)CC2)cccc2sccc12 32683,c1(C(N(C)CCOCCNC(C2(O)CC3CCC2C3)=O)=O)ccc2cn(C)nc2c1 32684,CCCCC(O)CC(=O)NC(C(N1CCCC(C)C1)=O)C1CC1 32685,N1(C(C2CCC(=O)N2)=O)CCCN(C(c2cc(-c3cccnc3)no2)=O)CC1 32686,C1(NC(CC(COC)C)=O)CC2CC1CN(C(c1ccncc1Br)=O)C2 32687,C(c1ccc(C(F)F)o1)=CC(=O)NCC(CCNC(C(c1cn(C)nc1)O)=O)O 32688,N1(C(C=C)=O)CCc2nc(C(N3CCC(NC(C)=O)CC3)=O)cn2CC1.c1cn[nH]c1 32689,C=C(C)C1OCCC1CNC(=O)C(C1CCCCC1)NC(C1C=CC1C(=O)OC)=O 32690,N1(C(C(N2CCCC(C)C2)=O)=O)CCCC(C)(C(=O)Nc2ncccc2OC)C1 32691,CC(CCCc1ccccc1)C(=O)N1CCC(N(C(=O)C2=C(Cl)CC2)C)CC1 32692,c1(OC)cc(C(N2CCC3(NC(=O)C=C(C)C(C)(C)C)CC3C2)=O)c(Cl)cc1Cl 32693,Cc1ccc(F)cc1C(N1CCOCC1CN(C)C(C1(F)CCCN(C)C1)=O)=O 32694,C(=O)(C1=NOC(CNC(=O)CC(C)n2ccnc2)C1)NC1(C(COC)O)CC1 32695,Cc1cc(CC(=O)NC2COCC2NC(=O)CC(C)F)ccc1CO 32696,C1(C2=CCOCC2)(CNC(c2sc(Br)nc2C2OCCO2)=O)CC1 32697,C(=O)(C(CCF)NC(=O)C(c1cnn(C)c1)=O)NCc1ncc(C)[nH]1 32698,c1(C(=O)NC(C2(O)CNC2)C2CC2)c[nH]nc1-c1ccccc1.CO 32699,Cc1ccc(CC(=O)NC2CC(NC(=O)C(C)(C)OC(C)C)C23CCC3)cc1O 32700,c1(CC)nc(C)c(C(=O)NC2CCCC(NC(=O)CCC#N)C2)c(C)n1 32701,C1(CNC(=O)NC(C#CC)(C)C2CCC2)(CNC(=O)OC(C)(C)C)CCC(=O)N1 32702,c1(CC)nc(C)c(CC(=O)NCCCCNC(C2CS(=O)(=O)CCO2)=O)c(C)n1 32703,c1(OC)ccc(CC(=O)NCCC2CCCC2(C)C)c(O)c1 32704,N1(C(C2N(CCCC)CCCC2)=O)CC(NC(c2cc(C)[nH]c2C)=O)C(C)(C)C1 32705,C(=O)(C1=CCCN(C(=O)CC=C(Cl)Cl)C1)N1CC(C)(OC)C1 32706,C1(C)(C(N(C(N(CC(C)O)C(C)C)=O)C(C)C)=O)CCN(S(C)(=O)=O)CC1 32707,c1(C(=O)NC(CC)CNC(=O)C=CS(C)=O)cnc2cnc(Cl)cc2c1 32708,N1(C(c2c(C)coc2)=O)CCC2(CCN(C(=O)CC3COCCOC3)C2)C1 32709,c1(C(N(C)CC2CCN(C(c3nccnc3N)=O)C2)=O)cncc2nc[nH]c12 32710,C=C(Cl)C(C)(C)C(=O)NCC(C1CCCN(C(c2ncncc2F)=O)C1)(C)O 32711,C(CC(O)CNC(c1n[nH]cc1Br)=O)NC(C1CC(C(=O)OC)C1)=O 32712,c1(CC)conc1CC(=O)N(CC(O)CNC(c1sncc1C)=O)C 32713,C1(NC(c2cc(F)c(Cl)cc2F)=O)CCCCCN(C(c2cc(CO)[nH]n2)=O)C1 32714,C=CCC(CC(F)F)C(=O)NC(CNC(c1cc(CC)cc(N)c1)=O)C(C)(C)C 32715,c1(C(N2CC(CNC(C3(C)CC3)=O)OCC2)=O)cc(F)c(C#N)c(F)c1 32716,CC1CN(C(=O)CCCF)CCC1CNC(c1cc(Cl)ccc1Cl)=O 32717,c1(CN(C(C2CC(CCNC(c3ccc[nH]3)=O)C2)=O)CC)cnc[nH]1 32718,C(CCCCCC(=O)NCCC1CC(C)=NO1)NC(c1n(CC)nc(C)c1)=O 32719,c1(C(=O)NC(C2CCCN(C(=O)CCNC(=O)CO)C2)C)ncnc(O)c1F 32720,CC(CO)(C1CCC1)NC(=O)NC1CCC1OC(C)(C)C 32721,C1(C(C)C(=O)NC(C)(CO)C2CCCC2)CCN(C(=O)COC2CCCOC2)C1 32722,N1(C(CCOC(C)C)=O)CCCC2(NC(c3cc(Br)nn3C)=O)CC2C1 32723,C=Cc1ccc(C(=O)NC(C)CC2CCN(C(=O)C(CC)NC(N)=O)CC2)cc1 32724,C1(CCC(=O)N(CC(C)N(C(CCCC)=O)C)C)CCCC(O)C1 32725,N1(C(CC(=C)C)=O)CCN(C(c2ncc(F)cc2N)=O)C2CC12 32726,C=C(Br)CC(C)(C)C(=O)NC(c1ccccc1)CNC(c1cccc(C)n1)=O 32727,c1(C(=O)NCC(C)(CNC(c2cncs2)=O)OC)cc(Cl)cnc1C 32728,N1(C(C(CC2CCCCC2)OC)=O)CC2CCC(C1)N2C(=O)C1=CC(O)CCC1 32729,C1(N(C(C(C)NS(CC)(=O)=O)=O)Cc2ccn(C)n2)CC2CCC(C1)N2 32730,C1(NC(C2(OC)CCCCC2)=O)CCN(C(c2cc(Cl)c[nH]2)=O)CC1C 32731,n1(C(C)C)ccnc1C(=O)NC(C)(C)CC=CC(=O)NC1(c2cccnc2)CC1 32732,S(=O)(=O)(c1cc(C)c(C(=O)O)o1)N(CCOC)CCO 32733,CC1=C(CNC(=O)CC2C=CC(NC(=O)C(c3ccccc3)O)C2)COCC1 32734,c1(C(N2C3C(NC(C4CC(=C)C4)=O)CC(CC3)C2)=O)ccc2cc(Cl)ccc2n1 32735,c1(C(N2CCC(N(C(=O)C3=CCCO3)CC)C2)=O)cccc2nccn12 32736,Cc1nnc(CCC(=O)NC2CC(CNC(=O)C(c3ccc(Cl)cc3)=O)C2)n1C 32737,C(=O)(CCC(C)(C)NC(c1cccc(F)c1N)=O)N(CC(O)C1CC1)C 32738,N1(C(c2cn(CCC)nc2C)=O)CCC(C)(NC(c2n[nH]c(C)c2C)=O)CC1 32739,C(CCO)(C(C)(C)O)NC(C1(CNC(c2c(COC)cc[nH]2)=O)CCCO1)=O 32740,CCC(O)C(C)(C)C(=O)NCC(CNC(=O)COC(CC)CC)C(F)(F)F 32741,c1(C(N2CC(N3CCC3)CC(C)C2)=O)ncc2cc(Br)ccc2n1 32742,N1(C(CC(CC)C2CC2)=O)CCC2C(NC(c3c(C)nn(CC)c3Cl)=O)CC12 32743,Cc1cc(Cl)ccc1C(N1CC(CNC(c2cnc3n2CCC3)=O)C2(CC2)C1)=O 32744,c1(C(=O)NCC23N(C(C(C)=C4CCC4)=O)CC(C2)C3)ccc(C)cc1N=[N+]=[N-] 32745,c1(C(=O)NCCCNC(c2c(C)ccc(OC)n2)=O)nccc2c1NCCC2 32746,c1(NCC2(NC(=O)CNc3ccncc3)CCCCC2)ncc([N+](=O)[O-])cn1 32747,CC(C)(C)CC(=O)NCC12COC(CNC(=O)CSc3cccnc3)(C1)C2 32748,c1(N(c2c(OC)c(F)ccc2)C(C2CC3CCCCN3C2)=O)ccnc2ccnn12 32749,c1(COC)nc(NC)cc(N2CCC(CCCO)CC2)n1.C(C(C(C)C)N(C)C)OC 32750,N1(CC(N2CC3C(C(N4CCC(C(=O)OC)C4)=O)(C3)C2)=O)C(=O)CCCC1=O 32751,c1(CCC)ccccc1C(=O)NC(C)C(C(C)C)NC(c1ccc(O)nn1)=O 32752,C1(C(=O)NC(CNC(c2c(C)cc(CC)o2)=O)(C)CO)CCCCCN1C 32753,CC1OCCCC1C(N1CCC(N2CCN(C(=O)C(C)(C)C3CC3)CC2)C1)=O 32754,Cc1cc(=NC2CN(CC3CC3)C2)[nH]c(N2CCc3n[nH]cc3C2)n1 32755,CCC(CC)CC(=O)NCC(C1(O)CN(C(=O)CCF)C1)(C)C 32756,C(C(C)C)(C(O)C(=O)NCC=CC(=O)NCC1CCC(C)(C)CC1)OC 32757,C1(C(=O)NC2CN(CC)C(=O)C2)CCC(C)(C)N(C(=O)CN(C)C2CC2)C1 32758,N1(C(c2cn(CCCC)nn2)=O)CCC2(CCCCN(C(=O)C(C)C(F)F)C2)C1 32759,Cc1cc(N)cnc1C(=O)NCC(C)NC(c1cnsc1C)=O 32760,CC1CC(NC(c2cnc(-c3cccnc3)s2)=O)CN(C(=O)CC2CC=CC2)C1 32761,C(C)(C)(CCC(=O)NCCCCOC(C)C)NC(C(COCC)C)=O 32762,C1(CNC(C(C)OCC=C)=O)CCN(C(C2CC2c2cccc(Cl)c2)=O)CC1 32763,C1(NC(c2cnn(C(C)(C)C)n2)=O)CCC(C)(CNC(=O)C=Cc2ncc[nH]2)C1 32764,C12(CCNC(=O)C=Cc3cnc[nH]3)CCC1CN(C(c1cc3sccc3[nH]1)=O)C2 32765,N1(C(C(CC=C)C)=O)CCC2CN(C(c3ccccn3)=O)C(C)C12 32766,C(CCC(C(=O)N1CCN(CCF)CC1)NC(=O)CC1CCOC1C)OC 32767,C1(C(N2CC(N(C)C(c3cnn(C)c3)=O)C(C)(C)C2)=O)(OC)CCCCCCC1 32768,C1(C(=O)NC(C(C)C)CNC(=O)CC2CCN(C)C2=O)CC(=O)OC1(C)C 32769,C1(C(=O)NC(C2N(C(c3c(CC)c[nH]n3)=O)CCC2)C)CSc2ccccc2O1 32770,CC1(C)OC2(CNC(C3(C4CCCO4)CCCO3)=O)CC1(NC(=O)CCF)C2 32771,n1(CCN(CCCC)CC)cc(C(C)(C)F)nn1 32772,N1(C(CS(CCOC)(=O)=O)=O)CCC2(CC1)CN(C(C1CC1OC)=O)CCO2 32773,C1(C(N2CC(COC)OCC2)=O)C(C(=O)O)C2CCC1(C)C2(C)C 32774,CCCC(CNC(=O)CC1CC(C)=NO1)NC(=O)C=C(C)C(C)C 32775,C1(NC(c2ccc(C)cc2C)=O)CN(C(=O)CC2CN(C)C2)C2(CCCC2)C1 32776,C1(NC(c2nc(CCC)sc2)=O)CC2CCC1C(NC(c1cc(C#N)cs1)=O)C2 32777,c1(C(CN(C(C)C)Cc2cccs2)=O)ccc2c(c1)CCCN2 32778,c1(C(N(CCC)CCNC(=O)CN2CCOCC2)=O)ccc(O)cn1 32779,CCCC(C)(c1nnnn1CCCF)NC1CCC1(C)C 32780,C1(NC(CCn2c(C)cc(C)n2)=O)CC2CCC(C1)N2C(c1ncccc1C)=O 32781,c1(CC)oc(C)cc1C(=O)N(CCCC(=O)NCCC(F)F)C 32782,c1(C(=O)NC2CCCN(C(=O)C(C3(O)CCCC3)F)C2)cc2nc(F)ccc2o1 32783,Cc1sc(=O)n(CC(=O)NC2CCC(C)N(C(=O)CNS(=O)(=O)C3CC3)C2)c1C 32784,N1(C(=O)COC2COC2)CCC2CCN(C(=O)COC(=O)CO)C2C1 32785,c1(C(=O)NC(C)C(CO)NC(c2ccc[nH]2)=O)cccc(-c2cnco2)c1 32786,C(=O)(C1CCCc2nnn(C)c21)N1CCCN(C(c2c(C#C)c[nH]n2)=O)CC1 32787,N1(C(Cc2c(C)cc(C)s2)=O)CC2(CNC(C3(C)CCCCC3)=O)CC(F)(C1)C2 32788,CC1(C)CCOC1CNC(C1CCCN(C(=O)CNC(N)=O)C1)=O 32789,c1(C(N(C(C)CNC(=O)CCCc2cncs2)C)=O)cc2c(O)ncnc2cn1 32790,Cc1cc(NC(=O)CC2C(NC(C3C(C)(C)C3(F)F)=O)CC2O)cc(CO)c1 32791,C(=O)(C1Cc2ccc(C)cc21)N1CCN(C(c2cc(COC)on2)=O)CC(O)C1 32792,N1(C(c2c(C)nc(CC3CC3)o2)=O)CC2(CCN(C(=O)C3=CSCS3)CC2)C1 32793,N1(C(CN(C)CC)=O)C2CCC1CC(CCNC(c1cnn(C)c1C(C)C)=O)C2 32794,C1(=O)C(C(C)(C)C)n2cc(nn2)C2CCN12.c1(CC)n[nH]c(C)c1C(C)C 32795,C(=O)(C(F)CC(C)C)N(C1CCN(C(=O)CN(C)C(N)=O)CC1)CCCC 32796,C=CC(CC)CC(=O)N1CCC(C)C(CC(=O)NCC(C)CC2CCCC2)C1 32797,C1(NC(CCn2ccc(C)n2)=O)C2CC3CN(C(C4OCC4(C)C)=O)C1C3C2 32798,C1(C(N2CC(NC(=O)C=C3CCCC3)C2)=O)CC12CCCc1ccccc12 32799,C1(NC(C2CC(OCC)C2)=O)CC(NC(C2(C(C)(C)C)CCCC2)=O)C12CCC2 32800,C(=O)(CC(O)CCSC)NC1CCN(C(c2ccc(CC)nc2)=O)C1C1CC1 32801,C12(NC(c3nc(C(C)(C)C)oc3)=O)CCCN(C(=O)C3=CCC3)CC1C2 32802,c1(CNC(C2ON=C(C)C2)=O)cccc(CNC(c2cnc(C3CC3)[nH]2)=O)c1 32803,c1(CN(CC(c2ccccc2)(C)C)CC)c(SC(C)CO)cccc1F 32804,c1(-c2n(C)ncc2)cccc(C(=O)NC2CC(NC(=O)C=CC(F)F)CC2O)c1 32805,CC12CN(CCO1)C2=O.C1(CNC(=O)CC2CCCCC2)COCCN1C=O 32806,N1(C(Cc2nnc(C)o2)=O)CCC(NC(=O)CCC2CCCN(C)C2)CC(O)C1 32807,c1(C(N2C(C(=O)NCC3COCCO3)CCC2)=O)cc([N+](=O)[O-])cs1 32808,c1(OCC(=O)N(C2CCN(C(C(C)=CC3CC3)=O)C2)CCO)c(C)cccc1Cl 32809,C1(C)(C(=O)NCCCN(C(C2CCc3ncnn3C2)=O)CC)CC(C2CC2)=NO1 32810,N1(C(C(C)(C)OCC)=O)CCN(C(c2c[nH]cc2CC)=O)CC(O)C1 32811,O=S(=O)(c1cccnc1NCC1CC2(C1)OCCO2)N1CCCC1CF 32812,c1(C(N2CC(C)N(C(C3OCCO3)=O)CC2)=O)ccn2ccnc2n1 32813,Cc1onc(-c2cccc(F)c2)c1C(=O)NC1CC1NC(c1coc(Cl)n1)=O 32814,c1(NC(C2C(CNC(Cc3n(C)ccc3)=O)C2)=O)cnc2[nH]cnc2c1 32815,c1(CNC(=O)NC(c2cn(C)nn2)c2cccs2)cc(Cl)ccn1 32816,c1(-c2cn(CC3N(C(CC(CC)C(F)F)=O)CC3)nn2)ccc2nccnc2c1 32817,C(=O)(CCS(=O)(=O)c1ccc(OC)cc1)NC(CNC(C(CCCC)(C)F)=O)C 32818,c1(C(=O)NC(C(C)NC(c2cccc3ccsc23)=O)C)ccc2c(c1)CCOC2 32819,c1(C(=O)OCC(=O)NC2C(Cc3cc(C)no3)=CC=C2)cc(F)c(O)c(Cl)c1 32820,N1(C(CCC(=O)OC)=O)CCCC(C2CC2NC(=O)Cn2nccn2)C1 32821,c1(C(=O)NC2CN(C(C3CCN(C)C3)=O)CC2F)cccc2c1CCC2 32822,N1(C(CC23C(C)(C)C(CC2)CC3)=O)CCCC(C2(NC(=O)C(O)C3CC3)CC2)C1 32823,c1(CN2CCC(c3n(CCSC)nnn3)(NC(C)=O)C2)n[nH]c2c1CCCC2 32824,c1(C(N2CCC(N(C(CN(CCC)C)=O)C)CC2)=O)ccc2c(c1)C(C)C(C)O2 32825,C1(C(N2C(C(=O)NCc3cccnc3O)CCC2C2CC2)=O)CC2(C1)CC(O)C2 32826,C1(C(N2CCC(N(C(C(N3C(=O)CCC3=O)C)=O)C)CC2)=O)C(C2CC2)C1(F)F 32827,c1(-c2c(C)cc(C(N3CC(C)(C)OCC3C3CC3)=O)s2)ccc2c(c1)ncn2C 32828,CCC(C(=O)OC)NC(c1csc(CNC(c2cnn[nH]2)=O)c1)=O 32829,CC(C)C(C)C(CNC(C1CCSCC1)=O)NC(c1cc(=O)n(C)o1)=O 32830,N1(C(C2(C)SCCCS2)=O)C(CC(=O)NC(C)(C)CC(C)(C)O)C2CCCC12 32831,C(=O)(C1=CC2(CCOC2)C1)NCC1(NC(c2c(C)ncnc2)=O)CCCCCC1 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32867,C(CC(O)CC(=O)NCCC1(O)CCCN(C(c2cn[nH]c2)=O)C1)SC 32868,N1(C(c2ccccc2)=O)CCCC(C2CCCN(C(C3CC(O)C3)=O)C2)C1 32869,N1(C(COCC)=O)CCCC(C)(CNC(=O)C2=CCCC2C)C1 32870,C=C(C)CCC(=O)NCC(C1CCCCC1)NC(=O)COCc1cccnc1 32871,c1(C(N2CC(N(C)Cc3n(C(C)C)c(S)nn3)C2)=O)ncc(Br)cc1Br 32872,c1(C2N(C(C3CC4(CC4)C3)C(=O)NC3COC3)CCC2)ccc(Cl)c(F)c1 32873,C1(C(=O)NC(COC(C)C)C)CC1C1CN(C(C2CC(C(C)C)C2)=O)C1 32874,CC1=CN2C(C(=O)NCCCCN(C(=O)CC3CC4CC4C3)C)(C=C1)CC2 32875,N1(C(c2c(C)ccs2)=O)CC2CC(CNC(=O)CCc3cncc(F)c3)CC1C2 32876,Cc1ccc(C(=O)NC(C)CCNC(=O)COCC2CCCO2)c(N)c1F 32877,c1(C(N2CCC(NC(CCS(=O)(=O)NC)=O)C(F)C2)=O)cnc2c(c1)CCCO2 32878,C1(NC2(CS(C)(=O)=O)CC2)CCN(C(c2coc(-c3csc(C)n3)c2)C)CC1C 32879,c1(C(C)F)ccc(C(=O)NCC(C)N(C(=O)CSCC(N2CCCC2)=O)C)cc1 32880,C(=O)(C(O)C(F)(F)F)NCC1CC(C)N1C(=O)CC(C)(C)C 32881,CCC(Cc1ccccc1)C(=O)N1CC(C)(NC(=O)CCC(=O)NC)C1 32882,N1(C(C(=O)NCc2ccc(F)cc2)CC2CCCO2)CCCC2CC(O)CCC12 32883,Cc1nc(O)ccc1C(N1CCC(C)C1C(=O)Nc1cnn(CCF)c1)=O 32884,C1(NC(C(C=C)O)=O)CCN(C(c2c(OC)noc2C2CC2)=O)CC12CCC2 32885,c1(OC)ccc(C(=O)NCC2CN(C3CC3)C(=O)O2)nn1 32886,CCCC(F)C(=O)NCCOCCCN(C)C(C1CCC1C#N)=O 32887,C(C(=O)N1CCOC2(CCC2NC(c2ccoc2)=O)C1)(c1ccccc1)=C(C)C 32888,CC(C)CC(CC(C)C)C(=O)NCCC(C)N(C(=O)CCc1ncc(F)cn1)C 32889,CN1CC=C(CCNC(=O)C(O)CNC(=O)CC(=O)N(C)C)CC1 32890,c1(SCC(N2C3CC(NC(C=CCC)=O)CC2CC3)=O)nc2ccc(C)cc2[nH]1 32891,C1(CNC(C(C)(C)SC)=O)CN(C)CCN1C(c1cc(Cl)sc1Cl)=O 32892,C1(=CCNC(C(C)C2CCCC2)=O)CCN(C(=O)CN2CCCCCC2)CC1 32893,CC(F)(F)C(C)(C)CC(=O)NC1(C)CCCN(C(=O)CCCNC(N)=O)C1 32894,C(=O)(C1Cc2ccccc21)NC(CCC(C)C)C(=O)NC(CO)C(=O)NC1CC1 32895,c1(C(N(CCC(=O)NCCSC)CCC)=O)cn(C2CC2)nc1C 32896,N1(C(CC2CCC(=O)C2)=O)CC2(CCC(CNC(c3ccoc3)=O)O2)C1 32897,C1(C(=O)NCC2(NC(c3cnc(-c4cccnc4)s3)=O)CC2)CCC2(CC2)C1 32898,C1(O)(CN(C(C2CCN(C)C2)=O)C)CCN(C(=O)CCc2cnn[nH]2)CC1 32899,c1(NC(c2ccn(CCO)n2)c2nnnn2CCC2CC2)cccc2[nH]ccc12 32900,C1(C)(COC)CC(NC(C2CN(C)C2)=O)CN1C(=O)CCc1nncs1 32901,CCCC(CCC)CC(=O)N(C(C)C(=O)NCCCCCO)C1CC1 32902,c1(C(=O)NC2(CNC(C3C(CC)C3)=O)CC2)cncc(Cl)c1C 32903,N1(C(c2c(CC)noc2)=O)CC2CC(C)N(C(c3cn(C)nc3Br)=O)C2C1 32904,c1(OC)cc(F)cc(C=CC(N2CCCC2CNC(c2cc(Cl)cc(Cl)n2)=O)=O)c1 32905,c1(C(N2CC3(CC(NC(C4(F)CC4)=O)C3)C2)=O)ccc2nc(O)oc2c1 32906,C#Cc1cc(F)c(CN2CCN(C)C(CO)C2)c(F)c1 32907,N1(C(C2(SCC)CC2)=O)CC2CCCC2(NC(c2csc(S(N)(=O)=O)c2)=O)C1 32908,C1(OCC)CC2(CCN(C(=O)CC=CC(C)(C)C)C2)C1.C12C(C1(C)C)NC2=O 32909,c1(NC2CC(NC(C(C)Sc3ccccn3)=O)C2)ccnc2ncnn12 32910,CC(C)(CNC(=O)CC1(C(=O)NS(C)(=O)=O)CCCC1)CNC(C1C=CCC1)=O 32911,C1(C)(C(=O)NCC(COC)OC)CCCN1C(c1c[nH]c(=O)cn1)=O 32912,C(=O)(N=c1c(Cl)c[nH]cc1Br)C1C=CC(NC(c2c(C)noc2)=O)C1 32913,C(=O)(CCCCN=[N+]=[N-])NCC=C(C(N1CCC(C(=O)OC)CC1)=O)C 32914,Cc1cc(C(=O)NC2C3CC2N(C(=O)C(C)OCc2ccncc2)C3)cc(C)n1 32915,N1(C(=O)NC2C3(CCC3)C23CCC3)CCC2CCC(O)C1C2 32916,Cn1nncc1CC(=O)N(CCO)CCNC(N)=O.C(C(F)(F)F)O.C1C(=O)N1 32917,c1(C(N2CCC(CNC(C3C(OCC)C3)=O)C2)=O)ccc(-c2ccc(Cl)s2)cn1 32918,C1(NC(c2ccsn2)=O)C2CC3C1C3C2C(N1CC(n2cccn2)C1)=O 32919,N1(C(C2CN(C(Cc3nc(C)sc3)=O)C2)=O)CCN(c2ccc(F)cc2)CC1 32920,C(=O)(C(O)C(F)(F)F)N(C)CC1COCCN1C12CC1(CC)CC2 32921,c1(CNC(C2CCCN2C(=O)C2=C(Cl)CCC2)=O)ccc(NC2CC2)cc1Cl 32922,c1(N(C)CCn2cccn2)ccnc(NCC2CC2(F)F)n1 32923,C1(N(C(C2(CC)CCC2)=O)C)CC2CCC(C1)N2C(c1occ2c1CCC2)=O 32924,C1(OC)CC(CNC(=O)CCNC(=O)CO)(NC(=O)CC2CCCC2C)C1 32925,C=CCCCCCCCCC(C(=O)NC1CCC1)N(C)Cc1cnn(C)c1C 32926,N1(C(C(=O)NCC(=C)C)C2=CCSC2)CCc2c(C)cccc2C1C 32927,N1(CC)CCC(C(=O)NC(c2nocc2C(=O)N(CC(O)C2CC2)C)C)C1 32928,c1(CN(C)C(N)=O)cn(CCCN(C(=O)CN2CCCC2)C2CC2)nn1 32929,c1(N2CCC(CNC(C(C)CN3CCOCC3)=O)C2)cccc(O)n1 32930,S(=O)(=O)(c1ccc(Br)cc1)NCC(=O)NCCNC(c1cccc(CO)c1)=O 32931,N1(C(c2c(CSCC)cccc2)=O)CC(C2CN(C(=O)CCCCC(N)=O)C2)C1 32932,N1(C(c2cnc(Br)s2)C(=O)NCCSC)CCCC(n2cc(C)cn2)C1 32933,N1(C(CCCCSC)=O)CC(NC(c2nc(C3CC3)ncc2Cl)=O)C(C2CC2)C1 32934,c1(CC(=O)NC(CC)CN(C(=O)C(C2CC2)SC)C)cc(F)ccc1C 32935,N1(C(c2ccc(CSC)cc2)=O)CCCN(C(=O)COC(F)(F)F)C(CO)C1 32936,N1(C(c2ccn(C(C)(C)C)n2)=O)CCOC(CCNC(c2nocc2Cl)=O)C1 32937,C(C(C(C)(C)C)NC(C1(C)CCCO1)=O)NC(=O)Cc1csc(C(F)(F)F)n1 32938,CCC(C)(C)CC(C(=O)NCc1ccc(F)cc1)N1CCN(C)CC(CO)C1 32939,c1(CC)ccc(CNC(=NCC2CCCCO2)NC2CC(OC)C2)cc1 32940,Cc1c(CC(C)NC(C)(CC(C)C)c2nnnn2C2CCCCC2)cccc1Br 32941,N1(C(C(c2cc(C)c(C)s2)NC(=O)OC(C)(C)C)=O)CCCC(C2(C)CC2)C1 32942,C(CCF)(C(=O)NCCF)NC(C(CC)NC(=O)CCC)=O 32943,C(=O)(C1=C2CCCN=C2NN1)NC(CCCOC)c1cccnc1 32944,C1(C(N2CCC(=CCNC(C(CCC)NC(N)=O)=O)CC2)=O)CCCS(=O)(=O)C1 32945,C1(COC)CN(C(c2cc(C#N)oc2C)=O)CCN1C(=O)C1=C(Cl)CCC1 32946,C1(OC)CCn2cc(C(=O)NCC3CCC(NC(=O)CC(C)(C)C)CC3)nc2C1 32947,C(c1cncnc1O)=CC(=O)NCC1(CNC(=O)CC(F)(F)F)CCOC1 32948,N1(C(c2ccc(CC)nc2)=O)CCOCC(CNC(=O)CC2CCC(F)(F)C2)C1 32949,N1(C(c2n(C)cnc2)=O)CCOC(C2CN(C(C3CC=CCC3)=O)C2)C1 32950,C1(CC)CCC(O)(C(N2CC(N(C)C(c3ccc(-c4ccccn4)s3)=O)C2)=O)C1 32951,N1(C(C(C)N(C(C(CCCC#C)C)=O)CC)=O)CC2CCC1C(O)C2O 32952,c1(C(N(CCCCNC(C(CCC)O)=O)C)=O)cc(F)cc2c1NCCC2 32953,C1(C(N(CC(CNC(C(C)C2(O)CCC2)=O)(C)C)C)=O)CCCC1P(C)(C)=O 32954,c1(C(=O)NCCCOCCN(C)C(c2nnn(C)n2)=O)cc2ncn(C)c2cn1 32955,c1(CN2CCC(N(C(=O)CCCN3CCCCC3)CC)C2)ccc2nonc2c1 32956,Cc1cc(C(=O)NCC2CCC(NC(=O)CCCCNC(N)=O)C2)c(C)cn1 32957,Cc1nn(CCC#N)c(C)c1C(=O)NCCCc1cn(CCCS(N)(=O)=O)nn1 32958,CC(C(C)(C)C)=CC(=O)NCCCOCCC(=O)NCC1=CCCC1 32959,c1(C(=O)NCC(C)NC(C(c2cccc(OC)c2)O)=O)cc2nc(F)ccc2o1 32960,C1(NC(CC2C=NN(C)C2=O)=O)C2CC3C1C3C2C(=O)NCCCOC(=N)O 32961,[N-]=[N+]=NC1CCCN(C(c2csc3ccccc23)=O)C1 32962,C(c1cnc2ccccc2n1)=CC(=O)NC1C2CN(C(CC(C)(C)O)=O)C1CC2 32963,c1(C(=O)NCCCOCCN(C)C(c2ccccn2)=O)cc(Cl)cs1 32964,Cc1cc(C(=O)N(C2CN(C(=O)CN(C)C)CC2(C)C)C)c2nc(C)n(C)c2n1 32965,C1(C(=O)NC2COCC2CNC(C2CCCCC2(C)C)=O)(CC)CCC(O)CC1 32966,S(=O)(=O)(c1ccc(Br)cc1NCC12CC(C1)C2)NC(c1ccccc1)(CC)C 32967,C(c1cccc(F)c1)=CCC(=O)NC1COCCC1NC(c1cccnc1)=O 32968,c1(N(CC(c2ccccc2)O)C)ncnc(N(C)Cc2nnc(C)s2)c1C 32969,Cc1cc(=NC2CCS(=O)(=O)C3(CCOCC3)C2)[nH]c(NC2CCCCCC2)n1 32970,N1(C(CNC(COC)=O)=O)CCC(O)C(C)C1.C12CCC(CC1)C(=O)N2 32971,N1(C(C(CC=C)C)=O)CC(NC(c2cccc(C(F)F)n2)=O)C2(CCOCC2)C1 32972,c1(C(N2CC(C=C)C(NC(c3[nH]c(C)nc3C)=O)C2)=O)nn(C)c2c1C(O)CCC2 32973,N1(C(c2cnc(C)n2C)=O)CCn2ncc(CNC(C3CCS(=O)CC3)=O)c2C1 32974,N1(C(C2C(C)CC(=O)N2)=O)CCC2(C1)CN(C(=O)CC1CCCC(F)(F)C1)C2 32975,c1(CNC(=NC)N(C)Cc2conc2CC)cccc2c1OCCO2 32976,c1(SCC2(C(=O)NC(C(=O)OC)CO)CN(C(C)=O)C2)ccc(N(C)C)cc1 32977,CC(CC(C)(C)C)C(=O)N1CC2(CCN(C(C3(C(=O)N(C)C)CCC3)=O)C2)C1 32978,C1(C(N2CC(N(C(CCC#C)=O)C)C3(C2)CC3)=O)CC2CCC1CC2(F)F 32979,n1(CCCC)ncc(C(=O)NCC2(Nc3nnc(C(C)(C)C)s3)CC2)c1C 32980,N1(C(CNC(CCC)=O)=O)CCC(C(C)C)CC1CNC(=O)C(F)(F)C(F)F 32981,C(=O)(C(C)(O)C(F)(F)F)N1CC(C(C)C)C(C(N2CCC(C)(C)C2C)=O)C1 32982,C(=O)(C(C)CC(F)(F)F)NCC1CN(C(c2c(C(C)C)ncs2)=O)CC1(F)F 32983,N1(C(C2N(C)CCC2)=O)CCC(CC(N)=O)(NC(=O)CCc2nccn2C)CC1 32984,CCC(CC)CCCC(=O)NC(C1CCCC1)CNC(C1CC(=O)N(OC)C1)=O 32985,N1(C(C(CC(C)C)=O)=O)CCc2nc(O)cc(C(=O)NCCc3nccs3)c2C1 32986,C(=O)(CCCS(N)(=O)=O)NCC1C(NC(c2ncc(C)cc2C)=O)CCCC1 32987,N1(C(C2(Nc3ccccc3)CC2)=O)CCOCC(NC(c2ccsc2)=O)C1 32988,c1(C(=O)NCCC(C)NC(c2c(OC)cncc2)=O)cc(Br)c(C)nc1O 32989,C(=O)(C(CC(C)(C)C)OC)NC1C(OC)CN(C(=O)CSC2CC2)C1 32990,c1(C(N2CCC(NC(C3CN4CCN3CC4)=O)C2)=O)cc(F)c(F)cc1F 32991,Cc1nc2sccn2c1C(N1CCC(C)(CNC(C2CC3CC3C2)=O)C1)=O 32992,C1(CCNC(CC(C)(C)C)=O)CN(C(C2CC2c2cccc(F)c2)=O)CCCO1 32993,N1(C(C)=O)CC2OC(=O)N(C3CCN(C(c4cc(O)n(C)n4)=O)CC3)C2C1 32994,C1(NC(=O)C2=CCCC2)C2CC3C1C3C2C(=O)NCc1cccc(F)c1O 32995,C(=O)(C(C(C)C)n1cc(Br)cn1)NCC(C)N(C(=O)CSC(C)(C)C)CC 32996,C1(Sc2ccccc2)CC1C1CCCC1.c12ccccc1CSC(C)CO2 32997,N1(C(CCC)=O)CC(OC)CC1(C)CNC(c1ccc(C)nc1O)=O 32998,C1(CNC(c2c(CC)nco2)=O)CN(C(=O)Cc2c(C)nn(C)c2Cl)CCN1C 32999,C1(O)(C(C)NC(=O)CCN(S(C)(=O)=O)C)CCN(C(=O)C2CC2)CC1 33000,C1(C(c2n(CCCC)nnn2)NC(C)(C)COC(C)C)(OC)CCCOC1 33001,C(C(C)(O)CC(=O)N1CC2(CC2)CC1CC(=O)N(CC(C)CO)C)OC 33002,N1(C(Cc2nc(C)sc2)=O)CCC(C)C(NC(=O)CCNC(=O)C(C)(C)C)C1C 33003,c1(C(=O)NC2C(NC(C3(CCC)CCC3)=O)COCC2)cnc2c(c1)OCCN2 33004,c1(C(=O)NCC2(OC)CN(C(C(CSC)O)=O)C2)cc(C)c2nc(C)nn2c1 33005,C#CC1(C)CCCN(C(=O)C(C2CC2)NC(c2cccc(CO)c2)=O)C1 33006,N1(C(C2CC(OC)C2)=O)CC(NC(c2cc(C)cc(O)n2)=O)C2(CCC2)C1 33007,N1(C(c2n(CC)ncc2)=O)CC2CC(C1)CN(C(=O)COC1CC1)C2 33008,C1(CC(=O)N(CC(C)O)CCNC(C=C(CCC)C)=O)CCCC(F)(F)C1 33009,C1(C(=O)NCC2(C)N(C(c3c(C)noc3C)=O)CC2)CCCCN(C)C1=O 33010,C1(COC)(NC(c2cnn(C)c2F)=O)CCN(C(=O)CC2CCCO2)CC1 33011,N1(Cc2n(C)ccc2)CC2CCC(C1)N2C(c1ncccc1F)=O 33012,CC(C)CCC(C(=O)N(C(C)CO)C)NC(=O)CCc1cccnc1 33013,Cc1cc(Cl)c(C(=O)NC2CC2NC(=O)Cn2cnc([N+](=O)[O-])c2)c(Cl)c1 33014,CCCC(C)CCCC(=O)N(CC(O)CNC(c1nonc1CC)=O)C 33015,C1(CC(=O)OC)CCCC2(CN(C(=O)CCc3cnn(C)c3)C2)O1 33016,c1(C(C(=O)NC)N(CCCCN2CCCCC2C)C)cc2c(Br)cccc2o1 33017,c1(C(N2CC(CNC(C(C)(C)C3CCC3)=O)C3C2C3)=O)cccc2c1CCC2=O 33018,C1(C(=O)NCCN(CCC)C(c2c[nH]c(=N)s2)=O)COCCN1CC(F)F 33019,C1(CNC(=O)Cn2cncn2)CN(C(C2CC3CC(=O)C2O3)=O)CC1(F)F 33020,c1(C(N(CCNC(=O)C(C)OCC(F)(F)F)CC)=O)cn2nc(C)cc2[nH]c1=O 33021,c1(C(C)C)ccc(C(=O)NC(C)C(C)NC(c2ccc(C3CC3)nc2)=O)cc1F 33022,Cc1cc(C(N2CCC3(CC3C(=O)NCCCC3CCCCC3)C2)=O)nc(C)n1 33023,CN1N=C(C(=O)N2CC(NCc3c[nH]c4cccc(F)c34)CC(F)C2)CCC1=O 33024,C(=O)(CCC(F)(F)F)NC(C)(C)CNC(c1ncccc1NC(N)=O)=O 33025,N1(C(C2C(OC)C2)=O)CCCN(C(c2cc(C(=O)OC)c(C)o2)=O)CC1C 33026,N1(C(=O)Cn2ccc(C(F)F)n2)CC2CN(C(C3CC3(F)F)=O)CC2C1 33027,Cn1cnc2c1CCCC2C(=O)NC1CCN(C(=O)CN2CSCC2=O)CC1F 33028,C1(NC(C(C)NC(=O)CN2CCCC2=O)=O)CN(C)NC1=O 33029,c1(C(=O)NCC(CO)NC(CS(C)(=O)=O)=O)cccc(S(=O)(=O)C(F)F)c1 33030,C1(CCNC(Cn2ncc(C)c2)=O)CN(C(C2C(C)(C)OC2(C)C)=O)CC(C)O1 33031,C(CC(C(C)C)NC(=O)CCc1ccc(Cl)nc1)N(C(c1c(CC)ccs1)=O)C 33032,c1(SC)cc(Br)ccc1C(N1CCC1CNC(=O)C#CC(=O)N(C)C)=O 33033,N1(C(C2CC(OC)CN2C(c2ccc([N+](=O)[O-])o2)=O)=O)CC2CC1CN2C(C)C 33034,C(=O)(C(C(C)C)NC=O)N(C1CCN(C(=O)C(c2ccccc2)SC)CC1)CC 33035,c1(C(=O)NCC2C(NC(C(C)OCC=C)=O)CC2)c[nH]c2c(C#N)cccc12 33036,N1(CC(=O)OCC(=O)Nc2ccc(OC)c(F)c2)C(=O)CC(C)(C)C1=O 33037,c1(C(N2CCC(NC(C3N(N=O)CCC3)=O)C2)=O)cc(C2CC2)cc(F)c1 33038,Nc1cc(Cl)ccc1C(N1CC2(C1)CN(C(c1coc(C(N)=O)c1)=O)C2)=O 33039,CCCCC(O)C(=O)NCCCC(CCC)NC(c1cc(CCC)n(C)n1)=O 33040,c1(C(C(=O)NC2C(NC(c3cn(CCC)nc3)=O)CC2)C)ccc(C#N)cc1 33041,c1(CN(C)Cc2nc(CCC)sc2)cccc(I)c1 33042,C1(OC)CN(C(c2ncn(C)c2C)=O)CC1NC(c1ccnc(OC(F)F)c1)=O 33043,Nc1c(F)ccc(F)c1C(N1CCCOC(CNC(c2ccc(Cl)cn2)=O)C1)=O 33044,c1(-c2cc(C(=O)NCC3CCC(NC(c4nnc(C)s4)=O)C3)sc2)ccc(F)cc1 33045,Cc1nc(N(C(C)CCNC(C2(C3CCCO3)CC2)=O)C)[nH]c(=N)n1 33046,C1(NC(C)=O)CCC(C(=O)NCCN2CCCC2=O)OC1 33047,c1(C(=O)NCC2N(C(CC(=O)NCC)=O)CCOC2)c(OC)ccc(Br)c1F 33048,c1(NC2CC3CN(CC4(CC)CCCC4)CC32)ncnc2cccnc12 33049,CC1(CNC(c2cc(C(F)F)no2)=O)CCN(C(C23CC(O)C2C3)=O)CC1 33050,c1(CC(=O)NC(C)CNC(=O)Cc2ccoc2)csc(CS(C)(=O)=O)n1 33051,c1(-c2nc(C(C)SCC)nn2CC)cnn2c1CC(C)CC2 33052,c1(CCC(N2CCC(C)(CNC(C(C)OCC#C)=O)C2)=O)c(O)nc(=N)[nH]c1C 33053,c1(N(C)C)ccc(C(=O)NC2(CCCNC(=O)CC(Cl)Cl)CC2)nc1 33054,C1(NC(C(N2CCNC2=O)C)=O)C2CC1N(C(C1CCSC1)=O)C2 33055,C1(NC(CCCC#CC)=O)CN(C(c2ccc(CC)[nH]2)=O)CC2(CCOCC2)C1 33056,C(c1cccc(F)c1)=C(C(=O)NC1C=CCN(C(c2c(CC)onc2C)=O)C1)F 33057,Cc1cccc(C(O)C(N2CCOC(CN(C(=O)Cc3nnc(C)s3)C)C2)=O)c1 33058,N1(C(c2cc(OC)ncc2)=O)CCC(N=c2nn[nH]n2C)C(C)C1 33059,C1(C(=O)NC2CC(F)(CNC(CCSCCCC)=O)C2)CCC(C(=O)NC)CC1 33060,C1(C(N(C)CC2OCCN(C(c3n(CC)ncn3)=O)C2)=O)CCCCC12CCC2 33061,C(CC(O)CC(=O)NCCCN(C(=O)CCCC(N)=O)Cc1ccccc1)SC 33062,c1(CC)cc(C(N(CC)Cc2ccc(-c3nn[nH]n3)cc2)=O)cc(O)n1 33063,c1(C(=O)NC(CNC(c2scc(COC)c2)=O)C(C)C)ccc(COC)nc1 33064,CCCCC(C(=O)N1CCCOC(CNC(=O)CCc2scnc2C)C1)N(C)C 33065,Cc1ccc(C(N2CCC(NC(=O)C(O)Cn3cncn3)C2)=O)cc1 33066,Cc1scc(CNC(=O)C(C2CC2)NC(=O)C(C)NC=O)c1C 33067,c1(N2CCC(CC)(CO)C2)nc(=NCC(C)(C)N2CCCC2)[nH]c2ncn(C)c12 33068,C1(n2cc(C(C(C)(C)C)O)nn2)CCCN(C(=O)COCC2CC2)C1 33069,c1(OC)cccc2c1OCCC2NS(=O)(=O)c1c(Br)cc(Br)cc1Br 33070,c1(OC)ncccc1C(=O)N(CCCC(=O)NC(c1cnc(C)s1)C)C 33071,N(C(=NC(C)C)N1CCCCC(S(C)(=O)=O)C1)Cc1cc(C)sc1.[nH]1ccnc1 33072,N1(C(c2c(OC)cc(C)cn2)=O)CC(NC(=O)C2=CCCC2C)C(N=[N+]=[N-])C1 33073,CC1CN(C(=O)CSc2nccn2C)CC1(C)CNC(c1ccc(CO)s1)=O 33074,C(=O)(C#CC1CCCOC1)NC1C2CCN(C(c3cc(C(C)=O)c(O)cc3)=O)C21 33075,c1(C(N(C)CC2CCN(C(=O)Cc3cncc(F)c3)C2)=O)cnc(N)c(N)c1 33076,Cc1ccc(C(=O)N(C)CC2CCCN2C(=O)CC2CC(CF)C2)cc1N 33077,c1(-n2cc(C3OCCN(C(=O)NCC4(O)CCOC4)C3)nn2)ccc2c(c1)CC2 33078,C#CCCC(C(=O)NC1(CC)CC(C)(C)C1)NC(C1CC2(C1)CC(C)C2)=O 33079,N1(C(=O)OC(C)(C)C)Cc2ccc(CNC(c3ccc4nn[nH]c4n3)=O)cc2C1 33080,c1(C(=O)NCC2N(C(c3c(C)con3)=O)CC(O)C2)ccc2nc[nH]c2n1 33081,N1(C(C2CCC(CC)C2)=O)CCCN(C(c2cnn(CC)c2)=O)CCC1 33082,N1(C(CCC=C)=O)CCOC(CC(=O)N(C2CC2(C)C)C)C1 33083,C12(NC(C3CCc4cnnn4C3)=O)CCCC1N(C(=O)C=Cc1cscn1)CC2 33084,N1(C(c2n(CC)cnn2)=O)CC2CCCC2(NC(=O)Cc2n[nH]c(C)n2)C1 33085,C1(CCCCNC(C(C)N(C(C)=O)C)=O)CCN(C(=O)Cc2ncoc2C)CC1 33086,C1(NC(CNS(CC)(=O)=O)=O)CN(C(C2CCS2(=O)=O)=O)CCC1C(F)(F)F 33087,C(CC(C(=O)NC1CCN(C(C)=O)C1)NC(C1CCCSC1C)=O)=CC 33088,CC1(NC(=O)CC2CCCOC2)CN(C(=O)CC2(O)CC2)C1 33089,C1(F)(CNC(c2c(C(F)(F)F)nc(C)s2)=O)CCCN(C(=O)C(C)O)C1 33090,CCC(C)C(CO)NC(=O)C(CC1CC1)NC(c1cc(C#N)cs1)=O 33091,CCC(C)CCCCC(=O)NOCC(=O)NC(C)C(C)C(=O)OC 33092,C(=O)(C(C)(C)CO)NC(C)C(C)NC(=O)CCOc1cccc(Br)c1 33093,C(=O)(CCCCc1cnc[nH]1)NC1CC(NC(CCN(C(C)=O)C)=O)C1 33094,C1(NC(CC(CC)C)=O)(CC)CCN(C(=O)CC23CCC(CC2)CC3)CC1 33095,Cc1cc(C(=O)Nc2ccccc2CN2CCC(n3cc(I)cn3)CC2)ccn1 33096,C1(N(C(c2csnn2)=O)CCSc2nc(C3CC3)cs2)CCN(CC)CC1 33097,CC1CC(NC(c2ccns2)=O)CN1C(c1cc(Cn2cccn2)on1)=O 33098,c1(C(=O)NCC(CNC(=O)CCSC(F)(F)F)OC)cc(C(C)(C)O)ccn1 33099,N1(C(c2c(C)ncs2)=O)CCOC2(C1)CN(C(C1CC(C)(C)CO1)=O)C2 33100,n1(CC)c(C)cc(C(=O)NC2(CO)CCN(C(C3CC(C(F)(F)F)C3)=O)C2)c1C 33101,N1(C(c2n(C(C)C)ncc2)=O)CCOC2(C1)CN(C(=O)C(C)CS(C)=O)C2 33102,CCC(C(=O)OC)C(=O)NCC(CC)NC(C1(c2cc[nH]n2)CCC1)=O 33103,c1(COC(C(=O)N(C2CCN(C(C3(OC)CC3)=O)C2)CCC)C)ccncc1 33104,N1(C(C2(CC)CCOC2)=O)CCCC(C)(CNC(c2csc(CC(C)C)n2)=O)C1 33105,c1(OC)ccc(CCC(=O)NCC2CN(C(c3cnco3)=O)C3CC23)c(OC)c1 33106,C(=O)(CC1OCCc2ccccc21)NCCCNC(c1csc2nnsc12)=O 33107,C1(OC)CC2CCC(C1)N2C(=O)CCCN(C)C(C1(C)CNC(=O)C1)=O 33108,c1(C(N(C2CCCN(C(C3C=CCC3)=O)C2)C)=O)cc(Br)cc2nc[nH]c12 33109,N1(C(C2CCCO2)=O)CCN(CCn2ccnc2)CC1 33110,O=C(C1=CC2(CCOC2)C1)N1CCCCC(CNc2cnc(F)cn2)C1 33111,c1(C(=O)NCC2(NC(C(C)Cc3ccco3)=O)CCCC2)cn(C)nc1C1CC1 33112,c1(OC)nccnc1C(=O)NC1CN(C(C2C=CCS2)=O)CC1C(N)=O 33113,CCC(C#N)(CC)C(=O)NCC12CC1CN(C(=O)Cn1nc(C)c(C)c1C)C2 33114,c1(C(=O)NCC(=C)CCNC(C23CCCCC2C3)=O)cc(C)cc(C)c1C 33115,N1(C(C(C)N(C(=O)CC(C)CC)CCC)=O)CC(N(C)C)C(C)(C)C1 33116,C1(NC(CC(CC2CC2)NC(c2cc(C)[nH]n2)=O)=O)CC2C(O)C(O)CC12 33117,c1(C(=O)NC(CC(C)C)CNC(=O)CC2(O)CCOC2)ccc(F)cc1C1CC1 33118,C(C)(CCC(=O)NC1CC(C(=O)NC(c2nnc(O)n2C)C)C1)OCC 33119,c1(C(N2CCC(NC(C(C)(C)CC#N)=O)(CO)C2)=O)cc(Br)cc(F)c1F 33120,N1(C(CCSC)=O)CCCC2(CCN(C(c3c(N)cc(Cl)cc3Cl)=O)C2)C1 33121,CN1N=CC(CC(N2CCOCC2CC(=O)NCCc2cccc(F)c2)=O)C1=O 33122,C1(CC(C)C)(C2(CC)CC2)CCN(C(=O)Nc2cccnc2)C1 33123,c1(C(N(CCN(C(=O)Cc2cc(Cl)cs2)C)C)=O)csc(S(N)(=O)=O)c1 33124,Cc1c(C(N2CCCC2Cn2cc(CC3(O)CCSC3)nn2)=O)sc2nccn12 33125,c1(CNC(N2CC(c3ccccc3F)C2)=O)cc(C(F)(F)F)cnc1O 33126,c1(C(N2C3CC(CNC(C(CCC)(C)C)=O)C2CC3)=O)cc2n(n1)C(C)CCC2 33127,c1(C(C(=O)NCC(C)NC(CCOc2ccc(C)cc2)=O)O)ccc(F)c(F)c1 33128,C(CC(=O)Nc1ccc(OCF)cc1)(C(F)F)NC(CCC(=O)NCC)=O 33129,C(CC(=O)NC(C1CN(C(c2nc[nH]c2C(F)(F)F)=O)C1)C)(C(F)(F)F)OC 33130,N1(C(C2C3CCC(F)C23)=O)CC2CCCC2(C(N2CCCCC2CO)=O)C1 33131,c1(CC(=O)NC)nc(CC(C(=O)CCSc2ccc(F)cc2)=O)n(C)n1 33132,N1(C(CC(C=C)(C)O)=O)CC(NC(c2cnn(C(C)C)c2Cl)=O)C(N=[N+]=[N-])C1 33133,C1(C)(C(=O)NC2CC(C)(NC(CC(C)SC)=O)C2)CC(C)=NO1 33134,N1(C(C(C)SCC)=O)CCCC12CCCN(C(C1(C)CCCCCC1)=O)C2 33135,C1(C(=O)NCC(C)(F)CNC(=O)CCOC(C)C)(OC)CCSC1 33136,Cn1cc(C(=O)NCC2CCC(NC(C3COCC3(C)C)=O)C2)ccc1=O 33137,N1(C(c2c(OCC)n[nH]c2)=O)CCN(C(=O)C=CC(C)(C)C)C(CCOC)C1 33138,c1(OCCCNC(=O)NCC2CCOC(c3ccccc3)O2)c(Cl)cccc1Cl 33139,CCCC(C(=O)NC(C)CC)NC(=O)CC1CC2CC2C1 33140,C1(NC(=O)CCc2cnccn2)CC2CN(C(c3cscc3Cl)=O)CC2C1 33141,n1(CC(C)C)ccc(S(=O)(=O)NNC(=O)c2ccc3c(c2)NCC3)n1 33142,c1(C(=O)NC(CNC(CC(C=C)C)=O)CC)c(C=CC(=O)OC)cnn1C 33143,C1(C(N2CCC(CC)C2)=O)N(C(c2scnc2Cl)=O)CCC1(C)C 33144,c1(C(N(CCN(C(C2NC(=O)OC2C)=O)CC)CC)=O)ccc(C(C)C)cc1F 33145,c1(C(=O)NC(CCCC)CNC(=O)CCCCC(C)C)coc2cc(F)ccc12 33146,c1(OC)cc(C#N)ccc1-c1ncsc1C(=O)Nc1ccc2c(c1)OCO2 33147,C1(C(=O)NC2CC(CNC(c3cn(C)c(=O)cn3)=O)C2)CCCC1S(C)(=O)=O 33148,CC1CCC(C)(NCC(N2C(=O)CCC2=O)C)CC1 33149,C(CS(=O)(=O)CC(=O)N(C1CN(C(=O)CCc2ccncn2)CC1(C)C)C)OC 33150,C1(NC(CSC)=O)CC2CC1CN(C(=O)Cc1c(C)cccc1F)C2 33151,C(=O)(C1c2c[nH]nc2CN1C(c1ccccn1)=O)NCC(CC(C)C)(C)C 33152,C(=O)(C1=C(Cl)CCOC1)NCC1C(C)CCN(C(C(n2cc(Br)cn2)C)=O)C1 33153,C1(N(C(c2c(C)nco2)=O)C)CCCC(NC(=O)C(c2cc(Br)co2)=O)C1 33154,N1(C(C(C)OCC#C)=O)CCC2(CC1)CC2CNC(=O)C(C)(C)C(N)=O 33155,N1(CC(=O)OC)CCN(C(C(=O)NCCCC2CC2)C2CC2C)CC1(C)C 33156,C12(C(N3CCC(C(=O)NCCN=c4[nH]ncs4)CC3)=O)CCCCC1OCC2 33157,N1(C(C=CC(C)C)=O)CCC(NC(C2CCS(=O)(=O)C2)=O)C12CCC2 33158,CCCC(C(=O)NOC)NC(C1CC1OC(C)=O)=O 33159,C1(NC(C2C(C)C2C)=O)CC2CCC1CC2NC(C1CCC(=O)N(C)C1)=O 33160,c1(N(CC(N2CCCC(C3(C)COC(=O)N3)C2)=O)C(C)=O)cccc(O)c1 33161,Cc1nc(NCC2CC(C)N(C(C3CCCOCC3)=O)C2)c2c(C)c(C)sc2n1 33162,C1(C)(C(N(CC#C)CC=C)=O)CC(O)CN1C(c1cnnn1CC)=O 33163,C1(CN2C(C(c3cnn(C4CCC(CO)CC4)c3)=O)CCC2)COC2(CCC2)CO1 33164,C1(C2(O)CN(C(c3oc(SC)cc3C)=O)C2)(CNC(C(C=C=C)C)=O)CC1 33165,c1(CNC(CNC(=O)OCC)=O)cc(OC)c(Cl)cn1.C12CC(C1)NC2=O 33166,N1(C(Cc2ccc(NC(C)=O)s2)=O)CC(C)CN(C(=O)COCC(F)F)CC1C 33167,c1(N2C(CCNC(c3n[nH]cc3Cl)=O)CCC2)cc(C(F)F)ncn1 33168,c1(C(N2CCN(C(=O)C=CBr)C(CC3CC3)C2)=O)cccc2nonc12 33169,C1(CNC(CSCC)=O)N(C(c2cc(C(C)(C)C)on2)=O)CCCC1(C)C 33170,C1(C(=O)NCCCCN(CCCNC(C(C)OCC)=O)C)CC(=O)N(OC)C1 33171,N1(C(C(CC)NC(C)=O)=O)CCCN(C(c2ncccc2C(=O)OC)=O)CC1C 33172,C1(CNC(C(CC)OC)=O)CC(C)N(C(C2CC(C)=NO2)=O)C1 33173,C1(CCC)CCCN1S(=O)(=O)CCC1CCOC1 33174,C1(C(N(CC(=O)Nc2cn[nH]c2)C)=O)C2CCC(C2)C1NC(=O)CCCCC1CC1 33175,N1(C(CC(C)n2cccn2)=O)CCC(N(C(=O)Cc2ccc(Cl)s2)CCO)CC1 33176,c1(C(N(CC(C)N(C(c2cc(C)no2)=O)C)C)=O)c(C)cc(F)cc1Br 33177,N1(CC(=O)NCc2ccsc2)CCC(C2CNC2)CC1 33178,N1(C(c2n(CC)ncc2)=O)CC2CCCC1C2CNC(C1(C)CCCO1)=O 33179,C1(C(=O)NC(CC)(C)C)CCC2(CC2)N1C(c1ccc(C)c(O)n1)=O 33180,Cc1ccc(NC(C2CN(C(c3sc(Cl)nc3Cl)=O)CCC2(F)F)=O)c(C#N)c1 33181,Cc1cc(CNC(C2(CNC(C3C=CCS3)=O)CCCCC2)=O)c(C)s1 33182,C1(NC(c2n(C)c(S)nc2)=O)CC(O)CN(C(=O)C=Cc2ccco2)C1 33183,C(=O)(C(O)C(C)(C)C)NCCO.C12CC(C1)N(C(N(C)C1CC1)=O)C(=O)C2 33184,C1(Nc2ccc(CCC(=O)OCC)cc2)C2C=CC(C2)C1CO 33185,Cc1ccc(C(C)C(=O)NCC2CN(C(=O)C=Cc3cn(C)cn3)CCO2)cc1 33186,n1(CCC)cc(C(=O)NCc2c[nH]nc2C2CCN(C(=O)C(F)OC)C2)cn1 33187,Cc1cnc(C(=O)NCC2CCCN(C(c3cncnc3C)=O)C2)cc1C 33188,C1(CNC(C(C)N(CC)CC)=O)(CO)CCCN(C(c2nc(C3CC3)cs2)=O)C1 33189,Cn1ccnc1S(=O)(=O)N1CCCC(C(=O)Nc2nc(F)ccc2C(N)=O)C1 33190,c1(C(N2CCC(C)(NC(C(CC#C)C)=O)CC2)=O)ccc2sncc2c1 33191,N1(C(CS(C)(=O)=O)=O)CCC2CCC12CNC(=O)CCOc1ccc(F)c(Cl)c1 33192,CCC(F)(F)CC(=O)NCCn1cc(C(=O)NCC2CC(=O)NC(C)C2)nn1 33193,N1(C(C2N(C(=O)CN3CCC(C)C3)CCC(C)C2)=O)CCCC(C2(C)CC2)C1 33194,N1(C(CCN(C)CC)=O)C2CCC1CC(CN(C(=O)CC1(CC(=O)OC)CC1)C)C2 33195,C12CC(C(O)C1)N(CC)C2=O.c1(CN2C(C(=O)NC)CCC2)cccnc1 33196,Cn1cnc2cc(CC(=O)NCC3CC(NC(C4CC4F)=O)C3)ccc12 33197,C(C(=O)N(CC(C)(C)CNC(c1nocc1C1CC1)=O)C)(C(C)C)SCC 33198,C1(C(=O)NC(C)C(=O)N2CCCC2)(COC)C=CCN1C(c1cn(CO)cn1)=O 33199,CN1N=C(C(=O)NCC(O)CNC(C2CC(OC)CN2C(N)=O)=O)CCC1=O 33200,C1(CC(=O)NC2CN(C(CN3CCN(CC)CC3)=O)CC2O)CCCC(C)(C)O1 33201,C1(C)(C(N2CC(CC)C(NC(C3(C(=O)NC)CC3)=O)C2)=O)CC2(CCC2)C1 33202,c1(C(=O)NCC(CC=C)NC(=O)C(C)(C)C(=C)Cl)cc2c(C)cc(Cl)cc2[nH]1 33203,C1(C(N2CCC(N(C(=O)C(C)(C)C3CCCCO3)C)C2)=O)C(C)(C)OC1(C)C 33204,N(C1CCc2c1ccc(F)c2F)C(CCNc1ccc(C)cc1O)=O 33205,N1(C(c2c(C)ccnn2)=O)CC(F)(F)CC1CNC(=O)C(N1C(=O)CCC1=O)C 33206,n1(CC)cnnc1C(=O)NC(C1CCCC1)CNC(=O)C(C)NS(=O)(=O)CCC 33207,c1(CC)nc(C)c(CC(=O)NC2(C)CCCN(C(=O)C#CC3CCC3)C2)c(C)n1 33208,c1(C(=O)NC(CNC(c2cc(C)ncc2)=O)(C)C)cc(N2CCCC2)nc(Cl)c1 33209,CCS(=O)(=O)CC(=O)NC1(CNC(C2CC2(C)C)=O)CC1 33210,N1(C(C=C(CCN(C)C)Cl)=O)CCOC2(C1)CN(C(C1CCCN1N=O)=O)C2 33211,c1(C(=O)NCC(=C2CN(C(C3CC3(F)F)=O)C2)F)n[nH]c(C2CC2)n1 33212,C1(NC(c2ccnc(Cl)c2F)=O)CCCN(C(C2CC3(CC3)C2)=O)CC1 33213,N1(C(CC(C(F)(F)F)c2n(C)ccn2)=O)Cc2ccnc(Cl)c2C1 33214,C(=O)(C1CSc2ccccc21)NCC1CCN(c2ccc(C(C)=O)cn2)CC1 33215,Cc1ccc2[nH]cc(CC(N3CC(NC(C4(C(N)=O)CC4)=O)CC(O)C3)=O)c2c1 33216,c12ccc(cn1)C(c1nnnn1C)N2.C1(COC)CCCC1Oc1ccccc1 33217,C1(C(=O)NCC2(C(N)=O)CN(C(c3ccc(F)c(Cl)c3)=O)C2)CC2C(C1)C2(C)C 33218,C12(CCCCC1)C(=O)NC2.n1(C)cc(CC(=O)NCC2C(CC)C2)nn1.OC 33219,C1(NC(C=CC(CC)=CC)=O)CCCN(C(=O)CCc2ccncc2)CC1F 33220,c1(CC)cnc(O)c(C(=O)N(C)CC2CCCN2C(c2n[nH]cc2OC)=O)c1 33221,c1(C(N2C3CC(NC(C4CCCN(C)C4)=O)C3CC2)=O)cc(Cl)cc2c1OCC2 33222,CC(C)CC(CNC(c1cocc1C(N)=O)=O)C(=O)NC(C)CC1CCC1 33223,c1(OCCC)cccc(C(=O)NC2CN(C(=O)C(C)=C3CCC3)CC2C)c1 33224,CCCC(CCCNC(=O)CC1CCCCCO1)NC(=O)CNC(=O)C(C)(C)C 33225,N1(C(c2scc(CNC(c3c(C)ocn3)=O)c2)=O)C2CCC1COC2 33226,Cc1cc(C(=O)NC(C)CN(C(=O)CC(=O)Nc2nccs2)C)c(C)nc1C 33227,c1(C(=O)NCC2CC(NC(CC3CCCC(C)(C)O3)=O)C2)cccc2nncn12 33228,C1(F)(C(=O)NCCN(CCOC)C)CCN(C(c2cnc(S)[nH]2)=O)C1 33229,N1(C(C2C3(CN(C(c4c(C)nn(C)c4C)=O)C3)C2)=O)C2CCC1CN(C)C2 33230,c1(CC)cccc(C(=O)NCC(O)CN(C)C(c2ccns2)=O)c1N 33231,CC1(C)Cn2[nH]c(=NC(=O)NCC3CC(F)(F)C(=O)N3)cc2CO1 33232,CN1CCC(NC(=O)CN(C(C2CCC(N(C)C)C2)=O)CC2CC2)C(C)(C)C1 33233,c1(C(c2n(C)nnn2)NCC(C)(C)OCCO)cc(Br)c(Br)o1 33234,C(=O)(CC(C)(C)C)N(C(C)C(N1CCC(Nc2cc(Cl)ncn2)CC1)=O)N(C)C 33235,N1(CC)CCOCC1CC(=O)N(CCC(C)NC(=O)CN1CCN(C)CC1)C 33236,C(CCN=C(NCc1cccnc1Cl)NC1CSC(C(F)(F)F)C1)SC 33237,c1(CC)cccc(C(=O)OC)c1NC(=O)C(N1CCOCC1C1CCCOC1)=O 33238,c1(C(N(C(CC)CNC(=O)C(F)OC(F)(F)F)C)=O)cccc2nsnc12 33239,C(CCC(=O)NCCCN(C(=O)C(C)CN(C)C(=O)OC(C)(C)C)C)=CCC=C 33240,C1(C(=O)NCC2(C(C)NC(c3cnsc3)=O)CC2)CCc2nnc(O)n2C1 33241,c1(C(=O)NCC(CC)(CC)NC(c2nnsc2C)=O)cc2ccccc2c(O)n1 33242,N1(C(C2(C)CCOCC2)=O)CCC2(CC1)CC2C(=O)NC1CC2(CCCO2)C1 33243,C1(CNC(c2c(C)nco2)=O)CN(C(=O)CC2CCC3(CCC3)O2)CCN1C 33244,N1(C(c2cc(C)cc(Cl)n2)=O)CC(C)CN(C(=O)C(C(C)C)NC(C)C)CC1C 33245,C(=O)(C(C)(O)CC)N(C1CCCCO1)C(C)(C)C.C1CCC(=O)N2CC(C2)S1 33246,C1(NC(C2C(CCC)C2)=O)CN(C(c2ccc(-n3cnnn3)cc2)=O)C(C)(C)C1 33247,C(CCS(C)=O)(C(=O)NC1CCCC1CNC(C12CC3CC1C2C3)=O)N(C)C 33248,c1(CC)onc(C(=O)NCC2(C)CCN(C(c3ncc[nH]c3=O)=O)C2)c1C 33249,C1(CNC(c2ccc(SC)o2)=O)C2CC1N(C(=O)CN1CCN(C3CC3)C1=O)C2 33250,C(=O)(C1CCCc2ccnn21)N1C(C)CC(NC(C2(OC)CCS(=O)(=O)C2)=O)C1 33251,Cc1nccnc1NC(c1nnnn1C1CC(F)(F)C1)CCC1CCCC1 33252,c1(C(=O)NC2CCC(CCNC(CC(C=C)C)=O)C2)c(C)nc2sccn12 33253,c1(C(=O)NC2C(C)CN2C(=O)C=Cc2ccco2)ccnc(OCCO)c1 33254,C(CC1=CCOCC1)NC1(c2nnnn2CSc2ccccc2)CC(CCF)C1 33255,N1(C(CSCC=C)=O)CCC(NC(c2cc(C3CC3)[nH]c2C)=O)CC1C 33256,C1(c2onc(-c3c(C)cccc3)n2)CN(SC2CCCCN(C)C2=O)C2(CCC2)C1 33257,N1(C(C(CC=C)(C)O)=O)CC=C(C(=O)NC(c2nc[nH]n2)C2CC2)CC1 33258,CC(=Cn1ccnn1)C(=O)NCC12CCC(CN(C(c3cccnc3O)=O)C1)C2 33259,N1(C(Cc2cc(C)on2)=O)CC2(CCN(C(=O)CCC3CCCC(O)C3)CC2)C1 33260,c1(OC)cncnc1C(=O)NCCC(=O)N(C1CCCCC1C)C1CC1 33261,C1(C(=O)NC2N(CC)CCC2)CCN(CC(=O)N(C)C2CC2)CC1 33262,c1(C(=O)NCC(CNC(C2N(C(C)=O)CCC2)=O)O)cc2c(O)ccc(F)c2[nH]1 33263,c1(C(C)NC(c2cc(NC(N)=O)on2)=O)cc2cccc(F)c2o1 33264,C(=O)(C(C)OCC(F)(F)F)NCC(C1CCCC1)NC(COCC(C)C)=O 33265,CCN=c1[nH]cc(C(=O)NC2COCC2NC(c2nc(C)oc2C)=O)s1 33266,c1(CN2CC3N(C(C4CN(C)C4)=O)C(C3)C2)c[nH]c2ncc(Br)cc12 33267,N1(C(C2CCN(CC#C)CC2)=O)C2CCC1CN(C(C1CC3CCC1O3)=O)CC2 33268,C1(NC(C(F)OC)=O)CCSC12CN(C(=O)Cc1cnnn1C)C2 33269,CC1(C(=O)NCC2CCCCN2C(c2ccn(C3CCC3)n2)=O)CC2CCC1C2 33270,CCC(CC(F)(F)F)C(=O)NC(CCN(C(=O)CC(C)(C)O)C)C(C)C 33271,N1(c2n(CC=C)c(C(O)CCOC)nn2)CCC(C)CC(C)C1 33272,C1(NC(c2c(C)con2)=O)CN(C(=O)Cc2ccns2)CCC12CCC2 33273,Cc1cc(C(N2CCN(C(c3ccccc3OC(F)F)=O)CC2)=O)nc(C(F)F)n1 33274,Cc1nc2sn(CC3CC(OC(F)F)C3)c(=O)c2c(C)c1C 33275,C1(NC(c2cnc(C)o2)=O)CCOC12CCN(C(c1cc(Br)c[nH]1)=O)CC2 33276,N1(C(c2nc(CCC)sc2)=O)CC2ON=C(CNC(c3nc(C)oc3C)=O)C2C1 33277,CC(C)CC(CNC(C1(F)CC1)=O)NC(C1(CC2CC2)CC1)=O 33278,CCCC(C)(O)CC(=O)N1C2CCC1C(CNC(=O)CN(C)CC)C2 33279,N1(C(=O)CCc2nccs2)CCCCC1C(N1CCOC2CC12)=O 33280,c1(CC(=O)NC(C(C)NC(c2cc(C)c(C)nn2)=O)C)ccc2ncsc2c1 33281,c1(C(C(=O)N(C)CC2N(C(CN(C)CC)=O)CCC2)O)cccc(C)c1 33282,N1(CC(N2CCC(NC(=O)Cc3nc[nH]n3)(CO)C2)=O)CCS(=O)(=O)CC1 33283,N1(C(CC(=O)NC2CC2)=O)CCC(C(=O)NCc2cccc(F)c2)C12CCC2 33284,N1(C(CC(CC)OC)=O)CCCCC2(CCN(C(=O)OC(C)(C)C)C2)C1 33285,c1(NC(CN2CCCC(CNC(C(C)C)=O)C2)=O)ccc(F)c(Br)c1 33286,c1(C(CC)(C)NC(=O)NC2(Cn3cnnc3)CC2)ccc(F)cc1 33287,Cc1cc(CN2CC(F)(F)CC2C(=O)Nc2nc(Cl)nc(Cl)n2)cnc1Cl 33288,C=CC(CCC)CC(=O)NC12CCC1CN(C(=O)C(O)CC(F)(F)F)C2 33289,N1(C(CC2(C(=C)F)CCC2)=O)CCC2(CNC(=O)CCC3CCC3)CCCCC12 33290,N1(C(CSC)C(=O)OC)CC(CCO)OCC12CC2 33291,C(C)(C)(CCCNC(=O)C(C)(C)C1CCCN1C(C1CCCO1)=O)OC 33292,CCCCCC(O)CC(=O)NCC(C(C)(C)C)NC(=O)C(F)C1CCC1 33293,C1(OC)CC(CC(=O)NCCC2CN(C(=O)CC(C)C)CCO2)C1(C)C 33294,N1(C(c2scc(C)c2Cl)=O)CCC2(CC1)OCCC2NC(C12CC(F)C1C2)=O 33295,C(=O)(CCC1=NNC(=O)CC1)NCCC(=O)NC1(C)CC(NC(=O)CO)C1 33296,S(=O)(=O)(c1cc(F)cc(Br)c1)N(C(=O)C(C)Oc1ccc(F)cc1)C(C)C 33297,N1(C(CCCn2c(C)ncc2)=O)CCCN(C(=O)CCN(C)CCO)CC1CO 33298,c1(N2CCCC3(NC(c4ncc(F)cc4F)=O)C(C2)C3)ncc2cccnc2n1 33299,C(C)(C)(CCCCNC(C1(n2nccn2)CC1)=O)NC(C(CSC)OC)=O 33300,c1(C(N2CC=CC(NC(c3c(C)ccc(C)c3)=O)C2)=O)nn(C)c2c1CCCC2 33301,c1(C(=O)NCC2C(NC(c3c(CC)occ3)=O)CC2)cncnc1C1CC1 33302,c1(C(=O)NCCC(CNC(c2n(C)nc(C3CC3)c2)=O)O)ccc(F)cc1O 33303,C1(C#N)(OC)CC(C(=O)NC(CNC(c2c(Cl)n[nH]c2C2CC2)=O)C(C)C)C1 33304,N1(C(CCC=C)=O)CCc2ccccc2C1CCNC(c1cnc(Cl)s1)=O 33305,N1(C(C(COC)C)=O)CC(NC(c2cc(=O)n(C)o2)=O)CC12CCCCC2 33306,C1(C2CC2)(CNC(CCCNC(C)=O)=O)CCN(C(=O)C2=C(C)OCC2)C1 33307,C=CCN=C(NCCCCC1CCCCC1)N1CCCC(CC)C1 33308,c1(CSC)cccnc1C(=O)NCC(C)NC(=O)Cc1cnc(C)[nH]1 33309,CCC(O)C(C)C(=O)NC1CCC(CNC(c2cccc(C#N)c2)=O)CC1 33310,N1(C(C2CC(OC(F)F)CN2)=O)CCCN(c2cccnn2)CC1 33311,C(=O)(CS(=O)(=O)C1CC1)NC(C(C)C)CCN(C(=O)Cc1ccn(C(F)F)n1)C 33312,Cc1cncc(NC(c2cnc(CNC(=O)CC3CSCCO3)nc2)=O)c1 33313,C1(C(N2CC(Cn3cc(-c4cccc(CN)c4)nn3)C2)=O)CC1C1CCCCC1 33314,CN1CC(C(=O)NCC(C)(C)NC(=O)C=CC(F)F)CCC1=O 33315,N1(C(C(C(C)C)NC=O)=O)CCC2(CCN(C(c3ccc(O)c(N)n3)=O)C2)C1 33316,c1(CNc2c(OC)cc(N3CCCCC3)cc2)nc2ncc(Br)cn2n1 33317,C1(NC(C=CCCC)=O)CCCC2CN(C(=O)CCc3cnn[nH]3)CC12 33318,C1(CNC(C2N(CC)CC2)=O)CCC2(CCC2)CN1C(=O)C(Cl)=CCl 33319,c1(CC)nnsc1C(=O)NCC(F)CNC(c1cn(CCF)nn1)=O 33320,c1(C(CN(C(=O)CCCOC(F)(F)F)C)O)cccc(C#N)c1 33321,C1(CCNC(c2cscn2)=O)CCN(C(c2cc(O)ncc2F)=O)CCC1(F)F 33322,c1(C(=O)NCC2(C)CC2(Cl)Cl)ccnc(-n2cccn2)c1 33323,Cc1cc(Cl)nc(N)c1C(=O)NCC1CC(C)CCN1C(C1CCC(C)(C)C1)=O 33324,C(=O)(CCCCCN(C)C(C1CC12CCCCC2)=O)NCC1CN(CC)C(=O)O1 33325,Cc1ccc(CNC(C2C3CN(C(=O)CCc4ccoc4)CC23)=O)c(O)n1 33326,c1(C(=O)NCCCC(C)NC(=O)C2CC2)cccc(OCc2ccccc2F)c1 33327,CCCC(C#N)NC(C12CC(n3cc(C4CCC4)nn3)C1C2)=O 33328,C1(C(N(CCCNC(c2ccnn2C(C)C)=O)CC)=O)CCCC(CF)C1 33329,C(c1ccoc1)=CC(N1CCC(NC(=O)C(Cl)(Cl)Cl)C1)=O 33330,C1(OC)CC(C(=O)NC2CCC(C(F)(F)F)CC2)(NC(=O)OC(C)(C)C)C1(C)C 33331,N1(C(Cc2cc(C)ns2)=O)CCCN(C(=O)CCC(CF)CF)C(C)C1 33332,c1(NC2C(C(=C)C)OCC2)nccc(=NCCN2CC(OC)CC2=O)[nH]1 33333,N1(C(CN(CCCCCC)C)=O)CC(NC(=O)C=CC2CCC2)C2(CCC2)C1 33334,c1(NCC2(NC(CCOCC#C)=O)CCC2)nccc(Oc2ccccc2F)n1 33335,c1(C(=O)NCC2N(C(C=CCCCCC)=O)CC(OC)C2)cnc2sccc2c1 33336,C(C(CC(F)(F)F)NC(c1cccc(O)c1Cl)=O)NC(C(CC)N(CC)CC)=O 33337,N1(NC(CCC2CCN(C(c3c(C)con3)=O)C2)=O)CC(=O)NCC1C(N)=O 33338,C#Cc1cc(C(=O)NCC2CC3(C2)CN(C(=O)CC(C)CC)C3)cc(N)c1 33339,C1(C(N2CCC(C)(NC(c3cc(C)c(C)o3)=O)C2)=O)CCCC2(CCC2)O1 33340,N1(C(c2ncccc2C)C(=O)NC)CC2CC3CC2C1C3O 33341,C1(CNC(c2cnnn2C2CC2)=O)CN(C(C2C3(CC3)C23CC3)=O)CC12CC2 33342,CC1CC(C(=O)N2CC(O)(C3CCCN3C(=O)C#CC3CCC3)C2)=NO1 33343,CC1CN(C(=O)C(c2ccc(Cl)cc2)O)CC1NC(=O)C(C)C1CCOC1 33344,C1(CNC(CC=CC)=O)C=CCN1C(=O)CCc1ccc(C)s1 33345,c1(OCC)ccccc1C(=O)NCC1CC1OC1CC=CC1.C12CC(C1)NC2=O 33346,c1(CCCCC)ccc(C(=O)NCC(CCOC)NC(=O)C(C)=CC(C)(C)C)o1 33347,C1(NC(c2c(CC)noc2C)=O)CC2CC(NC(=O)C(C3CCOCC3)F)C2C1 33348,Cc1cccc(C(=O)NCC2CC(C(=O)N3CC(CO)C(O)C3)=NO2)c1C 33349,Cc1ccc(CNC(C2C(O)CCN2C(C2CCC(C)(C)OC2)=O)=O)c(O)n1 33350,N1(C(C(C#N)C2CC2)=O)CCOC2CN(C(c3c(F)cccc3F)=O)CC12 33351,N#CCS(=O)c1ccc(C(=O)NC(C)(CNC(c2cnsn2)=O)C2CCC2)cc1 33352,c1(OC)cc(F)c(C(N2CCCCC(CNC(C3SCCS3)=O)C2)=O)c(F)c1F 33353,C(=O)(CC(C(F)F)NC(c1conc1C)=O)N1CC(F)(CC)C1 33354,N1(C(c2cncc(OC)n2)=O)CC(C(=O)NCC(O)C(C)(C)C)CC(C)C1 33355,N1(C(C(C)=C2CC2)=O)CC(N(C(=O)Cc2c[nH]nc2C)C)C(C)(C)C1 33356,N1(C(c2cc(C)[nH]c2C)=O)C2CCC1CN(C(c1cccc(C3CC3)n1)=O)C2 33357,CC1=C(C)CC(C(=O)NCC2COCCN2C(c2csc(C)c2C2CC2)=O)CC1 33358,N1(C(C(C2CCOC2)NC(c2nc(CCC)oc2)=O)=O)CCC12CCCC2 33359,c1(C(=O)NC2CC(NC(c3coc(Br)n3)=O)C2)ccc(-n2ccnc2)cc1 33360,c1(COCC)nc(C(=O)N(C(CNC(c2ccc(Cl)o2)=O)C2CC2)C)cs1 33361,c1(CN(CC(C)CS(C)(=O)=O)C)c[nH]c2cccc(Br)c12 33362,Cc1ncnc(C(N2CCC(CO)(NC(=O)C(F)C3CCOC3)CC2)=O)c1C 33363,C(C(O)CCNC(=O)CCNS(C)(=O)=O)NC(CCSCC(C)C)=O 33364,C1(C(=O)NCCn2c(C)cnn2)CCC(C)(C)N(C(=O)COCCCN(C)C)C1 33365,C1(O)(CCNC(C=CC(C)(C)SC)=O)CCN(C(=O)CC2C=CCCC2)C1 33366,c1(C(N2C3C(NC(c4c(Cl)ccc(SC)c4)=O)C(C3)C2)=O)c(N)ccc(F)c1C 33367,C1(C(=O)NC(CC)(CNC(c2csc(CO)n2)=O)CC)CCC2CC2CC1 33368,C12(C(=O)OC)CN(C(C3CCCOC3)C(=O)NC3CCCC3)CC1S(=O)(=O)C2 33369,C1(NC(c2c(OC)noc2C)=O)CC2CC1CN(C(c1ccccn1)=O)C2 33370,C1(NC(COCCC=C)=O)CC2CC(C1)N(C(C1CC(C(C)=O)C1(C)C)=O)C2 33371,C(=O)(C1=CCOCC1)NC(CNC(C1CC(=C2CC2)C1)=O)C1CCC1 33372,C1(CN(C(C2CC(N(C)C)C2)=O)CC)CCCN(C(c2cscc2C)=O)C1 33373,C1(C(=O)NCC2(CNc3ncc(C)cn3)CCCC2)(OCC)CCOCC1 33374,C(=O)(CCCC(C)(C)NC(=O)CCCCOC)NCCC(CC)(F)F 33375,Cc1ccc(C=CC(N2CC(C3(NC(=O)COc4ccccn4)CC3)C2)=O)cn1 33376,N1(C(c2cnn(C)c2)C)CCC2(CC1)CC(CNS(=O)(=O)c1ccncc1)C2 33377,Cc1cn2cc(C(=O)NCC3CC(F)(F)CN3C(=O)C(C)N(C)C)cc(F)c2n1 33378,c1(C(=O)NCC(C)NC(c2c(OC)ncc(Br)c2)=O)cnc2ccnn2c1 33379,C(=O)(CC(O)CC(C)(C)C)N1CC2C(NC(c3nc(OC)c(C)s3)=O)(C2)C1 33380,C12(CCCOC1)C(=O)N2.C(=O)(CC(C)COC)OC.c12cn(nn1)CC(C)NC2 33381,C1(CC=C)(NC(C2CC(N(C)C)C2)=O)CN(C(c2cc(C3CC3)on2)=O)C1 33382,C1(CC#C)(C(=O)OCCSCC(C)O)CCCC1 33383,Cc1cc(C(=O)NC(C)(C)CCNC(=O)Cc2ccsc2Br)ncc1F 33384,C1(C(=O)NC2CC(C)(NC(c3ccn(CCC)n3)=O)C2)NC(=O)CC1C(F)(F)F 33385,CCC(C)C(C(=O)NC(CCO)CC(C)C)NC(=O)Cc1c(C)cnn1C 33386,N1(C(C(CC)NC(C)=O)=O)CCN(C(=O)CC2CC2)C(C2CCCC2)C1 33387,C(N=c1cc(C(F)(F)F)nc[nH]1)C1C(C)CN(C(=O)COCC2CCCC2)C1 33388,c1(C(C)C)ncc(C(c2nnnn2CC(F)F)NCC2CCCCC2)[nH]1 33389,N1(C(C(OC)OC)=O)CCCC(O)(CCNC(C23CC2COC3(C)C)=O)C1 33390,c1(C(=O)NCCCN(C(=O)CCCl)CC)cc(Br)c(OC)s1 33391,N1(C(C)=O)CCC(NC(=O)COc2cccc(F)n2)C(c2ccc(F)cc2)C1 33392,c1(C(N2CC(Cn3cc(C(C)O)nn3)OCC2)=O)nccc2cc(Br)ccc12 33393,CC1=C(C(=O)NC(C2CCN(C(C3(C)SCCCS3)=O)CC2)C)C(C)(C)CCC1 33394,c1(CC(Cn2cc(CO)nn2)NC(=O)Cc2ccccn2)ccc(Cl)cc1 33395,C(=O)(CC(C)C(F)F)NC(C)C(C)(C)NC(c1cnc(C(C)(C)C)s1)=O 33396,Cc1ccc2c(C(=O)NCC(C)CNC(=O)C(C(C)C)C3CCC3)n[nH]c2c1 33397,c1(CNC(Cc2cc(C)no2)CNC(=O)OC(C)(C)C)ccc(I)c(O)c1 33398,CN1CCN(C(=O)C(F)C2CCCC2)CC1C(=O)NCC1CC12CC2(F)F 33399,C(C1CCCc2cccnc21)c1n(-c2c(OC)cccc2)nc(-c2cc[nH]n2)n1 33400,c1(OCCC(=O)N(C(Cn2c(C)ncc2)C)CC(C)C)cc(F)ccc1F 33401,c1(CC(c2c(C)nnn2C)=O)cc(F)cc(Cl)c1 33402,N1(C(C(C)(N(C(C(N2CCOCC2)C)=O)C)C2CC2)=O)CCn2ccnc2C1 33403,c1(CCC)nc(C(N)=O)co1.C12(CCC1)C(=O)N2.C12CCC1C2.C1=CCNC1=O 33404,n1(CC(=O)NCC2COCC2NC(=O)C(O)CC(F)F)cc([N+](=O)[O-])ccc1=O 33405,C1(C(=O)NC(C)CC(C)NC(c2sccc2F)=O)(Cc2cnn[nH]2)CCOCC1 33406,C12(C(=O)Nc3c(CCC)cccc3)CC(CO)(CN1C(=O)CSc1nc[nH]n1)C2 33407,c1(C(CC(=O)O)NCc2cccc(C3CC3)c2)cccc(F)c1Br 33408,C1(COC)(NC(=O)C(C2CC2)SC)CCCN(C(C2(O)COC2)=O)C1 33409,CC(C)C#CC(=O)NC12CC1CN(C(C1CCCN1C1CCOCC1)=O)C2 33410,c1(C(=O)NC(C)CN(C(=O)Cn2cnnn2)C)ccccc1-c1ncc[nH]1 33411,N1(C(C(C)=C(CC)C)=O)CCCC2C1CCN2C(=O)C(C(C)(C)C)NC(N)=O 33412,N#Cc1cnc(C(F)(F)F)cc1NC1CCC(OCCO)CC1 33413,C#CCCCC(C)C(=O)NC1CC(C)N(C(c2ccc3nccn3c2)=O)C1 33414,C1(C(N(C2CCC(CNC(C=CC=CCC)=O)CC2)C)=O)CCOCC1(C)C 33415,CCC(CNC(=O)C(C)OCC1CC1)NC(=O)CC1(C#N)CC1 33416,c1(C(=O)OCC)cc(CNC(C23CCC(C(F)F)(CC2)CC3)=O)ccc1[N+](=O)[O-] 33417,c1(CN(C(=O)CCC2(NC(c3cc(Cl)no3)=O)CCCC2)C)cccnc1 33418,c1(C(=O)NCC(CC)NC(=O)C(C)OCCC(C)C)ccnn1CCOC 33419,c1(CNC(=O)Cc2cnc[nH]2)cc(F)c(CO)c(F)c1.C12COCCN1C2=O 33420,N1(C(c2cccn(C)c2=O)=O)CC2CN(C(c3cnns3)=O)CC(F)(F)C2C1 33421,CC1CCCCN1CC(=O)N(C(=O)COc1ccc(C(N)=O)cc1)C1CC1 33422,c1(OC)ccnc(C(=O)NC2COCC2CNC(=O)C(C)OCC2CC2)c1 33423,c1(CC)nn(C)c(NC(=O)CC2CCCC(NC(c3cccnc3O)=O)C2)c1Cl 33424,c1(OC)cc(Cl)c(Cl)cc1C(=O)NCCC(C)NC(C1C(C)C1C)=O 33425,C1(NC(COC(CC)(C)C)=O)CCC2(CC2)N1C(=O)CN(C(=O)COC)C 33426,C1(C)(N(C)C)CCN(C(C2CC(=O)CN2C(C2(N(C)C)CCC2)=O)=O)C1 33427,C1(C(N2C(CNC(=O)C#CC(C)C)CC(OC)C2)=O)Cc2ccc(C)cc2S1 33428,c1(CC(=O)NCc2c(C(=O)NC(CC)CN3CCCC3)cco2)c[nH]nc1C 33429,C=C(Cl)C(C)(C)C(=O)NCC(O)CCNC(C1CC1CCC)=O 33430,C1(CNC(CCSCCC)=O)CC2(CO1)CN(C(=O)CCC=C(C)C)C2 33431,c1(C(C)(C)C)c[nH]cc1C(=O)NC(C)(C)CNC(=O)CCN1CCOC1=O 33432,CC1SCCCC1C(=O)NCCN(CCCN(C)C)C(=O)CC1(C)CC1 33433,C(=O)(C(C)(C)NC(C)=O)N1CC(C(C(=O)NCCCN(C)C)OC)C1 33434,CC1=NS(=O)(=O)NC=C1C(=O)N1CC(CCNC(C2CCCC3CCCN23)=O)C1 33435,c1(C(=O)NCC2C(NC(C(c3cn(C)nc3)O)=O)CCC2)ccnc(S)c1 33436,C12(C(=O)NCC(CCNC(C=C(CCC)CCC)=O)O)CC1CCC2(F)F 33437,Nc1ccc(F)cc1C(N1CC2CC2(CNC(=O)CCC2CCCCCC2)C1)=O 33438,C1(NC(c2cccnn2)=O)CC1C1CCCN(C(c2cc(F)c(F)c(F)c2)=O)C1 33439,C1(NC(=O)CCc2cc(F)ccc2Br)CN(C(C2(F)CC2)=O)CC(F)(F)C1 33440,N1(C(C(C(C)C)n2cnnc2)=O)CCN(C(=O)C(N)=O)CC(O)C1 33441,CC1CN(C(=O)CCc2cn[nH]c2)CCC1NC(=O)CCc1cnn(C)c1 33442,c1(C(N2CC(C(=O)Nc3cc(Cl)ncc3Cl)C2)=O)ccc2c(c1)CCO2 33443,c1(C(N2CC(NC(c3cc(F)cnc3O)=O)C(F)C2)=O)c(F)ccc(F)c1Cl 33444,c1(C(N(C(C)CCNC(=O)C=CC2C(C)C2(Cl)Cl)C)=O)n[nH]c2c1CCCC2 33445,c1(CC)nnc(C)cc1C(=O)NCC1CN(C(c2cnc3n2CCC3)=O)CCO1 33446,C(=O)(C1COc2ccc(Cl)cc21)NC1C(NC(c2c(CC)occ2)=O)CCC1 33447,N1(C(C2CCC(CNC(C3CC4CCC3O4)=O)CC2)=O)CCC(O)C(F)C1 33448,C1(CCC2CCCN2C(c2ccccc2)=O)(NC(C(C=C)O)=O)CCCCC1 33449,N1(C(c2c(OC)cccc2F)=O)CCc2ccccc2C(NC(=O)C(C)(F)F)C1 33450,c1(C(=O)NC(c2ccc(Cl)cc2)CNC(C(C)O)=O)cnc(O)cc1C(F)(F)F 33451,C(=O)(C1c2c[nH]nc2CN1C(=O)CC1CCOC1=O)NCc1c(C)cc(C)nc1 33452,C1(CC(=O)N(CCCCCNC(c2c(C)cncc2)=O)C)CC2CCC1CC2 33453,c1(N(C)Cc2c(C)ccc(Cl)c2)nc2c(c(=NCCC3CC3)[nH]1)SCC2 33454,CCC(C)C(O)C(C)C(=O)NCC12CC(CO1)N(C(C1(C)CCC(=O)C1)=O)C2 33455,N1(C(Cc2ccn(C)n2)=O)CCCC(C)(C)C1CNC(=O)Cc1ccsn1 33456,CC(C)(C)CCC(=O)NCCCC1CCCCN1C(C1CCC2(CCC2)C1)=O 33457,c1(CNC(c2ncc(-c3ccco3)cn2)=O)c(Cl)cccc1[N+](=O)[O-] 33458,Cn1ccnc1C(=O)NC1(C2CCCN2C(=O)CCSCc2nccn2C)CC1 33459,C1(CNC(CCc2ncc(C)[nH]2)=O)CC(NC(c2sc(C)cc2Cl)=O)C1(C)C 33460,n1(C(C(=O)OC)C)cc(C2(NCCCC(=O)N(C)C)CC2)nn1 33461,C1(C(=O)NCC(CNC(c2cn(C(C)C)nn2)=O)C)CCCC(=O)O1 33462,C1(NC(C(C(C)C)SCC)=O)CC2(CCN(C(=O)C=CCOC)C2)C1 33463,Cc1nc(C(=O)NC2CC(NC(=O)CC3CCC(=O)NC3=O)C2)c(C)n1C 33464,C1(NC(C(C(C)NC(CC2(OC)CCC2)=O)C)=O)C2CCCC1COC2 33465,C(=O)(C(O)CCS(C)=O)N(C(C)C)CCNC(c1sccc1OC(F)F)=O 33466,C1(CC)C(NC(=O)C(c2cn(C)nc2C)C)CCN1C(=O)C=CC1CCC1 33467,Cc1nn(CC(=O)NC2CC2NC(C2(C)CC(C)(C)C2)=O)c(C)c1Cl 33468,c1(C(=O)NC2(CNC(CP(C)(C)=O)=O)CC2)cc2cc(Cl)cnc2[nH]1 33469,c1(CC(=O)NCC(C)(O)CNC(=O)CCc2cnc[nH]2)c(F)cccc1F 33470,C1(C(N2CC3C(NC(C4CC5COCC5C4)=O)(C3)C2)=O)CC2(C1)CC(F)(F)C2 33471,c1(COCC(C)=CCOC(C2C(Br)(C(=O)OCC)C2)=O)cccnc1 33472,C1(NC(c2n(C)ccc2)=O)CCCC2CN(C(=O)C#CC3(C(F)(F)F)CC3)CC12 33473,N1(C(c2cn(CC(C)C)nn2)C)CC(=O)N(Cc2ncnn2C)C1=O 33474,C(=O)(CCCC(=O)NCCC1(NC(=O)C(C)NC(N)=O)CCCC1)NCC 33475,C1(NC(c2ccon2)C)CC(NC(=O)CNC(=O)Nc2ccco2)C12CCC2 33476,c1(CCC)nc(C(=O)N(CCCCN(C)C(C2(C)CCC2)=O)C)cs1 33477,c1(C(=O)NCC2N(C(CC(=O)OC(C)(C)C)=O)CCOC2)cc2ncccc2s1 33478,c1(OC)cccc(OC)c1NC(=O)NCCOc1ccc(C)cc1Br 33479,C1(C(N(C2CC(C#N)C2)CC(=O)NCC(C#C)OC)=O)CCOC1(C)C 33480,c1(C(C)C(=O)NCc2cc(C(F)F)no2)ccc(C(F)F)cc1 33481,C1(C(=O)NCc2c(OC)n(C)nc2)C2CC(O)C(C2)N1C(=O)CC1(C)CCOC1 33482,C(=O)(CCCN=[N+]=[N-])N1C2(C(=O)NC3CN(CCC)C3)CC2CC1 33483,C1(C(N2C3(CN(C(C4CCOCC4)=O)C3)CC2)=O)CC2CC(O)C(C1)C2 33484,C(CCCCCN(C)C(C1CCC(CO)CC1)=O)NC(CCNC(=O)NC)=O 33485,CCCCC(CC)C(=O)N1CCC(=CCNC(C2CC3CC3C2)=O)CC1 33486,N1(C(CC(CC#C)NC(=O)CC2CCCCC2O)=O)CC(=O)NC2(CC2)C1 33487,N1(C(CCc2cccc(C)c2)=O)CCN(C(=O)CCc2ccncc2)C2CCC12 33488,c1(C(=O)NC2CN(C(C(CO)NC(C(C)C)=O)=O)C2)ccc2c(c1)CCN2C 33489,C1(O)(CC(=O)NCCSC)CCN(Cc2ccc(F)c(OC)c2)CC1 33490,C(=O)(CC(C)(C(F)F)N(C)C)NC(CN(C(c1ccc(C)cn1)=O)C)C 33491,Cc1cc(CC(N2CCCC2CNC(=O)C(C)N(C)C)=O)ccc1Cl 33492,C1(NC(CCC(=O)OCC)=O)CS(=O)(=O)CC1NC(=O)CC1CCCCCCC1 33493,c1(CC)cc(C)c(C(=O)NC2COC(C3CCNCC3)C2)o1 33494,CC1(NC(=O)C(c2cccs2)=O)CCN(C(c2ccc(OCC3CC3)cc2)=O)C1 33495,c1(SC(C(=O)NC(CNC(c2cc(CCC)on2)=O)C)C)ccc(F)cc1 33496,C1(C(=O)NC2CN(C(C3CC(CF)C3)=O)CC2C(F)(F)F)SC2C=CC1CC2 33497,C(=O)(CC(C)(C(F)F)N(C)C)NC1C(O)CCN(C(CC=CC=C)=O)C1 33498,N1(C(CCC=CC)=O)CCCC1(C)CCC(N1C2CSCC1C2)=O 33499,N1(C2CCN(C(C3CC34CCOC4)C(=O)NCCC)CC2)CCN(CC)CC1=O 33500,C12(N(c3cccc(C)c3)C(=O)C(O)CC)CCCN(c3ncc(F)cn3)CC1C2 33501,C1(CC#C)CN(C(=O)COC2CN(C(=O)CSC(C)C)C2)CCO1 33502,c1(CNC(=O)Cc2ccco2)noc(-c2cnn(-c3cnccn3)n2)n1 33503,C(C(CC(F)(F)F)NC(=O)C1=NOC(C)C1)NC(C(NOC)=O)=O 33504,c1(CNC(c2nc(CC)oc2C)=O)ccc2c(c1)CN(C(=O)CCOC)C2 33505,N1(C(C(C)OC)=O)CCC(N(CC(C)C)C(=O)C=CC2CCCCC2)CC1 33506,c1(CC)cccc(CC(=O)NCC(F)CNC(=O)Cn2ccccc2=O)c1 33507,N1(C(C2N(CC)CCOC2)=O)CCCCC(N(C(=O)Cc2ccccc2C)C)C1 33508,C(=O)(CCC(C)(C)NC(=O)C(C1CC1)SC)N(CCN1CC=CC1)CC 33509,c1(CC)cncc(NC(C2(CNC(=O)C(C)NC(=O)C3CC3)CCCO2)=O)n1 33510,C1(C(=O)NCC(O)C(N)=O)(OC)CCN(C(C2CC(O)CN2C)=O)C1 33511,C(=O)(C#CC1CCCO1)NC(CNC(c1c(SC(C)C)cccc1)=O)(C)CO 33512,N1(C(=O)NC2C(C(N)=O)CCCC2)CCOC2(CCS(=O)(=O)C2)C1 33513,Cc1cc(O)nnc1C(=O)NCC1(C)CCN(C(=O)CC2CCC(C)C2)CC1 33514,C1(C(N2CCC=C(CNC(C3(F)C(C)OCC3)=O)C2)=O)CCn2cncc2C1 33515,C1(NC(c2[nH]c(=NC)sc2)=O)CN(C(c2ccnnc2S)=O)C2(CCCCC2)C1 33516,C1(C(=O)NCCc2ccc(Br)cc2)CC1C1CCNCC1 33517,CCCCS(=O)(=O)CC(=O)NC(C)CN(C(C1CCCN1C1CC1)=O)CC 33518,N1(C(CCCCN(C)C)=O)CCC2(CCCN2C(C2CCC(C)(C)C2)=O)CC1 33519,N1(c2nc(C)c(Br)cn2)CC(NC(c2ncc(Cl)s2)=O)CC(C)(C)C1 33520,N1(C(c2c(OC)oc(C)n2)=O)CCC12CN(C(C1CC3CCC1O3)=O)C2 33521,Cc1cc(C(=O)NC(CO)C(C)NC(C2CC(F)(F)CS2)=O)cc(C)c1Cl 33522,Cc1ccc(C)c(OCC(N2CC(O)(CNC(c3csc([N+](=O)[O-])c3)=O)C2)=O)c1 33523,C1(n2cc(C(CSCC)C)nn2)CN(C(=O)Cn2cccn2)CC1C 33524,Cc1ncc(C(F)(F)F)cc1C(=O)NC1CCCCN(C(C2(C(F)F)CC2)=O)C1 33525,c1(CNC(c2ocnc2C(=O)NC2(CC)CCSC2)=O)oc(C)nc1C 33526,c1(C(N2CC(CCNC(c3c(CC)nns3)=O)(OC)C2)=O)cc(C(C)C)nn1C 33527,c1(C(=O)NC2CCC(NC(c3cn(CC(N)=O)nn3)=O)CC2)ccc(O)nc1Cl 33528,CCC(C(=O)NCCC(O)CNC(=O)C(C1(C#N)CCCCC1)CC)C(F)(F)F 33529,N1(C(c2nc(CCC)oc2)=O)CCN(C(C)CNC(C23CC(CCO2)C3)=O)CC1 33530,Cc1nc(C(=O)NC2N(C(C(C3CC(C(=O)N(C)C)C3)F)=O)CC2)c(C)o1 33531,C1(CN(C(=O)Cn2cnnc2)C)CCC(CNC(=O)C=CCn2cncn2)CC1 33532,Cc1nn(C2CCOCC2)cc1C(=O)NCC1(NC(=O)C=CS(C)=O)CCCC1 33533,c1(CN2CC3CCC(CC(=O)OC)(C2)C3)cc(F)cc(F)c1Br 33534,CCCCCC(C)CC(=O)NC1CCCCC1NC(=O)CN1CCNC1=O 33535,N1(C(C2(C)CCN(C)C2)=O)CCN(C(c2cc(Cl)c(Cl)s2)=O)CC(CO)C1 33536,c1(C(N2CC3CCCC3C2)=O)cc(S(=O)(=O)O)ccc1O 33537,C(=O)(C(C)C(F)(F)F)N1CCC(C(C)NC(c2cccc(C)n2)=O)CC1 33538,C1(NC(C=CC=CC)=O)CCCC12CN(C(c1cccc(C(F)(F)F)n1)=O)C2 33539,c1(C(=O)NC2(C)CCCN(C(c3cc(C)on3)=O)C2)cc2cnccc2o1 33540,c1(C(N2CCC(c3ncc(C(=O)O)s3)C2)C)cccnc1 33541,C(CCCOC)(C(=O)N1CC(CF)C1)NC(c1nn(CC)nc1C)=O 33542,c1(C(N(C)CC2CCN(C(c3cn(CCO)nn3)=O)C2)=O)cc2cnccc2o1 33543,N(C(=NCCCCc1ccc(Cl)s1)NCc1ccccc1Cl)CC1CS(=O)(=O)C1 33544,C1(CC(=O)NCC(CO)NC(=O)C(C2CCCC2)C2CCCC2)CCOC1 33545,N1(C(C(N2CCC(C)C2)=O)=O)CCC(O)(NC(=O)Cc2ccccc2)CC1 33546,C1(C(=O)NCCCCCO)(CC)CCCN(C(=O)COCC(F)F)C1 33547,c1(C(=O)OCC)nc(=NC2CC(F)(CNC(=O)C(C)COC)C2)cc[nH]1 33548,Cc1c(Cl)cc(C(=O)NCCCC(=O)N(CCCN)C)cc1Br 33549,CCC(C(=O)N1CC(NC(c2csc(C)c2OC)=O)C1)C(C)C 33550,C1(CC)CN(C(=O)CC(C)C(C)C)CCN1C(C1CC(F)C1)=O 33551,C1(C(=O)NCC2CCC(NC(=O)CCCC3OCCO3)C2)C2CCC1CC2 33552,C#CC1(NC(=O)CCCC(C)NC(c2coc(C(N)=O)c2)=O)CCCCC1 33553,C1(NC(c2ccccc2-n2cnnn2)=O)CN(C(C2CC2(F)F)=O)CC1C(F)F 33554,C(=O)(C1=C(Cl)CCCC1)N1C(CNC(C2C(C(N(CC#C)C)=O)C2)=O)CC(F)C1 33555,C1(NC(c2nc(C(C)NC(CC(C)C)=O)oc2)=O)CCN2CCC1C2 33556,C(CC(O)CCC(C)(C)C)NCCc1cn(CCOC)nn1 33557,CCC(C)C(C(=O)NCC1COCCN1C)N(C(=O)CCC(C)OC)C 33558,N1(C(c2ccc(C(C)C)o2)=O)CC2CC(NC(=O)C(F)(F)C(C)O)C1C2 33559,C1(CNC(C(CCOC)C)=O)CCC2(CN(C(C3CCOC(C)C3)=O)C2)O1 33560,C(=O)(CCc1ccc[nH]1)N(C(C)C(=O)NC(C)C(=O)NC)CC 33561,c1(CC)ccc(C(=O)NCC(=C2CN(C(c3nnc(C(C)C)s3)=O)C2)F)c(O)c1 33562,c1(C(N2CC(CC(C)NC(=O)CCC3CCOC3)C2)=O)ccc(C(F)F)cc1 33563,N1(CC(=O)Nc2cnc(C)s2)CCN(C(c2cc(-c3ccco3)on2)=O)CC1=O 33564,C#Cc1ccc(C)c(NC(=O)C(CCC=C)NC(c2sncc2C)=O)c1 33565,Cc1cc(-n2cc(CN3CCC(c4ccc(C(=O)O)cc4)C3)nn2)cc(=O)o1 33566,CC(C)(CS(N)(=O)=O)C(=O)N1CCN(C(c2ccn(C3CC3)n2)=O)CC2(CC2)C1 33567,C(C(CC(C)C)C(=O)NCC(C)CN(C)C(C1CCCN1C)=O)OC 33568,C=CC(C(=O)NCC1CCN(C(=O)Cc2cnccn2)C1)NC(=O)OC(C)(C)C 33569,C(N=c1nnc(C)c(C)[nH]1)C1CN(C(c2ccc(C)c(F)c2)=O)CC1C 33570,N1(CC(=O)NCC(CC(C)C)NC(C2CCC23CCC3)=O)CCc2sccc2C1 33571,N1(C(c2cc(C(C)=O)sc2)=O)CCN(C(=O)C(F)(F)c2cccnc2)CC1C1CC1 33572,c1(N(CCOC)C)nc(=NCCc2nc(CO)n[nH]2)[nH]c2cc(OC)ccc12 33573,c1(C(C(=O)NCCN(C(=O)C(C)C(C)C)CCC)O)cccc(Br)c1 33574,C(CC(C)C(=O)N(C1CCN(C(C2(n3cc(Cl)cn3)CC2)=O)C1)CCO)=CC 33575,C1(C(=O)NCC(C)NC(c2cc(Cl)ncc2N)=O)CCc2cc(F)ccc2O1 33576,CC1CC(NC(=O)Cc2ccc(F)cc2)CN1C(=O)CC1CCS(=O)(=O)C1 33577,CCCC(CCCNC(=O)CN1CCOCC1)Nc1ncncc1I 33578,Cc1cccc(C)c1NC(=O)C(c1cc(Br)ncc1F)N1CCC(C(F)F)CC1 33579,C(=O)(CC(CC)CCC)NCCC1CCCN(C(C(C#C)(C)C)=O)C1 33580,CC(C)CCC(F)C(=O)NC1CC1CNC(c1cc(C(N)=O)n(C)n1)=O 33581,c1(SCC(=O)NCCC2CCCN(C(C=C(C)C)=O)C2)nc2ccccc2s1 33582,Nc1nc(C(N2CC(NC(c3cnns3)=O)CC(O)C2)=O)cnc1Br 33583,C(=O)(C(C)(F)CCCC)NCCCCC(C)NC(C(C=C)(C)CC)=O 33584,c1(CN(CC(C)C)N(C)C(C)c2nncn2C)nnc2n1CCOCC2 33585,c1(C(N2CC3(CC3C(N3CCC(c4cn[nH]c4)CC3)=O)C2)=O)cccc(Cl)c1Cl 33586,c1(C(N(CC(CC)NC(C2(CF)CCC2)=O)C)=O)c(C)nc2sc(C)nn12 33587,C1(CNC(C2CCCN(C(C)=O)C2)=O)CCCCN(C(C23CC(C2)C(C)O3)=O)C1 33588,CCCC(CC)C(=O)N1CC2C(CC(=O)NC3CCN(OCC)CC3)C2C1 33589,N1(C(c2nc(CCC)sc2)=O)CC(CNC(=O)C=CC2CC2)C2CC12 33590,Cc1cccc(-c2cccnc2NCC(N2CCN(C)CC2)=O)c1C 33591,N1(C(CSCCC)=O)CCN(C(c2cnc3ccsc3c2)=O)C2CCCCC12 33592,CC1(C)CC(C(N2CCOC(CF)C2)=O)CCN1C(=O)CCc1nncs1 33593,C1(NC(CC2C(C)CCO2)=O)C2CC3C1C3C2C(N1CCC(F)(CF)C1)=O 33594,CC1CCN(C(=O)CNC(=O)Cc2cnn(C)c2)CCS1 33595,c1(NC(C2C(C)CCCC2)=O)cnc2ccc(F)cc2c1 33596,CC1CCN(C(c2cc(O)nn2C)=O)C1CNC(c1ccc(C2(C)CC2)cc1)=O 33597,c1(C(C)(CO)OC(C2CCN(C)C2)=O)cccc(CNC(=O)NC(C)(C)C)c1 33598,c1(N2CCC(CCOC)C2)ncnc(NC(COC)CC(C)C)c1C 33599,C1(C(=O)NC(C(C)NC(=O)CCN2CCCCC2)C)CC2COCC2C1 33600,c1(C(N(C2CCCC(NC(C=C(C)c3cccs3)=O)C2)C)=O)cnc(C)c(N)c1 33601,Cc1cnc(C(N2CCC(NC(C3CC(CN(C)C)C3)=O)C23CC3)=O)cc1C 33602,C1(C(=O)NC2COCCN(C(CN3CCC(C)(C)C3)=O)C2)CCCC2(CCC2)O1 33603,Cc1cc(F)cc(C)c1C(N1CC(NC(c2[nH]cnc2C#N)=O)C1)=O 33604,c1(N2CC(CC=C)(NC(=O)CC3CC(O)C34CCC4)C2)nc2ccc(Br)cc2o1 33605,N1(C(c2cn(C)nc2)=O)CC=CC(NC(C2CCCC2(C)C)=O)C1 33606,Cc1cc(C(=O)N(C(C)CN(C)C(C2CC2Cc2ccccc2)=O)C)on1 33607,c1(NC(C(c2c(OC)cccc2)N(C)CCSC)=O)n[nH]c2c1CCCC2 33608,C1(C(=O)NCC23C(CN(C(C=CC(N)=O)=O)C2)C3)COc2ccccc2O1 33609,C#Cc1ccc(C(=O)NC2(COC)CCN(C(=O)C(C(C)C)NS(C)(=O)=O)C2)nc1 33610,C=CCCCC(=O)NCC(CC=C)NC(=O)C(=C1CCCCC1)F 33611,c1(C(=O)NC2(C)CCN(C(c3cccc(O)n3)=O)C2)oc2ccccc2c1Cl 33612,N1(C(c2nc(CC)oc2C)=O)CCC2CN(C(c3cn(C)nc3OC)=O)CC12 33613,C=C(C)CCC(=O)NCC(CO)NC(=O)CC(C)C 33614,C(=O)(C(C(C)O)NC(=O)Cc1cn[nH]c1)NCC1(C(C)C)CCCC1 33615,C1(NC(c2ccc(-n3ncc(S(C)(=O)=O)c3)cc2)=O)CCCC12CCCCC2 33616,C(=O)(C1=CCCCO1)N1CCN(C2CCCN(C(CSC)=O)C2)CC1 33617,c1(C(=O)NC2C(C)N(C(=O)Cn3ncnn3)CC2)cc2c([nH]1)CCOC2 33618,CC(C)(CCC(=O)NC1CCC(C(N)=O)C1)NC(C1CC=CC(O)C1)=O 33619,CCCCC(CCCC)C(=O)NC1(CNC(=O)C(O)CC(C)C)CCCC1 33620,Cc1nncc(C(N2CCCC2C(C)NC(C2CC23CCC3)=O)=O)c1C 33621,C(C)(CNC(C1CCNC1=O)=O)(CO)NC(C=C(CC)CC)=O 33622,C1(N(c2ccc(-c3ccc(C)nc3O)cc2)C)CCCCCC1C(F)(F)F 33623,c1(C(N2CC(NC(C3N(CC)CCC3)=O)C2)=O)nc2ccc(C)cn2c1N 33624,C(CC(C)(C)N(C1CCC1)C(c1ccncn1)=O)N(C)C(C1(N(C)C)CC1)=O 33625,c1(C(=O)NCC2C(NC(c3c(OC)cccc3)=O)CCC2)ccc(C)c(C)c1 33626,C=CC(CC)CC(=O)N1CC(O)(C(C)(C)CNC(C2CCCN(C)C2)=O)C1 33627,c1(C2(N(C(Cc3nnc(C)o3)=O)CC3CC3)CCCC2)ccc(OC(F)F)cc1 33628,CC1(C(=O)NCC2CC(NC(=O)CCc3cnoc3)C2)CC(C#N)C1 33629,c1(OC)ccc(NCc2cc(C)c(-c3cccnc3C(F)(F)F)cn2)cc1C 33630,C1(N(C)C)(C(=O)NCC(O)CCNC(=O)CCC2CCC2)CCOCC1 33631,C12(NC(C3CCOC3)=O)CCC(C1)N(C(c1cc(Cl)ccc1-n1cccc1)=O)C2 33632,c1(C(N(C)CCn2cc(COC3CCCC3)nn2)=O)cc(C(=O)O)ccn1 33633,C1(C2CCCC2)(NC(C2C(C)CCN2C(=O)C(C)c2cc[nH]n2)=O)CC1 33634,C(C(=O)NCc1cccs1)(C(C(C)C)OC)N1CCCC(C(=O)OC)C1 33635,C(=O)(C1=NOC2(C1)CN(C(=O)OCC(C)(C)C)C2)NCC=C(C)C1CC1 33636,c1(N(C)Cc2ccoc2)ccc(S(=O)(=O)NC2CC3CCC(C2)S3)cc1F 33637,c1(C(=O)NCCCN(C(C(CSC)O)=O)C)ccc2c(c1)CC(=O)NC2 33638,C=CC(C)(O)CC(=O)N1CCCC1C(C)NC(c1cc(CC)nn1C)=O 33639,C1(NC(C(C(=C)Cl)(C)C)=O)CN(C(=O)C(C)CC(=C)C)C2(CCC2)C1 33640,C1(CNC(C(C)Sc2nncn2C)=O)CCCC(NC(=O)CCn2cccn2)C1 33641,N1(CC)CC(C(=O)NCC2CCN(C(=O)C(=CC3CCCC3)C)C2)NC1=O 33642,N1(CC)CCCCC1C(=O)N(C1CCN(C(=O)CCSc2ccccc2C)C1)C 33643,c1(C(=O)NCCC23C(CN(C(CCOCC)=O)C2)CC3)sc2ccccc2c1C 33644,c1(C(=O)NCC(C)CNC(=O)CCn2cc(Cl)cn2)ccc([N+](=O)[O-])c(O)c1 33645,c1(N2CCC(NC(C3(C)ON=C(C)C3)=O)C2)nc(C)c(C#N)cc1Cl 33646,c1(C2(CNc3cncc(C(=O)OCC)c3)CC2)ccc2c(c1)OCCCO2 33647,N1(C(c2ccn(C(C)C)n2)=O)CCCC2(NC(=O)C(C)n3ccnc3)CC2C1 33648,c1(C(=O)NC(CCN(C(C(CSC)OC)=O)C)C)c[nH]cc(Br)c1=O 33649,N1(C(c2nc(C)n(C)c2)=O)CCCC(NC(c2[nH]ncc2C#N)=O)CC1 33650,CCCC(CC)C(=O)NCc1cccc(C(=O)N(C)CC2CCN(CC)C2)n1 33651,N1(C(c2ccn(CCC)n2)=O)CCCC2(CCCN2C(c2cc[n+]([O-])cc2)=O)C1 33652,N1(C(C(c2ccc(OC)cc2)C)=O)CC(C2CCN(C(=O)C(O)C3CC3)CC2)C1 33653,c1(-n2c3nc(n2)N2C(=O)CC3C2)cc(C)ccc1OC.CCC(C)C 33654,CC(C)(C)C1=NOC(C)(C(=O)NC2CCCCC2NC(=O)Cn2cnnc2O)C1 33655,CC1CN(C(C2CCCN2C)=O)CC(C)CN1C(=O)CCc1ccco1 33656,CN=c1ncc(-c2csc(C(N3CCOC3=O)=O)n2)c[nH]1 33657,c1(NC(CCC)=O)ccnc(C(N2CC(CO)(NC(C3CCC4CC34)=O)C2)=O)c1 33658,C1(CCC(=O)NC(CN(C(C(C)=C(CC)C)=O)C)CC)CCC(=O)NC1 33659,C1(C(=O)NCC2(COC)CN(C(C(C=C)C)=O)C2)CCC2(CCC2)C1 33660,C(=O)(C(O)CC(C)(C)C)N1CCC(N(C)C(c2cc(-n3cnnc3)ccn2)=O)C1 33661,N1(C(C2(CNC(c3cc(C)sn3)=O)CCC2)=O)CC(C)(C)OC(C)(C)C1 33662,Cc1cnc2c(C(=O)NCC(CO)NC(C3CC34CCCCC4)=O)cnn2c1 33663,CS(=O)C=CC(=O)NCC1C2CN(C(C3CC(O)(c4cccnc4)C3)=O)CC12 33664,c1(C(=O)NCC(C)NC(=O)Cn2cc([N+](=O)[O-])cn2)ccc(N)cc1Cl 33665,CC1Cc2cccc(C(=O)N(CCCCNC(c3ncc(C(F)F)s3)=O)C)c2O1 33666,c1(C(N(CCN(C)Cc2c(OC)ccc(Br)c2)C)=O)cncc2nc[nH]c12 33667,c1(C(N(CC(=O)O)CC2CC2)=O)ccc(-n2cc(-c3cncc(CO)c3)nn2)cc1 33668,c1(CNC(N(C(C(=O)OCC)C)C)=O)ncncc1C 33669,C1(C(=O)NCC2CCCC2C(C)C)(NC(COC(C)=O)=O)CC(F)(F)C1 33670,S(=O)(=O)(c1ccc(N(C)C)cc1Cl)NCCNC(C)Cc1nc(C(F)(F)F)cs1 33671,C(c1cccc(F)c1Cl)=CC(=O)NC1C(CNC(Cc2cn(C)nn2)=O)COC1 33672,c1(CC(=O)NCC(CCNC(C(C2CC2)SC)=O)O)cc(C)ccc1C 33673,c1(C(=O)NCC23CC(NC(C4CCC45CCCO5)=O)(C2)C3)cnc2c[nH]nc2c1 33674,C1(O)(C(C)NC(=O)CC(C)C2CCCO2)CCN(C(=O)CC(C)n2ccnc2)C1 33675,CCCC(CCCNC(=O)CC1COCC1(C)C)NC(c1cnc[nH]1)=O 33676,C1(NC(C(CC)CC)=O)CCC(C)N(C(=O)C(c2cccc(Br)c2)C)C1 33677,c1(OC)c(C(=O)NC2COCC2NC(=O)Cn2nc(C)nc2C)ncnc1C 33678,Cc1cccc(Br)c1-c1ccc(CNC(=O)C(N2CC(F)CC2CO)=O)o1 33679,c1(N2CCN(C(C34CNCC3(F)CCOC4)=O)CC2)ccc2c(c1)C1(CC1)C(=O)N2 33680,Cc1cccc2c1OCCN(C(=O)C(C)(N)CC(C)C)C2 33681,CCCS(=O)(=O)C(C)C(=O)NC1CN(C(c2cc(C(F)F)[nH]n2)=O)CC1C1CC1 33682,C1(CNC(C2(CC)CCCC2)=O)CC2(C1)CN(C(=O)Cc1cc(C)on1)C2 33683,c1(C(=O)NC(CNC(c2cncc(CC)c2)=O)CO)cc(C(C)C)ccc1N 33684,N12CC3CCC(C3)(C1)C2=O.Cc1sc(C(=O)NC(=O)C(C)CO)c(C2CC2)c1C 33685,N1(C(C2C(CC)OCC2)=O)CCC(F)(CNC(C23CC2C3)=O)CC1 33686,CC(CC(F)(F)F)C(=O)NCCNC(C1CCCN(C(=O)C#CC2CCC2)C1)=O 33687,C=CC1(C(=O)NC2C3CCCC23)CCN(C(c2ccc(C)[nH]2)=O)C1 33688,C1(NC(CC2(OC)CC2)=O)CCCCCC1NC(c1ccc(N)c(SC)c1)=O 33689,C1(COC)(CNC(=O)COC(C)C)CCN(C(=O)CNc2ccncc2)CC1 33690,c1(C(=O)NCCC2(C(=O)NCCC(=O)NC3CC3)CC2)cnc(C(F)(F)F)o1 33691,Cc1ncc(CC(=O)NCC(C2CC2)NC(=O)C(C)N2CCC2)[nH]1 33692,c1(OC)ccc(C(F)(F)F)cc1C(=O)NC1CN(C(C2COC(=O)N2)=O)C1 33693,C(=O)(N=c1cc2ccccn2[nH]1)C1(C)C=CCN1C(c1cc(Cl)cs1)=O 33694,c1(OC(C)(C)C)ccc(C(=O)NC2CCN(C(c3coc(Br)n3)=O)CC2)cn1 33695,c1(C(N(CC(C)NC(=O)CC#N)C)=O)cnoc1C1CCOCC1 33696,N1(C(CSC(C)(C)C)=O)CCN(C(=O)C(F)C(C)(F)F)CC1c1cn[nH]c1 33697,Cc1cc(C(=O)NCC(C)(CO)NC(=O)C=Cc2nccs2)ccc1Cl 33698,C1(CCNC(=O)CCCn2cncn2)(OC)CN(C(=O)C(c2ccc(C)s2)C)C1 33699,c1(-c2ccc(NCc3c(C)nc(F)cc3)nc2)c(C(F)(F)F)[nH]c2ccccc12 33700,c1(C(c2ccco2)O)nn2c(c1CNCC(O)COc1ccc(Cl)cc1)CCC2 33701,c1(CC(=O)NCC(CC)NC(=O)CC2(O)CCCN(C)C2)c(F)cncc1Cl 33702,CN1C(=O)CCC(C(N2CC(c3ccccc3F)C2)=O)C1c1ccccc1 33703,N1(C(COCC(C)C)=O)CCC(C)(CCNC(C2CC(C)C2)=O)C1 33704,Cc1nn(C)c(C)c1C(N1CC2CC(C1)C2NC(=O)C(C)N1CCC1)=O 33705,C1(CCNC(c2cc(C)on2)=O)CCN(C(C2CCCN2C=O)=O)CC1(F)F 33706,C12C(C1(C)C)C(=O)N2.C1(CCNC(C2CC(N(C)C)C2)=O)CC(F)(F)C1 33707,N1(C(c2scc(C)c2C)=O)CC(C(N2CCCC(O)(C(N)=O)C2)=O)C2(CC2)C1 33708,Cc1ccoc1CN(C(=O)C(C)(C1CC1)N(C)C(c1cnn(C(C)C)n1)=O)C 33709,C1(CC)CN(C(C2(NC(=O)CC(C)CN(C)C)CCOCC2)=O)CC(=O)N1 33710,c1(CSC)cccnc1C(N1CCOC(CNC(C2CCC(=O)N2C)=O)C1)=O 33711,S(=O)(=O)(c1cccnc1N1CCC(OC)CC1)NC.C1(N)CCCOC1C(C)(C)C 33712,CCCCC(F)C(=O)N(C1CCCN(C(c2c[nH]c(=N)c(C)c2)=O)C1)CC1CC1 33713,CCC(C)(C)C(=O)C(=O)N1CC(F)(C(=O)NC2(C(C)O)CC2)C1 33714,c1(C(=O)NC2C(CNC(c3c(CC)c[nH]c3)=O)CCCC2)cn(C)c(=O)cn1 33715,c1(C(N(C(CNC(C2CCC(=O)O2)=O)C2CC2)C)=O)cc2ccccn2n1 33716,C1(C)(C(=O)NCC(CCOC)NC(=O)CCCn2cccn2)CC(=O)N(C)C1 33717,c1(CC)cccc(N(C)C(c2cc(CNC(=O)CC3CC=CCC3)no2)=O)c1 33718,C(=O)(C(S(C)(=O)=O)C1CC1)N(C(C)CNC(c1ccc(Cl)o1)=O)CC 33719,C1(OC)CCCC(CNC(=O)CN(CC(C)C)C(=O)Cn2cncn2)C1 33720,C1(C2CCCC2)(C(=O)NC2C3(CCN(C(c4cc(Cl)nnc4O)=O)C3)C2)CCC1 33721,C(=O)(C(O)C(C(C)C)OC)N(C)CC1N(C(c2cc(CC)n(C)n2)=O)CCCC1 33722,CC1COCCCN1C(C1CN(C(C2CCCC2)=O)C(C)(C)C1)=O 33723,Nc1cnc(Cl)c(C(N2CCOCC(NC(c3ccc(F)s3)=O)C2)=O)c1 33724,c1(C(N(CC#C)C)=O)cccc(-n2cc(CNC(C3(CSC)CC3)=O)nn2)c1 33725,c1(C(N(C)CC2CCN(C(C3CCC(C)(C)C3)=O)CC2)=O)cc(O)c(O)c(O)c1 33726,c1(C(N(C2CCC(NC(C3CCC(F)C3)=O)CC2)C)=O)cc2cnn(C)c2s1 33727,C1(c2n(CC)nnn2)(NCCc2cncc(OC)c2)CCN2CCCCC12 33728,C1(CNC(C2(CC)CCN(C(C3CCCSC3)=O)C2)=O)CCC(C)(C)CC1 33729,c1(CCC(=O)Nc2cccc(NC3CCCC3)c2)ccc(Cl)c(Cl)c1 33730,N1(C(CCC(=C)C)=O)CCN(C(=O)C(C)CCC)C(c2cn[nH]c2)C1 33731,c1(C(=O)NC(C)(C)CSCC)cnc(CC)[nH]1.C(=O)(COCCOCCOC)N 33732,c1(C(=O)NCC2CN(C(=O)C=CCF)C2)cccc2cncn12 33733,C#Cc1cc(C(=O)NCCNC(C2CC[Si](C)(C)CC2)=O)cc(F)c1 33734,N(C(=NCCOc1ncccc1Cl)NC(C1CC1)C1CC1)CC1CCC(C)O1 33735,C1(c2nn(C(CC)C)c(-c3nc(C)c(C)s3)n2)CCC(F)(F)CC1 33736,c1(CNC(C2N(CC)CCC2)=O)sc(OC)nc1Cl 33737,c1(Nc2ccc(OC)cc2CC(N)C(=O)O)nc(C)nc2scc(CC(C)C)c12 33738,C1(NC(CSC(C)C)=O)COCCC1NC(c1cccnc1-n1nccn1)=O 33739,c1(CNC(=O)NCC2C(NC(=O)OC(C)(C)C)CC2)ccc(Cl)o1 33740,C=C1CCN(C(c2nscc2C)=O)C(C(=O)NCCC2CC=CCC2)C1 33741,Cc1ccc(C(=O)NCc2cc(C(=O)NCC3CCCC3)no2)c(O)n1 33742,c1(NCC)cccc(C(N2CC(F)(CNC(=O)C(C)OCCC(C)C)C2)=O)c1 33743,c1(C(N(C(CNC(CC=C)=O)C)CC)=O)cnc(Br)c(N)n1 33744,N1(C(c2c(CNC(C3C(C)CC3)=O)n[nH]c2)=O)CC2(CNC(=O)OC2)C1 33745,c1(CC(=O)NCC(Cn2cc(CCO)nn2)OC)cc(Cl)cc2c1OCC2 33746,CC1(C)OCCOC1C(=O)NCC1(O)CN(C(c2ncsc2C2CC2)=O)C1 33747,N1(C(c2ccc(C)[nH]2)=O)CCN(C)C(CNC(=O)C(c2cccnc2)O)C1 33748,N1(C(C(C)=CC)=O)CC(C)(C)CC1CNC(=O)CC(=O)N(C)C 33749,C1(CNCCOC(C)=O)CN(C2CCCCC2)C(=O)O1 33750,C1(C)(OC)CCCN(C(=O)C(C)(CNC(c2ncoc2C)=O)CC)C1 33751,CN1CCOCC1CC(=O)NCCCOCCNC(=O)Cc1cc(C2CC2)no1 33752,CCC(CC(C)C)C(=O)NCCN(c1ncc([N+](=O)[O-])cn1)CCOC 33753,N1(C(C(C(CC)C)OC)=O)CC2CCC(C1)N2C(=O)C(N1CCN(C)CC1)(C)C 33754,c1(C(=O)NC2C(Cn3cc(CN(C(C)=O)C)nn3)CCC2)cc(F)cnc1O 33755,C(=O)(C(CC(C)C)NC(c1c[nH]c(C#N)c1)=O)NC(C(CC)CC)C 33756,C1(NC(C2(NC(=O)C3=COCC3)C(C)C2)=O)CCC(C2CCC2)CC1 33757,C1(CC(=O)NCC(CNC(=O)CCc2nccs2)F)CCCCC12CC2 33758,N1(C(C(CC)c2ccccc2)=O)CC(CNC(=O)CC(C)(F)F)C2(CC2)C1 33759,c1(CN(C(C2C(CNC(C(CN(C)C)N(C)C)=O)C2(C)C)=O)C)cccc(O)c1 33760,c1(C(=O)NC2CCCC(NC(CNC(=O)NC)=O)C2)cc(C)cc(F)c1 33761,c1(CNC(C2(CC(C)C)CC2)=O)ccc(CN(C)C(C2C(F)(F)C23CC3)=O)cc1 33762,c1(C(=O)OCCN(CCN(C)C)C)cc(C#N)c(Br)s1 33763,CC1CCN(C(=O)OC(C)(C)C)C1C(=O)NCC1CCC(CC(C)(C)O)CC1 33764,N1(C(C(=O)NC(c2ccc(C)cc2)=O)=O)CCC(NC23CC(CO2)C3)C(C)C1 33765,C1(C2CC2)(CNC(c2sc(C)c(C)c2C)=O)CCN(C(=O)C2=CCOC2)C1 33766,c1(C(N2C(CCN(C(=O)Cn3nccn3)C)CCCC2)=O)c[nH]c2nccc-2c1 33767,c1(OC)ccc(O)c(C(C)NCc2ccccc2Cn2cc(Cl)cn2)c1 33768,Cc1ccc(CCC(N2CC(C)(NC(c3cc(Cl)c(Cl)[nH]3)=O)C2)=O)cc1Cl 33769,C(CCC(C)NC(=O)CN1CCOC1=O)NC(C(C)SCC)=O 33770,Cc1nnc2n1C(C(=O)N1CCN(C(c3csc4nnsc34)=O)C(C)C1)CC2 33771,N#Cc1cnn(CC(=O)OCCOc2ccc(Cl)cc2)c1 33772,C1(NC(C(C)=C(C)C)=O)CC2CCC1N(C(=O)C=Cc1ccc(C#N)cc1)C2 33773,C1(CNC(C2N(C)C(=O)NC2)=O)C(O)C(O)CN1C(c1ccc(F)cc1)=O 33774,c1(OC(C)C(N2CCC(C)(CNC(=O)C=C3CCCC3)C2)=O)cc(Cl)cc(Cl)c1 33775,O=S(N1CCCCCC1CC1CC1)C1CCNCC1 33776,C1(CC(N2CCC(NC(=O)CC3CC=CC3)(CF)C2)=O)CN2CCN1CC2 33777,C=CCCC(CC(C)C)C(=O)NC(C)CN(C(=O)COc1cccc(C)c1C)C 33778,N1(C(c2ncc(OCC)nc2)=O)CCCC(NC(=O)CCc2csc(C)n2)CC1 33779,Cc1cccc(C(N2C(C(=O)NCC=CC3CC3)CCC2C2CC2)=O)c1F 33780,c1(CN2CCC(N(C(C=CC(C)C)=O)C)CC2)ccc([N+](=O)[O-])cc1O 33781,C(CCCC(=O)NC1(C)CCN(C(=O)C(C)(C)c2cccnc2)C1)OCCC=C 33782,c1(C(N(CC(C)NC(CC(=C)Br)=O)C)=O)ncccc1S(=O)(=O)CC 33783,N1(C(C2(CCN(C)C)CC2)=O)CCC2(CC1)CC2NC(=O)C(c1cccnc1)O 33784,c1(C(N2CC(C)(C)N(Cc3ccccc3)CC2)=O)nc2c(F)cc(Cl)cc2s1 33785,N1(C(c2c(CC)con2)=O)CCC(NC(=O)CCCN(C)C)C1C1CC1 33786,Cc1ccc(C#N)cc1NC(=O)C(C)N(C(=O)CSc1nc[nH]n1)C1CC1 33787,C(CC(C)C(=O)NCC1CC1NC(c1ccnnc1C)=O)=CCC 33788,Cc1cc(Cl)c(Cl)cc1C(=O)NCCN(C(=O)CC1(C)CC1F)C(C)C 33789,N1(C(c2cc(CCCCC)[nH]n2)=O)CCCOC(CNC(=O)C=CC=C(Cl)Cl)C1 33790,C1(C)(C(=O)NC(C(=O)N2C(CC)CC2)CO)CC(=O)N(C)C1 33791,C1(CCC)CNC(=O)CN1C(C1CCC(NC(=O)NC2CC(=O)N(C)C2)CC1)=O 33792,C(CC(CC)C(=O)N1C(CC(=O)NCc2cnc(C)n2CC)C2CCCC12)=CC 33793,C1(CC(N2CCC(O)(CN(C(=O)CSCC(N)=O)C)C2)=O)CC2CCC(C1)N2C 33794,N1(C(C2(C(C)=O)CC2)=O)CC2(CCN(C(=O)Cc3nnc(C)o3)C2)C1 33795,C12(CNc3ccnc(C)n3)CC(NC(=O)C=Cc3ccncn3)(C1)C(C)(C)O2 33796,c1(OC)ccc(C(F)(F)C(N2CC3CC3(CNC(=O)C(C)C3CCC3)C2)=O)cc1 33797,O=C(C1=NOC2(CCN(S(=O)(=O)C3CCCC3)C2)C1)N1CCc2ncncc2C1 33798,C#CC1CCC(CNC(=O)CC2CCN(C(C3(CC)CCC3)=O)CC2)CC1 33799,CCC(CC(=O)NCCC1CN(C(=O)C(C)(C)CCOC)C1)CC(F)(F)F 33800,C1(C(N(CC(CC)(C)OC)C)=O)(C(C)C)CCN(C(c2coc(C3CC3)n2)=O)C1 33801,C1(CC(N2CCC(NC(COCCN(C)C)=O)(CO)C2)=O)CC2CCC1CC2 33802,c1(C(N(CCCNC(=O)C2=NNC(=O)CC2)C)=O)ccc2nc(Br)nn2c1 33803,S(=O)(=O)(c1cc(C(N2CCN(C(=O)CSC(F)F)C(C3CC3)C2)=O)co1)N(C)C 33804,N1(C(C(C)SC(C)C)=O)CC2CC2(C(=O)NC2CC3CCC2O3)C1 33805,C1(NC(C2C(C)CCOC2)=O)CCCCCC1C(=O)NCC1CC12CCC2 33806,c12[nH]c3ccccc3c1CC1(CC)COCC(CCCNC2=O)CNC1=O 33807,N1(Cc2cccc(C(=O)NCC(C(C)(C)C)SC)c2)CCC(S(N)(=O)=O)C1 33808,c1(OC)cc([N+](=O)[O-])cc(CN2Cc3[nH]nc(C(N)=O)c3C2)c1O 33809,C1(C)(C(=O)OC)CC(NC(=O)C=CC(=O)NC(=O)C(c2cnn(C)c2)C)C1 33810,CCC(O)CC(=O)NC(C)CC(=O)NC1(CCCCO)CC1 33811,N1(C(C2(COC)CCCC2)=O)CCOCC(NC(=O)CC2CCOC2=O)C1 33812,c1(C(=O)NCC2(O)CN(C(C3(C(=O)NC)CC3)=O)C2)cc(Cl)c(OC)cc1Cl 33813,C1(NC(CC=C=C)=O)CCC2(CC1)CC(NC(=O)COCC)C2 33814,c1(C(N(C(C)CNC(c2sccc2CN(C)C)=O)C)=O)ncc(Cl)nc1Cl 33815,Cc1c(I)c(C(=O)OCc2cc(C3CC3)on2)nn1C 33816,O=C(CCS(=O)(=O)N1CCOCC1)N1C2CC2C2CC12 33817,Cc1cc(C(=O)N(CCCNC(=O)CC(=O)NC2CC2)CC2CC2)ccc1O 33818,C(C)(C(CO)NC(c1cscn1)=O)NC(C1(C(C)C)CC1)=O 33819,C(=O)(C(F)(F)CC(C)C)N1CC(CC)N(C(c2cnn(CC)c2)=O)CC1 33820,c1(C(=O)NC(c2cccn2C)C(=O)OC)c(C)ccc(C)c1CN 33821,c1(C(N2CCN(C(C=C(CC)CC)=O)C3C2CC3)=O)cnc2c(c1)CCC(=O)N2 33822,CC1CCN(C(=O)C=C(Cl)Cl)C1N(C(c1ccc(C2CC2)o1)=O)Cc1nc[nH]n1 33823,N1(C(CCSC)=O)CC2CC3CC2C1C3NC(c1cc2sc(C)cc2[nH]1)=O 33824,CC1CCC(c2cn(CC3CCSC3)nn2)CC1 33825,c1(C(N(CC)CC2CCOC2)=O)n[nH]cc1CNC(=O)C(C)=CC1CC1 33826,C(=O)(C(F)CC(C)(C)NC(=O)CCC1CCOCC1)N(C)Cc1nccs1 33827,Cc1ccc(C=CCNC(=O)C(C)CCCc2nc(C(C)C(C)C)no2)cn1 33828,Cc1c(N)ccc(C(=O)NCCN(C(c2csc(Cl)n2)=O)CC2CC2)c1C 33829,N1(Cc2nc(C(C)OC)sc2)CC2CC1CN2C(C1CCCN(C(C)=O)C1)=O 33830,N1(C(CC(CCC)C)=O)CC2(CNC(=O)C(F)OC(F)(F)F)CC1CCO2 33831,CC1CC(C(N2CCC(NC(c3coc(Cl)n3)=O)C(C)C2)=O)CC(=O)N1 33832,c1(NC(c2ccc(COC)o2)c2nnnn2C(C)(C)C)cncc(OC)c1 33833,C(c1ccc(OC)cn1)=CC(N1CCC(CNC(CC=C)=O)C1)=O 33834,CCCC(C)(CC)C(=O)NCC(C(C)C)NC(=O)CC1=CCOCC1 33835,CCCC(C(=O)N(C)CCN(C(C1(OC)CCSC1)=O)C(C)C)C(C)C 33836,C1(NC(=O)CC2CSC2)CC(O)CN(C(c2cnn(-c3nccs3)c2)=O)C1 33837,C1(NC(C=Cc2ccc(CC)o2)=O)CC1C1CCN(C(=O)CC2CCOC2)CC1 33838,N=c1nc(N2CCCC(C3CC3(F)F)C2)[nH]c(=NCCC2CC3(CCC3)CO2)[nH]1 33839,Cc1cc(C)c(C(=O)NC2CCN(C(c3cc(C(C)C)[nH]n3)=O)C2)c(=O)o1 33840,Cc1n[nH]c(C)c1C(C)C(=O)NCC1(CO)CCN(C(C2(C)CSC2)=O)C1 33841,C(CC(F)F)(C(=O)N1CCC1C(=O)N(C)C)NC(c1cc(CC)on1)=O 33842,C1(NC(c2sc(CC)c(C)c2)=O)CC2CCC1N2C(=O)COCC1CCCCO1 33843,C1(NC(c2c(C)cnn2C)=O)CC2CCC1C(NC(=O)C(C)OC1CCCC1)C2 33844,C1(CC(N2CCC(C)C2CNC(c2cc(Cl)c(Cl)n2C)=O)=O)CC2CCC1CC2 33845,CCC(F)(F)CC(=O)N1CC2(CNC(c3nccn3C(C)C)=O)CCC1C2 33846,CCC(CC(=O)N1CCC1COC)NC(=O)CCc1ccccc1O 33847,c1(CC)ncc(Cl)c(C(=O)NC2(CC)CCN(C(C3CCOC(=O)N3)=O)CC2)n1 33848,C1(O)(COC)CCN(C(C2CCC(C)N2C(C2OC3CCC2C3)=O)=O)C1 33849,CC1(C)OC2CC(C(=O)NC3CCCN(C(=O)C4=CSCCO4)CC3)CC2O1 33850,C1(C(N(CCN(C)C)Cc2c(F)cccc2Cl)=O)C2(CCC2)C12CCC2 33851,c1(C(=O)NC(c2cccnc2)CC)cc2n(n1)CCN(C(=O)OC(C)(C)C)C2 33852,N1(C(c2c(OC)ccs2)C(=O)NCc2c(C)ncn2C)CC2CCCCC2C1C 33853,O=C1NCCc2cc(F)c(N3CC4C5COCC5C4C3)cc21 33854,c1(CC)nc(C)ncc1C(=O)NCC1(F)CCN(C(=O)CCC2CCCO2)CC1 33855,N1(C(C2CC(C)OC2)=O)C(C)CC2CN(C(C3CC(N(C)C)C3)=O)CC12 33856,N1(C(c2ccc(CCCCC)o2)=O)CC2C(C(=O)NC(C)C)C2C1 33857,C1(NC(C23C(C)(C)C(CC2)CC3)=O)CCCC2CN(C(c3cc(Br)co3)=O)CC12 33858,C1(CC)CN(CCNc2ccc3c(c2)O3)C(C)CO1.c1(OC)ccccc1C 33859,Cc1nccc(C(=O)NCCCN(C)C(C2CNC(=O)N2C)=O)n1 33860,N1(C(COCCOC)=O)C(C(=O)N(CCCC(=O)OC)C)CCC12CC2 33861,C(=O)(CCCC(=O)N1CCOCC(CNC(=O)C(C)CC(F)F)C1)OCC 33862,C1(O)(C(N2CC(O)(CCNC(C3(C)CCC(C)C3)=O)C2)=O)CCCC(C)(C)C1 33863,CC(C)C(C)C(CNC(c1cnc[nH]1)=O)NC(C1CSC1)=O 33864,CC1OC(C)(C)OC1(C)C(=O)NC12CC(NC(c3c[nH]cc(F)c3=O)=O)(C1)C2 33865,C(CC(N)=O)(C(=O)NCC1CC1(F)F)NC(CN(C(C(C)C)=O)C)=O 33866,Cc1cc(Cl)c(C(=O)N(C(C)(C)NC(c2cc(F)ccc2C)=O)CCO)cc1F 33867,C#CCC(C)(C(=O)NC1CN(C)CC12CC2)NC(=O)CSCC(F)F 33868,c1(CNC2C(C(=O)Nc3ccc(OC)c(O)c3)C2)cnc2ccc(Br)cn12 33869,c12ccc(cc1)oc2=O.C(=O)(C(C)=NOCC#N)N1C(c2c(C)ccs2)CCC1 33870,N1(C(C2=NOC(C)C2)=O)CCC2(CC1)CN(C(c1cn(C)cc1C(F)(F)F)=O)C2 33871,c1(NCc2c(OCC)cccc2)[nH]c(=NC(COC)C(C)C)nc2c1cnn2C 33872,N1(C(=O)CCCn2cccc2)CCOC(c2ncc[nH]2)C1.c12ocnc1c(=O)[nH]o2 33873,c1(OCC)ccc(C(=O)NCC2(CNC(C3(C)CC3(C)C)=O)CCCC2)cn1 33874,c1(C(=O)NC(CC)CNC(C2CC3(CCC3)C2)=O)ccc(F)c(C)c1O 33875,CC(C)CC(C)CC(=O)NC(CNC(=O)Cn1cc(CN(C)C)nn1)CC(C)C 33876,c1(C(N2CCCC(CNC(C3(OC)CCC3)=O)C2)=O)cc(=N)[nH]c(Cl)n1 33877,C=CCC(CC(=O)NCCC1CC(OC)C1)NC(=O)C(N1CCNC1=O)C 33878,C(=O)(C#CC1CC1)N1C(C(=O)NCCN2CCC(CO)C2)C(O)CC1 33879,N1(C(CN(C)C)=O)Cc2ccccc2C(NC(C23CCC(CO)(CC2)CC3)=O)C1 33880,N1(C(C(CC)n2ccnc2)=O)CCN(C)C(CNC(=O)CCc2cncs2)C1 33881,Cc1nc(N2CCC(NC(c3n[nH]cc3C3C4CC5C(C4)C35)=O)C2)sc1C 33882,C1(C(=O)NCc2sccc2Cl)CC(F)(F)CN1C(c1ccccc1O)=O 33883,Cc1c(NCc2cscc2Cl)ncnc1N1C2C=CCC1CC2 33884,C1(C)(NC(C)=O)CN(c2ncccn2)C1 33885,N#CCCCC(=O)NC1C=CCC(C(N2CCN(C3CCC3)CC2)=O)C1 33886,C1(N(C(=O)CCN(CC(C)(C)C)C)CC)CCC(NC(=O)CC2CCOC2)CC1 33887,C1(CNC(=O)Cc2cccnc2)CC2(CO1)CN(C(=O)CCOC1COC1)C2 33888,CCC(CC(=O)N1CCN(C(=O)CCC(C)(C)OC)CC(O)C1)C(F)F 33889,C(=O)(N=S(C)(=O)C1CC(O)C1)c1nc(N(C2CCc3cncn3C2)C(C)=O)cs1 33890,C1(CN(C(=O)CC2(CO)CC2)C)COCCN1C(c1cc(-n2cccc2)ccn1)=O 33891,N1(C(=O)CN2CCCCC2)CC2(CCC2)CC1C(=O)NCC=Cc1cccnc1 33892,C1(OC)CC(CNC(=O)C(F)C(C)C)N(C(C2CC(F)C(=O)N2)=O)C1 33893,C1(NC(CNC(=O)CC2CCCC2)=O)CCCCN(C(c2ncsc2Br)=O)C1 33894,CC(C)C(C)(C)CNC(c1conc1C(C)NC(c1ncc(F)cn1)=O)=O 33895,Cc1cc(C(=O)NC2CCN(C(c3coc(N(C)C)n3)=O)CC2F)cc(F)c1C 33896,c1(OC)cccc2c1CC(C(N1CC(N(C(=O)CCSCC(F)F)C)C1)=O)CO2 33897,c1(C(=O)NCC(CNC(c2c(C)nc(COC)s2)=O)(C)C)ccc(OC)cc1Cl 33898,C1(NC(C(C(=O)OC)OC)=O)CC2CN(C(c3ccc(CO)nc3)=O)CC2C1 33899,CC(CC(=O)NCCN(C)C(c1cnc2sccc2c1)=O)P(C)(C)=O 33900,N1(C(CC)=O)CCC(C2CCN(C(c3cc(F)c(Br)c(F)c3)=O)C2)CC1 33901,C(=O)(C(C)S(N)(=O)=O)N(CCOC1CCN(C(C=Cc2ccc(C)o2)=O)C1)C1CC1 33902,c1(-c2c(SC3(C(=O)OC)CCC3)ncnc2)ccccc1S(=O)(=O)NC 33903,C(C(C)CC(=O)N1CC2C(CNC(c3ccncc3SC(C)C)=O)C2C1)OC 33904,C1(CS(=O)(=O)NCC2CC(OCC(F)(F)F)C2)CC2C(C1)C2(F)F 33905,C(=O)(C1CCc2scnc21)N1CC(CNC(C(c2ccn(C)c2)C)=O)C2(C1)CC2 33906,N1(C(COC)=O)CCc2nc(CNC(C3CCC4C(C3)C4(F)F)=O)sc2C1 33907,C1(NC(c2n(C)ncc2)=O)CC2CC1CN2C(c1ccncc1F)=O 33908,c1(-n2c(CNC(c3n(CCCC)nnn3)C(C)C)nnn2)ccc(F)cc1 33909,c1(N2CCC(NC)CC2)cc(C)c(S(=O)(=O)NCC(C2CCCC2)OC)cn1 33910,N1(C(COCC=C)=O)CC(NC(C2CCCCC(=O)N2)=O)CC12CCOCC2 33911,N1(C(c2cc(OCC)n[nH]2)=O)CCC2(CCCN(C(=O)CC3(CO)CC3)C2)C1 33912,C1(NC(c2cc(C)c(F)cc2)=O)CCN(C(c2ccns2)=O)CC(O)C1 33913,C1(O)(CNC(C2C(C)CC2)=O)CCCN(C(c2ccc(F)c(C(F)F)c2)=O)C1 33914,c1(NC(N2C(C3(O)CN(C(=O)CC4CCCO4)C3)CCC2)=O)ccnc(Cl)c1 33915,C(=O)(C(C)(C)O)N(CC(C)(C)CC1CCOCC1)CCOCCOC 33916,c1(NCCC2(c3ccc(-c4cn(CCCC)nc4)cc3)CC2)c(C)cccc1F 33917,CC(C)CC(CC(C)C)C(=O)N(C)CC1CN(C(C2OCC2(C)C)=O)CC12CC2 33918,C1(NC(C=Cc2cc(OC)ns2)=O)CC2CCC(C1)N2C(C)=O 33919,c1(C(N2CCC(COC)(CNC(=O)C(F)CC3CC3)C2)=O)cn2c(n1)CCC2 33920,CC(C)CCC(C)N=c1[nH]c(=NC2COC3(CCC3)C2)c2ccc(CO)cc2[nH]1 33921,CP(C)(=O)C(CC(=O)NC1CC1NC(c1ccncn1)=O)c1ccccc1 33922,N1(C(c2n(C)c(=O)ccc2)=O)CCCC(C2CCN(C(C3CNC(=O)C3)=O)C2)C1 33923,C1(NC(Cn2c(C(C)C)nnn2)=O)CCC(N(C)C(C23CCCC2C3)=O)CC1 33924,c1(C(=O)NC2CCN(C(c3ccc([N+](=O)[O-])[nH]3)=O)C2)csc2c(Cl)cccc12 33925,C12(CNC(C3CCCC(NC(c4nc(C(C)C)oc4)=O)C3)=O)CCC(CC1)OC2 33926,c1(CC(C)C)ccc2cc(C(=O)NC3CCNCC3)[nH]c2c1 33927,c1(C(=O)NC2CCCCN(C(C(C3CC(F)(F)C3)OC)=O)C2)cc2c([nH]1)CCOC2 33928,N1(Cc2ccc(OCCO)cc2)CCC2CN(c3ncc4sccc4n3)CCC12 33929,c1(C(=O)NC2CCN(C(c3c(OC)ccs3)=O)C2)ccc(C2CC2)c(OC)c1 33930,N1(C(=O)CC2CCC2)CC2(CCN(C(C3(CC4CC4)CCCO3)=O)CC2)C1 33931,C1(CNC(CN(C)S(N)(=O)=O)=O)CN(C(=O)Cc2ccsc2)CC1O 33932,C1(C(=O)NCCC2CC(C)(C)C2)CC1C1CN(C(=O)CNC(N)=O)C1 33933,C(CO)(CCF)NC(CCN(C(=O)Cc1cc[nH]c1)C(C)C)=O 33934,CC1CCC=C1C(=O)N1CCN(C(CNC(=O)CCC2CCCC2)C(F)F)CC1 33935,c1(C(C(=O)NC2C3(CN(C(c4n(C)cnc4)=O)C3)CC2)O)cccc([N+](=O)[O-])c1 33936,Cc1csc(C(=O)NC2CN(C(=O)CCc3ccc[nH]3)CC2F)c1Cl 33937,c1(C(C)(C)C)cc(=NC2CCCC(NC(C3(C)CCCCCC3)=O)C2)[nH]c(Cl)n1 33938,N1(C(CCCC(C)=O)=O)CCN2C(=O)C(NC(c3ncn(C)c3C)=O)CC2C1 33939,CC(C)(C)C(C)(O)C(=O)N1CCCN(C(c2coc(C(F)(F)F)n2)=O)C(CO)C1 33940,c1(S)ccnc(OC)n1.C(=O)(C=CSC)N(CC=C)Cc1ccccc1.C12CCN1C2=O 33941,C1(C(N(CC)Cc2ccc(O)cc2)=O)CCCN(C(c2cnoc2C)=O)CC1 33942,c1(C(N(c2cnn(CCCC)c2C)C2CCOC2)=O)cc([N+](=O)[O-])ccc1Cl 33943,C1(C(N(CC)Cc2cccnc2)=O)C(C)C=CC2C(=O)N(C)C(=O)C12 33944,C1(CNC(c2c(C)cc(O)nn2)=O)CN(C(c2ccc(F)cn2)=O)CCC1(F)F 33945,CC1(C)CN(C(=O)OCCOC(c2ccccc2)=O)CCC1C(=O)NCCCN 33946,C1(CNC(c2c(C)scn2)=O)CC(NC(c2sccc2CC#N)=O)C1(C)C 33947,c1(OCC)cc(NC(=O)C(C)NC(C)(C)C)c(Br)cc1Br 33948,C(c1cccc(F)c1F)=CC(=O)NC1CCCC(CNC(C(C)O)=O)C1 33949,CCC(C(C)C)C(C(=O)NCc1ccccc1Br)N1CCC(CCCO)CC1 33950,C1(C(=O)NCC(C)(CO)NC(c2ccc(NC)cn2)=O)CC(=O)N(OC)C1 33951,C1(CC)CN(C(=O)C(F)OC(F)(F)F)CC1C(=O)N(C)Cc1ccc(F)cc1 33952,Cc1ccc2c(C(=O)NCCCN(C(C3SCCCS3)=O)C3CC3)c[nH]c2c1 33953,N1(C(CNC(C)=O)=O)CCN(CCN(C)C(C2CC2Cl)=O)CC1 33954,C1(NC(N(C)C)=O)CC(CNC(c2coc(N(C)C)n2)=O)C12CCC2 33955,N1(C(Cc2cccc(C)c2)=O)CCN(C(=O)Cc2ccccc2F)CC(CO)C1 33956,C1(NC(CC2CC(OCC)C2)=O)CCN(C(=O)CSc2ccc(C)nc2)CC1F 33957,N1(C(C(C)NC(N)=O)=O)Cc2ccccc2C1C(=O)Nc1nn[nH]n1 33958,c1(SC)nc(N2CCN(C(C3CC=C(C)CC3)=O)CC2)c(Br)c(C)n1 33959,c1(NC(c2n(CCC)nnn2)c2ncc[nH]2)cccc(CSCC)c1C 33960,c1(OC)ccc(CC(=O)NC2CC(NC(c3csnn3)=O)C23CCC3)c(F)c1 33961,c1(C(N2CCN(C(CN3C(=O)CCCC3)=O)CC2)=O)cc2cc(Cl)cnc2[nH]1 33962,C1(C(=O)NC(COC)C)CC(O)CN1C(=O)CN1CCOCC1 33963,n1(CC(N2CCC(NC(C(C)=O)=O)C(C)C2)=O)[nH]cc2c(=O)ncnc1-2 33964,N1(C(CN(CCC)C)=O)CC2CCCC2(C(=O)NC2(CC3CC3)CCC2)C1 33965,C1(C(=O)NC2CN(C(C3(SC)CC3)=O)CC2CC2CC2)CC(C)(C)OC1(C)C 33966,N1(S(=O)(=O)c2cccc(Br)c2)CCC2(CCCC2N2CCNCC(F)(F)C2)CC1 33967,C1(CN(C)C(c2cnn(CCO)c2)=O)CCCN(C(c2[nH]nnc2C(F)F)=O)C1 33968,N1(C(CC(C)C(F)F)=O)CC2(CCN(C(=O)C=Cc3ccn(C)c3)C2)C1 33969,C1(CCOC)(NC(c2ccon2)=O)CCN(C(C2CCOC2C)=O)C1 33970,C#CCCCC(C)C(=O)NC1CC(F)(CNC(c2cc(F)c(F)cc2F)=O)C1 33971,N1(C(CN(CC)Cc2ccccc2)=O)CCCCC1C(C)Nc1cnccn1 33972,C1(C(=O)OC)COC2(CCC2)CN1CCC(C)F 33973,N1(C(Cn2ncc(CC)c2)=O)CC2CCCC(C1)N2C(C1CC12CC(O)C2)=O 33974,N1(C(c2cccc(N)n2)=O)CC2CCN(C(C3CCN(S(C)(=O)=O)CC3)=O)C2C1 33975,C12(CNC(c3ccc(Cl)cn3)=O)CC1CN(C(c1cccc(=O)o1)=O)C2 33976,N1(C(C2(OCC)CCC2)=O)CC(NC(c2cnc(C3CCCO3)s2)=O)C2(CC2)C1 33977,N1(C(CC(CNC(c2ccc(Cl)o2)=O)O)=O)CC2(CCCC2)C1 33978,c1(C(=O)NC2CC(NC(CCCC)=O)C23CCC3)cc2cnc(Cl)cc2s1 33979,c1(N2CCC(NCc3cccc(C(C)C)n3)C2)ccc(S(=O)(=O)N(C)C)cn1 33980,c1(CCC)nc(=NCCCCC(C)NC(=O)C=C2CCCCCC2(F)F)s[nH]1 33981,c1(C(=O)NC2CCC(CNC(c3cc(C)oc3)=O)C2)ccc([N+](=O)[O-])n1C 33982,C12(NC(C(C)OCC=C)=O)CCCC1(F)CN(C(c1[nH]nc([N+](=O)[O-])c1Cl)=O)C2 33983,N1(C(c2c(COC)nn(C)c2)=O)CCC(C)C(NC(=O)COC(C)C)C1C 33984,c1(OC)cccc(C(N2CCC(N(C(=O)C=Cc3ccsc3)CCO)C2)=O)c1F 33985,C1(C(=O)NCC(C2CCCC2)NC(CCC#C)=O)CC2CCC(C1)C2F 33986,CC1CN(C(=O)CCCOC(C)(C)C)CCCN1C(=O)C(C)C#N 33987,C1(N(C)C)(C(=O)NCC(CNC(=O)C(F)=C2CCCC2)CO)CCCOC1 33988,C#CC1(C(=O)NCC2CSCCN2C(=O)CC2CCCCC23CC3)CCCCC1 33989,N1(C(C2(C)CCCCNC2=O)=O)CCOC2(CCN(C(=O)C(O)C(C)(C)C)C2)C1 33990,C=CC(C)(O)CC(=O)NCC(C(=O)NCc1sc(C)cc1C)OC 33991,c1(OCCC)ccc(Cl)cc1CC(N1CC2C(NC(=O)C3=C(Cl)CC3)C2C1)=O 33992,c1(CNC(NC(CC)CC)=NCC2CCOC2)cc(P(C)(C)=O)ccn1 33993,c1(OC)ccc(CNC(C(C)(C)OC)c2nnnn2CC(F)F)cc1C#N 33994,O=C1CCCC(CNC2COCCC2CC(=O)O)C1 33995,C1(CN(C2CC2)Cc2cccc(-n3cc(C(=O)O)nn3)c2)CC2(C1)CC(F)(F)C2 33996,c1(C(=O)NC2(CCNC(c3cn[nH]c3)=O)CC2)ccc(C2CCCCO2)cc1 33997,C1(C(N2C(C)CC(CNC(C(C)(C)NC(=O)OC)=O)C2)=O)Cc2cccnc2C1 33998,C(=O)(C(C(=O)Nc1cccc(CNC(=O)C(COC)OC)c1)C(C)C)OCC 33999,N1(C(C)=O)CCCC1CC(=O)N(CC(C)(C)CNC(C1(C(F)F)CCC1)=O)C 34000,C#Cc1ccc(CCC(=O)NC2CCN(C(c3cnn(C)c3)=O)C23CC3)cc1 34001,c1(C(=O)NCCNC(C(F)OC)=O)c(Cl)c([N+](=O)[O-])nn1C 34002,N1(C(C2CC23CCOC3)C(=O)NC(C)C)CCc2ccc(F)c(F)c2C1 34003,C1(C2CCN(C(c3cc(C)n(C4CC4)n3)=O)C2)(NC(CCOC)=O)CC1 34004,C1(NC(c2c(CC=C)cccc2)=O)CCCN(Cc2cn(C)nn2)C1C 34005,CCC1=NOC(C(=O)NC2CC2NC(c2cn(CCO)nn2)=O)C1 34006,C1(NC(c2ncn(CC)n2)=O)CN(C(c2sccc2CC#N)=O)CC1C 34007,CC(C)(N=[N+]=[N-])C(=O)NCc1occc1C(=O)NCc1ccccc1O 34008,CCCCC(C(=O)NC1CC2CC1CC2CO)NC(=O)CC1CC=CCN1C 34009,c1(OC)ncnc(Cl)c1NC(=O)CC1(Nc2ccc(C)cc2Cl)CCC1 34010,C1(CNC(CCC(=C)C)=O)CN(C(C2CC2C(=O)OC(C)(C)C)=O)CCC12CCC2 34011,C1(CNC(c2cc(C)cc(O)n2)=O)CC2CCC(C1)N2C(=O)CC(C)N(C)C 34012,Cc1ccc(Cl)c(C(=O)NC23CC2CN(C(c2ccc(C4CC4)nc2)=O)C3)c1 34013,CC1(C)OCCC1(O)C(=O)NC1CCC(CC(=O)NC2CC23CCC3)CC1 34014,c1(C(=O)NCC2C=CC(NC(c3c(C)csc3)=O)C2)nc(C)n(C)n1 34015,N1(C(c2nc(C)oc2C)=O)CCCC2(C1)C(NC(=O)C(C)NC(N)=O)CCN2C 34016,c1(C(=O)NC2(C)CN(C(C=CCOC)=O)C2)ccc(S(=O)CC#N)cc1 34017,CC1(NC(C2CN(C(c3cc(N)cc(F)c3)=O)CCO2)=O)CN2CCC1CC2 34018,c1(C2(C(N(C(=O)C(CCc3ccccc3)C3CC3)C)=O)CC2)cc(Cl)cc(Cl)c1 34019,C1(NC(C(C)OCCN(C)C)=O)CCSC12CN(C(=O)CCC1CCCO1)C2 34020,N1(C(=O)OC(C)(C)C)CC(C(=O)OCC#CCNS(C)(=O)=O)OC(C(F)(F)F)C1 34021,c1(C(C)NC(c2c(C)n(C)cn2)=O)ccc2c(c1)CN(C(=O)C(F)C(C)C)C2 34022,Cc1c(C(N2CCCC2C2CN(C(=O)COCC3CCOCC3)C2)=O)cnn1C 34023,c1(OC)cnnc(C(=O)NCC(O)CC(=O)NCCN(C)C)c1 34024,C1(NC(C2CCC3(CC2)CC3)=O)CCCN(C(c2cc(F)c[nH]2)=O)CC1F 34025,N1(C(CC=C)=O)CCCC2(C1)CN(C(=O)CC1OCCOC1(C)C)CCO2 34026,C(N=c1ccc(Sc2n(C3CCCC3)nnn2)c[nH]1)c1c(C)cccc1 34027,C1(C(=O)NCC(C(=O)N(CC(=O)NCCC)C)(C)C)CCOC(CC)C1 34028,c1(CC(=O)NCC2(CNC(CCOCCN(C)C)=O)CC2)nn(C)cc1Br 34029,Cc1nsc(C(=O)NCC2CCCN(C(=O)C(C)(C)C3CCC3)C2)c1N 34030,CCC(C)CCC(=O)NCc1ccc(C(N2CC(OCCF)C2)=O)s1 34031,CCC(CC(=O)Nc1cnn(CC2CC2)c1)N(C(=O)CC1(C)CC1)C 34032,C1(N(C(C(C)OCC)=O)C)CCCN(C(c2ccc(SCc3nccs3)cc2)=O)C1 34033,N1(C(c2c(C)n[nH]c2)=O)CC(NC(=O)CCc2nnc(C(C)C)o2)C2CC12 34034,C1(C(N(CC(C)(C)NC(=O)OC(C)(C)C)C)=O)CC(C2CC2)=NO1 34035,C=CC(C)(CC)NC(=O)CONC(c1c[nH]nc1C1CC1)=O 34036,N1(C(c2cnn(C)c2)C(=O)NC(C(=O)OC)CC(C)C)CCCC(C2CCC2)C1 34037,N1(C(CN(C(C)C)C)=O)CC2CCC(NC(c3cnn4ccncc34)=O)C2C1 34038,C1(N(C(=O)C(=O)NC2CC2)C)CCC2CCN(C(c3ccccc3CO)=O)C1C2 34039,c1(OCC)cncc(C(=O)NCCC2CN(C(=O)Cc3cc(Cl)cs3)C2)c1 34040,C1(C)(CNC(C2CC(CCC)C2)=O)CCN(C(=O)Cc2ncoc2C)CC1 34041,C(=O)(CS(=O)(=O)C(C)C)N1C(CNC(C=CC=CCC)=O)(COC)CCC1 34042,c1(NCC(C(C)C)(C)NC(C2COCCO2)=O)ncnc2scc(Br)c12 34043,C1(CN(C2CNCCC2C)CCC)CCC=CCC1 34044,Nc1nc(Cl)ccc1C(N1CC2CC2(CNC(=O)CCC2CC2(Cl)Cl)C1)=O 34045,N1(C(=O)Oc2ccc(Cl)cc2)CCC2COCCC12 34046,CCC(C)(C)C(C)OC(C1CCCN1C(=O)OC(C)(C)C)=O 34047,C#CC1(NC(C2CC(NC(c3csc(F)c3)=O)C23CCC3)=O)CCCCC1 34048,N1(C(c2cc(OCC)n[nH]2)=O)C2CCC(C2)C1CC(=O)NC(CO)C(C)(C)CO 34049,C1(O)(CNC(c2cc(-c3ccc(Cl)cc3)no2)=O)CCN(Cc2ccsc2Br)C1 34050,C1(C#N)(C(=O)NC(C(C)NC(c2cccnc2C(F)(F)F)=O)CO)CC1(C)C 34051,Cc1csc(Cl)c1C(=O)NCCCN1CCN(C(=O)CSc2ccncc2)CC1 34052,c1(Cn2cc(CNc3cc(C)cc(C)c3)nn2)ccc2c(c1F)OCCO2 34053,Cc1c(C(=O)NC2CC(NC(=O)CC(C)C3CCCO3)C2)cnc2ncnn12 34054,n1(CC(=O)NCC(CNC(CC(CC)OC)=O)C)cccc([N+](=O)[O-])c1=O 34055,c1(C(C(C)C)SCC)nc(CC(C)(C)C)nn1-c1ccc(Br)nc1 34056,O=C(C(c1cccs1)=Cc1cccs1)NCC1CCC(CO)O1 34057,C1(CC(=O)N(C(COC)C)C)CCN(C(=O)CC=C(Cl)Cl)C1(C)C 34058,C(=O)(C1=CCCCCC1)NC1CCCCCC1CNC(CCCC=C)C 34059,c1(-c2nn(CCOC)c(COC3CCCCC3C)n2)ccc2ccccc2n1 34060,N1(C(=O)C=CC(F)(F)F)CCC2CCCC12C(=O)NCc1ccc(O)nc1 34061,C(=O)(C(C)(C)CC(=O)NC1CN(C(=O)CCCOCCOC)CC1C)OCC 34062,N1(C(C2ON=C(C)C2)=O)CCC2C(C1)CN2C(=O)CCCN1C(=O)CCC1=O 34063,c1(C(=O)NC2C(C)CCN(C(=O)C=Cc3ccccc3)C2)cc2occc2n1C 34064,CC1C(NC(C2CCCCS2(=O)=O)=O)CCCN1CCC1CCCC1 34065,C1(C)(CC)C=C(C(=O)N2CC(NC(c3cc(C)ccc3OC)=O)C(C)C2)C1 34066,c1(C(=O)NCC2CCCN2C(C2CC(CF)C2)=O)cc2c(F)c(Cl)ccc2[nH]1 34067,c1(C(=O)NC(COC)CNC(c2cnnn2C2CC2)=O)cnc(Cl)n1C 34068,c1(CS(N)(=O)=O)ccccc1C(=O)NCCCN(CC(=O)O)C1CC1 34069,N1(C(C2CCN(c3n(C)ccn3)C2)=O)CC2(CCN(C(C3CC3(C)C)=O)CC2)C1 34070,C(=O)(CCCS(=O)(=O)C(=O)NC1(c2nc(C)no2)CC1)OC 34071,C1(NC(COCCCCCC)=O)CCC2(CC1)CN(C(=O)Cc1conc1C)C2 34072,C1(CC(=O)NC(c2cc(C(N3CC(NC(C)=O)C3)=O)n[nH]2)OC)CCCCN1C 34073,C1(F)(C(=O)OC)CCN(C(=O)COC)C1.c12ccc(cc1)OC(=O)N2 34074,N1(C(C2(SC)CN(C(=O)CN3CC4CC4C3)C2)=O)CCc2oc(C)nc2C1 34075,c1(C(=O)NCC(C)NC(=O)C(c2ccccc2F)C)cccc(N)c1Br 34076,C1(NC(=O)NCc2ccc(S(C)=O)cc2)CCC(F)(F)C(C)(C)O1 34077,c1(C(=O)NCC(CCOC)NC(C2(COC)CCOC2)=O)oc(C(C)C)nc1C 34078,CC1CCCCN1CCC(=O)NCC1CC1NC(c1ccc(CC(N)=O)cc1)=O 34079,C(=O)(C(CC(C)C)NC)N1C(C(N2CCCC(CCC=C)C2)=O)(C(C)C)CCC1 34080,N1(C(Cc2ccn(CC)n2)=O)CCCCCC1CNC(=O)C(C)(CC)CO 34081,C(=O)(C1OCCc2ccccc21)N(CCCOCC(F)(F)F)C(C)C 34082,N1(C(c2ccn(CCC)c2)C(=O)NC(C)C(=O)OC)CC(CO)C1(C)C 34083,c1(C(=O)NC(C)CCNC(C2(C)CC3CC3C2)=O)c(F)cccc1F 34084,N1(C(C(CCOC)C)=O)CC(N(C)C(c2cc3n(n2)CCC3)=O)C(C)(C)C1 34085,c1(CC(=O)NCCNC(C2CCS2(=O)=O)=O)noc2ccc(Br)cc12 34086,N1(C(C2N(C)CCN(C(CCCOCCC)=O)C2)=O)CCCC(C)(C)CC1 34087,C(CC(C)(C)C#N)(C(=O)NC)S(C)(=O)=O.N12CCC(CC1)CC2=O 34088,Cc1c(C(=O)NCC2CCCCC2NC(C2CC2CC2CC2)=O)cnn1C1CC1 34089,c1(Cc2cc(C3CC3)on2)nc(CCn2ccnc2)nn1Cc1ccccc1 34090,C1(C(=O)Nc2c(C)cccc2CO)CCN(C(=O)CNC(=O)C2CC2)C12CCC2 34091,C(=O)(C(CC)C(C)(C)CC)NCC(CC=C)NC(=O)COC1CC=CC1 34092,C1(C(N2CCCC(Cn3cc(C(CC)O)nn3)C2)=O)CCc2nc(O)[nH]c2C1 34093,c1(N(CCCC)C)ccc(C(F)(F)F)cc1S(=O)(=O)N1CCCC2CC2C1 34094,CC(C)C(C)C(C)CC(=O)NC(C)CC1CCN(C(=O)Cn2cnc(=N)[nH]2)CC1 34095,N1(C(CCC(N)=O)=O)CC(CNC(=O)CC(O)Cc2ccccc2)C2(CCC2)C1 34096,C1(NC(C(COCC)(C)C)=O)COC2CN(C(=O)C(F)C(C)(F)F)CC12 34097,C(=O)(C1CC(=O)c2ccccc21)N1C(C)(CNC(C(C)NC(N)=O)=O)CCC1 34098,Cc1cc(C(=O)N(C2CN(C(C3(C)CCCCCC3)=O)CC2(C)C)C)nc(C)c1 34099,C=CC(C)(CC)C(=O)N(CCCNC(=O)CNC(=O)COc1ccc(F)cc1)C 34100,Cc1cncc(C(=O)NC2CCCC2NC(=O)CCF)c1Cl 34101,c1(C(=O)NC(C)(CNC(=O)CC2CC=CCC2)CO)cc(Cl)ccc1O 34102,C1(C(=O)NCC(n2ccnn2)C)CN(C(=O)CN2CSCC2=O)CC(C)(C)C1 34103,Cc1oc(Cl)nc1C(=O)NC1(CCCC(=O)NC2CC(C(F)F)C2)CCC1 34104,CC1CC(NC(=O)C(C)S(N)(=O)=O)CN(C(=O)C(C)(C)F)C1 34105,N1(C(=O)Cc2c[nH]nc2O)CCC2CCN(C(c3ccc(Cl)cc3O)=O)CC2C1 34106,N1(C(c2c(C)[nH]cc2)=O)CC(NC(C2CCC(N(C)C)CC2)=O)C2CC12 34107,C1(NC(C2CCC3CC23)=O)CN(C(c2cnc(Br)s2)=O)CC12CC2 34108,C1(NC(=O)COC2CCOC2)CC(F)CN(C(c2c[nH]nc2C(F)(F)F)=O)C1 34109,C1(NC(C2(P(C)(C)=O)CC2)=O)CN(C(c2cocn2)=O)C2(CCCOC2)C1 34110,C(=O)(CCC(=O)NCC1(CNC(C2CC2C(F)F)=O)CC1)c1cn(C(C)C)nc1 34111,CC(C)CC(C)(O)C(=O)NCC(C1CC1)NC(c1ccn2ccnc2c1)=O 34112,C(=O)(C(C)(C)Cc1cnn[nH]1)N1CC(CNC(c2cc(COC)[nH]n2)=O)(OC)C1 34113,c1(CNC(C2(C)CCN(C(c3cc(C(C)=O)cn3C)=O)C2)=O)ccn(C)c(=O)c1 34114,CC1=CC(O)CN(C(=O)N(C)C)C1.c12nc(cs1)C(C)C(=O)N2 34115,C1(CNC(=O)CN2CCOCC2)CC(F)(F)CN1Cc1ncc(Cl)cn1 34116,c1(C(=O)NC2CCCN(c3n(CCOC)ncc3)C2=O)cc2ccc(Cl)cn2n1 34117,c1(CC)ncc(C(=O)NC(CO)C(C)NC(c2ccncc2C)=O)c(O)n1 34118,Cc1cc(C(=O)NC2CCCC23CN(C(=O)C(F)C(F)(F)F)C3)cc(N)c1Cl 34119,C1(NC(c2cc(-c3ccccc3)c[nH]2)=O)CCCC1NC(C1CC(O)C1)=O 34120,C(=O)(C(F)C(C)(C)O)N1CCC(CC(C)NC(C2(COC)CC=CCC2)=O)CC1 34121,c1(OC)cc(C2CCN(C(=O)C=CC(C)C)CC2)cnc1NC(=O)OC(C)(C)C 34122,C1(C(=O)NCCN(C(=O)C(C)N2CCC2)CC)CCC(NC(N)=O)CC1 34123,c1(CC)noc(C(=O)N(C2CCN(C(C3CC(OC)C3)=O)CC2)C)c1C 34124,c1(C(=O)NCC(C)CNC(=O)Cc2cccc(F)c2O)cnc2c(c1)nnn2C 34125,c1(CN(C(=O)C(c2cccc(OC)c2)OC)CCC)cn(C2CC2)nc1C 34126,CCC(O)C(C)(C)C(=O)N1CCN(C(=O)C(C)(Cl)Cl)CC(O)C1 34127,c1(C(=O)NC2C(C(=O)NC(CC=C)C(=O)OCC)CC2)cc(C)nc(O)n1 34128,c1(COC(c2cccc(COCc3ccccc3)c2)=O)cc(CCO)cc(Br)c1 34129,Cc1ccsc1C(N1CCCC1CCCNC(=O)C(C)CN(C)C)=O 34130,C1(CNC(C(N2CCC(O)(C(=O)NC)CC2)=O)=O)CC(CC(=O)CC(C)(C)O)O1 34131,N1(C(C(C=C)(C)CC)=O)CCCCC12CN(C(C1CC3C=CC1C3)=O)C2 34132,O=C(C1Cc2ccccc21)N1CCC(N2CCN(C(C3(CO)COC3)=O)CC2)C1 34133,N#CC1(C(=O)NCCCOCCNC(C2CC2C2CC2)=O)CCSCC1 34134,N1(C(CCCOC(C)C)=O)CCC(NC(=O)CC2CCCN(C)C2)CC1C 34135,N1(C(C(CSC)OC)=O)CC(O)CC1C(=O)NC1CC=CCC1C 34136,c1(C(N2CCC(Cn3cccc3)CC2)C(=O)NCC=C)nn(C(C)C)nc1Br 34137,Cc1ccc(OCC(=O)NCC2CC(NC(=O)CC3(O)CCC3)C(O)C2)c(C)c1 34138,N1(C(C2(CNC(=O)CC(C)(C)O)CC(=C)C2)=O)CCCCC(C)C1 34139,C1(C)(C(N2CC(NC(c3c(C)occ3C(F)(F)F)=O)C2)=O)OC(C)(C)OC1C 34140,C(=O)(C1CSc2ccccc21)NCCC1(C)CCN(C(C2CC(O)C2)=O)C1 34141,C1(CNC(CCCC#CC)=O)CC12CCN(C(C1CC3CCC(C1)N3C)=O)CC2 34142,C1(C(N2CC(C3CN(C(C(C(=O)OCC)F)=O)C3)C2)=O)CCc2cn(C)nc2C1 34143,N1(C(CC(COC)(C)O)=O)CCCC2(NC(=O)C=CS(C)(=O)=O)CCCC12 34144,N1(C(c2cnc(C3CCC3)o2)=O)CCN(C(c2cnn3c2OCC3)=O)C(CO)C1 34145,c1(SC)ncc(C(=O)NC2CC3CN(C(c4ocnc4C4CC4)=O)CC23)c(O)n1 34146,CC1(C)CCCC(C(N2CC3(CC(CNC(=O)Cc4cn[nH]c4)C3)C2)=O)C1 34147,C(C(=O)NCC1CC(NC(=O)Cc2ccc(OC)cc2)CCO1)(C(C)C)OCC 34148,c1(C(=O)NCC(=CC(=O)NC(CC=C)CO)C)n[nH]c(C)c1Cl 34149,C1(NC(c2coc(C(F)F)c2)=O)(CF)CCN(C(c2cncnc2)=O)C1 34150,C(C1=NCC(O)CN1)N(c1ccccc1)Cc1c(OCC)cccc1 34151,C1(CCNC(C(C)(C)OC)=O)CN(C(=O)C(C)NC(c2ccoc2)=O)CC1C 34152,N1(C(C2C(C)OCCO2)=O)CCCC(C)(NC(=O)C=CC(=O)OC(C)(C)C)C1 34153,CC1CC(NC(=O)CC(C)(C)F)CN(C(=O)CC2CCC(=O)CC2)C1 34154,c1(C(=O)NCC2CCN(C(C(CCOC)OC)=O)C2)cnn2c1CCC2 34155,c1(NC(C2CC3CC3N2C(=O)CCN2CCOCC2)=O)cccc(C(F)(F)F)c1 34156,N1(C(CC=C=C)=O)CC2CC1C2NC(c1ccccc1)=O 34157,N1(C(c2n(COC)ncc2)=O)CCCC1(C)CCC(=O)NCC(C)COC 34158,c1(CNC(CCCOC)=O)nnn(C)c1C(=O)NC1C=CCCCC1 34159,C1(c2nnnn2C)(NC(CCN(c2ccccc2)C)=O)CCCN(C(CF)CF)C1 34160,c12ncccc1-c1cn(nn1)CC1CCCN1C2=O.C1(C(=O)OC)C2CCCC12 34161,C1(CNC(c2c(C)nsc2)=O)C2CN(CC(=O)NCc3ccco3)CC12 34162,CCC(CCOC)C(=O)N1CCC(CN(C)C(C2COC(=O)N2C)=O)C1 34163,C(=O)(C(C)(C)CC(F)(F)F)N(CCNC(C(CCC)N(C)C)=O)CCC 34164,N1(C(C(c2cccc(Cl)c2)C)=O)CCN(C(c2ccc(Cl)cc2N)=O)CC1C 34165,c1(C(=O)NCC2N(C(c3c(CC)nns3)=O)CC(O)C2)cnc(C)cc1Cl 34166,C1(C(=O)NC)COCCN1C(c1cccc(-c2cc[nH]n2)c1)=O 34167,c1(C(=O)NCCC2(O)CCN(C(C3(CC#C)CCCO3)=O)C2)cccc(=S)n1O 34168,c1(C(N(C2CN(C(c3ccc(C)nc3C3CC3)=O)C2)C)=O)cc(F)c(F)cc1C 34169,c1(C(=O)NC(C2(O)CN(C(C(CC)N(C)C)=O)C2)C)cc2nccnc2cc1C 34170,C=Cc1cncc(C(=O)NC(C2CCOC2)CNC(c2c(C)cnnc2O)=O)c1 34171,N1(C(C(C2CCN(C(c3cnn(C4CC4)c3)C)C2)F)=O)CCC2(COC(C)C2)C1 34172,c1(C(=O)NCC2CCN(C(CN(C(COC)=O)C)=O)CC2)ccc(Cl)cc1Cl 34173,C1(NC(C2CCC=CO2)=O)CN(C(=O)COc2ccon2)CC12CCOCC2 34174,c1(OC)c(F)ccc(F)c1C(=O)NCC1CCC2(CCC2)C1NC(=O)C1=CCC1 34175,C1(NC(C2(C)CCN2C(=O)C(CN)c2ccccc2)=O)CCc2n[nH]cc2C1 34176,c1(CN2CC(C)CC(NC(CC=CCC)=O)C2)coc2ccccc12 34177,C(=O)(C(F)(CNC(C1(C#N)CCCOC1)=O)C(C)C)NC(C(=O)N(CC)CC)C 34178,N1(C(c2c(C)con2)=O)CC(NC(c2cccc3cnsc23)=O)C2(CCC2)C1 34179,C(C(CC(C)C)C(=O)Nc1cnc(C)c(C#N)c1)NC(C1(OC)CCC(C)C1)=O 34180,N1(c2nc(C)nc(O)c2C)CCC2(CC1)OCCC2NC(C1CNC(=O)N1)=O 34181,c1(CN2CC(OC)C(NC(=O)CNC(=O)CC(C)C)CC2)ccc2nc[nH]c2c1 34182,C1(CNC(c2scnc2Cl)=O)CCCC1NC(=O)C(Cc1ccccc1)C1CC1 34183,N1(C(c2nnc(C)s2)=O)CCN2CCOCC2(CNC(=O)C(C)CCC(C)C)C1 34184,CC(C)CCC(C)N(C(=O)CCCOc1cccnc1)C 34185,Cc1cc(C(N2CCCC(N(C(=O)C(C)CC3CC3)C)C2)=O)ncc1Cl 34186,CC1OC(=O)NC1C(=O)NCC1(CNC(=O)CCC2CCCCC2)CC1 34187,c1(SC)cc(NC2CCN(C(=O)C(C(C)C)C3CCC3)CC2C)nc(SC)n1 34188,N1(C(C2CCC(=C)CC2)=O)CCC2CCN(C(c3cc4sc(Cl)cc4[nH]3)=O)CC12 34189,Cc1noc(C)c1C(C)C(=O)NCCC(C)NC(=O)C(C)C1CCCO1 34190,c1(N(C(C2C(NC(=O)C=CCN3CCCCC3)C2)=O)CCCl)cnncc1Cl 34191,N1(C(C2N(C(C3C(C)CCCC3)=O)CCCC2(C)C)=O)CC23CCC2(COC3)C1 34192,c1(C(=O)NCCC(C)N(C(C(c2cncnc2)C)=O)C)cnc2cnn(C)c2c1 34193,CC(N=c1ccnc(N2CCc3nn(C)cc3C2)[nH]1)c1ccc(Br)o1 34194,Cc1ccc2nc(CNC(=O)NC3COCCN(CC(F)(F)C(F)F)C3)cn2c1 34195,C(=O)(CC(CNC(=O)CC1CSC1)C1CCC1)NC1(CN(C)C)CC1 34196,C1(O)(C(NOC)=O)CCCN(CC(C)OC)CC1 34197,N1(C(Cc2c(C)noc2)=O)CCC2C1CCCN2C(C1CCCCO1)=O 34198,C(CC(O)C(=O)NC1(c2ccccc2)CN(C(c2cc(C)on2)=O)C1)OC 34199,c1(C(C(=O)Nc2ccccc2)N(CCC(=O)OCC)C)nc(Cl)sc1Cl 34200,C=CC(CC)C(=O)NCC1(C(=O)NCC2CC2Cl)CCC1 34201,C(CC(C(=O)NC(CCO)c1ccco1)NC(C1CN(C(C)=O)C1)=O)SC 34202,S(=O)(=O)(c1ccc2c(c1)CCN2CC)NC(CCCC)C(=O)NC 34203,c1(SC(F)F)cccc(-c2cncc(CNCc3ncccc3Br)c2)c1 34204,c1(C(=O)NCC2N(C(C=NOC)=O)CCC2)cccc(C#N)c1 34205,N1(C(C(C)O)=O)CCC(C2CC(NC(=O)CCc3ccn(C)n3)C2)CC1 34206,N1(C(c2c(C)nc(C)o2)=O)CC2CCN(C(=O)CC3CCCNC3=O)CC12 34207,c1(C(=O)NCCN(C(c2c(C)ccc(C)c2)=O)C)nc2ccccc2cc1CO 34208,C(=O)(C(C)(C)S(C)(=O)=O)NC(C(C)NC(c1c(OC(C)C)cccc1)=O)C 34209,C(=O)(C1CCc2c[nH]nc21)NCC(C1CCCCC1)NC(C(=O)NC(C)C)=O 34210,C1(NC(C2(CC)CCOC2)=O)CCCCCC1NC(=O)CC1(CO)CC1 34211,C1(C)(COC)CCN(C(C2(NC(=O)CN3CCNC3=O)CC(F)(F)C2)=O)C1 34212,N1(C(COCCCC#C)=O)CCC(F)(F)C(CNC(c2sccc2COC)=O)C1 34213,C(N=c1cc2n([nH]1)CCCC2)(c1cccc(OC)c1)c1nnnn1CC(F)F 34214,C(=O)(C(C#N)C(C)C)N1CC(CNC(Cc2c(C)cnn2C)=O)C(O)C1 34215,C1(CC)CN(C(C2(CO)CCCC2)=O)CCN1C(c1csc(-c2cccs2)n1)=O 34216,N1(C(C(C=CC)O)=O)CC=C(C(C)(C)C(=O)NCC2CC(C3CC3)=NO2)C1 34217,C=CCC(CN1C(=O)C1C)OC.C1(CC(=O)NC2CC2)(NC(=O)NC)CCC1 34218,C1(OC)(CNC(c2cnoc2C)=O)CCN(C(=O)C2=COCCC2)CC1 34219,N1(C(c2c(SCC)cncc2)=O)C2CCC1C(CNC(=O)Cn1ccnc1C)C2 34220,N1(C(CC2C=CC(NC(=O)CC3CCCOCC3)C2)=O)CCC12CCSCC2 34221,c1(CC(=O)N(CC(C)C)CCN(c2ccccc2)C)ccccc1-c1nn[nH]n1 34222,C1(CNC(C=CC2N(C)CCC2)=O)CN(C)CCN1Cc1ccccc1 34223,C=CC1CN(C(=O)COCCC)CC1NC(=O)CCCc1ccccc1F 34224,c1(C(=O)NCCCNC(C2CC(P(C)(C)=O)C2)=O)n[nH]c2ccc([N+](=O)[O-])cc12 34225,N1(C(c2cn(CC(=O)N(C(C)(C)C)C3CC3)nc2I)=O)CC2(C)CC1CCO2 34226,N1(C(C2CCN(Cc3c(OC)ccc(Br)c3)CC2O)=O)CCC2(CC1)CN(C)C2 34227,NS(=O)(=O)c1ccc(C2(C(=O)NC3CCC3NC(C3(CO)CC3)=O)CCC2)cc1 34228,C1(CC(=O)OC(CC(C)N(C(=O)C(=O)NCC)C)OC)CC2(CCOCC2)CO1 34229,Cc1nccc(C(N2CCC(NC(c3cc(Cl)cnc3O)=O)C(C)C2)=O)c1C 34230,C1(C(=O)NCCC(C)N(C)C(c2cn(C)nn2)=O)CCC(C)(C)C1 34231,C1(NC(Cn2nc(C)n(C)c2=O)=O)CC12CCN(C(C1OCCC1(C)C)=O)CC2 34232,N1(C(c2cc(C)oc2C(F)(F)F)=O)CCN(C(c2cnc(O)o2)=O)CC(C)(F)C1 34233,Cc1cc(NC(=O)NC2(c3ccccc3)CCOC2)cnc1C 34234,CCC(C(=O)NCC(C)CN(C(=O)C1=NOC(C)C1)C)C(C)C 34235,c1(CCC(=O)NC(C2CCN(C(c3c(C)nn(C)c3)=O)C2)C)c(Cl)cccc1Cl 34236,CCCN=C(NCc1ccc(C(=O)OC(C)(C)C)c(Cl)c1)NCC.C12CCN1C2 34237,C1(C(N2CC3C(CN(C(=O)Cc4ccccc4)C)C3C2)=O)C2CCC3C(C2)CC13 34238,C1(NC(C(n2c(C)ncc2)C)=O)CN(C(=O)Cc2cnsc2)CC12CCC2 34239,C(=O)(C1=C(C)OCCS1(=O)=O)NC1CN(C(C(CC)CC(F)F)=O)CC1C 34240,c1(C(=O)NC2CC3(C2)CC3NC(c2ncccc2F)=O)cc(F)c2cn[nH]c2c1 34241,C1(CC)CCC(C(N2CCCC(CNC(c3nnn(C(C)(C)C)n3)=O)C2)=O)CC1 34242,C1(NC(c2c(C(C)C)scn2)=O)CN(C(c2c[nH]ccc2=O)=O)CC2(CCC2)C1 34243,C(C(C)C(=O)NC(C(=O)NC(C1CCOC1)CO)C1CCCC1)OC 34244,C1(C(N(c2ccccc2)CC=C)=O)CC12CCN(CC1CCCC(C#N)C1)CC2 34245,Cc1cc(Br)ccc1CC(=O)NC1CCC1NC(C1CCCCN1C)=O 34246,c1(SC(CC)C(=O)NC)ncc(Br)cc1OC1(n2cc(C3CC3)nn2)CCOCC1 34247,C1(C(=O)NCCCCC2CN(C(c3c(C)cc(C)[nH]3)=O)C2)CC12CCCOC2 34248,c1(OC)cc(C(=O)NC2CN(C(c3coc(C)n3)=O)C2)c(N)c(Br)c1 34249,C=CCC(C(=O)N1CC(C(=O)N(CCCN(C)C)CC)CC(C)C1)C(C)C 34250,C1(C(CC)=O)CCCC1OC(=O)CC 34251,Cc1nc2cc(C(N3CCCC(F)(F)CC3)=O)ccc2n1C(C)CO 34252,C1(C(N(CC(=O)NCC)C)=O)CCCN(C(=O)COC2CC2)CC1 34253,N1(C(CCC(=O)OCC)=O)CCC2(CCCN2C(=O)Cn2cc(C)cn2)C1 34254,CCCC(C(=O)NCCCOCCNC(C1CCc2nncn2C1)=O)S(N)(=O)=O 34255,N1(C(C(F)=CCC)=O)CCCC(NC(=O)COCC2CCCO2)C1C 34256,N1(C(c2nc(F)ccc2Cl)=O)CC(C2(N=c3[nH]nc(C4CC4)o3)CC2)C1 34257,C1(C(=O)NCC(C)CN(C)C(c2ncsc2C2CC2)=O)COC2(CCC2)C1 34258,C(=O)(C(CNC(=O)Cn1cccc1)CC(C)C)NC1CC(OC)C1(C)C 34259,N1(C(Cc2c(C)noc2C)=O)CCCC(F)(C(=O)NCc2cn(C)nc2C)C1 34260,N1(C(C(C(C)(C)O)F)=O)CC2OCCN(C(c3c[nH]c4nccc-4c3)=O)C2C1 34261,C1(C(F)(F)F)(C(=O)NC(CCNC(Cc2c(C)scc2)=O)C)CC2CCC1C2 34262,CC(C1OCCc2ccccc21)N(C)C(c1cncc(F)c1Cl)=O 34263,N1(C(CC2(C)N(C(c3cnc(CC)o3)=O)CC2)=O)CC(=O)NC(C)C1 34264,c1(C(=O)NCC(CC)NC(c2cc(F)cs2)=O)ccnn1C(F)F 34265,N1(C(C(C(C)(C)C)SC)=O)CCCC(C2CN(C(=O)CN3CCC3)C2)C1 34266,N1(C(c2c(CC)nn(C)c2)=O)CC2CC1CN(C(c1nocc1Cl)=O)C2 34267,Nc1cc(Cl)nc(Cl)c1C(N1C2CCC1C(NC(=O)CC1CC1)C2)=O 34268,C(CC(C)C(=O)NC(C1CN(C(=O)CCc2conc2C)C1)C)=CC 34269,CC1CN(C(C2CCCN2C=O)=O)CC1NC(C1(N(C)C)CCC1)=O 34270,CC1OCCC1(C)C(N1CCC(C(=O)NCC(C2CC(C)(C)C2)O)CC1)=O 34271,C1(NCc2nnc(-c3sccc3)o2)CCN(C2CCCCC2)C1=O 34272,C1(OC)CCCN(CC(=O)N(C2CCOCC2)C2(c3nncs3)CC2)CC1.CO 34273,c1(CSCC)ccccc1C(=O)NC(CNC(C1(C)CC=CC1)=O)CO 34274,c1(C(N(CC(C)NC(C(CNC(C)=O)(C)C)=O)C)=O)cc2sccc2cn1 34275,c1(NCCCCN(C)C2CC2)[nH]c(=NCC2(C3CC3)CCCO2)nc2sccc12 34276,c1(C(N(C(c2ccccc2)CNC(c2onc(C)n2)=O)C)=O)ccc(O)nn1 34277,c1(C(=O)NC2C(CNC(C(CC)CC3CCCC3)=O)CC2)ncc2ccccn12 34278,C(N=c1ccnc(C(C)C)[nH]1)c1c(NC(CN2CCN(CC)CC2)=O)cncc1 34279,c1(CN(C(C2CCCN(C(c3coc(C)n3)=O)C2)=O)CC)ccc(O)cc1 34280,N1(C(C#C)C)CCCN(C(=O)Nc2ccc(CC)c(C(F)(F)F)c2)CC1 34281,c1(OC)cc(NC(c2ccnn2C)c2nnnn2C2CCCC2)sn1 34282,N1(C(CC(C)(C)O)=O)CC2(CC(C(=O)Nc3ccc(F)c(F)c3)CO2)C1 34283,c1(C(=O)NCCCCC(C)NC(C2CCN2C(C)(C)C)=O)cccc(F)c1O 34284,C(=O)(CC(C)CC(F)(F)F)NC(C)CCN(C)C(c1cc2cc(Cl)ccn2n1)=O 34285,C1(CCNC(C(CC)C)=O)CCCCN1C(c1cccc(N2CCCC2=O)c1)=O 34286,N1(C(c2c(C)cccn2)=O)CC(C)CN(C(c2ccc(F)c(N)c2F)=O)C(C)C1 34287,N1(CC)CCCC(C)(CN(C(C2(C(F)(F)F)CC=CC2)=O)Cc2ccccc2)C1 34288,c1(C(C)C(=O)NC2CCC(NC(C3(F)CC3C)=O)CC2)ccc(S(N)(=O)=O)cc1 34289,c1(C(=O)NC2CN(C(C=NOC)=O)C3C2C3)ccc2c(c1)C=CS2(=O)=O 34290,C1(CNC(=O)CCCCCO)CN(C(c2cncc(F)n2)=O)CCC12CCOC2 34291,C1(NC(CCC=C)=O)CN(C(=O)COc2ccon2)CCC1C 34292,C(C(CO)(CO)NC(c1cccnc1)=O)N(C)C(C1CNC(=O)N1C)=O 34293,C(=O)(CCCCc1ccccc1OC)NC(CC)(C)C#N 34294,N1(C(CN(C)C2CC2)=O)CCCC(C)(C(=O)NC(C)(C)C(O)CO)C1 34295,c1(CC(=O)NC2CCCN(C(=O)CCN3CCCCC3)CC2)c(F)cncc1Cl 34296,C1(C(N(CC(C)NC(CCCNC(=O)OCC)=O)C)=O)CCc2nc(C)cn2C1 34297,C(=O)(C(C(CC)CC)OC(=O)C(c1cnn(CC)c1C)=O)N(CCC#N)CCC 34298,c1(C(=O)NC2C(NC(C=CCOC)=O)C2)cccc2oc(C)cc12 34299,c1(C(=O)NCC2CCC(NC(c3c(C)ocn3)=O)C2)cnc2c(c1)CCOC2 34300,C1(NC(C2C(NC(c3c(C)ccnc3C)=O)CCOC2)=O)CC(C2CCCC2)C1 34301,C1(c2ccc(Br)cc2)(NC(c2c(CC)nc(C)s2)=O)CCC(C)(C)C1 34302,C1(COC)(NC(=O)CCC=C(C)C)CCN(C(=O)C(c2ccccc2)SC)C1 34303,c1(C(=O)NC(C(C)(C)OC)C)ccc(CNC(=O)Cn2cc(C#N)cn2)nc1 34304,c1(C(N(CC(=O)OC)CC)=O)cnc(CNC(c2ccnn2CC)=O)nc1 34305,N1(C(C(C2SC(=N)NC2=O)C)=O)CC2OCCN(C(C3CN(C)CCO3)=O)C2C1 34306,C(c1cccc(C)c1)=CC(=O)NCC1(COC)CN(C(=O)C2=CCCC2C)C1 34307,N1(C(c2cc(COC)no2)=O)CCN(C(C2CCC(=O)O2)=O)CC2(CC2)C1 34308,C1(NC(C(CC)(C)CC)=O)CCN(C(C2CCC2)=O)CC(C)(C)C1 34309,N1(C(C2(Cl)C(C(C)=O)C2)=O)CC(C(=O)NC2CCCC2(C)C)C(F)(F)C1 34310,c1(COC)nn(C)cc1C(=O)Nc1cccc(-c2nc(C)co2)c1 34311,N1(C(c2nc(CC)oc2)=O)CCC(CC)C1CNC(=O)Cn1nnnc1C1CC1 34312,N1(C(C2CCOC2NC(=O)NC2CC2)=O)CCCOC(CC(N2CC(OC)C2)=O)C1 34313,N1(C(C2CC=CC2)=O)CCOC2(CCCN(c3ncc(Cl)cc3[N+](=O)[O-])C2)C1 34314,n1(CC(=O)NC2CC(NC(C3(C)C(C)OCC3)=O)C2)nc2c(n1)CCCC2 34315,c1(OC(C)C(=O)NC(C)(C)CO)cccc(C(F)(F)F)c1 34316,CCCCC(C)(F)C(=O)NCC(C)N(C(=O)CN1CCOCC1)C 34317,N1(C(CCN(C)CC)=O)CCC2C(NC(c3nn(CC)cc3Cl)=O)C2CC1 34318,N1(C(C(CC)N(CC)CC)=O)CC2CCC(CNC(=O)C=CSC)CC2C1 34319,C1(NC(c2ccc(SC(C)C)cc2)=O)CC2CC1CN2C(=O)CN(C)CCO 34320,c1(C(=O)NCC(CN(C(CNC(=O)NC)=O)C)O)ccc(-n2cncn2)c(F)c1 34321,N1(C(c2c(CC)n[nH]c2)=O)CC2CN(C(c3sccc3COC)=O)CC(C1)O2 34322,c1(C(N(CC(CC)NC(=O)CCNS(C)(=O)=O)CC)=O)cc(CC)cc(F)c1 34323,C(=O)(C1CCCc2n[nH]cc21)NC(c1cccc(OC)n1)C 34324,c1(CC(=O)NCC(CC)NC(=O)COc2ccsn2)csc(C(C)(C)C)n1 34325,CCCCC(CC)(c1nnnn1CCCCCC)NCC1CCCC(SCC)C1 34326,c1(C(=O)NCC2(NC(C3(CO)CCC3)=O)CCOC2)ccn2ccnc2n1 34327,c1(NC(C2(OC)CCN(C(C3CC4(CC4)CO3)=O)C2)=O)cc(C)cnc1C 34328,c1(C(N2C(CC)C(NC(c3cnn(C(C)(C)C)c3)=O)CC2)=O)ccc(=N)[nH]c1Cl 34329,N1(C(c2c(C)nc(CCCC)s2)=O)CCN(C(c2cnc(Cl)c(N)c2)=O)C2CC12 34330,C1(CNC(CC2CC(SC)C2)=O)CCCCC1NC(c1nnccc1C)=O 34331,N1(C(C(=O)NC(C)C)=O)CC2CC(NC(=O)CC3CC3)C1C2 34332,c1(C(=O)NCCC(=C)CNC(c2ncccc2C)=O)nn(C)nc1Br 34333,C1(CNC(c2n(CC)nc(C)c2)=O)CCCCN(C(C23CC(O)C2C3)=O)C1 34334,c1(CNC2C(NC(C(c3ccccc3)OC(C)=O)=O)COC2)ccncc1C 34335,C1(N2CCN(c3cc(NCC4CCC(C#C)C4)ncn3)CC2)CCCCN1N=O 34336,CC(C)CCCCCCC(=O)N1CCC2C(NC(=O)C(O)CN(C)C)C2C1 34337,c1(N2CC(C(=O)NC)OCC2)ccc(S(=O)(=O)NCc2csc(Br)n2)c(Cl)c1 34338,C=CC(F)(F)C(=O)N1CC(OC2CCN(C(=O)C(C)N(C)C)CC2)C1 34339,Cc1cc(Cl)cc(C)c1OCC(=O)NC(C)CCCNC(=O)CSc1cccs1 34340,CCC(C)CCC(=O)NCC(C)(CO)NC(C12CC(C)(C1)OC2C)=O 34341,C(=O)(NNC(=O)C(O)c1ccccc1)Nc1c(C)cccc1Cl 34342,C(=O)(C(CCSC)NCC(C)C)N1CC(=CCC)C1.c1(C=O)ccco1 34343,CCCCC(C)(c1nnnn1C)NCc1ccc(OC)nc1 34344,c1(CCn2cc(CC(C(N3CCC(=C)C3)=O)O)nn2)ccncc1OC 34345,N1(C(CSC)=O)CCN(CC2CCCN(C(=O)C(C)CF)C2)CC1 34346,CCC(CCC(=O)NCCCC(C)(C)C1CC1)NC(C1CC2C=CC1C2)=O 34347,C1(C(=O)NCC(C=C)(C)C)CN(C(=O)CCc2ccnn2C)CC1F 34348,N1(C(CC=C)=O)CC(C)(C)CCC1CNC(c1cccc(OCCOC)c1)=O 34349,c12noc(n1)C1CC21.c1(C(C)OCCOC)cc(-c2ccccc2)[nH]n1 34350,CN1CCOCC(NC(=O)CCOCCNC(=O)CC2CCCN(C)C2)C1 34351,c1(C(N2CC(NC(CCCOCC=C)=O)C(OC)C2)=O)cncc2n[nH]cc12 34352,C1(C(=O)NCC(C(C)C)NC(C=C(C)c2cccs2)=O)CCc2nncn2C1 34353,c1(C(N(CC(=O)N(C)CC2CCCN2C)CCOC)=O)nocc1Cl 34354,C1(OC)C2CCN(C(c3cncc(C)c3)=O)C2C1(C)C 34355,C1(NC(C)=O)CCN(C(C2CC(NC(c3ccns3)=O)C2)=O)C1 34356,C1(NC(c2cc(C)c(Br)o2)=O)(CO)CCCN(C(c2nonc2N)=O)C1 34357,c1(C(CNC(C(n2cc(CSC)nn2)C)=O)O)cccc(C#N)c1 34358,C12(C(=O)NC(C)C)CCN(C1)S(=O)(=O)C2 34359,c1(OC)cc(C)c(C(N2CCC(C)(CCNC(C3CCC(=O)N3)=O)C2)=O)c(C)c1 34360,C1(F)(C(N(CCNC(C2(N(C)C)CCCOC2)=O)C2CC2)=O)CC2(CCC2)C1 34361,Cc1ccc(C(=O)NCC2N(C(=O)Cc3cnc[nH]3)CCC2(C)C)c(C(C)C)n1 34362,N1(C(C2C(CCOC)C2)=O)CCC(C)(C)C1CC(N1CC(S(C)=O)C1)=O 34363,c1(C(N(CCCNC(=O)C=C(C)C)CC)=O)cc(F)c(F)c(O)c1F 34364,c1(C(=O)NC(C(=O)N(CC=C)CC)C2CCCO2)c[nH]c(=NC)s1 34365,c1(C(=O)NCC2(CC(=O)NCC(CCC)O)CC2)c(C)n[nH]c1C 34366,Cc1c(Cl)ccc(C(C)(C)C(=O)NC2(CNC(C3(C#N)CC3C)=O)CCC2)c1F 34367,S(=O)(=O)(CC(=O)N1CC(C(C)NC(=O)C(C)N2CCC2)C1)NCC 34368,N1(C(C(C(C)C)C)=O)CCC(CNC(c2ccccc2CO)=O)C(C)C1 34369,c1(CCC)c(C(=O)N(CCCOCCNC(=O)C=C2CCC2)C)cnn1C 34370,C(=O)(C(C)(CC)OC)NCC1C(C(=O)NCCC#CCC)C1(C)C 34371,C(=O)(C(O)CN(C)C)NCCN(C(C)C)C(c1csc(-c2ccccc2)n1)=O 34372,c1(CCC)cc(C(=O)NC(C)CC(C)NC(c2cccnc2F)=O)nn1C 34373,N1(C(c2scc(C(N)=O)c2)=O)CCC(C2CN(C(=O)CC3CCCCO3)C2)C1 34374,c1(C(=O)NCC(CN(C(CNS(NC)(=O)=O)=O)C)O)cnc(O)c(C)c1 34375,N1(CC(=O)Nc2c(C)cccc2)CCCN(C2CCN(C(=O)C(C)(C)Br)C2)CC1 34376,N1(C(c2cc(OC)n(C)n2)=O)CCN(C(C2CCNC2=O)=O)C(C2CCCC2)C1 34377,Cc1ccc(N2CCCC3(NC(C4CCCC(F)(F)C4)=O)CC3C2)c([N+](=O)[O-])c1 34378,c1(C(=O)NCC(CO)NC(c2n(CC)ncc2)=O)c(F)cc(C)cc1F 34379,CC(C)CC(F)(F)C(=O)N1CCN(C(c2c[nH]nc2[N+](=O)[O-])=O)CC1 34380,Cc1cnn(C)c1C(=O)N(C)CC1(CNC(C2COCC(C)O2)=O)CC1 34381,c1(C(N(C2CCN(C(c3cc(C)ns3)=O)C2)CCO)=O)nc(=O)n(C)[nH]1 34382,N1(CC(COCC(C)C)O)CCC(CNC(=O)C(F)Cc2ccccc2)C1(C)C 34383,c1(C(N(CC(=O)NC(C)C(O)C(C)C)CC)=O)ncnc(O)c1F 34384,Cc1ccc(O)c(C(=O)NC(C)(C)CN(C)C(C2CC2(C)C(C)C)=O)n1 34385,C1(N(C(c2nccc(C)n2)=O)C)CN(C(=O)C(O)C2CCCC2)CCC1C 34386,C1(CNC(=O)COC2CC2)CCC(CNC(c2csc(C(F)(F)F)c2)=O)CC1 34387,CC(C)CCCCCC(=O)NCC1CCN(C(C2CC(C)N(C)C2)=O)C1 34388,c1(C(=O)NCCC(C)N(C(CC2(CC)CCOCC2)=O)C)ccc2cnoc2c1 34389,CC(CN(C)C)CCC(=O)N1CCCC(C(=O)NCC2CC3OC2C2CC32)CC1 34390,C(N=c1nc(-c2ccccc2)[nH]s1)C1(C)CCN(C(C(CCSC)O)=O)C1 34391,c1(C(N(CCNC(C(c2cn(C)nc2)O)=O)C2CC2)=O)c(Cl)ccc2c1OCO2 34392,c1(CC)cc(C(=O)NCC(O)CN(C(=O)C(F)=C2CCC2)C)ccc1Br 34393,C1(CC(=O)NCC2COC(=O)C2)COCCN1C(c1ccc(CO)s1)=O 34394,c1(C(=O)NC(C2CN(C(c3ccc(C)n3C)=O)C2)C)n[nH]c2ccc(Br)cc12 34395,c1(C(=O)NC2(C3N(C(C(OC)OC)=O)CCC3)CC2)cc(C)cnc1F 34396,C12(C(=O)NCCNC(CC(CC)(C)C)=O)CCC(C)(C(=O)O1)C2(C)C 34397,C12(CCNC(c3cc(OCC)ncc3)=O)CCC1CN(C(=O)CC1CCOC1)C2 34398,c1(C(=O)NC(C2(O)CN(C(=O)Cc3cncs3)C2)C)cc([N+](=O)[O-])n(C)n1 34399,CC1(C)CC(C(=O)NC2CCCC(O)C2O)CCN1C(=O)C1=CCSC1 34400,N1(C(C(CC=C)NC(C)=O)=O)CC2CC(C(=O)NCCOC3CCCC3)(C2)C1 34401,CCC(CC(=O)NC12CC1CN(C(c1cocc1C)=O)C2)c1ccccc1 34402,c1(NCCC(C)NC(C2CCOC3(CCC3)C2)=O)cc(=O)n2ccccc2n1 34403,N1(C(CC(OCC)OCC)=O)CC(CNC(c2ncccc2F)=O)N2CCC1C2 34404,N1(C(C(=O)NCC=C)C2CC2)CCC(N(C)CCN(C)C)C1 34405,N1(C(c2cnc(COC)s2)=O)CCCC(CNC(=O)COCCCF)CC1 34406,C1(C2CCN(C)CC2)(C(=O)NC(CNC(C=Cc2cccc(C)c2)=O)CO)CC1 34407,C#CCCCCC(=O)NCCC.C1(=O)CCCC(=O)NCCC2CCN1C2 34408,Cc1cc(CC2CN(C(=O)C(=O)N)CC2C)ccc1F.OC 34409,c1(NC(C(Cc2cnc[nH]2)NC(c2[nH]cc(C)c2)=O)=O)cc(C)ccc1CO 34410,Cc1oc(CNC(c2ccn(C(C)C)n2)=O)nc1C(=O)NCCC1(C)CC1 34411,C1(C(=O)NCC2(C(=O)NC3(c4ncc(C)o4)CC3)CCC2)CCC2(CC2)C1 34412,N1(C(C2(C#C)CN(C(=O)C(O)C3CCCC3)C2)=O)CC(C(N)=O)CCC1C 34413,C(=O)(CS(=O)(=O)CCO)NC1C2CCN(C(CC3CCC(C)(C)CO3)=O)CC21 34414,c1(CN(C(C(=O)NC(CC)(C)C)c2ncco2)C)c(Br)ccc(C)c1F 34415,C(C(C)(C(C)C)NC(=O)C(N)=O)NC(C(c1cccnc1)OC)=O 34416,CC1CC(C)(C)CCC1NC(CCOC)(C)c1nnnn1C1CCC(F)(F)CC1 34417,O=CN1CCOCC1C(=O)NC1CN(C(=O)Cn2nc(O)ccc2=O)CC1F 34418,c1(OC)cc([N+](=O)[O-])ccc1CCN=C(NCC(O)CNC(N)=O)NCC(F)F 34419,c1(C(N(CC(CNC(COC)=O)O)C)=O)ccc(Oc2ccc(SC)cc2)cc1 34420,C12(C(=O)NCc3cn(C4CN(C(CSCC=C)=O)C4)nn3)CCCCC1C2 34421,c1(C(N2CC(C)C(NC(=O)CCC3CC3(Cl)Cl)C2)=O)csc2c(O)ccnc12 34422,N1(C(C(CC)C(C)C)=O)CC2CC(O)C1C2NC(=O)C=Cc1cscn1 34423,c1(CNC(C2(COC)CN(C(C3CC(C)(C)CO3)=O)C2)=O)ccc(F)cc1F 34424,N1(C(C2CC2C2CCCCC2)=O)CCC(C#C)(CNC2(C3CC3)OCCO2)CC1 34425,C1(C(=O)NCCC2CCCCC2)COCCN(CC2CCC(F)(F)C2)C1 34426,N1(C(CC(C)O)=O)CC2CCN(C(=O)C=CC3CCOCC3)CC12 34427,N1(C(C2(C)N(C(CN(C(=O)OC)C)=O)CC=C2)=O)CCC2(CC1)CC2 34428,C1(F)(CNC(CC2CC(C)C2)=O)CC(C(=O)OC(C)(C)C)C1 34429,Cn1nc(C(F)(F)F)c(CN2CC(F)CC2C#N)c1Cl.N12CCC(F)(CC1)C2=O 34430,CC(CNc1ccccc1)C(=O)NC1COCC1NC(C1(N(C)C)CC1)=O 34431,C#CCC(C)(C)C(=O)N1CCC(C)(CCNC(c2cncc(NCC)c2)=O)C1 34432,c1(OCC(=O)N(CC(C)O)CCNC(C2CCC(=O)O2)=O)ccc(Br)cn1 34433,c1(N2CCCC(C(C)NC(=O)C=CBr)C2)cc(Cl)nc(-c2ccccn2)n1 34434,N1(C(CC(CC)(C)C)=O)CCCN(C(c2cnccn2)=O)CC1C(C)C 34435,c1(C(=O)NC(C2CN(C(=O)C3=COCC3)CCO2)C)cc(Cl)cc(Br)c1 34436,c1(C(=O)NCc2nnc(SC)s2)ncnc2c(C)csc12 34437,Cn1cc(C(=O)NCC(C)(C)CC2CN(C(C3CC3c3cccs3)=O)C2)nn1 34438,c1(N2CCN(C(c3cn(C)nc3)=O)CC2=O)ccc(F)cc1C(N)=O 34439,C1(C(N2CC(C(C)NC(=O)COC(F)F)OCC2)=O)CC2(CCCC2)C1 34440,C1(F)(C(N(C(CC)C)C)=O)CN(C(=O)COc2ccn(C)n2)C1 34441,N1(C(CC)=O)CCN(C(c2cc(-c3cccc(Cl)c3)on2)=O)CC(CO)C1 34442,c1(CNC(C2(OC)CNC2)C)ncc(C(C)(C)C)[nH]1 34443,c1(CCC(=O)NCC(CCOC)NC(CC2CC(OCC)C2)=O)ncccc1C 34444,c1(C(=O)NC(CNC(CC(CC)SC)=O)C)ccc2c(c1)CCN2C(C)=O 34445,N1(C(CCOCC#C)=O)CCC(C(=O)NCC(O)COCC)C12CC2 34446,C1(N(c2ccc(C(N)=O)cc2)C)CC2CC1CN2S(=O)(=O)C1CC1 34447,CCCC(C(=O)N1CCC(NC(=O)CNC(=O)C(C)(C)C)C12CCC2)C(C)C 34448,C1(CCNC(C=CCCC=C(C)C)=O)CC(F)(F)CN1C(c1ccc(Cl)s1)=O 34449,C(=O)(C1=CCN(C(c2ccn(C)n2)=O)C1)N(CC(O)C(F)(F)F)C 34450,CC1CN(C(=O)CCNC(=O)CO)CC1CC(=O)NC1CC1C1CCCO1 34451,N1(C(c2cncnc2)=O)CCC2(CCC(NC(=O)C(F)(F)C(O)C3CC3)C2)CC1 34452,C1(C(=O)NCc2c(CC)cncc2)CCCN1NC(=O)C(C)c1cnsc1 34453,CC1C(NC(=O)C=CC2CCOCC2)CCCN1C(C1CC2(CCC2O)C1)=O 34454,C(=O)(C(C(C)(C)C)OCC(=O)NC)C1C(C(=O)OCC)CCCC1.C(C(=O)N)NC 34455,C(=O)(CCCCC(C)C)NC1(C(N2CC(c3nc(C)on3)C2)=O)CC(C(F)F)C1 34456,c1(C(N2CC3C(NC(=O)CC(C4CC4)C4CC4)(CC3)C2)=O)cn2c(n1)CCCC2 34457,C1(NC(CCC=C=C)=O)CCC2CCN(C(c3ccc(F)c(C)c3Cl)=O)C1C2 34458,c1(C(N2CC(N(C(C3N(C(C)=O)CC(O)C3)=O)C)C2)=O)cc(F)ccc1F 34459,c1(OC)ccc(Cl)c(C(=O)NCC2(O)CN(c3nccc(C#N)n3)C2)n1 34460,C(CNC(=O)CC1CCCC1C)(CCNC(C1(C(C)C)CCC1)=O)OC 34461,CC(O)C(F)(F)C(=O)NC1COCC1NC(c1cc([N+](=O)[O-])n[nH]1)=O 34462,N(C(=NCC1=CCCCC1)NCC1(C#N)CCC1)CC1N(CC)CCC1 34463,C(=O)(C(C)(C)C(C)O)NCC(CNC(COCc1c(C)ncs1)=O)F 34464,N1(C(C(C)OCC=C)=O)CC(NC(c2nocc2C2CC2)=O)CC1(C)C 34465,N1(C(C(C)C2CC2)=O)CCN(C(=O)CN(C(c2ccco2)=O)C(C)C)CC1 34466,N1(C(CN(C(c2c(CCC)n[nH]c2)=O)C)=O)CC(N(C)C)C(C)C1 34467,Cc1ncc(C(=O)NC(C)(C)C(=O)NCCC2CCCCO2)cc1C#N 34468,N1(C(c2cc(C)c(F)cn2)=O)CCC2OCCN(C(=O)CC3CCCOC3)C2C1 34469,c1(C(=O)NCC2(CNC(c3ccc(NC)c(F)c3)=O)CC2)nn(C)cc1[N+](=O)[O-] 34470,C1(CN(C)C(C2CC(C#N)C2)=O)CCCN(C(=O)C(O)CF)C1 34471,N1(C(C2CC(C)(C)C(N)CC2)=O)CCC(S(=O)(=O)C(F)F)C1 34472,C(=O)(CCC(C)NC(c1c(Br)noc1C)=O)OCC 34473,c1(NC(C2N(Cc3ncn(C)c3)CCC2O)=O)ccc(N=Nc2ccccc2)cc1 34474,C1(C(=O)Nc2cccn(C3CCSC3)c2=O)CN2CC3CC2(CO1)C3 34475,n1(C(C)C)cncc1C(=O)N(CCC(=O)N(C)CC1CCCOC1)C 34476,N1(C(c2cc(OC)cc(C)c2)C(=O)NC(CC)C)CC(C)c2ccccc21 34477,C1(O)(CC(=O)NCC2C(NC(C3(C(=O)OC)CC34CC4)=O)CC2)CCCCC1.C=O 34478,c1(Cn2nnnc2C2(NCc3cn(C)nn3)CSC(C)C2)cnc2ncccn12 34479,N1(C(C2CCN(CC)CC2)=O)CCCC(CNC(c2cc(F)ccc2O)=O)C1C 34480,[N-]=[N+]=NC1CCC2(C(=O)NC(CO)CCCNC(c3cncc(F)c3)=O)CC12 34481,N1(C(C=NOC)=O)CCCC(C2CC2NC(=O)Cc2cc(C3CC3)nn2C)C1 34482,C1(CNC(C2CCC(CC)CC2)=O)CN(C(=O)C(CC(C)C)N(C)C)CCCO1 34483,c1(C(=O)NCC2CC(OC)CN2C(c2csc(C(F)F)c2)=O)nnc(O)cc1O 34484,C1(C)(CNC(C2(SC)CC2)=O)CCCC1NC(=O)CCS(C)=O 34485,c1(O)cccnc1.c1(COC2C(COC(C3(COC(C)(C)C)CC3)=O)C2)cccs1 34486,C=CC(C)(CCOC)C(=O)NCCN(C(=O)C1=COCCO1)CCC 34487,c1(C(=O)NC(C)C(CO)NC(C2CC3CCC(C2)O3)=O)cccc2c1ncn2C 34488,C(C(O)CC(=O)NCC1CC12CC2)NC(=O)CCc1ncccn1 34489,C1(N(C(CC(C)CF)=O)C)CCC2(CC1)CCN(C(c1ccc(F)cc1O)=O)C2 34490,c12ccccc1CCC(=O)N2.Cc1nn[nH]c1COC(C1CC=CCC1)=O 34491,C1(NC(CC(c2ccc(C)cc2)C)=O)CCN(C(C2(C)COC2)=O)C12CCCC2 34492,CC1(C)NC(=O)CC1C(N1CCCC(C(=O)NC2CC(C)C2)CC1)=O 34493,CC(C)CC(CNC(=O)CCCC#N)C(=O)NCCCC1CC1C 34494,CC(C)CC(C)CC(C)C(=O)NC1CC(C(C)NC(=O)Cc2cncnc2)C1 34495,C1(N(C(COCC=C)=O)C)CC2CCC(C1)N2C(C1(C(F)F)CCOCC1)=O 34496,N1(CC(=O)NC(c2cc(OC)cc(Cl)c2)c2ccco2)CC(=O)N2CCCC2C1 34497,c1(CC)ccc(C(N2CCC(C)(CNC(=O)C(C)(C)CO)C2)=O)c(C)n1 34498,C1(CNC(C(C(C)C)OC)=O)CN(C(c2c(C)cc(O)cc2C)=O)CC(C)(C)O1 34499,c1(C(=O)NCC2C(C)CN(C(C3CCCCO3)=O)C2)cc(Br)c(F)cc1N 34500,CCCN(CCCc1ccccc1)N1CCC(C(O)C(F)(F)F)C1 34501,C1(CCC#C)CCCN1C(=O)C(C1CCN(C(C2CC(=O)C2)=O)C1)C 34502,N1(C(c2cn(CC)nn2)=O)CCCCCC1CNC(=O)C(C)C(C)C 34503,c1(SCC(=O)NCC2CCC2NC(=O)CC2CCCSC2)ccccn1 34504,CC1(CCO)CCN1C(=O)C(C1CCOC1)NC(C1CC(F)C1)=O 34505,CC1CC(NC(=O)CC(F)F)CN(C(=O)Cn2cnc(Br)c2)C1 34506,c1(C(N(CCNC(C2CCC(CC)C2)=O)C2CC2)=O)cc(N)cnc1C 34507,C1(NC(c2coc(C3CCC3)n2)=O)COC2(C1)CN(C(c1cc[nH]n1)=O)C2 34508,C1(NC(CC(COC)C)=O)CC1C1CCCN(C(c2cnn(C)c2Cl)=O)C1 34509,N1(C(C2(C3CC3)CCC2)=O)CCCC(C2CCN(C(C3CCCO3)=O)CC2)C1 34510,C(=O)(C#CC1(C)COC1)NCC1CN(C(Cn2ccc(C)cc2=O)=O)CC1O 34511,N1(C(C2C(OCC)C2)=O)CCC(NC(=O)CCn2cccnc2=O)C(CO)CC1 34512,C1(NC(C(CNC(c2cccc(=O)o2)=O)O)=O)C(O)C2CCOC12 34513,c1(OC)cc(OC)cc(C(C)NC(N2CCNC(=O)C2)=O)c1 34514,C12(CNC(c3cc(CC)n(C)n3)=O)CC(CO1)N(C(=O)C(C)CO)C2 34515,C(=O)(CCCC(C)CC)NC1(C(N2CCCCC(CCC)C2)=O)CCOCC1 34516,c1(-c2ccccc2CNC2CCSC2)n[nH]c2c1CCC2 34517,c1(C(N(C)CCN(C)C(C2CCCS(=O)(=O)C2)=O)=O)cncc2n[nH]cc12 34518,C=Cn1nccc1C(=O)NC1CC(C(F)C(=O)NCCOC2(C)CCC2)C1 34519,C1(C#CC(=O)N2CC(NC(C3(C(C)(C)C)CCCCC3)=O)CC2C)(CC)COC1 34520,C1(C2CC2)(NC(CCNC(c2nn(C)c(O)c2)=O)=O)CCOC1 34521,c1(OC)cc(NCC(C2CC2)N(C(=O)C(C)CC(F)(F)F)C)ccc1[N+](=O)[O-] 34522,CCC(CC(=O)NC1(CCC(=O)NCc2cn(C)cn2)CCCC1)C(C)C 34523,N1(C(C(C)O)=O)CCC(n2cc(CN(CCC(F)(F)F)CC(F)(F)F)nn2)CC1 34524,C1(OCc2cn(CC(=C)CC)nn2)CCCN(C(=O)CC2CCCC(O)C2)C1 34525,C=CC1CN(C(c2ncsc2C)=O)CC1NC(=O)C(C)(C)C1CC1 34526,C1(NC(c2c(C)ccn2C)=O)CC2(C1)CC(CNC(=O)CN1CCC(C)C1)C2 34527,CC1(C2CC2C(N2CCCC2C(C)(C)C(N2CC3CCC2CC3)=O)=O)COC1 34528,n1(CC(=O)NC(C(=O)NCCC2COCCO2)C2(O)CCC2)cc(CO)nn1 34529,C(=O)(CC(CC)CCCC)NC(CC#C)CC(=O)NCC1(C)CC(C)=NO1 34530,CCC(CC(=O)NCC1(C(=O)NCc2ccco2)CCCO1)C1CC1 34531,Cc1nn2cc(C(N3CCC(N(C(=O)C(c4ccccc4F)C)C)C3)=O)nc2s1 34532,N1(CC(N2CCC(NC(=O)CC3CCSCC3)C2)=O)C(=O)CNC1=O 34533,N1(C(c2c(SC)nccn2)=O)CCC2(CCC(NC(=O)Cc3nccs3)CC2)C1 34534,CC1C(NC(=O)C(CCN(C)C)NC(=O)Cc2ncccc2F)CCCN1C 34535,n1(CC(=O)N(C(CN(C(C2N(CC)CC2)=O)C)C)C)cc(C(F)F)cn1 34536,C1(CC)CCC(C(N2CCC2CC(=O)NCC(C)O)=O)CC1 34537,C(=O)(C1=Cc2ccccc2C1C)NC(C)CCCNC(=O)C1=C(Cl)CC1 34538,Cc1ccc(C(N2CC=CC(NC(=O)C(c3ccccc3)O)C2)=O)cc1F 34539,Cc1cc(C(N2CCOC(C(=O)NCCCCC3CCCC3)C2)=O)c(C)s1 34540,N1(C(c2cc(C)ncn2)=O)CCC(CO)C(NC(c2csc(C(F)(F)F)c2)=O)C1 34541,C(=O)(C1=CS(=O)(=O)CCC1)N1CCC(N(C(=O)C(C)Cc2cnc[nH]2)CC)CC1 34542,c1(C(=O)NC)cc(Cl)c(NC(c2c(F)ccc(-c3nn[nH]n3)c2C)=O)c(Cl)c1 34543,c1(C(C(=O)N(CC(C)NC(=O)COC2CCCCC2)CC)C)ccc(F)c(F)c1 34544,N1(CCC)CCSC(C(=O)N(CCC2CCCCC2)C(C)=O)C1 34545,C1(C(=O)NCC2N(C(C3(CCCC)CC3)=O)CC2)CCC(F)C1 34546,N1(C(CCCN(C(=O)OC)C)=O)CCN(C)CC1CNC(C12CC(F)C1C2)=O 34547,c1(NC(N2CCC(C)(c3cn(CC4CC4)nn3)C2)=O)cnc2ccccc2c1 34548,C1(n2cc(C(C)O)nn2)CCCN(N2CC(CCOc3ccccc3)C2)C1 34549,N1(C(=O)Cc2c(C)cnn2C)CCCC(C)C1CCNC(c1c(OC)scc1)=O 34550,c1(C(=O)NC2(CNC(=O)CCF)CCC2)cc(Cl)c2c(c1)OCCO2 34551,N#Cc1ccnc(NCC(c2ccccc2F)NC(C2(C(F)(F)F)CC2)=O)n1 34552,c1(NC(C2CN(C(CCS(C)(=O)=O)=O)CC2C2CC2)=O)cccc2cnccc12 34553,C=CCC(CNC(C1C2CCCC12)=O)C(=O)N1C2CCC1CC2 34554,c1(CC(N2CC(NC(C=CS(C)=O)=O)CC2(C)C)=O)ccc(Br)cc1C#N 34555,CCCCC(C(=O)N(C)CC1CCC(=O)N1)NC(c1n[nH]c(=N)[nH]1)=O 34556,NS(=O)(=O)N1CC(C(=O)NCC2C3CN(C(=O)CCCN4CCOCC4)CC23)C1 34557,C12(CNC(C3C=CCC3)=O)CC1CN(C(C1(c3cncc(Br)c3)CCC1)=O)C2 34558,C1(N(C2CCCCC2)C)CCN(CC2CCCC2(C)C)CC1 34559,Cc1cc2cccnc2nc1C(=O)NC1CN(C(c2cnc(S)[nH]2)=O)C1 34560,C1(NC(Cc2c(C)ccs2)=O)CCCN(C(c2ccccc2CO)=O)C1C 34561,C1(NC(C2N(CC)CC2)=O)CCSC12CN(C(C1CCN(CC3CC3)CC1)=O)C2 34562,c1(CNC(c2ccnn(C)c2=O)=O)ccc([N+](=O)[O-])cc1.C12CN(CC1F)C2=O 34563,N1(C(c2c(C)ccs2)=O)CCC2CN(C(C3COCCO3)=O)CCC12 34564,Cc1cc(NC(C2CN(C(c3cnc(C)c(C)c3)=O)CC2(F)F)=O)c(C)cc1O 34565,C1(NC(=O)C=CCN2CCOCC2)CC2(C1)CN(C(C1CCC3(CCC3)C1)=O)C2 34566,N1(C(NC2COc3ccccc32)=O)CCc2c(cc(F)c(F)c2F)C1 34567,c1(C(=O)NCCCC(C)NC(C2CN3CCC2CC3)=O)nn(C)c2c1CCCC2 34568,c1(CC(N2C(C)CC(Nc3nccc(CO)n3)C2)=O)cn2ccccc2n1 34569,C(=O)(CC(F)(F)CC)NC(C(C)NC(C(CCC)NC(=O)OC(C)(C)C)=O)CO 34570,Cc1cnc(N)c(C(N2CC(F)CC2CN(C)C(C2CCC3(CCC3)O2)=O)=O)c1 34571,Cc1nn2cc(C(=O)NCC(CC(C)C)NC(C3COC(=O)N3C)=O)nc2s1 34572,C#Cc1cccc(C(N2CCN(C(c3cc(C)nnc3O)=O)C(CC)C2)=O)c1Cl 34573,N1(C(C(CC)(C)C)=O)CC2CCCC(C1)N2C(=O)Cc1cccc2c1CCC2 34574,CC1CCN(C(c2cn(CC3(C)COC3)nn2)=O)CC1NC(c1cnn(C)c1)=O 34575,N1(C(C(CC)n2cncn2)=O)CC2CCC1CN2Cc1cccnc1 34576,c1(C(=O)NCC2(NC(c3nc(CCCCC)sc3)=O)CC2)cc(COC)ncn1 34577,c1(OC)ccccc1C(=O)NCC(C(C)C)NC(c1cnn(C(F)(F)F)c1)=O 34578,N1(C(=O)OC(C)(C)C)CC2CCCN(Cc3cccc(F)c3Cl)C2C1 34579,c1(C(CC(=O)N(C2CCN(C(=O)COCC3CC3)CC2)CC)C)ccc(F)cc1 34580,C(=O)(C(C)(C)CCC(=O)NC1CC2C1CCN2C(=O)C(C)NS(C)(=O)=O)OC 34581,CCC(O)C(C)C(=O)NC1(CO)CN(C(=O)C=CC(C)C)C1 34582,Cc1ocnc1CC(=O)N(CCCCCNC(=O)CC(C)n1cccc1)C 34583,C(CCCC(CO)NC(c1cc(C)nnc1CC)=O)NC(CC=CC)=O 34584,c1(CC(=O)NC2CCCC(CN=c3[nH]nc(O)s3)C2)cccc(Cl)c1Cl 34585,c1(OC(C)C)cccc(C(N2CCC(F)C(NC(=O)C(C)N(C)C)C2)=O)c1F 34586,C1(NC(C)=O)CCCCC12CCN(C(c1cc3c(Cl)cc(F)cc3[nH]1)=O)C2 34587,c1(NC(=O)OCC)ccc(C(=O)NCC2CCC(NC(=O)C(C)O)C2)cc1 34588,c1(C(=O)NCC(C)N(C(=O)C(C2CCC2)OC)CC)cc(C)ccc1OC 34589,n1(CC(=O)OC)cnc(C)c1C(=O)NCCCCNC(=O)C(C)Cn1cccn1 34590,N1(C(c2ncn(CC)n2)=O)CCC2CC12C(=O)NCCCc1c[nH]nc1C 34591,C1(C(=O)NCCOC2CN(C(CC3(C=C)CC3)=O)C2)CCS(=O)(=O)C(C)C1 34592,N1(C(C23CC(OC)C2C3)=O)CC(NC(c2cc(C(C)C)on2)=O)C(O)C1 34593,CC(=O)CCN=C(NCCCCCF)N1CCC(C2CC2)C1 34594,N1(Cc2c(OC)cccn2)C2CCCC1CC(NC(C1(C)CCCC1)=O)C2 34595,C#Cc1ccc(F)c(C(N2CCC(C)C(CNCc3ccc(CSC)o3)C2)=O)c1 34596,CC(C)(CCNC(=O)C=CCOC(C)(C)C)NC(C1CCC1F)=O 34597,C1(C2CCN(C(c3coc(Cl)n3)=O)CC2)(NC(C2(C)CC2)=O)CC1 34598,C1(CCOCCC(=O)NCC(C)N(C)C)CCCNC1 34599,N1(C(CCOCCOCC)=O)CC(O)CC1C(=O)N(C1CCC(OC)CC1)C 34600,c1(C(=O)NC(C(=O)N(CC#C)C(C)C)C2(C)CC2)ccc(CC)o1 34601,c1(CC(=O)NC2CCN(C(C(CC)F)=O)C2(C)C)ccc2nc(O)[nH]c2c1 34602,N1(C(c2cc(COC)on2)C(=O)NCCCC)CCOC(c2n[nH]c(C)n2)C1 34603,C1(C(=O)NCC2CC(NC(C3CN(S(CC)(=O)=O)C3)=O)C2)CCC(F)(F)CC1 34604,CC(C)CC(F)C(=O)N(CCCCCNC(c1nn(C)cc1Br)=O)C 34605,Cn1cnc(C(N2CCCCC2CNC(C2CCCC2(F)F)=O)=O)cc1=O 34606,C12(NC(c3ccc(O)nc3)=O)CCCC1N(C(c1ccc3nccn3c1)=O)CC2 34607,N1(C(c2c(C)nc[nH]2)=O)CCOC(CNC(=O)C(F)(F)c2ccsc2Cl)C1 34608,CC1CN(C(C2CCCN2C)=O)CCN1C(c1cc(Cl)ns1)=O 34609,Cc1c(CN(C(N2CCC2C2CCCCC2)=O)CC2CC2)oc2ccccc12 34610,C(=O)(C(CC(C)(F)F)C(C)OC(C)(C)C)NC(C(C)NC(CC=C=C)=O)CO 34611,c1(-n2c(CSC)nc(Cc3cccc(OCC)c3)n2)ccc2[nH]ncc2c1 34612,c1(C(=O)NC2CCCN(C(C3C(C(C)C)CCC3)=O)CC2)cnc2c(c1)CCC2 34613,Cn1ncc(=NC(=O)C2CC23CCN(Cc2ccc(C(=O)O)s2)C3)[nH]1 34614,c1(C(=O)NC2CCCC(NC(C3CC(F)C3)=O)C2)c(F)c(F)c(F)c(F)c1F 34615,N1(C(C(C2CC2)OC)=O)CCC2(CCCN2C(C2(c3ccccc3)CC2)=O)CC1 34616,Cc1cnc2n1CCCC2CNC(c1n[nH]c2c1CCC(F)(F)C2)=O 34617,N1(C(C2(COC)CCCC2)=O)CCC(C2CC2)(NC(=O)C(O)C2CCCC2)C1 34618,C1(C2(O)CCOC2)(C(N(C)CC2CCN(C(c3ccc(C4CC4)o3)=O)C2)=O)CC1 34619,C1(NC(C(C2CCCO2)NC(c2cc(C)n(C)n2)=O)=O)CC(C2CCC2)C1 34620,C1(NC(COCCC)=O)CC2CN(C(C3CC(Cl)(Cl)C3)=O)CC2C1 34621,C1(NC(c2c(C)n[nH]c2)=O)CC2CCC1N2C(=O)C=CC1CCOC1 34622,C=CCC(CC(C)C)C(=O)NC1CCN(C(=O)CC2CCSC2)C1C 34623,N1(C(C(CC)F)=O)CCN(C(=O)CSc2cccs2)C2COCC12 34624,CC(CC(=O)N1CCC(C(=O)OCC)O1)N(C)C.C(C(C)(C)N(C)C)N 34625,C1(NC(CC2(COC)CCC2)=O)CCN(C(C2CC3(CSC3)C2)=O)C1C1CC1 34626,C1(NC(c2cc(C(C)=O)on2)=O)CCCCC1NC(=O)CCc1cncnc1O 34627,c1(CC)oc2ccccc2c1C(N1CC(CNC(=O)C(C)CSC)C(F)(F)C1)=O 34628,CC(Cc1nccn1C)N=c1[nH]c(=NC(C)c2nc[nH]n2)[nH]c2ncn(C)c12 34629,Cc1nc(CC(=O)N(C)CC2(O)CN(C(C3(NC(N)=O)CC3)=O)C2)co1 34630,C(=O)(CCCCBr)NC(CC(=O)Nc1nccs1)c1ccccc1 34631,c1(OCCC(C)NC(=O)Nc2nn(C)cc2-c2cn[nH]c2)cccc(F)c1 34632,CCCC(C)CC(=O)NCC1(O)CCCN(C(=O)CCc2nc(C(C)C)no2)C1 34633,C(=O)(CCCCCCO)N1CCC(O)(CNC(c2ccc(Cl)cc2C(F)F)=O)C1 34634,c1(C(N(C)CCNC(C2CS(=O)(=O)CC(=O)N2)=O)=O)cccc2cnnc(O)c12 34635,Cc1sc(Cl)nc1C(N1CCCCC1CN(C)C(C1CC1CF)=O)=O 34636,c1(C(=O)OC)cc(=O)n(CC(=O)N(C2(C)CCCC2)C)cn1 34637,C1(CC(=O)N(CCCN(C(=O)CC=C(C)C)CCC)C2CC2)CCC(C)C1 34638,c1(C(=O)NCCCCCN(C(=O)CC2CC2(C)C)C)cnn2c(Cl)cccc12 34639,Cc1cc(C(=O)NCCC(C)N(C(=O)COCc2nccn2C)C)cc(C)c1Cl 34640,CC1CN(C(=O)CSS(C)(=O)=O)CC1NC(=O)CCCc1ccsc1 34641,n1(CC)cc(Cl)c(C(=O)NC2CCC2NC(c2cnc[nH]2)=O)n1 34642,N1(C(c2n[nH]c(C)c2Cl)=O)CCCC(C)(CNC(=O)CC2CC(C)(C)CCO2)C1 34643,N1(C(c2cc(CCC)[nH]n2)=O)CCN(C(C2CCC(=O)N2)=O)CC1C(C)(C)C 34644,S(=O)(=O)(c1c[nH]c2nc(Cl)ccc12)NCC1CCC(CC)C1 34645,C1(CNC(CCNC(=O)OCC)=O)CC2(CCC2)CN1C(C1CC1(Cl)Cl)=O 34646,C1(NC(CCC2N(C)CCC2)=O)CC=C(C(=O)Nc2ccc(C3CC3)nc2)C1 34647,O=S(=O)(c1ccncc1)NC1C2CCC1CC(CO)C2 34648,CC(CS(C)(=O)=O)C(=O)N1CC2CC(NC(c3ccc(N(C)C)nc3)=O)C(C2)C1 34649,C1(NC(=O)C(C2(O)CCCC2)F)CCSC12CN(C(c1ccc(F)cc1Cl)=O)C2 34650,CC(CCC(C)(C)C)N=c1[nH]c(N2CC3C4CCC(C4)C3(C)C2)nc(=N)[nH]1 34651,Cc1c(C(=O)N(CC(O)CNC(C2CC3(CCCO3)C2)=O)C)sc2nccn12 34652,c1(CC(=O)NC(CC)(C)CNC(=O)Cc2cccs2)ccc2scc(C)c2c1 34653,c1(CC)nnc(C)cc1C(N1CC(O)(CNC(c2nn(C)c(C)c2Cl)=O)C1)=O 34654,CC(C)CC(C)(CNC(c1ccc(F)cc1F)=O)NC(C1CC(OC(C)(C)C)C1)=O 34655,C=C(Cl)C(C)(C)C(=O)N1CC(n2cc(-c3cccc(N)c3C)nn2)C(C)C1 34656,OC1COC2(C1)CN(CC1(F)CCNCC1)C2 34657,c1(CCC(=O)NCCOCCCN(C(=O)C(=O)C(C)(C)C)C)cc(Cl)cc(Cl)c1 34658,CC1CC2(CCO1)CC2C(=O)NCCN1CCN(c2ccncc2[N+](=O)[O-])CC1 34659,N#Cc1ccc(CC(=O)NCC2CCN(C(=O)CCN3CCCC3)C2)cc1 34660,C(c1ccc(F)cc1)=CC(=O)NCC1CC(F)(CNC(C2(F)CC2(F)F)=O)C1 34661,N(C(=NC1CCCC1)N(C)C1CCSCC1)C(C#C)Cc1cccc(F)c1 34662,c1(CCC(=O)N(CC)Cc2cn(CCN3CCOCC3)nn2)ccc(Br)cc1 34663,N1(CC(=O)NCC=C)CCN(C2CCN(C(=O)CC(C)OC)C2)CC1 34664,C1(CN(C(C(n2ccc(C(F)(F)F)n2)C)=O)C)CC(F)CN1C(c1ccns1)=O 34665,N1(C(C(=O)NCC)=O)CCC(C)(C)C(CNC(c2c(C)noc2C2CC2)=O)C1 34666,N1(C(CSC(C)=O)=O)CCC2(CCC(C(=O)NCCNn3nccn3)O2)CC1 34667,CN(C)N(C(=O)C1CC12CCOCC2)S(=O)(=O)c1cc([N+](=O)[O-])ccc1Cl 34668,C1(c2n(C)ccn2)CCCN(C(=O)C(C)(N)C(F)F)CC1 34669,N1(C(c2ccc(OC)c(C(C)C)c2)C(=O)NC2CCCC2)CCOCC12CCC2 34670,C1(C(=O)NC(C2CCN(C(Cc3ncc(C)o3)=O)CC2)(C)C)CCCC(C)(C)C1 34671,C(=O)(C1=CC2CCCCC12)N1C(C(C)(C)NC(c2c(OC)cccc2)=O)CCC1 34672,c1(C(=O)NCC23C(CN(C(C(CC)NC(C)=O)=O)C2)C3)cccc2c1CCO2 34673,Cc1c[nH]c(C(=O)NCC(C)(C2CC2)NC(c2cnc(C(N)=O)s2)=O)c1 34674,Clc1ccc(CNc2cnn(C3CCOC3)n2)c(I)c1 34675,N1(C(C2CCC(COC)C2)=O)CCN(C(c2cnc(C)s2)=O)CC(O)C1 34676,C(C(O)CS(=O)(=O)c1cccs1)NC(c1ccc(-n2ncc(C(=O)O)c2)cc1)=O 34677,CC1CCN(C(C2CCC=CO2)=O)CC1NC(=O)CC1CCC(C(C)(C)C)CC1 34678,C12(C(N3C4CN(C(C5C(CC)C5)=O)CC3CC4)=O)CCCCC1CCCC2 34679,C#CC1CC2CCC1N(C(c1ccccc1OC1CCCCC1)=O)C2 34680,c1(C(C(C)(C)C)NC(N(CC2(OC)CCC2)CC2CCCO2)=O)cccc(C)c1 34681,c1(C(N2CCC3(NC(C4COC4)=O)C(C2)C3)=O)cc[nH]c2nccc1-2 34682,c1(C(N2CCC(O)(c3onc(C)n3)C2)=O)nc(C(F)(F)F)ccc1Br 34683,n1(CC(=O)NCC2CCCN(C(=O)CCc3cncnc3)C2)cc([N+](=O)[O-])cn1 34684,c1(CN(CC(=O)NC(CNC(CN(C(=O)OC)C)=O)(C)C)C)nnc(C)n1C 34685,C(CCOCC)(C(=O)N(C(C(N)=O)C1CC1)C)NC(C=CCC)=O 34686,C1(c2cccs2)(CN(CC(C)(C)CO)CC=C(C)C)CCCC1 34687,CCC(CC)(C(=O)N1CCC(NC(c2nonc2N)=O)C1)c1ccccc1 34688,Cn1c(Br)cnc1NC(N1CCN(c2ccc(Cl)nn2)CC1)=O 34689,c1(OC)ccc2c(c1)CCC2(C)CNc1nc(OC)ncc1Cl 34690,C(=O)(C#CC1CCCCC1)N1CC(N(C)C(c2ccc(Cl)c(F)c2)=O)C1 34691,c1(OC)ccccc1C(=O)NC(CNC(=O)C(C1CCCC1)OC)CO 34692,Cn1cc(C(N2CCC(O)(CNC(C3CCC(=O)N3)=O)C2)=O)c2cc(F)ccc12 34693,Cc1cc(C(N2CCC(C)(C(=O)NCC3(C)CC4CCC3C4)CC2)=O)c(C)n1C 34694,C#CC1CCC(NC(c2csc(CNC(c3ccc(CO)cc3)=O)c2)=O)C1 34695,N1(C(C(N2C(CC)CCC2)=O)=O)CCOCC1CN(C(=O)Cc1ccsc1)C 34696,C(=O)(CCC(=O)NN(C)C)NC1C(CO)CCN(C(COCCCC)=O)C1 34697,c1(C(=O)NCC2CC(F)CN2C(c2cnn(C(F)F)c2)=O)cccc2cccn12 34698,c1(C(=O)NCC(C(C)C)NC(C2(F)CC2C)=O)ccc(SC(F)(F)F)nc1 34699,N1(C(C2ON=C(C)C2)=O)CC(NC(=O)C2=CCCSC2)CC12CCCC2 34700,C1(NC(C=CSC)=O)C(C)CN(C(=O)CN2CCCNS2(=O)=O)CC1C 34701,c1(CC(C)NC(=O)C(N)=O)ccccc1CNC(=O)CC1(O)CCOC1 34702,N1(C(CCC=C)=O)CCCC2C1CCN2Cc1cc(Br)cnc1OC 34703,c1(CC(=O)NCC2C(NC(C(CC)O)=O)CC2)c(C)nn(CC(C)C)c1C 34704,CC(C)C(CC(=O)N(C1CC(CO)C1)C)NC(C1CC2CC(=O)C1O2)=O 34705,C(CCC(C)C(=O)NCC1(C(=O)O)CCOC1)OC 34706,c1(C(N2C(CNC(C3C(C)=CCS3)=O)CC(O)C2)=O)cnn2c1CCC2 34707,CC1(CNC(=O)C=CCO)CC(F)(F)CN1C(C1CCC2(CC2)C1)=O 34708,C1(NC(Cc2nc(C)[nH]n2)=O)CNCCOC1 34709,C1(NC(CC(=C=C)C)=O)CN(C(=O)CC2CCCOC2)C2(CCOCC2)C1 34710,c1(CC)nc(C(=O)NCC(C)(C)NC(C2CC(F)(CO)C2)=O)c(C)o1 34711,C(C)(C(=O)NC1(C)CCC(C)C1)(C(C)C)NC(C)=O 34712,c1(C(=O)NC2CC(CNC(=O)COC3COC3)C2)cc(Cl)ncc1F 34713,N12CCOC(C)(C1)COC1CC1C2=O.c1(C(=O)OCC)ncnc(OCC)c1F 34714,c1(C(N(C2CCN(C(C3CC34CC4)=O)CC2)CC#CC)=O)ncncc1Cl 34715,c1(C(N2CCC(C3CC3)(NC(C(F)=CC)=O)C2)=O)ccc2cnnc(O)c2c1 34716,C(CC(C(=O)NC(c1cncc(F)c1)C)NC(=O)Cc1nc(=N)[nH][nH]1)=CC 34717,c1(C(N2CC(NC(c3n(CC)nnc3)=O)C3C2C3)=O)cnc(N)c(N)c1 34718,Cc1ccc(CNC2CC3(C2)CC(C(=O)NCc2ccc(C#N)cc2)C3)c(O)c1 34719,N1(C(c2c(OC)nsc2)=O)C2COCC1CC(NC(=O)C(C)=NOCC#N)C2 34720,c1(C2(OC)CCCC2)nnc(N2CCC(CO)C2)n1Cc1ccc(C(N)=O)cc1 34721,C1(C(C)C)CN(C(c2cnc(O)o2)=O)CC1C(=O)NC1CCC(C(C)O)CC1 34722,c1(NC(C(n2cc(COC)nn2)C)=O)ccccc1F 34723,C(=O)(C(O)C(C)(C)CC)N1CC(NC(CCC=CC)=O)C2(C1)CC2 34724,C1(C(=O)NCCOCCN(C)C)(CNC(c2nonc2N)=O)CCOCC1 34725,C1(NC(c2c(C)nsc2)=O)CCCC(C(=O)NCCC2CCCC(C)C2)CC1 34726,N1(C(C(c2nc(C)sc2)=O)=O)CCOC(C)(CNC(=O)CCCc2cnn[nH]2)C1 34727,c1(C(=O)NC(c2c(C(=O)NC3(C(=O)NC)CCC3)con2)C)cc(O)nc(C)n1 34728,CN=S(C)(=O)c1cccc(CNC2CCN(C(=O)OC(C)(C)C)CCC2CO)c1 34729,C#Cc1ccc(C(=O)NC2CC(C(C)NC(c3cn(CCC)nc3C)=O)C2)cn1 34730,c1(C(N2CCC3CN(C(=O)CCc4cc[nH]n4)CC32)=O)ccc2nc(S)oc2c1 34731,CC1(C)OCCOC1CC(=O)NCCOCCCNC(=O)CC1OCCCO1 34732,N1(C(C)C=CC(F)(F)F)C(=O)CN(CC2(c3cccs3)CC2)C1=O 34733,C1(C(C)C)CCOC1C(=O)NCC1CC1C(=O)N(CC1=CCSC1)C 34734,C1(NC(C2(C)N(C)CCC2)=O)C2CCC(C2)C1C(=O)NC1COCC1O 34735,Cn1cnc(CNc2cccc(OCC3CCCCC3)c2)cc1=O 34736,c1(CNC(=O)NC(C)CCc2ccccc2Cl)c(Cl)ccc(Br)c1F 34737,c1(C(=O)NCCCCCN(C(=O)CC2CCCC(F)(F)C2)C)cc(=O)n(C)cn1 34738,C1(C(C(=O)NC(CC)CNC(c2ccoc2CC(N)=O)=O)F)CCC(=O)CC1 34739,C1(C2CCN(C(=O)CC3(C)CC3(F)Cl)C2)(NC(c2n[nH]c(C)c2C)=O)CC1 34740,c1(C(=O)NCC2(OC)CN(C(C3(CC)CCCCO3)=O)C2)ccc(C)cc1Cl 34741,c1(NC(N(CCC(=O)OCC)CC)=O)ccc(C)cc1OCCCCCC 34742,C(=O)(C(CCC(C)C)NC(=O)Cc1c(C)n[nH]c1C)N1CCC(SC)C1 34743,N(C(=NCCC(=O)N(C)C)N1CCCC(O)CC1)Cc1c(C)nc(Cl)cc1 34744,C#CCCC(=O)N(CCC(C)(C)NC(C1CC(NC(C)=O)C1)=O)C 34745,c1(OC)ccc(S(=O)(=O)NC2C3CN(C(=O)CCCC(F)(F)F)CC23)cn1 34746,C(CC(C(=O)N(C)Cc1nc(C)no1)NC(=O)CCCc1ncco1)OC 34747,c1(CC(=O)NCC(C)NC(CC(c2cccc(OC)c2)C)=O)ccc(F)c(C)c1 34748,N1(C(CSCCC)=O)CCc2cc(CNC(c3ncoc3C3CC3)=O)ccc2C1 34749,C12(C(=O)NC3CCCCN(C(C=CCCC)=O)C3)CCOC1CCOC2 34750,N1(C(C(CC#C)C)=O)CC2CCC1C(CNC(C1(c3cccc(Cl)c3)CC1)=O)C2 34751,N1(C(C2CC3(CCC3O)C2)=O)CCCC(F)(C(N2CCCC(CC3CC3)C2)=O)C1 34752,c1(C(=O)NC(CC(C)NC(c2c(C#C)c[nH]n2)=O)C)noc2c1CCCC2 34753,Cc1nc(O)nc(O)c1CC(N1CCCC(CNC(C2(C(N)=O)CCC2)=O)C1)=O 34754,c1(N(C)C)ncc(C(N2CC(O)(CCNC(c3cc(C(F)(F)F)n[nH]3)=O)C2)=O)s1 34755,N(C1CC2(CCC2)Oc2ccc(F)cc21)C(c1n(C)c(Cl)nc1)c1nnnn1CC 34756,C1(C(N2CC(C(C)(C)O)C2)=O)CN(C(=O)CCc2cncs2)CC2(CCC2)C1 34757,c1(C(=O)NCC(C)NC(=O)Cc2ccc(Br)cc2)nccc(C#N)c1F 34758,c1(CC(=O)N(C2CCCCC2NC(C2CC(F)C2)=O)C)c[nH]c2cc(Cl)ccc12 34759,c1(OC)ccccc1NC(C1CCCN(C(C2(C)CC2)=O)C1)=O 34760,CCCCCCCCC(F)C(=O)N1CC(NC(=O)C2=CCCOC2)C(O)C1 34761,c1(C(=O)NCC2CC(NC(CCCCCC#N)=O)C2)ccc2c(O)nncc2c1 34762,C=CC(C)CC(=O)NCCOCCOCCNC(C1CCCCO1)=O 34763,N1(C(CCC(C)OC)=O)CCCC(F)(C(=O)NC2CC(C)C2)C1 34764,C1(CC=C)CCCCN1C(C1CCN1C(=O)CC1CCOC1)=O 34765,N1(C(C(CC)(C)F)=O)CCC2(CC1)CN(C(C1CC(=C3CCC3)C1)=O)C2 34766,O=C(C1=CC(O)CCC1)NCC(C1CCCC1)NC(c1cccc[n+]1[O-])=O 34767,C(c1ccccc1)=C(C(=O)NCC1C(NC(CCC=C)=O)CCC1)CC=C(C)C 34768,n1(CC)cccc1C(c1nnnn1C1CCOC1)NCc1cncs1 34769,c1(C(=O)NCCCNC(C(C(C)O)N(C)C)=O)nnc2n1CCCCC2 34770,Cc1coc(C(C)(C)C)c1C(N1CC(N(C(=O)C(F)C2CCOC2)C)C1)=O 34771,c1(NC(c2n(C)cc(NC(c3ccc(Cl)nc3)=O)n2)=O)cc(Cl)c(F)c(Cl)c1F 34772,N1(C(C2(C)N(C(c3c(CC)noc3)=O)CCC2)=O)CCc2ncncc2C1 34773,C1(C(=O)NC(C)CNC(=O)CC2(C)CC(F)(F)C2)CC2(C1)C(F)(F)C21CC1 34774,C(CO)(CC(F)(F)F)NC(C(c1n(C)ncc1)NC(C1OCCC1(C)C)=O)=O 34775,C(=O)(CC1=CCN(C(C23CCC(OC)C2C3)=O)CC1)N(CCC=C)CC 34776,C1(CCNC(c2coc(Cl)c2)=O)CCCN(C(C2CCCCN2CC(F)F)=O)C1 34777,N(C1CCOc2ccc(Cl)cc21)C(c1c(C)sc(-c2ccc(F)cc2CO)n1)=O 34778,N1(C(c2c(C)scc2)=O)Cc2nccn2CC(NC(c2ccn(O)c(=O)c2)=O)C1 34779,C#Cc1ccc(CC(=O)NCC2(NC(c3coc(C(F)(F)F)c3)=O)CC2)cc1 34780,N1(C(c2c(C)snn2)=O)CCN(C(c2cccn2C)=O)CC1CCO 34781,CC(C)S(=O)(=O)CCCN1CCCC1C1CCCN(C(=O)C(=O)NC2CC2)CC1 34782,CC(C)(Cc1ccccc1)C(=O)N1CCOC(CNC(=O)C(C#N)C2CC2)C1 34783,c1(COC)cc(C(N2CCC2CNC(c2ccccn2)=O)=O)on1 34784,c1(-c2nnc(C(N(CC(C)(C)CN)C3CC3)=O)o2)ccc(Cl)cc1.C#CC1(C)CC1 34785,S(=O)(=O)(c1ccncc1)NCC1CCN(C(c2ccc(CC)cc2)=O)CC1O 34786,CC1c2c[nH]nc2CCC1C(N1CCC(CNC(=O)CC2=CCCC2)C1(C)C)=O 34787,N1(C(C(CCC)NC(C)=O)=O)CCN(Cc2cnc(OC)c(C)c2)CC1C#N 34788,c1(C(=O)NC(C)C(=O)NC(c2nc[nH]n2)CO)cc[nH]c2nccc1-2 34789,c1(C(=O)NC2CN(C(c3ncc(C)c(C)c3)=O)C(C)C2)ccc([N+](=O)[O-])n1C 34790,C1(CC(N2CCC(O)(CNC(c3cnc(C(C)C)s3)=O)C2)=O)OCCCC1(C)C 34791,c1(C(=O)NCC(CC)NC(c2snnc2C)=O)cccc2cnsc12 34792,C1(C(N2CC3C(CNC(C4(CCOC)CCC4)=O)C3C2)=O)CC2(CCC2)CO1.CO 34793,Cc1ccc(C(=O)NC(C2CCN(C(C34CCC3C4)=O)C2)(C)C)cc1 34794,c1(C(=O)NC2C(SC)CN(C(=O)CN3CCSCC3)C2)nccn2cc(C)nc12 34795,N1(C(=O)CCN2CCCC2)CCC(C(N2CCCC(CN(C)C)C2)=O)CC1 34796,C1(C(N2CCN(CCN(C(=O)Cn3ccnn3)C)CC2)=O)CCCC12OCCO2 34797,C1(C(=O)NCC2CC(CNc3nccc(OC)n3)OC2)CCCCCS1(=O)=O 34798,N1(C(CNC(CC)=O)=O)CC(NC(=O)Cc2ccccc2C)CCC1C 34799,N1(C(C23NC(=O)C4CC(C2)CC34)=O)CCCC2CN(C(c3coc(Cl)n3)=O)CC12 34800,C1(C(=O)NCCSCC(N2CC=CC2CF)=O)C=CCCC1 34801,C(C(Cl)C(C)(F)F)N1CC1=O.CN1CC(C(N2CCC2CO)=O)C1 34802,C(=O)(C(CCN(C)C)NC(c1cnnc(O)c1)=O)N1CCC(CC)C1 34803,c1(C(CNS(=O)(=O)C2(C(C)C)CC2)OC)ccc(O)cc1 34804,C1(C(N2CC(C)C(C)(CNC(C3(C#N)CCCC3)=O)C2)=O)CC1C1CCOCC1 34805,CCC(COC)C(=O)NC1CC(CNC(=O)C=CC(=O)OC(C)(C)C)C1 34806,c1(CCC)nc(C)c(C(=O)N(C2CCCC(NC(c3cn(C)c(O)n3)=O)C2)C)o1 34807,N1(C(C)C(=O)N2CC(c3cnn(-c4ccccc4)c3)C2)CCCCC1=O 34808,C1(CC#C)CCCCN1C(C1CCCN1CCCN(C)C)=O 34809,N1(C(CC=C)=O)CCN(C(C2(C)CC2(Cl)Cl)=O)CC1.C1(NCC)CCCN(C(C)=O)C1 34810,Cc1nc(O)nc(C)c1C(=O)NC1COCCN(C(=O)CCC(=O)OC(C)(C)C)C1 34811,C12(C(=O)NCCCCCNC(C(CN(C)C)(F)F)=O)CCCN(C1)S(=O)(=O)C2 34812,c1(C(=O)NCCC(C)CO)ccc2ncc(-c3cc(F)c(F)cc3O)n2c1 34813,c1(C(=O)NCCN(CC(=O)NCC(=O)OC(C)C)CC)ncc[nH]1 34814,N1(C(c2c(OC)nccc2)=O)CCCC(N(c2cnc(C#N)cn2)C)CC1 34815,c1(C(N(C2CCN(C(=O)C(C)(C)C)C2)CCC)=O)c2c(nn1CC)CCCC2 34816,c1(C(N2C3CN(C(=O)Cc4cn[nH]c4)C(C3)C2)=O)nc2cnccc2s1 34817,C(CC(C)(C)S(C)(=O)=O)CN1CC1=O.c1(CN(c2ncccn2)C)ccccc1 34818,Cc1cn(C)cc1C(=O)NC1C=CCN(C(C23CCC(CO2)C3)=O)C1 34819,c1(Cc2ncc(C(C)O)s2)ccnc2cc(Cl)ccc12.C1(=O)CCCN1 34820,CC1(C(=O)NC2CC2NC(=O)C(c2ccc(F)cc2)(F)F)CCC(O)CC1 34821,N1(C(COCC)=O)CCN(C(C2CCCCN2C(=O)CN(C)C)=O)CC1CO.N(C)C 34822,c1(C(N2CC(C=C)C(NC(=O)COc3cn[nH]c3)C2)=O)csc2ccc(F)cc12 34823,C1(NC(C(CC=C)C)=O)CC1C1CCCN(c2ncncc2Br)C1 34824,Cn1ccc2nc(N3CCC(CC(N4CCC(CO)C(F)(F)C4)=O)CC3)ncc12 34825,C1(NC(CCCSC)=O)CC(CC(=O)NC(c2ccc(CO)cn2)=O)C1(C)C 34826,c1(NC(N=c2n(-c3c(OC)cc(Cl)cc3)[nH]nn2)=O)cccc2c1nc(O)n2C 34827,c1(C(=O)NCC2(NC(c3cncc(O)c3)=O)CCC2)c(Br)ccc2c1OCO2 34828,CC1=NNC(=O)C1CCC(=O)NCCOC1CCN(C(c2ocnc2C)=O)C1 34829,c1(CC)c(C(C)OC(c2nn(C)cc2C)=O)oc2ccccc12 34830,C1(NCc2scc(CN(C)C)n2)CCC2(CCCNC2)C1 34831,c1(C(N2CC(C(C)NC(c3cnc(CC)s3)=O)OCC2)=O)cc(O)ccc1N 34832,CC1CN(C(C2CC2c2ccc(Br)cc2)=O)CCN1S(=O)(=O)c1cccs1 34833,C=CCN=C(NCCC1CC(C(=O)NC)C1(C)C)NCC(C)(C)NC(C)=O 34834,Cc1cccc2nc(C(=O)NC(C)(C)C(C)NC(C3CNC(=O)N3)=O)cn12 34835,c1(C(N2CCC(OCCOC)CC2)C(=O)NC(C)C)cnc2cnccn12 34836,c1(C(=O)NCC(C(C)(C)C)NC(c2c(C)cc(CO)o2)=O)cc(C)c(O)c(N)c1 34837,CCC(CC)C(C)C(=O)N1CCC(C(=O)NCc2nnc(O)o2)(CO)C1 34838,c1(C(=O)NC(C2CCN(C(=O)Cc3n[nH]c(=N)s3)C2)C)cc(OC(F)F)n(C)n1 34839,C1(C(=O)NCc2c(C)ccs2)C2CC3C(C2NC(=O)C(C)C(F)F)C13 34840,c1(CCC)nsc(N)c1C(=O)NC1CC1NC(=O)Cn1cccn1 34841,N1(C(CCC2CC(NC(Cc3cc(C)sc3)=O)C2)=O)CCCCC1C 34842,Cc1ccc(CCNC(c2occc2CNC(c2scc(C)c2C)=O)=O)cc1 34843,O=C1CCCC(CC(=O)NCC(CC2CC2)C(=O)NC2CC(C(F)(F)F)C2)C1 34844,C1(NC(Cn2ncc(C#C)c2)=O)CN(C(=O)C(C)CC(F)F)C(C)(C)C1 34845,c1(CC)cnc(C)nc1N1CCC(CNC(=O)CN(C)CCOC)C1 34846,C1(CN(C)C(c2cc(CO)[nH]n2)=O)CN(C(c2cc(Cl)cn2C)=O)CCO1 34847,CC1CCC(C)(C(=O)NCC(=C2CN(C(C3CC4CCC3C4)=O)C2)F)CC1 34848,Cc1c(C)c(C)c(CSCCC(C)(F)F)c(C)c1C 34849,c1(C(=O)NCCC2N(C(CCCC#C)=O)CCC2)ccc(OC)c(C(C)C)c1 34850,c1(C(=O)NCC(C(=O)NCc2ncc(C)[nH]2)C)cncc(C#N)c1 34851,Cc1ccc(CC(CO)NC(c2cnc[nH]2)=O)nc1 34852,c1(C(N2CC(CC)N(C(=O)CC3C=CS(=O)(=O)C3)CC2)=O)nccn2ccnc12 34853,C1(CC(C)NC(=O)C#CC2CC2)CCN(C(=O)CC23COC(C)(C2)C3)CC1 34854,C1(NC(C(C)n2ccnc2)=O)CCN(C(c2ccn(O)c(=O)c2)=O)C1(C)C 34855,c1(C(N2CC(C)C(NC(c3csc(O)n3)=O)CC2)=O)cncc2c(O)nccc12 34856,C(CCC(C(=O)NCCc1cccc(C)n1)N(C)C)NC(C1C(=C)C1)=O 34857,n1(CC(=O)N(C2CCN(C(=O)C=CC(F)(F)F)C2)CC2CC2)cnnc1O 34858,Cc1cc(C(=O)NC2CCC(C)N(C(C3SC4C=CC3CC4)=O)C2)ccc1O 34859,C1(CCC)CN(C(c2cc(F)ccc2F)=O)CCN1C(c1cc2[nH]ccc2s1)=O 34860,C1(C(=O)NC(C(C)NC(c2ccnnc2)=O)C2CC2)CC(C)(c2ccccc2)C1 34861,C1(CCC)CCCCC1NC(c1csc(CNC(C2(CO)CCCCC2)=O)c1)=O 34862,CC1(CNC(=O)CCF)COCCN(C(=O)CC2=NNC(=O)C2)C1 34863,c1(NC2C(NC(C3(C)CCC(F)(F)CC3)=O)CCC2)ccc2c(n1)CCCC2=O 34864,c1(CC(=O)NCC(CO)NC(c2coc(C(F)F)n2)=O)cnc(C2CC2)[nH]1 34865,C(=O)(C1=C(Cl)CCCC1)NCC1(COC)CCCN1C(C1CC12CCC2)=O 34866,c1(C(N2CCC(COC)(NC(C3(CF)CC3)=O)C2)=O)cc(Cl)cc(C(F)(F)F)n1 34867,N1(C(C(C(C)C)C2CCC2)=O)CCC(C)(NC(c2nnc(O)nc2O)=O)CC1 34868,c1(OC)c(Cl)ccnc1NC(C1CN(Cc2ccc(F)c(F)c2)CCS1)=O 34869,N1(C(c2cn(CCOC)nn2)=O)CCC(CO)(NC(C2CN(C)CCO2)=O)CC1 34870,C(CC(C)(C)C(=O)NCCN(S(C)(=O)=O)C)OC.N1(CC)CCN(CC)CC1 34871,N1(C(=O)NC(C)C(=O)NC2CC2)CCN(C2CCCC2)C(C)C1 34872,C1(NC(c2ccc(OC)cc2)=O)C2CC(O)C1N(C(=O)Cn1cnccc1=O)C2 34873,C1(NC2C(OCC)CCCC2)CC(C2CCOC2)C1 34874,N1(C(C2(C)CNC(=O)C2)=O)CCCN(CCNC(=O)C=Cc2ccsc2)CC1 34875,CN1CCC(CC(N2CCCC(CCNC(C3CC3OC(C)(C)C)=O)C2)=O)CC1 34876,C(C(N=[N+]=[N-])C(=O)N1CCC(C)(NC(=O)CC2CCC(C)(C)O2)C1)OCC 34877,N1(C(CC2(N(C)C)CC2)=O)CC2CC(Nc3ncnn4cccc34)CC1C2 34878,Cc1cc(F)ccc1CC(=O)NC(CNC(=O)CC1CCCC(=O)N1)CC(C)C 34879,C(C(O)C(=O)NCC#CCCO)NC(=O)Cc1ccccn1 34880,c1(C(=O)NC)c[n+]([O-])c(C)cn1.C1(=O)CC(NC(C2(CSC)CC2)=O)CN1 34881,C1(CC(=O)NC(CCNC(c2c(C)nco2)=O)C(C)(C)C)CC2(CCCC2)CO1 34882,c1(NC(Cn2c(C)cnc2)=O)cccc(CNC(c2cncc(N)n2)=O)c1 34883,N1(C(c2c(N)cc(Cl)nc2Cl)=O)Cc2nccn2CC(NC(C2(F)CC2)=O)C1 34884,Cc1cc(C(=O)NCCC2CCN(C(C3C4CCCC34)=O)CC2)cc(C)c1N 34885,N1(C(c2nccc(C)c2N)=O)CCOC2CN(C(=O)CC3C=CCCC3)CC12 34886,c1(C(N2C(C)CC(CNC(CC(C)C3CCCO3)=O)C2)=O)coc(S(C)(=O)=O)c1 34887,CCCCCC(C)CC(=O)NCC1(O)CCCN(C(C2(CO)COC2)=O)C1 34888,C(CNC(c1cncs1)=O)(C(C)C(C)C)NC(c1c(C)cn(C)n1)=O 34889,C=CC1(C(=O)NCC(C)(C)CNC(c2ccn(C3CC3)c2C)=O)CCCCC1 34890,C1(NC(C2CCCCC2)=O)C2CCC1N(C(c1ccc(C(F)F)cn1)=O)C2 34891,CC(C(C)(C)C(=O)NC1(C)CCCCC1)NC(=O)COc1ccsn1 34892,CC(C(=O)N1CCN(C(=O)CN(C)CCO)C(c2ccncc2)C1)C(C)(C)C 34893,Cc1cccc(CCNC(=O)CC2CCCOC2)n1.ONC(=O)Cn1cccn1 34894,c1(C(=O)NCCCCC(CO)NC(C(C)SCC)=O)ncc2ccccn12 34895,N1(C(C(C(=O)OC)(C)C)=O)CCC2(CC1)OCCC2NC(c1ccc(C)cc1)=O 34896,C(=O)(C(C)(C)C(F)F)NCC1CN(C(c2ccc(CSCCC)o2)=O)C2CC12 34897,C1(C(C)NC(C2CNC(=O)C2)=O)CN(C(=O)CN2CCCCC2)CCO1 34898,c1(C(N2C(CNC(CN3C(C)CC3)=O)C=CC2)=O)cn(C)nc1C(F)F 34899,CC(CC(=O)NCC(O)CNC(C1(F)CCCC1)=O)NC(C1CCCC1)=O.C(N)(=O)N 34900,c1(C(=O)NCC(CNC(c2ccc(C(C)C)nc2)=O)(C)O)cc(CO)ccc1Cl 34901,N1(C(C(CCC)OC)=O)CCC(CO)(NC(=O)CCOc2ccc(F)cc2)CC1 34902,c1(CC)ccc(C(=O)N(CC(C)NC(=O)C(c2ccccc2C)C)C)c(C)n1 34903,N1(C(c2c(CC)occ2C)=O)CC(C(=O)NCc2csc(C)c2C)CCC1(C)C 34904,C(CNC(C1CC(=O)NC1(C)C)=O)(C(=O)N=c1cc(C)n(C(C)C)[nH]1)OC 34905,C(=O)(C1=C(C#N)CCC1)N1CCC(C(N(C)CC)=O)C1C(C)C 34906,c1(CNC2CC(NC(Cc3onc(C)n3)=O)C2)cccc(C(F)(F)F)c1Cl 34907,C1(C(=O)NC(C2CCN(C)C2)C)(CO)CN(C(C2CCN(S(C)(=O)=O)C2)=O)C1 34908,c1(N(C(=O)CCCC(F)(F)F)C2CNCC2F)ncnc2n[nH]c(Br)c12 34909,Cc1cc(C(=O)NCCC2CCCN(C(=O)Cc3cnc[nH]3)CC2)cc(F)c1C 34910,C#Cc1ccc(C(N2C(C(=O)N(C)OCc3ccccc3)CC3CC23)=O)o1 34911,N1(C(C(C)C(C)(F)F)=O)CC2(CCCC2CNC(=O)C(C2CCOCC2)O)C1 34912,C1(C(N2C(CCN(C(=O)C#CC3CCC3)C)CCCC2)=O)CC2(CCC2=O)C1 34913,CCC(CC(=O)N(C)CCOCCC(N1CC=CC1C(=O)NC)=O)OC 34914,Cc1ccccc1CCC(=O)NC1(CNC(=O)C(C)C#N)CCCC1 34915,CC(C)S(=O)(=O)C(C)C(=O)N1CC(O)(CN(C(=O)CCCCNC(N)=O)C)C1 34916,c1(C(=O)NCCCCNC(=O)C(c2ccccc2)F)cn(C2COC2)nn1 34917,c1(OC)cc(Cl)ncc1C(=O)Nc1c[nH]nc1C(=O)Nc1cc(I)ncn1 34918,CC1CC2CN(C(c3cccnc3O)=O)CC2N1C(=O)CCCC1CCCO1 34919,C1(C(N(C(CNC(C(Cc2ccccc2)OC)=O)C)C)=O)CCC(=O)N1C 34920,N1(C(Cc2cc(C)on2)=O)CCCC(C)(CNC(=O)C(C2CCOCC2)C)C1 34921,c1(C(N2C(C3CN(C(=O)C=CC4CCOC4)C3)CCCC2)=O)ccc2ccnn2c1 34922,CCC(F)(F)CC(=O)NCC1CC1NC(=O)C(c1ccnn1C)O 34923,c1(C(=O)NC2CCCC(C(=O)NC3CC3)CC2)cccn2nccc12 34924,C1(C2CCN(C(c3c(C)noc3C3CC3)=O)C2)(NC(C2CC(CCC)C2)=O)CC1 34925,C(=O)(C(C)(C)C(F)(F)F)NC(C(=O)Nc1c(Cl)ccc(OC)n1)C 34926,c1(C(=O)NCCOC2CN(C(C3CC34CCCOC4)=O)C2)cn2cccnc2n1 34927,CCC(C)(CNC(c1cc(C)c(F)cn1)=O)C(=O)NOCC=CCl 34928,c1(SC)ccc(C(=O)NCCC2CCCCN2C(=O)C(Cl)=CCl)c(Cl)c1 34929,C1(CC)(CC)CC(C(=O)NCCCOCCC(=O)NCC2CCCOC2)C1 34930,CCC(C)CCC(O)CC(=O)NC1(C)CN(C(c2csnc2OC)=O)C1 34931,N1(C(Cc2ncc(CC)[nH]2)=O)CC(C)(C)CC1CNC(C1CC(O)CN1C(C)=O)=O 34932,C1(N(C(c2c(C)cc(C#N)s2)=O)C)CCCCC1S(C)(=O)=O 34933,c1(COC)ccc(C(=O)NCCCN(C(=O)C=C(C)C2CC2)C)o1 34934,N1(CCCCOC)CCN(C(=O)NCCCC(C)(F)F)CC1 34935,Cc1nn(C)c(C)c1CC(=O)NC1CN(C(C2CC2F)=O)CC1C 34936,Cc1nc(=NC(=O)C2CCCN(CC(C)C)C2)n(-c2cccc(C#N)c2)[nH]1 34937,N1(C(COCCOC)=O)CCC1CNC(c1cnsc1)=O 34938,N1(C(C=CCN(C(c2c(CC)con2)=O)C)=O)CCC12CCCSC2 34939,C(C(C)(C)CCC=C)NC(CCC=CC)(C)c1nnnn1CC(F)F 34940,N(C(=NCCc1cccc(C#N)c1)NCc1cc(C)c(CC)s1)C(C=C)C 34941,N1(C(CC(C)c2cnn(C)c2)=O)CC(CNC(=O)CC(O)CC2CC2)C(C)C1 34942,C1(C(N2C(CC(=O)NCc3ccccc3F)CC2)=O)Cc2ccccc2C1 34943,O=C1CCN(C(=O)CCc2ccc3ccccc3n2)c2ccccc2N1 34944,C1(C2CCN(C(=O)CC(Cl)Cl)C2)(NC(C(C)O)=O)CC1 34945,C=CC(C)(CC)C(=O)NCCC(F)(F)Cn1cc(C2CC23CC3)nn1 34946,c1(C(=O)NC2C(OC)CN(C(=O)CC(F)F)C2)cc(S(N)(=O)=O)c(F)c(F)c1F 34947,c1(C(=O)NC(CCNC(CC2CCC(C#N)C2)=O)(C)C)cc(F)cc([N+](=O)[O-])c1 34948,C1(C2CCN(C(=O)CNC3CC3)CC2)(NC(c2c(C)ccc(F)c2O)=O)CCC1 34949,Cc1nc(Cl)[nH]c(=NC2CC(CNC(c3cncnc3C3CC3)=O)C2)c1F 34950,c1(C(C(=O)NCC)N(C)Cc2cccc([N+](=O)[O-])c2)cnc2c(c1)c(C)nn2C 34951,C1(C(=O)NC23CC2CN(C(c2ccsc2Cl)=O)C3)CCCC1C1CC1 34952,Cc1[nH]nc2cc(C(N3CC4(C3)CN(C(c3coc(C(N)=O)c3)=O)C4)=O)ccc12 34953,C(=O)(CC(C)(C)OC)N(CCCNC(c1csc(-c2cn[nH]c2)n1)=O)CC 34954,C(=O)(C(O)(c1ncnn1C)SC)NCC(CC)NC(=O)C(C)(C)c1ccccc1 34955,Cc1cc(=O)cc(C)n1CCCC(=O)NCC(C)CNC(=O)C(C)c1cccs1 34956,CCCC(CNC(C1Cc2nccn2C1)=O)C(=O)NOCC(C)CC 34957,c1(C(C)NC(=O)CNC2C=CC(C(=O)NC3(c4cccs4)CC3)C2)ccccc1 34958,C1(CNC(C(C#C)(C)C)=O)CN(C(=O)CCn2ccnc2)CC(C)(C)O1 34959,CCCC(C)CCCC(=O)N1CC=C(CNC(=O)C(CC)OC)CC1 34960,C1(C(=O)NCC2CCC(C(=O)N(C)Cc3c[nH]nc3C)CC2)(OC)CCCOC1 34961,N1(C(=O)CC2CCC(F)(F)C2)CCC2CN(C(c3ccc(Cl)cc3Cl)=O)CC2C1 34962,c1(C(=O)NCC2(CNC(=O)CCOCC3CC3)CCC2)occ2c1CCCC2 34963,c1(CC)noc(CC)c1CC(N1CC(NC(=O)CC2CCCCO2)C(O)C1)=O 34964,C1(NC(C=CSC)=O)CCC2CC1CN2C(=O)CC1CCOC(C)(C)C1 34965,Cc1nc(C(C)C)nc(O)c1C(N1CC2(COC(CNC(C3CCO3)=O)C2)C1)=O 34966,C1(NC(C(C2CC2)SC)=O)CCCC1NC(=O)Cn1ccc(Br)n1 34967,CC(C)CC(F)(F)C(=O)N1C2CCC1CC(CNC(C1CCCCC(=O)N1)=O)C2 34968,C#CCC(C)(C(=O)NCCC1CC1C)NC(c1cc(C#N)cs1)=O 34969,C1(C(N2C(C)CC2)=O)CCc2ncnc(C)c2C1.C1(N2CC(=O)N2)CCCC1.CO 34970,CCCCCCC(F)C(=O)NC1CC1CNC(c1ccon1)=O 34971,C(C1=CCN(C(=O)C(c2ccc(F)cc2)F)CC1)NC(C(CC)N(C)C)=O 34972,CC1=C(C(=O)N2CC3(C(=O)NCC4CCCCN4C)CC2CO3)CCCO1 34973,CC1C(NC(=O)CCC2CCC(C)O2)CCCN1C(c1cn(C)c(=O)n1C)=O 34974,C(=O)(CC1c2ccccc2C(=O)N1C)NCCCCNC(CC1CC(SC)C1)=O 34975,Cc1ccc(C(C)CC(N2CCC(C)C2CNC(C2CCCC(=O)N2)=O)=O)cc1 34976,S(=O)(=O)(c1ccc(=NCCS(=O)C(C)(C)C)[nH]c1)NCc1nc(C)sc1 34977,c1(-c2cn(C3CN(C(CCC)=O)CC3O)nn2)cc(Cl)cc(F)c1Cl 34978,Cc1cc(C(N2CC(C)CCC2CNC(c2cn(CC)nn2)=O)=O)c(C)nc1C 34979,C(C)(C(O)C(=O)NCc1nnc(-c2ccc(C(F)(F)F)cc2)o1)OC 34980,C(=O)(C1=CCCC1C)N1CC2(C(C(=O)OCC)C2)C1.CCSC 34981,C12(C(NOCCOCC#C)=O)CC(CN(C(=O)CC3C=CCC3)C1)C2 34982,CC1CCN(C(C2(CF)CC2)=O)CC1NC(C1CCN(C2CC2)CC1)=O.C(C(F)F)N 34983,CC1CN(C(=O)CCc2nc[nH]n2)CC1NC(C1(F)CCCOC1)=O 34984,C12(COC)CC(NC(=O)Cc3cccnc3)(CN1C(=O)CN1CCSCC1)C2 34985,C12(CC(=O)NC(CNC(C(C)(C)F)=O)C(C)(C)C)CC3CC(C1)CC(O)(C3)C2 34986,CCCC(C(=O)NOC(CO)C(C)C)NC(=O)C(F)F 34987,c1(C(N2CCC(N(C)C(C3CCCCCCC3)=O)CC2)=O)c2c(nn1C)CCSC2 34988,c1(C(N(c2ncc(CCC)cn2)C2CC(N)C2)=O)cc(C(F)(F)F)ccc1F 34989,c1(C(=O)NC(CN(C(C(C)SCCCC)=O)CC)C)cnc(CC(C)C)[nH]1 34990,C1(OC)C=CCN(C(C2(C(C)NC(c3cocc3C(N)=O)=O)CC2)=O)C1 34991,Cc1cnc[nH]c1=NCCCC(C)NC(c1cnn(CCN(C)C)c1)=O 34992,c1(NC2C(C)CCN(C(c3c[nH]c(C(N)=O)c3)=O)C2)ncnc2sccc12 34993,C1(C(=O)NC(CCCCC)C)CN(C(C2(O)CCOCC2)=O)CC12CC2 34994,c1(CCC(=O)N(c2cccc(CCC)n2)C2CC3CC2CN3)ccc(F)cc1Br 34995,c1(C(=O)NCC2(CC)CC2)occc1CN(C(C1CCN1C(C)(C)C)=O)C1CC1 34996,N1(C(C2C(CN(C)C)C2)=O)CC2(C1)C(NC(=O)C=CCO)CCS2(=O)=O 34997,C=CCC(C)(C)CC(=O)NC1CCCC1NC(=O)C=C(C)C1CC1 34998,CCC(CC(=O)NC(CCOCC)C(=O)N1CCC=C(Br)C1)C1CC1 34999,c1(OC)cc(Cl)cc(N)c1C(=O)NCC(N1CCCCC1C)C 35000,C1(C(N(C)Cc2ccns2)=O)CCC(C2CC2)N1C(c1ccc(C#N)s1)=O 35001,c1(C(N2CCC(C#N)C2)C(=O)NCc2cccc(Br)c2)ccc2ccccc2n1 35002,CCCCCC(O)C(=O)NCc1cc(-c2ccc(C#N)cc2)nn1C 35003,C1(CN(C(=O)Cc2sccc2C)CC)CCCCN1C(=O)CN1CCC(F)(F)C1 35004,c1(C(N2CCC(CCNC(C(C)CC(F)F)=O)C2)=O)cccc2c1CC(=O)N2C 35005,C1(OCCCNC(CC(=O)NCC#C)=O)CCN(C(=O)C(C)COC)CC1 35006,N1(C(C2(CC)CCC2)=O)CC2CC2(CNC(=O)C(C)Sc2ccc(OC)cc2)C1 35007,c1(C(C)C)ccc(C(=O)Nc2cccc(NC(=O)CCC3CNC(=O)N3)c2)cn1 35008,Cc1oc(-c2ccccc2F)nc1C(=O)NCC(O)CN(C)C(c1cncs1)=O 35009,C(=O)(NNC(=O)Cc1ccccc1C(F)(F)F)c1c(C)ccs1 35010,Cc1c(C(=O)NC2CN(C(=O)CC(C)NC(N)=O)CC2F)cnc2ncnn12 35011,N(C1CCCc2c1cnn2Cc1ccccc1)Cc1cc(C)cc(I)c1 35012,C(=O)(C1CCSc2ccccc21)N1C(C)CCN(C(c2cnn[nH]2)=O)CC1 35013,c1(C(N2C(C(N3CCC(C(C)(C)O)CC3)=O)CC2)=O)cc([N+](=O)[O-])n[nH]1 35014,C1(NC(C2CCC(NC(CCC3C(C)C3)=O)C2)=O)CC2CC1CC21CC1 35015,C(CC(C)C(=O)OC(c1ccc(Cl)cc1)C(F)(F)F)=CCC 35016,C(=O)(CC(C(F)(F)F)NC(=O)Cc1ncccc1F)N1CCC(F)(C(N)=O)C1 35017,O(NC(=O)C(C1CC=CCC1)NC(C1C2CCC(F)C12)=O)CC(C)(C)O 35018,c1(NC(C2C(C(=O)Nc3c(C#N)ccs3)C2)=O)cccnc1[N+](=O)[O-] 35019,N1(C(Cc2c(C)non2)=O)CC2(CCC2NC(=O)Cc2cc(Cl)cc(Cl)c2)C1 35020,c1(N(C2CC(N)C2)C(c2c(F)ccc(Cl)c2Cl)=O)ncnc2cc(Br)sc12 35021,CCCC(C)CCCC(=O)NCC1CN(C(c2cc(Cl)nnc2O)=O)CC1(C)C 35022,CC1CN(C(=O)NCC2CCCCC2)CC(C)N1C(c1csc(Cl)c1Cl)C(=O)O 35023,Cc1cc(C=CC(N2CC(F)CC2CNC(=O)C(C)OCC2CC2)=O)on1 35024,C(C(C)S(N)(=O)=O)NC(C1N(C(C2C(C(C)C)OCC2)=O)CCC1)=O 35025,c1(OC)ccc2ccccc2c1NC(C1CNCCN1Cc1cncs1)=O 35026,C(=O)(CCC(C)(C)[N+](=O)[O-])N1CCC(CNC(C2(CC)CC2(F)F)=O)C12CC2 35027,N1(C(C(COC)OC)=O)CCN(C2CCCN(C(=O)C=C(C)C(C)C)C2)C(=O)C1 35028,C12(C(=O)NCC3CCN(C(c4cccnc4S)=O)C3)CCC(O1)c1ccccc12 35029,C1(NC(C2(CC)CCC2)=O)CN(C(=O)C(C)CSC)CCC1CO 35030,N1(Cc2ccc(N(S(CC)(=O)=O)CCC#N)cc2)CCC(C(F)(F)F)C(F)(F)C1 35031,c1(CC)cc(C(=O)NC2CC2CNC(c2cncc(N)n2)=O)cc(O)n1 35032,CCC(C)C(=O)C(=O)NC1COCCC1C(=O)N(CCC(N)=O)CC 35033,N1(C(CNC(C2C(C)C2)=O)=O)CCC(C(=O)N(C2CSC2)C)(CF)C1 35034,c1(C(=O)NCC2C(N(C)C)CN(C(CC3C(CC)C3)=O)C2)c(Cl)ccnc1C 35035,S(=O)(=O)(c1c[nH]c(=NCCN(C)C2CC2)cc1C)NCC1CCN(C(CC)C)C1 35036,C12(C(=O)NC3C(OC)CN(C(C(CC=C)C)=O)C3)CC3(F)CC(F)(C1)CC(F)(C2)C3 35037,Cc1cc(C(=O)NCCCC2(NC(=O)C(C)N3CC(C)C3)CC2)ncn1 35038,c1(C(=O)NCCOC2CCCOC2)c(F)cc(Cl)cc1Cl 35039,c1(OCC)ccc(Cl)cc1C(=O)NCCOC1CN(C(c2cc(C)sn2)=O)C1 35040,c1(OC)ccc(F)cc1CC(N1CC(NC(c2cn(C)cn2)=O)C(C)C1)=O 35041,c1(C(=O)NC2(CNC(C(C)CCN(C)C)=O)CC2)csc2ccccc12 35042,c1(C(=O)NCC2N(C(c3c(Cl)c(C)n(C)n3)=O)CC2)cncc2c1CCCC2 35043,N(C1CCOc2ccc(O)cc21)C(c1c(C)cco1)C 35044,Cc1ccc2c(c1)C(=O)N(CC(=O)NCC1COCCN1C(=O)C=C1CC1)C2=O 35045,N1(C(c2cccc(OC)n2)=O)CC=C(C(=O)Nc2cncnc2O)C1 35046,n1(CCOC(C)C)nc(Cc2ccccc2Br)nc1-c1cncn1C1CC1 35047,N1(C(C(=O)C(=O)C)=O)CC(CO)OC(C)(C)C1.c1(NC)ccccc1 35048,N1(C(c2ccc(CCC)cc2)=O)CCCC(C)(NC(C2CCC3CC2CO3)=O)C1 35049,CCCCC(CNC(c1cc(C)cs1)=O)NC(=O)CC(c1ccccc1)N(C)C 35050,C1(NC(CC2CC(C)(C)OC2=O)=O)CN(C(c2ccnc(O)c2)=O)C2(CCC2)C1 35051,Cc1noc(CCNCc2ccn(CC(=O)OC(C)(C)C)n2)n1 35052,C(CN=c1[nH]c(=NCC2(C(F)(F)F)CC2)[nH]c2cccnc12)c1ccc(C)nc1 35053,C(CCCC(=O)N1CC(O)CC1C)NC(c1c(CCC)[nH]cc1)=O 35054,C1(C(=O)NC2CCN(C(C(=C(C)C3CC3)F)=O)C2C)CC(C(C)C)=NO1 35055,C1(C(N(CC(C)(C)NC(COCCCC(C)C)=O)C)=O)CCCCC1(F)F 35056,N1(C2CCN(C(CC3C(C)C3)=O)CC2)CCC(NC(C2(CN(C)C)CC2)=O)CC1 35057,N1(C(C2C(CCC)C2)=O)CCC(O)C(N(C(=O)CC2CCN(C)C2)C)C1 35058,c1(OCC)nccc(C(N2CCC2CNC(c2nc(C)n(C)c2C)=O)=O)c1F 35059,CC1CC(c2ccc(Br)cc2)CN1C(=O)Cc1cncs1 35060,N1(CC(CC)CC)CCC(NC(=O)CCCc2ccccn2)C(O)C1 35061,C(=O)(CC(C)C(=O)OC)N1CCC(NC(c2cc(CC)ncc2)=O)(COC)C1 35062,c1(NC(c2c(C(C)C)nns2)=O)ccccc1I 35063,c12cc(Cl)nnc1[nH]c1ccc(cc1)[nH]c2=O.C1(SCCO)CCCCC1 35064,C1(C(=O)NCC(CC)NC(=O)N(C)C)CC(O)CN1C(=O)Cc1ccc(C)cc1 35065,C1(C)(NC(c2cn(CCN(C)CC)nc2)=O)CCCN1C(=O)CCc1ccsc1 35066,c1(C(=O)NC2C3CN(C(c4ccc(C(C)=O)cc4)=O)CC32)c(F)cc(F)cc1Cl 35067,N1(C(C(CSC)(C)C)=O)CCC(CNC(C2CCCC(CF)C2)=O)C(O)C1 35068,c1(C(N(CC(CNC(C(C)SCCCC)=O)C)C)=O)ccc(-n2ccnn2)cc1 35069,c1(C(N2C(CC(=O)NCC(C)C3CC3)C3CCCC32)=O)cc2ccccc2o1 35070,CC1CCC=C1C(=O)N1CCN(C)CC1CNC(=O)CN1CCOCC1=O 35071,c1(C(C)=O)cccc(NC(C2CCC(NC(=O)CCN3CCCC3)CC2)=O)c1O 35072,O=C(O)CCC(F)(F)C(=O)N1CC2CC1CN2Cc1ccc(F)cc1 35073,c1(C(=O)NC(C)CNC(=O)C(C)N2CCCC2)cc(Cl)cc(Cl)c1 35074,N1(C(CCOCCC)=O)CCCC2CN(C(c3cncc(NCC)c3)=O)CCC12 35075,C=CCC(C)C(=O)N(C1CCCN(C(=O)C=C(CC)CC)C1)CCF 35076,c1(OC)cc(C(=O)NC(C)CC(C)NC(c2cnn(CCO)c2)=O)ccc1Cl 35077,C1(C(N2CCC(O)(COC)C2)=O)COCCN(C(=O)CN(C(=O)C(C)C)C)C1 35078,C1(C(=O)NCC2N(C(c3c(OC)nsc3)=O)C3C(C2)C3)Cc2ccccc2S1 35079,C1(CN(C(C(C2CCCC2)NC(C(C)=C(C)C)=O)=O)C)C(C)(C)C1(C)C 35080,CC(C(=O)N1CCC(O)(CN(C(=O)C(C)(C)C)C)C1)C(F)F 35081,C(=O)(C(F)(F)C(C)O)NC(C)CCCNC(c1cc(F)cc(Cl)c1)=O 35082,c1(NCCOCCOCCOC)ccc(-n2cnnn2)cn1.C1CCO1 35083,C=C=C(C)CC(=O)NC1(CC=C)CCN(C(c2cnn(C(C)CC)c2C)=O)C1 35084,C(CC(C)(C)C(=O)NCC(N1CCOCC1)=O)NC(C=CC=CC)=O 35085,c1(NC(C2C3CN(C(CCCC(C)C)=O)CC32)=O)cc(Cl)c(Cl)cc1C#N 35086,N1(C(c2cnn(C3CC3)c2)C(=O)NCC2CCCO2)CC2CC(O)C(O)CC2C1 35087,c1(OC)ccc(CNC(=O)Nc2ccnn2-c2c(F)cccc2F)c(O)c1 35088,C1(C(=O)NCCCC2CCCN2C(=O)CN2CCSCC2)CCCCCC1(F)F 35089,N1(C(C2CC(C)SCC2)=O)CCN(C(=O)Cn2cccc2)CC1CO 35090,c1(NCc2nc3ccc(OC)cc3[nH]2)[nH]c(=NCC2CC2)nc2ncn(C)c12 35091,c1(OCCCC)c(C(=O)N(CC(C)C)Cc2cnc(C)nc2C)cccc1Br 35092,C(C)(CC(=O)NC1(CCC(=O)NCC(O)CCC2CC2)CCCC1)=C(C)C 35093,Cn1cncc1C1CC1NC(=O)CC1(C)CCN1C(=O)CNC1CCC1 35094,C1(NC(C=C(C)C(C)C)=O)CCN(C(=O)C(C)SC(F)(F)F)C1C1CC1 35095,N1(C(CCN(C(C)=O)C)=O)CCC(CN(C(=O)C(F)(F)c2cnccn2)C)CC1 35096,N1(CCC)CCCCC1C(=O)N(C(CNC(=O)CSC(C)C)CC)C 35097,CCC(CC)CCCC(=O)N1CCC2CN(C(c3cccc(Cl)c3)=O)C2C1 35098,N1(C(C(C)C(F)F)=O)CCC(C)(NC(c2cc(C3CC3)cc(F)c2)=O)CC1 35099,Cc1ccc(CCCC(=O)NC2CCCC2CNC(=O)Cc2cn(C)nn2)s1 35100,C1(C)(CNC(CNS(CCOC(C)C)(=O)=O)=O)CCCN1C(=O)CSC(F)F 35101,N1(C(c2c(C)noc2)=O)CCN(C(=O)CCn2cccn2)CC1CO 35102,C(=O)(C1=CS(=O)(=O)CCC1)NCC1CN(C(c2c(SC)scc2)=O)C(C)CC1 35103,CCC(C)CC(C)C(=O)N1CCC(F)(CNC(=O)CC2(C(F)F)CC2)CC1 35104,c1(CC(=O)Nc2ccc3c(c2)OCC3)noc2ccc(Cl)cc12 35105,N1(C(C(C2CCCCC2)C)=O)CCCC1(C)CNC(C1(CCF)CCOCC1)=O 35106,C1(CNC(C(N2CC(C)C2)C)=O)(CNC(C2(C)CCSCC2)=O)CC12CCC2 35107,c1(C(=O)NCC2(OC)CN(C(c3cc(C)ncc3C)=O)C2)ccn(O)c(=O)c1 35108,C1(C)(C(=O)NC2CCC(N(C(c3ccc(CC)[nH]3)=O)C)C2)CCC(C)(C)CC1 35109,C(=O)(C(CO)C(C)(C)C)NCc1c(C(=O)NCC(C(=O)NC)(C)C)occ1 35110,C1(NC(c2c(C(C)C)n[nH]c2)=O)CCCN(C(=O)C(C2CCC(=O)N2)C)CC1 35111,c1(C(=O)OC)cc(F)c(Br)c(S(=O)(=O)NC(=O)COc2ccc(C)cc2F)c1 35112,O=C(CCCNC(c1cccnc1)=O)NCC1CN(C(c2cc(Cl)c[nH]2)=O)C1 35113,c1(CN(C)C)c[nH]c(C(=O)NC2CC2NC(=O)COCC2CCCO2)c1 35114,N1(C(C2(COC(C)C)CC2)=O)CC(C2CCCCN(C(C3COCCO3)=O)C2)C1 35115,c1(C(=O)NC2CC(NC(c3cn(CC)nc3C(F)(F)F)=O)C2)nnc(O)cc1O 35116,N1(Cc2c(C)cccn2)CC2(CN(C(c3ccc(Br)cc3CO)=O)CCO2)C1 35117,C(=O)(CCCCC(=O)NC1CN(C(=O)CSc2nnnn2C)CC(C)(C)C1)NC 35118,N1(C(COCCNC(C(C2CCCCC2)C)=O)=O)CCC2(CC(F)C2)C1 35119,N1(C(C2C3(CC(OCC)C3)C2)=O)CCC(O)(C(=O)NC)CC1 35120,CC(C)CCCOCC(=O)NCC(C)N(C(=O)CC1CCN(C)C1)C 35121,N1(C(C(C)(C)NC(=O)NCC)=O)CC(NC(c2nnccc2C)=O)C(C)(C)C1 35122,C12(C(=O)NC3(C(F)F)CCOC3)CC(CNC(CCOCC)=O)(C1)OC2C 35123,O=C(CCCC(F)(F)F)NC1CC(O)CN(C(=O)COC2CCOC2)C1 35124,c1(OCC)oc2ccccc2c1C(=O)NCC(CC)NC(C1CC2(C1)CC2F)=O 35125,c1(NC(=NCC2C(C)CC(C)C2O)N(C)C)ccc2cccnc2c1 35126,c1(C(C(=O)NC2CCOC2)N(C(C)C)CC2CCCO2)nc2c(s1)CC(C)CC2 35127,CCCCCCC(C)C(=O)NC(C(=O)NC1CC(F)(F)C1(C)C)C(C)C 35128,C12(C(N(CCC(=O)NC(CC=C)C3CC3)C)=O)COCC1C2 35129,N12CCCCC1Cc1nccc(c1)C2=O.CC(C)(C)C(O)c1cn(COCC=CC)nn1 35130,C1(CNC(C2CC(OC)C2)=O)COCC1NC(=O)CCOc1cccnc1 35131,CN=c1ccc(C(=O)NCC(C2CCN(C(=O)CC3CCC(C)C3)CC2)O)c[nH]1 35132,c1(OC)cc(C2(C(N3CCCC(C)(NC(=O)CCC(N)=O)C3)=O)CC2)ccc1C 35133,c1(C(N2CC(CC=C)(NC(c3ncc[nH]3)=O)C2)=O)cnn(C(C)C)c1C 35134,N1(C(c2cccc(Cl)c2)=O)CC(C2CCCN(C(C3CCCCS3)=O)C2)C1 35135,c1(C(=O)NC(Cn2c(CC)ncc2)C)ccc(Br)cc1N=[N+]=[N-] 35136,c1(NC(N2CCOC(C3CCCOC3)C2)=O)cc(F)c(N2CCC2)c(F)c1 35137,C1(F)(C(=O)OC)CN(C(=O)CONC(c2cccnc2)=O)C1 35138,N1(C(C(CC)OCC)=O)CC(N=c2nc(C(C)(C)C)[nH]s2)CC(C)(C)C1 35139,N1(C(C=Cc2c(C)nsc2)=O)CCCC2(NC(=O)CSC(C)C)CCCC12 35140,N1(C(C2N(C(C)=O)CC(O)C2)=O)CC(NC(c2[nH]cnc2C)=O)CC(C)C1 35141,N1(C(COCC=C)=O)CC2CCC(C1CO)N2C(c1ccc2c(n1)CCCC2)=O 35142,c1(C(N2CCC(NC(C(C)OCCCC)=O)C2)=O)ncccc1C(F)F 35143,[N-]=[N+]=NCC(C(=O)NC1(C2CC2)CC1)NC(=O)Cc1cnoc1 35144,C12(NC(CCc3c(C)cccc3)=O)CCN(C(=O)CCOCC3CC3)CCC1C2 35145,C#CCCC(C(=O)NCC(C)C#N)NC(=O)CCCCCN(C)C 35146,n1(CC(=O)NC2C(CNC(CN(C3CCC3)C)=O)C2)cnc(Br)n1 35147,C1(NC(C(C)C)=O)CCCC12CCN(C(=O)C(C)CS(C)(=O)=O)CC2 35148,c12ccc(Br)c(c1)CS(=O)(=O)N2.N1(CC)CC(=O)N(CC(=O)OC(C)(C)C)C1=O 35149,O=S(=O)(c1cccc(F)c1F)N1CCC(OCc2ccccc2)C1 35150,c1(C(=O)NCCCC(=O)NCC2CCC(=O)NC2)c[nH]nc1[N+](=O)[O-] 35151,N1(C(c2cnc(COC)s2)=O)CCN(C(=O)CC2CN(C)C2)C(C)CC1C 35152,N1(C(COCCC=C)=O)CC2(CC2)CC1CNC(=O)CSCCC(F)(F)F.C(CCC)O 35153,C(=O)(C1=CCCSC1)NC(C(C)(C)NC(C1CCCN(CCC)C1)=O)C 35154,Cn1ccc(C(N2CC(C(=O)NCC=CCl)CC2(C)C)=O)cc1=O 35155,C1(C(=O)NCC2CCN(C(CC3C(C)(C)C3)=O)CC2)CCOC2(CCOCC2)C1 35156,CC1(C)CC(O)(C(=O)NCC(C2CCCC2)NC(=O)CC2CCCOC2)C1 35157,C1(C(=O)NCc2cc(C(=O)NCC3(C)CC3)n[nH]2)(OC)CCC(C)C1 35158,Cc1cc(F)c(C(N2CC3CN(Cc4cncc(C)n4)C3C2)=O)c(F)c1 35159,Cn1nc(C(=O)NC2CCCC2NC(C2CCC3CC23)=O)c2c1CCC(C)(C)C2 35160,N1(C(C(CC)C)=O)CC2CCC(C(=O)NCCc3ncn(C)n3)(C2)C1 35161,Cc1nccc(C(=O)NC2(CNC(C34CC5CC3C4C5)=O)CCOC2)c1N 35162,N1(C(C)C)CCCC1C(N1CC(CN(C)C(c2nccn2C)=O)C1)=O 35163,c1(CC(=O)NC2CN(C(CC(c3c(C)n[nH]c3C)C)=O)C2)c(F)cccc1Cl 35164,S(C1CCc2c(F)ccc(F)c21)CC(CNC(N)=O)O 35165,C1(C(N2CC3CCN(C(C4CC(OC)C4)=O)CC23)=O)CC2(CCC(CO)CC2)C1 35166,C(CC(C(=O)N1CCC(C(=O)OC)C1)NC(=O)COCc1nc[nH]n1)=CC 35167,CCCCCC(C)CC(=O)N(C(CNC(=O)CN1C(=O)C(C)C(C)C1=O)CC)C 35168,CCC(C)C(O)C(C)C(=O)N1CCC(N=[N+]=[N-])(C(N2CC3C=CCC(C3)C2)=O)C1 35169,CCC(C)(C)C(C)CC(=O)NC1(CNC(=O)C=Cc2cc(Cl)ccc2Cl)CCC1 35170,C1(CNC(C2CCC(CC)O2)=O)CC(NC(c2cnc[nH]2)=O)CC1O 35171,N1(C(=O)CN2CCCC2)CC2CN(C(c3cccc4cc[nH]c34)=O)CC2C1 35172,N1(C(CC(COC)C)=O)CCCCC(CNC(=O)C=C2CCC(C)(C)CC2)C1 35173,N1(C(c2c(C)cccc2F)=O)CC(NC(=O)Cc2ccon2)CC2(CC2)C1 35174,CCCCCCC(F)C(=O)N(C)CC1CCCN1C(=O)CC12COC(CF)(C1)C2 35175,c1(C(=O)NCC2N(C)CCN(C(=O)C=C3CCC3)C2)cnn2ccn(C)c12 35176,C=CCCCCC(=O)N1CCC(OCC(=O)NC(CCF)C(=O)OC)C1 35177,C=CCC(CC)C(=O)NC1CC(C(=O)N(C(C)C(N)=O)C)CC1O 35178,c1(CO)cc(C(F)(F)F)ccc1Nc1n[nH]c(-c2ccccc2)n1 35179,Cn1nccc1C(=O)NCCC(O)CNC(c1c[nH]c(Br)c1)=O 35180,CC1CCN(CCCOCCCCCCNC(=O)Nc2cccc(CO)c2)CC1 35181,CCC(CCCC(=O)N1CCCCC1CCO)NC(=O)C(C)(C)SC 35182,Cc1nn(C)c(C)c1CNc1nccc(SCC(=O)N(C(C)(C)C)C(C)C)c1F 35183,N(C(=S)N1CC(CO)CC(C)C1)c1ccc(OC)c(Cl)c1 35184,CC(C)CC(CNC(=O)C1=CCCCO1)C(=O)NC(C1(O)CCCC1)(C)C 35185,S(=O)(=O)(c1cc(C(=O)NC2(CCNC(c3cnsc3C)=O)CCC2)co1)NC 35186,c1(CC(=O)NCC2C=CC(NC(C3C(C(C)C)(COC)C3)=O)C2)nc(C)c(C)s1 35187,C1(C(=O)NCC2N(C(C(C(=O)OCC)(C)CC)=O)CC2)CCc2ncnc(C)c2C1 35188,C1(C(=O)NCCOCCC(=O)N(CCC#C)CCO)C(C)(C)C1(F)F 35189,C(C1=NOC2COCC12)NC(CCN(C(=O)CCCC1CCC1)CC1CC1)=O 35190,CC1CCC(CO)N(C(=O)NN2CCC(c3ncc[nH]3)CC2)C1 35191,Cc1cccc(-c2cccc(NC(C3CC(C)N(c4ccccc4)C3)=O)c2)c1 35192,C12(CNC(c3c(CC)noc3)=O)CCCN(C(c3c(C)n[nH]c3C)=O)C1C2 35193,c1(C(N2CC3(CCN3C(C3(F)CCCCC3)=O)C2)=O)ccc(Cl)c(F)c1F 35194,c1(OCCN(C(=O)C(=O)N(CCC(F)(F)F)CCN)C)ccc(Br)cc1 35195,C1(CC(N2CC(C3CC3)C2)=O)CN(C(C2(O)CC2)=O)CC12CC2 35196,N1(C(c2cc(C)ncc2)=O)CC2CN(C(c3ccc(Cl)cc3F)=O)C2C1 35197,N1(C(C(CO)N(C)C)=O)CCC2(C1)CN(C(=O)CS(=O)(=O)C(C)(C)C)CCO2 35198,N1(C(c2ccn(C)n2)=O)CC2CC1C2NC(c1cccc(-n2cncn2)n1)=O 35199,c1(OCC)cc(C(N2CCC(CCNC(=O)Cc3cc(C)ns3)C2)=O)[nH]n1 35200,N1(Cc2c(OC)cco2)CCCC(NC(c2cnc(Cl)cc2I)=O)CC1 35201,C(=O)(C(C)(C)CC(F)F)NCc1c(C(=O)NCC(C#C)OC)con1 35202,c1(CN2C(CN(c3ccccn3)C)C=CC=CC=C3C(CCN3C)C2=O)ccccn1 35203,C(=O)(C(O)C(F)(F)F)N1CCC(CCC2N(C(C=CC)=O)CCC2)CC1 35204,c1(N2CC(C3N(C(C(C(C)C)F)=O)CCCC3)C2)ncnc2cccc([N+](=O)[O-])c12 35205,c1(C(N2C(CNC(CSCC)=O)CC(C)CC2)=O)n[nH]c2cc(C)ccc12 35206,N1(C(C2(COC)CCC2)=O)CC2CCC1C2NC(=O)CCc1ccc(Cl)cc1 35207,C1(CNC(C(c2ccc(F)cc2)OC)=O)CN(C(c2ccc[nH]2)=O)C(C)(C)C1 35208,C1(N(C(=O)CCc2nncs2)C)CN(C(c2cnc(N)c(N)c2)=O)CC12CC2 35209,C(C1OCc2ccccc21)S(C)(=O)=O.n12nnnc1CNC1CC2C1 35210,C1(NC(CCCCOC)=O)CC2(C1)CN(C(=O)CC1C(C(=O)OC)C1(C)C)C2 35211,C1(C)(CNC(C=CC(C)C)=O)CCC(NC(C2CC3(C2)CC(F)C3)=O)CC1 35212,C1(NC(C2C(C)CCS2)=O)CCC(NC(=O)C(C)(C)c2ccc(Cl)s2)CC1 35213,c1(NC(C2CC(C)CN2C(c2c(O)cccc2O)=O)=O)cccc2sccc12 35214,N1(C(c2c(CC)[nH]cc2)=O)CCCC(NC(c2csc(S(N)(=O)=O)c2)=O)C(F)C1 35215,N1(C(C(C(CC)C)O)=O)CCCC2(C1)CN(C(c1nc(O)[nH]c(=O)n1)=O)CCO2 35216,c1(COC)cc[nH]c1C(=O)NC1(CNC(=O)C(C)NC(C2CCC2)=O)CCCC1 35217,C(c1cccc(O)c1)=CC(N1CCC(C2CCCN2Cc2cccnc2Cl)C1)=O 35218,c1(C(N2C(CNC(CNC(=O)OC)=O)CCCCC2)=O)sc2cccnc2c1N 35219,N1(C(C(c2ccc(Cl)s2)C)=O)CCC(NC(=O)Cc2ccc(O)c(Cl)c2)CC1C 35220,Cc1cc(C)n(CCCC2CCCN2)n1.C1(c2cn(CC(CO)(C)C)nn2)COC(C)(C)C1 35221,c1(CCN=C(NC2CC(CC)C2)NCC2CCCO2)ccc(S(N)(=O)=O)cc1 35222,c1(OCC(N2CC3(CN(C(Cn4ccc(C)n4)=O)C3)C2)=O)cc(N)cc(C)c1F 35223,c1(NCc2ccc(Oc3ccc(Br)cc3)nc2)cccc2ncsc12 35224,CCC(C(=O)NCC1CC(C)CN(C(=O)C(n2nccc2C)C)C1)C(F)(F)F 35225,CN1CCN(C(=O)COC2CN(C(=O)C(F)C(C)(F)F)C2)CC12CCC2 35226,N1(CC(C2CC2)OCC)CCC2(CCCCN(C(c3cn(C)cn3)=O)C2)C1 35227,C1(C(=O)NC(c2ccncc2F)C)CC12CCN(C(=O)CCc1cncn1C)C2 35228,c1(C(C)(C)C)nnc(C(=O)NCCCNC(C2CN(C3CCOCC3)C2)=O)s1 35229,C(=O)(C(CC(N)=O)SC)NC(C1(OC)CCN(C(c2ccc(C(F)F)o2)=O)C1)C 35230,c1(OC)ccc(C(N2CCC(CCNC(C)=O)CC2)C(=O)NC2CCC2)c(Cl)c1 35231,C(N=c1cc(NCC=C(C)C(C)(C)C)nc[nH]1)C1(Cc2ccccc2)CCCC1 35232,C(=O)(CCCCN(C)C)NCC1C(NC(COC(C)=O)=O)CCC1 35233,CCCC(C(O)C(=O)N1CCc2c[nH]nc2C1)NC(=O)C=Cc1cncn1C 35234,N1(C(c2nc(CC)[nH]n2)=O)CC(NC(C2(C(C)C)CC2)=O)CC1C 35235,N1(C(C(CC)C#N)=O)CC(O)(C2CCN(C(=O)Cc3cn4ccsc4n3)CC2)C1 35236,CC(C)(C(=O)NCC1CC(NC(=O)C(C2CC(F)(F)C2)O)C1)C(F)(F)F 35237,N1(C(CC2N(C(C3CC(=O)NC3)=O)CC2)=O)CCOCC(CO)C1 35238,c1(C(N2CC3C(NC(CC(=O)OCC)=O)C3C2)=O)cc2cc(F)ccc2o1 35239,C(C)(C)(CCCC(=O)NC(CO)C1CC1)NC(c1ccc(OC)cc1)=O 35240,c1(N(C)CC2C3CN(C(C4CCC(C)CO4)=O)CC32)nc2cc(F)ccc2s1 35241,C1(CC)CCCCCCN1C(C1CCOCCN1C(C1CCSCC1)=O)=O 35242,N1(C(c2cncc(C(N)=O)c2)=O)CC2CC(C1)N(C(=O)CC1CC=CCC1)C2 35243,C1(C(=O)NC(c2nocc2C(=O)NCCc2cccc(F)c2)C)CCCCC1O 35244,C12(CNC(C3(C)COCCO3)=O)CCC1CN(C(c1cc3occc3[nH]1)=O)C2 35245,C12(CNC(CC3CC(=O)C3)=O)CCC(C1)N(C(=O)CCCCN1CCCC1)C2 35246,c1(C(=O)NCC(C)(C)OCC(=O)NCC(=O)NCC=C)ccccn1 35247,C(CC(=O)NC1CN(C(c2nc(Br)sc2C)=O)C1)(C(F)(F)F)OC 35248,Cc1cc(C(=O)NCCN(C(=O)C(c2ccc(Cl)cc2)C)C)c(C)[nH]1 35249,C1(C(=O)NC2C(OC)CCOC2)C2CC3C(C2NC(c2cnnc(C)c2C)=O)C13 35250,N1(CC(=O)NC(C)CN(C(=O)CCc2cscc2Br)C)CCCCCC1 35251,N1(C(c2c(C)nc(CC)o2)=O)CCC(NC(=O)C(C)NC(=O)NC)C(CO)CC1 35252,c1(CC(=O)NC(C(C)C)CCN(C)C(C2CC(C)(C)C2)=O)ccccc1[N+](=O)[O-] 35253,Cc1cc(Br)ccc1CCNC(C1CC2CC2N1C(=O)CNC(=O)CC(C)C)=O 35254,c1(N(C)CC)ccc(C(N2CC(n3cc(C(C)(O)CCO)nn3)C(C)C2)=O)cc1 35255,c1(C(N2CCCC2c2ncc(-c3c(F)cccc3F)[nH]2)C)cccc2c1OCO2 35256,c1(C(=O)NC(CC(C)NC(C2CC(CC)C2)=O)C)ccnc(C(F)F)c1 35257,c1(OC)cc(C(=O)N(CC(C)N(C(=O)CN2CCCC2C)C)C)[nH]n1 35258,c1(NC2C(C)SCC2)ccc(S(=O)(=O)NCC(C)(C)CO)c(Br)c1 35259,C12(NC(COCC)=O)CN(C(c3ccc4n[nH]cc4c3C)=O)CC1CS(=O)(=O)C2 35260,C1(C(=O)NCC23OCC(NC(C4(C)CC4)=O)C(C2)C3)COc2cc(Cl)ccc2C1 35261,CC1CNc2c(C(=O)NCCN(C)C(C3CCC(N=[N+]=[N-])CC3)=O)cnn2C1 35262,C1(N(C2CCOC2C)C(c2cccc(OC(C)=O)c2)=O)CCNCC12CC2 35263,C(C1CN(C(=O)CCN(c2ccncc2)C)CC1C(=O)NC(C)CC)=CC 35264,c1(C(C(=O)NC(CC)(C)CNC(=O)Cn2cc(C3CC3)nn2)C)ccccc1F 35265,N1(c2c(C(C)=O)cccn2)CCC(NC(=O)C(C)n2cnnn2)C(O)C1 35266,Cn1nc(C(=O)NCC2(C(=O)NCC3CCCNC3=O)CCCO2)cc1Cl 35267,c1(C(C)(C)C)cc(C(=O)NCC(O)CNC(=O)CCOCC(F)F)cs1 35268,C1(C(C#C)NC(C2CCOCC2)=O)(CC)CCN(C(=O)CCc2conc2C)C1 35269,N1(C(C(CC)F)=O)CC2CCOC2(CNC(c2cc(OC(C)C)ccc2Cl)=O)C1 35270,N1(C(c2c(CC)ncs2)=O)C(CNC(c2cc(C(C)C)on2)=O)CC2CC12 35271,C(=O)(C1CCCc2cn(C(C)C)nc21)NCC1N(C(c2c(C)nns2)=O)CCC1 35272,c1(OC)ccc(C(C)=CC(=O)NC2CCC2NC(c2csc(CO)n2)=O)cc1 35273,CC(C)C(C(=O)NC1CN(C)CCN(C)C1)C(C)NC(C1CCCCC1O)=O 35274,c1(CC(=O)NC2CCCCN(C(C(CCCC)=O)=O)C2)csc2cccc(F)c12 35275,C1(NC(CCC(=O)NC)=O)(CNC(c2cccnc2N)=O)CCCCC1C 35276,N1(C(C2CCCSC2)=O)CCCCC2(CCN(C(=O)C(C3CCOCC3)O)C2)C1 35277,c1(C(=O)NC2C(CNC(=O)Cn3cnnc3O)C2)cc2ccc(Cl)c(F)c2[nH]1 35278,c1(C(=O)NCCC2CCC(NC(c3c(CC)occ3)=O)C2)ccc(Cl)cc1NC 35279,Cc1ccc(S(=O)(=O)NC(Cn2ccnn2)C(=O)N(C)C)cc1C 35280,C1(CNC(c2cnn(C)n2)=O)C(C2CC2)CCN1c1ncnc(Cl)c1F 35281,CC1(C)C(CNC(C2CCCCCC2)=O)CCN1C(C1C(C)(C)C1(F)F)=O 35282,C(C(C(=O)NCC1(O)CC(NC(=O)CC2CC(=C3CCC3)C2)C1)NC(C)=O)OC 35283,N1(C(c2ccn(CCC)n2)=O)CC2CC2C1CNC(c1ccnnc1C)=O 35284,Cc1ccc(N)cc1S(=O)(=O)NC(c1ccc(OC(C)(C)C)nc1)=O 35285,c1(C(=O)NC2CN(C(C3(C(C)C)CNC(=O)C3)=O)C2)nn(C)c(Cl)c1Cl 35286,c1(NCC2CN(C(c3[nH]cc(CC(C)C)c3)=O)CC2C)ncnc2c1nnn2C 35287,CON(C(=O)CC1=CCN(C2CC2)CC1)C(C)C1C2COCC12 35288,N1(C(CC2CC(=C)C2)=O)CC2CCN(C(c3cc(N)cc(OC)c3OC)=O)C2C1 35289,c1(C(N(CC(CC)NC(C2(c3cccs3)CC2)=O)C)=O)cnc(O)n(C)c1=O 35290,O=C(C1=CCCSC1)NC1CCN(C(c2ncc(F)cn2)=O)CC1CO 35291,C12(C(=O)NCC3C(C(=O)OCC)CCO3)CC3CC(C1)CC(F)(C3)C2 35292,Cc1c(C(=O)N(C)CCC2CCCCN2C(=O)C#CC2CC2)cccc1CO 35293,c1(C(=O)NC(CCCC)CNC(c2ccco2)=O)cccc(OC)c1OC 35294,C(CC(=O)NC1CC(CCNC(C2(CC)CCC2)=O)C1)OCCC 35295,c1(C(=O)NCCC(=C)CNC(c2cc(Br)c(C)o2)=O)cccc(CC)n1 35296,c1(NC(=O)C(=O)NC2CC(C3CCC3)C2)cc(F)c(Br)c(Cl)c1 35297,C12(NC(c3c(C)cncc3)=O)CC(CNC(C3C=CCC3)=O)(C1)OC2C 35298,C(=O)(C1=NOC2COCC12)N1C(C)CN(C(C(C)=NOCC#N)=O)C(C)C1 35299,Cc1ccc(NNC(=O)CNC(=O)CC2CCC(C#N)C2)cn1 35300,N1(C(c2ccc(NC(C)=O)nc2)=O)C2CCC1CN(C(=O)COC1(C)CCC1)C2 35301,c1(C(N2C(CN(C(=O)COCC3CC3)C)CCC2)=O)ccc(F)c2ccncc12 35302,C=CC(C)(O)CC(=O)NC1C2CC(NC(c3nc(CC)c[nH]3)=O)CC12 35303,C1(COC)CCCCN1C(=O)C(N1CCC(CCn2cncn2)CC1)=O 35304,c1(C(=O)NC(CNC(C2(C)CCC(C)C2)=O)C)cnn2ccccc12 35305,C1(C(N(CCC)CC2CC2)=O)CC12CCN(C(=O)Cn1ccnc1C)C2 35306,c1(C(N2CCCC(CN(c3ncncc3Br)C)C2)=O)cncc2c1CCCC2 35307,N1(CC(c2ccc(F)cc2)NC(=O)Nc2ccc(I)cc2)CCCS1(=O)=O 35308,CC1(F)CCC(C(=O)NC2CCCC2NC(c2ccc([N+](=O)[O-])o2)=O)CC1 35309,CC1(C)CCC(CC(=O)O)N(C(=O)C(O)Cc2ccncc2Br)C1 35310,c1(C(=O)NCC2N(C(C(C)NS(CC)(=O)=O)=O)CC(O)C2)cccc(F)c1C 35311,CC(C)(C)C(O)C(=O)NCC1CN(C(c2ccnc(C(F)(F)F)n2)=O)CC1(C)C 35312,Cn1nc(C(=O)NC2CCC(NC(c3coc(CC4CC4)n3)=O)C2)cc1C#N 35313,N1(C(C2(CC)CC2)=O)Cc2cccc(CNC(=O)Cc3cn[nH]c3)c2C1 35314,c1(OC)ccc(S(=O)(=O)OCC(=O)Nc2cc(Cl)cs2)cc1[N+](=O)[O-] 35315,N#Cc1ccc(C=CC(N2CC(CO)(NC(c3cn4c(n3)CCC4)=O)C2)=O)cc1 35316,CC(C1COc2ccccc21)CN(CCC(=O)O)C(c1cnc(C(F)(F)F)nc1)=O 35317,Cc1nc2cc(C(N3CC(NC(C4CNC(=O)N4)=O)C3)=O)ccc2n(C)c1=O 35318,CSC1=C(C(=O)NCC(C2CC2)N(C(=O)C(CO)c2ccccc2)C)CCCC1 35319,C1(C(=O)N(CCNC(c2c[nH]cc2C2CC2)=O)C2CC2)(COC)CC1(F)F 35320,C1(NC(=O)NCC(C)OC)CCN(C)C2(CC2)C1 35321,C1(N(C(CC)C(=O)NCC)CC)CCN(C(=O)CCCn2ccnc2C)C1C 35322,c1(C(N2CC3C(CC)C3C2)=O)c(OC)cc(NC(=O)OC)cc1I.C1(=O)CN1 35323,c1(C(=O)NCC(CC)N(C(=O)C(c2csc(C)n2)=O)C)cc(C2(C)CC2)n[nH]1 35324,C1(NC(=O)NCCN(C)CC)C2CCC(C2)N1C(=O)OC(C)(C)C.C1COC1 35325,C12(C(=O)NC(c3ccc(F)cc3)CNC(CC(C)(C)F)=O)CC=CC(C1)OC2 35326,C=Cn1nccc1C(N1CC(N(C)C)C(CNC(=O)C(O)CC)C1)=O 35327,c1(C2C(C(N3C(C(=O)NCCC(=O)O)CC3)=O)C2)ccccc1OC(F)(F)F 35328,Cc1ncncc1C(=O)NCCn1cc(CNC(C2CC2C(C)(C)C)=O)nn1 35329,N1(CCNC(c2c(C)occ2)=O)CCC(NC(c2c[nH]c(=S)cn2)=O)CC1 35330,C1(NC(C(C)C2(O)CCC2)=O)CCCCCC1NC(c1cc(F)cc(Cl)c1)=O 35331,CC1CC(C(=O)NC2C3CCC2N(C(=O)Cc2ccon2)C3)=NO1 35332,C(CCN(C)C)(C(=O)NCCOC1CC1)NC(C1(COC)CCCO1)=O 35333,C1(NC(C=CC(=O)OCC)=O)C2CC(O)C1N(C(=O)Cc1csc(NC=O)n1)C2 35334,CC1(CNC(=O)C=Cc2ccco2)CN(C(=O)CCN2CCC(F)C2)CCO1 35335,C(=O)(C#CC(C)(C)CNC(C1(C)CC1(F)F)=O)NC1C(C)COCC1 35336,CCCN=c1cccc(S(=O)(=O)NCC(c2ccc(F)cc2)(C)C)[nH]1 35337,c1(C(=O)NC2C(NC(=O)Cc3ccnnc3O)CCCC2)ccc([N+](=O)[O-])o1 35338,N1(C(c2nc(C)oc2C)=O)CCN(C(c2cc(=O)c(O)c[nH]2)=O)CC(O)C1 35339,N1(C(C=CC)=O)CCC2(CC1)CC(NC(=O)C(C)Sc1nnnn1C1CC1)CO2 35340,CCC(C)(CCNC(=O)C(F)C1CCCC1)NC(=O)CC1(N2CCCC2)CC1 35341,C(=O)(C(C(C(C)C)OC)N1CC(O)CC1CN(C)C)NCC.C1(=O)C(C)N1 35342,C(C(C)(COC)CO)NCc1ncc(CC)[nH]1 35343,c1(C(=O)NC(C(N2C(C(N)=O)CC2)=O)c2ccco2)ccc(Cl)cc1Cl 35344,C1(C(N2CCC(CNC(CCS(C)=O)=O)C23CC3)=O)COc2cc(F)ccc2C1 35345,N1(C(c2cc(OCC)cc(F)c2)=O)CC2(CC(NC(=O)Cc3ccsc3)CO2)C1 35346,c1(C(N2CCCC(NS(CC(=O)OCC)(=O)=O)C2)=O)ccc2nccn2c1 35347,C1(OC)CC(NC(c2ccccc2CO)=O)CN(C(=O)CNC(N)=O)C1 35348,c1(C(=O)NCC2(CN(C(C3C(CC)C3)=O)C)CC2)cncc(C#N)c1 35349,c1(NC2CC(NCc3cc([N+](=O)[O-])sc3)C2)ncnc2c1CCC2 35350,CC1C2C(CCN2C(=O)COC2CCOC2)CN1C(=O)CN1CCCC(O)C1 35351,c1(C(N2CCC(OCC(=O)NC3CC3C3CCCC3)C2)=O)ccc([N+](=O)[O-])[nH]1 35352,C1(C(=O)NC(C(C)NC(C2CC2c2cccc(F)c2)=O)(C)C)CCCC(=O)N1C 35353,C(=O)(C1=CC2CCCCC12)N1CC(CNC(=O)CC2(O)CCC2)C(C(F)(F)F)C1 35354,c1(C(c2ccc(C)cc2)NC2CC3CCC2CC3)ccc(-c2nc[nH]n2)c(F)c1 35355,N1(C(c2cc(C)ncc2C)=O)CC2CCCC(C1)N2C(c1cccc(N)c1O)=O 35356,C1(C(N2CC(NC(C3CCCN(C(=O)OC)C3)=O)C2)=O)CCC12CCOCC2 35357,C(=O)(C1CCCn2ccnc21)NC1C(NC(=O)CCN2CCCS2(=O)=O)CCC1 35358,C(=O)(C1CCCc2sccc21)NCC(CNC(c1c(CC)cccc1CC)=O)C 35359,N1(C(CC=C)=O)CC(C)(C)CC1CC(=O)NC(C)C(O)C(F)F 35360,N1(C(C(C)Sc2nncs2)=O)CCn2c(nc3ccccc23)C1 35361,C1(CC(=O)NCC2CCCN2C(c2ncoc2-c2cccs2)=O)CCCS1(=O)=O 35362,C1(N(C(c2ccc(C(C)C)cc2)=O)CC)CCCN(C(C2(C3CC3)CC2)=O)CC1 35363,c1(C(N2CC(O)(C(C)NC(C(C)S(C)(=O)=O)=O)C2)=O)n[nH]c2c1CS(=O)(=O)CC2 35364,N1(C(Cc2ncc(CC)[nH]2)=O)CC(CCNC(=O)CC(=O)NC2CC2)OC(C)C1 35365,C(C(C(F)(F)F)N1CCN(C(=O)CC2C=CCC2)CC1)NC(CN(C)CCO)=O 35366,c1(C(N2CC(N(C(=O)CC3CC(C(F)F)C3)C)C2)=O)coc(Cl)c1 35367,C1(C(N2CCC(CN(C(=O)CN3CCC(C)(C)C3)C)CC2)=O)CCCCC12CC2 35368,c1(C(=O)NCCC(C)NC(c2ccc(Cl)o2)=O)oc2ccccc2c1CS(C)=O 35369,c1(N2CCC(NC(c3cnn(CC)c3C)=O)C2)cccc(F)c1C#N 35370,C1(C(=O)NCC(C(C)C)NC(c2cn3c(n2)SCC3)=O)CCC(S(C)(=O)=O)CC1 35371,C(=O)(C(F)CCC(C)(C)C)N1CCN(C(C2N(CC)CC2)=O)C(COC)C1 35372,c1(CCC)ccc(C(=O)NC2COCCC2NC(C2CC(F)C2)=O)cc1[N+](=O)[O-] 35373,C(=O)(CC(O)C(C)(C)C)NC1CCC(NC(C2ON=C(C)C2)=O)CC1 35374,CCCCC(C(=O)NCC=C(C)C)NC(=O)CCC(N)=O 35375,c1(C(N(C2CCN(C(=O)CSC3CC3)CC2)C)=O)nnc(-c2ccccc2)n1C 35376,c1(C(N2CCCC(CC(=O)Nc3nccc(C)c3)C2)=O)cc(Br)cnc1O 35377,c1(C(=O)NC2CN(C(C3(O)CCOC3)=O)CC2O)cc(F)cc(Cl)c1 35378,N1(C(C(C)(C)SC)=O)CCN(CCCNC(=O)C(=Cc2cccs2)C)CC1 35379,c1(CC(N2CCCCC(N(C(CC(C)CF)=O)C)C2)=O)cccc2nsnc12 35380,C(=O)(C1=C(Cl)CCC1)NC(C1CCC1)CNC(C(C)Cn1cccn1)=O 35381,c1(C(N2CCN(C(=O)C=Cc3ccco3)C(CO)C2)=O)ccc2c(c1)COCO2 35382,CCCC(C)(O)CC(=O)N1C2CCC(C2)C1C(=O)NC(c1ccccc1)CF 35383,N1(C(CCC(C)C)=O)CCOCC2(COCCN2C(=O)C2=CC3CCCC23)C1 35384,c1(CC)ccc(C(=O)NC2CCC(NC(C3(F)CCC3)=O)C2)[nH]1 35385,C(C(CC(C)(C)C(=O)OC)NCc1cn(-c2cc(C)cc(C)c2)nn1)OC 35386,C12(CNC(C(C(C)C)C)=O)CCC(CN(C(=O)CCCc3n[nH]c(=N)s3)C1)C2 35387,Cc1[nH]c(C#N)cc1C(=O)NCC1C(C)CCCN1C(C1CCCC1O)=O 35388,C(=O)(CC1=CCCC1)NC(CCC(=O)NCC1(C(=O)OC)CC1)C 35389,C1(C2CC2)(CNC(C=C(C)C(F)F)=O)CCN(C(c2c(C)ccc(F)c2O)=O)C1 35390,c1(OC)cnc(F)cc1C(=O)NCC(C)(CO)NC(=O)C=Cc1ccc(O)cc1 35391,Cc1cccc(CC(N2CCC(CNC(C3(C)CCCCO3)=O)C2)=O)c1Cl 35392,C(=O)(C1=NOC2(CCN(C(C3C4C=CSC34)=O)C2)C1)Nc1cc(C(C)C)no1 35393,N1(C(C(C)n2cnnn2)=O)CCN(C(=O)C#CC2CC2)C(CC(F)F)C1 35394,c1(C(=O)NC(CC)CNC(=O)CCc2ccc(F)nc2)cncc2cccnc12 35395,C1(C(=O)NCC2(NC(c3cc[nH]c3)=O)CCC2)CC12CCSCC2 35396,C(=O)(C(O)C(C)OC)N(C1CCN(C(C2(CF)CCC2)=O)CC1)CCC 35397,c1(C(=O)NC2CC3CN(C(C4(CSC)CC4)=O)C2C3)ccc(S(N)(=O)=O)nc1 35398,C#CC1(O)CN(C(=O)CN(C(C2CCC2(OC)OC)=O)C2CC2)C1 35399,C1(CC)C(C(=O)N(CCC(=O)N(C)CC2CCCCO2)CCO)CCN1C 35400,c1(C(C)=O)ccc(C(N2CCC(C3CCCN3C(c3csc(CO)n3)=O)C2)=O)o1 35401,c1(CC)nn[nH]c1C(=O)N(C)CC1(NC(=O)C(COC)OC)CC1 35402,c1(C(=O)NCC(CC)NC(=O)CCC(C)OC)ccc(N)c(CC(C)C)c1 35403,C(=O)(CCCS(C)(=O)=O)NC1CCCC(N(C(=O)C=C2CCC(C)(C)CC2)C)C1 35404,N1(C(c2c(C)snc2)=O)CCC(NC(=O)Cc2cncn2C2CC2)C12CCC2 35405,c1(CNC(C(C(C)O)NC(=O)CC(C)(C)O)=O)ccc(C#N)cc1 35406,c1(C(N2CCC(NC(c3scnc3Cl)=O)CC2C2CC2)=O)cncc2sccc12 35407,c1(CCC(=O)NC2CC(NC(CCS(C)=O)=O)C2)nnc(S)nc1O 35408,CC1(C)CC2(CC2C(=O)NCC2(NC(c3ccc(F)c(C(F)F)c3)=O)CC2)C1 35409,C(=O)(CCC(C)(C)F)NCC(CCNC(C1N(C(CC(C)C)=O)CCCC1)=O)O 35410,C1(NC(=O)CSc2ccsc2[N+](=O)[O-])CCN(C(=O)COC2CCC2)C12CCC2 35411,c1(CC(=O)NC(C2CCCN(C(=O)CC3CC3)C2)C)ccc(F)c(F)c1 35412,C1(C(N2CCC(NC(C(CC)=CC)=O)C(C)C2)=O)CCCC2CCCN12 35413,CC1(C)CCCC(C(=O)NC2CCCC23CN(C(c2snc(Cl)c2Cl)=O)C3)CC1 35414,CC1(C)CCC(=O)NCc2cn1nn2.c1(-c2ccccc2)nc(=O)o[nH]1 35415,c1(CC(C(=O)NC2(CCNC(CC3CC(OC)C3)=O)CC2)C)ccc(F)cc1 35416,N1(C(c2nc(C)sc2C)=O)CCC(C2(O)CN(C(=O)C(C)S(N)(=O)=O)C2)CC1 35417,N1(CC)C(=O)CCC1CC(=O)NCCOCCCNC(=O)CN1C(=O)CNC1=O 35418,C1(C)(CCC(=O)NCCCN(C(C)C)C(C2CC(F)(F)C2)=O)CCC(=O)N1 35419,n1(CC(=O)NC2(C)CC(NC(C3(CC)CCNC3=O)=O)C2)c([N+](=O)[O-])cnc1C 35420,O=C(CCC(=O)N1CC(O)(CNC(C2(F)CCOC2)=O)C1)OCc1ccccc1 35421,C12(C(=O)NC3CCC(CCNC(c4cnc(OC)nc4)=O)C3)CC(C)(CCO1)C2 35422,Cn1cc(C(CO)NC(=O)CNn2cc(-c3cnn(C)c3)nn2)nn1 35423,c1(C(=O)NC2CC(O)(CNC(=O)CC3CCCS3(=O)=O)C2)cc2c(s1)CCC2 35424,CC(C)S(=O)(=O)CCCN1CC=CC(NC(c2coc(Cn3cccn3)c2)=O)C1 35425,C(=O)(CC(C)(C)N(C(=O)CC1CCC(=O)N1C)C)NC(c1ccccn1)CC 35426,C=CC1CN(C(C2(Cc3ccccc3)CC2)=O)CC1NC(c1cc(C)c(C)[nH]1)=O 35427,N1(C(C(C2CCOCC2)OCC)=O)CCC2C1CCCN2C(c1cnc(O)s1)=O 35428,C=C(Cl)CC(C(=O)NOCC)NC(C1CN(C(=O)NC2CC2)C1)=O 35429,C1(C(=O)NCCC(O)C2CCCC2)(CC)CCN(C(=O)C=Cc2cocn2)C1 35430,Cc1ccc2n[nH]cc2c1C(=O)NC1CCN(C(c2cnc(O)c(Br)c2)=O)C1 35431,N1(C(CC2CC(OC)C2(C)C)=O)CC2CCC(N=c3ccc(C(F)(F)F)n[nH]3)C2C1 35432,N1(C(c2c(C)nc(CC)s2)=O)CC(CNC(c2ccsc2C#N)=O)CC1(C)C 35433,C(=O)(C1CCCc2c[nH]nc21)NC1(CNC(C23OCC(C)(C2)C3)=O)CC1 35434,c1(CC(=O)NC(C)CCNC(=O)C(C)C2CCCO2)ccc2nonc2c1 35435,C1(C(=O)OCC)CC2CC(C1)CN(C(=O)Nc1cc(F)cc(F)c1Cl)C2 35436,C1(C(=O)N(C)CCSC)(CC)CCCN(C(c2cc(CCO)on2)=O)C1 35437,c1(C(=O)NC2C(NC(c3c(C)nc(COC)s3)=O)C2)cc([N+](=O)[O-])c(C)cc1Cl 35438,c1(C(=O)OC)ccc(C(=O)NC2CCC(NC(=O)CS(N)(=O)=O)CC2)nc1 35439,c1(CCC(=O)NC(CC)CNC(C2CCC(F)(F)CO2)=O)nc2ccccc2o1 35440,C(C1(C)COC1)=CC(=O)NCCN(C(C1C(Cl)(C(=O)OCC)C1)=O)CC 35441,N1(C(C2CCCN(CC)C2)=O)C2CCC(C2)C1CNC(c1ccc(O)nc1)=O 35442,N1(C(C(C)=C(C)C)=O)CC2(COC(CNC(c3cc(C(F)(F)F)n(C)n3)=O)C2)C1 35443,N1(C(C(C)(C)C2(O)CCC2)=O)CCCC(Cn2ccnc2)C1 35444,CCC(CC(C)C)C(=O)NCC1(O)CN(C(=O)Cc2ccn(CC(F)(F)F)n2)C1 35445,O=C1CCc2cccc(C(=O)NC3CCCC3CNC(c3coc(Cl)c3)=O)c21 35446,C1(C)(NC(C(CCCNC(C=C(C)C(F)F)=O)O)=O)CCC(=O)NC1=O 35447,C1(N(C)C(C2(C(C)(C)C)CCC2)=O)CCN(C(=O)COc2ccsn2)C1 35448,c1(C(=O)NCC2C(C(=O)NCc3c(C)nccn3)CCO2)ccn(C)c(=O)c1 35449,C1(C(=O)NC(C(=O)NC)(C)C)CC2CC1CC2NC(=O)C(CO)N(C)C 35450,N1(C(C(Cn2ccnc2)NC(=O)CNC(C2CCCO2)=O)=O)CCC(O)CC1 35451,C=C1CCN(CCn2nc(C)oc2=O)CC1 35452,C1(CC)CN(C(=O)C=Cc2cccnc2)CCN1C(=O)COCC(=O)NC 35453,N1(C(c2c(C)ncs2)=O)CCCC2C1CCCN2C(C1CCC(N(C)C)CC1)=O 35454,c1(NC(C(C2CN(C(C(COC)O)=O)C2)OC)=O)cncc(N2CCCC2)n1 35455,N1(C(C2CCN(C(c3n(CC)ccn3)=O)C23CC3)=O)CCC(O)CC(C)C1 35456,N1(C(C(CCOC)OC)=O)CCN(C(=O)CCCSC)C(C)C1 35457,CC1CS(=O)CCN1C(C1CCCC(NC(=O)CCc2nccs2)C1)=O 35458,C12(C(N(C(c3cccc(F)c3)C)Cc3ccco3)=O)CC(CN)(C1)OC2C(F)(F)F 35459,C(CNC(=O)C(C)(C)n1ccnn1)(CC(F)(F)F)NC(c1cccc(OC)c1)=O 35460,c1(C(=O)NCCCC(C)NC(CCNC(COC)=O)=O)ccc(C)nn1 35461,Cc1ncc(C#N)cc1NC(=O)C=CCN(C)C(C1(O)CCOC1)=O 35462,N1(C(C(C)=C(C)C)=O)CCC2CN(C(C3(C)C=CCC3)=O)CC2CC1 35463,C1(CC)CN(C(=O)CC2CS(=O)(=O)C2)CCN1C(=O)COc1cnn(C)c1 35464,C(=O)(CC(C)CNC(=O)C(C)c1ccco1)NCc1n(CC)cnn1 35465,C(CC(C)C(=O)N1CCN(CCNC(=O)Cc2n[nH]c(=NC)s2)CC1)=CC 35466,CC(C)CCC(F)C(=O)NC1(CCC(=O)N(C)Cc2ccsc2)CCCC1 35467,c1(OC)ncnc(C(=O)NC2(C)CN(C(C3CCOC(=O)CC3)=O)C2)c1F 35468,N1(C(C2CCC(C)(C)CC2)C(=O)NCC=C)CCCC2OCCC2C1 35469,CCC(O)C(C)C(=O)N1CC(C2(NC(c3c(OCC)cncc3F)=O)CC2)C1 35470,CCCC(CC)C(=O)NCC(O)CCNC(c1cc(=O)c(Br)c[nH]1)=O 35471,N1(C(CC2CC(=O)OC2)=O)CC=CC(C(=O)NC2CC(CO)C3CC23)C1 35472,CC(CC(C)NC(=O)CS(=O)(=O)NC1CC1)N=c1[nH]c(Cl)nc2ccccc12 35473,CC1(C(=O)NCC2CC(NC(C3CC(=O)N(O)C3)=O)C2)CS(=O)(=O)C1 35474,C1(CC(=O)NC2CC(NC(C)=O)C2)CN(C(=O)CCC(=O)NCC2CC2)CCO1 35475,C(CC(=O)NCCCC(F)F)(C1CC1)NC(C(C)c1cc[nH]n1)=O 35476,CCCC(C)(CCCNC(N1CCCC(F)(F)C1)=O)C1OCCO1 35477,N1(C(c2cc(C)n(C)n2)=O)CC(F)(F)CC1CCNC(c1cc(Cl)c[nH]1)=O 35478,c1(C(N2CC3CN(C(C(CC(=O)OC)C)=O)CC3C2)=O)c(O)nnc2c1CCC2 35479,C(C)(CCCNC(=O)C=CCOC1CCOCC1)NC(CSCCCC)=O 35480,C(=O)(NNc1cccc2ccsc12)C1N(C(=O)OC(C)(C)C)C(C2CC2)CC1 35481,N1(C(c2cc(Br)cs2)C(=O)NCC2CC2)CC2CCCCN2c2ccccc21 35482,c1(C(=O)NC2C(C)CCN(C(c3csc4cncn34)=O)C2)cc2occc2n1C 35483,c1(C(=O)NC2CC(F)(CNC(C(N3CCOCC3)C)=O)C2)c(F)ccc(F)c1N 35484,N#CC1(C(N2CCC2CNC(C2(S(N)(=O)=O)CCC2)=O)=O)CC2CC2C1 35485,N1(C(C2CCN(CC(C)C)C2)=O)CCN(C(=O)C2=CSCS2)CC1C1CCC1 35486,Cc1cc2[nH]c(=O)c(NC(=O)NC3CCN(c4ccccc4)C3C3CC3)cn2n1 35487,CC(=O)CC(C)(C)C(=O)N1CCC(C)C(CNC(C2CN(C)CC(C)O2)=O)C1 35488,C1(C(N2CCC(C(C)OC)CC2)=O)CC2CCC1N2C(c1csc(C)c1)=O 35489,CN=c1[nH]c(=NCCCc2nc(C)cs2)[nH]c(=NC2CCOC(C(C)C)C2)[nH]1 35490,c1(C(N(CCCCN(C(CCn2c(C)ncc2)=O)C)C)=O)ccc(F)c(Cl)c1F 35491,c1(C(=O)Nc2c(C(N3CCC(C)CC3)=O)cc(OC)nc2)cc2ccccc2s1 35492,N1(C(c2c(C)ccnc2)=O)CCCC(C)C1CNC(=O)C(F)C1CCOC1 35493,c1(C(=O)NCC2=CCN(C(c3ccn(COC)n3)=O)CC2)cn2cc(C)sc2n1 35494,N1(C(Cc2nnc(C)o2)=O)CC2(CCC(NC(c3cc(Cl)c(F)cc3F)=O)C2)C1 35495,C1(CNC(CC2C(C)CCO2)=O)CCC2CN(C(c3cnc(Cl)[nH]3)=O)CCC2C1 35496,N1(C(CN(C(=O)C(C)c2cccs2)CC#C)=O)CCC(C)(CO)C1 35497,C(=O)(C(C)C(O)CC(C)C)NCC1(O)CN(C(Cc2c(F)ccc(C)c2)=O)C1 35498,c1(OC)cc(F)c(C(=O)NC2CC2CNC(c2cocn2)=O)cc1Br 35499,C=CCC(CNC(C1(C)CC(=C)C1)=O)NC(c1csc(C2CC2)n1)=O 35500,C=C(Cl)CC(C(=O)NC(c1nccn1C)C)NC(=O)Cc1ccn(CC)n1 35501,C1(NC(C(F)=C(C)C)=O)C2CC3CN(C(c4cc(O)c5ccoc5c4)=O)C1C3C2 35502,Cc1ccc(C(=O)NCC(C)(CO)NC(=O)CC2CCC2C)c(O)n1 35503,c1(OC)c(C(N2CCCCC(Cn3cc(C4CCC4)nn3)C2)=O)ccc(Cl)c1Cl 35504,c1(OCC)cc(C(N2CCC(=CCNC(=O)CCC3(C)CC3)CC2)=O)cc(F)c1 35505,Cc1ccc(Cl)c(C(=O)NCC(C2CC2)NC(=O)Cc2ccc(F)cn2)c1N 35506,N1(C(c2c(C)nc(C)o2)=O)CCC(C(=O)NC2(C(O)CO)CC2)C(O)C1 35507,C1(NC(C(C)NC(C2CNC(=O)N2)=O)=O)(CO)CC2CCCC12 35508,CCCCCCCCCC(=O)NCC1CC2(CC2)CN1C(=O)C(O)C(F)F 35509,N1(CCNC(c2nc(C(C)C)oc2)=O)CCCN(C(C2CC2(F)Cl)=O)CC1 35510,CC1CC(C(F)(F)F)n2nc(-c3nc(C4CCC(O)CC4)no3)cc2N1 35511,n1(CCCC)nnnc1C(c1cc(C(F)(F)F)cs1)N(C1CCC1)CC 35512,Cc1nc([N+](=O)[O-])cn1CC(=O)NCCC(C(C)C)NC(C1CCOC(=O)N1)=O 35513,C1(CC(=O)OC(c2ccc(F)cc2)C)COC2(CCC2)CO1 35514,c1(C(=O)NCC2(CNC(C(C(C)C)OC)=O)CC23CCC3)ccc(Cl)c(F)c1O 35515,O(C1CCCc2ccccc21)CC(=O)N(C(C)C)Cc1n[nH]c2c1CCCC2 35516,C(=O)(C(O)CCCc1ccccc1)N(CCNC(C1CCN(C)C1=O)=O)C1CC1 35517,N1(N2CCn3c(O)nnc3C2)CC2C(CO)C3CCC2(C1)O3.O=C(O)CSCC=O 35518,N1(Cc2ccc(-c3nc(CC)c(C)cn3)s2)CCC2(CCOC2)CC1 35519,C1(NC(C2(C)N(C(CCc3c(C)noc3)=O)CCC2)=O)(CO)CC2CCCC12 35520,c1(C(=O)NCC(C)CNC(C23CC(C)(C2)C3)=O)cc2c(o1)CCCNC2=O 35521,C1(CNC(c2c(N)c(Cl)ncc2)=O)CCC2(CCC2)C1NC(c1ccoc1Cl)=O 35522,N1(Cc2n(CC#C)cnc2)CC(CC(=O)OCC(C)(C)C)c2ccccc21 35523,Cc1cn2cccc(C(N3CC(C4(NC(=O)Cc5csc(S)n5)CC4)C3)=O)c2n1 35524,C1(C(=O)NCC2C3CN(C(=O)C(C4CCCCCC4)O)CC23)(CC)CCCCC1 35525,n1(CC)cccc1C(=O)NC1CC1NC(=O)C(c1ccccc1)OCCC(C)C 35526,C1(CNC2(COC)CCN(C(C(CCN(C)C)(C)O)=O)C2)CC2CCCC(C1)C2 35527,N1(C(CN(C)CC)=O)CCC(C)N(C(=O)COc2cccc(Cl)c2)CC1 35528,CN1CCN(C(=O)CCc2cc(F)ccc2Br)C(CNC(=O)C(N)=O)C1 35529,c1(OC)ccc([N+](=O)[O-])cc1-n1cc(CN(C(=O)C(C2CCC2)OC)C)nn1 35530,c1(C(N(C)CCC2CCCCN2C(=O)CCC(N)=O)=O)ccccc1P(C)(C)=O 35531,N1(C(c2c(OC)ccnc2)=O)CCCC(NC(=O)CC(C)(C)C#N)C1C 35532,N(C(=NCCCC1CCOC1)NCC1CC2CCC2C1)CCc1cn(C)nc1 35533,CCCCCCCCOCC(=O)NCC(C)NC(C1C2CCCOC12)=O 35534,n1(CC2CCN(C3CCCN(C)C3=O)CC2)ncc(Cl)c(Cl)c1=O 35535,Cc1ccc(Cl)cc1C(=O)NCC(O)CN(C(=O)CN1CCC(C)C1)C 35536,CC1CN(C(C2CC(O)(CNC(C3(C)CCC3)=O)C2)=O)CC(C)(C)C1 35537,CC1(NC(C23CC(CN2C(C2(CCN=[N+]=[N-])CC2)=O)C3)=O)CCOC1=O 35538,C1(CNC(C(c2ccc(C)o2)C)=O)CN(C(=O)C=Cc2cccs2)C(C)(C)C1 35539,C1(NC(=O)Cc2ccc(Br)s2)CN(C(=O)CCC2CC2)CC1O 35540,c1(C(N2CCC(C(N(CCC(=O)OC)C)=O)C2)=O)ncc(F)cc1F 35541,C(N=c1nc(N2CCCC(Cn3ccnn3)C2)cc(C)[nH]1)C1(OC)CCC1 35542,N1(C(C2(CC)CC2)=O)CCN(C(c2csc(C(C)(C)C)n2)=O)CC2(CC2)C1 35543,c1(C(=O)NCCC(C)N(C(Cc2c(C)n[nH]c2)=O)C)cc2c(cnn2C)nc1C 35544,C1(COC)CN(C(C2(C)CCN(C(C)=O)C2)=O)CCN1C(=O)CC1CC=CC1 35545,N1(C(C2CC(C)SCC2)=O)CC(NC(C2COC(C)(C)C2)=O)CC(C)(C)C1 35546,C=C(Cl)CC(C(=O)NCC1C(CO)C1(F)F)NC(=O)C(CSC)OC 35547,N1(C(c2c(CC)noc2)=O)CC(CNC(c2cccc(C)c2)=O)CCC1C 35548,c1(C(=O)NCc2occ(C(=O)NCC(C(CC)C)C)c2)ccnc(C)c1N 35549,c1(C(N2C(C(C)NC(CCCCCC=C)=O)CCC2)=O)cc(N)c(F)c(F)c1Cl 35550,c1(C(N(CC(C)NC(=O)CCOCC(F)(F)F)CC)=O)cncc(Br)c1 35551,C(c1cn(CCCN(C)C(C2CCN(c3ccc(Cl)cn3)CC2)=O)nn1)=CC 35552,C1(C(N(C(CNC(C(C)O)=O)Cc2ccccc2)C)=O)CCC(F)CC1 35553,C12(C(=O)NC(CNC(c3cc(C)cc(O)c3)=O)(C)C3CC3)CCC(C)(CC1)OC2 35554,N1(C(C23N(C(C(=CC4CCCC4)C)=O)CC(C)(C2)C3)=O)CCC2CC1C(=O)O2 35555,C1(NC(C(N2CCSCC2)C)=O)CC(F)CN(C(c2cc(C3CCC3)on2)=O)C1 35556,Cc1ccc2sc(C(N3CCN(C(=O)C(C)C4CCOC4)CCC3C)=O)cc2c1 35557,N1(C(c2c(C)nc(C)o2)=O)CC2CCCC(C1)N2C(=O)C(C)n1ccnc1 35558,c1(CC(=O)NCCOC2CN(C(CC(C)OC)=O)C2)cnccc1Cl 35559,C(=O)(CCC(=O)N1CC(CCNC(C2(SC)CCC2)=O)C1)Nc1nnc(CC)s1 35560,C12(C(N(CCN(C(C3CC3(C)C(C)C)=O)CC)CC)=O)CC(C)(C1)OC2(C)C 35561,CC1(C)CC(NC(=O)Nc2ccnc(I)n2)C(=O)O1 35562,C1(NC(=O)CCC(F)(F)F)CCCC2CN(C(=O)CC3CCOC3)CC12 35563,C1(Nc2ccc(CC)cc2)CC2c3ccccc3C1c1ccccc12 35564,Cn1nnc(CNC(=O)C(c2ccccc2)NC(c2cc(F)c[nH]2)=O)n1.[nH]1ccnn1 35565,N1(C(c2c(C)occ2)=O)CCC2CC(CNC(C3CCC(C)CC3)=O)CCC2C1 35566,CC(C)CC(C(=O)N(C(C)CC(N)=O)C)ONC(=O)C1(C(N)=O)CC1 35567,C1(C(=O)N(CCCCC(=O)NCC2(C)CCCCO2)C)(CC)CCNC1=O 35568,C1(NC(c2cccc(F)c2OCCF)=O)CN(C(=O)COC(F)F)CCC1CO 35569,c1(C(CC)O)nc(C2CCC(=O)N2C)n(-c2nc(C)nn2C)n1 35570,N1(C(COCC#C)=O)CCN(C(=O)C2CC2)C(C)C1C 35571,C1(F)(C(=O)OC)CN(C(=O)NCCc2cccc(F)c2)CC1C1CC1 35572,N1(C(c2onc(CC)n2)=O)CC2(CCN(C(=O)Cc3cccs3)CC2)C1 35573,c1(C(=O)NC2C(CNC(C(C)NC(c3ccoc3)=O)=O)CC2)cc(Cl)c(Cl)n1C 35574,c1(OC)ccc(F)cc1C(=O)C(=O)NC1CCN(C(c2ccc(C)o2)=O)C12CC2 35575,N1(C(C(=O)NCC)=O)CCOCC(CNC(c2ccc(C)[nH]2)=O)C1 35576,C1(C(=O)NCC(CC=C)NC(c2cc(CCC)oc2C)=O)CC2C=CC1C2 35577,CC(C(=O)NC(C(=O)NCC1(CO)CCC1)c1cccs1)OC1CCCC1 35578,C(=O)(CCCC(C)(C)C)N1CCC(CN(C(=O)Cc2cn3ccsc3n2)C)C1 35579,Cc1cc(O)nnc1C(=O)NCCCCN(C(=O)C(C)(C)c1ccsc1)C 35580,c1(CC)c(NC2(C)CCCN(C(=O)CCC3CC3)C2)nc(C)nc1Cl 35581,N1(C(c2nnn(CC)c2C)=O)CCC(C2(NC(c3[nH]c(O)nc3C)=O)CC2)CC1 35582,[N-]=[N+]=NCCCC(=O)NCC1(O)CC(CNC(=O)CCc2csc(=N)[nH]2)C1 35583,c1(C(=O)NC2CC(NC(C3OCCN(C)C3)=O)C2)cc2c(C3CC3)cccc2[nH]1 35584,C1(CN(C)Cc2cccnc2)CCCN1C(=O)N(C(=O)C(C)(O)C1CCC1)C 35585,N1(C(C(CC)OCC)=O)CCC2(CCCN2C(c2cc(C(F)F)no2)=O)CC1 35586,n1(CC)nc(C)cc1C(=O)NCC1CC1NC(=O)C(C)(C)n1ccc(C2CC2)n1 35587,C1(CC)CCN(C(c2ccc(SC)s2)=O)C1C(=O)Nc1cnn(C)c1SC 35588,N1(C(CNC(C2C(C)(C(F)F)C2)=O)=O)CCC(Cc2ncncc2Cl)C(O)C1 35589,N1(C(c2c(C)nc(C)o2)=O)CC2(COC(CNC(c3ccns3)=O)C2)C1 35590,N1(C(c2cnn(CC)c2Cl)=O)CCC2CN(C(c3cnccc3Cl)=O)CCC2C1 35591,C(=O)(CCS(=O)(=O)C1CCCC1)NCC(CCOC)NC(=O)COC(C)(C)C 35592,C=CCC(C)C(=O)NN(CCNC(C1(C(=O)OC)CC=CC1)=O)C 35593,CC(C)(C(=O)NCC(O)CNC(C1CC(n2ccnn2)C1)=O)C(F)(F)F 35594,Cc1c(F)ccc(Br)c1C(=O)NC1CCC(C)(NC(c2cnccn2)=O)CC1 35595,C1(NC(C(C)OCCCCCC)=O)C=CCN(C(=O)CC2(C3CC3)CC2)C1 35596,Cc1cc(C)c(C=CC(=O)NC2(CO)CN(C(c3csc(CO)n3)=O)C2)cc1C 35597,C(=O)(C1=CC2(CCN(C(=O)Cn3cccn3)C2)C1)NC1C(C)CCCCC1 35598,C1(c2cn(C3CC(=CCC=C)C3)nn2)COCCN1C(c1ccccc1Cl)=O 35599,N1(c2nnc(-c3nc(C(=O)OCC)oc3)n2CC2CC2)CC2CCC2(C)C1 35600,c1(C(=O)NC2CCC(NC(=O)C3=C(Cl)CCC3)C2)c(Cl)ccc2ccoc12 35601,c1(NC(c2cc(CC)on2)=O)ccc(S(=O)(=O)N(CCOC)CC)cc1 35602,CCC(CC)CCCC(=O)N1CC2CCC1CC2NC(C1C=CC=CC=C1)=O 35603,N1(C(c2scc(CNC(C(C=CC)O)=O)c2)=O)CCc2c(cnn2C)C1 35604,CC(=O)CCN=C(NCC1COC(C)(C)O1)NCc1cccc(C(N)=O)c1 35605,C12(CNC(C3CCN(C(C4CCNC4=O)=O)CC3)=O)CCC(CC1)O2 35606,C(N=c1nc(C(=O)OC)c(Cl)c[nH]1)C1CCCC(NC(C(CCC)(C)CC)=O)C1 35607,c1(OC)cc(C(=O)NC(CNC(C2CCCC23CC3)=O)C2CC2)c(F)cc1N 35608,C(=O)(C(C)C(O)CC)N(CCN(C(C(C)(C)OCC)=O)C)C 35609,C1(CNC(C=Cc2n(C)cnc2)=O)CCN(C(=O)C=CC(=O)NC2CC2)C12CC2 35610,c1(C(=O)NC2CN(C(C(C)(C)OCC(F)(F)F)=O)CC2F)cc2sccc2[nH]1 35611,c1(C(=O)NCC2(F)CCC(NC(CC(COC)C)=O)C2)c([N+](=O)[O-])cnn1C 35612,C1(CNC(c2c(C(C)C)noc2)=O)CN(C(C2CC3CC3C2)=O)CCC1C 35613,Cc1cc(C(N2CCOC(C(C)NC(C3CCCCCC3)=O)C2)=O)cc(C)c1F 35614,C1(NC(COCCOC)=O)CS(=O)(=O)C2CN(C(c3nn[nH]c3Cl)=O)CC12 35615,C1(C(=O)NC2CC(NC(C3CC4(CC4)C3)=O)C2)CCC12CCCO2 35616,c1(C(=O)NC2C(NC(c3nncc(OC)c3)=O)COCC2)cc(C)c(Cl)cn1 35617,S(=O)(=O)(c1ccnc(C(F)(F)F)c1)Nc1ccc(C(=O)NC2CC2)[nH]1 35618,C12CCC(C1)n1cc(nn1)C1(CCCC1)CNC2=O.C1(CO)(CC2CCC2)CC1 35619,N1(C(c2c(C)con2)=O)CCC2(CC1)CN(C(c1csc3nccn13)=O)CCO2 35620,c1(C(=O)NCC2CC(NC(c3c(CC)ncs3)=O)C2)ccc2c(c1)C(=O)CCO2 35621,C1(c2nnnn2C(C)C)(Cc2cn(CC)nc2)CC(C)(C)C1.C1(=O)NCCN1 35622,CC1CC(CNC(=NCCN2CCCC2(C)C)NCc2ccccc2)CC(C)O1 35623,N#Cc1ccncc1NCc1cc(C(=O)NCc2ccc(Br)cc2Cl)ccn1 35624,C1(C2CCOCC2)(C(=O)NC(CCC(C)C)CO)CC1 35625,C(C(C(=O)NCCN(C(=O)C(C)(C)n1ccnn1)C)C(C)(C)C)OCC=C 35626,C(=O)(CCCC(=O)NCc1ccc(C(=O)NC)nc1)N(CCCCN(C)C)CC 35627,Cc1c(C(F)(F)F)n[nH]c1C(=O)NCCCCNC(=O)Cn1cnnc1O 35628,C(=O)(CCCCCC#N)N1CC(NC(c2cc(C)ncc2C)=O)C(C)C1 35629,c1(C(=O)NCCCC(C)NC(c2ccncc2Cl)=O)cccn(C)c1=O 35630,c1(C(N2CC(NC(C3(COC)CC3)=O)C(C3CC3)C2)=O)oc2ccccc2c1C 35631,c1(CNCC2N(CC(C)C)CCC2)n[nH]c2cc(F)ccc12 35632,c1(C(N2C(CN(C(C3C(C=C)C3)=O)C3CC3)CCC2)=O)nc2cccnc2s1 35633,CCC(CCC(=O)NCCN(C)C)N(C(=O)CN(CC(C)(C)C)C)C 35634,C1(CC(C)NC(C=C(COC)C)=O)CCN(C(=O)C(N2CCCCCC2)C)CC1 35635,c1(C(N2C(CNC(C(N3CCCCCC3)C)=O)COCC2)=O)ccc(C#N)n1C 35636,C1(CNC(C(C)(CO)OC)=O)CN(C(=O)CCc2nnc(O)nc2O)CC1(C)C 35637,c1(NC(CC2CCN(Cc3cc(OC)cc(OC)c3)C2)=O)[nH]nc2ncccc12 35638,c1(C(N2C(C(=O)N(C3CCCCCC3)C)CCC(C)C2)=O)cc[nH]c2nccc1-2 35639,N1(C(C(CN=[N+]=[N-])NC(=O)CCCn2ccnn2)=O)CC2CCC(O)C2C1 35640,n1(CNC(c2cc(OC)c(OCC3CCCO3)cc2)C#N)cnc2ccccc12 35641,c1(CC)ncc(C(=O)N(C2CCCCC2)Cc2cccnc2)c(C)n1 35642,c1(OC)nccc(C(=O)NCc2occc2C(=O)NC(c2ccccc2)C)n1 35643,C1(F)(CNC(CN(C2CC2)CC)=O)CCCN(C(=O)CS(C)(=O)=O)CC1 35644,c1(C(=O)Nc2cncc(C(=O)NCC(N)=O)c2)cccc2ccnn12 35645,c1(CN2CCN(C(c3ccncn3)C)CC2)ccc(C(F)(F)F)c(F)c1.C1CC1 35646,C1(C(=O)NCC(CNC(C(CC)=CC)=O)F)CCCC(NC(=O)OC(C)(C)C)C1 35647,N1(C(c2[nH]c(=NC)sc2)=O)CCC2(CC1)CN(C(C1CC1C(C)O)=O)CC2CO 35648,c1(CC(N2C(C)CC(NC(CC(CC)C3CC3)=O)C2)=O)ccc(O)c(C)c1 35649,C(=O)(CCCCCNC(=O)CCCOc1ccc(Br)cc1)N(C)C 35650,c1(CC(=O)N(CCOC)CCNC(C2CCC2)=O)cccc2cccnc12 35651,NC(=O)C1CN(C(C2(O)CCCCC2O)=O)Cc2ccccc21 35652,C(C)(CCC(=O)N1CCN(C2CCN(C(=O)C=C3CCC3)CC2)CC1)OC 35653,c1(C(=O)OCC)cc(Br)c(Cl)nc1N.c12cc(ccc1C)C(=O)N2 35654,C1(C(=O)NC(C)C)CCCCCC1NC(C1CC1(F)F)=O 35655,C(C)(C)(CC(=O)NC(C1CN(C(=O)CC2CCCS2(=O)=O)CCO1)C)SC 35656,c1(C(=O)NC2C(NC(C(C)(C)NS(C)(=O)=O)=O)CCCC2)cc(N)ccc1Cl 35657,N1(C(CSc2cn(C)nc2)=O)CCC(CO)C(NC(=O)CCOC2CC2)C1 35658,C1(C(=O)NCCNC=O)CCN(c2cnccn2)C1.C12CC1C2.COC 35659,c1(C(N(C2CCCOC2)CC)=O)cc[n+]([O-])cc1 35660,N1(CC(=O)N(CC(C)CNC(=O)CCC2CCCCN2C)C)CCC(=O)NC1=O 35661,c1(OC)cc(C(N2CC(C)(NC(=O)C=Cc3ccccc3)C2)=O)cc(N)c1N 35662,C(=O)(CC(C(C)C)Cn1cncc1NC(C1CN(CC)CCO1)=O)OC.C(C)=O 35663,C1(C(=O)NC2C(NC(C=CC(=O)OCC)=O)CC2)CC(=O)N(c2cnn(C)c2)C1 35664,C1(C)(OC)CCCN(C(C2CN(C(c3cnc(C)nc3)=O)CCO2)=O)C1 35665,C(=O)(CS(=O)(=O)CCC)N1CC(CCNC(CCC=CC)=O)OC(C)C1 35666,C1(NC(C2N(CC)CCC2)=O)CCCC(NC(=O)Cc2ncc(Cl)s2)C1 35667,N1(C=O)CCCN(C(N)=O)CC1.Cc1ccc(CC(=O)NC2(C3CC3)CCC2)o1 35668,C12(C(=O)NCCOCCNC(C3(CC4CCOC4)CCC3)=O)CCC1C2 35669,Nc1cc2[nH]c(O)nc2cc1C(N1CCCC1CF)=O 35670,Cc1nc(NC(C2CC(C)CN2Cc2cnn(C)c2C)=O)cc(Cl)n1 35671,C1(CNC(C(CC=C)(C)C)=O)CC2CCC(C1)N2C(=O)CC1CC(C)C1 35672,Cc1c(NC(C)CCC2CC2)ncnc1NCCOC(C)(C)C 35673,c1(CN(C)C)ccc(C(=O)NC2COCC2CNC(=O)CN2CCCC2=O)o1 35674,C1(CC(=O)Nc2cnc[nH]2)CC2(CC2)CO1.C1(=O)CCC2CC(C2)N1C 35675,CC1=CC(C(=O)NC(C)C(=O)N(CCc2ccsc2)C(C)C)SC1 35676,CC1CC2CN(C(=O)CCCCNC(=O)CCNC(=O)CCC(CF)CF)CCN2C1 35677,N1(C(CN2CCN(C(CN(C3CCC3)C)=O)CC2)=O)CC2(COCC(=O)N2)C1 35678,N(C1CSCc2ccc(Br)cc21)C(=O)NC1(OC)CCCCC1 35679,C(=O)(CCC1CCc2ccccc21)NCc1c(N(C)C)cc(C(=O)O)nn1 35680,C1(NC(=O)C=CC2CCCC2)CCN(C(C2CCCS2)=O)CC1F 35681,c1(NC(C(C2CC2)OC)C)[nH]c(=NCCc2nncs2)nc2scnc12 35682,n1(CC)cnc(C(=O)NC2CC2CNC(=O)C(C)NC(=O)OC)c1 35683,N1(C(C=C2CCC(C)C2)=O)CCCN(C(=O)CN2CCN(C)CC2)C(C(C)C)C1 35684,C(=O)(CC1=CCOCC1)N1CCC(C(C)(C)NC(=O)Cc2cccc(C#N)c2)C1 35685,C(N=c1cc(NCCc2ccccc2Br)nc(C(F)(F)F)[nH]1)C1(F)CCOCC1 35686,Cc1ccc2cc(C(N3CCC4CCC(C3)N4C(=O)COCCF)=O)ccc2n1 35687,CCC(C)CCC(=O)NC1CC2(NC(c3cccc(N(C)C)c3)=O)COC1C2 35688,C1(C(c2n(C)ncc2)C2CC2)CCN(C(=O)C(=O)NC(COC(C)(C)C)=O)CC1 35689,c1(C(=O)NCC(CC)(C)NC(=O)Cn2cccc2)cccc(C2CC2)n1 35690,c1(CC(N2CC(OCCNC(C(C)=CC)=O)C2)=O)ccc2ncccc2c1 35691,N1(C(C2CN(C(=O)OC)C2)=O)CC2CC1(CO)CN2C(=O)CC1(CO)CC1.CSC 35692,c1(C(C(=O)NCCC)N(c2ccccc2)CC)ccc(CC2CCOCC2)cc1 35693,C1(CCC)(C(=O)NCC(CCOC)NC(=O)CCCCSC)CCNC1=O 35694,N1(C(COCCC=C)=O)CC2ON=C(CNC(c3cccc4ncnn34)=O)C2C1 35695,CCCC(C)CC(=O)NCCC(C)NC(=O)CSc1cc(F)ccc1F 35696,c1(C(=O)NC(C2N(C(CCCC(=C)C)=O)CCC2)C)ccc2cc[nH]c2n1 35697,c1(OC)ncc(CNC(=NCC2CCCCC2)NC2CCC(C)(C)C2)cc1Cl 35698,c1(N2C3CN(c4nccc(OC)n4)C(C3)C2)ncnc2cc(C(C)(C)C)sc12 35699,n1(CC(=O)N(C(CC)CN(C)C(C2CN(CC(F)(F)F)C2)=O)CC)cnc(=N)[nH]1 35700,CN=c1[nH]c(=NCc2ccccc2N(C)C)[nH]c(=NCCC2CC3CCC2O3)[nH]1 35701,N1(C(C)=O)CCC2(CCC2NC(c2ccc3ncccc3n2)=O)CC1 35702,C#CCCCCCC(=O)NC1(CCOC)CCN(C(=O)Cc2ccnc(C)c2)C1 35703,C1(NC(COCCC)=O)(CF)CCN(C(c2sc(C(C)C)nc2C)=O)C1 35704,N#Cc1cccc(CN2CCC(Nc3ncnc4n[nH]cc34)C(O)C2)c1Cl 35705,c1(C(=O)NCCC(C)NC(c2c(CC)nns2)=O)ccc(C#N)n1C 35706,N1(C(c2c(OC)cc(C)cc2)C(=O)NC2CCCCC2)CCCC2CN(C)CCC12 35707,C1(NC(c2cnc(O)c(Br)c2)=O)CC12CCN(C(=O)CCCCBr)CC2 35708,C(C(C(=O)N(C)CC1CCCCN1C(C1CCOC(=O)CC1)=O)C(F)(F)F)OC 35709,Cc1ccc(C=CC(=O)NCCCNC(c2c(-c3cccs3)noc2C)=O)cn1 35710,c1(OC)ncc(Cl)cc1C(N1CCN(C(c2cc(C)co2)=O)CC1C(F)F)=O 35711,C(=O)(C(C)(C)CN(C(=O)Cc1ccsn1)C)NCCS(CC)=O 35712,N1(C(C2N(C(C)C)CCC2)=O)Cc2ccccc2C(NC(c2nsnc2O)=O)C1 35713,CC1(C(N2CCC(O)(CCNC(C3CCC4(CC4)C3)=O)C2)=O)COC(=O)N1 35714,c1(OCC(=O)NC(c2nocc2C(N2CCC(CC3CC3)C2)=O)C)cccnc1 35715,c1(C(=O)NC2(CC=C)CN(c3ncc(C#N)cc3F)C2)cnc2c(c1)ncn2C 35716,c1(NC(=O)NC(CC2CCCC2)CO)cccc2nc(O)nc(O)c12 35717,CC(C)CC(CNC(=O)CC1CCCCOC1)C(=O)NCC1(C)COCCO1 35718,N1(C(C2C(CC)CCCC2)=O)Cc2[nH]nc(C(N3CCCC3CN(C)C)=O)c2C1 35719,N1(C(CC2(CSC)CC2)=O)CC2COCC2(C(=O)NCC(O)C(C)(C)C)C1 35720,C1(C(=O)NCC(C2CC2)SC)CCN(C(=O)CC2CCCC(C)O2)O1 35721,C1(NC(C2CCCN(C(N)=O)C2)=O)CN(C(=O)CC2CCCCO2)CC2(CC2)C1 35722,c1(C(=O)NCC2C(NC(=O)C=CC3CCC3)CC2)cnc2[nH]ncc2c1 35723,Cc1c(C(N2CC(C(C)(C)O)(CNC(C3CCSC(C)C3)=O)C2)=O)[nH]ccc1=O 35724,CC(C)C(O)C(=O)N1CCCC1C1(C(N2CCOC(C(C)(C)C)C2)=O)CC1 35725,N1(C(CCC)C)CCC2(CC1)CC2C(=O)NC(C)CN(C)C 35726,CN1CCC(C)(C(=O)NCC2CCN(C(=O)Cc3cn[nH]c3)CC2O)CC1 35727,c1(C(=O)NCCN(CCOC)C(C2CC(=C3CCC3)C2)=O)c(C)n[nH]c1C 35728,C(C(C(=O)N1CCOC2CC12)C(C)(C)C)NC(COC(CC)C)=O 35729,c1(C(=O)NC(C)C#N)ccc2c(-c3cscc3C#N)nn(C)c2c1 35730,N1(C(CC2CC(C(C)(C)C)C2)=O)CC=CC(NC(C23CSCC2C3)=O)C1 35731,C1(NC(C2N(C)CCC2)=O)CC2CC1N(C(=O)Cc1cccc(C3CC3)c1)C2 35732,Cn1cc(C(=O)NC2CCC(NC(C3(C)COC3)=O)CC2)c(C(F)F)n1 35733,C#CC1CN(C(=O)CCC2CCCCN2C(c2cc(Cl)no2)=O)CCO1 35734,C1(C(N(C2(CC(=O)NC(C#C)CC3CC3)CC2)C)=O)Cc2ccccc2C1 35735,C(=O)(C(C)(C)F)N(CC(C)N(C(CC1CC(OC)C1)=O)C)C 35736,N1(CC)CCC(NC(=O)CCC(C)NC(=O)CS(C)(=O)=O)C1=O 35737,c1(C(C(N2CC(C(C)(C)O)(CNC(CCOC)=O)C2)=O)C)ccc(N(C)C)cc1 35738,C12(C(=O)NC(C(C)F)C)CC(CCO1)N(C(C1CN(C)C(=O)N1)=O)C2 35739,CCC(C)(C)C(=O)NCC1C2CN(C(=O)CNC(c3cccs3)=O)CC12 35740,c1(C(N2CC(NC(C3(CC)CC3(F)F)=O)C2)=O)ccccc1S(C)(=O)=O 35741,CCCC(C)N=c1ccc(Br)c(S(=O)(=O)NCc2cccc(Br)c2)[nH]1 35742,c1(C(=O)NCC2CN(C(C3CCC(=O)NC3)=O)CC2O)[nH]cc2c1CCC2 35743,N1(C(Cn2nnc(C)n2)=O)CC=C(C(=O)N2CCC(OC3CC3)CC2)CC1 35744,C(=O)(CCCCC(F)(F)F)NC12CC(NC(CC(C=C)C)=O)(C1)C2 35745,C(CC(C(C)(C)C)NC(=O)CC1CN(C)C1)N(C(c1c(C)c[nH]c1)=O)C 35746,CCCCCCC(c1nnnn1CCCOC)NC(c1ccc(F)cc1)C(C)C 35747,Cc1cnc(F)c(CNc2cc(NCCN3CCC(C)(F)C3)ncn2)c1 35748,Cc1nnsc1C(=O)NC1(CNC(C2(C(C)C)CC2)=O)CC1 35749,CN1C(=O)OCC1C(=O)NC1CC(CNC(c2cccc(=O)o2)=O)C1 35750,c1(C(=O)NCCCN(C(C(C(=O)OC)OC)=O)C2CC2)cc2n(n1)CC(F)C2 35751,C12(C(=O)OC)CC1CN(C(=O)CC(O)CNC(c1cc(C3CC3)[nH]n1)=O)C2 35752,c1(C(N2C(C(N)=O)CCC(C)C2)=O)coc2c1CN(C(=O)CC1CCC1)C2 35753,C1(CC(N2CCCC(O)C2)C(=O)NCCC2CC2)CCC(F)(F)CC1 35754,N1(C(C(C)=CC)=O)CCC(C2CCCN(C(C3CS(=O)(=O)C3)=O)C2)C1 35755,c1(C(=O)NCC(CC)N(C)C(c2cnsc2C)=O)n[nH]c(C)n1 35756,C(=O)(C1=CCCCCC1)NCC(CNC(c1c(C(=O)OC)c(C)[nH]n1)=O)CO 35757,n1(C(C)C)ncc(C(N2CCCC2CN(C(=O)CSCc2ncc[nH]2)C)=O)c1N 35758,CC1=C(C(=O)NCC2CCC(N(C(=O)CN3CC(C)(C)C3)C)CC2)COCC1 35759,CCCC(C)CC(=O)NCC(O)CNC(=O)COc1ccc(CC#N)cc1 35760,N1(C(C=CC(=O)OCC)=O)CC2CC(NC(=O)Cc3cnco3)CC2C1 35761,C1(NC(=O)CC2CC(C(F)F)C2)CN(C(=O)Cc2cncs2)CC1C1CC1 35762,N1(CC)C(C)CN(c2nnc(CC3CCOC3)n2CCCN2CCCCC2)CC1C 35763,Cc1ccc(C=CC(=O)NC2CC2NC(c2cnc(C(C)(C)C)s2)=O)cc1Cl 35764,c1(C2(C(=O)NCC(C)CN(C(=O)C(C)C3CCC3)C)CCC2)ccccc1 35765,c1(OCC)ccc(NC(=O)CC2CC(NC(c3occc3COC)=O)C2)cn1 35766,N1(C(C(CC)(C)COC)=O)CC(NC(c2cnn3ccccc23)=O)C2(CCC2)C1 35767,C1(N(C)C)CCC(C(=O)NC(C2CCCC2)CNC(=O)C=CC2CCCC2)CC1 35768,C1(C)(OC)CCN(C(=O)C(O)CCCNC(c2csnc2Cl)=O)CC1 35769,C1(CN2CC(F)(C(=O)NC3CC(NC(=O)CC4CC4)CN3)C2)CC(C2CC2)=NO1 35770,CC#CCC(C(=O)N(CCOCC)CC)NC(C1C2CC3C(C2)C13)=O 35771,Cc1cc(F)cc(Br)c1C(=O)NC1CC2CCC1N2C(C1CCC(=O)C1)=O 35772,c1(C(=O)NC(CC(F)F)C(=O)NCC(O)(CO)CO)ccnc2cc[nH]c12 35773,c1(C(=O)NCC2CCC(C)N(C(c3ccon3)=O)C2)cccc([N+](=O)[O-])c1Cl 35774,c1(C(=O)NCC(CC(F)(F)F)NC(CSC)=O)c(C)c(C)cc2ccccc12 35775,C#CC1(Nc2ccccc2)CCN(CCC2CN(C)C(C)(C(=O)N(C)C)C2)CC1 35776,c1(CN(C)CCOCCNC(c2cc(Cl)c[nH]2)=O)ccc([N+](=O)[O-])cc1 35777,C1(S(C)(=O)=O)(NC(=O)NCCc2c(OC)ccc(C(F)(F)F)c2)CC(O)C1 35778,c1(C(C)C)nnc(C(=O)NC2CN(C(=O)C(C)(C)C3CCCCC3)C2)s1 35779,c1(C(=O)NC2CC(NC(C3CCCO3)=O)C2)c[nH]cc(F)c1=O 35780,N1(C(C(C)O)=O)CCC2(CCC(NC(c3ccc(=O)oc3)=O)C2)CC1 35781,CC1(C)CCC(C(N2CC3CC3(CNC(c3ccc(Cl)o3)=O)C2)=O)O1 35782,N1(C(c2scc(C(C)=O)c2)=O)CC(O)CC1CNC(=O)CCOC1CCOCC1 35783,c1(NCC(C(C)C)O)cc(S(=O)(=O)NCCc2cn(C)nn2)ccc1C#N 35784,CCC1=NOC(C(=O)NCCC(O)CNC(=O)C(F)(F)CO)C1 35785,CC1(F)CN(C(=O)C(O)C2CCC2)CCN(C(c2c(Cl)ccnc2F)=O)C1 35786,c1(CC)ccc(C(N2CC(CF)(NC(=O)C=Cc3cncn3C)C2)=O)cc1CC 35787,N1(C(CC(C)SC)=O)CC2CC(C(=O)N(CCCO)C)C(C2)C1 35788,C1(CN2CCCC(C)(SC)C2)CCCCN(C2CCC2)C1.c12cn(nn1)C2 35789,CCCCCCCCCC(=O)NC1CN(C(=O)Cc2ccsc2)CC12CCC2 35790,C(=O)(CCCCCNC(C1C(C)(C)C1(F)F)=O)NCc1nc(CC)sc1 35791,C12(C(N(C(CC)CO)CC)=O)CC(C)(CN1C(c1ccccc1C#N)=O)C2 35792,C(=O)(C(CO)C(F)(F)F)NC(CCC=C)C(=O)NC1CCOC1C 35793,C(=O)(C(O)CC(F)(F)F)N(C)CCNC(C1CCC(Oc2ccncc2)C1)=O 35794,C1(C(N(CCCF)C)=O)CCCCN(C(C2(N(C)C)CC2)=O)C1 35795,CC1CC(=O)NC(C(N2CC(NC(c3cn(CCC(C)(C)C)nn3)=O)C2)=O)C1 35796,c1(C(N2CCOCC(C(=O)OC)C2)C(=O)NC)ccn(C(C)C)c(=O)c1 35797,c1(NC(N2C(CC)CN(C)CC2)=O)ccc(S(=O)(=O)N(C)C)cc1 35798,c1(CN=C(NC(C#C)C(C)(C)OC)NC2CCC2)ccc(C#N)cc1Cl 35799,CCC(C)C(C(=O)N(CC(C)(C)C(=O)NCC1=NOCC1)C)OC 35800,Cc1cc(C)c(C(=O)N(C(C)CNC(=O)COCCN(C)C)C)[nH]1 35801,C=C(CNC(C1CC1CN(C)C)=O)CCNC(c1ccoc1C)=O 35802,CCCCCC(CC)C(=O)NC(CNC(c1nocc1C)=O)CO 35803,c1(C(=O)NC(CNC(C(CC)n2nccc2C)=O)C2CC2)cc2cccnn2n1 35804,c1(C(=O)NC2C(NC(C(C)O)=O)COC2)cnc(C2CCC2)nc1O 35805,CCCC(C(=O)NC)NC(=O)CC1(N(C)C(C2CC(C)(C(N)=O)C2)=O)CC1 35806,N1(C(CCNC(=O)C=CCl)=O)C(CNC(=O)C(O)c2cnc[nH]2)CC2CCCC12 35807,c1(CCCN(C)C(N2CCC(SCC)C2)=O)nccc(C)n1 35808,C1(CC)CCCCN1C(=O)COCCNC(=O)CCC1CC1(C)C 35809,N1(C(CCS(C)=O)=O)CC(NC(c2cccc3c2CCC3)=O)C(C2CC2)C1 35810,C(C(C)C(C)C(=O)NCC1CN(C(C2CCC(=O)N(C)C2)=O)CCO1)OC 35811,C1(CN(CC(C)(C)Cn2cc(-c3c[nH]c(C(=O)O)c3)nn2)C(C)(C)C)C(F)(F)C12CC2 35812,CCC(Cc1ccccc1C)C(=O)N1CC(NC(c2csc(CO)n2)=O)C(C)C1 35813,C1(N(C(c2cnc(CC)s2)=O)C)CCN(C(c2c[nH]nc2-n2cnnn2)=O)CC1 35814,c1(C(N2CCC(NC(C3CCCOCC3)=O)CC2)=O)cc(F)c(O)c(Cl)c1 35815,C1(NC(c2ccnc(CO)c2)=O)(CF)CCN(C(=O)CC2CCCC2(F)F)C1 35816,C1(C=O)(COC)CN(C(c2ccc(CO)o2)=O)C1.N(CC)CC1CC1 35817,N1(C(C2N(C(CCC)=O)CC=C2)=O)CCC(N=[N+]=[N-])C1 35818,N1(C(C(C)N=[N+]=[N-])=O)CC2CCCC2(CNC(c2cnnc(O)c2)=O)C1 35819,C(=O)(C(C)(C)CCCO)NCCC1CCN(C(C(C(C)(C)C)NC(N)=O)=O)CC1 35820,Cc1nocc1NC(=O)CNC(=O)CNC(c1ccc(F)s1)=O 35821,N1(C(CC2CC(=C)C2)=O)CCCC(O)(CN(C(=O)CCCn2cccn2)C)C1 35822,C1(C(=O)NCC(CN(C)C(C2CC(F)C(=O)N2C)=O)(C)C)C2C3CCC(C3)C12 35823,N1(C(C2N(C(c3c(C#C)cn(C)n3)=O)CCC2(C)C)=O)CC2(COCC(=O)N2)C1 35824,N1(C(C(=O)N(C)CC2CCCN2)=O)CC2CCCC(N)C2C1 35825,c1(C(N2CC3C(CNC(C4C(=C)C4)=O)C3C2)=O)ccc2c(c1)nc(C(F)F)n2C 35826,c1(OC)cc(C(=O)NCC23CC2CN(C(c2n[nH]cc2C)=O)C3)nc(Br)c1 35827,C1(C)(CNC(CN(C)C(N)=O)=O)CN(C(=O)CC2CCCC23CC3)CCO1 35828,C1(CNC(CCC(C)OC)=O)CN(C(c2nnn(C(C)C)c2C)=O)CC(C)(C)C1 35829,N1(C(CC(C)OC)=O)CC2CCN(C(c3nccc4[nH]ccc34)=O)C(C2)C1 35830,c1(NC(CCCN(CCOCC)C)=O)cccc(F)c1CNC(=O)COC(C)=O 35831,c1(C(=O)NCC2(C(N)=O)CN(C(C3C4CCCOC34)=O)C2)ccc(Cl)c(F)c1F 35832,c1(OC)cccc(C(=O)N(C2CCCC(N(C)C(c3nnsc3C)=O)C2)C)c1F 35833,N1(C(Cc2c(C)n(C)cn2)=O)CC(NC(C2(Cl)CC2(F)F)=O)CC(C)C1 35834,C1(CN2CCC(F)(CN3CC(CC(=O)OC)C3)C2)C2CCC1(c1ccccn1)C2 35835,c1(CC)ccc(C(=O)NCC(CO)NC(c2ccc(C)cc2C)=O)cc1C#N 35836,n1(CC)cncc1CNCc1cc(C)on1 35837,c1(CC)c(C(C)NC2CCN(C3CCCC3O)CC2)oc2ccccc12 35838,c1(C(N2CCC(N3CCN(C(CC)=O)CC3)CC2)=O)c(F)cc(F)cc1Br 35839,CC1(C)CCC(C(N2CCOC(Cn3cncn3)C2)=O)O1 35840,CC(C)(CC1CCOC1)C(=O)NCC1CCN1C(=O)COCC1CCOCC1 35841,N1(C(=O)C(F)C2CCCC2)CCC(N(C(=O)C(F)C2CC2)CCO)CC1 35842,C1(NC(C2(OCC)CCSCC2)=O)COCCN(C(c2csnc2Cl)=O)C1 35843,N1(C(=O)CCc2cc[nH]n2)CCC2(CCCN2C(c2ccccc2Cl)=O)C1 35844,O=C(C1=CC2CCCCCC12)N1CCN(C(c2ccc3c(n2)CCCC3)=O)CC1 35845,N(C1=NC2CC3CC3C2N1)c1ccc(OC(C(F)F)(F)F)cc1 35846,C(C(C)(C)CNC(=O)C(CC1CC1)NC(=O)CCOC(C)=O)OC.C(C(C)C)O 35847,c1(C(=O)NC2CC(NC(C3(O)CCCC3)=O)C23CCC3)nnn2c1CSCC2 35848,C(=O)(C1=CCS(=O)(=O)C1)NC1C(N(C)C(C2CCCC(=O)N2)=O)CCCC1 35849,C#CCC(CC(=O)NCc1cccc(C#C)c1)NC(c1cnn(C)c1Cl)=O 35850,c1(NCc2cn(CC3(n4ncc(C)c4)CCCOC3)nn2)ccc(F)cc1Cl 35851,Cc1nn(CC(N2CCCC(C(C)NC(=O)Cn3nnc(=O)[nH]3)C2)=O)c(=O)o1 35852,C1(C(N(C(CC)C2CC2)C)=O)CC2C=CC1N(C(=O)CCNC(=O)CO)C2 35853,N1(C(C2CCC(C)O2)=O)CC(CNC(c2cc3ccccc3o2)=O)OC(C)(C)C1 35854,C1(N(C(CN(c2ccccc2)CC)=O)C)C2CN(C(=O)C(F)=C3CC3)CC12 35855,N1(C(CC=CC)=O)CCC2(NC(c3cccc(Br)c3C)=O)CCCCC12 35856,c1(CN2CCC(CC(=O)Nc3cnc(Cl)c(Cl)c3)C2)cnc2ccccn12 35857,N(C1CCc2cc(CNC(C3(O)CCCCC3)=O)ccc21)C(C(CCC#C)O)=O 35858,c1(CC)ccc(CNC(N2CCCC(C)(N(C)C)C2)=O)c(C(F)(F)F)c1 35859,c1(C(=O)NC2CC3CN(c4nc(COC)nc(C)c4)CC32)ccc2ncsc2c1 35860,C1(c2cn(C)nc2)CSCCCN1c1nc(Cl)ns1.c12ccccc1S2 35861,C1(C(=O)NC2COCC2NC(c2cnc(O)s2)=O)(OC)CCOCC1 35862,Cc1cc2cc(C(N3CC4CC3(CNC(=O)CN(C)C(N)=O)C4)=O)[nH]c2cc1Cl 35863,C(CC)(CC(=O)NCC1(CO)CCCC1)NC(CC=C)=O 35864,S(=O)(=O)(c1ccccc1)NC(C(=O)NCC(CNC(c1c(C)cnn1C)=O)O)C 35865,Cc1cc(F)ccc1C(=O)NC1CCCN(Cc2scnc2C)C1 35866,Cc1cc(C(=O)N(CCCCNC(c2ccc(C(F)F)nc2)=O)C)c(Cl)cc1F 35867,N1(C(C(C2CCCN(C(C3CNC(=O)CN3C)=O)C2)C)=O)CC2(CO)CC2(CO)C1 35868,C(CC(=O)NCCC(COC)OC)(C(C)C)NC(C(CC)(C)C)=O 35869,CC(=O)n1ccc(-c2nc(COC(c3ccccc3F)COC(C)(C)C)cs2)c1 35870,c1(OC)nccc(C(=O)NCC2CN(C(C3(n4cncn4)CC3)=O)C2)c1F 35871,c1(NC(C2C(NC(c3c(SC)cccc3)=O)CCC2)=O)cccc2c1OCO2 35872,C(c1cnn(C)c1)=CC(=O)NCC(COC)NC(c1csnn1)=O 35873,c1(C(=O)NC(C)C(CO)NC(c2cnc3cccnn23)=O)cccc2nn[nH]c12 35874,c1(C(=O)NCCN(C(CCC#C)=O)CCOC)cc(Br)c(OC)s1 35875,CCCCN=C(NCC1(O)CCC1)NCC1CCCCN1S(C)(=O)=O 35876,CC1CN(C(=O)CCCC2CCC2)CCC1NC(=O)CCc1cncc(Br)c1 35877,C(=O)(CC(C)COC(C1(CNC(=O)OC(C)(C)C)CC1(F)F)=O)OC 35878,C1(NC(c2cc(CC)sn2)=O)C=CCN(C(c2nonc2CC)=O)C1 35879,c1(C(=O)NCCN(C(CCC(=C)Cl)=O)CC)cc(C(=O)OC)cc(C(F)(F)F)c1 35880,c1(NC2CCC(CCCC)C2)ccc(F)c(NC(=O)N(C)C)c1 35881,CCC(C)CC(C(=O)NCC1(COCC)CC1)NC(C1CCN(C2CC2)C1)=O 35882,CCC(C)(C)OCC(=O)NCC(C)CN(C)C(C1(C(C)(C)O)CC1)=O 35883,N1(C(c2c(C)nccn2)=O)CCN(C(=O)CC2(O)CCOC2)C(CC2CC2)C1 35884,C1(NC(CCCC(N)=O)=O)CC2CC1CN(C(C1(c3cnccc3Cl)CC1)=O)C2 35885,N1(C(C2(CC)CCCC2O)=O)CC2CCC1CN2C(=O)Nc1c(C)cccc1C 35886,C1(N(C(c2cscc2Br)=O)CC)CCCN(C(=O)CC2CCCC(O)C2)C1 35887,C1(C2CCN(C(=O)CCOCC(F)(F)F)CC2)(NC(CC2C(C)CCC2)=O)CC1 35888,CC1(CNC(C2CC(C(F)(F)F)C2)=O)CCN(C(C2(O)CC(F)(F)C2)=O)C1 35889,Cc1ncc2n1CCC(C(=O)NC1(CF)CCN(C(c3ccncc3Cl)=O)C1)C2 35890,C#CCCCCCC(=O)N1CCC2CN(C(=O)CSCC(C)C)CC12 35891,CCCCC(C)CCC(=O)N(CC(=O)NCCOCC1CCOCC1)CC 35892,c1(C(=O)NCC2C(NC(COCCCOC)=O)CC2)sc2ccccc2c1Cl 35893,c1(OC)cccc(C(N2CCCNC(=O)C2)C(=O)NC(c2ccccc2)C)c1Br 35894,c1(OC)ccc(C(N2CCC(C)(C)C2CNC(=O)C#CC(=O)N(C)C)=O)cc1C 35895,C12(CNC(CC(C)SC)=O)COCCN1CCN(C(C1CN3CCN1CC3)=O)C2 35896,CSC1=C(C(=O)NCC2(CCNC(=O)C(n3ccnc3C)C)CC2)CCCC1 35897,c1(CC)noc(C)c1C(=O)NC1CCCC(N(C)C(c2ccn(CC)n2)=O)C1 35898,N1(C(Cc2cn(C)nc2)=O)CC(NC(C2CC3CCC3C2)=O)C2(CC2)C1 35899,C1(C(=O)NCC=C2CCN(C(C3(C(N)=O)CCC3)=O)CC2)CNc2ccnn2C1 35900,C1(C(=O)OCC)CCN(C(=O)OC(C)(C)C)C1C(=O)N(c1ccc(C)cc1)CC 35901,C1(NC(C=Cc2ccc(SC)s2)=O)CN(C(C2(CO)CCCCC2)=O)CC12CC2 35902,c1(C(C(=O)O)NC(C2CN(C(=O)NCN)C2)=O)ncccn1 35903,C1(CNC(C2(CC(=O)OC)CC2)=O)C2CCCC1N(C(c1[nH]cnc1C)=O)C2 35904,c1(OC)ncnc(OC)c1N1CCN(C2CCC(F)(F)CC2)CC1 35905,CCCCCC(CC)C(=O)N1C2CCC1CC(CNC(c1cc[n+]([O-])cc1)=O)C2 35906,N1(C(C2(CC(C)C)COC2)=O)CCC2(CC1)CC2(CO)CNC(C1CC(=O)N1)=O 35907,Cc1nc(C(=O)NC2CC(C)(NC(C3(C)CCN(C)C3=O)=O)C2)c2ccccn12 35908,Cc1c(C(=O)NC2(C3CCCN(C(C4CCO4)=O)C3)CC2)oc2ccc(F)cc12 35909,c1(-c2ccc(CNC(C(C)(C)C)=O)cn2)ccc2c(c1)OCCN2 35910,C1(NC(c2c(CC)noc2)=O)CC(CNC(c2cccc(F)c2)=O)C1(C)C 35911,c1(CC)cc(C(=O)N(CCCC(=O)NCCC2CC2C2CC2)C)ncn1 35912,c1(C(=O)NC2C(NC(c3cc(C)nc(C)c3)=O)COC2)cc2nccn2c(O)n1 35913,C1(C(=O)NC(C2CCCN(C(c3c(C)nn(C)c3)=O)C2)C)CCc2nc[nH]c2C1 35914,N1(C(C2ON=C(CC)C2)=O)CCC2CCCC2CC1.N12CCN(CC1)C(=O)C2 35915,C1(NC(=O)CC2CC2C(F)(F)F)CCCCN(C(=O)C=Cc2ccccc2)C1 35916,CCCC(C(=O)NCC1(C)CCCN1C(=O)C(F)C(C)C)OCC 35917,C(C)(CC(C)(C)N1CCCC1)(c1n(CC)nnn1)NCCSc1cncn1C(C)C 35918,S(=O)(=O)(c1ccc(C2CC2)cc1F)N(C(C)C)C1CC1 35919,CCCC(C)(O)CC(=O)N1CC(C(C(=O)NC2CN(c3ncco3)C2)OC)C1 35920,N1(C(C(C)=C2CC2)=O)C2CCC1C(C(=O)NC(c1ccns1)C)C2 35921,c1(C(C)=O)cc2ncc(C(C)C)cc2[nH]1.c12cc(C(F)(F)F)ccc1N2 35922,N1(C(C2CC=C(C)CC2)=O)CCN(Cc2cc(Cl)ccc2F)C2CC12 35923,N1(C(c2c(C)n3c(n2)scc3)=O)CCC(C2CC(NC(C3SCCCS3)=O)C2)C1 35924,c1(C(=O)NCC(CN(C)C(c2ccnn2C(F)F)=O)O)coc2ccc(O)cc12 35925,CC(CCc1ccccc1)CC(=O)N1CCCC1CNC(=O)C=CC1CC1 35926,Cc1[nH]nc(CNC(=O)C(c2cccs2)NC(=O)C=Cc2cncs2)c1C 35927,c1(CC)cc(C(N2CCC(CC(=O)N(CC(C)C#N)C)C2)=O)on1 35928,N1(C(C=NOC)=O)CC2CC(NC(C3(C4CCCO4)CC3)=O)C2C1 35929,C1(COC)CN(C(c2cc(Br)c(C)cn2)=O)CCN1C(c1cnc(O)o1)=O 35930,c1(C(=O)NCCC2N(C(CSc3onc(C)n3)=O)CCC2)c(C)cccc1C 35931,Cc1c(C(=O)N(C)CCOCCNC(=O)C(C)C(C)C)cnn1C1CCOCC1 35932,Cc1ccc(C(N2CCCC(C)(NC(c3cscc3F)=O)C2)=O)c(Cl)c1 35933,C1(CNC(C2(C(CC)(F)F)CC2)=O)(NC(C2CC3C=CC2O3)=O)CC(F)(F)C1 35934,N1(C(c2ccc(C(=O)OC)o2)C(=O)NC(C)C)CCOC(C2CC(F)(F)C2)C1 35935,C(=O)(C1CCCn2ccnc21)NCCOC1CCN(C(CC2CC(=O)C2)=O)CC1 35936,n1(CC(N2CCN(C(C(=O)NC)C)CC2)=O)ccc2ncc(Br)cc12 35937,N1(C(CCC2C(C)(C)C2)=O)CCOC2(CCC(Nc3ncc(Br)cn3)CC2)C1 35938,N1(CC)CCCC1C(=O)NC1CC1CNC(C1CC2CC2C1)=O 35939,C1(CN(C(CC(C)O)=O)C)COCCN1C(c1cncc(C(C)(F)F)c1)=O 35940,c1(C(=O)NC(CC(C)NC(c2c(C)cn(C)c2)=O)C)ccc(Cl)cc1F 35941,[N-]=[N+]=NC1CN(C(C2OCCO2)=O)CC1NC(c1c[nH]nc1-c1ccc(Cl)s1)=O 35942,Cc1[nH]c(C)c(C(=O)NCC2CN(C(c3cn(C(F)F)cn3)=O)CC2O)c1C 35943,c1(CC)onc(C)c1C(N1CCCC(C(=O)NCCCCC(=O)NC)C1)=O 35944,Cc1ncc(Cl)cc1C(N1CC(CC(C)NC(c2cncc(F)c2Cl)=O)C1)=O 35945,N1(C(C(C(CC)C)O)=O)CC(NC(C2OCC2(C)C)=O)CC(C)(C)C1 35946,c1(C(=O)NCCC(C)(C)NC(C(C)OC2CCOCC2)=O)ccc2c(c1)COC2 35947,c1(C(N2CCN(C)CC2CNC(C2CCS2(=O)=O)=O)=O)ncnc2c1ccn2C 35948,C1(CC)(CO)CCN(C(=O)C(CNC(=O)C(F)(F)COC)CC2CCCC2)C1 35949,c1(C(=O)OC)cc2c(N3CCC(=CCN(C(=O)CC4CC4)CC)CC3)[nH]cnc-2n1 35950,c1(C(=O)NC(CNC(c2ccc(C)nc2O)=O)(C)CO)nccc2ccccc12 35951,C1(C(N2CCCC(=C)C2)=O)CC1C1CN(C(C2(C)CNC(=O)C2)=O)C1 35952,Cc1cc(F)ccc1CNC(C1CC2(CC2)CN1C(=O)C(Cl)Cl)=O 35953,O=C1NC(=O)C2(CN(C(C3CCCC3CNC(=O)CCC3CCOCC3)=O)C2)N1 35954,CC(C)=C=CC(=O)NCCc1ccc(CNC(=O)CN2CCCC2)cc1 35955,C(C(C(=O)N1CC(C(N)=O)C1)C(C)C)NC(C1(CC(C)C)CC1)=O 35956,C12(CC(CO)C1)C(=O)N2.c1(C(=O)NC(C23CC(CO2)C3)C)cc(Cl)no1 35957,C1(SC)CN(C(=O)CCN2CCCS2(=O)=O)CC1NC(=O)C#CC1CC1 35958,C1(N(C(=O)CCc2nnc(-c3ccncc3)o2)C)CN(C(=O)CC2CC2)CC1F 35959,C1(NC(CN(CC(=O)NC(C)C)C)=O)CCCCN(C(=O)CC2CCOCC2)C1 35960,CC(CC(=O)NC1C=CC(CNC(c2cc(Cl)n[nH]2)=O)C1)n1cccn1 35961,c1(NC(c2cnc(Br)s2)=O)cc([N+](=O)[O-])c(Br)cc1OC(F)(F)F 35962,C#CCCCCCC(=O)NCCCN1CCN(C(=O)CC2CSCCO2)CC1 35963,Cc1nc(C(C)NC(C2CCN(C(c3c[nH]nc3C)=O)C2)=O)n[nH]1 35964,c1(C(=O)NCCCCNC(C2CCCN(C(C)=O)C2)=O)cc(F)c(F)c(F)c1 35965,C1(C(N(C(CCC)Cc2ccccc2)C)=O)CC2CC(=O)C1O2 35966,C1(COCC)CCCN(C(=O)C(C2CCOC2)NC(=O)CC2CN(C)C2)C1 35967,C(=O)(CCCCC(C)(C)C)N1CCC(NC(COCc2ncc(C)o2)=O)C1(C)C 35968,Cc1nc(C2CCCCC2)nc(O)c1C(=O)NCC(C)C1CC1 35969,c1(C(N2CCC(NC(c3c(C=C)cnn3C)=O)C2)=O)c(Cl)ccc(F)c1F 35970,N1(C(CCOC)=O)CCC(C)C1C(=O)N(C)CCn1ccnc1C 35971,C1(O)(C(=O)NC2CCN(C(C3C4(C(=O)OC)CC43)=O)C(C)C2)CCC(C)(C)CC1 35972,N1(C(C(CN(CC)CC)F)=O)CCC(F)(NC(C2CCOC2=O)=O)CC1 35973,C1(NC(C(=O)N(C)C)=O)CCCN(C(c2coc3c2COC3)=O)CC1 35974,n1(CC(N2C(C(=O)OCCCC(=O)c3ccncc3)CSC2)=O)ccccc1=O 35975,N1(C(CCN(C(C)=O)C)=O)C2CCCC1CN(C(C13CC(C)(CCO1)C3)=O)CC2 35976,N1(C(CCCOC(C)=O)=O)CC(F)(F)CC1CCNC(=O)COC1CC1(F)F 35977,Cn1nc(C(=O)NCCC2CCC(NC(C3(CF)COC3)=O)C2)cc1Cl 35978,C1(NC(C2(CO)CN(C(C(SC)SC)=O)C2)=O)CC2(CCC2)C1O 35979,c1(OC)cc(C(=O)NCCN(C(=O)CCCF)Cc2cccc(Cl)c2)cc(Cl)n1 35980,C1(C(=O)NCC2(OC)CC2)CCCCC1NC(=O)C(C)(C)C1CC1 35981,C1(C(=O)NC2CCC(NC(Cc3ccn(C(C)C)n3)=O)C2)CC2(CCO2)C1 35982,Cc1cccc2c1CC(C(N1CCC(NC(c3occc3Cl)=O)C1)=O)O2 35983,Cc1c(CCC2CCCN2C(c2ccc(SCC#N)cc2)=O)cccc1F 35984,c1(C(N(CC(C)NC(CC2ON=C(C)C2)=O)C)=O)cn(C)c(C)cc1=O 35985,N1(CCn2c(C)ncc2)CCCC(C(=O)NCC2=CCCCC2)C1 35986,O=C(C1=C(Cl)CCCC1)NC1CCCC1C(N1CCC(c2nc[nH]n2)C1)=O 35987,N1(C(C(c2ccccc2)C)=O)CCCC1CCCNC(=O)CCc1cccnc1 35988,CN1CCC(C)(C(N2CCOCC2CN(C(=O)C(C)(C)c2ccns2)C)=O)C1=O 35989,C1(CNC(c2c(SC)cccn2)=O)CN(c2cnc(F)cn2)CC2(CCC2)O1 35990,c1(CNC(C(C2CCN(C(CC3(CC)CCC3)=O)C2)(C)C)=O)cc(C)c(C)[nH]1 35991,c1(CC)cc(C(=O)NCC2CCCN(C(=O)CC3CC(F)C3)C2)cc(O)n1 35992,N1(C(C2(COC)CCCO2)=O)CCCN(C(c2cnn(C3CC3)c2C)=O)CCC1 35993,C1(CNC(C2(CC)CC(C)(C)C2)=O)CN(C(=O)CC2CCCC2)CC12CCC2 35994,N1(C(CCC=CC)=O)CCOC(C)C1C(=O)NCCC(C)C(C)C 35995,[N-]=[N+]=NC1COCC1NC(=O)Cn1cc(CN2CC3CC3C2)nn1 35996,C1(C(c2n(CC(=C)C)nnn2)NCC2(OCC)CCCOC2)CC2(CCC2)C1 35997,n1(CC)cc([N+](=O)[O-])c(C(=O)NCC(O)CN(C(=O)CNC(=O)OC)C)n1 35998,N1(C(c2nc(O)cc(C(C)(C)C)n2)=O)CCC2CCC(C1)S2 35999,C1(C(=O)NC(CCC)C(=O)N(C)CC2CCOC2C)CCCCC1(C)C 36000,Cc1ccnc2ccc(C(=O)NCC34CC3CN(C(C3CCC3(F)F)=O)C4)cc12 36001,N1(CC(=O)NC(CNC(C2CN(C(N(C)C)=O)C2)=O)C2CC2)CCCCC1 36002,C1(NC(C2CC(=C)C2)=O)(COC)CCCN(C(c2ccc(F)c(Cl)c2)=O)C1 36003,c1(CC)cc(C(N2CCC(C(C)NC(c3cn(C(C)C)cn3)=O)CC2)=O)nn1C 36004,C(=O)(C(C)CCC(C)(C)C)N(C)CC1CCC1.c1(C(=O)OC)ncc(F)cn1 36005,CC(O)C(C(=O)NCC1(n2ccnc2)CC1)NC(=O)COc1cccnc1 36006,c1(NC(c2ncccc2Cl)C)nccc(NC2CC(C(N)=O)C2)n1 36007,N1(C(c2n(CC#C)ccc2)=O)CC(NC(c2cc(CC)cc(F)c2)=O)C2CC2C1 36008,c1(C(=O)NC(C2(CN(C)C)CC2)C)ccc(CNC(=O)Cn2cnnc2)o1 36009,N1(C(c2ccc(C(C)=O)cc2)=O)CCC(CO)C(NC(c2cc(C)[nH]n2)=O)C1 36010,S(=O)(=O)(c1ccccc1C(=O)O)NC(c1ncc(OC)nc1)(C)C.C(=O)OC(C)=O 36011,Cc1ccc(C)c(C(=O)NCC2CCCN2C(=O)Cc2cc(F)ccc2Cl)c1 36012,N1(C(C(C)C)=O)CC(C)(C)OCC1CNC(=O)C(C(C)C)n1cccc1 36013,C(=O)(C(F)C(C)(C)O)NCCOCCN(C(CC1C(C)C(=O)CC1)=O)C 36014,N1(C(Cn2ncc(C)c2)=O)CC2CC1CN2c1cc(-n2ccnc2)ncn1 36015,c1(NC(C)=O)c[nH]c(C)c1C(=O)NC(C)CCNC(C1(F)CCOC1)=O 36016,N1(C(C(C(C)(C)C)n2cc(C3(O)CCC3)nn2)=O)CCCOC2CCCC12 36017,Cc1nn(C)c(N2CCN(C(=O)C3CC3)CC2)c1CNC(=O)CNS(=O)(=O)C1CC1 36018,C(=O)(C(CC1CC1)OC)NCC(CNC(C1(c2ccno2)CC1)=O)OC 36019,C(=O)(CC(C(F)F)NC(=O)Cc1ncn(C)c1C)N1C(COCC#C)CCC1 36020,c1(CNCCCNC(=O)Nc2cnc(N(C)C)nc2)ccc(F)c2ccccc12 36021,C(=O)(C(O)C(C)(C)C)NCC1(O)CN(C(C2(CC=C)CCC2)=O)C1 36022,Cc1cc(C2CCN(C(c3nccn3C(C)C)C(=O)NCCCF)C2)cc(C)c1 36023,C=CCC(C)(C)CC(=O)NCC1CCCC(NC(c2cncc(C)c2)=O)C1 36024,N1(C(C2C(C(C)C)CCO2)=O)CC2(CC(NC(=O)C=CCOC(C)(C)C)CO2)C1 36025,n1(CC(N2C(CNC(=O)Cc3cnccn3)CC2)=O)c(-c2cccs2)nnc1S 36026,C(c1c(Cl)nc2sccn12)=CC(N1CC(NC(C2CC3C=CC2O3)=O)C(O)C1)=O 36027,c1(CCNC(c2n(CCC)nnn2)c2cnc(C3CCCO3)s2)cccnc1C 36028,Cc1nc(O)nc(C)c1CC(N1CC=C(CNC(=O)CCCN(C)C)CC1)=O 36029,Cc1ccc(F)cc1C(N1CCC(C(F)F)(CNC(=O)Cn2cncn2)C1)=O 36030,CCCN=C(NCC1(C2CC2)CC1)NC1CCN(CC)C(C)C1 36031,CC1CCN(C(=O)CC2(C)CC2(Cl)Cl)CC1NC(c1ccnc(N(C)C)c1)=O 36032,Cc1cc(C(=O)NCC2(O)CCCN(C(=O)C=C(Cl)Cl)C2)c(C)n1C1CC1 36033,c1(-n2c(CCCOc3ccccc3)nc(CC(C)(C)C)n2)cccc2nc[nH]c12 36034,C12(NC(c3n(C=C)nnc3)=O)CCN(C(c3c(Cl)cnn3CC)=O)CC1C2 36035,c1(C(N2CC(NC(C3CN(C)C(=O)C3)=O)C(O)CC2)=O)nccn2nccc12 36036,c1(C(=O)NCC2CCCN(C(C3CC(C)C3)=O)CC2)cn(C)c(=O)nc1O 36037,C(CCCCC(=O)N1CCOCC(CNC(C2CC23CC3)=O)C1)OCC 36038,C1(NC(C=C(C)C(C)C)=O)CCCCCC1C(N1CCC(C)C1)=O 36039,C1(C(=O)NCC(CNC(CC2CCC(=O)C2)=O)CO)CC2(CCOCC2)C1 36040,C1(N(C(=O)C(F)Cc2ccccc2)C)CCCN(C(=O)OC(C)(C)C)CC1 36041,C1(NC(C2CC2C2CCCN(C(C3CC34CC4)=O)C2)=O)CCCCC12OCCO2 36042,C1(NC(C2C(C)=CCS2)=O)CN(C(c2csc(C)n2)=O)CC1(C)C 36043,C12(CNC(C3CC(=C4CCC4)C3)=O)CCC(C1)N(C(=O)COc1ccsc1)C2 36044,N1(C(C(C)c2cccs2)=O)CCC2(CCN(C(c3cnn(C)n3)=O)CC2)C1 36045,c1(SCC#N)cccc(C(=O)NCC(O)CNC(=O)CCN2CCCC2)c1 36046,Cc1cc(C(N2CCC2C(=O)Nc2cnc(Br)c(C)c2)=O)ccc1O 36047,CCCCC(F)C(=O)NCC1C(C(N2CCCC(OCC3CC3)C2)=O)C1(C)C 36048,c1(C(=O)NC2CCCN(Cc3ccc(Cl)cn3)CC2)cn2c(Cl)cccc2n1 36049,c1(C(=O)NCCC#N)cnc(C(C)(C)C)nc1N1CCC(O)C1C(C)C.CO 36050,C1(NC(CC(COC)C)=O)CC2CCC(C1)N2C(c1cnc(O)c(Cl)c1O)=O 36051,N1(C(C2=CCCC2(C)C)=O)CCC2CCN(C(c3ccc(CO)nc3)=O)CC12 36052,CC1C(NC(C2C=CCC2)=O)CCN1C(=O)Cc1cn(C)nc1Cl 36053,C=CC(C)(CC)C(=O)NCC(C)(C1CC1)NC(=O)CCc1nc(N(C)C)no1 36054,C(=O)(CCC(C)(C)NC(=O)CN1CCOCC1)N(CCN(CC)CC)C 36055,N1(CC(=O)NC23CC(CNC(Cc4c(C)n[nH]c4)=O)(C2)C3)C(=O)C(C)C(C)C1=O 36056,c1(C(N2C(CNC(C3CC3C3CCCCC3)=O)CCC2)=O)nc2cnccc2s1 36057,c1(CC)nn(C)cc1C(=O)NC1CCN(C(=O)Cc2ccoc2C)C1C(C)(C)C 36058,C12(NC(c3c(C)ccs3)=O)CCCN(C(C3(CS(C)(=O)=O)COC3)=O)CC1C2 36059,C1(C(=O)NCc2c(C(=O)NCCC(COC)O)nco2)OCCCC1(C)C 36060,CCCCC(O)C(=O)NCC1(C)CCN(C(=O)CCCC(O)c2ccccc2)C1 36061,N1(C(CN(CCCNC(Cc2c(C)scc2)=O)C)=O)CCOC2CCCC12 36062,C(=O)(CN=c1[nH]c(C)cs1)N1CCC(CNC(c2c(OC)nccc2)=O)C1(C)C 36063,C1(COC)CC(C)(C)CN1C(CC)C(=O)NC1(C)CC1 36064,N1(C(C(C(C)C)c2ccncc2)=O)C2CCC1C(CNC(=O)C=C1CCC(C)C1)C2 36065,C(CCCCNCCc1cc(C(=O)OC)no1)SC 36066,c1(C(=O)NC(CCNC(c2c(CC)nns2)=O)C)cc(Cl)ccc1OC 36067,c1(C(=O)NCC(C2CCCCCC2)NC(CCOCC#C)=O)nnc(O)cc1O 36068,N1(C(C2CCCCCN2C(c2n[nH]c3c2CCC3)=O)=O)CC2CC3CC2C1C3 36069,Cc1snnc1C(=O)NCCOC1CCN(C(c2cnn(-c3nccs3)c2)=O)C1 36070,C1(NC(CN(C)CC)=O)(CC)CN(C(=O)CC(C)c2ccccc2)C1 36071,CCC(C)(COC)C(=O)NC1CN(C(c2cccc(F)c2C)=O)CC1F 36072,CC1Oc2ccc(-c3ccc(NC(C4(C)CCCS4(=O)=O)=O)cc3)cc2NC1=O 36073,N1(C(CC2C(C)(C)OCC2)=O)CCC2CN(C(c3ccnc4ccnn34)=O)CC12 36074,c1(C(=O)NCc2ncoc2CCNC(C2(Br)CCC2)=O)ccnc(S)c1 36075,c1(OC)ccc(Cl)c(C(=O)NC(C)CCNC(C2CC(C3CCC3)C2)=O)c1 36076,c1(C(=O)NCC2CC(NC(c3ncccc3F)=O)C2)cc2c(cc1O)CCC2 36077,c1(-c2c(C(=O)NCCCC3N(C(CC#N)=O)CCC3)cno2)ccc(F)cc1 36078,c1(NCC2C(CC)C2)ccc(S(=O)(=O)N2CCCN(C)CC2CC)cc1Cl 36079,N1(C(CSCC)=O)CCC(NC(c2ccc3c(c2)CCO3)=O)C(F)(F)CC1 36080,n1(CC)ncc(C(=O)NCC(n2cc(CNC(c3c[nH]c(=N)s3)=O)nn2)C)n1 36081,CCC(C)CC(C)N(C(=O)CCN(C)C(c1cn(C)cc1C)=O)C 36082,c1(C(=O)NCC2C(C)CN(C(c3cscc3Cl)=O)CC2)cc2ccsc2c(=O)[nH]1 36083,c1(CC(=O)NCC(C(C)C(C)C)NC(C(C)C)=O)nn(C)cc1[N+](=O)[O-] 36084,N1(C(=O)Cn2ncnn2)CCCC1C1(C(=O)NCCn2cncn2)CC1 36085,c1(CNC(N2CCN(CC(=O)OC)C(=O)C2)=O)ccc2n[nH]cc2c1 36086,C1(NC(C(CC)NC(N)=O)=O)CN(C(=O)C(C)OC)CC2CC12 36087,c1(C(=O)NCC(CN(C(C2CCN(CC(C)C)C2)=O)C)C)cc(S(N)(=O)=O)co1 36088,C(=O)(CC(C)C(F)F)NCC(CC)(C)NC(=O)CCc1nc(C(C)(C)C)no1 36089,CC1(C)CCCCCC1NC(C1CCCC1NC(C1CCCCC(=O)N1)=O)=O 36090,Cc1ccc(F)c(C(N2CCC(NC(c3ncsc3S(N)(=O)=O)=O)CC2)=O)c1F 36091,C1(CC(=O)OC2(c3c(OC)ccc(F)c3)CC2)CC(O)C12CC(F)(F)C2 36092,CC(CC(=O)NCC1CCN(C(=O)CN2CC(C)(C)C2)C1)NC(=O)OC(C)(C)C 36093,C=C(Cl)CCC(=O)N1CCC(C(C)(O)CNC(c2ccn(CCOC)n2)=O)CC1 36094,C(=O)(C(CC)CC(F)(F)F)N1CCCC(N(C(CS(CCC)(=O)=O)=O)C)C1 36095,O(C1CCCc2ccccc21)CC(=O)N(CCCNC(C1CCO1)=O)C 36096,Fc1cc(CNc2nccc(CSC3CCCC3)n2)cc(C(F)(F)F)c1 36097,c1(N(C(C)C(=O)N(C)CCCN)S(C)(=O)=O)ccc(F)cc1 36098,C1(C(=O)NC2CC(C)OC2=O)CN(C(C2CCC(O)C2)=O)CC(C)(C)C1 36099,N1(C(C2CCC(CCC)CC2)=O)CCCC2CN(C(=O)Cc3ccsn3)CCC12 36100,c1(OCCC(N2CCC(N(CCO)C(C3(n4cccc4)CC3)=O)C2)=O)ccccc1 36101,C1(NC(c2cc(OC)ncc2)=O)CC2CN(C(C3CCOC3)=O)CC2C1 36102,C1(C)(CNC(Cc2nnc(C)o2)=O)CCCN(C(=O)CC2COC3CC2C3)C1 36103,c1(CC(=O)NCC2(C(C)NC(C3C=CC(C(=O)OC)C3)=O)CC2)ccc(Cl)cn1 36104,CC(C)=C=CC(=O)NCC1(NC(=O)C(c2ccccc2)F)CCOCC1 36105,C12(C(=O)NCC3(C(C)NC(c4n(CCC)ncc4)=O)CC3)CCC(OC)(CC1)C2 36106,N1(C(C=CCOC)=O)CC2CCC1C(CNC(=O)C(CO)NC(=O)C(F)(F)F)C2 36107,N1(c2ccc(S(=O)(=O)N(C)C)s2)CCc2[nH]nc(O)c2C1 36108,c1(C(=O)NC(CN(C(c2ccn(C3CCC3)n2)=O)CC)C)nc(C)sc1C 36109,C1(CC(N2C(CN(C(c3cnc(S)n3C)=O)CC)CCC2)=O)C=NN(C)C1=O 36110,c1(C(=O)NCC(C)(C2CC2)NC(c2ccc[nH]2)=O)cccc(S(=O)(=O)CCO)c1 36111,C12(NC(CCc3n(C)cnc3)=O)CN(C(c3cccs3)=O)CC1CS(=O)(=O)C2 36112,Cc1cc(C)c(C(=O)NCC2(O)CC(NC(=O)Cn3cc(C(F)F)cn3)C2)o1 36113,C1(C(=O)NCCN(CCCF)C)CN(C(=O)OCC(C)(C)C)C(C)(C)C1 36114,c1(C(=O)NCCC(C)NC(=O)CSC2CCCCO2)cc(F)cc(Cl)c1 36115,CCC(C(=O)NC(CC1CCC1)C(=O)NC1CCOCC1O)C(F)(F)F 36116,C1(CN(C(c2nc(OCC)oc2)=O)C)CN(C(c2csc(O)n2)=O)CCO1 36117,N1(CCNC(CCCOC)=O)CCN(C(c2ccc(C(N)=O)s2)=O)CC1 36118,C(C1CCN(C(=O)CCCN=[N+]=[N-])CC1)=CC(=O)NCc1cccc(CC)c1 36119,N1(C(c2c(NC(CCN(C)C)=O)cn(C)n2)=O)CCCC(C)(C(N)=O)C1 36120,C1(C(=O)NCC(C)(C)OCC(=O)NCCc2cccs2)Cc2ccccc2C1 36121,C1(NC(C2(C(C)(C)OC)CC2)=O)COCCN(C(=O)CCC2CCCOC2)C1 36122,CCCC(C)CC(=O)N1CCC(C2CCCN2C(=O)COCC2CC2)CC1 36123,c1(C(=O)NC2C(NC(C(C(C)C)N(CC)CC)=O)CC2)c(F)cccc1Cl 36124,n1(CC(=O)NC(CN(C(=O)C2=NNC(=O)C2)CC)C)sc2ccccc2c1=O 36125,CN1CC2(CCN(C(C3CCCN(c4ccc(F)cc4)C3=O)=O)C2)CC1=O 36126,N1(C(CSCC=C)=O)CCC2(CC(C(=O)NC3CC4CC3C(O)C4O)C2)C1 36127,C1(C(N(C(C(C)SC)C)C)=O)C2CC1N(C(c1cc(C(C)C)on1)=O)C2 36128,C1(NC(c2cnn(C3CC3)c2)=O)CC2CN(C(=O)C3=COCCO3)CC2C1 36129,N1(C(c2c(N)cn(C)n2)=O)CC(NC(=O)Cc2cc(Cl)n(C)n2)CC2(CC2)C1 36130,N1(C(COC2CN(C(C)=O)C2)=O)CCC(NC(c2nnc(C)s2)=O)CC(C)(C)C1 36131,C1(C(N(CCN(C)C(c2ncoc2C2CC2)=O)C)=O)C2CS(=O)(=O)CC12 36132,N1(C(c2ccon2)=O)CC2CCC(C1)N2C(=O)C(c1cccc(Br)n1)(F)F 36133,c1(C(N(CCCCNC(COCCC=C)=O)C)=O)cc(C#N)ccc1Br 36134,c1(SC)ccc([N+](=O)[O-])c(C(=O)NC2CC(CCNC(=O)CC(C)C(C)C)C2)c1 36135,C(=O)(CCC(=O)N1CCCCC1C(C)NC(C1CN(CC(C)C)C1)=O)NCCC 36136,C1(C(=O)OC(C)(C)C)CCN(Cc2cccc(I)c2N)CC1F 36137,C1(NC(C(C)NC(CC)=O)=O)CCCCN(Cc2cc(Br)ccc2C)C1 36138,C1(NC(CSC(C)C)=O)CC2(CCN(C(c3csc(C4CC4)c3)=O)CC2)C1 36139,CN1C2CCC1CN(C(=O)C(=O)Nc1cc(Cl)c(N(C)C)c(Cl)c1)C2 36140,Cc1cc(CNC(=O)CC2C=CC(NC(c3ncc[nH]3)=O)C2)n(C)n1 36141,C1(C(=O)NCc2ccc(C)c(C)c2)N(C(=O)CC=C(Cl)Cl)CC12CCCC2 36142,Cn1ncc(Cl)c1C(=O)NCC1C=CCN1C(=O)CCn1ccccc1=O 36143,C1(C(=O)NC2CC(C3CNC3)C2)CNc2ccnn2C1 36144,c1(CCC)ccc(C(=O)NC2CC(F)(CNC(C3(C)CCC(=O)N3)=O)C2)cc1 36145,c1(OC)cc(CC(N2CCC(C)(NC(c3ccnn3C(F)F)=O)C2)=O)cc(Cl)c1 36146,N1(C(CCCCOC)=O)CC2(CCCCN2C(C2(C)CC3CCC2O3)=O)C1 36147,N(C1CCCn2cnnc21)C(=O)Nc1ccc(C2CCC2)nc1 36148,Cc1ccc(C(=O)NC2CC(CNC(=O)CNC(c3cccs3)=O)C2(C)C)n1C 36149,Cc1ccc(S(=O)(=O)N2CC(C)NC(C)C2)cc1NC(=O)C(F)(F)C1CCNC1 36150,c1(C(N2C(C(C)NC(C3CC4(C3)CC4F)=O)CCC2)=O)nn(C)c2ccccc12 36151,C1(C(C)C)N(C(=O)CC(C)(O)C(F)(F)F)CC12CCN(C(C1CC1(C)C)=O)CC2 36152,C(=O)(CC(CNC(=O)CN1CCC(=O)CC1)C1CCC1)N(C1CCN(C)C1)CC 36153,C(=O)(CC(c1ccccc1)C1CC1)NC1C(NC(C(=O)NCC(F)(F)F)=O)CC1 36154,c1(CCC(N2CCC(NC(C3(F)C(C)C3)=O)C23CC3)=O)ccc([N+](=O)[O-])cc1 36155,C(=O)(CCS(=O)(=O)c1ccccc1)NC(CC)CN(C(=O)C(C)CC1CC1)CC 36156,CCCC(CC)CC(=O)NC1CN(C(=O)CNc2cccc(C#N)c2)CC1O 36157,C1(F)(C(N(CCC)CCNC(C2CC2C(F)(F)F)=O)=O)CC1C 36158,C(=O)(CCCN(C)N=O)NCCC1CC(OC)CN1C(=O)C(C)NC(N)=O 36159,C(=O)(CCCCN=[N+]=[N-])NCC(CN(C(C1(C2(C)CC2)CC1)=O)CC)(C)C 36160,Cc1cnc(C(=O)NC2CC(NC(=O)CC3CC4(COC4)C3)C2)nc1 36161,N1(C(C2N(C(C3C(C=C)OCC3)=O)CCOC2)=O)CC(C2CC2)(COCC)C1 36162,N1(C(c2ccc(C)c(F)c2)=O)CCCCCC(NC(C2(C)CC2(F)F)=O)C1 36163,C#CCCC(C(=O)NC1CC12CCC2)NC(c1cc(C)no1)=O 36164,N1(C(CC2CCC(NC(c3occ(C)c3)=O)C2)=O)Cc2cccc(C)c2C1 36165,Nc1ncc([N+](=O)[O-])cc1C(=O)NC1(CO)CCN(C(C2CC2(F)F)=O)C1 36166,c1(C(N2C(CN(C)C(c3scc(Cl)c3Cl)=O)CCC2)=O)cccc(=O)n1C 36167,CCCC(C(=O)NC(C)CN(C(=O)CC1(OC)CCOCC1)C)c1ccccc1 36168,N1(C(CCC(=O)NC)=O)CCN(C(c2coc(C#N)c2)=O)C(C)C1 36169,C1(C(N2CCC(N(C(c3c(Cl)ccc(OC)c3)=O)C)C2)=O)CCc2nccn2C1 36170,Cc1cc(C(N2CC(C)(NC(=O)CC3CCCOCC3)C2)=O)cc(N)c1 36171,C(=O)(C1CCCn2ccnc21)N1CCC(CNC(c2ccc(O)cc2F)=O)CC1 36172,N1(CC)CC(NC(=O)CCCNC(C2CSC2)=O)C(C)C1 36173,c1(NC(CN2C(C)CC2)=O)cccc(NC(=O)Cn2ncc(Br)n2)c1 36174,C1(COC2CCN(C(C(C)O)=O)C2)CCN(C(C2CC(F)C(=O)N2)=O)CC1 36175,CC1CC=C(C(=O)N2CCCC(CC(=O)NC3(C)CCCC3C)C2)CC1 36176,c1(CN2CC(CCC)C(C(=O)OC)C2)ccc(CN2CCCCC2)c(C)c1 36177,N1(C(c2cc(CC)oc2C)=O)CC2(CCCC2)C1C(N1C2CCC1CC(F)C2)=O 36178,C1(C(C(=O)NCC=CCOC)C)CCN(C(c2cc(CO)sn2)=O)C1 36179,C=CCC(F)(F)CN(C(=O)C(C1CCN(C(=O)C(C)C2CC2)CC1)C)C 36180,c1(C(=O)NCCOCCN(C(C2(CC#C)CC2)=O)C)cc2c(cc1Cl)CCCC2 36181,c1(C(=O)NC2CCC(CCNC(c3c(OC)csc3)=O)C2)cn(C)c(=O)cc1C 36182,Cc1ccc2c(c1)CC(N(C(=O)COc1nc(C(C)OC(C)C)no1)C)C2 36183,C1(CNC(c2ccc(N3CCC3)nc2)=O)CN(C(c2nccnc2Cl)=O)CCO1 36184,N1(C(C)=O)CC(C)OC2(CCN(C(c3c(C)nc(C(C)(C)C)nc3S)=O)CC2)C1 36185,c1(CC)nc(C)c(C(=O)N(C)CCOCCN(C)C(c2nc(C3CC3)cs2)=O)s1 36186,C12(CNC(CSCC#C)=O)CCC(CN1C(c1ccc(C)nc1OC)=O)C2 36187,c1(C(=O)Nc2cccc(Br)c2)cnc2n1CCN(C(=O)Nc1occc1Br)C2 36188,C1(CNC(=O)COCC2CCOCC2)CC2CC2N1C(c1ccnc(CO)c1)=O 36189,C1(NC(C=Cc2cc(OC)ns2)=O)CCCN(C(c2cccc(F)c2F)=O)C1C 36190,c1(C(C)NC(C2CN(C)C2)=O)ccc(CNC(c2ccc(C#N)[nH]2)=O)cc1 36191,N1(C(c2ccc(OC)s2)=O)CCC2(CCCN(Cc3cccc(C)c3)C2)CC1 36192,N1(C(c2cccc(C#C)c2)=O)CC(C2CN(C(=O)C(C)(C)CCCO)C2)C1 36193,c1(C(=O)NC2C(CNC(c3ncc(Cl)s3)=O)CCCC2)cnn2c1C(=O)NCC2 36194,C1(C(=O)NCc2ccc(C(N(CCCC=C)CC)=O)s2)CC(C)(C)CN1C 36195,C(=O)(CCCCC#N)N(CCC(C)NC(=O)CC1CCC(F)(F)C1)C 36196,C1(CNC(C(C#C)(C)C)=O)CCCC2(CCN(C(c3nc(C)oc3C)=O)CC2)O1 36197,c1(C(=O)NCC(CN(C)C(C2CN(C3CCCCC3)C2)=O)O)cc(F)ccc1O 36198,N1(C(C(C)OCCC#C)=O)CC(NC(=O)CCn2cc(C)cn2)C(C)C1 36199,n1(CC)cccc1C(=O)NCC(F)CNC(c1cc(C2CC(F)(F)C2)[nH]n1)=O 36200,c1(CC(=O)NCCC(C)NC(CC(CC)OC)=O)cccc(F)c1F 36201,c1(OC)ccc(F)c(C(=O)NCC2CC3(CC3)CN2C(=O)CC2CNC(=O)C2)c1 36202,C1(NC(C(CC)CC(C)C)=O)CCCC12CCN(C(=O)CC1CC(F)(F)C1)CC2 36203,N1(C(c2c(C)[nH]cc2)=O)CCC(CO)C(NC(=O)Cc2cn(C)cn2)C1 36204,C(=O)(C(O)CCN(C)C)N(C)CC1(CNC(=O)Cn2nnc(=O)[nH]2)CC1 36205,C=CC1CN(C(=O)CC(C)=C(C)C)CC1NC(C1CN(C(C)C)CCO1)=O 36206,C1(C(C)C)CN(C(c2cc(O)cc(O)c2)=O)CCN1C(=O)C(C)c1cccs1 36207,C=C(C)CC(=O)NCC(C)NC(=O)C(C1CCCCC1)NC(C1CCCCC1)=O 36208,N1(C(C2CSCCS2)=O)CC2CCN(C(C3(O)CCSCC3)=O)CC12 36209,N1(C(C(C)(C2CC2)OC)=O)CCN(C(C23CC2COC3(C)C)=O)CC(O)C1 36210,N1(C(C(c2ccccc2)C)=O)CC(NC(c2c[nH]c(=O)cn2)=O)C(C)C1 36211,N1(C(C2(CC)CC(C)(C)C2)=O)CCC12CN(C(=O)CC1C=CCC1)C2 36212,CCCCCC(C)(C)C(=O)NCCC(C)NC(=O)C(n1cc([N+](=O)[O-])cn1)(C)C 36213,C(CCCCCCCO)=CC(=O)NC1COCC1CNC(=O)CCCCCC#N 36214,C#CCC(CC(=O)NC1CC2(NC(c3cn(C)nn3)=O)COC1C2)c1ccccc1 36215,C(=O)(CC(C)C(C)C)NC1(CN(C)C(C2(OC)CCCC2)=O)CCC1 36216,c1(C(N2CC=CC(NC(C=CCN(C)CC)=O)C2)=O)cc[nH]c2nccc1-2 36217,C(c1cccc(C)c1)=CC(N1CC(NC(C(CC)Oc2ccccc2Cl)=O)C1)=O 36218,C1(C(=O)Nc2cccc(NC(c3cnn(C)n3)=O)c2)CC2(C1)CC2(F)F 36219,C1(C(=O)NCC2(SC)CC2)CC12CC(NC(=O)CCC1CCCO1)C2 36220,c1(OCC)ccccc1OCCN1CC2C(C(=O)NC(CC)CO)C2C1 36221,C1(CNC(=O)COC2CCCC2)C(C2CC2)CCN1C(C12CCC(F)(CC1)C2)=O 36222,C(CC(CC)C(=O)NC1(CCC(=O)NC(COCC)C(C)C)CCC1)=CC 36223,Cc1ccc(C(CNC(C2(n3ccnn3)CC2)=O)NC(=O)CSC(F)F)cc1 36224,O(NC(=O)C(O)CNC(=O)C(O)C(F)(F)F)C(C=C)C 36225,n1(CC(=O)NCC(CC)N(C)C(c2cnc(C3CC3)s2)=O)nnc(C2CC2)n1 36226,c1(C(=O)NC2CC3(CC(NC(C4C(C(=O)OC)C4)=O)C3)C2)ccnc2[nH]cnc12 36227,N1(C(c2ccc(CCC)s2)=O)CCCCC(NC(C2CCN2C2CCCC2)=O)C1 36228,C(=O)(C1CCCc2ncc(C)n21)N1CCC(NC(CCc2nnc(CC)o2)=O)C1 36229,c1(OC)ccc(C(=O)C(=O)NC2CCC(NC(C3CC3(F)F)=O)C2)cc1OC 36230,CC1CC(F)(F)CN1C(=O)C=CC(C)(C)NC(=O)C=CC1CCC1 36231,CCCC(C(=O)N1CCC(C(C)NC(c2ccoc2)=O)C1)S(N)(=O)=O 36232,C(C1CCOCC1)=CC(=O)NC1CC(NC(C2(C(N)=O)CCC2)=O)C1 36233,c1(C(=O)NCC2CCC(CNC(CCOC)=O)CC2)ncnc2sccc12 36234,C=C=CC(C)C(=O)NC1(C)CC(NC(=O)CCc2nc(-c3ccoc3)no2)C1 36235,C(=O)(C(C)(C)CC#N)NC1C(NC(c2c(SC)cn(C)n2)=O)COCC1 36236,N1(C(C(N2CCC(O)CC2)C)=O)CCCC(CNC(=O)Cn2cncn2)C1 36237,c1(C(=O)NCCOC2CN(C(C=C(C)C(F)F)=O)C2)cc2oc(C)c(C)c2[nH]1 36238,c1(OCC)ccccc1C(=O)NC(c1cnc[nH]1)C 36239,C1(C(=O)NC2C(OC)CN(C(c3ccnc(N(C)C)c3)=O)C2)CCCC(=O)N1C 36240,c1(C(=O)OCCCC#C)nnc(C(F)F)s1 36241,C1(C(=O)NC2CCC(NC(=O)Cc3ccccc3F)CC2)(COC)CCOCC1 36242,C=CC(CCC)CC(=O)NCC1CC(F)CN1C(c1cc(F)c(N)c(F)c1)=O 36243,N1(C(C2CCN(C)C2=O)=O)CC2CN(C(c3cnc4ccsc4c3)=O)CC2(C)C1 36244,C1(C2(C(=O)NC3(CC)CN(C(=O)C(C(C)C)c4cncs4)C3)CC2)CCCCC1O 36245,N1(C(C(=O)NCC(=O)NCC(=O)NC2(CC(C)C)CC2)C)CCOC1=O 36246,C1(C(=O)NCC2(NC(c3ccc(C)o3)=O)CC(OC)C2)CC12CCCCC2 36247,c1(C(=O)NCC2N(C(c3cc(C4(C)COC4)no3)=O)CC=C2)ccc([N+](=O)[O-])cn1 36248,CCC(CNC(C1(NC(=O)CCn2cncn2)CC1)=O)CCO 36249,Cc1ccc(C(=O)NCC2(F)CCN(C(=O)CC3CC=CCC3)CC2)c(O)n1 36250,N1(C(C(C)SC)=O)CC(NC(C2CCC(C(F)(F)F)O2)=O)C(CO)C1 36251,C(=O)(C(COC)CC(C)C)NC1(CC=C)CN(C(=O)C(C)=CC(C)(C)C)C1 36252,C12(C(=O)NCC3(C)OCCN(C(Cc4nnc(C)o4)=O)C3)CCCCC1C2(F)F 36253,Cc1ncnc(N2CCC(CCNC(c3ccc(=O)n(CC4CC4)c3)=O)C2)c1F 36254,C1(NCc2ccccc2Cl)CCCN(c2ncccn2)C1.C12(CC1)N(C)C2=O 36255,c1(CC(=O)NC(CNC(C(C)OC)=O)(C)C)c(Br)ccc(Cl)c1F 36256,C(C)(C)(CC(=O)NC(C)(C)CCCNC(=O)Cc1cc(Cl)cs1)SC 36257,c1(C(N2CC(CNC(c3[nH]nnc3C3CC3)=O)C2)=O)cc2c(F)cc(F)cc2[nH]1 36258,c1(C(=O)NC2CC(CNC(C(CC)n3cncn3)=O)C2)cc(C)nc(O)n1 36259,C1(C(N(C2CCN(C(=O)C=Cc3cn(C)nn3)C2)CCC)=O)CCCCN1C 36260,C(=O)(C1COc2ccccc21)NCCN(C(CSCCC)=O)CCOC 36261,CC1CCC(CNC(c2coc(CNC(C3(C)CSC3)=O)c2)=O)N1C 36262,c1(C(N(CC(C)NC(=O)C(C(=O)OC)OC)CC)=O)cc2nc(=O)ccn2[nH]1 36263,N1(N(C(C)(C)C)C(=O)NC(CCCn2ncc(C)c2)C)CCN(C)CC1(C)C 36264,CC1(C(=O)NCCCCCNC(=O)CNC(c2ccncc2)=O)CCC(=O)NC1 36265,C1(C(N(CC#CC)CC#C)=O)CC(C)CN(C(c2c[nH]nc2[N+](=O)[O-])=O)C1 36266,c1(CNC(NC(COC)C)=NCCc2cn3c(n2)SCC3)ccc(C#N)c(F)c1 36267,c1(NC(C(=O)Nc2c(CC)scc2)=O)ccccc1N1CCNC1=O 36268,C=C=CC(C)C(=O)NC(CNC(c1cc(C)n(CC(F)(F)F)n1)=O)CC=C 36269,n1(CC(=O)NCC2C(NC(=O)CCC3CCC3)CCC2)ccc(O)nc1=O 36270,C1(NC(c2cncc(OC)n2)=O)CN(C(c2cc(C)c(C)o2)=O)C(C)(C)C1 36271,C(=O)(C#CC(C)(C)C)N(C(=O)C(N1CCN(C(C)C)CC1)C)OC(C=COC)=O 36272,CC1(CNC(=O)CC2CCSCC2)CCCN(C(C2CC3(C2)CC32CC2)=O)C1 36273,c1(C(=O)NC(CNC(c2cc(C(C)C)on2)=O)(C)CO)ccc(S(=O)(=O)NC)o1 36274,N1(C(CCOCC#C)=O)CC2OC(C1)C2.C(=O)(C(C)OC)NCC1CC1 36275,Cc1cc2cc(F)ccc2n1Cc1ncc(F)cn1 36276,CC(C)CC(O)CC(=O)N1CC(C)C(C)(CNC(C2(C(C)C)CC2)=O)C1 36277,Cc1ccc(C(=O)NC2CCC(C)N(C(c3ccnc(F)c3F)=O)C2)cc1N 36278,Cc1ccc(CC(=O)NC2CC2CNC(C2C(C)(C)C2(F)F)=O)cn1 36279,C1(CNC(c2c(COC)cccc2)=O)(NC(=O)CSS(C)(=O)=O)CCCCC1C 36280,N1(C(c2cc[nH]c2)C)CC2C(C(=O)N(C)Cc3ccc(Cl)cc3)C2C1 36281,c1(C(N2CCCC(CN(C(C(CC#C)C)=O)C)C2)=O)c(C)nn(CCO)c1C 36282,CC1CCCN(C(C2(C)CC(O)CN2C(c2ccn(C)c(=O)c2)=O)=O)CC1 36283,C1(CC)CCC2(CC1)NC(=O)N(C(=O)Cc1ccc(Cl)s1)C2=O 36284,Cc1cc(C(=O)N(CC(C)C(=O)NCc2nn[nH]c2C2CC2)C)n(C)n1 36285,c1(OC)cc(CC(N2CCC(NC(C3CCCOCC3)=O)C2(C)C)=O)ccc1C 36286,C1(CNC(CCC(=C)Cl)=O)CN(C(c2c(N)cc(Cl)cc2F)=O)CC2(CCC2)O1 36287,CCC1=C(C(=O)NCCN(C2CCCC2)C(C2CCCC(F)C2)=O)SCCO1 36288,Cc1cc(O)ncc1NC(C1CCC(C2CC2)N1C(c1nnn(C)c1N)=O)=O 36289,CC(C)C(CN(C)C)C(=O)NC(CC(F)F)C(=O)NCC1CCC(=O)NC1C 36290,C1(NC(CSc2cccc(OC)c2)=O)CC(F)(F)C12CCC2 36291,N1(c2nccc(=NCc3c(C)occ3)[nH]2)CCN(C)CC2(C)CCCC12 36292,C1(CNC(c2n(C(C)C)ccn2)=O)CC(C)N(C(=O)C(N2C(=O)CCC2=O)C)C1 36293,N1(C(CSCCN(CC)CC)=O)CC2CCC1C2CNC(c1[nH]cc(C)c1C)=O 36294,Cc1cc(C(N2CC(NC(c3cc(C4CCCC4)[nH]n3)=O)C3CC23)=O)c(C)cn1 36295,C(=O)(C(CNC(C)=O)CC(C)C)NC1C(C(N2OCC(=C)C2)=O)CCOC1 36296,C(=O)(C(CNC(c1oncc1CC)=O)CC(C)C)NC1(CC#C)CCC1 36297,C1(N(C(=O)CC2CCC3CC23)CC)CCN(C(=O)Cc2ccccc2F)CC1 36298,CC1CN(C(c2cc(CCCO)on2)=O)CC(C)C1NC(=O)C1CC1 36299,N1(C(C2CCOC2)=O)CCCC(Cn2cc(C3CC=CCC3)nn2)C1 36300,C=CCC(CC)C(=O)N1CC2CCC2(NC(=O)COc2cncc(Cl)n2)C1 36301,C1(NC(CCCC=C)=O)CC2CC1N(C(=O)CCc1ccsc1Cl)C2 36302,N1(C(C(CC)(C)O)=O)C2CCC1CC(CNC(=O)C(C)(C)Nc1ccccn1)C2 36303,c1(OS(CC2C(C)(C)OC2(C)C)(=O)=O)c(-c2ccccc2)nc2ncccn12 36304,c1(C(N(CC(=O)NCC(F)(F)C(F)(F)F)C)=O)ccnc2ccccc12 36305,c1(C(N2CCN(C(C=CC(=O)OCC)=O)C(CF)C2)=O)cccn2c(O)nnc12 36306,CCC(C)(C)C(C)CC(=O)NC1CCC1CNC(=O)Cn1cnc(C#N)n1 36307,CCC(CCC(=O)N1CCC(C(C)(F)F)CC1)OC 36308,C(C(O)CC(=O)NCCCCCF)NC(CCC1C(C)(C)C1)=O 36309,C1(C(NOCCOC(C)C)=O)CC(NC(=O)CCC2CCCN2C)C1(C)C 36310,C1(CSc2c(OC)cccc2)COC(C)(C)CN1c1nc(C)cc(NC(C)=O)n1 36311,C(=O)(C(F)CC(C)(C)NC(=O)CCCCCF)N1CCCC(C(C)C)CC1 36312,c1(NC(C2N(C(C(C)OCCCCCC)=O)CCC2C)=O)cnc(F)cc1C 36313,C1(NC(C(CC#C)C2CC2)=O)COCCN(C(=O)CCOCC#C)C1 36314,c1(OC)ccc2[nH]cc(C(=O)NC(C)CC(C)NC(=O)CSC3CC3)c2c1 36315,N1(C(C(C)OCC(C)C)=O)CCC2(CCC2)C(NC(=O)CSC2CC2)C1 36316,C#CC1CN(C(=O)Cc2ccc(Cl)s2)CCN1C(c1cc(C(C)(C)C)[nH]c1C)=O 36317,C#CC1(C(=O)NCCC(=C)CNC(=O)CN2CCC(OC)C2)CCCCC1 36318,Fc1cc(F)c(CCNC(c2ccncc2)c2nnnn2CC(F)F)c(F)c1 36319,C(CCCC(C)(C)C)c1nnc(CC(C)(C)OC(F)F)o1 36320,c1(CNC(CC2N(C(CC(C)c3ccco3)=O)CC2)=O)ccc(O)cc1 36321,C1(NC(CCOC)=O)CC=C(C(=O)NCC2CC3C=CC2O3)C1 36322,N1(C(Cn2c(C)nc(C)n2)=O)CCC2(CC1)CCN(C(C1(C(F)F)CC1)=O)CC2 36323,N1(C(C(=O)NCC=C)C(C2CC2)OCC)CCC2(CC1)NC(=O)NC2=O 36324,c1(C(N(C(=O)CSc2ncn(C)n2)CC)=O)ccc(-c2cccs2)nc1C 36325,CN1CCN(C(c2cc(CNC(=O)CCc3ccsc3)[nH]n2)=O)CC1CO 36326,Cc1nc(N)c2c(C)c(C(=O)Nc3ccc(CN(C)C4CC4)cc3)sc2n1 36327,N1(C(C(C)SCC)=O)CCc2sc(CNC(c3cc(F)c(C)cc3O)=O)nc2C1 36328,c1(CC)ncc(C(=O)NC2COCC2NC(=O)CCC2CC2(F)F)c(C)n1 36329,C1(C(=O)Nc2scc(C(C)C3CC3)n2)C(C2CC2)CCN1C(=O)OC(C)(C)C 36330,C(C)(C)(C(=O)NC1CCC1NC(=O)CN1CCCC1C)OC(C)C 36331,C(C(=O)Nn1cccn1)N(C(C)CC(N)=O)CC 36332,N1(C(C2CCC=CO2)C(=O)NC(C(=O)OC)C)CCC(S(=O)(=O)C(F)F)C1 36333,c1(C(N(C2CCN(C(C3CCNC(=O)C3)=O)CC2)C)=O)ccnc2ncccc12 36334,C1(CC)CN(C(=O)C(C2CCC2)NC(c2ccnnc2C)=O)CCO1 36335,N1(C(CCCc2cc(C)no2)=O)CCC2CCN(C(c3ncoc3C)=O)C2C1 36336,c1(NC2(CNC(C3CC(CC)OCC3)=O)CCC2)ncc(S(C)(=O)=O)cc1Cl 36337,C#CCN(OC)C(=O)CC1(OC)CN(C(c2ccn3ccccc23)=O)C1 36338,CCC(O)C(C)(C)C(=O)NCC1CCN(C(=O)CSCCC(C)C)C1 36339,Cc1c(C(=O)N(CC(O)CNC(C2COC(=O)N2)=O)C)[nH]c2c(C)cccc12 36340,C1(CCC)CN(C(c2c(F)cccc2Cl)=O)CCN1C(c1cc(COC)c[nH]1)=O 36341,CC1(C)C(CNC(C2CCCC2)=O)CCN1C(=O)CC1COC(=O)C1 36342,c1(CNC(C(CCC)CC)=O)ccc2c(c1)CN(C(C1CCN1S(C)(=O)=O)=O)C2 36343,C#Cc1cnn(C)c1C(N1CCC(N(C(=O)CSc2cnn(C)c2)C)CC1)=O 36344,C1(C2CCN(C(Cc3c(C(C)C)con3)=O)C2)CCCCN1C(c1cccs1)=O 36345,N1(C(C(=O)N(C)C)=O)CC2CCCCC2(CNC(C2(C)CCCCNC2=O)=O)C1 36346,c1(NC(C(CC)(C)OC)c2nnnn2CCCF)ccc(C)c(S(C)(=O)=O)c1 36347,O=C1CCC(C(=O)N)=NN1.C1(C2CCN(CCN3CCCCCC3)C2)CCC(O)C1 36348,C(=O)(C(C)(C)CCCOC)NC1CCC(NC(c2cc(OC)ns2)=O)C1 36349,C#Cc1ccc(C(N2CC(C)CC2C(=O)Nc2cnn(C)c2)=O)cc1C 36350,Cc1nc[nH]c1CC(O)C(=O)N(C(C1C2CCCC12)=O)C(C)C.C12CCN(C1)C(=O)C2 36351,C(C)(N=c1[nH]c(=NCC(CO)C2CCCC2)c2c(ncn2C)[nH]1)c1ncc(C)s1 36352,C1(C(=O)NC(CC)CNC(c2snnc2C)=O)CCN(S(=O)(=O)NC)CC1 36353,C(=O)(C1=CC2C=CC1C2)NC1CCN(C(C(C)NC(C)(C)C)=O)C1C1CC1 36354,C1(CNC(c2c(OC)n(C)nc2)=O)C(C2CC2)CCN1C(c1nnn(C)c1C)=O 36355,C1(C(=O)NC2(CNC(Cc3scc(C)n3)=O)CCOC2)CCc2c(cnn2C)C1 36356,n1(CC)ccnc1C=CC(=O)NC1CC(NC(=O)CCOC2CCCC2)C1 36357,C(CCCCNC(=O)C(c1ccnn1C)C)NC(C(C1CCC1)OCC)=O 36358,Cn1cc(C(=O)NC2CCCN(C(=O)Cc3ccns3)C2)c(O)n1 36359,NS(=O)(=O)c1ccc(C(N2CCC(CNC(c3nsnc3O)=O)C2)=O)cc1F 36360,N1(C(C(CC)C)=O)CC(CNC(c2sccc2C)=O)OC(C)(C)C1 36361,Cc1cc(N2CCC(C)C2CNC(C2(C(N)=O)CCC2)=O)n2ncc(C)c2n1 36362,C(=O)(C(O)CCC(C)C)N1CC(C)(NC(C2CCCC(OC)C2)=O)C1 36363,N1(C(C(C)OCC(C)C)=O)CCOC(C(N2CCCC(C)(C)C2)=O)CC1 36364,c1(NC(C)=O)cnc(C)c(C(N2CCCC2CNC(C2OCC2(C)C)=O)=O)c1 36365,C(N=c1nc(N2CCN(C)CC(C)C2)c2[nH]ccc2[nH]1)c1c(C)cccc1Cl 36366,c1(C(=O)O)cc(F)c(C(c2ccncc2)NS(=O)(=O)C(F)(F)F)cc1F 36367,Cc1sccc1C(=O)NC(C1CCCN1C(=O)CSS(C)(=O)=O)C 36368,CC1CN(C(c2ccc3sccc3c2)=O)CC(C)CN1C(c1nn(C)cc1N)=O 36369,N1(C(C(C)OCC)=O)CC(NC(=O)CCc2cnc(O)[nH]2)C2(CCOCC2)C1 36370,c1(OCC(=O)NC2CCC(NC(C(C(C)C)SC)=O)CC2)cc(C)ccc1F 36371,c1(C(=O)NC2CCC(NC(C(CCCC)O)=O)C2)cc2sc(N3CCCC3)nc2s1 36372,c12cc(N(C)C)ccc1OC2=O.C1(N(CC)CC)CCS(=O)(=O)C1 36373,c1(SC)nc(N2CCCCC2CNC(c2cncc(F)c2)=O)cc(Cl)n1 36374,CCC(C)CC(C)C(=O)N(CC(=O)NC1C2CCN(CC2)C1C)C1CCC1 36375,c1(C(C)C(=O)N2CC(C(C)N)C2)c[nH]c2ccccc12 36376,C1(O)(CNC(C(C)(F)F)=O)CCCN(C(C23CCC(CF)(C2)OC3)=O)CC1 36377,c1(C(c2n(CC(=C)C)nnn2)NCCc2cccc(F)c2)cc(F)c(F)cc1F 36378,S(=O)(=O)(C1CCN(CC#Cc2cccnc2)CC1)NC 36379,c1(OC)ccc(CN2CC3CC3(C(=O)Nc3ccc(C4CC4)nc3)C2)c(C)c1 36380,C1(CNC(C2(NC(C)=O)CCC2)=O)CCCN(C(c2cccnc2O)=O)C1 36381,N1(C(c2coc(CO)c2)=O)CCCN(C(=O)C2=C(Cl)CCC2)C(CO)C1 36382,c1(CC)cc(C(=O)NCCCC(=O)NC(CO)(CO)CO)c(C)o1 36383,Cc1nccc(C(=O)N(C(C)CN(C)C(C2(CN3CCC3)CCCC2)=O)C)n1 36384,C1(O)(CN(C)C(c2ccc(OCF)cc2)=O)CCCN(C(c2ns[nH]c2=O)=O)C1 36385,N1(C(C(CC)OCC)=O)CCC(O)(C(C)CNC(=O)CCc2cnco2)C1 36386,c1(CNC(CCCCCC)C)cc2ccc(C(=O)OC)cc2o1 36387,C1(NC(c2nc(N(C)C)oc2)=O)CCC(C)(CNC(c2ccc(C(N)=O)s2)=O)C1 36388,C1(C(=O)NC(C)CCCCNC(c2cc(O)cc(F)c2)=O)CCCCC(C)(C)C1 36389,c1(NC(c2cc(-c3c(OCOC)cc(F)cc3)[nH]n2)=O)c(C)cc(C#N)cc1Cl 36390,c1(OC)ccc(Cl)c(OC)c1C(=O)NCC1(C)CN(C(c2cc(C)nn2C)=O)C1 36391,N1(C(CN(C(c2n[nH]c(O)n2)=O)CC)=O)CCCC1C 36392,c1(CC)cncc(C(=O)NCC2CCC(NC(=O)CCc3cnn(C)c3C)C2)c1 36393,Cc1cn(C)nc1C(N1CCCC1CCNC(c1c(C)ccn1C)=O)=O 36394,C1(C(N2C3CN(C(CC4(C)CC4)=O)CC2CCC3)=O)CCCC12NC(=O)NC2=O 36395,N1(C(C2CCOC2)=O)CCCN(C(c2cscn2)=O)C(c2ccccc2)C1 36396,C1(C(=O)NCCCCNC(CSCCC)=O)(N(C)C)CCCCC1 36397,C1(C(=O)NC2C(NC(c3cc(C)c(C)s3)=O)CCC2)CC12CCOCC2 36398,C1(NC(C(C)N2CCCC2)=O)CC2CCC1(C(N1CCCC1C)=O)C2 36399,c1(C(=O)NC2CC3N(C(C(C)SC)=O)C(CC3)C2)csc2c(O)ccnc12 36400,C1(NC(C2N(C(c3c(C)nsc3)=O)CC2C)=O)(CO)CC2CCCC12 36401,c1(C(N(C2CCN(C(c3cccc(F)c3I)=O)C2)C)=O)cc(F)c(Cl)cc1Cl 36402,C1(CC)(CC)CCN(C(=O)CSCCNC(c2ccnc(OC)c2)=O)C1 36403,Cc1cc(C)c(C(N2CCOC(CCNC(=O)C(C)(F)F)C2)=O)c(O)n1 36404,C(c1ccc(Br)cc1)=CCC(N1CCC(C)(CCNC(=O)C(F)F)C1)=O 36405,CC1(C)CN(C(C2(c3ccno3)CC2)=O)CCN(C(C2(C)CCC(=O)NC2)=O)C1 36406,c1(CNC2CC(NC(c3cn(CCC)nc3)=O)C2)cc(OCC)ncn1 36407,C#CCCCCC(=O)NC(C1CCOC1)CNC(C1(C(F)(F)F)CC(=C)C1)=O 36408,N1(C(C=CSC)=O)CC2CCC(CNC(C3C4CCCCCCC34)=O)(C2)C1 36409,C1(OC)CC(NC(=O)C(C)C(F)(F)F)CN(C(c2c(C)nc(C3CC3)n2O)=O)C1 36410,c1(C(=O)NC2C(NC(C3(CCN(C)C)CC3)=O)CC2)cccnc1C(F)(F)F 36411,c1(NCC2C(C)CN(C(c3ccc(=O)oc3)=O)CC2)c(F)cccc1[N+](=O)[O-] 36412,c1(CC)ccc(C(=O)NC(C2CCCCC2)CNC(C2COC(=O)O2)=O)s1 36413,N(C(=NCc1cc(C)nn1C)N1CCc2ccc(Cl)cc2C1)C(C=C)C 36414,Cc1cccc(NC(N2CCCC(c3nc[nH]n3)C2)=O)c1OC 36415,N1(C(C2(C(C)C)CCN(C(=O)CN(C)C3CC3)C2)=O)CC(C)CC(C)(C)C1 36416,Cc1c(C(N2CCCC2CN(C)C(C2(O)CC2)=O)=O)sc2cc(F)ccc12 36417,C12(NC(c3nocc3Cl)=O)CCCC1N(C(c1ccc(OC(F)F)cc1)=O)CC2 36418,C1(CNC(C(C)(C)OCC)=O)CCN(C(c2coc3c2COC3)=O)CC1O 36419,C1(c2nnc(CNC(C(C)SC)=O)s2)CCN(C(C2CCC(=O)NC2)=O)CC1 36420,c1(OC)cc(P(C)(C)=O)ccc1NC(=O)NC1CCN(c2ccc(F)cc2)C1 36421,Cc1cc(F)c(C(=O)NCC(O)CN(C(=O)Cc2c[nH]ccc2=O)C)cc1F 36422,Cc1cccc(-c2nc(C(C)N(C)C)nn2C2CCCCC2C)n1 36423,Cc1[nH]c(C)c(C(N2CCOC(CNC(=O)CC(C)C(F)F)C2)=O)c1C 36424,c1(C(N2CCC(N(C(C3(OC)CCCC3)=O)C)CC2)=O)cc(S(N)(=O)=O)c(C)o1 36425,C1(CC(=O)NCc2c(C)cc(C)s2)CCCN(C(c2ccccc2)=O)CC1 36426,C(=O)(C(C(=O)Oc1cccc(NS(C)(=O)=O)c1)c1ccccc1)OCC 36427,C1(N)CN(C(=O)COC(C)(C)C)CC12CC2.c1(CN(C)C(=O)O)ccc(N(C)C)cc1 36428,C#CC1(O)CC(C(=O)NC2CCOC(c3ccncc3)C2)C1 36429,N1(C(c2c(CC)noc2)=O)CCN(C)CC1CNC(=O)Cn1nccc1N 36430,N1(C(COC)=O)CCC(CNC(=O)C(c2cncnc2)C)C(F)(F)C1 36431,c1(C(=O)NCCCCC(CO)NC(c2nc(C(N)=O)sc2)=O)cnc2[nH]cncc1-2 36432,C(C(C(=O)NCC1CC(C)(NC(=O)C(C)Sc2nncn2C)C1)NC(C)=O)OC 36433,C1(C(=O)NCc2cc(C)ncc2)COC2(C1)CN(C(C1CCC(=O)C1)=O)C2 36434,NC(=O)CCC(C(=O)N=c1ccn(-c2ccncc2)[nH]1)n1cc2nnncc2n1 36435,c1(OC(=O)NCCC=C)ccccc1C1(C(C2CCCC2O)=O)CC1 36436,C(=O)(N=c1[nH][nH]c2c1CN(Cc1ccc3c(c1)OCC3)C2)c1c(C)cccc1O 36437,C1(C)(C(=O)NCC(C)N(C(C2CC2(Cl)Cl)=O)CC)C2CC3CC(C2)CC1C3 36438,C1(C(=O)OC(C)(C)C)C(NC(=O)NCCCCCNC(C2CCCC2)=O)C1(C)C 36439,C(=O)(C(C)(C)c1cccs1)NC(C1CC(NC(=O)Cc2cnc[nH]2)C1)C 36440,C1(NC(CC(=O)N(C)C)=O)CN(C(=O)CCCc2ncc(Br)cn2)CC1O 36441,c1(C(=O)NC23C(CN(C(Cc4ccc(C)s4)=O)C2)C3)ccc2ncc(=O)[nH]c2c1 36442,CCCC(C(=O)N1CCC1C(=O)N(CC(C)(O)C1CC1)C)OC 36443,CC1CCN(CC(=O)NCCCC(C)NC(C23CC4CC2C3C4)=O)CC1 36444,C(=O)(C(C(C)C)c1cnc(C)s1)NCCC1CC(NC(CC(C)C)=O)C1 36445,CC1CN(C(c2nncs2)=O)CC1NC(C1CCC(N(C)C)CC1)=O 36446,N1(C(C(C)n2ccnc2)=O)CCC2(CCC2)C(NC(=O)CCc2cnoc2)C1 36447,C1(O)(C(C(=O)NC2CC(NC(c3c(C)snn3)=O)C2)(F)F)CCOCC1 36448,N1(C(c2c(C)nc(CNC(C(CCC)NC(N)=O)=O)o2)=O)CCC2(CCCN2C)C1 36449,c1(C(N2CC(OCCNC(CS(CC)=O)=O)C2)=O)cc(C(=O)OC)cc(O)c1 36450,c1(C(N2CC(C3(NC(C4C(CC)CCO4)=O)CC3)C2)=O)cc(S(C)(=O)=O)c(C)o1 36451,C1(C)(NC(C(C2CC2)NC(CC)=O)=O)CCCC1(F)F 36452,N1(CC(=O)NC2CCC(CNC(C3(N(C)C)CCC3)=O)C2)C(=O)CC(C)(C)C1=O 36453,C1(C(=O)NCC(C(=O)N2CC(OC(C)C)C2)O)CC2CCC2C1 36454,c1(C(N2CC(C)C(C(=O)NC3(C4CCCO4)CC3)C2)=O)cc2ncccc2[nH]1 36455,C(CC(O)C(F)(F)F)NC(C1(C)CCN(C(c2cc(F)cc(F)c2)=O)C1)=O 36456,Cc1nn2c(c1CNC(C1(F)C(C)(C)C1(C)C)=O)CN(C(C1(C)CC1F)=O)CC2 36457,c1(CNC(c2c(C)coc2)=O)nn(C)c2c1CN(C(C1CC1C(F)F)=O)CC2 36458,C1(CNC(C2(SCC)CC2)=O)CCN(C(C2C3CCCCC23)=O)CC1 36459,CC1=C(C)CC(C)(C(N2CC(O)(CNC(c3cc(F)c(O)c(F)c3)=O)C2)=O)CC1 36460,c1(C(=O)NCc2c(C(N(C(CCC)C)C)=O)scc2)cc(OC)n(C)n1 36461,C1(CC)COCCN(C(c2cc(CCNC(=O)C(C)SC(C)C)on2)=O)C1 36462,C1(C)(CC(=O)OC)CCN(C(c2ccc(C)c(I)c2)C(=O)NCC(C)C)CC1 36463,c1(C(=O)NCC(CC)(CC)NC(c2ccn(C)n2)=O)c(O)cc(F)cc1F 36464,C(=O)(C(O)Cc1ccccc1)NCCCN(C(=O)CC1CCCO1)C(C)C 36465,c1(-c2c(OC)nc(Cl)nc2C)ccc(S(=O)(=O)CC)cc1 36466,C1(NC(CC(C)(C)SC)=O)CN(C(C23CCC(N=[N+]=[N-])C2C3)=O)CC(C)(C)C1 36467,C1(NC(Cc2c(SCC)cccc2)=O)CN(C(=O)OC(C)(C)C)CCC1C#N 36468,c1(NCCc2c(C)cccc2)[nH]c(=NC2CC2c2ccccc2)nc2scnc12 36469,Cc1ccc(C)c(C(=O)NC2CC(C)N(C(C3CC(O)(C(F)(F)F)C3)=O)C2)c1 36470,c1(C(C(C)NCc2cnn(C(C)(C)C)c2)O)ccc(F)cc1F 36471,C=CC(CC)CC(=O)NCCC1CSCCN1C(c1n[nH]c(C2CC2)c1Cl)=O 36472,c1(OC)nc(C(=O)NCC(C)CNC(=O)CCC(=O)c2ccccc2)cc(O)n1 36473,NS(=O)(=O)c1cc(C(=O)NC2CC2NC(C23CC4CC2C3C4)=O)c(O)cc1F 36474,Cc1cn2c(CC(=O)NCC(C)NC(=O)CC3(C#N)CCC3)csc2n1 36475,C(=O)(C(CC(F)F)C1CCC1)NC1CC(CNC(=O)CCn2cncn2)CC1O 36476,C1(F)(C(=O)NCC(CO)NC(C(c2ccccc2)OC)=O)CCOCC1 36477,c1(C(N(CCCCN(C(C(CSC)O)=O)C)C)=O)ccc2nnnn2c1 36478,N1(C(c2c(OC)cccc2)=O)CCC(C)C(CNC(=O)CCc2cccs2)C1 36479,CN1CCC(C(N2CCC(CNC(C3CCCC34CCC4)=O)CC2)=O)S1(=O)=O 36480,Cc1cc(C)n(C(C)CNC(N2CCCC2Cc2ccncc2)=O)n1 36481,c1(OC)cc(F)c(F)cc1NNC(=O)NCCCCCS(C)(=O)=O 36482,c1(C(=O)NCC(C2CCC2)NC(CC(=O)NCC)=O)ncncc1Cl 36483,C(CCCCC(=O)NCC1(C(C)(F)F)CC1)N(C(c1ccc(CC)cc1)=O)C 36484,C1(NC(C2CCOC(C)C2)=O)CCCC(C(=O)NC2(OC)CCOC2)C1 36485,c1(CC(=O)NCCC(C)N(C(CC(C=C)C)=O)C)cc(Cl)cc2c1OCC2 36486,C(=O)(C(O)C(C)(C)C)N1C(C(=O)NCC2CC3CCC3C2)CC(C)C1 36487,Cn1nnnc1SCCCNC(CCNC(=O)COC1CCOC1)=O 36488,c1(C(=O)NCC2CN(C(c3n(CCC)ncc3)=O)C3C2C3)cc(F)ccc1OC 36489,C1(C)(CC(=O)N(CCCNC(C2(CC(F)(F)F)CC2)=O)CC)CCS(=O)(=O)N1 36490,C(CCCCC(=O)N(CC(C)O)CCNC(C1CC(O)CN1C)=O)OCC 36491,C(=O)(C(C(C)C)OC)NCC1C(NC(C(COC)C)=O)CCC1 36492,C1(NC(C2N(S(C)(=O)=O)CCC2)=O)CCN(C(C2CC3(CCCO3)C2)=O)CC1F 36493,N(C1CCCc2ccoc21)C(C1N(C(=O)C(=O)NCC2CCC2)CCN(C)C1)=O 36494,C1(CNC(C2CC(CCC)C2)=O)CN(C(c2ncnn2C(C)C)=O)CCC1(C)C 36495,C(C(C)C(C)C)NC(C(C)NC(C)=O)=O.C12CC(C1)CCNC2=O 36496,N1(C(C)C)CCCN(C(C2CCC(C(C)C)N2C(=O)C2=CCOCC2)=O)CC1 36497,CC1=CCSC1C(=O)NCc1ccsc1C(=O)NCCC(C)N(C)C 36498,C(=O)(CC1=NNC(=O)C1)NC(C1N(C(c2c(C)cc[nH]c2=N)=O)CCCC1)C 36499,C1(O)(CNC(CN2CC(C)C2)=O)CCCN(C(=O)CCS(C)=O)C1 36500,c1(N2CCC(N(C)C(C3CCCC(NC(N)=O)C3)=O)C2)ccc([N+](=O)[O-])cc1C#N 36501,c1(C(=O)NCC(C2CC2)NC(c2ccc(CC)c(N)c2)=O)cccc2scnc12 36502,c1(C(N2CCC3(CN(C(C(CC(C)C)OC)=O)C3)C2)=O)cc2nc(=O)ccn2[nH]1 36503,C1(C(=O)OC)CN(C)CCN1C(=O)CN(c1cccc(I)c1)C 36504,c1(C(N2CC(NC(C3C(=C)CC3)=O)C3(C2)CC3)=O)cc(Br)c(OC)cc1N 36505,c1(CC)cccc2[nH]c(C(N3CC(CNC(C4COCCO4)=O)C(O)C3)=O)cc12 36506,CC1=CCC(C(N2CC(O)(C(C)(C)CNC(=O)CC(C)(C)C)C2)=O)CC1 36507,c1(C(N2C3(C(N(C4CCCCC4)CCC)=O)CC(C2)C3)=O)cc2ccccn2n1 36508,C1(NC(CN(C)C(=O)C2CC2)=O)CC(N(C)C)CN(C(c2cccc(CO)n2)=O)C1 36509,c1(C(CC)C)nccc(N2CC(C)(C)C2C2CCN(C(c3cncs3)=O)CC2)n1 36510,C1(CNC(CCN2CCN(C)CC2)=O)CCN(C(C2C=CCC2)=O)C12CCC2 36511,c1(C(N(CCCNC(c2cccc(CN(C)C)c2)=O)C)=O)coc2ccccc12 36512,N1(C(C2CCC(CC)C2)=O)CCC(C=CC(=O)NC(CCO)C(F)F)CC1 36513,N1(C(C2CC(C#C)(O)C2)=O)CC(NC(c2cnn(CC(F)(F)F)c2)=O)CC1(C)C 36514,C(=O)(C(CC)CC=CC)N1CC(CN(C(CC2CC(=C)C2)=O)C)OCC1 36515,N1(C(CC2(CSC)CC2)=O)CC2C(NC(=O)C(c3ncccc3F)(F)F)C2C1 36516,C1(CNC(=O)CC2CCC3(CCC3)O2)CN(C(c2ccsc2)=O)C2(CCC2)C1 36517,C1(C(=O)NCC2(CNC(c3cnc(C)nc3)=O)CCCC2)CCC(C)(C)CC1 36518,C(=O)(CCCCCCCCC)NCC(CNC(C1C(=C)CC1)=O)(C)C 36519,c1(C(N2CCC3(CCN(C(C45CC(F)(C4)C5)=O)C3)C2)=O)cnc2ncnn2c1O 36520,CCC(C)CC(C(=O)Nc1ccc(NC)nc1)NC(c1cnc2n1CCCC2)=O 36521,CCC(CC)C(C)C(=O)NC(C)(C(=O)NCC1=CCCCC1)C1CCC1 36522,C1(O)(CNC(c2cnc(C(F)F)s2)=O)CN(C(c2cn(C3CCC3)nn2)=O)C1 36523,C1(CNC(c2c(C)scc2)=O)C(C2CC2)CCN1C(c1coc(C(C)C)n1)=O 36524,C1(NC(C(CC#C)C2CC2)=O)CC2CC1CN(C(=O)CC1CCS(=O)(=O)CC1)C2 36525,CC1CCC(NC(=O)C(C)(C)c2cncnc2)CN1C(=O)C=Cc1ncc[nH]1 36526,C1(CC#N)C(=O)C(C)OC(=O)N1.C(=O)(C(C)NC(=O)OC(C)(C)C)OC 36527,C1(C(=O)NCCN(C2CC2)CC)CC2(CC2)CN1C(C1CCCC(=O)C1)=O 36528,N1(C(C=Cc2cnc(C)s2)=O)CCCC2C1CCCN2C(=O)C#CC1(C)CC1 36529,CCC(C)(C)CC(=O)N(CC(C)N(C)C(C1CSCN1C(C)=O)=O)C 36530,C1(O)(C(=O)NC2(CNC(=O)Cc3cc(C)ns3)CC(OC)C2)CC2CCC1C2 36531,C#CCC(CC#C)NC(=O)C(C)(C1CCC1)NC(c1cc(=N)[nH][nH]1)=O 36532,N1(C(c2c(CC)cccn2)=O)CCC(F)(F)C(C(=O)Nc2cc(O)ccc2Cl)C1 36533,C1(C(N(C)C(=O)C2CC2)=O)CC(N)C1(C)C.c1(C(=O)NC)ncoc1C1CCC1 36534,C1(CC)(NC(=O)C(c2ccc(F)c(Cl)c2)C)CCN(C(=O)C(C)S(N)(=O)=O)CC1 36535,CC(CC(F)F)C(=O)N(C1CCC(NC(=O)C(C)N2CCC2)CC1)C 36536,N1(C(CCCCC)=O)CC2CCC(C1)C2CNC(C1(F)CCOCC1)=O 36537,C1(CCOC)CCCCN1C(N1CCC(C)(O)C1)=O 36538,C1(N(C=O)Cc2nscc2Br)CCc2nncn2C1 36539,c1(C(N2CC(NC(C(CCC)(C)CC)=O)C(C)C2)=O)nnc2ccccc2n1 36540,CC1(C)OC(=O)CC1C(=O)NC1CCCN(C(=O)CSCC(F)F)C1 36541,N1(C(C(CCNC(C2(CCC)CC(=O)C2)=O)O)=O)CC2(C1)CC(C)(F)C2 36542,N1(C(C=CSC)=O)CCC2(CC1)CN(C(C1(C)C=CCCC1)=O)CC(C)O2 36543,C1(NC(=O)CCF)CCCCC1NC(c1coc(Br)c1)=O 36544,CCCC(C(=O)N1CC(CNC(c2cocn2)=O)(COC)C1)C(C)C 36545,C1(NC(=O)CC2CCCCC2)CC(F)CN(C(=O)C(F)F)C1 36546,C1(NC(c2c(C(C)C)nns2)=O)CCN(CCNC(C2CC2(Cl)Cl)=O)CC1 36547,N(C(=NCCC(=O)NC1CCCCC1C1CC1)NCc1ccccc1C#N)CC 36548,C(CCN=c1cc(C)nc(CC)[nH]1)N(CC)CC.c1ccc(C(F)(F)F)cn1 36549,C1(NC(=O)C=Cc2cccnc2)CC2CCC1(NC(=O)CCC1CC(F)(F)C1)C2 36550,N1(C(C(=O)NCC)=O)CCC2(CC1)COC(CNC(c1c(Cl)nn(C)c1C)=O)C2 36551,Cc1c(Cl)ccc(C(=O)N(C2CCCN(C(c3cccc(=O)n3C)=O)C2)C)c1O 36552,C1(NC(COCC(C)C)=O)CCN(C(C2CC(N(C)C)C2)=O)C(C)C1 36553,Cc1nc(Cl)nc(N2CCC3(CC2)CN(C(C2CC(=O)N2)=O)CCO3)c1[N+](=O)[O-] 36554,C(=O)(C(C)(c1ccccc1)OC)N(C1(CC(=O)NCC2(C(=O)OC)CC2)CC1)C 36555,Cc1nnccc1CNCc1cccnc1N1CCCCC1 36556,c1(C(=O)OCC)nnc(CNCC(c2nnc(C)o2)C)s1 36557,n1(CC(=O)NCC(C2CC2)NC(c2ccccc2)=O)nc(Cl)ccc1=O 36558,CC1CN(C(c2scnc2C(F)(F)F)=O)CCN1C(C1CC2(CCOC2)C1)=O 36559,c1(CN2C(C3CCN(C(C(CC=C)C)=O)CC3)CCC2)ccc([N+](=O)[O-])cc1F 36560,c1(C(N2CCC(C)(c3cccs3)CC2)C(=O)NCC(C)C)cc(S(N)(=O)=O)cs1 36561,Cc1ccc2c(C(=O)N(C3CCN(C(=O)COc4ccsn4)C3)C)ccnc2c1 36562,c1(Cn2c(C(=O)OCC3(CS(C)(=O)=O)CC3)ccn2)ccc(Br)cc1F 36563,CC1CCC(NC(=O)CN2CC3CC3C2)CN1C(c1cc(N)ccc1F)=O 36564,C1(COC)CCN(C(c2cc(CNC(=O)C(CO)OC)cs2)=O)C1(C)C 36565,C1(NC(C2(C=C)CCC2)=O)COCCC1NC(C1(Cc2cccc(Cl)c2)CC1)=O 36566,c1(C(=O)NCC(CCCC)NC(=O)C(C)SCC)ccnc(F)c1OC 36567,c1(CC)cc(C(N2CCC(CCNC(=O)CC3CCCO3)C2)=O)ccc1OC 36568,Nc1ccc(F)c(C(=O)NC2CCC(NC(c3snc(O)c3Cl)=O)CC2)c1F 36569,N1(C(C=C(C)C)=O)CCCC(C)C1C(=O)C(C)N(C)C 36570,C1(CNC(c2ncoc2-c2ccon2)=O)CN(C(=O)CCOCC(F)F)CC1O 36571,c1(OCC)ccccc1CCNC(=O)NC(C)Cc1cccc(N)c1 36572,C12(C(=O)NCC3N(C(c4c(C)ccnc4)=O)CCC3)CCCN(CC1)C2 36573,Cc1cc(C(=O)NCc2cc[nH]c2C(=O)NCC=C(Cl)Cl)cc(C#N)c1 36574,N1(C(c2occ(C)c2)=O)CCCC(O)(Cn2cc(CC3CCCCC3)nn2)C1 36575,N1(C(CN(C(=O)Cn2nc(C)nc2C)CC#C)=O)CCCC(C)C1CO 36576,C1(C(N2CCN(C(C3CC3C(F)(F)F)=O)C(CF)C2)=O)CC2CCC1CC2 36577,C(CN=C(NCc1cc(O)cc(O)c1)NCc1cc(C)ccn1)N(CC)CC 36578,c1(CC(=O)N(C2CC(C(=O)NCC(C)Cc3cn[nH]c3)C2)C)cccn1C 36579,c1(C(=O)NCCCOCCN(C(=O)CC2COC(=O)C2)C)c(Cl)cnn1C 36580,c1(NC2(CNC(CC(=O)OC)=O)COC2)cc(Br)c(F)cc1OC 36581,C1(OC)CC(NC(C2CC=CC2)=O)CN(C(C2CCC(=O)N2C2CC2)=O)C1 36582,C1(C(=O)NC2CCC(NC(c3ccncc3O)=O)C2)CCCC1(F)F 36583,Cc1nncc(C(=O)NC2CCC2NC(=O)CC2CCCCN2C)c1C 36584,C1(C(=O)NCC(CNC(CC2C(OCC)COCC2)=O)C)CC(=O)NC1(C)C 36585,N1(C(Cc2ncc(CC)[nH]2)=O)CC2(NC(=O)CCCn3cccc3)CC1C2 36586,c1(CN2C(C(=O)Nc3c(OC)cc(C)cc3)CCC2)cc([N+](=O)[O-])cc(O)c1O 36587,N1(C(Cc2nc(C)sc2)=O)CCCN(C(=O)Cc2cccc3nonc23)C(C)C1 36588,C(CCC(N)=O)(C(=O)NCC1CCN1C(=O)CCN1CCCS1(=O)=O)NC(C)=O 36589,C(C(COC)C(C)C)NC(c1cccc(C)c1)(c1n(CCCSC)nnn1)C(C)C 36590,C(=O)(CCC(=O)NN(C)C)NC1CC(C)CN(C(c2cc(O)ncn2)=O)C1 36591,c1(CC)nc(C)c(C(N2CC(C(=O)NCCC3C=CCC3)(CC)C2)=O)o1 36592,C1(C(N2CCC(CO)C2)=O)CCCN(C(C2CC23CCCC3)=O)CC1 36593,CC1(C)CCCC(CC(=O)NCC2COCCN(C(c3ccoc3Cl)=O)C2)C1 36594,c1(C(=O)NCC2C(NC(COCC)=O)COC2)c(F)cccc1[N+](=O)[O-] 36595,N1(Cc2onc(-c3cc(C)c(F)cc3)n2)CCN(C)C(C)C1C 36596,c1(CNC(N2CCC(c3c(C(=O)OC)c[nH]n3)C2)=O)cc(C)n(C)c(=O)c1 36597,C(=O)(C(C)(O)CC(C)C)N1CC(CCNC(=O)CCS(=O)(=O)N(C)C)(OC)C1 36598,C(=O)(C#CC1CCOCC1)NC1CCC(CNC(C(c2ccccc2)C)=O)CC1 36599,C(CC(C)C)(C(=O)N(CC(=O)NCC1CCC(C)(C)CO1)C)NC(C)=O 36600,C1(NC(CP(C)(C)=O)=O)CN(C(c2cc(O)ncc2Br)=O)CC12CCC2 36601,CCCS(=O)(=O)c1ccccc1C(=O)NCCCCCNC(C1CC1F)=O 36602,Cc1nc(C(=O)NC2CC2CNC(=O)C=CC2CCCCCC2)c(C)n1C 36603,n1(COC)nccc1C(=O)NC1CCC1CNC(C1CCC(C(=O)OC)C1)=O 36604,C1(CNC(c2n(CCSC)nnn2)c2ccncc2)CC2CCC1CC2 36605,c1(OCC)ccc(C)cc1C(NC(=NCC1(C#N)CCOCC1)NC(C)C)C 36606,Cc1ccc(S(=O)(=O)N2CCC2C(=O)Nc2cc(C)cnc2Br)c(F)c1 36607,N1(Cc2ncc(CC)o2)CC2(C)CN(C(=O)CCC(C)OC)CC2(C)C1 36608,c1(C(=O)NCC2N(C(c3cnc(=N)[nH]c3)=O)CCCC2)ccc2c(c1)CCCS2 36609,C1(N(C(CCN(C(CC(C)SC)=O)CCO)=O)C)CCOC(C)(C)C1 36610,C1(C2CCN(CC(=O)N(c3cnsn3)C)C2)CCCCN1Cc1ccc(O)nn1 36611,C1(C#CC(=O)NCC(O)C(=O)NC)(CC)COC1.C1CCC(=O)NC12CCC2 36612,C12(CNC(C3OCCN(C)C3)=O)CCC(CNC(C3CC3(F)F)=O)(CC1)CO2 36613,c1(C(C(=O)NCCCCCC)N(CC(F)(F)Cl)C)ccc(Br)cc1OC 36614,N1(C(C)=O)CCC(CC(=O)O)C(NC(=O)Cc2cc(C)nn2C)C1 36615,C(=O)(NNC(=O)C1OCCC1Cn1cc(C)cn1)OCC 36616,N1(C(c2c(OC)cnnc2)=O)CC(C(=O)NCC2CCCN2CC)CC12CCC2 36617,CC(C)C(O)C(C)C(=O)NCCCC(C)(C)NC(c1cc(C2CC2)on1)=O 36618,c1(SC)ccc(C)c(C(=O)NC(C)C(C)(C)NC(=O)CN2CC(C)(C)C2)c1 36619,CC1CCc2nc(C(=O)NCC3CCCC3NC(=O)CC(C)(C)O)ccc2C1 36620,C1(NC(c2nc(-c3c(C)cccc3)sc2)=O)(CNC(=O)C(N)=O)CC2CCC1C2 36621,Cc1ccc(F)cc1CC(=O)NC(C)C(C)(C)NC(C1CC2(CCC2)CO1)=O 36622,n1(CC)ncc(Br)c1C(N1CC(NC(=O)CC(C)CF)C(C)C1)=O 36623,c1(C(N2CCC(NC(c3ccc(S(C)(=O)=O)s3)=O)C2)=O)cccc2nc(Cl)cn12 36624,C(=O)(N=c1[nH]nc(C2CC2)s1)N(c1ccccc1CCSC(C)(C)C)C 36625,C1(COC)(NC(=O)C=CC(F)(F)F)CCN(C(=O)Cn2cnc(=N)[nH]2)CC1 36626,Cc1nc(F)ccc1C(C1CC1)NC(=O)CC1CCN(C(=O)C=CCO)C1 36627,CCC(N=c1ccnc(NC2CCN(CCC(C)(C)C)CC2)[nH]1)C(C)C 36628,C1(CC(=O)N(CCn2c(C)ncc2)C)COCCN1C(C1CCC(C)(C)C1)=O 36629,CC(C(=O)N1CCCC1CCNC(c1c[nH]cc1C(F)(F)F)=O)C(F)(F)C(F)F 36630,CCCCCCCCC(C)C(=O)NC(C1CCN(C(C2(C)CCC(=O)C2)=O)C1)C 36631,N1(C(C(C)N(C(C)=O)C)=O)CC(=O)NCC1C(=O)NCC1(O)CCN(C)C1 36632,N1(C(COC)=O)CCCC(C)(C)C1CNC(C1(Cc2ccc(F)cc2)CC1)=O 36633,c1(CC(=O)NC2C(NC(c3cc(C(C)C)nn3C)=O)C2)cn2ccccc2n1 36634,C1(CN(C(CCCOCC)=O)C)CCCC(NC(c2nnc(C(C)(C)C)s2)=O)C1 36635,c1(N2CC(c3nc(C)[nH]n3)OCC2)ncnc2sc(C(C)(C)C)cc12.C1C(=O)N1 36636,c1(N2CCCC(CCNC(CC3C(C)CCC3)=O)CC2)ncc([N+](=O)[O-])c(=N)[nH]1 36637,C1(C(=O)NC(CCCNC(CCC(=O)NCC)=O)C)COCC(C)(C)O1 36638,N1(C(C2CCC(C)O2)=O)CCC(C(C)C(=O)NC(C2CCCC2)CO)CC1 36639,CC(C)(C)CC(=O)NCC1CC(CNC(=O)Cc2ccn(C3CCCC3)n2)CO1 36640,C1(C(=O)NCC(C)CN(C)C(c2cnn(C3CCCC3)c2)=O)OCC1(C)C 36641,C1(NC(c2ccc(OC)c(Br)n2)=O)CCc2ncc(Br)n2C1 36642,c1(C(=O)NCCC2CN(C(c3c(CC)nccn3)=O)C2)cc2c(=O)[nH]ccn2c1 36643,n1(CC)cnc(C(=O)NC(CO)C(C)NC(=O)CCNC(C2CCOCC2)=O)c1 36644,C(=O)(C(F)CCC(C)(C)C)NCC1CCCN(C(C(CC)NC(C)=O)=O)C1 36645,Cc1cc(C(N2CCC(F)(CNC(C3CCCN3C3CC3)=O)C2)=O)nnc1C 36646,CN=c1[nH]cc(C(=O)N(C)CCN(C(=O)Cc2cnn(C(F)F)c2)C(C)C)s1 36647,C(c1ccc(F)nc1)=CC(=O)NC1CCCCC1CNC(c1cncc(Cl)c1Cl)=O 36648,C1(N(CCCC)C(=O)C=Cc2cscn2)CCN(C(c2cc(C)cs2)=O)CC1 36649,c1(OC2CN(CC(c3ccc(CC)cc3)O)C2)ccc(Cl)cc1[N+](=O)[O-] 36650,C1(C(N(CC(C)(C)N(C)C)C)=O)CCN(C(C2CC(C)(C)C2)=O)CC1 36651,N1(CC(COCC(C)C)O)C2CCC1CN(Cc1ccc(C3CC3)o1)C2 36652,C1(C2CCOCC2)(C(=O)NCC(C(C)(C)C)NC(C(C)CC(F)F)=O)CC1 36653,C1(CNC(C(CC=CC)NC(c2cc(CN(C)C)on2)=O)=O)OC(=O)CC1(C)C 36654,Cc1cc(C)c(C(=O)NCCC2(O)CCCN(C(C34CCC3C4)=O)C2)c(=O)o1 36655,C(=O)(C1=CC2(CN(C(C3C(C)(C)C3(F)F)=O)C2)OC1)N(CCCO)CCC 36656,C1(NC(C(CCC)=CCC)=O)CCCC(C(=O)NCCN2CCCOCC2)CC1 36657,C(C(F)(F)C(F)F)NC(C1CC(CF)C1)=O.C12(CCC1)CC(=O)N2 36658,C1(CNC(C(CC)CO)=O)CCN(C(c2cnn(C3CC3(F)F)c2)=O)C1(C)C 36659,c1(C(=O)NCC(C)CNC(c2cccc(I)c2)=O)ccc2cnccc2c1 36660,c1(C(C)=O)cccc(OC(C)C(=O)NCCCCC(C)NC(=O)CSC(F)F)c1 36661,c1(CC(=O)NC(C(N)CO)C(=O)O)cc(Cl)ccc1I 36662,CCCC(C(=O)NCC1CCCCN(C(=O)CCN2CCOCC2)C1)S(N)(=O)=O 36663,Cc1noc(C(F)F)c1C(=O)NCc1cccc(CN(C(=O)C(C)(C)F)C)c1 36664,N1(C(C2(OC(C)=O)CC2)=O)CCC(C(C)(C)C)(CNC(C2CC(C)(C)CO2)=O)C1 36665,c1(CC(N2CC(O)(C(C)NC(C3CC(CCC)C3)=O)C2)=O)sc(C)nc1C 36666,N1(C(CC2(OC)CCC2)=O)CCN(C(c2ncnc(C)c2C)=O)CC(C)C1 36667,c1(C(=O)OC)c(C)ccc(NC(C2COCCN2CC2CCCC2)=O)c1C 36668,c1(N(C)CCC2CCCCC2)nc2c(c(=NCC3CCC=CCCC3)[nH]1)COC2 36669,CCC(C)C(=O)C1CC1.C12CC(C1)OCN(CCC)C2=O.C1C(=O)N1.C1(N)CC1 36670,N1(C(c2c(C)snc2)=O)C2CCC1C(CNC(=O)CCc1nc(C3CC3)no1)C2 36671,CC1(NC(c2nnsc2-c2ccccc2)=O)CCN(C(=O)CC(F)(F)F)C1 36672,C1(C(=O)NCC23CC(NC(c4ccc(CC)s4)=O)(C2)C3)CC(C)(C)C1C(F)(F)F 36673,N1(C(C(CSC)C)=O)CCC2CCCC12C(N1CCCCC(N(C)C)C1)=O 36674,C=C(Br)CC(C)(C)C(=O)N1CC(CNC(=O)C(C)NS(C)(=O)=O)C(C)C1 36675,C(=O)(C1=C(F)CN(C(=O)CC=C(Cl)Cl)CC1)NCc1c(C)ccc(O)c1 36676,C(CC(CNC(=O)CCF)NC(=O)CNC(c1cccs1)=O)Oc1ccccc1 36677,N1(CCNC(C(c2cscn2)N(C)C)=O)C(=O)NC(C)(c2ccc(Br)cc2)C1=O 36678,c1(-c2c(C(=O)NC(C)C(C)n3ccnc3)c[nH]n2)ccc2c(c1)CCCO2 36679,c1(C(N2CCC(NC(CCc3c(C)nccc3)=O)C2)=O)ccc(C(F)F)c(Cl)c1 36680,c1(C2C(C(=O)NC3C(NC(=O)CCc4ccon4)C3)C2)ccc(Cl)cc1 36681,c12ccc(Br)c(c1F)NC(=O)C2N(C(C)(C)C)CCN(C)C.C(COCC)OC 36682,C1(NC(C2C(CC)N(C(=O)CCC(C)(C)OC)CC2)=O)CC(C)(C)OC1(C)C 36683,C(=O)(C#CC1CCCCC1)NC1CC2CN(C(C(CCCOC)C)=O)CC21 36684,C1(C(=O)NCCOCCN(C)C)CNC(=O)CN1C(=O)CCn1cccc1 36685,C1(C(=O)NC2C(NC(C3(CC#C)CCCC3)=O)CCC2)CC2C=CC1C2 36686,c1(C(=O)NC2CCC(C)(CNC(=O)C3=C(Cl)CC3)C2)cccn2cncc12 36687,Cc1ccc([N+](=O)[O-])cc1C(N1CCC2CN(C(C3(C#N)CC=CC3)=O)CC12)=O 36688,c1(C(=O)NCCC2(CNC(C(C)O)=O)CCCC2)nccc2cc[nH]c12 36689,CCCCC(F)F.C(=O)(C(C)COC)N(Cc1ccccc1)C 36690,C12(C(=O)NCCN3CCCN(C(CP(C)(C)=O)=O)CC3)CCCCC1C2(F)F 36691,C1(CC(N2C3CN(C(C4(C)CC(=C)C4)=O)C(C3)C2)=O)CCc2ccccc2C1=O 36692,C(c1ccc(C)cc1C)=CC(=O)NC1CCCC(CNC(CN(C)CC)=O)C1 36693,Cc1cc(F)cc(C(N2CC(N(C)C(C3CCOCC3)=O)C3(CC3)C2)=O)c1O 36694,C=CCC(Cc1ccccc1)C(=O)NCCCOc1c(F)cccc1F 36695,N1(C(C(C)SCC)=O)CCC(CNC(c2cnccn2)C2(CO)CC2)C12CCC2 36696,N1(C(C=Cc2cc(C)no2)=O)CC2CCC(N(C(=O)C3=CCCSC3)C)C2C1 36697,c1(C(N2C(C)(C(=O)NC)CC(O)C2)=O)nccc2[nH]ccc12 36698,C(CNC(=O)Cc1ccccc1)(C(C)(C)C)NC(CCN(C)CCO)=O 36699,C1(C(=O)NCCCN2CC=CC2)CCC(O)CN1C(c1cc(C(F)F)[nH]n1)=O 36700,N(C(=NCc1ccccc1[N+](=O)[O-])N1CCC(C)(F)C1)Cc1cc(C)on1 36701,c1(OC(c2cncc(F)n2)=O)ccnc(NC(CNS(C)(=O)=O)C2CC2)n1.c1ccco1 36702,C1(OC)(CNC(c2n[nH]c(C)c2O)=O)CCN(C(c2cn(C)nc2C(C)C)=O)C1 36703,CC1CC2(CCN(C3CCN(C)C3=O)CC2)CN1C(C1CC1(Cl)Cl)=O 36704,c1(NC(=O)OC(C)(C)C)cccnc1ONS(=O)(=O)Oc1ccccc1 36705,N1(C(C2C(c3n(CC)ccn3)OCC2)=O)CC2CC(C)N(C(C3CCC3)=O)C2C1 36706,c1(C(N(CCCO)CC)=O)cc(CNC(=O)C(OC)OC)[nH]n1 36707,N1(C(CC2(OCC)CC2)=O)CCC(CCNC(c2cnc(C3CCC3)o2)=O)C1 36708,C1(NC(c2ccc(Br)cn2)=O)CC2CC1CN2S(=O)(=O)CCBr 36709,C#CC1(C(=O)NCC2CCC=CO2)CN(C(=O)CC2CCCC2O)C1 36710,N1(C(C=Cc2scc(C)n2)=O)CC(CO)C2(C1)CN(C(c1c(C)noc1C)=O)C2 36711,C(=O)(C(C)(C)CCCF)NCC(C(=O)NCc1c(C)cc(O)cc1)CC1CC1 36712,N1(C(C2C(COC)CC2)=O)CCCC(F)(C(=O)NCC23CCCC2CCO3)C1 36713,C1(CNC(C2CC3(C2)CC3F)=O)COCCN1C(=O)Cn1cnnc1O 36714,CC1CN(C(c2cncc(F)c2)C(=O)NC2(C)CC2)C12CCOCC2 36715,c1(C(=O)NC(CNC(C(c2c(C)nn(C)c2)O)=O)CO)cc(Cl)cc(Cl)c1 36716,CC(=O)C(C)(C)CC(=O)N(C1CCN(C(c2ccccc2[N+](=O)[O-])=O)C1)C 36717,C(CC(=O)N1CC(C)(C)C1C(C)C)(C(C)C)NC(c1cccc(OC)c1)=O 36718,N1(c2snc(CCC)n2)CCC(NC(c2cn(C3CCOC3)cn2)=O)C(C)C1 36719,c1(C(=O)NC2C(NC(=O)Cc3ccon3)CS(=O)(=O)C2)cc2cccc(Cl)c2[nH]1 36720,C1(CNC(C(C(C)C)SC)=O)CN(C(c2ccc(Cl)c(C)c2)=O)CC12CCC2 36721,C(=O)(CCCCCNC(C)=O)NCC1CC(NC(COCCC)=O)C1 36722,C(=O)(C(C)C(C)(C)C)NCCCN(C(=O)C=Cc1cccc(CO)c1)CC 36723,c1(C(N)=O)ccncc1NC(c1cc(CNC(=O)C(C2CCOCC2)O)on1)=O 36724,c1(CN2CC(F)CC(C(=O)NC(CCC)C(=O)NC)C2)ccc(F)c(NC)c1F 36725,C1(CNC(c2c(C)cn(C)n2)=O)COC(C)(C)CN1C(=O)CCCN1CCCC1 36726,N1(C(C(N)=O)=O)CC2CC1CN(C(c1cc(C(N)=O)co1)=O)C2.N1(C(=O)N)CCCC1 36727,C1(NC(C(=Cc2ccccn2)C)=O)C2CCC1N(C(c1cc(C(F)F)no1)=O)C2 36728,C1(C2CC2)(C(=O)NCC(c2ccccc2)CNC(C)=O)CC1 36729,CCCC(C)CC(=O)NCCCC(O)C(=O)NCc1cnccc1Cl 36730,C(CCCC(=O)N(C(C)C(=O)N(C1CCNC1=O)C)C1CC1)NC(C)=O 36731,c1(C(N(C)C(C2CCCN2C(C2CC23CC3)=O)C2CCC2)=O)cccc(F)c1 36732,Cc1c(NCCCN2CCCN(C)CC2)nc[nH]c1=NCC1CC2(C1)CC(O)C2 36733,N1(C(CCSCC)=O)CCC(NC(=O)CC2(C)CCOCC2)C1C(C)(C)C 36734,c1(NC(C)=O)ccc(C(N2CCCN(C(C3CC3(C)C(F)F)=O)CC2)=O)c(C)c1 36735,C1(C)(COC(C(C(C)C)n2cncn2)=O)CCCN(C(=O)OC(C)(C)C)C1 36736,c1(NCCCCC(N)=O)[nH]c(=NCCCC2CC2(Cl)Cl)nc2scnc12 36737,c1(C(N(CCCNC(C=CCCC)=O)CC)=O)c(OC)nsc1OC 36738,C#CCCCC(C)C(=O)N1CCOC(CC(=O)NC(c2n[nH]c(C)n2)C)C1 36739,C1(C(=O)Nc2cc(OC)c(O)cc2)CC12CCN(C(c1cc(O)n(C)n1)=O)CC2 36740,CCS(=O)(=O)c1cc(F)ccc1NC(=O)C(N1CCC2CSCC2C1)=O 36741,Cc1ccc(CC(N2CCC2CNC(=O)CN(S(C)(=O)=O)C)=O)c(Cl)c1 36742,C1(O)(CCNC(Cc2ccc(SCCCC)cc2)=O)CCN(C(=O)C=C(C)Cl)C1 36743,C(=O)(C=C1SCC(=O)N1C)NC1CCN(C(c2n(CCC)ccc2)=O)CC1O 36744,CC1CC(C(=O)NC2(CCNC(=O)Cc3ccc(Br)nc3)CCCC2)=NO1 36745,C(=O)(C1CCc2ccccc21)N1CCCC(C(C)NS(C(CC)C(C)C)(=O)=O)C1 36746,c1(CC(=O)NCCC(C)NC(C2CC23CC3)=O)c[nH]c2ccc(Cl)cc12 36747,N1(C(=O)CC2CCCN(C(c3cnn(C(F)F)c3)=O)C2)CCC(CO)C(F)C1 36748,CC(CCCCNC(C1CCCC12CC2)=O)NC(c1conc1C(F)(F)F)=O 36749,c1(C2C(C(N3CCC(N(C)C(c4scnc4Cl)=O)C3)=O)C2)ccccc1Cl 36750,c1(CNC(c2cc(C)ns2)=O)nc(C)c(C(=O)NCC(C)(C)N2CCCC2)o1 36751,CC1=NOC(C)(C(=O)NC(CO)C(C)NC(=O)Cn2nc(C)cc2C(F)F)C1 36752,C(C1=NOC(CC2CCOC2)C1)N(CC(c1ccccc1)OC)C 36753,C(CCC(=O)NNC(=O)C1CCCO1)n1cc(-c2cccc(NC)c2)nn1 36754,C(c1c(C)noc1C)=CC(N1CCC(N(CCC)C(C2CCCN2C=O)=O)C1)=O 36755,N1(C(CC(CC)C2CCC2)=O)CCN(C(C2CCc3c[nH]nc3C2)=O)CC(O)C1 36756,Cc1cc(NC(=O)C(CC2CC2)NC(=O)C2=CCCOC2)cc(CO)c1 36757,N1(C(C2(SC)CN(C(=O)C(C3CCOCC3)O)C2)=O)CC(C#N)(CCF)C1 36758,CC(CN=[N+]=[N-])NC(C1COCC1NC(=O)CC1(C)CCC1)=O 36759,C12(C(N(C)OC3CCCC3)=O)CC(C)(CN1C(c1cc(C(N)=O)co1)=O)C2 36760,Cc1ccc(CNC(c2nnnn2C(C)C)(C)CC2C=CCC2)c(F)c1 36761,c1(OC)ccc(NC(C2CC3(CC3)CN2Cc2ccnc(Cl)c2)=O)c([N+](=O)[O-])c1 36762,C1(CNC(CCC#CC)=O)CN(C)CCN1C(C1CC1Sc1ccccc1)=O 36763,C1(CC)CN(C(c2cc[nH]n2)=O)CCC1NC(=O)Cc1ccccc1Cl 36764,CC(C)(CCCO)C(=O)NCCCCC(C)NC(c1c[nH]nc1[N+](=O)[O-])=O 36765,C(=O)(C(CNC(C1(C)CCSCC1)=O)CC=C)NCCOCCC=C 36766,Cc1nc(N2CC3C(CNC(=O)CC(C)CC(C)(C)C)C3C2)c2cc[nH]c2n1 36767,c1(CC)ccc(F)cc1C(=O)N(CCNC(c1nn(C)cc1Cl)=O)CC1CC1 36768,N1(C(C(CC)OCC)=O)CC(NC(=O)C(c2cnn(C)c2)C)CC12CCOCC2 36769,C1(C(N2CC(O)(CCNC(=O)COCC(F)(F)F)C2)=O)CCC(C2CCC2)CC1 36770,N1(C(C(=O)OCC)=O)CCC(C(F)C(=O)Nc2ccc(SC)cc2)CC1 36771,C(=O)(CC(C)c1ccco1)N(C(CNC(=O)CC#N)C1CC1)C 36772,C=Cn1nccc1C(=O)NCC1CCC1NC(C1(C(N)=O)CC1)=O 36773,C1(NC(C(c2ccccc2)C)=O)CCCCN(Cc2ccncc2Cl)C1 36774,Nc1cc(=NCC2CC3(CCNC3)CO2)[nH]cn1 36775,C1(OC)CCC(CC(=O)NC2CCN(C(c3ccn(C)c3)=O)C2C(C)C)CC1 36776,c1(C(N2CCOCCC2C2CC2)C(=O)NC)ccc(S(=O)(=O)C(C)C)cc1 36777,c1(C(=O)NC(CNC(C2C(OCC)C2C)=O)C(C)(C)C)cnc(N)c(O)c1 36778,N1(C(c2c(CCCC)ocn2)=O)CCN(C(=O)Cc2ccns2)CC1CO 36779,C(C(O)CC(=O)N1CCCC1C(=O)NC1CC1)NC(=O)OC(C)(C)C 36780,Cc1c(C(=O)NC(C2CCCN2C(=O)Cc2cn(C)nc2Cl)C)sc2nccn12 36781,c1(C(N2CC(COC)N(C(c3ncncc3F)=O)CC2)=O)cc(C)cc(C)c1O 36782,O(C=CC(=O)N1CCCC1C1CCN(C(=O)C(F)CN(CC)CC)C1)CC 36783,c1(C(=O)NCC2(O)CCN(C(CC)=O)C2)ccc(C#N)cc1C 36784,C(=O)(CC1CCC(C)(C)c2ccccc21)NCCCNC(C(COC)O)=O 36785,CN=c1[nH]ccc(C(N2CCCC(NC(C3(F)CCOC3C)=O)CC2)=O)c1N 36786,c1(SC)ncc(C#N)c(N2CCCC(C(N3CCCC(CO)C3)=O)C2)n1 36787,c1(NC(C(C2CCCCC2)NC(C=CCOC)=O)=O)ccc(C)c(CO)c1 36788,c1(CC)n[nH]cc1C(=O)NCC(N1CCC(C(=O)NCCOC)C1)=O 36789,C(CC(C)C)(C(=O)N1CCC(C)C(C(=O)NOC(COC)COC)C1)OC 36790,C=CCC(C(=O)N(C(C)CN(C)C)C)NC(C)=O.C1(=O)C(C)N1 36791,N1(C(=O)CC2C=CCC2)CC2(CCN2C(c2cc(-c3ccncc3)on2)=O)C1 36792,C1(CC(N2CC(CNC(Cc3cccc(SC)c3)=O)C2)=O)CCC2(CCC2)CO1 36793,CCCC(CCOC(C(=O)OCCOC(C)(C)C)(C)C1(C)CC1)C1CC1 36794,Cc1cc(O)ccc1C(=O)NCC1CCCN(C(=O)CCC2CCCN2C)CC1 36795,Cc1nn(CC(F)F)c(C)c1C(=O)NC(C)CCCNc1ncncc1Cl 36796,CC(CC(F)F)C(=O)N(C)CC1CCCCN1C(=O)C(O)Cc1ccccc1 36797,N1(C(C2CC(=O)NCC2)=O)CCC(CNC(=O)CCc2ncc[nH]2)C(F)(F)C1 36798,c1(CNC(=O)CC2(NC(=O)CC3CCCOC3)CCC2)ccnc(O)c1 36799,Cc1nc(CO)sc1C(=O)NC1(C)CCN(C(=O)CSCc2csc(=N)[nH]2)C1 36800,C1(CN(C(C2CC(OC)(OC)C2)=O)C)CCc2nc(C(F)(F)F)cn2C1 36801,N1(C(C2CC(=O)NC2)=O)CC2(C1)CN(Cc1cc(Cl)ccn1)C2 36802,N1(C(C(CC)NC(C)=O)=O)CCN(C(=O)Cc2nc([N+](=O)[O-])n[nH]2)C(C(C)C)C1 36803,c1(C(C(c2nnnn2CCCF)NCC(C(C)C)OC)(C)C)ccc(F)cc1 36804,C1(C(C)NC(=O)CC2CC3CC3C2)CCN(C(C2(COCC)CCCO2)=O)CC1 36805,C1(NC(c2nc(CC)oc2)=O)CC2CC1N(C(C1CCC(F)(F)CC1)=O)C2 36806,N1(C(C2(C)CC(=O)C2)=O)CCC(C)(C)C(CNC(c2c(F)cccc2F)=O)C1 36807,N1(C(CCNC(CC(CC)C2CC2)=O)=O)CC2CCC(C1)O2 36808,N1(CCN(C(C(c2c(F)cccc2F)NCC)=O)C)CCN(S(=O)(=O)N(C)C)CC1 36809,N1(C(C(CC)N(C)C)=O)CC=C(CCNC(C2CN3CCN2CC3C)=O)CC1 36810,c1(CC(=O)NC2CCCCCC2NC(=O)CC(F)(F)F)cccc2c1OCCC2 36811,C1(C(=O)NC(Cn2cc(C3(CC)CCOC3)nn2)C)CCC(C)(C)CC1 36812,C1(CN)CCN(C(=O)Cn2cc(CN3CCCCC3)nn2)C1 36813,CC(C)CC(C)CC(=O)N1CCC1CNC(=O)CCc1nncn1C 36814,N1(C(c2c(C)nc(CC)s2)=O)CC2(CCCCN(C(C3CN(C)C3)=O)C2)C1 36815,C1(C)(NC(c2c(C)n[nH]c2)=O)CCCN(C(=O)C(C)Oc2cccc(C#N)c2)C1 36816,c1(N(C)CCOCC(C)(C)C(C)(F)F)ccc(S(=O)(=O)NC2CC2)cn1 36817,N1(CC(N2CC(c3cn(CCS(C)(=O)=O)nn3)(N(C)CC)C2)=O)CCOCC1=O 36818,c1(CC)cc(Cl)ccc1NC(c1nnnn1C1CCOCC1)CC1COC1 36819,c1(-c2nc(C)c(C(=O)Nc3cc(F)c(Cl)cc3F)cc2)ccc2c(C)[nH]nc2c1 36820,c1(OC)cc(SC)ccc1CNC(Cc1sccc1Br)C(=O)O 36821,C1(CNC(C=C(C)C)=O)CCC(CNC(=O)Cc2ccn(C)c2)CC1 36822,C1(NN(C(=O)CCCn2ccnc2)C(=O)Cc2cn(C3CC3)nn2)C=CCCCC1 36823,C1(NC(CSCCCC)=O)CC(OC)CN(C(c2cc(C)nc(C)c2)=O)C1 36824,c1(C(N2CCCC(F)(CNC(C3(Cl)C(C)(C)C3)=O)C2)=O)n[nH]c2cc(Cl)ccc12 36825,N1(C(C(c2ccc(CO)cc2)C)=O)CC2CCCN(C(=O)CCCN=[N+]=[N-])C2C1 36826,C1(NC(c2cccc(C)n2)=O)CC2CC1N(C(=O)C(F)(F)CCn1ccnn1)C2 36827,C(=O)(C(C)C(F)F)NCCNC(=O)NC1(C(C)=O)CCC1.c12ccc(s1)C(=O)NC2 36828,C1(C(=O)NCC(=O)NCC#C)CCC(CNC(c2csc(=N)[nH]2)=O)O1 36829,C(=O)(C1CCCc2ncccc21)N1C2CC(CN(C(C(CC)OC)=O)C2)C1 36830,c1(OCC)ncc(NC(=O)C(C2CCCN(C(=O)C(C)C(C)C)C2)(C)C)cn1 36831,CC(C)CC(F)(F)C(=O)NC1CN(C(c2c(Cl)nn(C)c2Cl)=O)CC2(CC2)C1 36832,C(=O)(CC(C)CC(=O)N(CCC(C)NC(c1ncc2ccccn12)=O)C)OC 36833,N1(C(C(C2(OC)CCCC2)=O)C)CCCC(Nc2ccn(O)c(=O)c2)C1C 36834,N1(C(c2cncs2)=O)CCCC(F)(C(N2CCCCC2CCCO)=O)C1 36835,c1(C(N2CCC(N(C(c3c[nH]nc3SC)=O)CC)C2)=O)cn2ccc(C)cc2n1 36836,C12CC(C13CCC3)CN2.C1(C(=O)NC)CC(CNC(=O)OC(C)(C)C)C1 36837,C1(C(=O)NC(c2nccs2)C)CCCC12CCN(C(c1ccc[nH]1)=O)C2 36838,c1(C(N2CC(C)C(CNC(c3cn[nH]c3)=O)C2)=O)nc(Br)c2ccccn12 36839,N1(C(CCCc2onc(CC)n2)=O)CCN(C(=O)C(O)CCSC)C(CC)C1 36840,Cc1ccc(C(=O)N(C2CCCC2)CCNC(=O)C(C)(C)C(N)=O)c(C)c1Br 36841,c1(C(c2ccc(C)[nH]2)=O)ccc(CCOCC2CC2)c(F)c1.C1CO1.C1CO1.OC 36842,C(=O)(C(F)CC1CN(C(=O)CSc2ccccc2)C1)NC(C1CCCO1)C 36843,C12(CNC(C3=NOC(C)C3)=O)COCCN1C(=O)CN(C(=O)CSCCC#N)C2 36844,c1(C(N2CC(O)(CN(C)C(c3cccn3C)=O)C2)=O)cccc(F)c1F 36845,CC1CN(C(=O)C(c2ccccc2)=O)CCC1NC(c1ccnc(C2CC2)n1)=O 36846,N1(C(C(c2ccnn2C)C)=O)CCC=CC1C(=O)NOCC1CCCO1 36847,C1(NC(=O)CCc2ccccc2Cl)CC2CC1CN(C(C1CC(F)C1)=O)C2 36848,c1(NC(C2(NC(C(C)OCC=C)=O)CCSC2)=O)c(C)ccn(C)c1=O 36849,c1(C(=O)NC2CCCC(F)C2)cc2oc(Br)cc2s1 36850,CCC(C)CC(=O)N1CCC(O)(CN(C)C(C2CC(OC)C2)=O)C1 36851,c1(C(N2C(C(=O)Nc3ccn(C)n3)CC(F)C2=O)=O)cc(Br)ccc1C(F)(F)F 36852,c1(CCCC(=O)NCC(CC=C)NC(C2(COC(C)C)CC2)=O)ccc(O)cc1 36853,c1(C(=O)OC)cc2sccc2s1.C=C1CC2N(C1)CC1N(CC(F)C1)C2=O 36854,N1(C(C(CC)N(CCO)CC)=O)CC2(CC(C(=O)NOC3CCCCC3)CO2)C1 36855,S(=O)(=O)(c1cnc(N(C)CC2CCCC2O)c(Cl)c1)NCCc1c(C)ncs1 36856,CC1(C)CN(c2nnc(O)s2)CC1NC(c1ccc(F)cc1N)=O 36857,C(C(=O)NC(C)(CNC(=O)C=Cc1cn[nH]c1)CO)(C(C)(C)C)SC 36858,c1(CC)ncc(C(=O)NCC(C)CN(C(=O)C(C(C)C)N(C)C)C)cn1 36859,C12(C(N(C)CC3CC(O)C3)=O)C(NC(C3CC4C=CC3O4)=O)C3CC1C2C3 36860,c1(C(=O)NC(CNC(c2c(C)nsc2)=O)(C)C)cccc(OC(F)F)c1 36861,C1(CNC(Cc2cc(OC)ncc2)=O)CCN(C(C2CC=C(C)CC2)=O)C12CC2 36862,C12(CC)CCC(C(=O)NC3CCC(NC(C4(C)CC(F)C4)=O)C3)(CC1)CO2 36863,N(C(=NCC1CC1)N1Cc2ccccc2C2(CC2)C1)CC1CCCS(=O)(=O)C1 36864,N1(C(c2c(N)ncc(C)c2)=O)CC2CC3CC2C1C3NC(c1csc(C)c1C)=O 36865,c1(C(C(=O)NCCCC(C)NC(CCCCC)=O)(F)F)ccccc1C#N 36866,CC1CN(C(=O)C=CC2CCCN2C)CC1(C)C(=O)Nc1ccc(F)c(CO)c1 36867,c1(N(C)CC2CCCN(C(C34CC(C)(CO3)C4)=O)C2)ncc(C#N)cc1F 36868,N1(C(C2C(OC)CN(C(C(CCOC)C)=O)C2)=O)CC2(CCC2(C)C)C1 36869,C(C(C)(C)C#CC(=O)NCC(O)CC(F)(F)F)NC(CC1CCCC(CC)C1)=O 36870,C1(C(N(CCOC)CCO)=O)CCN(C(C2(CO)CCCCO2)=O)CC1(C)C 36871,C1(NC(C(CNC(C2(CC#C)CCCO2)=O)C)=O)CCC(C#N)CC1 36872,Cc1c[nH]nc1C(=O)N(CCC(C)NC(=O)C(Cc1ccccc1)N(C)C)C 36873,C1(OCC)CN(C(c2nccc(C)n2)=O)CC1CNC(c1ccc(CF)cc1)=O 36874,C(CCCC(=O)N1CCC(NC(=O)CSc2ccc(F)cc2)C(C)C1)(OC)OC 36875,N1(C(C(CC)N(C)C)=O)CCSCC1CNC(=O)C(O)c1ccco1 36876,C(=O)(C1CCC(=O)c2ccccc21)N1CCCC(NC(CNC(CC)=O)=O)C1 36877,c1(C(=O)NC2CN(C(C(C)C)=O)CC23CCC3)nn(C)c2ccccc12 36878,c1(C(=O)NCC2(C)OCCN(C(C3CN(C(C)=O)C3)=O)C2)cc2ncccc2[nH]1 36879,c1(CNC(C2(CCC)CCC2)=O)cc(C(=O)NCCCCCF)co1 36880,c1(C(CNC(c2cnoc2C(C)C)=O)NC(Cc2c(C)nsc2)=O)cccc(Cl)c1 36881,C1(OC)CC(NC(c2cc(C)nc(O)c2)=O)CN(C(=O)C(C)Cc2cnc[nH]2)C1 36882,C(=O)(CC(O)C(C)C)NC1C(NC(C(CC#C)C)=O)CCCC1 36883,N1(C(C2(SC)CC2)=O)CC(CCC(=O)NC2(CC(C)C)CC2)C1 36884,N1(C(c2ccn(CC)n2)=O)C2CCC(C2)C1CNC(c1cc(C)c(C)o1)=O 36885,C(=O)(CC(F)(F)F)NC1CC1.C12(NC(C3CCC(C(F)(F)F)C3)=O)CN(C1)C2=O 36886,c1(C(N2CC(C)C(NC(c3ccc(N(C)C)nc3)=O)C2)=O)ccc2cncn2c1 36887,Cc1c(N)cc(C(=O)NCC(C)NC(=O)C(c2cccc(Cl)c2)O)cc1[N+](=O)[O-] 36888,c1(C(N2C(CNC(c3n(CC)ncc3)=O)CC2)=O)cc(C2CC2)nc2ccnn12 36889,C1(N(C)C)CN(C(C23CC2CCN3C(C2CC(N(C)C)C2)=O)=O)CC1(C)C 36890,N1(C(C(CNC(C2C=C(C)CS2)=O)OC)=O)CCOC(C)(C)C1C 36891,c1(CNC(C2(CC)CC2)=O)ncoc1CCNC(C1CC(C)(C)O1)=O 36892,Cc1cc(O)ccc1C(N1CC=CC(NC(=O)Cn2cccnc2=O)C1)=O 36893,c1(C(=O)NC2C3(CC(NC(c4c(C)cc(Br)o4)=O)C3)C2)cc[nH]c2nccc1-2 36894,C(=O)(CCC(=O)OCc1csnc1C1CC1)OCC 36895,c1(CC(N2CCC(C(C)NC(=O)C(N)=O)C2)=O)cccc2ncccc12 36896,C(=O)(C(C)(C)CCCNC(=O)C(c1cnn(C)c1)C)N1C(CC)CCOCC1 36897,C(C(C)(Cn1cccn1)NC(C1(C(C)C)CC1CNc1csnc1C)=O)OC 36898,c1(C(N(CC(CNC(c2c(COC)ncs2)=O)C)C)=O)cc2oc(C)cc2[nH]1 36899,c1(CC(=O)NC2(C)CCOC2)cccc(OCc2ccccc2O)c1 36900,CC1CCN(C(=O)C(c2ccns2)NC(=O)NCCC(=O)O)CC(C)O1 36901,CCCC(C)(C)C(=O)NCC1CC(C(N2CC(=O)NC(C(=O)OC)C2)=O)C1 36902,N1(C(c2nncc(OC)c2)=O)CC(F)(F)CC1(C)CNC(c1ccc(Cl)cn1)=O 36903,CC1(c2ccc(CN3CC(n4cc(C5CC56CC6)nn4)C3)cc2)NC(=O)NC1=O 36904,c1(C(C(=O)NCC2CCOC2)N(C)Cc2cnc(CCC)s2)ccc(C)cc1Cl 36905,C1(C)(CC)C=C(C(=O)N2CCOC(CC(=O)NCCOCC(C)(C)O)C2)C1 36906,C(=O)(C(CO)C(C)(C)C)NC(CCC#C)C(=O)NC(c1ncc(C)cn1)C 36907,C(=O)(C1CCc2c[nH]nc21)N(C(c1cn(CCC(=O)NC)nn1)C)C 36908,C1(NC(c2c(C)cn(C(C)C)c2)=O)CC(F)CN(C(c2nn(C)c(Cl)c2Cl)=O)C1 36909,C1(=Cc2cn(C3CCC(C(N(CC)CC4CC4)=O)C3)nn2)CCCCC1(C)C 36910,C1(O)(C(=O)OC)CC(NCCSCCc2ccccc2)C1 36911,C1(O)(CN(C(C=C(C)C(F)F)=O)C)CCN(C(=O)CC2(O)CCC2)CC1 36912,CC(=O)C(C)(C)CC(=O)N1CC=CC(C(=O)NCC=CCCOC)C1 36913,CCC(C)CCN=c1[nH]c(=NCC2(CO)CC3CCC2CC3)c2ncccc2[nH]1 36914,c1(SCC(N2CC(NC(COCCC#C)=O)C2)=O)cc(C)ccc1C 36915,c12cccc3c1CCN(CC3)C2.C1(OC(C)=O)CCSCC1 36916,c1(C(=O)NC2CC(CNC(C3CCC(CC)C3)=O)C2)ccc(OC2CCC2)nc1 36917,C(=O)(C1=COCCC1)NC(c1ccccc1OC)CNC(CS(CC)=O)=O 36918,C1(C(=O)NC(C2C(C(=O)OC)C2)C)CN(C(C2COCCC2C)=O)CC1F 36919,Cc1cc(C2(C(=O)NC3CCCN(C(C4(O)CCCCC4)=O)C3)CC2)cc(C)c1 36920,Cc1ccnc(NCCCCNC(=O)C(C)NC(c2cccs2)=O)n1 36921,c1(C(=O)NCC(C2(O)CN(C(CC=CC)=O)C2)(C)C)cnc(N(C)C)nc1 36922,N1(C(CSCCC=C)=O)CCCC(O)(CNC(=O)C(C(C)C)NS(C)(=O)=O)C1 36923,N1(C(CCCCC(N)=O)=O)CC(NC(c2cccnc2)=O)CC12CCCOC2 36924,C(C(C)CC(=O)NCCC(O)CNC(=O)C1=CCOC1)OC 36925,c1(C(=O)NC(CNC(C2(OCC)CCC2)=O)C2CC2)scc(C)c1C 36926,CCCCC(O)C(=O)N1CC=CC1CNC(C1(CC)CCCCCC1)=O 36927,C=C(C)c1cncc(C(c2nnnn2CC2CCCO2)NCC2(C#N)CCCC2)c1 36928,C(=O)(C#CC1(C)CCCO1)N(CCC(=O)NCC(CC)C(C)C)C(C)C 36929,c1(C(=O)NC2CC(C)(CNC(C3N(C)C(=O)CC3)=O)C2)cn(C)c(=O)nc1O 36930,c12cc(OC)c(OC(F)F)c(c1)NC2.C1C(C)(C)C(=O)N1.S(C)(=O)(=O)NC 36931,C1(O)(CC)CCN(C(=O)C=CC(C)NC(C2CCCC2O)=O)C1 36932,N1(C(c2ccn(CCCC)n2)=O)CCC2(NC(=O)C=CC3CC3)CCCCC12 36933,c1(OC)ccc(F)c(C(=O)NCC(C2CCC2)NC(C23CC(OC)C2C3)=O)c1 36934,C1(CNC(c2nnc(C)s2)=O)CCC2(CN(C(=O)C(c3cccc(O)c3)C)C2)O1 36935,c1(C(C)NCC(C(F)(F)F)N2CCN(c3nnc(C#N)s3)CC2)ccc(Cl)cc1Cl 36936,C=CCC(CC=C)C(=O)N1CCC(C(=O)N(CCCCC)C)(CC)C1 36937,C1(NC(C(C)(C)OC)=O)CCC(C)C(C)C1 36938,c1(C(=O)NCC2(C(C)(C)C)CCN(C(c3onc(C)n3)=O)C2)cnc2c[nH]nc2c1 36939,N1(C(C=CC=CCC)=O)CC(NC(c2nccnc2C)=O)CC1CO 36940,Cc1c(C(=O)NCC2CC(C)N(C(c3coc(C(F)F)n3)=O)C2)sc(Cl)c1Cl 36941,n1(CCC(=O)NCCCCCN(C(=O)CC2CC23CC3)C)ccc(O)nc1=O 36942,c1(C(=O)NCC2N(C(CC=CC=C)=O)CCC2)cncc(F)c1C 36943,c1(C(N(CC(CC)NC(c2cc(Cl)ns2)=O)C)=O)ccc(OC)cc1 36944,CCCC(C)CCCC(=O)NCCC1CCN(C(=O)CCc2cccc(O)c2)C1 36945,C1(NC(c2c(C)nco2)=O)C(C)(C)C(NC(C2CCOCC23CCC3)=O)C1(C)C 36946,C1(NC(CCCCCC)=O)CC2CN(C(=O)C(=Cc3cccs3)C)CCN2C1=O 36947,CCC(CC)C(=O)NCC1CCCCC1O 36948,c1(-c2nc(C(C)Nc3cc(S(C)(=O)=O)co3)[nH]n2)ccc2ccccc2c1 36949,c1(CC(=O)NCCC2C(C)CCCC2)cc(Br)ccc1Cl 36950,Cc1cc(C(=O)NCCCCC(C)NC(=O)CCC2(C)CC2)cc(N)c1 36951,N1(C(C(C)(C)NC(C)=O)=O)CCC(CC(=O)NC(C)C#N)CC1 36952,c1(C(=O)NCCC2OCCN(C(c3nc(C)oc3C)=O)C2)ncc(Cl)cc1Cl 36953,c1(OC)c(CN2CC(F)(C(=O)Nc3cccc(C)c3F)C2)cc(Cl)cc1Cl 36954,N1(C(C2(CCC)CC2)=O)CCC2CCCN(C(c3cn(C)nc3C)=O)C2C1 36955,C1(NC(C=NOC)=O)C2CCN(C(=O)C(C)Cc3cccnc3)CC12 36956,C1(C(=O)NCC2N(C(c3nc(C)sc3)=O)CCCC2)CC2CC1C1C2C1(F)F 36957,C#CCC(CC(F)F)C(=O)N1CCC(NC(=O)Cc2sccc2C)C1C1CC1 36958,c1(SC)cc(C(=O)NCC2CN(C(=O)CCSC(F)(F)F)C3CC23)ccc1F 36959,c1(C(N2C(CNC(c3c(CC)ncs3)=O)C=CC2)=O)cc2n(n1)CCC2 36960,c1(OC)ccc(Br)c(C(N2CCCC(O)(CNC(=O)C(C)SC)C2)=O)c1 36961,c1(CNC(C(=O)NCC(CC)(C)CC)=O)c(C)cc(C(C)(C)C)cc1C 36962,C1(OC)CC(NC(C(N(C)C[Si](C)(C)C)c2nnn(C)n2)=O)C12CCC2 36963,C1(CC)(CC)NC(=O)N(NC(=O)NC(c2sc(N3CCOCC3)nc2C)=O)C1=O 36964,c1(C(=O)NC(C2CCOC2)CC)ccc(Cn2cc(C(N3CCCC3)C)nn2)o1 36965,c1(C(=O)NCC2C(CNC(=O)C3=NOCC3)C2)cnn2cnnc2c1 36966,c1(-n2c(-c3onc(-c4nccc(C)c4)n3)ccn2)cc(Cl)ccc1Cl 36967,C1(NC(C(F)=C(C)C)=O)CCCC(NC(c2cc(Cl)n(C)n2)=O)C1 36968,c1(C(N2CC3CC2CN3C(c2nc3ccccc3o2)=O)=O)cccn2ncnc12 36969,CC1CCC(C)(NC(C2CCCN2C(c2cc(CO)on2)=O)=O)C1 36970,C1(C2CCN(C(=O)CC(C)c3ccco3)C2)(NC(CC(CC)CC)=O)CC1 36971,c1(C(=O)NC2CC(OCC(N3CCC(C)(OC)C3)=O)C2)c(C)nn(C)c1N 36972,CC(C)C(CC(=O)N1CCC(O)CC1)NC(c1cocn1)=O 36973,CCC(CC(=O)NC(C(=O)NCC1(CC)CCCO1)C(C)OC)OC 36974,CC(C)C1=NOC(C(=O)NCC2CC3CCC2N3C(C23CC(C)(CO2)C3)=O)C1 36975,CCC(C)C(O)C(=O)N1CCCN(C(c2[nH]c(-c3cccnc3)nc2C)=O)CC1 36976,c1(C(=O)NCCC(C)NC(c2cnnn2C)=O)c(Cl)c(Cl)cc(Cl)c1Cl 36977,c1(CC)cc(=NCC2CCCCC2NC(=O)C(F)C2CCC2)[nH]cn1 36978,N1(C(c2ccc(C)n2C)=O)CCCCC2(CCN(C(c3cncc(N)n3)=O)C2)C1 36979,CC1(C)CCCCCC1NCC1CCCNC1 36980,Cc1ccc([N+](=O)[O-])cc1C(N1CCN(C(=O)Cc2ccc(F)cc2)CC1C)=O 36981,C1(CNC(C2CCC2Cc2ccccc2)=O)CCNC(=O)CC1 36982,CP(C)(=O)C(O)C(=O)N(C1CCCN(C(=O)C=CBr)C1)Cc1ccccc1 36983,CC1CN(C(C2CC2C(C)(F)F)=O)CC1(C)C(N1CCC1c1ccccc1)=O 36984,C(C(C(=O)NOCCCC(=O)OC)C(C)(C)C)NC(C(CCC)C#N)=O 36985,N1(C(c2cc(OC)no2)=O)CC(CNC(=O)C(N2CCSCC2)C)C2(CC2)C1 36986,C1(C(=O)NCCCCN2CCOC2=O)Cc2ccc(Br)cc2N1 36987,c1(N2CC3CN(C(Cc4cc(C)cc(C)c4)=O)CC3C2)nc2ccc(Cl)cc2s1 36988,C=C(C)C(CC(=O)NCC1CCC1NC(=O)Cc1ccc(F)cc1F)OOCC 36989,C1(NC(C2CCCC(F)C2)=O)CCN(C(c2cnccn2)=O)CC12CCC2 36990,C1(C(=O)NCC=CCCC)(C(C)C)CCN(C(=O)CCC=C(C)C)C1 36991,c1(C(N2CC(F)CC(NC(C3(C)N(C)CCC3)=O)C2)=O)cc2ccccn2n1 36992,C1(NC(CC=CC)=O)C(CNC(=O)COc2c(C)cccc2Cl)CCC12CCC2 36993,C1(CC(=O)NCCOC2CCN(C(C(C)(C)CC3CC3)=O)C2)CCCCC(=O)N1 36994,Cc1nn[nH]c1C(N1CCCC1CN(C(=O)CC1(CS(C)(=O)=O)CC1)C)=O 36995,c1(C(=O)NC2CS(=O)(=O)CC2NC(c2cnccc2Cl)=O)cn2cnnc2cn1 36996,C12(C(=O)NCc3cccc(NC(C(CC)(C)CO)=O)c3)CC3CC(C(=O)N1)C2C3 36997,c1(C(=O)Nc2ccc(-c3cnn[nH]3)cc2)c(C2(C(F)(F)F)CC2)ccc(Cl)c1F 36998,N1(C(C=CC2N(C(C(C)N3CCCC3)=O)CCC2)=O)CCOC(C)(C)C1 36999,c1(C(N(C)CC2CN(C(c3ccncn3)=O)C2)=O)cc(N)cc(O)n1 37000,C1(C(N(CCOCCNC(c2c(C(C)C)scc2)=O)C)=O)CC2CCCC2C1 37001,C(=O)(C(C)(C)C(C)(F)F)N1CCN(C(c2cc(C)nc(O)n2)=O)C(CO)C1 37002,N1(C(C(CC)CC2CCCCC2)=O)CC2CCCC(C1)N2C(=O)C1=NOCC1 37003,N1(C(c2c(C)cccc2)=O)C2CCC1(CNC(=O)CCCC(=O)NC(C)C)CC2 37004,c1(C(=O)NC2(CC(=O)N(CCOCCOC)C)CCCCC2)cnccc1C#N 37005,C1(OC2(C(=O)NOC(C)(C)CO)CN(C(C(C)NC=O)=O)C2)CCCC1O 37006,CC(C)CC(CNC(C1(C(F)(F)F)CC(F)(F)C1)=O)NC(c1ccccn1)=O 37007,C1(CC=CC)CCCN(C(=O)CC2CC2CNC(=O)C(C)SCC)C1 37008,C1(NC(c2c(OC)cnc(Br)c2)=O)CC2(CCN(C(c3ccn(C)c3)=O)CC2)C1 37009,N1(C(CC(COC)C)=O)CC(NC(c2cccc(C(C)(C)C)n2)=O)CC12CCC2 37010,c1(OC)cnn2c1CN(C(=O)Cc1ccc(-c3nn[nH]n3)cn1)CC2 37011,C1(C(=O)NC23CC(NC(c4c(C(C)C)c[nH]c4)=O)(C2)C3)CC(=O)NC(C)C1 37012,c1(CC(C)CN2CCCC2)cc(C(=O)O)cc(Cl)c1 37013,CC1CN(CCNC(=O)N(C(C2CCCCC2)CO)Cc2ccccc2)CC1 37014,Cc1cc(F)ncc1NC(=O)NCC(C1CC1)NC1CCOCC1 37015,N1(C(c2cc(COC)[nH]n2)=O)CC2CCC(C1)C2NC(c1cc(COC)cs1)=O 37016,c1(NC(N2CCC(CCC=C)C2)=O)c(I)cnc(Cl)c1F 37017,c1cc(NC(C2C(C(=O)OCC)C2(F)F)=O)on1.c1(C2(CNC=O)CC2)cc[nH]n1 37018,c1(C2(C(=O)NC3CN(C(c4cn(CC)nc4)=O)C(C)C3)CC2)ccc(F)cc1F 37019,N1(C(c2[nH]nnc2CN2CCCC2(C)CNC)=O)CC2(C=C(C(=O)OC)CO2)C1 37020,c1(-c2cc(C)cc(O)c2)ccn2cc(C(=O)NCC(F)F)nc2c1 37021,N1(C(CN(C)C)=O)CC2CCCN(C(c3ccc4oc(O)nc4n3)=O)C2C1 37022,Cc1ccc(OCC(=O)NC2CCC23CN(C(=O)CCC(C)(C)C)C3)c(C)c1 37023,N1(C(CC(C)OC)=O)CCn2c(CNC(=O)CSc3nnnn3C)nnc2C1 37024,Cc1cccc(C(=O)NC2CCC(C)(CNC(c3cc(C(F)(F)F)no3)=O)C2)n1 37025,c1(C(CC)CC)cc(C(=O)NC2CC(CNC(=O)CN3CSCC3=O)C2)on1 37026,C=CC(CC)CC(=O)NCCN(C(=O)C(C)(C)CC)Cc1cccc(Cl)c1 37027,c1(SC)cc(C(=O)NC2COCC2NC(C2CCC2(F)F)=O)ccc1F 37028,c1(C(=O)NCCC(C(C)C)NC(c2nc(C)sc2)=O)c[nH]c2cc(F)ccc12 37029,c1(C(=O)NC2CN(C(C3(C=C)CCCCC3)=O)CC(C)C2)cc2ncccc2o1 37030,C1(F)(c2c(C)cccc2)CCN(C(=NCCC(=O)N(C)C)NC2CC2)C1 37031,c1(C(=O)NC2CCC(NC(c3c(SCC)nccn3)=O)C2)cc(CC)ccc1O 37032,N1(C(C2CC23CC3)=O)CC2(C(=O)NCCOCCF)CCC1CC2 37033,c1(NC(=O)N(CCCO)CCCO)cccc(CC2NC(=O)NC2=O)c1 37034,c1(C(N2CC(CN(C)C(c3ccsc3Cl)=O)OCC2)=O)cn2cc[nH]c(=O)c2n1 37035,n1(C(C)C(N2CCOCC2)=O)cc(CN(C2CCOCC2)C)nn1 37036,C(=O)(C1=CCCOCC1)NCC1(C)CCC(NC(=O)Cn2ccccc2=O)CC1 37037,c1(C(=O)NCCOCCNC(=O)CCc2ccc[nH]2)ccc(Cl)cc1Cl 37038,Cn1ccc(C2(C(N3CC(O)(CNC(c4csc(C(F)F)c4)=O)C3)=O)CC2)n1 37039,c1(NC(C2CC3CCCCC3N2C(c2ccoc2)=O)=O)ccc2nc(O)[nH]c2c1 37040,N12CCC(C1)N(C)C2=O.c1ccccc1.N1(C(C)C)CCCC1C(F)(F)F 37041,N1(C(C2N(C(C)=O)CCC2)=O)CCCCCC(NC(c2csc3cncn23)=O)C1 37042,c1(C(N(C2CCN(C(C3CC(CC)(CC)C3)=O)C2)C)=O)cc(C)c(Cl)cc1OC 37043,N1(C(CC2CC(OC)C2)=O)CCCC(C)C1CCNC(=O)CCC1CC(F)(F)C1 37044,C(=O)(CCCN=[N+]=[N-])NC1C(NC(c2nn(C(CC)C)c(C)c2)=O)COCC1 37045,N1(C(c2c(CC)non2)=O)CCC(CN(C(=O)CC2(COC)CC2)C)CC1 37046,c1(N2CCC3(CC(OC)C3)C2)nc(=NCc2cc(C)cs2)[nH]c2c1CCC2 37047,N1(C(CC#N)=O)CC2CCCC(CNC(c3cc([N+](=O)[O-])cnc3O)=O)(C2)C1 37048,c1(NC(c2c(CC)ncs2)=O)ccc(C)c(C(F)(F)F)c1 37049,C1(NC(c2ccn(CC)n2)=O)CC2(C1)CC2NC(=O)CCc1ccc(C(F)F)o1 37050,c1(C(=O)NCCC2CC(NC(c3cn(CCO)nn3)=O)C2)cc(Cl)ccc1O 37051,C1(CC=C)(NC(C2CC3CC3C2)=O)CCCN(C(C2CC(=O)N(C3CC3)C2)=O)C1 37052,C1(NC(Cc2c(C)n[nH]c2C)=O)CCCN(C(=O)CNC=O)CC1F 37053,c1(CC(C(=O)NC2CCC(NC(CCSCCC)=O)CC2)C)ccc(F)c(F)c1 37054,Cc1cc(=O)n(CCNC(N2CC3C(CSc4ccccc4)(C3)C2)=O)c(O)n1 37055,C1(C)(C(c2n(CCSC)nnn2)NCCCOC(C)C)CCOCC1 37056,C(C(C)(C)CNC(c1nonc1N)=O)N(C)C(C1CCCC1O)=O 37057,C1(C(=O)NCC(C2CCCC2)C)C2CN(C(=O)CC#N)CC12 37058,C(=O)(C1=CC2C=CC(C1)C2)NC(CC(CC)C)C(=O)N1CCC12CC(CN(C)C)C2 37059,c1(OCC(=O)NC2CCN(C(C(C)C(C)(C)O)=O)C2)ccccc1[N+](=O)[O-] 37060,c1(SC)ccccc1C(=O)NC(C1CN(C(=O)Cc2cncc(O)c2)CCO1)C 37061,C(=O)(C1=CS(=O)CCC1)N1C(CNC(C=Cc2c(C)ccs2)=O)COCC1 37062,c1(OC)nccc(C)c1NC(=O)CC(O)CNC(=O)CCCN(C)C 37063,c1(N(CC(=O)NCC(CCCC)NC(=O)CC(F)(F)F)C)ncnc2[nH]cnc12 37064,Cc1ccc2oc(C(=O)NC3CN(C(=O)CCNC(=O)CO)C4CC34)cc2n1 37065,C(=O)(C(=O)C(C)(C)C)NCc1c(NC(CC2(OC)CCOCC2)=O)cccc1 37066,CC(C)CC(C)(CNC(C1(C(C)(F)F)CCC1)=O)NC(c1cnc2n1CCC2)=O 37067,C1(CN(C(C(CC)C)=O)CC)CCCCN1C(=O)COCC(C)(C)C 37068,c1(NC(N)=O)cc(Br)cnc1N1CCCC(Cc2ccc(Cl)cc2)C1 37069,CCC(C)(C(=O)NCC(Cc1ccccc1)NC(=O)C=Cc1nnn(C)n1)CO 37070,C(=O)(C(CC)C(C)O)NCC(=C)CCNC(c1cnc(CC(C)C)s1)=O 37071,c1(CC)ccc(Oc2ccc(CNC(=O)CCC3CCC(=O)NC3)cn2)cc1 37072,N1(C(C2CC(N(C)C(=O)NC(C34CCC(CO3)C4)C)C2)=O)CCC2CC12C(=O)OC 37073,N1(C(=O)OC(C)(C)C)C(C(=O)NCCc2ccc3nc[nH]c3c2)CC2CCCC12 37074,c1(OC(CC)C(=O)NC2CCCN(C(=O)C=CBr)C2)ccccc1F 37075,C1(NC(CCOCC)=O)CCC(CC(=O)NCCCC2CCCC2)C1 37076,C(=O)(C(O)P(C)(C)=O)N1CCC(N(C(CN(CCC#C)C)=O)C)C1 37077,C1(NC(C=CCCC)=O)CCS(=O)(=O)C12CN(C(C1CN(S(N)(=O)=O)C1)=O)C2 37078,c1(C(c2n(C(CC)C)nnn2)NCCCOC2CC2)nc(C)c(C)n1C 37079,c1(CCC(=O)NCC2C(NC(COCC)=O)CC2)nc(CC)no1 37080,C1(c2nnnn2Cc2cccs2)(NCC2CCCC2)CN2CCCC2C1 37081,CCC(C(=O)NC1CC1NC(=O)CCc1sccc1Br)c1ccccc1 37082,Cc1cnc(C(=O)NCC2C(C)CCN2C(c2cc(C3CC3)n(C)n2)=O)cc1C 37083,c1(OC)cc(F)ccc1C(=O)NC(CO)C(C)NC(C1(C)CC(C)=NO1)=O 37084,c1(C(=O)NC(CNC(C(CC)n2cncn2)=O)C)ccccc1C(C)=O 37085,N1(C(C(C)=C(C)C)=O)CC(C)OC2(CCN(c3ncc([N+](=O)[O-])cc3Br)C2)C1 37086,CCCCC(C(=O)NC1CCN(C(c2cncc(N)n2)=O)CC1O)N(C)C 37087,N1(C(CCC2C(OC)CCC2)=O)CC(CO)C2(C1)CN(c1nc(C3CC3)ns1)C2 37088,C1(CNC(C2CN(CC)C(=O)C2)=O)C(C)CCCN1C(=O)CCc1cncn1C 37089,c1(N2CC(OCCNC(C3CC4CCCC34)=O)C2)ncc(F)c(C2CCC2)n1.NC 37090,C1(NC(C2(CC#C)CC=CCC2)=O)CN(C(c2ccco2)=O)CC1S(C)(=O)=O 37091,c1(SCC(N2CC(C(C)NC(=O)CCOC3CCCCC3)C2)=O)n[nH]c(O)n1 37092,Cn1nc(NCC2CC3CC(OC(F)F)C3C2)c(C(F)F)c1Cl 37093,C(=O)(C1=NOC2(CCN(C(=O)Cc3ccsn3)C2)C1)N1CCN(C)C(=O)C1 37094,Cn1c(C(=O)NCCCNC(c2c(F)cccc2Br)=O)cc2c1CCOC2 37095,C(=O)(CCCC#CC)NC1CCN(C(C(C)OCCC#C)=O)C1 37096,Cc1ccnc(C(=O)NCC2CCN(C(=O)C=C(Cl)Cl)C(C)C2)c1F 37097,c1(CC)ccc(C(N2CCN(C(=O)C=C3CCC3)CC2CC(F)F)=O)c(O)c1 37098,c1(C(=O)NC2CCCC(NC(C3CC(CC4CC4)C3)=O)C2)cccc2ccsc12 37099,CC(CC(=O)N(C)Cc1ccc(F)c(C(F)(F)F)c1)C(C)(C)C 37100,N1(C(c2cc(C)c(Cl)s2)=O)CCCC(NC(=O)C(c2ccc(F)cc2)(C)O)CC1 37101,C1(CC(=O)NCc2csc(CNC(C3CCC(O)C3)=O)n2)CCCCC1O 37102,C1(CC=C)(NC(=O)CC(C)(C)C)CCCN(C(=O)CSc2ccc(C)c(C)c2)C1 37103,CN1C(=O)C2CN(c3ncc(S(=O)(=O)NC4CC4F)cc3Cl)CCN2C1=O 37104,Cn1c(Cl)nc2cc(C(=O)NC3C=CC(C)(C)CC3)ccc12 37105,CCC(C)(C)CC(=O)N1CCCC(C(=O)NC2(C3CCCO3)CC2)C1C 37106,C(C1=NOC2CN(C(=O)C=Cc3cncs3)CC12)NC(=O)COCC1CC1 37107,Cn1ncc2c(NCC34CCCC3C4(F)F)[nH]c(=NCC3CCC=CO3)nc12 37108,C#Cc1cn(C)nc1C(N1CC2CC1CN2C(=O)CCCCN1CCCC1)=O 37109,c1(C(N2CC(CNC(=O)C=Cc3cn[nH]c3)C(O)C2)=O)cc(F)cc(F)c1 37110,C(=O)(CCC(N)Cc1ccccc1)N(C(CCC)C)C 37111,C(=O)(CCC(=O)NCC1(O)CC(C(=O)NC(CC2CCCC2)CO)C1)NCC 37112,C1(NC(C2CCC3(CCC3)OC2)=O)CC2CCCC(C1)N2C(C1CSC1)=O 37113,C1(CC=C)(C(N2CC(C#N)(SC)C2)=O)CCCN1C(C1CC1C1CCC1)=O 37114,C(=O)(CC(CC)CC)NC(CCCC)CNC(c1ccnn1CC(F)F)=O 37115,c1(CC(=O)NCC(CO)NC(=O)CN2CC3CC3C2)cc(Cl)c2c(c1)OCCO2 37116,N1(C(=O)C(O)c2ccsc2)CC2CC2(NC(C23CC(F)(C2)C3)=O)C1 37117,c1(C(C(=O)N(c2cn(CC=C)nc2)CC)N(CCC)CC2CC2)ccc(F)cc1 37118,c1(N(CCC(C)=O)C)c(Br)ccc(F)c1Br 37119,c1(CC)nc(C)cc(=NCC(CC(C)C)NC(C2CCCCO2)=O)[nH]1 37120,C12(CC(N3C4(CN(CC(c5cnc[nH]5)=O)C4)CC3)=O)CC3CC(CC(C3)C1)C2 37121,c1(NC(c2c(C)nc(NC(c3cnc(Cl)cc3Cl)=O)s2)=O)ccc(C#N)cc1 37122,C1(C(N2CC(c3cc(C)on3)(O)C2)=O)C=CCNC1=O 37123,N1(C(C2C(CC)OCC2)=O)CCC(CNc2cnc(N(C)C)nc2)CC1C.C=O 37124,c1(N2CCC(NC(N(CC(C(=O)OC)C)C(C)C)=O)C2=O)c(F)cccc1F 37125,C1(C(N2C(CC(=O)NC3CCCC(O)C3O)CC2)=O)CC2C(C1)C2(F)F 37126,c1(C(CCCOC)C)nc(C2CCCN(C)C2)nn1-c1ccc(F)cc1 37127,n1(C(CC)C)ncc(C(=O)Nc2nccnc2CO)c1C 37128,C1(Cn2cc(C(CC)N(C)C)nn2)CC(CC2CCOC2=O)CN1C(=O)CSC 37129,C1(C(N2C(C(=O)N(C)Cc3cncnc3)(CC)CCC2)=O)C2CC3C(C2=O)C13 37130,CCC(O)C(=O)NC1CC(F)(CNC(c2n[nH]cc2-c2cnn(C)c2)=O)C1 37131,C=CCC(C)(C)C(=O)NCC1CCC(NC(C2CC3CC2C3)=O)CC1 37132,C12(C(=O)NC(CN(C(COCCC)=O)CC)C)CCC(C)(CC1)CC2 37133,C1(NC(c2c(C)onc2)=O)C2CC1N(C(C1(n3cccn3)CCC1)=O)C2 37134,c1(NC)ccccc1C(=O)NC1CC1NC(c1cnc(Br)s1)=O 37135,C#Cc1cncc(C(=O)NCC(C(C)(C)C)NC(=O)Cc2ccsc2Cl)c1 37136,N1(C(c2c(CC)nnc(C)c2)=O)CC2(COC(CNC(=O)C=NOC)C2)C1 37137,C(C)(CC)(CCNC(=O)C(C)Cc1cnn(C)c1)NC(C(C)=C(CC)C)=O 37138,N1(C(C)C(=O)NCC2CC2NC(=O)COC2CCCC2)C(=O)CCC1=O 37139,c1(OC)nc(C)ccc1C(N1CCC(C)C1CNC(C1(C)CC(=O)N(C)C1)=O)=O 37140,C1(C(=O)NCCC2OCC(C)(C)C2)CCCCN(C(C2CCOCC2(C)C)=O)C1 37141,C1(NC(c2cc(C(C)O)n[nH]2)=O)CCN(c2ccncc2C(N)=O)CCC1CO 37142,Cc1sncc1C(=O)N(C(C(=O)N(C(C)C)Cc1ccccc1)C1CC1)C 37143,C1(N(CC(C)C)C(c2c(CC)n[nH]c2)=O)CCN(C(c2cscc2C#N)=O)CC1 37144,c1(CC(N2CC(C(=O)NCC3CC(=C)C3)(COC)C2)=O)ccc(C)c(F)c1 37145,c1(C(N(CCC)CCNC(=O)C(O)C2CC2)=O)ccc(Br)c([N+](=O)[O-])c1 37146,C1(CC(N2CCCC(N(C(C3C(C)CCC3)=O)C)C2)=O)OCCCC1(C)C 37147,Cc1cc(NC(=O)NC2CCN(C(N3CCOC3=O)C)C2)cc(C)c1Cl 37148,c1(C(=O)NC2C(CNC(c3cc(C)nn3C(C)(C)C)=O)C2)ccnc2[nH]ncc12 37149,C1(C(=O)NCC2CCC(NC(c3n(CC)ccc3)=O)C2)CCc2nc(O)[nH]c2C1 37150,S(=O)(=O)(c1cc(Br)ccc1F)N1CC(C(N2CCCC3CCCCC23)=O)OCC1 37151,Cc1nnc(CCCNC(=O)Nc2csc(-c3ccc(F)cc3)n2)n1C 37152,CC1c2cc(Br)ccc2CCN1CCSc1ccccc1F 37153,c1(CC(=O)NCCCN(C(C(SC)SC)=O)C2CCCC2)ccc(C)c(F)c1F 37154,C(C)(C)(C(C)NC(=O)CC(C)c1cnn(C)c1)NC(C(C)C)=O 37155,C1(C(=O)NC2(CC(=O)N(CC(C)C#N)C)CC2)CCNC(=O)C1 37156,CN1C(=O)OCC1C(=O)NC1CN(C(c2cn(Cc3ccccc3)cn2)=O)C1 37157,C1(CNC(c2c(C)ccnc2C)=O)CN(C(=O)Cc2cnn(C)c2)C2CCN1C2 37158,C1(CC)CN(C)CCN1C(C1(NC(=O)C=Cc2cn(C)nn2)CCSC1)=O 37159,N1(C(=O)NCc2ccnc(COC)n2)CCOC2COCCC12 37160,CCC(O)C(=O)N1CCCC1C(=O)NC(C)Cc1cn[nH]c1 37161,CC1(C)CCC(C)(NC(=O)CCNC(c2ccc(F)cn2)=O)C1 37162,c1(NC)nc(C)ccc1C(=O)N(C)CC1CCCC(NC(=O)Cc2ccsc2)C1 37163,CCC(CN(C)C)CC(=O)NC1CN(C(c2cc(C)nc(O)n2)=O)CC12CC2 37164,C12(NC(c3c(COC)scc3)=O)CC1CN(C(=O)C(O)Cc1cnc[nH]1)C2 37165,CC1CN2CCN1C(C(=O)NC(C1CCN(C(=O)Cn3cccn3)C1)C)C2 37166,N1(Cc2cc(C)n(-c3cc(OC)c(C)cc3)c2C)CCCC(C2(O)CCC2)C1 37167,Cc1ccnc(O)c1CC(N1CC(NC(C2CCC2)=O)C(O)C1)=O 37168,CCC(C(=O)OC)C(=O)NC1CN(C(=O)Cc2ccc(OC)cn2)C1 37169,c1(CC(=O)NCCN(C(c2ccc(CSC)o2)=O)C2CC2)ccc(F)cc1C 37170,Cc1ccc2ncc(C(=O)NCC3CC3CNC(=O)Cc3cnnn3C)n2c1 37171,C(=O)(CN=c1cc[nH]cc1)NC(CC)CNC(=O)C1=C(C)OCC1 37172,N1(C(c2nn(C)c(Br)c2C)C(=O)NCCCSC)CCC2(CNC(=O)N2)C1 37173,N1(C(C(n2c(C)ncc2)C)=O)CCC(C(=O)NCCC2(C)CC2)C1C 37174,C(=O)(C1=C(SC)CCCC1)NCC(CC)NC(c1ccc(Br)o1)=O 37175,N1(C(C(c2ccc(N(C)C)cc2)C)=O)CC(NC(=O)CC2CSC2)CC12CCC2 37176,CC1(C)CN(C(C2(C#N)CCCOC2)=O)CCC1NC(=O)CC(C)(O)C1CC1 37177,C#Cc1ccccc1CC(=O)N(C)CCNC(c1cc(C2CC2)on1)=O 37178,C1(NC(CCSCC)=O)CC2(CCN(C(c3cnn(C(C)C)c3Cl)=O)C2)C1 37179,c1(NCC(C)CNC(C2CCCC(C)(C)CC2)=O)cccc(F)c1[N+](=O)[O-] 37180,c1(N2CCC(CCCC)C2)nc2cccnc2c(=NC2CCCC2N(C)C)[nH]1 37181,N1(C(c2occ(C)c2C)=O)CCCC12CCN(C(=O)CC1CSC1)CC2 37182,C1(C(=O)NCCOCC(N)=O)(CC)CCN(C(=O)C(C)=C2CC2)C1 37183,c1(OC2(C)CN(C(C3CCC(C(N)=O)C3)=O)C2)cc(C(=O)NC)ccn1 37184,N#Cc1ccc(C(=O)NCC(CC2CC2)C(=O)NCCc2cncs2)o1 37185,C12(C(N(C(CC)CC)C)=O)CC(NC(=O)CN3CCCC3)(C1)C2 37186,N1(Cc2c(Br)ccc(C)n2)CC2C(C1C(N1CC3C(CO)C3C1)=O)C2(C)C 37187,C1(C(=O)NCC(C)(C)NC(=O)C=Cc2ccco2)CCC([N+](=O)[O-])CC1 37188,c1(C(=O)NCC2C=CC(NC(Cc3cc(C)on3)=O)C2)c(Br)nc2n1CCC2 37189,c1(C(N)=O)cc(NC(=O)C(=O)NC2CC2c2c(F)cccc2F)ccc1F 37190,c1(N2CCC(CC(C)C)CC2)nc(=NCCN(C)C(C)C)[nH]c2c1ncn2C(C)C 37191,C(c1ccc(C)cc1)=CCC(N1C(SC)C(NC(CNS(CC)(=O)=O)=O)CC1)=O 37192,c1(CNC(NCc2cc(C)on2)=NCc2cnn(CCF)c2)cc2occc2[nH]1 37193,c12cc(O)nc(n1)C(C)OC2=O.CCCC1C(=O)N(C2CC2)CCN1.OCC 37194,c1(CC)cnccc1C(=O)N(CC(O)CNC(c1nccnc1C(F)(F)F)=O)C 37195,c1(C(C)C(=O)N(C)C(c2ccc(Cl)cc2)C2CCCC2)ccc2c(c1)OCO2 37196,C1(C(=O)NC(Cn2cc(C(CC)(C)O)nn2)C)CC(C(=O)OC(C)(C)C)=NO1 37197,C1(NC(c2ccccc2)=O)CCC2CN(C(c3ccc(CCF)cc3)=O)CC2C1 37198,Cc1ncc(CC(N2CCC(NC(=O)C(C)NC=O)C(C)C2)=O)c(O)n1 37199,c1(C(N2CCC(C)(CNC(C3CC(=O)N(O)C3)=O)C2)=O)cc2nc(=O)ccn2[nH]1 37200,N(C1CCCc2cc(OC)ccc21)C(c1n(CC)nnn1)c1c[nH]nc1C 37201,Cn1cc(I)cc1C(N1CCCC2CC12)C(=O)NCc1ccco1 37202,C1(C(=O)NC(CCC)CCO)CCCCN(C(=O)CC2CC(OC)C2)C1 37203,C(=O)(C(C)(O)CC(F)(F)F)N1CC(C)C(n2cc(-c3ccc(CO)nc3)nn2)C1 37204,C(C)(N=c1nc(NCC(C)C(C)(C)C)c2c([nH]1)c(C)nn2C)c1c(C)nc(C)[nH]1 37205,C(=O)(CCC(C)(C)C)NCC1OCCC(NC(CCN2C(C)CCCC2)=O)C1 37206,c1(C(N2CC3C(CNC(Cc4c(C)noc4)=O)(C3)C2)=O)cnc2c(c1)CCCO2 37207,C1(OC)CC(NC(=O)CC(F)F)N(C(=O)CCCC2CN(C(=O)OC(C)(C)C)C2)C1 37208,CCC(CC(C)C)C(=O)N(CC(O)CNC(c1ccc(Br)c(Cl)c1)=O)C 37209,c1(C(C(=O)OCC2C(OC)CCC2)(C)C)ccc(C(F)(F)F)cn1 37210,C12(C(=O)NCC(=O)N(C)CC)CC1CCN2C(=O)CC1CC2(CCC2)C1 37211,c1(C(=O)NCC2C(NC(CC3(C)CCCO3)=O)CC2)nccc(Cl)c1F 37212,N(C1CCCc2n[nH]cc21)C(C1C2CCCCCC12)=O.CC1(C)C#CC(=O)NC1 37213,CCCCC(CCCC)C(=O)N1CC(NC(=O)C(C)(C)NC(=O)C(F)(F)F)C(C)C1 37214,C=CCN=c1nc(N(C2(c3ccccc3C)CC2)C)c2ccc(OC)cc2[nH]1 37215,Cc1c(C(=O)N(CCCNC(=O)C=CC(=O)N(C)C)C)c(C(F)F)nn1C 37216,N1(C(c2cn(C(C)C)nn2)=O)CCC(C)(C)C1CC(=O)NC(C(F)(F)F)C1CC1 37217,C1(NC(C(=O)NC(C2ON=C(C)C2)C2CC2)=O)CCC(C)(C)C(C)C1 37218,c1(C(=O)NC2C(NC(c3c(CC)nc(C)o3)=O)COC2)cc(C)nc(C)c1 37219,c1(NC)ncccc1C(N1CCC(F)(C(N2CCC(CN(C)C)C2)=O)C1)=O 37220,C#CC1CN(C(C2CC3(C2)CC(O)C3)=O)CCN1C(c1cc(C2CC2)on1)=O 37221,C1(NC(=O)CC2CCCCC2)CC1C1CCN(C(c2nnc(O)cc2O)=O)CC1 37222,C1(C(N(C2CCC(O)C2)C)=O)CCOC2(CCN(C(=O)OC(C)(C)C)CC2)C1 37223,CC1CN(C(C(=O)NCc2ccco2)c2cnsc2)CC(C2CC2)O1 37224,CCC(N=c1nc(N2CC3CC2CN3C)c2[nH]ccc2[nH]1)c1ncc(C)[nH]1 37225,N#Cc1ccc(CN2CCC(O)(C(=O)Nc3cc(Cl)ccc3I)C2)cn1 37226,N1(C(c2nnn(CC)c2C)=O)CC2CCC1C1CN(C(=O)C(Cl)=CCl)CC21 37227,c1(NC(CCC2CCC(NC(c3[nH]c(=N)sc3)=O)CC2)=O)ccc2c(c1)OCC2 37228,N1(C(CC2C(C)(C)C2(C)C)=O)CC=C(CC(=O)NC2C=CCCC2CO)CC1 37229,c1(CSC)cccnc1C(=O)N(C)CC1CN(C(=O)CC2COCC2O)CCO1 37230,C(=O)(C(C)(C)CCCC(=O)NC1CCCCC1CNC(=O)C#CC1CC1)OC 37231,C(=O)(C1=CCCCO1)N(C1CCCN(C(C(=CC2CCCC2)C)=O)C1)CC1CC1 37232,C1(C(=O)NC2(C)CC(NC(C3C(CCC)C3)=O)C2)CCC(O)(c2ccccc2)C1 37233,CC1(C)CC(O)(C(=O)NCC2CCCN(C(c3ccc(CO)s3)=O)C2)C1 37234,Cc1cccc(C)c1C(=O)NCC1CC(O)CN1C(=O)Cc1ccnc(O)c1 37235,c1(C(=O)NCC(CO)NC(c2scnc2C2CC2)=O)cccn2nncc12 37236,N1(C(=O)C=C2CCCC2)CCCCC(C2CN(C(=O)CC3CCOCC3)C2)C1 37237,C1(C)(CC)CCC(N=c2[nH]c3cccc(OC)c3o2)CC1 37238,N1(C(c2c(C(C)C)onc2)=O)CC2CCC2(CNC(C2CCS(=O)(=O)CC2)=O)C1 37239,N1(C(c2ccc(SC)cc2)=O)CC=C(CNC(=O)C(C2CCOCC2)O)CC1 37240,CCCCCC(=O)NCCC1(CNC(C)=O)CC1.C12CC(C1(C)C)NC(=O)C2 37241,CC(CNC(c1cc(CCO)on1)=O)C(F)C(=O)NC1CCC(O)C(O)C1 37242,C1(CNC(C(C2CC(F)(F)C2)OC)=O)C(C)CCCN1C(=O)C1=CCN(C)C1 37243,C1(C(N2CC(F)(CNC(C3C(C)CC3)=O)C2)=O)CC2C=CC1C21CC1 37244,C1(C(=O)NCCCCC(=C)C)(OC)CCS(=O)(=O)CC1 37245,C1(CC(C)(C)C)CN(C(c2scnc2C(F)F)=O)CC1NC(=O)C=CCF 37246,N1(CC)CC(C(=O)NCCCNC(=O)CCc2ncc(C)[nH]2)c2ccccc21 37247,C(=O)(CC1=CCCC1)NCC(C1CCOC1)NC(c1c(C)ncs1)=O 37248,C#Cc1ccc(Cl)c(C(N2CC(NC(=O)C(F)F)C(CC)C2)=O)c1 37249,N1(C(CC(C)(C)NC(C2C(C(C)=O)C2(C)C)=O)=O)CCCC2CC1C2(C)C 37250,CCCCCCCC(=O)N1CCC(C(=O)NOC(C)(C)C)C1C 37251,Oc1c(F)ccc(CN=c2cc(Cn3ccnc3)nc[nH]2)c1F 37252,Cn1nc2ccccc2c1C(N1CCCN(C(=O)Cn2cnnc2)C(CO)C1)=O 37253,N1(C(CC2N(C)CC=CC2)=O)CCC2CN(C(c3ncccc3Cl)=O)CC2CC1 37254,c1(C(CC(=O)NC(CCNC(c2c(OC)noc2C)=O)C)C)ccc(F)cc1F 37255,C1(NC(=O)NCC2OCCCN(C(=O)OC(C)(C)C)C2)CC2(CCOCC2)CO1 37256,c1(CNC2C(C(=O)OC)COCC2)nc2ccccc2n1CC(F)F 37257,C12CCC(C)(C)CN1C2=O.c1(C2(NC(CC(C)CF)=O)CC2)ccc(C#N)cc1 37258,CCCCC(C)C(=O)NCc1n[nH]cc1C(=O)Nc1cscc1CC 37259,c1(C(=O)OC)cc(C(=O)NC2CC(NC(=O)C(C(C)O)N(C)C)C2)c(F)cn1 37260,N1(C(C(=O)NCC)=O)CCC2CN(C(c3ncnc(OC)c3F)=O)CCC2C1 37261,C12(CNC(C3C(CC)OCC3)=O)CC(CO1)N(C(C1CCN(C)C(=O)C1)=O)C2 37262,Cc1nn(C)c2ncc(C(N3CCC4(NC(c5cccnn5)=O)CC4C3)=O)cc12 37263,N1(CC(N)=O)CCCC(N=c2[nH]c(=NCC3CCSC3)[nH]c3c2CSC3)C1 37264,C(=O)(CC(C)CCC(=O)NCC(CC(C)C)NC(=O)C=Cc1cnc(C)s1)OC 37265,C(=O)(CCCC(C)(F)F)NCCN(C(=O)CCOCC1CCCO1)C(C)C 37266,CC1(C)CC(NC(c2ccns2)=O)CN(C(=O)COCCO)C1 37267,C(c1cccc([N+](=O)[O-])c1)=CC(=O)NC(CN(C(=O)C(C)(C)C(F)(F)F)C)(C)C 37268,Cc1nc(CO)ncc1C(=O)NC(CNC(=O)CC1CC(F)(F)C1)C(C)C 37269,C12(C(=O)NC(COC)C(=O)OC)CC(C)(CN1C(=O)C(F)C(F)(F)F)C2 37270,c1(C(N2C(C)CC(CNC(c3cc(Cl)c(Cl)s3)=O)C2)=O)cc2ccccc2cn1 37271,N1(C(CC(CC)C)C)CCCOC(NC(C)(C)Cc2ccccc2)C1.C1C(=O)N1 37272,C1(CC(=O)NCC(CC(=O)OC)O)CN(C(c2ccccc2O)=O)CC12CC2 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37309,Cc1ccc(F)c(C(N2CCC(O)CC2C(=O)Nc2ccccc2)=O)c1Cl 37310,c1(C(=O)NC2CCCC2)occ2c1CCC2.Cc1cc(C(=O)N2CCC2)ccn1 37311,CC1CN(C(C2(CCCF)CC2)=O)CCC1C(=O)NCCC1CCC(C)(C)C1 37312,C1(CNC(=O)OC(C)(C)C)CN(C(=O)CC2CCCNC2=O)CCC12CCOC2 37313,C1(F)(C(=O)NC(C(=O)NC)C2CC2)CCCN(C(c2ccc(C3CC3)s2)=O)C1 37314,c1(C2(C(=O)NCCC3CN(C(C(C)NC(C)=O)=O)C3)CC2)ccccc1F 37315,C1(CNC(C(C)OCC(C)C)=O)C2CCCC1N(C(C1CCCS1)=O)C2 37316,C1(C(=O)NCCOCC(N)=O)CC(F)CCN1C(=O)CCC1CCOC1 37317,Cc1ccccc1-n1ccc(C(=O)Nc2ccc(C(=O)N(C)C)nc2)n1 37318,CCCCCCC(C)(CC)C(=O)NCCN(C(=O)C(F)C(CC)CC)CC 37319,N1(C(c2cc(OCC)n[nH]2)=O)CCC(C2(NC(=O)CN3CC4CC4C3)CC2)CC1 37320,c1(CCC)cnnc(C(=O)NC2CN(C(c3cc[nH]c3C3CC3)=O)CC2OC)c1 37321,c1(OC)cnncc1C(=O)NCC(O)CNC(C1(O)CCCCC1)=O 37322,C1(NC(=O)Cc2cscn2)CN(C(c2csc(O)n2)=O)C2(CCCCCC2)C1 37323,C1(NCCOCC=C)C(=O)NCC(CO)NC(=O)OC1C.C(C)(C)(C)SC 37324,C1(CNC(c2cc(CC)nn2C)=O)CCCC2(CN(C(=O)C3=CCSC3)C2)O1 37325,Cc1cccc(C(=O)NC(C2CCOC2)CNC(=O)CCCN2CCCC2)c1O 37326,[N-]=[N+]=NC1CCC(C(=O)NCC2CCCN(C(=O)CNS(=O)(=O)C3CC3)CC2)C1 37327,c1(C(=O)NC2CN(C(C(C(C)C)F)=O)CC2c2nccn2C)nc[n+]([O-])cc1Cl 37328,CCCCCC(=O)N1CCC(C(=O)N(CCCCN(C)C)C)C1C 37329,C1(CNC(=O)Cc2ccc(F)nc2)CC(F)(F)CN1C(C1C2CC3C(C2=O)C13)=O 37330,c1(SC)ccc(C(=O)NC2(CNC(=O)C#CC3CC3)CCCCC2)cc1 37331,CCCCCC(O)C(=O)NCC1=CCCN(C(=O)C(CC)C(=O)OC)C1 37332,c1(N(C)CC2CCN(CC)C2)nc(N(CCCCN(C)C)C)nc2ccsc12 37333,CCN=C(NCCc1ccsc1Br)NCC(c1ccoc1)O 37334,c1(C(=O)NCCN(C(=O)CC2(O)CCC2)CCOC)scc(C)c1C 37335,C(=O)(C1=CCCCO1)N1CCC(OCCNC(C2CC(Cl)(Cl)C2)=O)C1 37336,CC#CCCC(=O)NC1CCCC(NC(=O)CCOc2ccc(F)cc2)C1 37337,c1(C(=O)NC2(CC=C)CCN(C(=O)C(CCO)N(C)C)C2)oc2ccccc2c1C 37338,N1(C(CCCC#C)=O)C2CCCC1CC(CNC(c1ccccc1C)=O)C2 37339,c1(C(C(=O)N(C(CC)C2CC2)C)NC(=O)C(C2(C)CC2)SC)c(C)cccc1Br 37340,C1(N(C(=O)CC23COC(C2)C3)C)CCN(C(c2cn(C)nn2)=O)CC1 37341,c1(C(N2CCCN(C(C3(OC)CCSC3)=O)CC2)=O)cc2c(s1)C(C)(C)CCC2 37342,N1(C(C2=C(C)OCC2)=O)CC(NC(=O)C(C)CS(C)(=O)=O)C2(CCOCC2)C1 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37360,Cc1cc(=O)oc(C)c1C(=O)NC(C1CCCCC1)CNC(=O)C(C)(O)C(C)C 37361,c1(-c2ccc(NC(C34COC(C3)C4)=O)s2)cccc2ccccc12 37362,c1(C(=O)NCCN(C(C2(C(=O)OC)C=CCC2)=O)C)cc2c(cc1Cl)NC(=O)C2 37363,c1(CC)nc2ccccc2cc1C(=O)NC(CNC(=O)C(F)CC(C)C)C1CC1 37364,N1(C(C(CC=C)CC)=O)CCC2(CCC2NC(c2nncn2CC)=O)CC1 37365,Cc1cc(F)c(O)c(NC(C2CC2c2ccccc2F)=O)c1F 37366,N1(C(=O)CCc2ncccn2)CCN(C(=O)CC2CCCC2(F)F)CC1 37367,C12(C(=O)NC3CC(C)(CNC(C=CC)=O)C3)CCCCC(=O)N1CCC2 37368,N1(C(Cc2nc(COC)sc2)=O)CCCN(C(=O)C(C2CCOCC2)O)CC1C 37369,S(=O)(=O)(c1cncc(Br)c1)NC1CN(C(C2(C)CCCN2)=O)CC1F 37370,c1(C(=O)NC2C(CNC(CCC=C=C)=O)CCC2)ccc([N+](=O)[O-])c(N(C)C)c1 37371,Cc1ccc(C(=O)N(C)CCNC(C2CCOC2=O)=O)cc1OC(F)F 37372,C1(CC=C)CCCN1C(=O)CC(=O)OC(C)(C)C.CCC(=O)NC 37373,c1(NC(N(C2CC(OC(C)(C)C)C2C(F)(F)F)C)=O)cnccc1Br 37374,c1(C(N(CCN(C(C)C)C(C2CC23CC3)=O)C)=O)cccc2cc[nH]c12 37375,Cn1c(CC(=O)NCCOCCN)nnc1S 37376,C(=O)(C(CCC1CCN1C(=O)OC(C)(C)C)N(C)C)NC(C)CCc1cn[nH]c1 37377,N1(C(C2CC(n3cc(COCC)nn3)C2)=O)CC(CN(C)C)OC(C)(C)C1 37378,N1(C(C(F)=CC)=O)CCCOC(CNC(=O)CC2COC(C)(C)CO2)C1 37379,c1(C(=O)NCC(CO)NC(=O)CC2COCCO2)ccc(-c2nnc(S)o2)cc1 37380,C1(C(N2CCC(CN(C(COC(C)=O)=O)C)CC2)=O)CCC(C)=C(C)C1 37381,c1(C(=O)NCC(CNC(C2C(C)=CCS2)=O)(C)F)cc(N)c(O)c(F)c1 37382,c1(OC)ccc2ccccc2c1C(=O)Nc1csc(-c2cc(SC)ccc2O)n1 37383,C(CCCC(=O)NCC1(CC)CC(NC(=O)CCc2ccncc2)C1)OCC 37384,CC(C)CC(CNC(=O)CC1CCCCO1)NC(C1CC(O)CN1C(N)=O)=O 37385,C(CCCCCC(=O)NOCC1CC1)NC(c1c(C)nccc1)=O 37386,O=C1CC(C(N2CCC(OCCF)C2)=O)N(C(=O)C(=C2CCCCC2)F)C1 37387,N1(C(C(n2cc(CCCSC)nn2)C)=O)CC(C(N)=O)C(c2cnn(C)c2C)C1 37388,N1(C(c2ccc(C(C)C)cn2)=O)CC2(CCN(C(=O)CN3CCCCC3)C2)C1 37389,c1(CN(C2CC2)CC2(C)CCCC2)cncc(C(F)(F)F)c1 37390,C1(NC2CC(C)(C)CC(c3nnnn3C3CC3)C2)CCOC2(CCCCC2)C1 37391,c1(-c2cn(CCC(=O)NCC3(C)N=C(C)SC3)nn2)cc(C#N)ccc1C 37392,c1(C(C(N2C(C)C(CNC(=O)C(CO)N(C)C)CC2)=O)(F)F)cc(F)cc(F)c1 37393,Cc1cc(F)cc(Br)c1C(=O)NCC1(c2ccccc2)CCN(C)C1 37394,C(=O)(C(CCOC)OC)NCC(=O)NCCOCC(=O)NCC 37395,N1(C(=O)Cc2cccc(Cl)c2)CC2(CCC(NCc3cnccc3Cl)C2)C1 37396,N1(C(=O)CCN2CCCCCC2)CC2CN(C(c3cc4ccoc4s3)=O)CC2C1 37397,C12C3CC4CN(C1C4C3)N(C=O)C(=O)N2.CC1CCC(CN)O1.C(=O)C(F)(F)F 37398,c1(OC)ccc(CCNCC(O)C(C)c2ccccc2)c(F)c1F 37399,C(=O)(C1=CCCC1(C)C)NCCOC1CCN(C(CC2CCN(OC)CC2)=O)C1 37400,C1(C(=O)NCC(C)(C)NC(c2cc(OCC)n[nH]2)=O)C(O)C(=O)N(C)C1C 37401,C1(C)(C(=O)NC(C(C)NC(C2CCSCC2)=O)CO)Cc2ccccc2NC1=O 37402,c1(OC)ccc2c(c1)CC(C(N1CC3CS(=O)(=O)CC3(NC(C)=O)C1)=O)CO2 37403,c1(CC)ccc(F)c(C(=O)NCC2CCCC(NC(=O)CC3CCOCC3)C2)c1 37404,CC(C)CC(O)C(=O)N(C1CC(NC(=O)CCc2nc(C(C)(C)C)no2)C1)C 37405,N1(C(CCCCSC)=O)CCCC(C2CCN(C(=O)C3CC3)CC2)CCC1 37406,Cc1nc(C(N2CC(NC(c3ccnc(O)c3)=O)CC(F)C2)=O)c(C)n1C 37407,N1(C(CC)=O)CCOC(CN(C(c2csc(-c3ccccn3)n2)=O)CC)C1 37408,C1(C(=O)NCC2CC(NC(CC3(CC(=O)OC)CC3)=O)C2)NC(=O)OC1(C)C 37409,N1(C(Cc2cc(C)on2)=O)CCC(NC(=O)CN(C2CCSC2)C)C(C)(C)C1 37410,C1(CCOC)(NC2CCC3C(C(=O)O)C32)CCN(C(=O)OC(C)(C)C)CC1 37411,C1(CC(=O)OC(C)C(=O)NC(c2ccc(Br)cc2)C)CCCCCC1 37412,C1(NC(c2cncc(-c3ccc(Cl)cc3)c2)=O)CCC(O)(c2ccccc2)CC1 37413,N(C1CCc2cc(Br)ccc21)(C(c1ccc2c(c1)ncn2C)=O)CC 37414,CCCCCCCN=c1nc(N2CCC(C(N)=O)(N(C)C)C2)c2c([nH]1)COC2 37415,C12(NC(=O)Nc3cc(CN4CCOCC4)cc(F)c3)CCC(O)(CC1)CC2 37416,N1(C(CN(C(COC)=O)C)=O)CC=CC(NC(C2CC3CCC2C3)=O)C1 37417,Cc1cc(C(N2CCC(CCNC(=O)CCS(C)=O)C2)=O)c(C)s1 37418,N1(C(c2cc(C)cc(N)c2)=O)C2CCC1CC(CNC(c1cn(C)nc1Cl)=O)C2 37419,N(C(=NCCCCl)N1CCC2(CNC(=O)C2)C1)CC1C(C)(C)C1 37420,C(=O)(CC(C(F)(F)F)c1ccccc1)N1CCC(CNC(=O)CCCC2CC2)C1 37421,C1(OC)CN(C(c2cn(C)nc2Cl)=O)CC1NC(c1ccccc1O)=O 37422,C1(N(C)C(C2CC3(CCC3)C2)=O)CCC2CN(C(=O)CC3CCS(=O)(=O)C3)CC12 37423,CC1CN(C(=O)C(c2ccccc2F)O)CCN1C(=O)COc1ccon1 37424,Cc1ccc(C(C)NC(=O)C(=O)NCCC2COCC2(C)C)cc1C 37425,N1(C(C2CC(C(C3CCOCC3)C)OC2)=O)CCC(NC(=O)CC#N)C(C)(C)C1 37426,C12CC3CCC1CN(C3)C(=O)Cc1cn2nn1.n1(CC(=O)OC)ccc(OC)n1 37427,N1(C(C(N2CCSCC2)C)=O)CCCOC(CNC(=O)C=Cc2cccs2)C1 37428,Cc1sc(C(=O)NC2CCCC(NC(=O)CC(C)NC(N)=O)C2)cc1[N+](=O)[O-] 37429,c1(OC)c(C(=O)NCC2CCCN2C(c2ncccc2O)=O)c(C)nn1C 37430,c1(C(N2CC(CCNC(C3(OC)CC3)=O)(OC)C2)=O)cn2ccnc2s1 37431,Cc1cc(C(N2CC=C(CCNC(=O)CC(O)C3CC3)CC2)=O)c2n[nH]cc2c1 37432,C1(CCNC(C(C(=C)Cl)(C)C)=O)CCN(C(c2ccc(F)cc2O)=O)CC1(F)F 37433,C(CC(=O)NC1CN(C(c2cccnn2)=O)C(C)(C)C1)(C(C)C)OCC 37434,CCCCC(O)C(=O)N1CCCC(NCc2ccc(CC(=O)OC)cc2)CC1 37435,N1(C(C(c2ccc(C)o2)C)=O)CCC(C)N(C(=O)COc2cn[nH]c2)CC1 37436,C1(C(N(OC)C)=O)CCOCCN1C(=O)C(n1nccc1C)C 37437,C=CCC(CC)C(=O)N1CCC(C(=O)Nc2csc(Cl)c2)(CF)C1 37438,CCC(C)C=CC(=O)N(CC(=O)N(C1CCC1)CCOC)C1CCC1 37439,c1(NC(C)=O)c[nH]c(C)c1C(=O)N(C1CN(C(C2(C3CC(F)(F)C3)CC2)=O)C1)C 37440,Cc1ccc2[nH]cc(CC(=O)NC3CC(CNC(c4ccc[nH]4)=O)C3(C)C)c2c1 37441,c1(OCC)ccc2ccccc2c1NC(=O)C(=O)NC1CCc2nc(C)nn2C1 37442,CCCCC(C(=O)NCCCC(C)(C)C)NC(=O)C=CC(C)C 37443,N1(C(CSCc2cn(Cc3c(C(=O)O)cco3)nn2)=O)CC(F)(F)C(F)(F)C1 37444,C1(NC(=O)CCc2ccon2)COCC1NC(c1n[nH]cc1Cl)=O 37445,CC(C)C1=NOC(C)(C(N2CCC(C)(CNC(=O)C=C(C3CC3)C3CC3)C2)=O)C1 37446,N1(C(c2cncc(C)c2)=O)CC(NC(=O)Cn2ncn(C)c2=O)C(F)(F)C1 37447,c1(CCC(N2CCC(CO)(NC(C3CC(O)C3)=O)CC2)=O)cccc([N+](=O)[O-])c1 37448,C(=O)(CC(F)(F)C(F)F)NCC1C(NC(C(C)(C)C(F)F)=O)COC1 37449,C1(NC(C2CCN(C)C2=O)=O)CC(F)CN(C(=O)CN(C)Cc2ccccc2)C1 37450,N1(c2c(C(C)=O)cccn2)CCCC(C)(CNC(C2(C(F)F)CCCCO2)=O)C1 37451,C(C(C(=O)NCCC1CC(=O)N(C)C1)C(C)(C)C)NC(c1cn(CC)nc1)=O 37452,CN1CCN(C(C2(F)CCCN(C(c3cc(N)cc(F)c3)=O)C2)=O)C(C2CC2)C1 37453,c1(-c2occ(CC(=O)NC(C(C)NC(C3(CC#C)CC3)=O)C)n2)ccc(Cl)cc1 37454,C1(C(N(C2CCN(c3ncncc3C)C2)CCC)=O)CC(C)(C)CC(C)(C)C1 37455,C(=O)(CCCc1cncs1)NCC(CC)NC(=O)CSc1nc[nH]n1 37456,C1(C)(CNC(CC(C)O)=O)CN(C(=O)C(=O)C(C)(C)C)CCO1 37457,c1(C(=O)NCC2N(C(C(COC)C)=O)CC(O)C2O)cn2c(n1)COCC2 37458,C1(C(C)(C)C)CC(CNC(c2ccccc2)=O)CN1C(=O)CCN1CCCC1 37459,c1(-c2cc(C(N3CC(NC(C(CC)F)=O)C3)=O)on2)c(F)cccc1F 37460,Cc1nccc(=NCC2(CNC(=O)C(C3CCC(=O)N3)C)CC2)[nH]1 37461,N1(C(C2CC(N(C)CC)C2)=O)CC(C)(C(=O)NCCC(O)C(F)(F)F)CC1(C)C 37462,Cc1noc(C)c1CCC(=O)NCC(C)CNC(=O)C(C)(O)c1ccccc1 37463,Cc1sc(C(F)(F)F)nc1C(=O)N(CC(C)(C)NC(=O)CC1C=NN(C)C1=O)C 37464,c1(C(=O)NC2(C(=O)NC(c3ccnc(C)n3)C)CSC2)cc(O)nc(C)n1 37465,c1(CNC(C(c2sc(Cl)cc2Cl)N(CCC(=O)OC)C)=O)ccccc1Br 37466,CC(C(=O)N1CCC2(CC1)CN(C(C1CCCCO1)=O)C2)S(=O)c1ccccc1 37467,C(C(C(C)(C)C)NC(=O)C(O)C1CC1)NC(C=C(C)C(F)F)=O 37468,c1(C(CN(C(=O)NC(C2CC2(C)C)C)C)O)cccnc1 37469,CCS(=O)(=O)CC(=O)NC(C)(CNC(=O)C(c1c(C)nn(C)c1C)C)C1CC1 37470,CC1(CC(=O)NC2(CNC(c3cc4sccc4[nH]3)=O)CC2)CCS(=O)(=O)N1 37471,O=C(C1CCc2nccn21)NCC1CN(C(c2ncc3c(F)cccn23)=O)C1 37472,c1(OC)cc(N)c([N+](=O)[O-])cc1C(=O)OC(Cc1cnc[nH]1)C(N)=O 37473,c1(COCC(=O)NCc2cccc(CNC(=O)C3=CCC3)c2)cc(F)cc(F)c1 37474,c1(N2CCC(N(C(=O)Cc3cnsc3)CC)C2)ccc([N+](=O)[O-])cn1 37475,C(=O)(CCCCCS(N)(=O)=O)NC1CCCCN(C(c2c(Cl)cn(CC)n2)=O)C1 37476,c1(OC(C(CC)C)C)cc(C#N)ccc1NC(=O)OC(C)(C)C 37477,CCCC(C(=O)NCC1(O)CCCN(C(=O)C2=NOCC2)CC1)S(N)(=O)=O 37478,c1(C(N(C)CCNC(C2CC2C(=O)NCCO)=O)=O)cncc(-n2cccn2)c1 37479,c1(CCNC(c2n(C(C)C)nnn2)c2csc(-c3ccsc3)n2)ncccc1F 37480,c1(CC(=O)NCC2C(NC(C(C)OCCC=C)=O)CCC2)cn2ccccc2n1 37481,c1(CCC(=O)NC2C(NC(C)=O)CCCC2)nc2c(O)nc(=O)n(C)c2[nH]1 37482,c1(C(N2CC(NC(c3coc(Cl)n3)=O)C(O)C2)=O)nc2ccccc2o1 37483,N1(C(C(CC)(C)F)=O)CCC2(CC1)CN(C(=O)CC=CC(C)(C)C)C2C(C)C 37484,N1(C(CC(C)SC)=O)CCOCC(CNC(=O)C(C)Nc2nc(C)cs2)C1 37485,N1(C(c2cc(OC)n(C)n2)=O)CCC(O)C(N(C(=O)C=CCF)C)C1 37486,N1(C(C2CCC3(CC3)C2)=O)C2CCC1CC(NC(C13CC4CC1C3C4O)=O)C2 37487,c1(COC)nccc(=NC2CC(NC(c3cccn4ccnc34)=O)C2)[nH]1 37488,Cc1c(F)ccc(N)c1C(=O)NCC12CC(NC(=O)COC(F)(F)F)(C1)C(C)O2 37489,C=Cn1nccc1C(=O)NC1CC(C)(NC(C2CCCN(C(=O)OC)C2)=O)C1 37490,C(C(=O)N=S(C)(=O)c1cnn2c1CN(c1ncnc(C(C)(C)C)n1)CC2)=CC 37491,c1(C(=O)NC)cc(C)[nH]c(=NCC2CCC(NC(=O)C(C)(C)CC(F)(F)F)C2)n1 37492,N1(C(C(CC)OC)=O)CCCC(CNC(C2(OC)CC2)=O)CC1 37493,CN=S(C)(=O)c1ccc(C(=O)NCC2CCCCC2NC(c2cccs2)=O)cc1 37494,CC1CN(C(C2(F)CCN(C(=O)CNC=O)C2)=O)CC2(CCC2)O1 37495,Cc1cnc(F)cc1C(N1CC(NC(=O)Cc2conc2C)C(C)C1)=O 37496,N1(C(C(N2CC(C)C2)C)=O)CCC(C)(C)C(C(=O)NC2CC(C)(C)OC2=O)C1 37497,C1(NC(COCCCCC)=O)CC2C(NC(=O)C(C)OCC)C2C1.C1CCCC1 37498,CC1=NOC(C(=O)NCc2cn(CCNC(C34CC(C)C3C4)=O)nn2)C1 37499,c1(CC)c(NC(c2coc(C(C)NC(=O)CC(C)n3cccc3)n2)=O)cnn1C 37500,C1(NC(CC(C)(C)N(C)C(C2C=CCC2)=O)=O)CCCC(O)CC1 37501,N1(C(CC)=O)CC2CCC1CN2C(c1[nH]c(C(C)=O)cc1-c1ccccc1)=O 37502,N(C1CCCc2cc(F)ccc21)C(C1C(NC(C2C=CC(=O)N=N2)=O)C1)=O 37503,c1(CCC(=O)NC(C)(C)CNC(C2(N=[N+]=[N-])CC2)=O)cccc(F)c1 37504,C1(CNC(C(C)=C(C)C)=O)CCC(C)(C)CN1C(c1ccc(NC=O)cc1)=O 37505,N1(C(c2ccc(CNC(C3CC=CC3)=O)cc2)=O)CCC2CCCCC12 37506,c1(C(N2C(CNC(C(C)CSc3ccccc3)=O)CC2)=O)ccc(C(F)F)cn1 37507,C1(C(N2CCC(CC)C2C(=O)NCCCCCCO)=O)OCC2CCCC12 37508,CCC(CCOC)C(=O)N(CCCOCCN(C(=O)C(C)(C)n1cccn1)C)C 37509,CC1(C)CCCC(N2CCCC(Oc3ccc(C#N)cc3)C2)C1 37510,CCC(CC1CCCC1)C(=O)NC1CCN(C(C2CC(C)(C)CO2)=O)C1C 37511,C1(NC(=O)C(C2CC2)C2CC2)CCC2CCN(C(=O)C(O)c3ccsc3)C1C2 37512,n1(CC(=O)N(C)C(C2CCCCNC2)c2ccccc2)cc(C#N)cn1 37513,N1(C(Cc2c(C)nc[nH]2)=O)CC(NC(=O)Cc2cc[nH]c2)CC12CCCCCC2 37514,CCC(C)(CN)C(=O)NC1CCN(c2nnnn2Cc2cc(F)ccc2F)CC1 37515,C(=O)(C(CNC(c1cc(C#N)n(C)n1)=O)C(C)C)N1CCC(CSC)CC1 37516,C12(C(N3CC(C(C)NC(C(CC)(C)OC)=O)C3)=O)CCCC1C2(F)F 37517,CC1(C)CCCC(C(=O)NCCC2=CCN(C(c3ccc(C#N)[nH]3)=O)CC2)CC1 37518,c1(C(=O)NCC2(CCNC(C3CCCCO3)=O)CC2)cnc(O)c2ncccc12 37519,c1(C(N(CC(C)N(C(CC2CCC(C)O2)=O)C)C)=O)ncccc1Cl 37520,CCCC(O)C(=O)N1CCCC1C1CCCN(C(=O)COCc2ncc(C)o2)C1 37521,C(CS(=O)(=O)c1cccs1)NC(=NCC=C)NC(C)CNC(=O)OC(C)(C)C 37522,c1(C(N2C3CC(NC(C(CCC)OC)=O)C3CC2)=O)cccc2c1nnn2C 37523,N1(CCC)CCC(N(C)CC2(COC)CCC2)C1 37524,C(C(CCCC)NC(C12COC(CF)(C1)C2)=O)NC(CSCC=C)=O 37525,C=CCC(F)(F)C(=O)NC1CCCC(NC(=O)Cc2ccc(Cl)c(F)c2)CC1 37526,C(CC#CC(C)(C)C)NC(C(CNC(c1cc(C(N)=O)c[nH]1)=O)N(C)C)=O 37527,C1(C(=O)O)C(OCc2cn(C(C)C(=O)N(C)C)nn2)C2(C)CCC(C2)C1(C)C 37528,c1(C(N(C(C)C(=O)N(C)Cc2ccoc2)CCC)=O)cc(C(C)C)on1.C1CO1 37529,c1(NC(C2C(OC)CN(C(=O)C3=CCCCO3)C2)=O)c(C)cc(O)nc1C 37530,CC1(NC(=O)CONC(=O)C2CC(O)C2)CCCO1 37531,c1(C(=O)NC(CNC(C2CC(OC)C2)=O)C)ccccc1C1(C#N)CC1 37532,C=CC1CCN(C(C2(CNC(=O)C(F)F)CC(=C)C2)=O)C1 37533,N1(CC(=O)N(Cc2scc(CNC(CCC(=C)Cl)=O)n2)CC)Cc2ccccc2C1 37534,C1(NC(c2[nH]cc(C)c2)=O)CN(C(c2cncc(Br)c2C)=O)CC12CCC2 37535,C1(OC)CC(CNC(c2cc(C)nn2C2CC2)=O)N(C(c2cc(C)ccn2)=O)C1 37536,c1(OC)ccc(C(=O)NC2CC23CN(C(=O)OC(C)(C)C)C3)c(Cl)n1 37537,c1(C(=O)Nc2cccc(CNC(C(C)N(C)C)=O)c2)cc2c(cc1N)CCCC2 37538,c1(CC(=O)NCC2CCCN2C(C2CCC3(CC3)C2)=O)cn2cc(F)ccc2n1 37539,c1(CC(=O)NCCN(C(=O)C(C)CCN(C)C)CCOC)ccc(OC)cc1C 37540,C1(C(=O)NCC2OCCCN(C(C3CNC(=O)N3)=O)C2)Cc2cncn2C(=O)N1 37541,C#Cc1ccc(SCCCNC(N2CC3CC(O)C3C2)=O)cc1 37542,C(=O)(C(C)(CC)CC)NCC(C)(C)NC(C(F)=CC)=O 37543,C(=O)(C(F)C(F)(F)F)N(C(C)C)CCOc1ccccc1F 37544,Fc1cc(Br)c2[nH]c(=NCCn3cc(-c4ccc(Cl)cc4)cn3)ccc2c1 37545,CC1CN(C(c2cc[nH]c(=N)n2)=O)CCN1C(=O)C=Cc1ccncn1 37546,C12(F)CCC(C1)N2.c1(C(N(C)NC(C(C)OCC)=O)=O)ccc(C2(C)CC2)cc1 37547,c1(C(C(=O)NCC(C)N(C)C(C2(F)CCCCC2)=O)C)cncc(F)c1 37548,CC1OC2(CO)CC1(C(N1CCC(N(c3nnc(O)s3)CC3CC3)CC1)=O)C2 37549,N1(C(C(C)SCC)=O)CCCC(CNC(C2CCCN2S(C)(=O)=O)=O)C1 37550,c1(OC)ccc(CC(C)(C)C(=O)NCc2ccc(Cl)cc2Cl)cc1OC 37551,CC(C)CC(CNC(c1csc(F)c1)=O)C(=O)NCC(N1CCOCC1)C 37552,N1(C(C(C)NC(=O)OC)=O)CC2(CCCN(C(=O)CC3COCCN3C)C2)C1 37553,C(=O)(CS(=O)(=O)C1CCCC1)N(CCN(C(C(C)C1=CCCC1)=O)C)C 37554,Cc1cc(S(N)(=O)=O)oc1C(=O)NCCN(C(c1c(C)n[nH]c1C)=O)C1CC1 37555,N1(C(c2n(C)ncc2C#N)=O)CCC2(CC1)CCN(C(C1CC1CF)=O)C2 37556,c1(C(=O)NC2CN(C(C(C(=O)OCC)CC)=O)C2)cc(=O)n(C)c2ccccc12 37557,c1(CCC(N2CC(O)(CNC(c3ccc(F)nc3F)=O)C2)=O)c(Cl)cncc1Cl 37558,C1(C(=O)NCCC(C)NC(c2cnoc2C2CCOCC2)=O)CC(Cl)(Cl)C1 37559,Cc1cc(C(=O)NCC(C2CC2)NC(c2cnsc2)=O)cc(Cl)c1 37560,C1(CN(C(C=CCN(CC)CC)=O)C)CN(C(=O)Cc2cnc(C)s2)CC12CC2 37561,C(=O)(C1=CC2C=CC1C2)NC(C(=O)N(CC#C)CCOC)(C)CSC 37562,Cc1nccc(C(N2CCN(C(=O)CN(S(C)(=O)=O)C)C(C)C2)=O)c1Cl 37563,c1(OC)nccc(CNC(=O)CC2(NC(C3CC3(F)F)=O)CCCCC2)n1 37564,c1(COC(C2(COC)CCN(C(=O)OC(C)(C)C)C2)=O)ccc(F)cc1Cl 37565,CCC(C(=O)N1CC(C(N)=O)(CNC(=O)CC2(O)CCOC2)C1)C(C)O 37566,C1(C(=O)NCC2(CC)CCCC2)CN(C(C2(C(F)(F)F)CC2)=O)CC1(F)F 37567,c1(CC(=O)NCC(C2CCC2)NC(C(C)OCC=C)=O)ccc(Br)s1 37568,C1(CNC(C2N(CC#C)CCC2)=O)CN(C(C2CSC(C)=N2)=O)CCC12CCC2 37569,c1(CC(=O)NCC(CC=C)NC(c2n[nH]cc2Cl)=O)cnc2ccccc2c1 37570,c1(N2CCC(O)(COC)C2)cc(C)c(F)cc1[N+](=O)[O-] 37571,c1(CNC(NC(C)C)=NCCC2CC2C2CC2)ccc(C#N)cc1F 37572,Cc1nc(=N)[nH]c(C)c1C(=O)NCCC(C)NC(C1OC(C)CC1C)=O 37573,C1(C(N2C(C(C)(C)C(=O)NCCC3CCOC3)CCC2)=O)C2CCCCC12 37574,CC1=C(C(=O)NCC(C2(O)CCN(C(C3CCC3)=O)C2)C)CCC(C)(C)C1 37575,C(CN=c1[nH]c(=NC2CC3CCCCC23)c2ncccc2[nH]1)N1CCC(C)C1 37576,N1(C(C2(S(N)(=O)=O)CCC2)=O)CC2CCCC(C1)N2c1cnc(C(=O)OC)cn1 37577,c1(CC)cc(C)c(C(=O)NNC(=O)C2CCCN(Cc3ccccc3)C2)o1 37578,C=CC1(CC(N2CC(OC)C(NC(=O)C(C)C#N)C2)=O)CCOCC1 37579,c1(OCC)nccc(C(=O)NC2CCCCN(C(C3CC=C(C)CC3)=O)C2)c1F 37580,c1(CC)cc(OC)ccc1C(N1CCC(NC(=O)CN2CC(C)(C)C2)C1CC)=O 37581,C(=O)(CC(C)C(=O)c1ccccc1)N1CCC(C(CNC(COC)=O)(C)O)CC1 37582,c1(N(CC(C2CCC2)NC(=O)OC(C)(C)C)C(C2CC(F)C2)=O)ccc(Cl)cc1 37583,c1(C(=O)NCC2OCC(CNC(c3ccc(O)nc3)=O)C2)ccc2nn[nH]c2n1 37584,c1(CN(c2cccc(C#C)c2)CC)ccc2ccoc2c1.N12CCC(CC)CN1C2 37585,c1(OC)ccc(C(N2CC(N3CC(NC(c4cnsn4)=O)CC3=O)C2)=O)c(C)c1 37586,c1(CN2CCC(N(C(CC)C)C)CC2)ccc(Br)c(OC)c1 37587,N1(C(C=CCC)=O)CC2CS(=O)(=O)CC2(NC(c2cc3c(cn2)OCCO3)=O)C1 37588,O=C(CCN=c1[nH]c(=NCCF)[nH]c2c1COC2)N1CCOCC1 37589,C(=O)(C1CCC(N)c2ccccc21)N1C(COC(C)(C)C)CCCC1 37590,C1(C(N(CCNC(c2scc(C)c2C)=O)C)=O)CCC2(CCC2)C1 37591,N1(C(C=CCC)=O)CCN(C(=O)CC2C=NN(C)C2=O)CC1COC 37592,N1(CC(=O)Nc2ccc(-c3cncc(Br)c3)s2)CCC12CCN(CC1CC1)CC2 37593,N1(C(=O)C=Cc2cccnc2)CCC2CC2(C(N2CC(CO)(CO)C2)=O)CC1 37594,C1(N(C(=O)CC2(CO)CC2)C)CN(C(C2CCN(CC(C)C)C2)=O)CC12CC2 37595,CC1(C)CCC(C(=O)NCC2=CCCOC2)(NC(=O)C=CCN2CCC2)C1 37596,c1(-c2cc(CC(=O)NCC(C)CNC(c3nonc3N)=O)no2)cccc(F)c1 37597,N1(C(CNC(=O)NC)=O)CC2(CC(NC(=O)C(C)CCCOC)C2)C1 37598,c1(N2CCC(OCCNC(C3CC34CC4)=O)C2)nccc(-n2ccnc2)n1 37599,C(=O)(CS(=O)(=O)C(C)C)NCC1(NC(c2cc(C)cc(O)c2)=O)CCOC1 37600,CCCCC(O)C(=O)N1CCNC(C(=O)Nc2nc(F)ccc2Br)C1 37601,N1(C(Cc2ccc(C)nc2)=O)CC2CC(NC(C3CCCC3N(C)C)=O)CC2C1 37602,c1(NC(c2nncs2)C)[nH]c(=NCc2csc(Br)n2)nc2c1ncn2C 37603,N1(C(c2ccc(C(C)(C)C)nc2)C(=O)NC2CC2)CCC2(COC(=O)N2)C1 37604,C1(C)(C(c2nnnn2CSc2ccccc2)NC2C(C(C)C)C2)CCCC1 37605,N1(C(c2n(C=C)ncc2)=O)CCCC(NC(C2CC3CC3C2)=O)CC1 37606,C1(SC)CN(C(c2cnc(C(N)=O)s2)=O)CC1NC(=O)C=CC1CCC1 37607,c1(CC2CCCN(C(C(C)c3cc[nH]n3)=O)C2)ccc(F)c(F)c1 37608,c1(CC)cccc(F)c1C(=O)NCCC1CC(NC(=O)CC2(C)CCCC2)C1 37609,Cn1c(C(=O)Nc2csc(S(C)(=O)=O)c2)cc2c(=O)n3ccccc3nc12 37610,c1(NC(C(=O)NCC(CC(C)C)C)=O)ccccc1S(C)(=O)=O 37611,N1(C(c2ccc(SC)o2)=O)CCCC(C2CN(C(c3cc(O)cc(O)n3)=O)C2)C1 37612,c1(C(=O)Nc2c(C(=O)NCc3n(C)ccn3)n[nH]c2)ccc(I)c(O)c1 37613,C1(NC(C(C)OCC(C)C)=O)C2CCC1CN(C(=O)C(C)C(C)(F)F)C2 37614,C(CC(F)F)(C(=O)NOCCC(C)O)N(C(=O)CC(C)(C)C(F)F)C 37615,c1(C(=O)NC(c2cccc(OC(F)(F)F)c2)C2CC2)cccc2occ(Br)c12 37616,N1(C(N2C(C)(c3cn(C4CC(O)C4)nn3)CCC2)=O)CC(O)C2CCCCC2C1 37617,c1(C(=O)OCCCN=[N+]=[N-])cc(C(F)(F)F)ccc1-c1n[nH]cc1Cl.C1C(=O)N1 37618,c1(C(=O)NCC2CCCC2NC(C2CCOC2)=O)c[nH]c2ccccc12 37619,C1(C(=O)NC2CC(NC(c3ccc(C)s3)=O)C2)C2CC2C2CC12 37620,c1(OCCOC)ccc(C(N2CC(NC(=O)C(=O)c3ccco3)C3CC23)=O)cc1 37621,c1(C(=O)NC(CC(C)NC(c2n(C=C)ncc2)=O)C)cc(Cl)c(N)c(Cl)c1 37622,C(=O)(CCCN=[N+]=[N-])NCC(C)NC(=O)CSCc1ccncc1 37623,Cc1cc(F)c(C(=O)NC2(C3CCCN3C(=O)C(O)C(C)(C)C)CC2)cc1F 37624,n1(C(C)C)cc(CNc2ccc(CN3CCOC3=O)cc2)c(I)n1 37625,N1(C(c2ccc(SC)o2)C(=O)Nc2ccccc2)CCN(c2nccs2)CC1 37626,O=C1CC2(C1)CC(C(N1CCSCC1C(=O)NCC(CO)C1CC1)=O)C2 37627,N1(C(c2c(OCC(=C)C)cccc2)=O)CCN(C(=O)CCCCC2CC2)C2CC12 37628,n1(CC)ccnc1C(=O)NCC1CCCC1NC(=O)CCC=C(C)C 37629,c1(NC(=O)NCC(C)C)ccc(OCC(C)NC(c2cnn(C)c2F)=O)cc1 37630,N1(C(C(C(CC)C)O)=O)CCC2(CC1)CN(C(=O)COCCCOC)CC2CO 37631,c1(C(N2CCC(NC(c3c(N)cn(C)n3)=O)CC2)=O)cccc2ccccc12 37632,CS(=O)(=O)c1cc(C(=O)N=c2nc[nH]n2C2CCN(C(=O)OC(C)(C)C)C2)cs1 37633,C1(C(=O)OC)CCC(C(=O)NC(C)(C)C(C)NC(=O)CCCN(C)C(C)=O)CC1 37634,Cc1ccc(C=CC(N2CC(C(C)NC(c3cnn(CC(F)F)c3)=O)C2)=O)cc1 37635,c1(CC)c(C(N2CCC(C)C2C(=O)NCc2cnn(C(C)C)c2)=O)ccn1C 37636,c1(N2CCC(F)(C(=O)Nc3cc(OC)cc(Br)c3)C2)ncc2ccccc2n1 37637,N(C1CCCn2ccnc21)C(C1(C)CCCN1C(=O)CC1(O)CCOCC1)=O 37638,c1(C(N2CCC(O)(CNC(C(CC)(C)CC)=O)C2)=O)noc(C)c1[N+](=O)[O-] 37639,C12CCC(C1)C(=O)N2.c1(C(N)=O)cc(C(=O)NCC2CC(C(=O)OCC)C2)on1 37640,C(=O)(CCCC(=O)c1ccc(C)cc1)N(CC(CC)O)C1CC1 37641,CCC(O)CC(=O)N1CC(NC(c2coc(N(C)C)n2)=O)C(C)C1 37642,C1(NC(C2N(C(c3c(OC)csc3)=O)CCC2C)=O)CC2(C1)CC(C)(C)C2 37643,S(=O)(=O)(c1ccc(NC(C)CCc2ccc(Cl)cc2)c(F)c1)N1C(C)SCCC1 37644,C12(C(=O)NCC3C(CNC(c4c(C)onc4CO)=O)C3)CCCN(CCC1)C2 37645,C1(C(=O)NCc2cc(C(=O)NCC(N3CCCC3)C)n(C)n2)(OC)CCC(C)C1 37646,c1(C(N2CC(C)C(CNC(=O)CO)CC2)=O)c(Cl)ccc2ccoc12 37647,C(C(CC1CC1)C(=O)NCCC1COCC1O)NC(CSC)=O 37648,Nc1cc(F)cnc1C(=O)NCC(O)CC(=O)NC(CC1CC1)C1CC1 37649,C(=O)(CC(CC#N)c1ccccc1)N(C1COC1)CCc1cn(CCCC)nn1 37650,c1(OC)cc2c(cc1C(N1CCC(NC(=O)Cc3ccco3)C1)=O)OCO2 37651,C1(C2CC2)(CNC(c2cc(C)nc(O)n2)=O)CCN(C(=O)C(C)OCC(C)C)C1 37652,CCC(C)(C)CCCC(=O)NC1CCC2CCN(C(=O)CCC(C)C)C12 37653,c1(C(N2CCC(C)C(N(C(=O)CC3CCCSC3)C)C2)=O)ccc(N=[N+]=[N-])cc1 37654,C1(C(=O)NC2CCN(C(c3c(C(=O)OC)nccn3)=O)C2)COC2CCCCC12 37655,c1(C(N(CC(C)NC(c2cn(CC3CC3)nn2)=O)C)=O)cnn2ccn(C)c12 37656,c1(C(=O)NCC2(NC(c3cnn(C4CC4)c3)=O)CC2)cnc(S)n1C1CC1 37657,c1(C(=O)NC2C(C(=O)NC(C(=O)NC)CC(C)C)C2)cc(Cl)cc(Cl)c1[N+](=O)[O-] 37658,C(C(C(C)C)NC(C12CC(CO1)C2)=O)NC(C1C(C)C1C)=O 37659,c1(OC(c2c(Cl)cn(CC)n2)=O)cc(C)c(NC(C)=O)c(C)c1 37660,c1(CNC(C2CC(CC)C2)=O)nc(C(=O)N(CCCN=[N+]=[N-])C)c(C)o1 37661,c1(C(C)C)ccc2cc(C(N3CCC(O)(c4cnn[nH]4)C3)=O)ccc2c1 37662,CC(C)(O)C(=O)NNC(=O)c1cc(C(F)F)cc(F)c1 37663,c1(CS(Cc2ccc(-c3n(CC)ncc3)s2)=O)ccc(O)cc1 37664,C(=O)(CCC(C)(C)OC)N1CCC(CN(C)Cc2nnc(CC)o2)C1 37665,c1(C(N2CCN(C(C3C(OC)(OC)CC3)=O)C(CF)C2)=O)ccc2occc2c1 37666,N1(C(=O)NCc2cccc(C#N)n2)CCC2(CC1)CC(=O)NC2=O 37667,Cc1cscc1C(=O)NCC1(C(N2CCCC2C)=O)CC=CC1 37668,N1(C(c2c(C)onc2)=O)CCC2C(CCCN2C(=O)CN2CCC(C)(C)C2)C1 37669,c1(C(=O)NCCC(C)(C)NC(c2ccc(NC(C)=O)s2)=O)csc2nnsc12 37670,c1(OC)nc(N2CCCC(C)(NC(=O)CCCCCCBr)C2)nc2[nH]cnc12 37671,C1(CNC(c2ncc(F)cn2)=O)COCCN(C(c2ccc(F)c(Cl)n2)=O)C1 37672,C1(CC(=O)N(C)Cc2nc[nH]n2)C2CN(C(C3C4CCCC34)=O)CC12 37673,c1(C(N2CC(N(C)C(C3(C)CC=CCC3)=O)C2)=O)ccc(Br)cc1OC(F)(F)F 37674,C1(NC(C=CCC)=O)CC12CCC(NC(c1ccc(C(F)F)o1)=O)CC2 37675,C1(NC(CN(CC)CC)=O)CCCC(NC(=O)C(C(C)CC)OC)CC1 37676,C(C(C)(F)CNC(c1ccc(SC)o1)=O)NC(C(C1CC1)SC)=O 37677,C1(NC(=O)NCc2nc(C(C)(F)F)on2)CS(=O)(=O)CC1Cc1cccc(Br)c1 37678,c1(C(N2CC(CN(C)C(c3ccnn3C3CC3(F)F)=O)C2)=O)conc1C(F)F 37679,c1(C(=O)NCCC2CN(C(C3CC(C)(F)C3)=O)C2)cc(F)cc2cc[nH]c12 37680,O=C(C#CC1CCCC1)N(C1CCCCC1)CCNC(C12CCCC1(C(N)=O)C2)=O 37681,N1(C(C(C(C)(C)C)O)=O)CCC2(CC1)CC(NC(=O)C(C)(O)C(F)(F)F)C2 37682,C(C(O)C(C)(C)CO)CN(CC(c1cccs1)NC(=O)OC(C)(C)C)C 37683,O=C(C1Cc2ccccc21)NC12CC(C(N3CCC(C(F)(F)F)C3)=O)(C1)C2 37684,N1(C(C(CC)N2CCCC2)=O)CCN(C(=O)C(C)n2cccn2)CCC1C 37685,C(=O)(C(C)C(C)(C)C)NCCC1(OC)CN(C(c2n(CC)c(O)nc2)=O)C1 37686,N1(C(C(C)CF)=O)CC2CCC1C1CN(C(c3c(Br)nnn3C)=O)CC21 37687,C1(C)(NC(C(C(C)C)NC(c2sccc2CO)=O)=O)CCC(=O)NC1=O 37688,C1(C(=O)NCC(C2CC2)SC)C2CC2CN1C(c1cnccn1)=O 37689,C1(NCc2c(C)c(Br)ccc2F)CCN(c2ccnc(C3CC3)n2)CC12CCC2 37690,c1(C(N(CCCNC(c2cccc(OCC)c2)=O)C(C)C)=O)cc2[nH]ccc2s1 37691,C(C(=O)NC1CCN(CCC(F)(F)F)CC1)(C(C(C)C)OC)OC 37692,C1(C(N(C(C)CCNC(C2CNC(=O)C2)=O)C)=O)CS(=O)(=O)CC(=O)N1 37693,C(=O)(CC(C)CC(C)(C)C)NC(c1ccccc1)C(=O)NCCn1ncc(C)c1 37694,C1(C(=O)NC2CCCC2NC(c2cnco2)=O)(OCC)CCSCC1 37695,Cc1cccc2c1OC(C(=O)NCC(F)CNC(=O)CSCCC(F)(F)F)C2 37696,Cn1c(C(=O)NC2CCC(C(=O)Nc3ccc(Br)nc3)OC2)cccc1=O 37697,c1(C(=O)NC(C2(O)CN(C(CC(CC)C)=O)C2)C)cccc2nn(C)nc12 37698,C(=O)(CCCC(C)(C)C)N(C(C)CNC(=O)C(C)(O)Cn1cc(Br)cn1)C 37699,C1(C(N2CCCC(C(C(=O)NCCC(C(=O)OC)C)C)C2)=O)CCOC(=O)CC1 37700,N1(C(C(CCC)NC(C2CCOCC2NC)=O)=O)CCC(C)(C(C)C)CC1 37701,C1(C(N(C(CNC(=O)CC2CC2)C2CC2)C)=O)CCC(O)C1 37702,c1(C(=O)NCCCCCN(C(C(=Cc2ccco2)C)=O)C)nnc(S)n1C 37703,CC1(C)CC(C(=O)NC2CCC(CNC(c3cnn(C4CCOC4)n3)=O)C2)=NO1 37704,C1(C(=O)NCC2CN(CC)C(=O)O2)CC(NC(=O)CC2CC(C)=NO2)C12CCC2 37705,c1(NCC2CN(C(C3C(OCC)C3)=O)C2)cc(C(=O)OC)ncn1 37706,CS(=O)(=O)c1ccc(F)c(C(=O)NCC2(NC(=O)CC3CC=CC3)CCOC2)c1 37707,CC(C)(CNC(C1C=CCN1C(C1CC(=C2CC2)C1)=O)=O)CN=[N+]=[N-] 37708,C1(S(N)(=O)=O)(C(N2CC(CC)C(NC(c3[nH]c(O)nc3C)=O)CC2)=O)CCCC1 37709,C=CCC(CC(C)C)C(=O)NC12CC(CNC(=O)C3=CCCS3)(C1)C2 37710,c1(OC(C2C(C(=O)OCC)C2)=O)ccc(N2CCOCC2)cc1 37711,c1(C(N(CC(CNC(c2ccc(CC)cc2)=O)O)C)=O)c(Cl)cccc1[N+](=O)[O-] 37712,C(=O)(C1CSc2ccccc21)NC(C(C)NC(=O)CC(C)(C)C(F)(F)F)(C)C 37713,C(C)(N=c1[nH]c(=N)[nH]c(=NCc2nc(C(C)(C)C)cs2)[nH]1)C1CC(SC)C1 37714,N1(C(C(=O)N(C)CC)C)CCOCC(C(=O)NCC(n2nc(C)cc2C)C)C1 37715,c1(C(=O)NCC2CCN(C(c3c(OC)nsc3)=O)C2)ccc2nc(O)n(C)c2c1 37716,CN1CC(C(=O)N2CC(CNC(C3(F)C4CCCC34)=O)C2)c2ccccc2C1=O 37717,C(=O)(C(O)CC[S+](C)C)NCCOC1CCN(C(C(C)(C)OCC)=O)C1 37718,CN=c1nc(C(N2CCCC(CN(C(=O)CN3CCC3C)C)C2)=O)cc(C)[nH]1 37719,C(=O)(C(C(C(C)C)OC(C)(C)C)N(CC(C)(CC)CC)C)NCCC 37720,Cc1oc(-c2ccccc2)cc1C(=O)NC1CCC1NC(=O)C(C1CC1)C1CC1 37721,C(C(CC(F)(F)F)NC(C1CCCN1N=O)=O)NC(=O)Cn1cnnc1O 37722,C1(NC(C(C)(CO)CCN2CCC(C(N)=O)C2)=O)C2CC3C1C3C2C(=O)NOC 37723,CC1CC(NC(=O)C=Cc2ccc(C(F)F)o2)CN1C(c1ccc(C#N)o1)=O 37724,c1(C(=O)NCC(C)CN(C)C(c2cscc2C2CC2)=O)ccc(S(C)(=O)=O)o1 37725,C(=O)(CCC(CF)CF)N1CC(C)(C(=O)NC2CC3(C2)CC3(F)F)OCC1 37726,S(=O)(=O)(c1ccc(C)c(Cl)c1)N1CCN(C(c2ccc(C)cc2O)=O)C2C1C2 37727,c1(C(=O)NC(c2cccc(C)c2)CNC(C(CC#C)C)=O)ccc2c(c1)CC2 37728,C1(CNC(C(C)NC(C)=O)=O)CCN(C(C2CC2C(N)=O)=O)CC1C 37729,C1(C(=O)Nc2cccc(CO)n2)CCCC12CCN(Cc1cc(Cl)cnc1Br)C2 37730,Cc1nc(C(N2CC(OCCNC(C3CN(C)CC3C(F)(F)F)=O)C2)=O)[nH]c1C 37731,N1(C(CC=C)=O)CC(NC(c2ccc([N+](=O)[O-])cc2)=O)C(C2CC2)C1 37732,C1(C(C)NC(C2CN(C(C)=O)C2)=O)CCN(C(c2ncsc2C(F)(F)F)=O)C1 37733,N1(C(CC2CC(C(C)C)OCC2)=O)CCC(CO)(NC(C2C3CCCC23)=O)CC1 37734,c1(C(C(=O)NCC(C2CC2)NC(Cc2cc(C(C)C)no2)=O)O)ccc(F)cc1 37735,C1(O)(c2cn(C(C)CNC(C3CCSC(C)(C)C3)=O)nn2)CCC(F)(F)CC1 37736,c1(CC(N2CC(NC(c3cccnn3)=O)C2)=O)c[nH]c2cc(Br)ccc12 37737,c1(OCC)nc(C(=O)NC2(C(=O)NC(CN(C)C)CCO)CC2(C)C)co1 37738,c1(C(N(CCCNC(C2CC2C)=O)CCC)=O)cc2n(n1)CCN(C)C2 37739,c1(N2CCC(C#N)C2)nc(N2CCC(C3CCCCO3)CC2)c2c(n1)CCS2 37740,c1(C(C(=O)Nc2ccccc2)N(C(C)C)C)cccc(Cl)c1Br 37741,N1(C(c2ccc(=N)[nH]c2)=O)C2CCC1(CNC(C1CCN(C3CC3)CC1)=O)CC2 37742,c1(CN2CC(NC(C3(F)CCCC=C3F)=O)C2)ccc2cc[nH]c2c1 37743,CCCC(C)CCCC(=O)NCCCOCCCNC(c1cn(CCO)nn1)=O 37744,Cc1ccc(CC(N2CC(OCCNC(=O)C(C)CF)C2)=O)cc1Br 37745,c1(C(N2C(C3CCN(C(C4CCN(C)C4)=O)C3)CCC2)=O)cc2c(F)cccc2[nH]1 37746,N1(C(C(C)=C2CC2)=O)CCC(CC(C)NC(=O)C(c2ncccc2F)(F)F)CC1 37747,c1(C(=O)NCC(COC)NC(=O)CCCN2CCCC2)nccn2cnnc12 37748,N1(C(c2cc(C)on2)=O)CCCCC1CCCNC(c1cnc(O)o1)=O 37749,C1(NC(c2c(CNC(CCC(C)SC)=O)occ2)=O)CCC(C)(O)CC1 37750,C1(C(N(CCOCCN(C(C(C#C)(C)C)=O)C)C)=O)COC2(CCC2)CO1 37751,C1(C(N2CC(F)C(F)C2)=O)COC2(CCN(Cc3cncc(Cl)c3)CC2)C1 37752,Cn1nc(C2CC2)cc1C(=O)NCC1CCCC(NC(=O)COC(F)F)C1 37753,C1(C(N(C)CC2CCSC2)=O)CCN(C(=O)CCc2cncs2)CCO1 37754,CCC(C)(C)CCCC(=O)N1CC(NC(=O)Cn2ccc(C)cc2=O)CC1CO 37755,c1(C(C(=O)NC(CC)C)N(C)C(C2(C)CC2)C)csnc1OC 37756,CC(C)CCCC(=O)N1CCC1CNC(=O)COC1CCCC(C)C1 37757,c1(SC)ncc(N)c(C(=O)NC(C)(CNC(=O)CN(C2CCSC2)C)C2CC2)n1 37758,C(=O)(C1=C2CCCN=CN2NN1)N1C2C(NC(C3CC3C(F)F)=O)CC(C2)C1 37759,C1(S(N)(=O)=O)(C=O)CCC1.c1(C(=O)NCC(C)(C)OCC)cn(CC(F)F)cn1 37760,C1(C(N2CCCC(CNC(C=C(COC)C)=O)C2)=O)C(O)C(=O)N(C)C1C 37761,N1(C(C2CC(F)(F)C2)=O)CCC(CCNC(C2COCCO2)=O)CC1 37762,CCCCCC(CC)C(=O)NCCCOCCC(N1CCN(C(C)C)C(=O)C1)=O 37763,Cc1ccccc1CC(=O)NC1CCC(NC(=O)CCC2CCCCN2C)C1 37764,C1(CNC(CC2C(CNC(C3ON=C(C)C3)=O)C2)=O)CCC=CCC1 37765,N1(C(C(CCC)F)=O)CCCC(O)(CCNC(=O)CSc2nc(C)cc(C)n2)C1 37766,c1(C(=O)NCC(CC=C)NC(C2CCN(C(=O)CC)C2)=O)ccnc(OCC)c1 37767,C1(C(C(=O)NCC(C2CC2)OC)C)CCN(C(c2csc(C#N)c2)=O)CC1 37768,C(=O)(CC(C(C)(C)C)NC(=O)C(C)SC(C)C)NC1(COC)CC1 37769,C=CCC(C)(CO)CN=c1[nH]c(N2CCC(C3CCC3)C2)nc2c1SCC2 37770,N1(C(C(C)OCC)=O)CCC2(CCC(CNC(=O)NC3CCCOC3)CC2)CC1 37771,C1(O)(CNC(C(C)OCC2CC2)=O)CCN(C(c2nnn3c2CCC3)=O)CC1 37772,C1(OC)CN(C(C2(CN(C)C)CC2)=O)CCC1NC(c1cccc(C(C)C)c1)=O 37773,C(=O)(CCCC(=O)NCC(C)CNC(c1cc(C)nn1C)=O)NC 37774,Cc1cc(C(=O)NC2CN(C(=O)Cn3nc(Cl)ccc3=O)CC2O)ccc1Cl 37775,c1(C(N2C(CCC(=O)Nc3cnn(C)c3C#N)CCC2)=O)cc2ccoc2cn1 37776,CC(C)(CCCNC(=O)Cc1nc[nH]n1)NC(=O)CC1CC(F)C1 37777,c1(CC(=O)NCC2CC2NC(C2CC2F)=O)c(F)cc(F)cc1F 37778,Cn1cncc(C(N2CCC(F)(CNC(=O)CCN3CCOCC3)C2)=O)c1=O 37779,CC1(NC(c2ccc(Br)c(C(F)F)c2)=O)CCCN(C(C2CC2C#N)=O)C1 37780,c1(C(=O)NCCNC(c2cccn(C3CCSC3)c2=O)=O)ccn2ncccc12 37781,c1(NC(C(=O)NCCN(CCC(C)N2CCCC2)CC)=O)cnc(Cl)s1 37782,C(C(=O)NCCC1CN(C(C2(C(F)F)CC(F)(F)C2)=O)CCO1)(C(C)C)OC 37783,C1(NC(c2cccc(Cl)c2)=O)CCC2CN(Cc3ncc(C(F)F)s3)CC2C1 37784,C12(C(N3CC(NC(=O)NC)C3)=O)CCCC1C2 37785,C(=O)(CC(C)C(F)F)NCCN(C(=O)C(O)(C1CC1)C1CC1)CC 37786,c1(-c2nc(-c3cc(Cl)ncc3)n(CCC3CC3)n2)cc(F)cc(F)c1 37787,O=C1CN(C(c2ccc[nH]2)=O)C(C(N2CCNC(=O)C2CCO)=O)CN1 37788,N1(CCNC(CN(c2ccc(Cl)cc2)C)=O)CCN(C(C)(C)C(N)=O)CC1 37789,C1(C(N(C2CCCN(C(=O)C=CCF)CC2)CC)=O)CC(F)(F)CCC1(C)C 37790,c1(C(=O)NC2CCCN(c3ccnc(Br)n3)C2)cnn2c1CCCC2 37791,C(=O)(CC(C)(C)c1cccc(Br)c1)NCC1(CNC(C2(F)C(C)C2)=O)CCC1 37792,c1(OC)ccc(C(=O)NCC2CCN(C(=O)Cc3cc[nH]c3)CC2C)c(Cl)c1 37793,C12(C(N3CCN(C(c4cc(Br)c[nH]4)=O)CC3)=O)C3C4C1C1C2C3C41CO 37794,c1(C(=O)NC2(CNC(C(C)C3CC3)=O)CCC2)n[nH]c2c1COc1ccccc1-2 37795,C1(CC)(NC(=O)CC2CCCC2O)CN(C(C2CCC(C)O2)=O)C1 37796,CC(C)C(CCN(C(=O)C(C)C(F)F)C)NC(=O)Cc1ccc(Cl)cc1 37797,c1(C(C(=O)NCCOC)N(C2CCC(F)(F)C2)C)ccc(F)c(Br)n1 37798,Cc1ccc(C(=O)NCC2CCN2C(C2CCCC2C)=O)c(N)c1C 37799,c1(C(=O)OC)ccnn1C(C)(C)NC(C1CC1C1CCCC1)=O 37800,N1(C(=O)CC2CC3CC3C2)CC2CCC(C1)N2C(c1ccsc1C1CC1)=O 37801,N1(C(c2ccsc2)=O)CC2(C1)CN(Cc1ccnc(Cl)c1)CCO2 37802,C1(C(=O)NCCC2N(C(C(C=CC)O)=O)CCC2)C2CCC1(C)C2(C)C 37803,CC1C2C(CCN2C(=O)CCc2cccs2)CN1C(C12CSCC1C2)=O 37804,C1(CNC(c2nccc(C)c2)=O)CN(C)CCN1C(C1CCN(C)C1C)=O 37805,c1(C(N(CC(CN(C(CC(CCCC)O)=O)C)O)C)=O)cc([N+](=O)[O-])ccc1O 37806,C1(NC(C2CS(=O)(=O)C2)=O)CCCC12CN(C(c1c(O)cc(F)cc1F)=O)C2 37807,N1(C(CC2CC(=C)C2)=O)CCN(C(=O)C(N2CCOC2=O)C)C(CC(C)(C)C)C1 37808,c1(CC(=O)NCC(CNC(c2c(C)ncc(C)c2)=O)O)cc(Cl)cc2c1OCC2 37809,CS(=O)(=O)c1ccc(C(N2CCC(F)(F)C(NS(=O)(=O)C(F)(F)F)C2)=O)cc1Br 37810,c1(N(c2ccnc(-c3ccc(OC(F)(F)F)nc3)c2)C(=O)C2CC2)cnc(Br)nc1 37811,C1(C(N2CC(CC(=O)NCc3nccc(OC)c3)OCC2)=O)CC(=O)OC1(C)C 37812,c1(CC(=O)NC2CC3(C(NC(C(CC#C)O)=O)C3)C2)ccc(Cl)cc1F 37813,C(=O)(C(CNC(=O)CN1CC(C)(C)C1)C(C)(C)C)NCCc1c(C)ncs1 37814,CCCCCCn1nnnc1C(C(C)C1CCC1)NCCc1cccnc1 37815,CC1CN(C(=O)C(C)(C)N2CCOCC2)CC(C)C1Cc1cccc(O)c1 37816,Cc1c(C(=O)NCC(C(C)C)NC(c2c(Cl)cnn2C)=O)sc2ccccc12 37817,C(CC(=O)NCc1cccc(NC(C2CN(C(N)=O)C2)=O)c1)(C(C)C)OC 37818,Cc1cc(C(=O)NC23CC(NC(=O)C(C)OCCC(C)C)(C2)C3)cc(C)c1N 37819,N1(C(C(CC=C)OC)=O)CCc2nc(CNC(c3ccco3)=O)sc2C1 37820,c1(CC(=O)NCC2CN(C(C3CN(C4CCC4)C3)=O)CC2O)cccnc1Br 37821,C(=O)(C(F)(CC)C(=O)OC)N1C(C)CCC(NC(c2c(CC)ccc(Cl)c2)=O)C1 37822,c1(C(N2CCC(C)(NC(C3CCC(C)C3)=O)C2)=O)cc2c(s1)CN(C)CC2 37823,N1(C(CCCC(=C)C)=O)CCCC2(C1)CN(C(=O)CC1CCCCC1O)C2 37824,c1(C(=O)NC(CC=C)CNC(=O)C(CC)N2CCCC2=O)ccc(Cl)cc1F 37825,N1(C(C2CC(C#C)(O)C2)=O)CCN(C(C2(C(O)C(F)(F)F)CCC2)=O)CC1C 37826,c1(C(=O)NCc2ccc(C(NOC)=O)o2)ccc([N+](=O)[O-])[nH]1 37827,N1(C(C2(OC)CC(C)(C)C2)=O)CC(C(=O)NC2CC3CC3C2)C(F)(F)C1 37828,c1(OC(C)C)ccc(Cl)cc1C(=O)NCCC(C)NC(=O)CC1CC(=O)C1 37829,C1(C(=O)NCc2c(C)nc(CC)o2)CN(C(C2CC(C)(O)C2)=O)CCC1(C)C 37830,N1(C(C2CC(C)OCC2)=O)CCCCC2(CCOCC2)C1 37831,C1(NC(CC2(COC)CCCC2)=O)CCC(NC(c2nscc2N)=O)CC1 37832,c1(CNC(C2CC(CC)C2)=O)cc(F)c(F)c(F)c1.C12CCC(CO1)NC2=O 37833,c1(C(N2CC(CNC(c3nc(C(C)=O)sc3)=O)C(C)(C)C2)=O)c(C)nc(C)nc1C 37834,CC(CCC(=O)N1CC(n2cc(Cc3cccc(F)c3)nn2)C1)c1ccccc1 37835,C1(CNC(c2cc(C(N)=O)no2)=O)(CNC(=O)CC2CC23CC3)CC12CCC2 37836,c1(C(=O)NCC2(F)CC(CNC(C(CC)n3ccnc3)=O)C2)n[nH]c(C)c1Cl 37837,Cc1cc(CC(=O)NC2CCCN(C(=O)C(=O)NCC(F)(F)F)C2C)ccc1F 37838,C1(C(N(CCC)CCO)=O)CN(C(=O)CC(C)C(C)C)CCC1(C)C 37839,C#CCC(C)C(=O)NCC1(O)CC(NC(C2CCCN(CC(F)(F)F)C2)=O)C1 37840,N1(C(C2NC(=O)C3C2CC3)=O)C2CCC1CN(C(c1cc(C3CCC3)on1)=O)C2 37841,c1(C(N2CCCN(C(C(=O)NCC)=O)CC2CO)=O)[nH]c2ccc(F)cc2c1C 37842,N1(C(C)=O)CCCCC1CC(=O)N(CCNC(=O)Cc1ccccc1)CC1CC1 37843,N1(C(=O)Nc2n[nH]cc2-c2ccc(Cl)cc2)CCN(CCOc2ccccc2)CC1 37844,N1(CC(=O)NCCCC2(NC(C3CC3C(F)(F)F)=O)CC2)CCC(O)CC1 37845,c1(C(=O)NC2C(NC(C=C(C)C3CC3)=O)CC2)cnc(OCC(F)F)cn1 37846,C1(NC(C(C)C(C)(F)F)=O)CN(C(c2cc[nH]n2)=O)CC2(CCC2)C1 37847,c1(C(N2CCC(c3cnn[nH]3)C2)C(=O)NC(CC)C)cc(Cl)c(Cl)c(Cl)c1 37848,C(=O)(C(C)(C)N1CCCC1)NCC(C)N(C(=O)CCNC(N)=O)C 37849,C1(C)(C(=O)NC2CCN(C(Cc3c(C(C)C)con3)=O)C2)CC(C(F)(F)F)=NO1 37850,C#CC1(NC(=O)C(C(C)NC(=O)Cc2cccnc2F)C(C)C)CCCCCC1 37851,C1(NC(CSSC)=O)CCN(C)C12CCCN(C(=O)Cn1cc(Cl)cn1)C2 37852,c1(CC)ccc(C=CC(=O)NCCC(C)NC(=O)C=CCn2cncn2)o1 37853,N1(C(c2c(C)cc(Br)cc2F)=O)CCC2CN(C(c3ccc(O)cn3)=O)CC2C1 37854,CCCS(=O)(=O)N=c1cc[nH]c(-c2ccc3nn(C)c(C)c3c2)c1 37855,C1(NC(COCC(C)(C)C)=O)CN(C(C2CCOC(=O)CC2)=O)C(C)(C)C1 37856,c1(C(C)NC(C2(C)N(C(c3c(C)nn(C)c3)=O)CC2)=O)cccc2ccccc12 37857,c1(C(=O)NC2CN(C(CCCCC)=O)CC2C)ccc2c(c1)C(C)CO2 37858,C1(C(N(CC(C)NC(=O)CC2(N(C)C)CCCCC2)C)=O)CC(F)C(=O)N1 37859,C1(C(=O)NC(c2cnn[nH]2)C)CCCN1NC(=O)c1c(Cl)cnn1C 37860,CCCC(C)(O)C(=O)NCC(CC1CC1)C(=O)NCC1CC(CC)C1 37861,C1(C(=O)NCCC=CCCC)C2CCC(C2)C1NC(C1CC2CC1CC2=O)=O 37862,C(CS(=O)(=O)C1CCOCC1)C(C#N)C(=O)c1cnnn1-c1ccccc1F 37863,C(c1ccc([N+](=O)[O-])s1)=CC(=O)NC(CN(C(C=C1CCC(C)C1)=O)C)(C)C 37864,N1(C(COCC#C)=O)CCN(C(=O)CC(C)COC)CC1Cc1ccccc1 37865,c1(C(=O)NC2C3CN(C(c4ccnc(O)c4Br)=O)CC23)ccn2ncnc2c1 37866,C1(C(=O)NCC2C(NC(c3ccc(CCC)[nH]3)=O)C2)CC(=O)N(CC(F)(F)F)C1 37867,N1(C(C(=O)N(C)C)=O)CC2(CCC2NC(=O)CC2CCCC23CC3)C1 37868,C(C)(c1cccs1)=CC(=O)NCC(CC)NC(=O)C(c1cccnc1)O 37869,C(=O)(CC(F)(F)F)N(C1CCC(CNC(=O)CCNC(=O)OC(C)(C)C)C1)C 37870,c1(C(=O)NCC(CC)NC(c2cnsc2C)=O)cccc2c1OC(F)(F)O2 37871,C1(NC(c2ccc3ccnn3c2)=O)CCN(C(c2cccc(F)n2)=O)C12CCC2 37872,C1(C2CCC2)(CNC(C2C(C)OCC2)=O)CCN(C(c2cccc[n+]2[O-])=O)CC1 37873,CC1CC(CCNC(C2(C)CC2)=O)CCN1C(=O)Cn1cncn1 37874,CCC(CC(=O)N1CCCC(CNC(C2(n3cccn3)CCC2)=O)C1)C(C)C 37875,N1(C(C(C(C)C)CNC(=O)CSC(F)F)=O)CCOCC(C)(F)C1 37876,N1(C(c2c(C(C)(C)C)con2)=O)CCOC(CNC(c2cncn2C(C)C)=O)C1 37877,C=CCCCCCCCCNC1(c2nnnn2CC(F)F)CCCC1CCCC 37878,c1(CC(=O)N(CC(C)CNC(=O)C=Cc2ncco2)C)cn2cc(F)ccc2n1 37879,C(=O)(C(O)C(F)F)NCCC1CC(NC(COCCC=C)=O)C1 37880,c1(C(=O)NCC2CC(CNC(c3cc(Cl)no3)=O)C2)sc(F)cc1Cl 37881,C1(CNC(C(C(C)C)NC=O)=O)(NC(=O)CC2CC2(Cl)Cl)CCCCCC1 37882,c1(C(=O)NC2C(C(=O)NCC3CC(OCCOC)C3)CCC2)cccc(C#N)c1C 37883,C1(C(=O)NCC(C)(O)COC)(SC)CN(C(=O)CCCC2CC2)C1 37884,c1(CC(N2CC(C(=O)NCc3occ(C)n3)C(O)CC2)=O)ccc2c(c1)CCC2 37885,c1(NC)c(C(=O)N(C)CCNC(=O)Cc2ccc(Cl)nc2)sc2nccnc12 37886,C1(CC)CN(C)CCCN1C(=O)CC1(N(C)C(c2cc(C3CC3)[nH]n2)=O)CC1 37887,c1(NC(N2CC(NC(C3CCCC(CC)C3)=O)C2)=O)ncnc(C)c1C 37888,CC(C)(C)CC(O)C(=O)NCC1CC(CNC(=O)CNc2nccs2)C1 37889,C(=O)(C1COc2ccccc21)N(C)CC1CCN(C(=O)Cn2nnc(=O)[nH]2)CC1 37890,c1(CC2C(NC(C=CCN(C)CC)=O)COC2)nnn(C)c1C(=O)NN(C)C 37891,c1(C(N2CC(NC(C(CC)OC)=O)C2)=O)ccc(OC(C)(C)C)cn1 37892,Cc1ccc(C(N2CC=CC(NC(C3(C)CCCS3)=O)C2)=O)c(N)c1F 37893,CC1(CNC(=O)CCN2CCCCC2=O)CCCN(C(=O)Cn2cnnc2)C1 37894,C(C)(CN=c1[nH]nc(C(C)(C)C)o1)OC.c12c(OC)ncnc1N2 37895,n1(CC)nc(C)c(C)c1NC(=O)NCc1cscn1 37896,C(C)(CC(C)C(F)F)NC(CCN(CC#C)C(c1cnc(CC)o1)=O)=O 37897,c1(CC(=O)N(C2CCCCN(C(=O)C(O)C3CC3)C2)C)ccc2occc2c1 37898,c1(-c2c(C(=O)NCC3C(NC(CC(=O)OCC)=O)C3)c[nH]n2)ccccc1Cl 37899,Cc1nc2sccn2c1C(N1CCC(NC(=O)CC2CC2(Cl)Cl)C12CC2)=O 37900,C1(CCNC(C=CC(=O)OCC)=O)CSCCN1C(=O)CS(=O)(=O)NC 37901,c1(C(=O)NCC(C(C)C)NC(=O)C(C)Cc2cccc(F)c2)ncc[nH]c1=O 37902,c1(NCc2n(CC(=O)OC)ncc2)ccc2c(c1)CCC(C)C2 37903,Cc1cc(C(N2CC(n3cc(C4(N(C)C)COC4)nn3)C2)=O)c2c(Br)cccc2n1 37904,C1(CNC(CN(C)CC)=O)CCC(CNC(C2CCCN(C(N)=O)C2)=O)CC1 37905,C12CC(=O)N(C1)C2.C12(C(N3CC(CCCCNC(CCOC)=O)C3)=O)CC(F)C1C2 37906,c1(NC(C2CN(C(c3cnc(O)nc3O)=O)CCS2)=O)ccc(I)c(Cl)n1 37907,c1(OC)ccc(CN2CCC(O)C(C(=O)Nc3nc(C4CC4)cs3)C2)c(Cl)c1 37908,Cc1cc(CN(C)C(C2C=CCCN2C(c2cc(C(C)C)oc2C)=O)=O)n(C)n1 37909,Cc1cc(C(=O)NCC(N2CCOCC(O)C2)=O)cnc1C 37910,c1(CC(C(=O)N(C)CC2(CNC(C3(OC)CC3)=O)CC2)C)c(C)nn(C)c1C 37911,c1(C(N2CC(CN(C(C(CSC)(C)C)=O)C)C2)=O)cn(C2CC2)c(C)cc1=O 37912,CC(C)(C)C(C(=O)NCC12CC1CN(C(c1cc(C3CC3)cs1)=O)C2)C1CCC1 37913,CC(C)(C)CC(=O)N1CCC1(C)C(=O)NCCOc1ccc(Cl)cc1 37914,C(C)(C(=O)N1CC(CNC(=O)Cc2ccc(F)nc2)C2(CC2)C1)(C(C)C)OC 37915,C(=O)(CCC(=O)N1CCN(c2ccccc2CNC(C2(F)CC2C)=O)CC1)OC 37916,N1(C(c2n(CCC)ncc2)=O)CCC(C(=O)N(C(C)C(F)F)C)C(C)(C)C1 37917,N1(C(CC(COC)C)=O)CC(C)(CNC(=O)CSS(C)(=O)=O)CC1(C)C 37918,CC(C)CCC(O)C(=O)N1CCC(C(C)C(=O)NOC2CCOC2)C1 37919,S(=O)(=O)(c1ccc(NCc2ccncn2)c(Cl)c1)NCC(C)(C)CCCO 37920,c1(NCC(=O)NCC2(O)C(C)OCC2)ccc(=O)n(-c2ccncc2)n1 37921,Cc1ccc(NC(C2(NC(=O)CN3CC4CCC3C4)CCOCC2)=O)cc1C 37922,c1(C(=O)NC2CCN(C(C(n3ccc(Br)n3)C)=O)C2)ccc2ccccc2n1 37923,CC(C)C(C)(C)C(=O)NC1CC(NC(c2c[nH]nc2[N+](=O)[O-])=O)CC1O 37924,c1(N(CCC2CC2)CC)nnc(-c2oc(CO)cc2C)n1CCc1ccccc1 37925,C(=O)(C(CC(C)C)N(C(=O)CCCC1(OC)CCC1)C)N1C(C(=O)OCC)CC1 37926,c1(C(=O)NCC(CCCC)NC(C2(CC#C)CC=CCC2)=O)cc(F)ccc1N 37927,c1(C(=O)NC2C3(CC(NC(C(CCSC)O)=O)C3)C2)cc(Cl)ccc1O 37928,Cc1cnc(N2CCOCC2)nc1C(N1CC(SC(C)(C)C)C1)=O 37929,C(=O)(CC(CN(C)C)CC)NCC(CC)NC(c1ccc(CO)o1)=O 37930,c1(COC)nc(N2CCC(CNC(C3CCC(N=[N+]=[N-])C3)=O)C2)cc(Cl)n1 37931,C(=O)(CN=c1cc[nH]cc1)N1CC(CC(N2Cc3c[nH]nc3C2)=O)OCC1 37932,N1(c2ncc(C(=O)OC)c(C)n2)CCC2(CCCN(C(c3cccn3C)=O)C2)C1 37933,CCCCC(CNC(=O)COCCCOC)NC(=O)CC1CCS(=O)(=O)C1 37934,CCC(CN(C)C)CC(=O)N1CC2(C1)CN(C(=O)Cc1nc[nH]n1)C2 37935,c1(C(N2CCC(O)(CN(C)C(c3cc(F)n[nH]3)=O)C2)=O)[nH]c2ccccc2c1Cl 37936,C=CC1(C(=O)NOCc2ccc(C)cc2)CCN(C(c2csc(C#N)c2)=O)CC1 37937,C12(C(=O)NCC3CN(C(c4cccc(N)c4)=O)C3)CC1Cc1c[nH]nc12 37938,CC1(C)CCOC(C(=O)NCC2CCCCC2C(=O)NCc2ccc(O)cc2)C1 37939,C1(CCC)CN(C(=O)Cc2ccnn2C)CC1C(=O)NCC(N1CCCC1)=O 37940,N(C(=NCCC(=O)NC)NC1CCN(CC2CCCC2)C1)C(c1nnc(C)s1)C 37941,c1(C(N(C)CC)=O)cccc(C(=O)NCC2CN(C(=O)C(C)COC)CCO2)c1 37942,CCCCCC(C)NC(=O)CC1CCC(NC(=O)CCCC2CCCC2)CC1 37943,C(=O)(C1=CCCC1(C)C)NC(C(C)C)(C)CNC(=O)CCOCC1CCCO1 37944,c1(C(=O)NC2CC(C(=O)NCCc3cccs3)C2)cccc2nccnc12 37945,C(=O)(C1CCc2c[nH]nc21)N(C1CCCN(C(=O)CCc2cccs2)C1)CCO 37946,c1(NC2CCCN(C(C=Cc3c(C)cncc3)=O)C2)cc2nccn2cn1 37947,N1(C(CC2(C=C)CCC2)=O)CCN(C(=O)C(F)(F)C(C)O)CC1C 37948,c1(CC(=O)NCC2OCCN(C(c3c(C)n(C)nc3)=O)C2)ccc(F)cc1F 37949,C1(C(=O)NCCCCN(C(Cc2ccc(C)o2)=O)C)CCn2nncc2C1 37950,c1(C(N2CC3(OCC(NC(CCC=C=C)=O)C3)C2)=O)cc(C)c2c(c1)CCC2 37951,CN1CCc2c(C(N3CCCC3C(=O)NC3CC(F)(F)C3)=O)cccc21 37952,c1(C(N(C)CC2(CNC(C3C(CC)OCC3)=O)CC2)=O)cn2c(n1)C(C)CCC2 37953,N1(C(CSCCN(C)C)=O)CCC(N(C)C)(CNC(C2CCCSC2)=O)C1 37954,c1(CC)ccc(C(=O)NC(C)CNC(=O)CCC2CCOCC2)cc1S(C)(=O)=O 37955,c1(C(N(CCN(C(=O)CC(=O)OC(C)(C)C)C)C)=O)cnc(O)c(Br)c1 37956,C(=O)(CC(C)C(F)(F)C(F)(F)F)N1CC(C(=O)Nc2ccc(C=C)cc2)C(O)CC1 37957,c1(CC)cc(=NC(=O)C(CNC(C2(CC)CCC2)=O)CC(C)C)[nH]n1C 37958,C(=O)(C(=NOC)c1ccco1)NC1CCCCN(C(C2(CCC)CCC2)=O)C1 37959,N1(C(C=NOC)=O)CC2CC(NC(c3cc(O)ccc3Br)=O)C(C2)C1 37960,N1(C(C(CC)CN(C)C)=O)CC2(CCC(NC(=O)C(n3ccnc3C)C)CC2)C1 37961,c1(CC(N2CCCC(CNC(=O)CC3(O)CCOCC3)C2)=O)c(F)cccc1F 37962,c1(C(=O)NC2CCCC(C(=O)N(C3CCOCC3)CC)C2)ccc2c(c1)CCCS2 37963,c1(CC(N2CCCCC(NC(C3CCCS3)=O)C2)=O)cnc2cccnn12 37964,c1(CC)nc(C(=O)NCC(C)N(C)C(c2csc(-c3cn[nH]c3)n2)=O)n[nH]1 37965,C1(C(N(C)C)=O)(N(C(=O)NCC2CON(C)C2=O)C)CCCCC1 37966,c1(C(N2CC(NC(CCCC(C)=O)=O)CC2(C)C)=O)cc2ccc(F)cc2[nH]1 37967,N1(C(c2c(CC)noc2)=O)C(CNC(=O)CN2CC(=O)NC2=O)CC2CCCC12 37968,N1(C(c2cccc(C)n2)=O)CC(N=[N+]=[N-])CC1C(=O)N(CC(C)C(F)(F)F)C 37969,c1(C(=O)NCCN(CCC)C(C2(CF)CC2(F)F)=O)nccc2ccsc12 37970,Cc1cc(Cl)c(CN2CCOC(C(C)O)C2)c(Cl)c1 37971,C(=O)(C(C)(C)CO)N1C(c2n(C)ccn2)CCC1 37972,CC(C(=O)NCCC1CCN(C(c2ccc(C(F)F)cc2)=O)C1)C(F)F 37973,C12(NC(C3(CC=C)CC3)=O)CC1CN(C(C1(CCN(C)C)CCCC1)=O)C2 37974,N1(C(CC2CC(OC)C2)=O)CCCC(F)(CNC(=O)C(C)(C)c2ccccc2)C1 37975,c1(CCN=C(NCCC2(C)CC2)NCC2CC2)cnc2c(Cl)cnn2c1 37976,N1(C(C2N(C)CCC2)=O)CCC(C)(C)C1CC(N1CCC1CN=[N+]=[N-])=O 37977,Cc1cc(C(F)F)n(CC(N2CCCCC2C(C)NC(=O)C(C)(C)CO)=O)n1 37978,N1(C(CC2CC(CC)C2)=O)CCC2CCCC12CNC(c1ccnc(Cl)c1N)=O 37979,c1(C(N2CCC(O)(CNC(c3cc(CC)c(C)s3)=O)C2)=O)ccc(N)c(Cl)c1O 37980,C1(NC(CNC(=O)NC)=O)CCC2CN(c3cc(C(N)=O)nc(Cl)n3)CC2C1 37981,c1(-c2n(C)cnn2)ncccc1C(=O)NCCCCNC(C1CC2CC2C1)=O 37982,CCCCCCCC(=O)N1CC(CC(=O)NCCCCN(C)C)C2(CC2)C1 37983,C1(C(C)C)CCC(C(=O)NCC2CN(C(c3ccc(C4CC4)o3)=O)C2)CC1 37984,c1(C(=O)NC2CCN(C(C3(N(C)C)CC3)=O)CC2O)c[nH]c2cc(C#N)ccc12 37985,C1(NC(c2ncccn2)=O)CN(C(c2ccc(O)nc2)=O)C2(CCCC2)C1 37986,C1(C)(CC)CC(C(=O)NC(Cc2ccoc2)CO)CCO1 37987,C1(OC)CN(C(=O)Cn2nccn2)C(C)(CNC(c2ncc[nH]c2=O)=O)C1 37988,CC(C)(C)C(C(=O)N1CC(O)(CNC(C2(C#N)CCOC2)=O)C1)C1CCC1 37989,C12(C(=O)NCC3(O)CN(C(c4nc(C(C)C)oc4)=O)C3)CC(CO1)C2(C)C 37990,c1(C(=O)NCCC2N(C(c3ncn(C)c3)=O)CCC2)cnn(C)c1S(C)(=O)=O 37991,N1(C(COCC)=O)CC23CCCC2(C1)CN(C(=O)C(c1cc(F)c(F)c(F)c1)O)C3 37992,c12cccnc1C(=O)N1CCC(CC1)C(C)NC2=O.C1(NC(C)=O)SCCS1 37993,c1(CN2CCC(OCC)C(C(=O)O)C2)nc2cc(Br)ccc2n1C 37994,C(C1CC1)(C1CC1)=CC(=O)NCCCN(C(c1cc(SC)oc1C)=O)CC 37995,C1(CNC(C(N2CCSCC2)C)=O)CCCCC1NC(c1ccn(CC#N)n1)=O 37996,c1(C(N2CCC(CNC(C=COCC)=O)(OC)C2)=O)c(C)nn(C)c1OC 37997,C=CC1CN(C(C2(N(C)C)CC2)=O)CC1NC(=O)CNC(=O)CCC 37998,N1(C(C2(C#N)CC=CC2)=O)CCC(NC(c2ccc(Cl)nn2)=O)C(CO)CC1 37999,C(=O)(CCCCC(F)(F)F)NC(CNC(C=C1CCC(C)C1)=O)C1CCC1 38000,c1(C(=O)NCC(C)NC(C(CCCC=C)(C)C)=O)ccc2c(c1)NC(=O)CCC2 38001,N1(C(=O)CCc2cncnc2)CCC2CN(C(=O)NC3Cc4nccn4C3)C2C1 38002,N1(C(C(C)NC(C(CC2CC2)OC)=O)=O)CC(F)(F)CC1C 38003,N1(C(c2ccc(F)c(Br)n2)C(=O)NC)CCC(C)(C#N)CC1 38004,c1(C(=O)NC2(C)CC(NC(c3cccnc3O)=O)C2)cc2c(s1)CCOC2 38005,N(C(=NCC(C)N(c1ccccc1)C)NC(c1ccc(C)c(C)c1)C)C(C=C)C 38006,C12(C(=O)NCCC3CCN(C(C4CC5(CSC5)C4)=O)C3)CCC(CC1=O)C2 38007,N1(C(CCCC2C(C)C2)=O)CCCN(C(c2cc(O)nn2C)=O)CC1C 38008,c1(C(=O)OC)ccc2c(c1)CCN(C(=O)Nc1[nH]cc3c1CCC3)C2C 38009,C12(NC(=O)CCSC(F)(F)F)CCCN(C(c3ccc(F)o3)=O)CC1C2 38010,N(C(=NCCCN(C)C)NC1CC1(C)C(F)(F)F)C(C)C1CC1 38011,c1(C(N(CCNC(C2(C)CCC(=O)N2)=O)CC)=O)c(F)cc(Cl)cc1Cl 38012,c1(N2CCOCC(NC(c3cnn(CC)n3)=O)C2)ncc(Br)cc1C#N 38013,N1(C(C2C(C=C)OCC2)=O)CC2CCC(NC(c3ccoc3CCC)=O)(C2)C1 38014,Cc1cc(Cl)cc(C(N2CCCCC2CNC(=O)CC2CCCOCC2)=O)c1N 38015,c1(C(=O)NCCCN(C(c2cn(-c3ccccc3)nn2)C)CC)ncccc1Cl 38016,C1(COC(C2CCC(c3ccccc3)O2)=O)CCCCC1N1CCCC1=O 38017,CCC(C)C(C)CN=c1[nH]c(=NCCCc2nc(C)cs2)c2cc(Cl)ccc2[nH]1 38018,c1(C(=O)NC(C2(O)CCCCC2)C(=O)NCCCCN(C)C)cc([N+](=O)[O-])n[nH]1 38019,C1(C(=O)NCCCCCN(CC(=O)NC)CC)CC1(C)C(=O)NC(C)C 38020,C1(C)(CNCc2nc(C)n(C)c2C)CCCC(C)(C)C1 38021,N1(C(=O)CC2CC3CC3C2)CCN(C(c2cnc(C3CCC3)o2)=O)C(CCO)C1 38022,c1(C(=O)NCC2(NC(C3COCC(C)O3)=O)CCCCC2)cc(C#N)ccc1O 38023,CCCCCC(O)CC(=O)NC1CCC(CNC(=O)CCCN(C)C(=O)OC)C1 38024,CC(C)(C)C(C(=O)N1CC2(CCCO2)C1)NC(c1sccc1CO)=O 38025,C1(NC(C(CC=CC)CC)=O)Cc2ccccc2C1NC(=O)CCc1cn[nH]c1 38026,CCCN(OC)C(=O)CC(CNC(=O)C(CN(C)C)N(C)C)C1CC1 38027,n1(CC)cc([N+](=O)[O-])c(C(=O)OCCCN(C(=O)OC(C)(C)C)C2CC2)n1 38028,C(=O)(C1=CCCC1(C)C)NC(C(C)(C)NC(CC1(C=C)CCC1)=O)C 38029,N1(C(C(F)=CC)=O)CCC2CCN(C(=O)CCC3CCCCN3C)C2C1 38030,N1(C(C2(C)CC2(F)Cl)=O)CC2CCC(C1)N2C(c1cnns1)=O 38031,N1(C(COC(C)(C)C)=O)CCC2(C1)CN(C(=O)CC(F)(F)Br)CCO2 38032,Cc1nc(SCC(c2ccc(C3CC3(F)F)cc2)=O)n(C2CCS(=O)(=O)C2)c1C 38033,CCC(CC)(C(=O)NCC(C)(C)CC(=O)N(C)CC1(C#N)CC1)C(C)C 38034,C1(C(C)C)CN(C(=O)C(N)=O)CCC1NC(=O)CN1CCCC(CO)C1 38035,c1(N(CCC#N)C)cccc(C)c1.c1(CCC)cnc(CN)s1 38036,c1(N2CC(C)(NC(c3ccc(C#C)cc3)=O)C2)nc(CC)nc2sccc12 38037,C(=O)(C(O)C(C)(C)C)NC1CC(C)(NC(c2nc(CN3CCOCC3)cs2)=O)C1 38038,C#CCCCCCCCNC(=O)CC(CC)NC(c1cc(C)cc(C)c1)=O 38039,Cc1ccnc(F)c1NC(=O)NCCc1ccc(Br)cc1C(C)C 38040,C12(C(CNC(c3cn(C(F)F)cn3)=O)NC(c3ccoc3Cl)=O)CCC(CC1)C2 38041,O=C(C#CC1CC1)N1CCC1CNC(c1ccc(C(F)(F)F)[nH]1)=O 38042,N1(CCc2c(C)cccc2)C2CCCC1CN(C(C1CCC(C)(C)C1)=O)C2 38043,N#Cc1c(N2CC(C3(NC(=O)CCC4CCC(C(N)=O)O4)CC3)C2)cccc1F 38044,N1(C(=O)OC(C)(C)C)CCC(C2(O)CN(Cc3ccc(OCCO)c(Br)c3)C2)CC1 38045,CCCCC(C)CCC(=O)N(CC(C)O)CCNC(c1cccc(C)c1N)=O 38046,c1(C(N2CCC(NC(C3(CC#C)CC3)=O)C(O)C2)=O)ccc2nc(C)[nH]c2c1 38047,Cc1c(C(=O)NC2(C)CCN(C(=O)C(C)O)CC2)sc2[nH]cnc(=O)c12 38048,C1(C(=O)OCC)CCS(=O)(=O)C12CN(C(C1CCCO1)=O)C2.n12cc(nn1)C2.OC 38049,C(C)(C(C(=O)NC1CC(O)C1O)NC(C1OCCC1(C)C)=O)OC 38050,C1(NC(C2(NC(=O)CC3CCOCC3)C(C)(C)C2)=O)CCn2nnnc2C1 38051,N1(C(C2=CC(C)(CC)C2)=O)CCCC2(NC(=O)C(F)=C(C)C3CC3)CCCC12 38052,Cc1nn(C)nc1C(=O)NCC1(CNC(c2cc(Cl)cs2)=O)CCCC1 38053,O=S(=O)(c1cnc(Cl)c(C(F)F)c1)N1CCN(CCC2CC2(Cl)Cl)CC1 38054,c1(OC)cccc(-c2cc(C(=O)OCc3nnn(C)n3)c(C)o2)c1 38055,Cc1[nH]c(CN2CC3CC2C3C(=O)Nc2ccc(Br)c(Cl)c2C)c(C)c1[N+](=O)[O-] 38056,CCC(C)CC(C)C(=O)NCC1CC2CCC1N(C(c1cnnc(Cl)c1)=O)C2 38057,C1(C)(C(=O)NC(CCOC)C(N)=O)CCCN(C(c2ccco2)=O)C1 38058,N1(C(Cc2c(C)n[nH]c2)=O)CCC(n2cc(NC(=O)CC(C)(C)C)nn2)C1C 38059,N1(C(c2cc(OC(C)C)ncc2)=O)CCC(C)N(C(=O)C(O)C(C)C)CC1 38060,C1(CC(=O)NC(C)CCCNC(c2ccnn2C2CCC2)=O)CC2CCC1CC2 38061,C(C)(C(=O)NC1CCCC1NC(=O)Cc1ccoc1)(C1CCOCC1)NC(C)=O 38062,C1(C(=O)NC2C3CCC4C(C3)CC24)(C(=O)O)CSC(c2ccccc2)=NO1 38063,c1(CCC)c(C(N2CC(CN=[N+]=[N-])C2)=O)cnn1CCO 38064,c1(OC)cnc(C(=O)NC2(C)CC(NC(c3n[nH]c(C4CC4)n3)=O)C2)c(F)c1 38065,C1(Nc2ccc(C(C)=O)cn2)CCN(C(c2cnn(C(C)(C)C)c2)=O)C(C)C1 38066,C#Cc1ccc(C(=O)NC2C3CC2N(C(C2CCC(=O)N(C)C2)=O)C3)nc1 38067,C(=O)(CCCCc1cn(C2CCC(C(=O)N(C3CCN(C)C3)C)C2)nn1)OCC 38068,C1(C(N2C(C(=O)NCC(C)(C)CO)COCC2)=O)CCc2nc[nH]c2C1 38069,c1(OCC)ncc(C(=O)NCCCNC(=O)Cc2ccc(C(F)F)cc2)cc1Cl 38070,c1(C(N2C(C)(C(=O)NCCOCCCC)CC2)=O)ccc(C)c(C)c1 38071,C(=O)(CCN(OC)C(=O)CCCCCNC(=O)CC1CCCC2CC12)OC 38072,c1(C(=O)NC2(C)CC(C(N(CC(C)SC)C)=O)C2)cccc(F)c1F 38073,c1(C(=O)NCCN(C(C(C)C2CCCO2)=O)C2CCCC2)cnc2sccc2c1 38074,C1(CNC(C2(CC#C)CCCO2)=O)CC(C)CN(C(=O)C(OC)OC)C1 38075,c1(CCNC2CCCCC2)cc(C(=O)CCCNC(=O)OC(C)(C)C)no1 38076,C(CCC(CO)NC(=O)C(n1ccc(C)n1)C)NC(c1ccc(SC)s1)=O 38077,c1(C(=O)NC(CNC(c2ccc(C)nc2O)=O)C2CCC2)c(Cl)ccc(F)c1C 38078,C1(NC(=O)Cn2ccnn2)CC2CN(C(C3(C(F)F)CCC3)=O)CC12 38079,C(=O)(C(O)CC(C)(C)C)NCCCC(CCC)NC(C1CS(=O)(=O)C1)=O 38080,C(N=c1cc2c(c[nH]1)CCCC2)C1C(C(=O)O)C1.CC(C)(C)OC(=O)NC 38081,c1(C(=O)NC(C(C)(C)NC(C(CCSC)O)=O)C)ccc(C2=NOC(=O)C2)cc1 38082,CCCCC(N=c1cc[nH][nH]1)C(=O)N1CCNC(=O)C1 38083,N1(C(c2c(F)ncc(C)c2)=O)CC2CCC(CNC(C3CCNC(=O)C3)=O)C2C1 38084,C(=O)(C1CCCc2n[nH]cc21)NCC1(NC(=O)Cn2cccc2)CC(OC)C1 38085,c1(C(N2CCCC(N(C)C(c3cncs3)=O)CC2)=O)cc2cccc(F)c2s1 38086,c1(OCCOC)cccc(C(=O)NC(CNC(C2(Cl)CC2)=O)C2CC2)c1 38087,C1(NC(c2cc(-c3cccnc3)no2)=O)CC(F)CN(C(C2CCCSC2)=O)C1 38088,C=CCCCC(C)(C)C(=O)N1CC(CC(C)(C)CNC(=O)C(C2CC2)OCC)C1 38089,CS(=O)(=O)CCC(=O)NCC1CC(C(F)(F)F)CCN1C(C1CCC=CCC1)=O 38090,N1(C(C)=O)CCC2CN(C(=O)C(C)(C)c3cscc3Cl)CCC2C1 38091,c1(NC(C2C3(CCN(C(Cc4n(C)ncc4)=O)C3)C2)=O)nc2ccc(Cl)cc2[nH]1 38092,N1(C(C2N(C(C(C)C)=O)CCC2)=O)CCN(C(C2CCCS2)=O)C2(CC2)C1 38093,c1(C(C)(C)C(=O)NCCNC(=O)CC2CC2C2CC2)ccc(Cl)nc1 38094,Cc1cnnc(-c2ccc(CN3CC(C(=O)O)C(O)C3)c(F)c2)c1C 38095,Cn1nc2c(c1-c1c[nH]nc1C(=O)Nc1cc(O)ccc1Cl)CCC2 38096,C1(NC(=NC(NCC)=N)N(C)C)(C(=O)NC2(CO)CC2)CC2(CC(F)C2)C1 38097,CCCCC(F)C(=O)N1CCC1C(N1CCC(OC)C(F)C1)=O 38098,Cc1ccnc2c(C(=O)NCC(C)NC(C34CC(C)(C3)C4)=O)cnn12 38099,c1(OC)ccc2cc(C(=O)NC3CCCN(C(=O)C=CC(C)C)C3)sc2c1F 38100,c1(C(N(C2CCN(C(C3COCCO3)=O)CC2)CC)=O)cccnc1N 38101,c1(N2CCC(NC)CC2)ncnc(NC2CC(O)CN2CCC2CC2(Cl)Cl)c1C 38102,c1(CNC(=O)NCC(c2cccc(C)n2)CC)c(C)cc(C(=O)O)cc1C 38103,C(=O)(C1=NN2CCCN=C2N1)NCC(CN(C(C1(c2cccs2)CC1)=O)CC)(C)C 38104,C1(C(=O)NCC(C2CC2)SC)CC2(CCN1C(=O)C=C1CCC(C)CC1)CC2 38105,C1(C(=O)NC(c2cc(OC)c(F)cc2)C)CC2OC(C)CC2N1 38106,C(CC(=O)OC)(C(C)C)NC(CCc1n(NCC)nc(-c2ccc(F)cc2)n1)=O 38107,C1(NC(CN(C2CC(C#N)C2)C(=O)C=C(C2CC2)C2CC2)=O)CCn2nccc2C1 38108,N1(C(c2occ(C(=O)OC)c2)=O)CC2CC(NC(C3(N(C)C)CC3)=O)C1C2 38109,N1(C(CCCOC2(C)CN(C(C3(C#N)CCOC3)=O)C2)=O)CCc2cncnc2C1 38110,C1(NC(C(C2CN(C(COCCN(C)C)=O)C2)O)=O)CCN(C)CC1(C)C 38111,Cc1nn(C)cc1CCNC(C1CN(C(=O)CC2(O)CCCC2)CC1C)=O 38112,N1(C(C(=Cc2ccco2)C)=O)CC2(CC2)CC1CC(=O)NC(c1nc(C)no1)C 38113,C1(CCC)(NC(c2csnc2Cl)=O)CCN(C(c2cccc(O)n2)=O)CC1 38114,c1(-c2sc(C(N3CC(NC(C=C(C)C4CC4)=O)C3)=O)c(C)n2)c(C)nn(C)c1C 38115,c1(OC(CC)C)ccc(-c2nc(-c3cccnc3)nn2-c2ccnc(O)c2)cc1 38116,C1(C(N(CC(C)O)CCNC(=O)C(C2CC2)C2CC2)=O)CCc2nn[nH]c2C1 38117,c1(C(=O)NCC(CNC(CCN(C(CCC)C)C)=O)F)cc(O)cc(Cl)c1 38118,C1(C(C)C)COCCN1N1CCN(C(C)C)C(C2CC2)C1 38119,C1(OC)(OC)COC(CS(=O)(=O)Nc2ncccc2Br)C1 38120,Cc1ccc(C(C)NC(C2CC=CCN2C(c2cnn(C)c2Cl)=O)=O)cc1 38121,c1(CN2C(CC)CN(C(c3c(Cl)ccnc3Cl)=O)CC2)ccc2nc(O)[nH]c2c1 38122,C1(C)(C(=O)Nc2ccc(OC)c(Br)c2)CCCCNC1=O 38123,C(C(C)(C)S(C)(=O)=O)(c1nnnn1C(C)C)NCCSC.C(=O)(C1CC1)O 38124,c1(CC(=O)NC2CCN(C(c3onc(C)n3)=O)CC2C)oc2ccccc2c1C 38125,c1(C(=O)Nc2ccc(CC(=O)OCC)cc2)c(Br)cc(F)c(F)c1F 38126,CC(N=c1[nH]c2c(c(=NCCSC3CCOCC3)[nH]1)CCCCC2)c1ccco1 38127,CC1=NS(=O)(=O)NC=C1C(=O)NC1(CCCNC(C2(S(C)(=O)=O)CC2)=O)CC1 38128,C1(NC(c2c(C)noc2)=O)CC2CCC(C1C)N2c1ncccn1 38129,Cc1ccc2c(c1)CC(C(N1CC=CC(NC(=O)C(C)(Cl)Cl)C1)=O)S2(=O)=O 38130,C(=O)(CCCC(C)NC(=O)C(C1CCCCC1)F)NC(C(=O)OC)CO 38131,c1(C(=O)NCC2C3CN(C(C(C)n4cccc4)=O)C2C3)cc([N+](=O)[O-])ccc1Cl 38132,Cc1cn2c(C(=O)NCC3CCCCN3C(=O)CCC(N)=O)cnc2s1 38133,c1(CNC(=O)Nc2c(C)cncn2)ccnc2ccccc12 38134,Cc1ccc(N2CCC2)c(C(=O)NC2CCC2NC(=O)C(C)n2cncn2)c1 38135,N(C1CCc2sc(Br)cc21)C(=O)OC(C)(C)C.c12cccc(c1)CNC(=O)N2 38136,C1(CC)CCCCC1N(C(=O)C(=O)Nc1cncc(Oc2ccccc2)c1)C 38137,C1(CC(=O)NCCCCC2C(C)C2)CCCN(C(c2nonc2N)=O)C1 38138,C1(C(=O)NC(C)(C)CC(=O)NC2CCS(=O)(=O)C2)CC2(CCC2O)C1 38139,C1(O)(CNC(CC(=O)OC)=O)CCN(C(=O)C(C)Sc2ccccn2)C1 38140,C1(NC(CCC2(C#N)CCC2)=O)CN(C(C2CC(=O)CCO2)=O)CC(F)(F)C1 38141,C1(CNC(c2cnsc2)=O)CC2CN(C(C3(c4cccnc4)CC3)=O)CC12 38142,S(=O)(=O)(c1cnn2ccc(=NC(CO)C3CCC(F)(F)CC3)[nH]c12)NCCCC 38143,CCC(CC(=O)N1CC(N(C(=O)COCC2CCCO2)C)C1)C(C)(C)C 38144,N1(C(C(c2ccc(Cl)cc2)C)=O)CC(C)(C)CC1CNC(C1CC1F)=O 38145,N1(c2nnc(C(=O)NCC(C)(C)C)n2CCC#N)CC2(CCSCC2)C1 38146,C1(C(N(C(C)CCNC(C23CC(C#N)(C2)C3)=O)C)=O)CC(=O)C12CCC2 38147,N1(C(CCC#C)=O)C(C(=O)Nc2ncncc2I)CC2CCCCC12 38148,CC(C)(C)CCC(F)C(=O)N1CCCC(F)(CNC(=O)CCn2cncn2)C1 38149,C1(C(=O)NCC2N(C(C3CN(S(CC)(=O)=O)C3)=O)CC2)CCCC1OC 38150,C12(NC(C3N(C)CCOC3)=O)CCCC1CN(C(c1cc[nH]n1)=O)C2 38151,C1(NC(=O)NCCC(CC)C)CCCN(C(=O)OC(C)(C)C)C1c1cnn(C)c1 38152,C1(C(N2CC3CC(C2)O3)=O)CC2CC2N1C(C1CCNC(=O)C1)=O 38153,C1(CN(C(c2c(CC)cc[nH]2)=O)C)CCC(NC(C2CC=CCC2C)=O)CC1 38154,N1(CCC)CCCC(C(N2CCC(N(C(=O)C(F)OC)C)CC2)=O)C1 38155,c1(C(=O)NCCN(C)C(c2ccc(N3CCCC3)nc2)C2CC2)cccc(=O)o1 38156,c1(CNC(c2ccn(CCC)n2)=O)nnn(C)c1C(=O)N(CC(C)O)CC 38157,C1(C(N2C(C)(C(NOC(C=C)C)=O)C=CC2)=O)CC2CC(=O)C1C2 38158,C(=O)(C(CO)NC(=O)C=CC1CC1)NCC(C)(O)C1CC1 38159,c1(CCCCC)cc(C(=O)NCC23CC(NC(c4cnc(C)o4)=O)(C2)C3)n[nH]1 38160,c1(C(=O)NCc2cn(C3(C(N)=O)CC3)nn2)ccc2c(c1)CCCS2(=O)=O 38161,C1(C(=O)NCC=CC(=O)NCC2(CO)CCCCO2)(OC)CCOCC1 38162,CCCCC(CC)CC(=O)NCC(C)(C)C(=O)NCCS(C)(=O)=O 38163,C1(NC(=O)CN2C(=O)CCC2=O)CCCCN(C(C2CN3CCN2CC3)=O)C1 38164,Cn1nc(C(F)(F)F)c([N+](=O)[O-])c1N1C2CCC1C(NC(c1ccsn1)=O)C2 38165,c1(C(=O)NC2C3(CN(C(C4(C=C)CC4)=O)C3)CCC2)ccc2c(n1)OCC(=O)N2 38166,N1(CC(CCC)OC)CCCC(c2nn[nH]n2)(C(C)C)C1 38167,c1(CC(N2CC(C)C(NC(=O)Cc3nc[nH]n3)CC2)=O)c(F)ccc(Br)c1F 38168,N1(C(c2snc(C)c2N)=O)CCCC(CC(=O)N(CC(C)(O)C2CC2)C)CC1 38169,c1(CN2CC(N)C2)cn2cccnc2n1.C12CN(CCO1)C2=O 38170,C1(CNC(c2cc(C)oc2)=O)CN(C(=O)CSC(C)(C)C)CCC1C 38171,c1(SCCC)cccc(C(=O)NCC(O)CNC(=O)C(C)Sc2cccs2)c1 38172,c1(CNC(C2(CC)CN(C(=O)Cc3nonc3C)C2)=O)nc(C)c(C)s1 38173,C1(F)(CNC(CN(C)C(N)=O)=O)CCCN(C(=O)C(F)Cc2ccccc2)CC1 38174,CC(C)(C#N)CCC(=O)N1CCC(NC(=O)CSc2nc[nH]n2)C(F)C1 38175,CC1(C)CCCN(C(c2ccc(N)c(F)c2)=O)C1CNC(=O)C#CC1CCC1 38176,C1(NC(C2CCC(CC)O2)=O)CCC(N(C(=O)CC2CSC2)C)CC1 38177,Cn1cc(C#CCNC(C2CC(C)(C)CCN2C(=O)CP(C)(C)=O)=O)cn1 38178,CC1CCCCC1C(=O)NCC(CO)Nc1nccc(C(F)(F)F)n1 38179,c1(CNC(=O)COCCCF)ccc2c(c1)CN(C(c1cc(CO)ccn1)=O)C2 38180,C1(NC(C(CC=CC)C)=O)CCCOC12CCN(C(=O)Cc1cc(C)on1)CC2 38181,C1(C(=O)OC)(NC(C2CCCC23OCCO3)=O)COc2ccccc2C1 38182,c1(CNc2c(C(=O)OC)cc(C)c(C)c2)ccc2c(c1)C(CCOC)C(=O)N2 38183,c1(N(CCCOCCNC(c2cnn(C(C)C)c2F)=O)C)ncccc1C#N 38184,CC1CN(C(=O)CCSCc2ccccn2)CCC1NC(=O)C=Cc1cc[nH]c1 38185,c1(-c2n(C(c3cccc(F)c3)C)nc(Cc3ccccc3)n2)cc2ccncc2s1 38186,c1(N(C(CN2CCCC(COC)C2)=O)CC2CC2)cc(S(N)(=O)=O)cnc1C 38187,C1(C(=O)NOCCO)(CC=C)CCCN1C(C1CCC(F)CC1)=O 38188,c1(C(N(CCC(C(C)C)NC(=O)C=CBr)C)=O)ccc2c(n1)CCO2 38189,CCC(CC)CC(F)C(=O)N1CCC2CCCC12C(=O)NC(C)C1CC1 38190,c1(C(N(CCCCCN(C(C=CCOC)=O)C)C)=O)c(OC(C)C)ccnc1F 38191,N1(C(C(C=C)CC)=O)CCOC2(CCN(C(=O)Cc3ccco3)C2)C1 38192,C(=O)(C(F)(CNC(=O)C(C)(C)C(C)(F)F)C(C)C)NC(C#C)CC1CCCC1 38193,C(=O)(C(O)C(O)c1ccccc1)N(CCCCNC(C(=O)N(C)C)=O)C 38194,N1(C(C(c2ccc(F)cc2)C)=O)CCC(NC(c2occc2CN(C)C)=O)CC1 38195,C1(C(N2CCC3CC23)=O)COCCC1NC(C12CCN(CC1)C2)=O 38196,CCC(O)C(C)C(=O)N1CCN(C(C2CCCC2C(=O)OC)=O)CC1C1CC1 38197,c1(C(N2C(C)(CNC(=O)C=CC3CC3)CCC2)=O)occ2c1CCOC2 38198,c1(NC(C2C(C(N3CC4C(C(=O)OC)(C4)C3)=O)C2)=O)cncc(F)c1I 38199,c1(CC)cccnc1C(=O)N(CC(C)NC(c1ccc(-c2cccs2)[nH]1)=O)C 38200,C=C(C)C1OCCC1Cc1ccc(NC(=O)C(=O)Nc2cccc(Br)c2Cl)cc1 38201,CCC(C(=O)NCC1(NC(C2CCCC2O)=O)CCCC1)OC1CCCCC1 38202,c1(-c2cn(C3CN(C(C(C)c4cccs4)=O)CC3O)nn2)nsc2ccccc12 38203,c1(SC)cc(C(N2CC3CC2CN3C(c2cn[nH]c2)=O)=O)cc(SC)c1 38204,C1(CC)CN(C(C2(C)CC3CC3C2)=O)CC1NC(c1cccc(C(=O)OC)c1)=O 38205,C1(C(N(CCNC(c2c(C)nn(CC(F)F)c2C)=O)C)=O)CC2(C1)CC1(CC1)C2 38206,c1(CC(N2CC(=C(CNC(CC(=O)NCC)=O)F)C2)=O)coc2ccccc12 38207,c1(CN2CCC(C)(C(=O)NC(CC)C)C2)cc2ccccc2s1 38208,N1(C(C(c2ccccc2)C)=O)CC2CCC(CNC(=O)Cc3cc[nH]c3)(C2)C1 38209,c1(C(=O)NCCNC(C(C(C)(C)O)NC(=O)OC(C)(C)C)=O)cnc2[nH]ccnc1-2 38210,c1(C(C)=O)cccc(CC(=O)NCCC2CCN(C(=O)C=C3CCC(C)C3)C2)c1 38211,C(=O)(CCCNC(C)=O)NCC(COC)NC(=O)C(CC1CCC1)OC 38212,c1(N2CCN(C(C)=O)CC2)nc(N2CCC(C3CCCO3)C2)c2sccc2n1 38213,C(=O)(CC(C)C(C)C(C)C)NCC1(F)CC(NC(c2nnc(C)s2)=O)C1 38214,C1(CNC(CSC)=O)CN(C(c2cccc(N)c2N)=O)CCC1(F)F 38215,N1(C(=O)COCCF)CCC2CN(C(=O)COCCc3ccc(Cl)cc3)C2C1 38216,C12CCN(CC1)Nc1cnn2c1.C1(CN(C)C)CCCCC1C(=O)O 38217,N1(C(C(C)(C)C#N)=O)CCC(F)(F)C(CNC(C2(C)CNC(=O)C2)=O)C1 38218,N1(C(C=CC)=O)CCOC2(CCC(NC(C3CCCC(C(F)(F)F)C3)=O)CC2)C1 38219,c1(C(=O)NCC2N(C(CC(=O)OC)=O)CCN(C)C2)ccccc1N=S(C)(C)=O 38220,C1(C(N2C(C)(CNC(C(C)CSC(F)(F)F)=O)CCC2)=O)CCc2nn[nH]c2C1 38221,CC(CC(=O)NC(C)(C)CCN(C(=O)CC(C)n1ccnc1)C)c1ccccc1 38222,C1(CC)(CO)CCCN1C(C1C=CCN(C(=O)C(N2CCOC2=O)C)C1)=O 38223,c1(C(N2C(C(C(=O)NC3CC4(CN(C)C4)C3)(C)C)CCC2)=O)ccn2cncc2c1 38224,c1(OCC)cc(NC(c2ccc(-c3cn[nH]c3)cc2)C)cc(Br)c1 38225,C12(C(=O)NCC(=C)CCNC(C3COC(=O)N3C)=O)CC(CO)(C1)OC2(C)C 38226,C1(C(=O)NCC2(COC)CCCN2C(=O)CN=S(C)(C)=O)COC2(CCC2)C1 38227,c1(C(N(CCNC(C(CC)CC(F)F)=O)C2CC2)=O)ccc2c(c1)CCCC2=O 38228,c1(CCC)c(C(=O)NCC2(NC(=O)CCn3ccnc3C)CCOC2)cnn1C 38229,N1(C(C2(CO)CCN(C(CCCC#CC)=O)C2)=O)CCC2(CCOC2)C1 38230,CC1(C)COC(C(N2CCC(C)(NC(=O)CC3C=CS(=O)(=O)C3)C2)=O)C1 38231,C(=O)(C1CCc2cccc(=O)n21)NC1C(OC)CN(C(C2(C(=O)OC)CC2)=O)C1 38232,C(=O)(C(F)CC(C)(C)C)NCC1(NC(Cc2ccc(CCC)cc2)=O)CCCC1 38233,c1(C(=O)OC(C)(C)C)cccc(CNC(N2C(C)(CCC)CC2)=O)n1 38234,C(=O)(C(C(C)(C)C)OC(C)(C)C)N(C)CC1CCN(C(C2(C(N)=O)CCC2)=O)C1 38235,N1(CC)C(=O)CCC1C(=O)NC(C1CCCC1)CNC(=O)C(=C1CCCCC1)F 38236,C(C1CCN(C(C2CCC3(CCC3)C2)=O)CC1)=CC(=O)NC(CCC=C)C 38237,N1(C(c2c(NC(N)=O)cccc2)=O)CC2(CCN(C(c3cc(CO)[nH]n3)=O)C2)C1 38238,c1(OC)cccn2ncc(C(=O)NC3CC(NC(=O)C=CBr)C34CCC4)c12 38239,C1(CNC(CCCc2ncc(C)o2)=O)CC(NC(=O)CNC=O)C12CCC2 38240,Cn1cc(C(=O)NCC(CO)NC(=O)C2=CCSC2)ncc1=O 38241,CCC(C)CCCCC(=O)N1CCCC1CNC(=O)CCCCc1ccccc1 38242,C1(NC(C(CCC)CC2CC2)=O)COC2(C1)CN(Cc1cncs1)C2 38243,Cc1cc(C(=O)NCC2(NC(=O)C=Cc3ccc(=N)[nH]c3)CC2)c2c(c1)CCC2 38244,Cc1cc(F)ccc1CC(N1CCC(CF)(NC(=O)Cc2c(C)cnn2C)C1)=O 38245,Cc1ccnc(O)c1C(=O)NC(CNC(c1ccnn1CC(F)F)=O)C1CC1 38246,C(=O)(C(CC)(CC)CC)N1CCC(CC(=O)NC(C(=O)OCC)CO)C1 38247,C1(NC(=O)C(F)C2CCC2)CN(C(=O)CN2CCCCC2=O)CC12CC2 38248,N1(C(CC2N(CC)CCC2)=O)CCN(C(=O)C=C2CCCC2)C2CS(=O)(=O)CC12 38249,c1(OCC)ccc(Cl)c(C(=O)NCCOCCCNC(c2cc(O)n(C)n2)=O)n1 38250,C1(C(=O)NCCC(C)NC(c2cccc(-n3cccc3)n2)=O)CC=CCC1C 38251,c1(N2CCC(N(C)C)CC2)nc(=NCC2CC2Cl)[nH]c2c1SCC2.C(=O)C(C)(C)C 38252,CCC(C(=O)NCC(C)CNC(=O)Cc1cccc(OC)c1F)C(F)(F)F 38253,C1(C(F)(F)F)(OC)CCCN(CC2CCC(C#N)CC2)C1 38254,CC1(C)CC(CN2CC(c3cc(Br)sn3)C2)CN(C(=O)OCc2ccccc2)C1 38255,CCCCCS(=O)(=O)CC(=O)N1CC2CC2(NC(c2cc(F)c(N)c(F)c2)=O)C1 38256,CCC(C(=O)NC(CO)C(=O)NCCCCO)n1ccnc1 38257,Cc1cc(O)c(C(N2CCCC(C(C)NC(=O)Cn3nccc3C)C2)=O)cc1F 38258,c1(NC2CN(C(C(C)C)=O)CC2C)ncccc1S(C)(=O)=O 38259,c1(C(N(C(C)CNC(=O)CC2CC(F)C2)C)=O)c[nH]nc1Cl 38260,C1(NC(CC2CC(=C)C2)=O)CC(F)CN(C(=O)Cn2cccc(C)c2=O)C1 38261,C#CCC(C)(C(=O)NC(CC1CC1)CO)NC(c1ncn(C(C)C)n1)=O 38262,N1(C(C(C)Cc2ccccc2)=O)CC2(CCC2)C1c1cccnc1 38263,C1(NC(C(CC=CCC)C)=O)CCN(C(=O)CC2CN3CCC2CC3)CC1O 38264,c1(C(=O)NCCOC2CN(C(c3nn(CC)c(C)c3)=O)C2)sc(C)c(C)c1C 38265,c1(C(=O)NC2(C)CN(C(C3(C)CCCS3(=O)=O)=O)C2)ccc(F)c(C(F)F)c1 38266,C=CC1OCCC1C(N1CCC(CCN(C(=O)CC(O)CN(C)C)C)CC1)=O 38267,N1(C(C2C(C3C(C)C3)C2)=O)CCC(O)(CN(C)C(c2cn3ccsc3n2)=O)CC1 38268,C12(NC(CC3(NC(C)=O)CC3)=O)CCCC1CN(C(=O)Cc1c(C)cccc1Cl)C2 38269,c1(C(=O)NCCC(C)(C)NC(=O)C(O)CCS(C)=O)nnc(O)c2ccccc12 38270,c1(C(=O)NC(C(=O)NC(CC)CCCO)c2ccoc2)c[nH]c(C)cc1=O 38271,Cc1cc(F)sc1C(=O)NC(C(=O)N(C)Cc1cccnc1O)C1(O)CCC1 38272,N1(C(C2(C(C)C)CCC2)=O)CC2CC1CN2C(C1CC1(F)Cl)=O 38273,N1(C(C(OC)OC)=O)C2CCC1CC(NC(C1CCNC(=O)C1)=O)C2 38274,CC1CCN(C(=O)CC2CCC2(F)F)CCN1C(c1noc2c1CCCC2)=O 38275,n1(CC(N2C3CCN(C(C4(COC)CC4)=O)CC3C2)=O)c(C)nc2ccccc12 38276,Cc1ccc(C(=O)NC2(CNC(C3CC3c3cnn(C)c3)=O)CC2)c(C)c1Br 38277,c1(CCC(=O)NCCCNC(c2nc(OC)oc2)=O)ccc(O)nc1 38278,Cc1oc2ccccc2c1C(N1CCN(C(=O)CCC2CCCOC2)C(C)C1)=O 38279,C1(C(N2CCC(O)(Cn3cc(C4CCCC4O)nn3)C2)=O)CCCC2(CCC2)O1 38280,N1(C(C23CCC(C(=O)OC)(C2)C3)=O)CCC2CCCN(C(C3(C)CCC3)=O)C2C1 38281,N1(C(C2(C3(C)CC3)CC2)=O)CCOCC(C(=O)NCCN2CCC3CC23)C1 38282,C(=O)(C1=CCCCC1C)NC(CC=CC)C(=O)Nc1cc(Cl)ccc1C 38283,CCCC(C)(CCC)C(=O)NCCCNC(=O)C(C)OCC1CCCCO1 38284,C1(N=[N+]=[N-])(C(=O)NCC(CCC)(C)C)CCN(C(C2CCOC2(C)C)=O)C1 38285,c1(C(=O)NCC2CC(NC(C3(N(C)C)CCC3)=O)C2(C)C)ccc2c(c1)OCO2 38286,c1(CC(N2CC(OCCNC(C(CSC)O)=O)C2)=O)ccc(Cl)cc1C 38287,N1(C(c2cncc(N)c2)=O)CC2CCC1C1CN(C(c3cnc(O)o3)=O)CC21 38288,c1(C(CC)C(=O)N(CCCN2CCCC2)C)ccc2c(c1)OCO2 38289,Cc1conc1C(=O)NCC1CN(C(c2cnn(C(C)C)n2)=O)C1 38290,C1(C(=O)NCC2(C(C)(C)O)CN(C(CSCC=C)=O)C2)CCCCCC1(F)F 38291,CC(C(C)(C)C(=O)NCCn1cccnc1=O)NC(c1cnc2n1CCC2)=O 38292,C1(C(=O)NCc2c(CC)cncc2)CCCN1NC(=O)C(F)C(F)(F)F 38293,C1(C)(C(=O)NC)CCCN1C(c1cn(CCNC(=O)CC2(C#N)CC2)cn1)=O 38294,C(C(F)(F)C(F)(F)F)OCC(=O)N(CCCNC(=O)CC1CC1C)C 38295,C=CC(C)(CC)C(=O)NCCC1(C(=O)NC2(c3ccccc3)CCC2)CC1 38296,n1(CCOC)ccc2cc(NC(c3cccc4c3COC4)=O)ccc12 38297,c1(CC)cccnc1C(N1CC(NC(=O)C=Cc2nc(C)cs2)C(C)C1)=O 38298,Cc1csc(C)c1C(=O)NC1CCOCC1C(=O)NCCCn1ccnc1 38299,n1(C(C(=O)OCC)C)nnnc1C(c1nocc1CC)NC(C)CC1CCCO1 38300,C1(C(N(CC(=O)NC(C)C)C)=O)CN(C(c2cccn2C)=O)CC1(F)F 38301,c1(C(=O)OCc2cccnn2)nc(Br)sc1Cl 38302,c1(C(=O)NCC(CC)NC(C2(C3CC3)CCCO2)=O)[nH]c2ccc(C)cc2c1C 38303,C#Cc1ccc(OCC(=O)NCC(CO)NC(c2ccc(Cl)cn2)=O)cc1 38304,C1(CC(=O)NCCN(C2CCCCCC2)C(=O)C=C2CCC2)CCS(=O)(=O)C1 38305,C1(OC)CN(C(=O)CN2CSCCSC2)CC1NC(=O)CCn1ccnc1C 38306,N1(C(c2c(C)csc2)=O)CCCCC1CNC(c1ccc(-c2ccco2)s1)=O 38307,N1(C(C(CC=C)C)=O)CC(NC(=O)C(CC(=C)C)NC(C)=O)C(C)(C)C1 38308,Cc1n[nH]cc1C(C(=O)NC(C)C)N(C)CCC1CCCCC1 38309,C1(C(=O)NCC2(C)CC2(F)Cl)(COCC=C)CCCNC1 38310,C1(CNC(C(=O)N(C)Cc2ccn(CC)n2)=O)C2CCCCCC12 38311,N1(C(CC(CCC)C)=O)CC2CC(C1)N(C(=O)COCC1CCOCC1)C2 38312,C1(NC(c2c(C)onc2)=O)CC2CC(C1)N(CC(=O)NCC1CCOC1=O)C2 38313,N1(C(C(=O)N(C2C(C)OCC2)CCO)=O)CCN(S(=O)(=O)N2CCCC2)CC1 38314,C1(C(=O)NCC(CN(C)C(C2(C(F)F)CC2)=O)O)CCC=CCCC1 38315,C1(C(=O)OC)C(O)C(O)CCN1C(=O)NCc1ncc(OC)cn1 38316,CC1(C)CC(C(=O)NCCCCCC(=O)NC2CCCSC2)CCO1 38317,c1(CC)ccc(F)cc1NC(C1CC(NC(=O)Cc2ccc(O)nc2)C1(C)C)=O 38318,Cc1cc(C)c(C(=O)NC2CCC(CNC(c3cc(CO)[nH]n3)=O)CC2)cn1 38319,c1(C(=O)NCC(C=C)O)nc(CNC(=O)CN(C)C(C)=O)oc1C 38320,c1(C(N2CC(OC)C(NC(=O)C(CO)NC(N)=O)C2)=O)c(C)oc(C)c1Br 38321,c1(C(=O)NCCCCNC(c2c(SC)cccc2F)=O)ncnc2ccsc12 38322,n1(CC(C(N2CC(CNC(c3n(C=C)nnc3)=O)C2)=O)C)nnc2ccccc12 38323,C(CCCCC(=O)N1CC=CC1C(=O)NCCN1CCCCCC1)=CC 38324,CCCC(C(=O)N1CCCC(N(C(=O)C(C)OCC(C)C)CC)C1)N(C)C 38325,CC1(C)CC(C(F)(F)F)(C(=O)NCC2CCC2NC(=O)CSc2ccccn2)C1 38326,N#Cc1n[nH]c(=NC2CCCC23CN(C(C2CCCC(F)(F)CC2)=O)C3)s1 38327,CC1CC(CCC(=O)O)CCN1C(=O)Nc1ccnn1C 38328,C1(C(N2CCC(OC)C2C(C)C)=O)COC2(C1)CN(C(c1cccc(=O)o1)=O)C2 38329,C(=O)(C(C)CCCC(C)C)NC(CNC(C(=Cc1cn[nH]c1)C)=O)CO 38330,N1(C(C2COC(=O)O2)=O)CC23CCCC2(C1)CN(C(c1cnc(O)s1)=O)C3 38331,C1(CNC(c2cc(NC(C)=O)c(C)cc2)=O)CCN(C(=O)C(C)S)CCC1(F)F 38332,N(C1COc2c(Cl)cccc21)C(N(C)Cc1ccccc1I)=O 38333,C12(CNC(C3CCC(C)O3)=O)CCCC1N(c1ncc(C(C)(C)O)cn1)CCC2 38334,c1(C(=O)Nc2cc(C)cc(O)c2)cn(C)c2ccc(-c3cccc(F)c3C)cc12 38335,CC1CN2CCN1CC2C(N1CC(NC(C2NC(=O)C3CCC23)=O)C(C)(C)C1)=O 38336,CC1(C)CCN(C(=O)CC2(C#N)CC2)CC1C(=O)NCC1CC(O)C(O)C1 38337,C1(CNC(C2C(C)CCC2)=O)CCCN(C(=O)CC(C)(C)O)CC1 38338,C1(COC)(CNC(=O)CSc2cccs2)CN(C(=O)CC2CCCCO2)C1 38339,N1(CC)C(=O)CCC1CC(=O)NCc1nc(CNC(C2COCC2(C)C)=O)cs1 38340,C1(C(C)NCc2onc(C)n2)CCCN(c2ccccc2)C1=O 38341,N1(C(c2sc(C(F)(F)F)nc2-c2ccccc2)=O)CCS(=O)C(F)(F)C1 38342,c1(NC(C2CN(C(N(C)C)=O)C2)=O)nc(Cl)c(Cl)nc1Cl 38343,C(C(C)C(F)C(=O)NC12CC(C1)C2)NC(c1c(C(C)C)occ1)=O 38344,C1(CCOC)(NC(=O)C(c2ccccc2)F)CCN(C(=O)OCC)CC1 38345,C(=O)(NNC(=O)C(CN)CC(C)C)c1c(C)nc(-c2ccc(Br)cc2)s1 38346,N1(C(C(CC(C)(C)C)NC(c2cnn(CC)c2C)=O)=O)CC(C)C12CCOCC2 38347,Cc1nc(C(C(=O)NCc2ccc(F)cc2)N(C2CC2(C)C)C)sc1C 38348,c1(CCNC(C(C2CCN(C(c3ccn(C)n3)=O)C2)(C)C)=O)ccc(F)cc1 38349,CC1CN(C)CC(C(N2CCCN(C(=O)CN3C(=O)CNC3=O)CC2)=O)O1 38350,C1(OC)CC(CNC(c2cccnc2)=O)N(C(=O)CC(F)(F)Cl)C1 38351,c1(C(N(CCN(C(CCc2cnc(C)s2)=O)C(C)C)C)=O)ccccc1N(C)C 38352,C1(CNC(=O)OC(C)(C)C)(CC2CC2)CCSCC1.C12CN(C1)C(=O)N2C 38353,c1(CC(=O)NC(C2CC=CCC2)C(=O)NCC(C(C)O)O)ccccc1F 38354,C(=O)(C(C)C(O)CC)NCC1CCC(C(=O)NC2(CC=C)CCCCC2)CC1 38355,c1(CCC(=O)N(CC(C)CNC(=O)Cc2ccon2)C)ccc(O)c(Cl)c1 38356,C(C1=CCN(C(c2ccsn2)=O)CC1)NC(c1cn(C2COC2)nn1)=O 38357,C1(CNC(N2CCCN(c3nccs3)CC2)=O)CC2CCCCCC12 38358,C1(NC(c2cc(CCC)ncc2)=O)CCN(C(c2sccc2F)=O)CC1CO 38359,CC1(C)CC(=O)N(CC(=O)NC2C=CCN(C(c3cccc(Cl)n3)=O)C2)C1=O 38360,c1(C(=O)OC)cccc(NC(=O)NCc2ccncc2C(C)C)c1OC 38361,C=CC1CN(C(=O)C(c2cscc2Br)=O)CC1NC(=O)C(C(C)C)SC 38362,C1(C(=O)NCC(CC=C)(F)F)CC2CCC(C1)N2C(=O)C(C)(C)C(=O)OCC.O 38363,c1(C(N(C2CCCCC2NC(C2(C)COC2)=O)C)=O)ccc2c(c1)OC(C)(C)C2 38364,N1(C(C2CCC2C2CC(=C)C2)=O)CC2CCC2(Cc2cc(SCC)cc(F)c2)C1 38365,c12ccc(cc1)[nH]c2=O.c1(C(N2CC(N(C)C(N)=O)C2)=O)cnc(O)[nH]1 38366,C1(NC(c2c(CC)cco2)=O)CCN(C(C2(C)CCCN2C)=O)CC1O 38367,Cc1c(NCc2n[nH]c(=N)o2)ncnc1N1CCN(c2ncccc2F)CC1 38368,C1(C)(C(N(CCCNC(c2c(C(=O)OC)cco2)=O)C)=O)CCOC1C 38369,c1(C(N2CCC(O)(CCNC(C(COC)(C)OC)=O)C2)=O)cc(C)c(C)c(C)c1 38370,C1(NC(c2ccc(CCO)cc2)=O)CN(C(=O)C2=CCC2)C2(CCOCC2)C1 38371,C1(NC(C(CC=C)CNC(=O)C=C(C)C(F)F)=O)CC2CC1CC21CC1 38372,C1(NC(C2(C)N(C(c3ccc(N(C)C)c(F)c3)=O)CC2)=O)CCc2n[nH]cc2C1 38373,N1(C(c2ccc(CC)cn2)C(=O)NC(C)C)CCC(C2CCOC2)C1 38374,c1(C(N2CCC(N(C(c3ncc[nH]c3=O)=O)CC)C2)=O)cc2c(ccn2C)[nH]1 38375,C1(CC(=O)Nc2ccc(Cl)cc2)CCN(S(=O)(=O)CC2CC2CC(=O)O)C1(C)C 38376,c1(C(=O)NCCN(C(=O)Cc2cc(Cl)ccc2O)CC)cnc2ncccc2c1 38377,C1(C(=O)OC(c2onc(CC(C)C)n2)C)CCN(C(=O)NC(C)C)CC1 38378,N1(C(c2c(CC)nns2)=O)CCN(C(=O)Cc2ccc(C)c(C)c2)CC1C(C)C 38379,N1(C(C(CC)=CC)=O)CCC(CNC(=O)CCc2ccc(OC)c(Cl)c2)C(C)C1 38380,c1(C(N2CC(C)(C(=O)Nc3cncc(C(C)(C)C)c3)C2)=O)ccc(Br)nc1Br 38381,c1(C(N2CCCC(N(C)Cc3cc(C)no3)C2)=O)n[nH]c(C)c1[N+](=O)[O-] 38382,c1(C(N2C3CC(NC(c4n(CC)nnc4)=O)C2CC3)=O)cccc2c1OCCO2 38383,N1(C(c2ncn(CC)c2)=O)C2CCC1CC(CNC(=O)C(=Cc1cscn1)F)C2 38384,CCCCCCCCC(C)CC(=O)NC1CC(CNC(=O)C(F)(F)C(F)(F)F)C1 38385,C1(CNC(COC)=O)CN(C(=O)CC2CC(C)(C)OC2=O)C2CCCC2O1 38386,N1(C(c2c(C)nc(N(C)C)s2)=O)CCCC12CCCN(C(=O)C(O)C1CC1)C2 38387,c1(OC)ccc(OC)c(C(N2CCC(C)(CNC(C3(C)CC(C)(C)C3)=O)C2)=O)n1 38388,c1(C(=O)NCCC(C)N(C(=O)C(O)CC(N)=O)C)cccc(S(=O)(=O)C2CC2)c1 38389,c1(C(=O)NCCCOCCNC(c2c(C)nncc2)=O)nc(=O)cc(N)[nH]1 38390,C1(CNC(c2nc(CCC)sc2)=O)C(O)C(O)CN1C(C1CCCCS1(=O)=O)=O 38391,C1(NC(=O)CCOCCN(C)C)CCN(C(=O)CCC2CCC(O)CC2)CC1F 38392,c1(C(N2CCCC(=C)C2)C(=O)NCCOC)cccc(F)c1I 38393,C1(C(=O)NC(C#C)(C)C)(NC(=O)C(C)=C(C)CCC)CCN(C)C1 38394,C(=O)(CC(C1CC1)C1CC1)NC(CN(C(C(=O)NCC)=O)C)CC 38395,CC1(CNC(c2coc(Cl)n2)=O)COCCN(C(c2ccnc(O)c2)=O)C1 38396,Cc1cccc(C)c1CC(=O)NC1CC2(C1)CC(NC(C1(F)C3CCCC13)=O)C2 38397,c1(C(=O)Nc2cc(O)n[nH]2)cnc2n[nH]c(-c3cccnc3C3CC3)c2c1 38398,N1(C(C(CC#C)C)=O)CC2CCC2(CNC(=O)CCOc2ccc(OC)cc2)C1 38399,c1(C(=O)NC2(C)CCN(C(C3C(C)(CC)C3)=O)C2)ncc([N+](=O)[O-])n1C 38400,Cc1c(C(=O)NC2CC3CCC2N3c2cc(OC3CC3)ncn2)cncc1Cl 38401,C=CCC(CC(=O)NCc1ncoc1C1CC1)NC(=O)C(CCC)N(C)C 38402,C1(N(C(c2cccc(Br)c2)=O)CC)CN(C(=O)CN2CCC2C)C(C)(C)C1 38403,c1(C(C)NC2(C)CCC(=O)NC2=O)cccc(S(=O)(=O)C(=O)N(C)C)c1 38404,c1(C(N2CCN(C(C(C(CC)C)O)=O)C(CO)C2)=O)cc(C)c2[nH]nnc2c1 38405,c1(C(=O)NCCN(C(C2(N(C)CC)CC2)=O)C)c(Cl)nc2sc(C)cn12 38406,C1(CCN(C(CC=C)=O)C)CCCCN1C(c1nc(CC(F)(F)F)sc1C)=O 38407,N1(C(CC2C3CN(CC(=O)NCC4(C)CCCC4O)CC32)=O)CCn2cncc2C1 38408,c1(C(=O)NC2CC(CCNC(c3csc(C4CC4)n3)=O)C2)ccc2c(c1)CCN2 38409,C1(NC(CC(C)N(C)C)=O)CC2CCC1CN2C(=O)CCCCC1CC1 38410,C1(CC(=O)NCC(O)CF)C2CCCC2N1C(=O)CC1CC2(CCC2)CO1 38411,C1(NC(CCCC=C)=O)CCC2(CC1)CC2NC(c1c(SC)cnn1C)=O 38412,n1(CC(=O)NC(C2CCN(C(C3CN(C(=O)C4CC4)C3)=O)C2)(C)C)cc(Cl)cn1 38413,C1(C(=O)NC2CCC(C)N(C(=O)CCc3cnn[nH]3)C2)CCCC2CCCN12 38414,C=C(C)CCC(C(=O)Nc1ccc2c(c1)OCO2)N1C2CCC1CC(O)C2 38415,CC1COC(C(=O)NCc2csc(CNC(C3(CF)CC3)=O)n2)C1 38416,CCN=c1ccc(C(=O)NCC2(F)CCC(CNC(=O)CC3CC3)C2)c[nH]1 38417,c1(C(=O)NCCCn2cc(C(C)(C)C)nn2)ccc(CO)cc1F 38418,c1(C(N2CCC(CNC(C(C=C)O)=O)CC2C)=O)c[nH]c2c(F)cccc12 38419,O=S(=O)(CCCCC1CC1)NC1(c2cccc(F)c2)CCCCC1 38420,N1(C(Cc2ncc(C)s2)=O)CC2CC(NC(c3cn(C)nc3C(F)(F)F)=O)C2C1 38421,CC1=C(C(=O)N2CCC(C)(NC(C3CC4CC4C3)=O)C2)CCCO1 38422,c1(C(=O)NC2C(CNC(CC(=O)NCC)=O)CC2)ccc(-c2cccnc2)cn1 38423,c1(CC)oc(C(=O)NCCC2(O)CN(C(=O)CCC(C)OC)C2)cc1C(=O)OC 38424,c1(C(=O)NC2(CCOC)CCN(C(c3cnncc3O)=O)C2)c[nH]cc(C)c1=O 38425,Cc1cc(F)ccc1-n1cc(O)c(C(=O)OCC2C=CCC2)n1 38426,c1(NC(C2CCN(C(c3c(I)ccnc3F)=O)C2)=O)ccc(Br)cc1Cl 38427,CC1CCC(C)(C(=O)NC2CCCCC2NC(=O)CC2COCCO2)C1(C)C 38428,c1(CNC(C2CCC3(CN(C(CCC(C)C)=O)C3)O2)=O)ccc2ncccc2c1 38429,c1(C(N2CCC(CNC(C3(C#N)CCCO3)=O)C2)=O)cn2cc(Cl)cnc2n1 38430,C1(CC(N2CC(CC(C)NC(=O)Cc3cnsc3)C2)=O)OCCC1(C)C 38431,C12(C(N(C3CCCN(C(C(CC#C)O)=O)C3)CCO)=O)CCOC(C)(C1)C2 38432,CN=c1[nH]cc(C(=O)NC2CCOCC2C(=O)NCc2cc(Cl)ccn2)s1 38433,C12(NC(c3[nH]c4cc(C)sc4c3)=O)CCCCC1N(C(=O)Cn1cnnn1)CC2 38434,N1(C(=O)NC(c2nc(C(=O)OCC)c(N)s2)C)CC(C2CCC2)CCC1C 38435,C(=O)(CC(O)(c1ccccc1)C1CC1)NCCC(C)NC(c1c[nH]nc1F)=O 38436,c1(C(=O)NC2CC(C)N(C(=O)CC3CCCCCCC3)C2)coc2c1CCCC2 38437,C1(C(=O)NCC2CC3CC3N2C(C2SCCS2)=O)CCc2nc(O)[nH]c2C1 38438,C1(CC(N2CCC(C(CNC(c3c(C)cns3)=O)C)CC2)=O)CCCCC12CC2 38439,c1(C(=O)NC2CC(CNC(C3CC4CC4C3)=O)C2)cccc2ccnn12 38440,N1(CCC(=O)NC2C3(CCC(NC(C=CC)=O)CC3)C2)Cc2ccccc2C1=O 38441,N1(C(c2nn(C)c(=O)cc2)=O)CCC(NC(=O)CC2CC2C(F)F)CC(C)(C)C1 38442,N1(C(C=CC(C)(C)C)=O)CC2CC1CN2C(c1[nH]ccc1-c1ccccc1)=O 38443,c1(C(N2CCC(C3(NC(C(C)C(C)O)=O)CC3)C2)=O)coc2c(F)cccc12 38444,c1(C(=O)NC2(c3ccc(C)cc3)CCC2)cnc([N+](=O)[O-])cc1C 38445,O=C(CC(C(F)F)c1ccccc1F)NCC1CCC1NC(c1cocn1)=O 38446,N1(C(c2cc(OC)ncc2F)=O)CCCN(C(C2CC3CCC(C2)O3)=O)CC1C 38447,C1(C(N2C(Cc3c(C)cccc3)CCC2)=O)C2CC3C1C3C2F 38448,N1(C(CCC(=C)Cl)=O)CCCCC(CNC(C2CCCN(CC(C)C)C2)=O)CC1 38449,C(C(C)CC(=O)NCCCC(C)(C)NC(=O)C(F)C1CCC1)OC 38450,C1(N(C)C(c2ncoc2Br)=O)CCC(NC(=O)CN2CC=CC2)CC1 38451,C(=O)(CC(O)CNC(=O)CCc1ccsc1)N(C(C1CCCC1)CO)C 38452,C(CC(=O)NCC1(F)CCN(C)C1)(C(F)(F)F)NC(C1(OC)CCOC1)=O 38453,C1(NC(CNC(C(C)(C)C)=O)=O)CN(C(=O)Cn2nnc(=O)[nH]2)CC12CC2 38454,CCCC(C)(O)CC(=O)NCC1(C)CN(C(c2nc(C)c(C)s2)=O)CC1C 38455,N1(C(C(C)C2CCCC2)=O)CCOC(C)(CNC(c2cc(CF)on2)=O)C1 38456,C1(C(=O)NC2C(c3cn(C)nc3)C2)N(C(=O)CC2CCC=CCC2)CCC1(C)C 38457,C(=O)(C(CC(C)CCC=CC(C)C)N1CCC(C)(C=C)CC1)NCCSC 38458,Cc1ccc(CN2CCC(C(=O)NCc3cccnc3F)C(O)C2)cc1C#N 38459,CC(CN(C)C)N=c1[nH]c(N2CCC(C(C)(C)C)C2)nc2c(F)cccc12 38460,Cc1nc(O)nc(O)c1CC(=O)NCC1(O)CCN(C(C2CC2CF)=O)C1 38461,C(CNC(c1c(Cl)cnn1CCSCC)=O)(C(C)(C)C)NC(CSCC#C)=O 38462,N1(C(c2cnc(-c3ccccc3)o2)C(=O)NCC=C)CC(=O)N2CCCCC2C1 38463,C(=O)(CCCCO)N1CC(OC)(CNC(=O)CSc2ccc(C)nc2)C1 38464,C(C(C)(CNC(C1C=CC(NC(=O)CN2CCC(OC)C2)C1)=O)CO)OC 38465,C1(CNC(c2n[nH]c(C)c2O)=O)(NC(=O)C(C)SC(F)(F)F)CCC(C)(C)CC1 38466,CC(=O)CCCC(=O)N1C2CCC(C2)C1C(=O)Nc1cn(C)nc1Cl 38467,c1(OC)ccc2oc(C(=O)NC3CCCCC3NC(=O)C=CCF)cc2c1 38468,C1(N(C(C(CC)O)=O)C)C2CN(C(=O)CCCNC(=O)OC)CC12 38469,c1(OC)cc(C(=O)NC(C)C(C)NC(=O)CCc2cccc(F)c2Cl)ccc1F 38470,c1(C(=O)NC2C(CNC(CSCC(C)C)=O)CCC2)nnc(O)cc1O 38471,Cc1cc(=O)n(C)cc1NC(C1CC12CC(NC(=O)C(C)CN(C)C)C2)=O 38472,C(=O)(C(C)C(O)C(C)C)NCCCC(C(N1CCCC(C)(CC)C1)=O)O 38473,C1(NC(C2CCCN2C(c2cc(-c3ccccn3)[nH]n2)=O)=O)C2COCC12 38474,C1(NCC2CC(OCOC)C2)CC2(CCC(N)CC2)C1 38475,c1(OC)cc(C(N2CCC(F)(CNC(=O)C3=CCCC3)CC2)=O)cc(F)n1 38476,S(=O)(=O)(c1ccc(N2CCC3CCCC3C2)cc1Cl)NCC1N(C)CCC1 38477,c1(OC)ccc(C)cc1CNC(=O)Nc1cccc(N2CCCCC2=O)c1 38478,Cc1nnccc1C(N1CC=CC(C(=O)NCCc2ccc(O)cn2)C1)=O 38479,C12(CNC(C(C)NC(=O)NC)=O)CC1CN(C(=O)C=Cc1c[nH]nc1C)C2 38480,c1(C(N(C(C)CNC(c2c(Cl)cnn2C)=O)CC)=O)cncc(F)c1Cl 38481,N1(C(C(=C(C)C2CC2)F)=O)CCC(N(C(C2C(C)C2(F)F)=O)CC2CC2)CC1 38482,CC1(C2CCN(CC(N)Cc3ccccc3Cl)CC2)CC1 38483,C1(C(=O)NCC(CC)OC)C=CCN(C(C2(C)CC3CC3C2)=O)C1 38484,N1(C(C(=O)NC(C(CC)C)=O)CCO)CCc2sccc2C1 38485,N1(CC(N2CCCC(C3N(C(C(CC)CC)=O)CCC3)C2)=O)C(=O)CN(C)C1=O 38486,C1(C(N(CCCNC(=O)C(c2ccnn2C)C)CCC)=O)CC(O)CN1C 38487,N1(CC(=O)N(CCCNC(=O)CC2CCC2)C2CC2)CCCc2sccc2C1=O 38488,S(=O)(=O)(C1CC2C(C1)C2(F)F)N1CCC(N(C2CCCC2)C)C1 38489,c1(C(=O)NC(CNC(CC(CCC)C)=O)C(C)(C)C)ccc(C)c([N+](=O)[O-])c1 38490,C(CCCCNC(=O)C(C)NC(=O)NC1CC1)NC(C(C1CCOCC1)OC)=O 38491,C1(C(C)NC(=O)CSc2nncn2C2CC2)CCN(C(C2(C)CC2(F)Cl)=O)CC1 38492,N1(C(c2ccc(C(C)=O)o2)=O)CCC(O)(CCNC(C2CCNC2=O)=O)CC1 38493,C1(NC(C(C)SCC)=O)CCCN(C(C23CC(CC)(C2)C3)=O)C1 38494,N1(C(C=C2CCC(C)CC2)=O)CCC2CN(C(c3cccc4nonc34)=O)C2C1 38495,CC1CN(C(c2conc2C(C)NC(c2ncccc2Cl)=O)=O)CC1(F)F 38496,c1(C(=O)NC)cn(CC(N2CCC(CNC(C3(Cl)CC3(F)F)=O)C2)=O)nn1 38497,N1(C(C2(C)C(C(=O)OC)C2)=O)CCOC(CCNC(=O)CCNS(C)(=O)=O)C1 38498,c1(C(=O)NCC(CN(C(COCCOCC)=O)C)O)c(N)ccc(C)c1F 38499,C1(=CCNC(c2cc(CCC)on2)=O)CCN(C(=O)C(C)(COC)OC)CC1 38500,C=CC1CCCCN1C(=O)COC(C1CCN(C(=O)OCC)CC1)=O.C(C)(C)(C)O 38501,N1(C(C2(CCNC(C(N3CCCCC3)C)=O)CCC2)=O)CCC(O)CC(C)C1 38502,C(C(C)(C)C(=O)NOCc1ccc(F)cc1)NC(CCC1CCC(C)O1)=O 38503,N1(C(C(=O)N(CC(C)C)CCOC)=O)CCCC(C(C)C)CC1 38504,N1(C(c2c(CC)c(F)ccc2)=O)CCC2(CCN(C(C3CCC(C)O3)=O)CC2)C1 38505,N1(C(COCC(=O)OC)=O)CCN(C(=O)CC2(C(F)(F)F)CCC2)CCC1C 38506,CCC(CC(=O)N1CCC(C#N)(c2ccc(F)cc2)CC1)CC(C)C 38507,N1(C(C(CC2CC2)OC)=O)CCN(C(=O)Cc2cnn(C)c2C)CC(C)C1 38508,c1(C(=O)NC2CC(C)N(C(c3cncc(F)c3Cl)=O)C2)cccc2c[nH]nc12 38509,Cc1csc2c(C(=O)NC3(C4CCCN(C(C5(Br)CC5)=O)C4)CC3)ncnc12 38510,N1(C(C=C(C)C2CC2)=O)C2CCC1CC(O)(CNC(=O)C(F)CN(C)C(C)C)C2 38511,C1(CNC(c2c(C)ncs2)=O)CCC2CN(C(=O)C(C)(C)C3CCC3)CCC2C1 38512,C1(C(C)C)C(=O)N1.C1(COC)CCCCC1C(=O)C1CC1.C12(C(N)=O)CC(C1)CN2 38513,Cc1cc(NC(c2ccnc(CNc3ncc(F)c(C)n3)c2)=O)cc(C#N)c1 38514,c1(CC(=O)NC2C3CCN(C(c4nc(C)oc4)=O)C32)c(C)cccc1C 38515,C1(CCC#C)(CC(=O)NCC2CCN2C(=O)CCCC2N=N2)OCCO1 38516,C1(COC)(CNC(c2[nH]ccc2CO)=O)CCN(C(C2CN3CCC2C3)=O)C1 38517,c1(C(=O)NCC2N(C(C34CC(C)C3C4)=O)CC2)cccc(Cn2cncn2)c1 38518,c1(C(=O)NC(CCNC(C2CCC(C(=O)OC)C2)=O)(C)C)nc(C)sc1Br 38519,S(=O)(=O)(c1ccsc1C(=O)O)NCc1cc(N2CCCC(C)C2)ncc1 38520,C1(C(N(C(C)CC(=O)NCC(O)(C2CC2)C2CC2)C)=O)CC12CCOC2 38521,CC(CCCCNC(C1(N(C)C)CCCOC1)=O)NC(=O)CC1COC2CC1C2 38522,C1(NC(c2nnnn2CCOC)(CC)C2CC2)CCC2(CC1)CSC2.C1CCOC1 38523,c1(C(=O)NC2C(NC(C(C3CCC3)OC)=O)C2)ccc2cccc(Br)c2n1 38524,c1(NC)ncccc1C(=O)NCCC1CCN(C(=O)C2CC2)C1 38525,Cc1nc(C=CC(N2CC(NC(=O)CC3CCCCCO3)C(F)C2)=O)[nH]c1C 38526,C(=O)(CCCNC(=O)C1CC1)NCC(CNC(c1cnc(Cl)[nH]1)=O)OC 38527,CC(CN(C)C)CCC(=O)N1C(C(=O)NC2COC3(CCC3)C2)CCC1C1CC1 38528,C1(C(N2CC(OC)(CNC(C3(C)CC3(C)C)=O)C2)=O)CN2CCN1C(C)C2 38529,c1(N2CC(C)(C)C(CO)C2)nc(NCCN2CCOCC2)c2ncsc2n1 38530,CC1CCN(C(c2ccc(O)nc2)=O)CC1NC(c1cnc(C(C)(F)F)s1)=O 38531,c1(C(=O)NC2(C3CCCCN3C(=O)C(F)=CCCF)CC2)cc(Cl)c(F)c(Cl)c1 38532,c1(C(N2CCC(N(C(c3ncc(CC)nc3)=O)C)CC2)=O)c(C)oc(C)c1C 38533,C1(CNC(c2c(C)ncnc2)=O)C2CCCC1N(C(C1CCCN(C)C1)=O)C2 38534,c1(NC(CNC(CCC(=O)NCC)=O)(C)C)ncnc2sc3c(c12)CCC(C)C3 38535,N1(C(C(C(C)(C)C)OC)=O)CCC(C2(NC(c3scc4c3OCCO4)=O)CC2)C1 38536,CCC(CCC(=O)NC(CC)C(N)=O)NC(c1sc(F)cc1C)=O 38537,C1(c2n(CC)nnn2)(NCC2CCC3(CCCC3)C2)CC2(C1)CC(C)(C#N)C2 38538,Cc1cc(=NCC2(O)CCCN(C(C3(n4cncn4)CC3)=O)C2)[nH]c(C(C)C)n1 38539,CCC(CC(=O)N(CCNC(c1c(C)nnn1CC)=O)C1CC1)C(C)(C)C 38540,C1(CCCCNC(=O)CC2COCCO2)CCN(C(=O)CC2C=CCC2)CC1 38541,c1(NC(C(C)OCC)=O)c(C(=O)NC2CCN(C(C)C)C2)cnn1C 38542,N1(C(c2cc(C)c(C)nc2C)=O)CC(CO)C2(CCN(C(=O)CC(C)F)CC2)C1 38543,C1(NC(c2c(C)onc2CO)=O)CC2CC1N(C(=O)C(=CC1CCCCC1)F)C2 38544,C1(NC(C=CCC)=O)(COC)CN(C(=O)CCCSC(C)(C)C)C1 38545,c1(C(=O)NCC(c2c(C)nco2)=O)cccc(C(N)=O)c1 38546,N1(C(N2CCc3cccnc3C2)=O)Cc2cc(Br)ccc2C2CC1C2 38547,c1(CCC(=O)N(CCC)CCNC(C2CC3CC2C3)=O)ccc2c(c1)CCCO2 38548,c1(N(C2CC2)CC)nc(C(=O)OC)cs1.C1(=O)C(C)N1 38549,CC1(C)Cc2cccc(C(N3CC(CO)C(c4ccccc4)C3)=O)c2O1 38550,N1(C(C(CC)(C)O)=O)CC2(CC2)CC1C(=O)Nc1ncc(Br)nc1C 38551,C#CCC(C(=O)N1CCC1c1cn(CC2(n3ccnc3C)CC2)nn1)SC.OC 38552,N1(C(c2cnc(C(C)C)[nH]2)=O)CC2C(N(C(=O)COc3ccc(Cl)cn3)C)C2C1 38553,C=CC(C)(CCOC)C(=O)NC1CN(C(c2sc(C)cc2Cl)=O)CC1SC 38554,C1(NC(COCCNC(COCCC=C)=O)=O)CCC(C(C)O)CC1 38555,C1(CC(=O)N(C)Cc2ccn(CC)n2)CN(C(=O)CCc2nc(C)no2)CCO1 38556,Cc1cccc(C(CNC(c2ncncc2C)=O)NC(c2cn[nH]c2)=O)c1 38557,C1(C(=O)NC(c2ccccn2)C)CCN(C(c2ccc(=O)n(C)c2)=O)C(C)(C)C1 38558,CCC(C)CCCC(=O)NCCCC(C)(C)C(=O)N1CCC12CCCCC2 38559,c1(N2CCC(C)C2CNC(c2ccc[n+]([O-])c2)=O)nc(Cl)ncc1C(F)(F)F 38560,N1(C(c2c(C)ccs2)=O)CCCCC1C(=O)Nc1cccnc1C(N)=O 38561,c1(C(=O)OC)ccc(CC(=O)N(C2CN(C(=O)Cn3cncn3)C2)C)cc1 38562,N1(C(CCC2CCCC(=O)N2)=O)CCCN(C(C23CSC(C2)C3)=O)CC1 38563,c1(C(=O)NCCN(CCOC)C(C2CC=CCC2)=O)csc(O)n1 38564,C1(C(=O)NC(CC#C)CC)CCCCN1C(c1csc(O)n1)=O 38565,Cc1csc2ncc(C(=O)NC34CCCC3N(C(=O)COCCC(C)C)CC4)n12 38566,C1(C(=O)NC2CC(NC(c3cc(Cl)cc(Cl)c3)=O)C2)CCN2CCCC2C1 38567,n1(CCC)ccc(CCC(=O)CCCn2cc(-c3ccn(C4CC4(F)F)n3)nn2)n1 38568,Cc1ccc(C)c(OCCC(=O)NCC2CCN2C(c2nocc2C)=O)c1 38569,c1(C(N2CC(C(N3CCC(Br)C3)=O)SCC2)=O)c(O)cccc1O 38570,C1(NC(c2c(C)cno2)=O)CCC(CNC(=O)CN2CCOCC2=O)CC1 38571,C1(C)(C(=O)NCCCCN(C)C(C2CC2c2ccccc2)=O)CC(C2CC2)=NO1 38572,CC1CCN(C(=O)Cc2cnns2)CC1NC(=O)C=CC1CCCCC1 38573,c1(C(=O)NCC(CC)NC(=O)Cn2ccc(O)nc2=O)ccc2nccn2c1 38574,Cc1c(Cl)cc(CNC(C2CCN(Cc3ccccc3)C(=O)C2)=O)cc1Br 38575,C(CC(C)(C)C)(C(=O)N1CCC(CO)(NC(=O)CSC(F)(F)F)C1)OC 38576,C1(CNC(C(CCC)=CCC)=O)COCCN(C(C2(C)CC=C(C)CC2)=O)C1 38577,C1(NC(C#CC(OCC)OCC)C)CCc2nn[nH]c2C1 38578,Cc1ccc(CC(N2CCC(C(C)NC(=O)C(C)CCO)C2)=O)cc1 38579,c1(N2CC(CC=C)(NC(=O)CC3C=CCC3)C2)ncnc2[nH]c3ccccc3c12 38580,c1(NC)cccc(OC)c1C(N1CC(CO)(NC(C2CCCC2C)=O)C1)=O 38581,C1(CN(C)C(c2ccns2)=O)CCCN1C(=O)CCCc1nccs1 38582,Cc1nn(C(C)C)c(C)c1C(N1CC2CN(Cc3ccc(C#N)cc3)C2C1)=O 38583,C12(C(N3CCN(C(C(C)=CC)=O)C(CC(F)F)C3)=O)CCC(N=[N+]=[N-])C1C2 38584,N1(C(C(C=CC)O)=O)CC(C(F)(F)F)C(CNC(C2CC23CC(O)C3)=O)C1 38585,c1(CC)cccnc1C(=O)NC1CCC1CNC(c1ccn(CC(F)(F)F)n1)=O 38586,Fc1cc(SCC2CC(CCC(=O)N)NC2)ccc1Br.c1ccccc1 38587,CCCCC(O)C(=O)NCC(CC(C)C)NC(c1cnn(C)c1OCC(F)F)=O 38588,c1(OC)ccc(NC(C2CC2C2CN(C(c3c[nH]c(C)c3)=O)C2)=O)cc1C 38589,c1(NC(C(C)C)CCN(C)C(C2CCOC2)=O)ncnc2cnccc12 38590,C1(C)(NC(c2c(COC)cccn2)=O)CCCN(C(=O)C(c2cccnc2)O)C1 38591,C(C(C)(O)CC(=O)NCCNC(=O)CNC(c1ccoc1C)=O)OC 38592,C(=O)(C(CCC)C(=O)OC)OC(CCCC)C(=O)O 38593,CCCC(C#N)C(=O)NCC(CNC(=O)C(CSC)OC)OC 38594,N1(C(c2c(C)c(N)cnc2)=O)CC2CCCC2(NC(=O)Cc2ccccc2Cl)C1 38595,N1(C(C2C(NC(=O)OC(C)(C)C)C2)=O)CCC(N2CCSCC2)CC12CC2 38596,C1(NC(CCC=CC(C)C)=O)CC(C(=O)NCCN2CCCNC2=O)C1(C)C 38597,c1(OC)ncnc(C)c1C(N1CC(C(C)NC(=O)CCCCC2CC2)C1)=O 38598,c1(NC(C2(O)CCN(Cc3c(C)cccc3Cl)C2)=O)cc(F)cnc1C#N 38599,C=CCCCCCCC(=O)NCC(C)NC(c1c(N)cc(F)cc1F)=O 38600,c1(OC)ccc(C(N2CC3CC(NC(=O)C(C)n4cncn4)C3C2)=O)cc1N 38601,c1(NC(=O)C(C2CCCO2)C2CC2)cc(Cl)cc([N+](=O)[O-])c1O 38602,CC1CC2(CCN(C(=O)CC3CCCCO3)CC2)CN1C(c1nn[nH]c1Cl)=O 38603,c1(C(N2CC=CC(NC(c3cc(OC)ncn3)=O)C2)=O)cc2cccc(Cl)c2o1 38604,c1(C(N(CCC)CCNC(C2CCC2C)=O)=O)coc2ccc(OC)cc12 38605,C(C(=O)NN1CCSCC1)(C1CCCCO1)NC(=O)OC(C)(C)C 38606,c1(CC)c(OC)cccc1C(=O)NC(CNC(C1COCCC1(F)F)=O)C(C)C 38607,N1(CC(=O)N(CCC(=O)NCCC2CC2C)C(C)C)CC2CCC1C2 38608,N1(C(c2ccncc2)=O)CCC2(CCCN(C(c3ccc(Cl)nc3O)=O)C2)CC1 38609,N1(C(C(C2CCOC2)OCC)=O)CC2(CCCC2NC(=O)CC2CC2)C1 38610,N1(C(c2c(C)cc(N)cn2)=O)CC2COCC2(C(N2CCC(O)(C(N)=O)C2)=O)C1 38611,c1(OC)cc(OC)c(C(=O)NC2CN(CC3CC3)CCO2)cc1N 38612,CCC(CC(F)F)C(=O)NC1CCCCN(C(C2CCCN(CC(C)C)C2)=O)C1 38613,CCCCC(C(=O)NC1CC(CNC(c2ccoc2CC)=O)C1)NC(N)=O 38614,Cc1ccc(Cl)c(O)c1C(=O)NCCCCC(C)NC(c1c[nH]nc1C)=O 38615,N1(C(=O)C2=CCCC2)CCC2C(CCCN2C(c2cnc(-c3ccco3)s2)=O)C1 38616,c1(C(=O)NC2(CC=C)CN(C(C3CC(C(C)C)=NO3)=O)C2)ccc2n[nH]cc2n1 38617,C(c1cnc(C)nc1O)=CC(N1CC(C)CC(NC(CCCCC=C)=O)C1)=O 38618,c1(C(C(=O)NC2CCN(c3c(C)ccs3)CC2)=O)cc(F)cc(Cl)c1 38619,c1(C(N2CCC(N(C(=O)CNC(C3CCC3)=O)C)C2)=O)ccnc(O)c1 38620,C12(OC)CCCCC(C(=O)N(CC(C)NC(=O)CCn3ccccc3=O)C)(C1)C2 38621,C1(C)(NC(CCSC)=O)CCN(C(=O)C(C(C)C)c2cnc(C)s2)CC1 38622,c1(OCCc2cccc(CC)n2)cc(Br)c(F)cc1F 38623,c1(CN2CC(n3cc(Cc4nnn(C)n4)nn3)C2)cccc(OC(F)(F)F)c1 38624,c1(C(N2C(C3CCN(C(C(CC=C)C)=O)C3)CCC2)=O)ccc(C)c2cccnc12 38625,N1(C(C2=CCCC2C)=O)CCC(NC(c2cc(N)c(O)c(F)c2)=O)C(F)(F)CC1 38626,C1(F)(C(N(C2CCN(C(C(C)(F)F)=O)C2)Cc2ccccc2)=O)CCCOC1 38627,CN1CCC2CN(C(C3CCN(C(c4cc(Cl)ncn4)=O)CC3O)=O)CC2C1 38628,N1(C(CNC(C(CC)C)=O)=O)CC=C(C(=O)NC(CO)C2CC2)C1 38629,Cc1nc(Cl)[nH]c(=NCC2CC(CNC(=O)CCc3ccn(C)n3)CO2)c1Cl 38630,C1(NC(C(c2n(C)cnc2)O)=O)CC2(CCC(NC(C3(C)CC3(F)F)=O)CC2)C1 38631,c1(C(=O)NC2CC(C)(NC(CCC(C)OC)=O)C2)csc2cc(C)ccc12 38632,C(CN=c1[nH]cnc2c(Cl)cc([N+](=O)[O-])cc12)C1C2N(C(=O)OCC)CC(CC2)C1 38633,c1(CC)cc(C(N2CCC(NC(c3cc(O)ncn3)=O)C2)=O)ccn1 38634,Cc1cc([N+](=O)[O-])c(Cl)cc1S(=O)(=O)N.C1(C(F)(F)F)(NC(C)C)CC2(C1)OCCO2 38635,n1(CCC)cc(Cl)c(C(=O)NC23CC2CN(C(=O)C(C)CC)C3)n1 38636,c1(COC)nccc(=NC2CCC3CN(C(c4n[nH]c(C)c4C)=O)CC23)[nH]1 38637,Cc1nnc2n1CC(C(=O)NCC1CCC1NC(=O)C=CCO)C2 38638,C(=O)(CCCCN(C)C(C)C)NC1C(CNC(C(CC)=CC)=O)COC1 38639,C(=O)(C(C)(C)S(C)(=O)=O)NC(CC1CN(C(Cn2c(=O)ccc(C)n2)=O)C1)C 38640,N(C1CCCn2ccnc21)C(CC(C)NC(C1C(C(C)C)C1)=O)=O 38641,c1(C(N2CCC(c3cnccn3)C2)C(=O)NCCOC)cc(Cl)cnc1OC 38642,c1(OC)ccc(CCC(=O)NC(CNC(=O)C=CC(F)(F)F)C(C)(C)C)cn1 38643,N1(C(c2cc(OCC)cc(F)c2)C(=O)NCCC#N)CC2CCC(OC)C2C1 38644,C(=O)(C1Cc2ccccc21)NC(C1N(C(c2c(CC)ocn2)=O)CCC1)(C)C 38645,N1(C(C(C)SCC)=O)CCC(CNC(c2cnnc(C3CC3)c2)=O)C(F)(F)CC1 38646,C1(C)(COC)CCCN(C(=O)Cn2cc(CNC(C3(C#N)CC3C)=O)nn2)C1 38647,C1(CCNC(CCCOC(C)=O)=O)CCCN(C(=O)C(N2CCCC(O)C2)C)C1 38648,C(=O)(CCCCC(C)(C)C)N1CCC(NC(c2c(CC(C)C)onc2)=O)C1 38649,c1(OCC)cc(C(=O)NC2CCC(O)CC2)c(-c2nccs2)cn1 38650,N1(C(COC2C(CC)CCCC2)=O)CCN(C(c2ccnnc2O)=O)CC1C 38651,C(CCCCCC(C(=O)C(=O)OC(C)(C)C)N1CCOCC(C)(F)C1)N.C1(O)CC1 38652,C(=O)(C1=C(C)S(=O)(=O)CC1)N1CC(NC(CCCC)=O)C(OC)C1 38653,N1(C(C2C(=C)C2)=O)CCC2(CCCCN(C(C3CC4CCC(C3)C4(F)F)=O)C2)C1 38654,N1(C(C(C)=C(C)C)=O)CC(C(=O)NCC(N)=O)OC(C)C1 38655,C1(CCN(c2ccccn2)CCC#N)=C(Br)C2C(=CC=C1)OCCC2 38656,N1(C(c2nc(C)n(C)n2)=O)CCC(C2CCCN(C(=O)C(C)(O)C3CC3)C2)C1 38657,N1(C(C(CC)C)=O)CC2(CC(NC(c3coc(Br)n3)=O)c3nccn32)C1 38658,C(=O)(C(O)CCNC(=O)C(CSC)OC)NC(C#C)CC1CCC1 38659,c1(CC)nn(C)c(C(c2nnnn2C(C)C)NCCCC(C)(C)OC)c1Cl 38660,N#Cc1c[nH]c(C(=O)NCCC2CC(NC(C3(c4ccsc4)CC3)=O)C2)c1 38661,C(CCCCC(=O)N1CC(O)CC1(C)C(=O)N(C)Cc1ccncn1)OCC 38662,c1(C(N2CCN(CCCNC(C3C(=C)C3)=O)CC2)=O)nn(C)cc1[N+](=O)[O-] 38663,C1(C2CCCN(C(c3ccn4nccc4n3)=O)C2)(NC(CC(C)SC)=O)CC1 38664,C12(NC(C(CC)SC)=O)CCCC1N(C(c1c(OC)cccc1F)=O)CC2 38665,N1(C(C(CC)OCC)=O)CCCC(C2CN(C(c3cccc4[nH]ncc34)=O)C2)C1 38666,C1(C)(NC(c2n(C3(SCC)CC3)c(-c3ccnc(C)n3)nn2)=O)CCS(=O)(=O)N1 38667,c1(C(C)C)conc1CC(N1CC(CC(C)NC(c2c[nH]nc2C2CC2)=O)C1)=O 38668,C1(C(N2C3(C)CC3CC2)=O)C=CCCN1C(=O)CCOCC(F)F 38669,N1(C(C=C(C)C)=O)CCC2(CCC2)C(NC(=O)CCOc2cccc(Cl)c2Cl)C1 38670,N1(C(CCc2nnc(C)n2C)=O)CCCC(NC(=O)CC2CC(C(F)F)C2)C1C 38671,c1(NCC)ccc2c(c1)OCO2.c12cccc(c1)N(C(C)=O)C2 38672,c1(N(C)C)nc2cc(C(=O)NC3CC(C)(NC(C4CC4C#N)=O)C3)ccc2o1 38673,CCCC(CCC)CC(=O)NC(CCC1CC1)C(=O)N1CCC1CC(=O)NC 38674,N1(C(C(c2cc(C)oc2C)C)=O)CCC2CCN(C(c3cnn(C)c3)=O)C2C1 38675,c1(CC=CC)ccc(C(=O)NC2CC(C)(NC(=O)CC3CCC3)C2)cc1 38676,N1(C(C(C(C)O)N(C)C)=O)CCOCC(C)(CNC(c2coc(CO)c2)=O)C1 38677,c1(C2C(NC(C=Cc3ccc(OCCOC)cc3)=O)C2)ccc2cc[nH]c2c1 38678,C(C)(CNC(C1(C(C)(C)C)CCCCC1)=O)(C(C)C)NC(Cc1nnc(C)o1)=O 38679,C(=O)(C(C)(C)CCCNC(=O)C(F)C1CCOC1)NC(C)Cn1cnnc1 38680,N1(C(C2CN(C(C(CC)(C)COC)=O)CC(C)C2)=O)CCOC2C(O)CC12 38681,CC(CO)CCCNC(C1CCCN(C(=O)Cc2cccc(O)c2)C1)=O 38682,C(=O)(CCCCC(C)C)N1CCC(OC)(CNC(C2COCCC2(F)F)=O)CC1 38683,C1(C(N(C(CNC(C2N(CC#C)CCC2)=O)C)C)=O)CCc2nncn2C1 38684,C(=O)(C1=NN(C)C(=O)CC1)NC1CCN(C(CC)=O)C(C2CC2)C1 38685,c1(C(N2CCC(N(C(=O)CSc3nnnn3C3CC3)CC)C2)=O)cncc(N)n1 38686,C(Cn1cncn1)(C(=O)NCCCC1CCOC1=O)NC(=O)Cn1ncnn1 38687,N1(C(C(=O)NCc2nccc(OCCC)n2)=O)CCCN(CC(=O)OC)CC1 38688,C1(CC(=O)N(CC(C)C)CC(C)NC(=O)CC=CC(C)(C)C)OCCC1(C)C 38689,N1(CC(=O)Nc2cc(C(F)F)ncn2)CCC(C(F)(F)F)C(NCC)C1.C(F)(F)F 38690,c1(C(=O)NCC2(F)CCN(C(Cc3c(C)nsc3)=O)CC2)ccc(N)c(F)c1F 38691,C1(C)(C(=O)NC2CCC(C)N(C(=O)C=Cc3cscn3)C2)Cc2ccccc2C1 38692,C1(C)(CNC(C(C2CC=CCC2)NC(CN(CCOC)C)=O)=O)CCCO1 38693,Cc1ccc(C(N2CC=CC(NC(=O)CCC3CCN(C)CC3)C2)=O)c(Cl)c1C 38694,C1(NC(CC=CCCCCC)=O)C2CN(C(=O)OCc3ccccc3)CC12 38695,c1(C(=O)NC(CNC(c2ccc(C)cn2)=O)(C)C(C)C)cc(C2CC2)n(C)c1C 38696,Cc1nnc(N2CCCC2c2csc(C)n2)n1CC1CCN(C(C)(C)C)CC1 38697,C(CCCC(=O)N1CCC(C(C)NC(=O)CC2(C)CCOCC2)C1)N(C(C)C)C 38698,O(NC(=O)CC1(NC(c2ccn(CCF)n2)=O)CCCC1)CC(=O)OCC 38699,N1(C(c2n(CC)nnc2)=O)C2CCC(C(=O)NC3CCCCCC3F)C1CC2 38700,c1(OC)c[nH]c(C(=O)NC(C2CCN(C(C3CCC4(CC4)C3)=O)CC2)C)cc1=O 38701,c1(C(=O)Nc2cc(C(=O)NCCC3CC(O)C3)ncc2)ccc(F)cc1F 38702,C(CC(O)C(=O)NC1CCCC1NC(C1(C2CCCO2)CC1)=O)N(C)C 38703,c1(C(=O)NCCCCNC(CCC#CC)=O)cc2ccc(C(C)=O)cc2[nH]1 38704,N1(C(C(COC)O)=O)CCCC(CO)(NC(C2CCC(F)(F)CC2)=O)C1 38705,c1(OCC)cccc(C(C)NC(c2cnc(C3(C)OCCO3)s2)=O)c1 38706,C1(C(N2CCC(CN(C)C(c3ncc(F)cc3N)=O)CC2)=O)CCCC(F)(F)C1 38707,CC1(C)CN(C(=O)CCCCC2CCCC2)CC1NC(c1cnn(C(F)F)c1)=O 38708,C(=O)(N=c1[nH][nH]c(C)c1Cl)c1cccc(-c2c(OCCOC)cc(F)c(F)c2)n1 38709,c1(C(C)C)ccc(C(=O)NCC2CC(F)(CNC(C3(C)CC3(F)Cl)=O)C2)cc1 38710,C1(c2nnnn2CCCF)(Nc2cccc(SC)c2)CCCC(F)(F)CC1 38711,C(=O)(CC(=O)N(CCCC(=O)N1CCC1CC(C)C)C)NCC 38712,N1(C(Cc2ccc(C#C)cc2)=O)CC2CCC1CC2NC(c1c[nH]nc1CC)=O 38713,C1(CNC(C2(C)CCCC2)=O)CCCCCN1C(=O)C(F)CC1CCCC1 38714,c1(C(N(C)CC2N(C(COCCC=C)=O)CC(F)C2)=O)cc(N)c(Cl)cn1 38715,c12ccc(cc1)COCC(=O)NC1C(C1)NC(=O)C(C)N2.C1(CC)CCOCC1 38716,CC1CCN(C(C2CCCCC2O)=O)CC1CNC(C1(c2ccccc2)CC1)=O 38717,C1(NC(C(C)=CC)=O)CC2(CCCN(C(C3CC3CCC)=O)C2)C1 38718,C1(C(N2CC(C(CC)CC)C2)=O)(NC(c2ccn(CCF)n2)=O)CCSC1 38719,Cc1ccc2c(c1)C(C(=O)N1C(CNC(c3cc(O)n(C)n3)=O)CC3CC13)CC2 38720,C1(C(=O)NCCCOCCNC(=O)C=CC2CCCO2)CC(C2CCCC2)C1 38721,C1(C(N(CCCNC(c2ncoc2C2CC2)=O)C2CC2)=O)CCCC(O)C1 38722,C(=O)(CCS(C)(=O)=O)NCC1(C(=O)N(C2CCCC(C)C2C)C)CC(=C)C1 38723,N1(C(c2c(C(C)C)con2)=O)CCC2CN(C(c3cncc([N+](=O)[O-])c3)=O)C2C1 38724,N1(C(C=C(COC)C)=O)CCCOC(CNC(=O)CC2CC3CCC2C3)C1 38725,C1(C(N2C(C3CCN(C(C4CCCN4C4CC4)=O)C3)CCC2)=O)CC(=O)N(O)C1 38726,c1(NC(C)=O)n[nH]c2cc(-c3ccncc3)ccc12.c12ccc(c(C)c1)c(=O)[nH]2 38727,CC1(C)NC(=O)C2(CCN(C(=O)NCc3cc(C4CCC4)no3)CC2)O1 38728,C(=O)(CCC(C)CN(C)C)N1CCC(CC(C)NC(C(CC=C)C)=O)CC1 38729,N1(C(C(=O)NC(C)C)=O)CCC(C)(C)CC1C(=O)NC1CCC(C2CC2)C1 38730,CC1(c2nc(-c3cnn(CCO)c3)nn2-c2ccc(Cl)cc2)CCCC(F)(F)C1 38731,c1(COC(C2(C(N3CCN(CC)CC3)=O)CC2)=O)ccc(On2cccn2)cc1 38732,n1(CC)cc(NC(=O)CC(C)(C)N(C)C(c2cncc(C#N)c2)=O)ccc1=O 38733,C(C(=O)N=c1ccn(CCNC(C2CC3(CC3)CN2C)=O)[nH]1)=C(C)C(C)(C)C 38734,Cn1ncc(C(=O)NC(CNC(c2csc(=N)[nH]2)=O)C2CC2)c1S(N)(=O)=O 38735,c1(OC)cccc(OCC(=O)N2C(C3CCC3)CCC2)c1.C(=O)(C(O)C(C)C)OC 38736,Cc1c(Cl)ccc(C(N2CCC23CN(C(=O)Cn2nc(Cl)ccc2=O)C3)=O)c1Cl 38737,C(=O)(CCC(C)(C)[N+](=O)[O-])NCC(C)NC(=O)CSCc1ccccn1 38738,O=C1Nc2ccc(C(N3CC4CN(C(=O)CC5(O)CCC5)C4C3)=O)cc2C1=O 38739,N1(C(C(CC)N(C)C)=O)CCN(C(=O)C(O)Cc2[nH]cnc2C)C(CCO)C1 38740,C1(C2CCN(C(=O)CN3CCCC3C)CC2)(NC(CC(CC=C)(C)C)=O)CCC1 38741,C(CCCCC(=O)N1CCC(C)(C)C1C(=O)NC(C)C(=O)NC(C)C)SC 38742,CCC(O)C(F)(F)C(=O)N1CCC(C(C)NC(=O)CCCn2ccnc2C)CC1 38743,N1(C(COCC)=O)CC(C)N(C(=O)Cc2csc(NC(C)=O)n2)CC1C 38744,C1(C(N2CCCC2Cc2ccccc2)=O)CCC2(CCOCC2)NC1 38745,Cc1ncc2ccc(C(N3CC4(CC(NC(C5CCC(=O)N5)=O)CO4)C3)=O)cn12 38746,C1(NCC)COCCN(C(=O)COCn2nnc(C(=O)Oc3ccsn3)c2N)C1 38747,CCCC(C(=O)Nc1cnccc1OC)NC(=O)OC(C)(C)C 38748,N1(C(=O)Cn2ncccc2=O)CC2CCN(C(=O)CCc3ccncc3)C2C1 38749,C1(C(=O)NC(CN(C(=O)CCCOC(C)C)CC)C)OCCC1(C)C 38750,n1(CC)nncc1C(=O)NC1C=CC(CC(=O)NCC2(CC)CCC2)C1 38751,c1(C2(C(=O)NCCC(C)(C)N(C)C(C3COCCO3)=O)CCC2)c(F)cccc1F 38752,CCC(CCCC(=O)N(C(C1CCC1)C)CC)NC(=O)C(n1ccc(C)n1)C 38753,c1(C2CC2)nnc2n1CCC2.c1(COC)csc(C)n1.C1CNC(=O)N1 38754,C1(OCC)(CN)CN(C(=O)C(C)=CCOC)C1.C1(=O)CC1=O.OC 38755,c1(C(=O)NCC2C(CNC(Cn3c(C)nnn3)=O)C2)ccc(NC=O)cc1 38756,C(=O)(CCCS(C)(=O)=O)N(CCCNC(c1ccc(F)c(C(F)F)c1)=O)C(C)C 38757,Cc1[nH]c2ccccc2c1C(=O)NCC1CN(C(C2C3CCC23)=O)CCN1C 38758,N1(C(C(N)Cc2cscn2)=O)CCC2(CCN(C(c3cccc(N(C)C)c3)=O)C2)C1 38759,O=C(NN1CCSCC1)C(=O)N1CCCCC1c1ncc[nH]1 38760,C1(OC)CC2(CCN(c3ccnc4ccnn34)C2)C1 38761,C(=O)(CC(C)CC(C)(C)C)NC1CC(OCCN(C2CCCC2)C(=O)COC)C1 38762,N1(CC(=O)NCC2(CCNC(c3onc(CC)n3)=O)CC2)CC2C=CC1C2 38763,Cc1ccc(F)cc1CC(=O)NCC1(C)CCCN(C(C23CCN(CC2)CC3)=O)C1 38764,c1(SC)ccc(C(N2CC(NC(c3ccc(CN(C)C)[nH]3)=O)CC2C)=O)cn1 38765,C1(c2nnnn2C)(Nc2c(OCCOC)nccc2)CCOCCC1 38766,c1(SCC)nc(C)c(CC(=O)NC(C)(C)CCCNC(C2(C)CC2(F)Cl)=O)s1 38767,c1(NC(C2CN(S(CCC(=O)OC)(=O)=O)CC(F)C2)=O)ccc2c(n1)NC(=O)CC2 38768,c1(C(C)C(=O)NCC2CC(NC(c3occc3Br)=O)C2)cccc(C#N)c1 38769,CCC(O)(CC)c1cn(CCC(=O)N(CC(C)C#N)CC)nn1 38770,C(CC(CNC(=O)COC1CC=CC1)NC(C1CCCN1C(C)C)=O)OC 38771,C(=O)(C(C)C(O)CC)NCc1cc(C(=O)NCCC(=O)NCC)n[nH]1 38772,C1(C(=O)Nc2cc3cc[nH]c3cn2)CC2CCC1N(C(=O)CN1CCOCC1)C2 38773,C1(NCc2ccc(OCCOCC)c(OCC)c2)CCCC(P(C)(C)=O)C1 38774,C(=O)(C(F)(F)C(C)(C)O)N1CC2C(NC(c3c(C)n(C)nc3)=O)(CC2)C1 38775,C1(C(=O)NCCOC2CCN(C(C3C(OCC)C3)=O)C2)CCC(C)CC1 38776,C1(C#N)(C(=O)NC(CC)CNC(C2CC(=O)N2)=O)CC12CCCC2 38777,C1(NC(c2c(C)n(C3CC3)cc2)=O)CC2CC1N(C(c1cnc(C(C)O)s1)=O)C2 38778,CC1CCC(NC(=O)CCC2CC2)CN1C(c1cc(-c2ccccc2)[nH]n1)=O 38779,c1(C(=O)NCC(C)CNC(C2CCOC3(CCC3)C2)=O)cc(F)c(F)cc1F 38780,c1(C(=O)NC2CN(C(C3C(C)OCCO3)=O)CC2F)cn(C)c(=O)cn1 38781,n1(C(C(=O)NC(CC)CNC(c2cnccc2C)=O)C)cnc2ccccc12 38782,Cc1nc2cc(C(=O)NC(CNC(C3CCCC(=O)N3C)=O)C(C)C)cnc2[nH]1 38783,C1(C(N(CC(CCC)O)C)=O)CCC(C(C)C)N1C(C1CCCC(O)C1)=O 38784,CC1CC(C(=O)N(C)CCOCCNC(=O)C(C)(C)C2CCCCC2)C1(C)C 38785,Cc1ccc(C=CC(=O)NCC2(F)CC(NC(C3CCSC(C)C3)=O)C2)cc1C 38786,CCCC(C)CC(=O)N1CCC(C(C)CNC(C2(CF)CC2)=O)CC1 38787,c1(C2C(C(=O)NCC3(O)CN(C(C(c4ccsc4)=O)=O)C3)CC2)ccc(F)cc1 38788,C(=O)(CC(F)F)NCC1CC(NC(C=CC)=O)C1 38789,N1(C(C(CC)C)=O)CC2(CC(NC(=O)COc3c(C)cccc3C)C2)C1 38790,c1(OC)nc(N2CCN(C(=O)CCC3(OC)CC3)CC2)cc(C)n1 38791,c1(NCc2ccc(OCC#C)cc2)ccc(F)cc1C(=O)NC1CNC1 38792,c1(C(N2CCCC(N(C(C(CSC)O)=O)CCO)C2)=O)cc(F)ccc1F 38793,C(=O)(C1=CCCCC1C)NCC1N(C)CCN(C(c2cc(C)on2)=O)C1 38794,C1(COC)CCN(C(c2nc[nH]n2)=O)C(C(=O)N(CC(C2CCC2)OC)C)C1 38795,C1(C(=O)NC(CCN(CC)CC)C)COCCC1NC(C1CN(C)CCO1)=O 38796,C1(N(C(c2n(CC=C)ccc2)=O)C)CCCCC1N(C(=O)Cn1nccc1C)C 38797,c1(C(C)NC(=O)C(n2nnnc2C2CC2)CC2CCC2)ccc(Cl)cc1 38798,C(C(COC)CC(=O)N1CC(n2cc(NC(=O)CC(C)(C)O)nn2)C1)OC 38799,C(CC(F)F)(C(=O)NC1CC2C(C1)C2(F)F)NC(CC1(OCC)CCC1)=O 38800,c1(C(N2C(CN(C(C(CC=CC)C)=O)CC)CCC2)=O)cc(C)cc([N+](=O)[O-])c1 38801,Cc1cc(C(N2CCC(C)(CCNC(c3c[nH]nc3C(F)F)=O)C2)=O)cc(C)c1 38802,c1(OCCC(=O)NC(C(C)NC(c2ccncc2)=O)C)ccc(CC#N)cc1 38803,C1(C)(NC(CC2CC(CC)OCC2)=O)CCN(C(c2sncc2C)=O)CC1 38804,c1(CC)cc(NC(c2coc(CNC(=O)CCC3CC3(C)C)c2)=O)cc(O)c1 38805,c1(C(N2C(C)CC(NC(c3cncc(COC)c3)=O)C2)=O)ccc(N)c(Cl)c1O 38806,c1(N2CC(C(C)NC(=O)CCC3CC3(Cl)Cl)OCC2)cc(-n2cncn2)ncn1 38807,c1(C(C)=O)ccc(C(F)(F)F)nc1NC(C)(C)CNC(C1CC(C)OC1C)=O 38808,c1(-c2cc(NCc3c(C)c4c(s3)cccc4)ncc2)ccc2c(c1)OC(C)(C)O2 38809,C12CN(C(C3(O)CCN(C(=O)OC(C)(C)C)C3)=O)CCN1C2=O.C(C)(C)(C)O.CC 38810,C(C(F)(C(=O)NCCc1cocn1)C(C)C)NC(C(CC#C)O)=O 38811,c1(CC)cc(C(=O)NC2CCN(C(=O)CC3CC(C)=NO3)C2C(C)(C)C)n(C)n1 38812,Cc1cccc(C(C2CCCCC2)C(=O)Nc2cnccc2C)c1 38813,C(C(=O)NCC1CCCC(CNC(c2ccc(C#N)cn2)=O)C1)(C(C)(C)C)SC 38814,C(=O)(C(C(C)C)NC(N)=O)N(C(c1cn(Cc2c(C)nn[nH]2)nn1)C)C 38815,c1(COC)conc1C(=O)NCC1CCC(NC(C2CN(C3CCC3)C2)=O)C1 38816,Cc1c(C(=O)NC2CC(C)N(C(=O)CSc3nnnn3C)C2)noc1C1CC1 38817,Cc1c(N(CCCF)C)cccc1Cl.c1(C2C(=O)N2)cnn(C)c1 38818,N1(C(C2(CC#C)CCCO2)=O)CCC(C)N(C(=O)CC2(CC)CCC2)CC1 38819,C1(N(CC#C)C(C2CC2(F)Cl)=O)CCN(C(c2cocn2)=O)CC1 38820,N1(C(C(C)O)=O)CC(F)(C(=O)NCCCn2cncn2)C1 38821,C(=O)(C(CCC1CCC1)NC(c1cnsc1)=O)NC1(CC(C)(C)C)CC1 38822,C=C(Br)CCC(=O)NC1CCN(C(=O)CCc2cnccn2)C1C 38823,N1(C(C=C(CC)CC)=O)CCC2CN(C(c3cc(CC4CCC4)c[nH]3)=O)CC2C1 38824,Cc1cc(CNC(C)C(C)OCc2ccccc2)ccc1[N+](=O)[O-] 38825,N1(S(=O)(=O)CC2CC(CO)C3CC23)CCC(O)(C2(C(=O)O)CCC2)CC1 38826,C(C(C(=O)N(CC(=O)NC(C)C)C)C(C)C)NC(C1(CC=C)CCC1)=O 38827,Cc1ccc(C(N2CCN(C(=O)CC3=NNC(=O)C3)C3CC23)=O)c(F)c1F 38828,S(=O)(=O)(CCC(=O)NCC1CCN(C(c2cc(C)c(Br)o2)=O)CC1)NC 38829,CC1CN(C(=O)CN2CCN(C(C3CC3c3ccco3)=O)CC2)CC(C)(C)O1 38830,Cc1cnc(C(=O)NC2(CCCC(N3Cc4c[nH]nc4C3)=O)CCC2)c(C)c1 38831,c1(C(=O)NCC(C)(C2CCC2)NC(COC(C)C)=O)cn(CCO)nn1 38832,c1(CC(N2CC(CC(C)NC(c3ccc(C(N)=O)s3)=O)C2)=O)ccccc1O 38833,c1(CNC(c2nnnn2CCCF)(c2ccns2)C)ccc(OCC(F)F)cc1 38834,c1(CC)cnc2cc(C(=O)NC3(CCC(=O)OC)CCCC3)[nH]c2c1 38835,c1(OCCC(C)C)ccc(C(=O)NCC(O)CNC(C2CCCN2C=O)=O)cc1 38836,c1(C(=O)NC2CC(C)N(C(=O)CC3(O)CCCC3)CC2)noc2cc(F)ccc12 38837,n1(CC)cc(N)c(-c2noc(CCC3CCN(C4CCCC4)CC3)n2)n1 38838,N1(C(C(COC(C)C)NC(Cc2c(C)nsc2)=O)=O)CCC2(CC2)C1 38839,C(=O)(CC(C)F)NC(CNC(CC=CCC)=O)(C)C1CC1 38840,C1(NC(C(F)=CCC)=O)CCCC12CCN(C(c1ccc(Cl)c(Cl)c1N)=O)C2 38841,c1(COC2CC(C(=O)OC)C2)cccc2c1CCC2 38842,c1(C(=O)NC2(CCOC)CCN(C(=O)C(C)=C(C)C)CC2)scc2c1CCCC2 38843,C1(CC=C)OCCC1(c1nnnn1CC=C)NCC=CBr.C1(C)(CC)CC1 38844,c1(C(N2CCN(C(=O)CC(F)F)C3CC23)=O)cc2ncc(Br)cc2o1 38845,Cc1[nH]c(=N)[nH]c(=NCC2CCN(CCc3ccccc3)CC2)c1Cl 38846,N1(C(c2c(C)n(C)nn2)=O)C2CCC(C2)C1C(=O)NC1CC(C(F)(F)F)C1 38847,C(=O)(CCCCC(=O)OC)N1C(CCNC(C(CC)C(C)O)=O)CCCC1 38848,C12(CN(C(=O)C(CO)OC)C1)N(C)C2=O.N1(CC)CC=CC1 38849,C(=O)(CCC(CF)CF)NC(C(=O)NC1(C(=O)OC)CC1)CC(C)C 38850,N(C(=NCC1CCC1)NCc1ccsc1)C(c1ccccn1)C1CC1 38851,N1(C(Cc2c(F)ccc(C)c2)=O)CCCN(C(c2nc(C)ncc2Cl)=O)CC1C 38852,c1(C(=O)NCCCC(C)NC(C2CC3CCC2C3)=O)cc2sccc2s1 38853,N1(C(CC2(C(=C)F)CCC2)=O)CCC2(CCC2)C(NC(c2cn(C)c(=O)n2C)=O)C1 38854,N1(C(C=Cc2c(C)n[nH]c2)=O)CC(NC(c2cc(C#N)ccn2)=O)CC12CCC2 38855,CCCS(=O)(=O)C(C)C(=O)NCC1CC1CNC(=O)C=Cc1nccn1CC 38856,c1(C(=O)NCc2cc(C(=O)NCC(C(CC)C)OC)sc2)c[nH]c2ccccc12 38857,CC(c1ccco1)=CC(=O)NC1(C)CC(NC(=O)CC#N)C1 38858,C=C(C)CC(C(=O)N1CC=CC1Cn1cc(Cn2ccccc2=O)nn1)OC 38859,Cn1ncc(C2CC2)c1C(=O)NC1CCC1NC(=O)CC1(O)CCOCC1 38860,c1(C(C(=O)NC(Cc2c(OC)cccc2)C(C)C)OC)ccc(C#N)cc1 38861,C1(CCOC)(NC(c2ccc(Br)o2)=O)CCN(C(c2cccc(C(C)C)c2)=O)C1 38862,c1(CNC(CNC(C2(C)COC2)=O)=O)cc(=O)cc[nH]1 38863,Cc1ncc(Cl)cc1N(C1CCCCC1)C(c1[nH]c(C)c(C(=O)OCC)c1C)=O 38864,c1(C(N2CCC(CC(F)F)C2)C(=O)NC)cccc(S(N)(=O)=O)c1 38865,C=CCCCCCC(=O)NC(C)(CC)CCNC(C1COCCN1CC)=O 38866,N1(C(CCOCCOCC)=O)CC2(CCN(C(=O)CC3CCCC(C)C3)C2)C1 38867,c1(OC)ccc(C(N2CCN(C(=O)Nc3ccc(F)cc3)CC2)C2CC2Cl)cc1 38868,N1(C(c2c(OCC)n(C)nc2)=O)CCC(C2CCN(C(=O)C3=CCCOC3)C2)C1 38869,CS(=O)(=O)C1CCN(C(c2ccc(F)cc2)C(=O)NCCCC2CC2)C1 38870,c1(CNC(c2c(OC)csc2)=O)ccc(CNC(=O)C(c2nc(C)cs2)C)cc1 38871,CSC1=C(C(=O)NCC(CNC(c2cn(C3CCOC3)nn2)=O)CO)CCCC1 38872,CC(C)(C)C(C)(O)CNC(C1CC1CNC(c1csnn1)=O)=O 38873,c1(CC)nonc1C(=O)NC(C)(CNC(c1ccncc1)=O)CO 38874,CC1(C(N2CCN(C(=O)Cc3cocn3)CC2)=O)C=CCCC1 38875,N1(C(CNC(CCC(C)C)=O)=O)CC(N(C(=O)C=C2CCCC2)CC)C(C)(C)C1 38876,c1(OC)c(F)ccc(F)c1C(=O)NC1CC(C)N(C(c2cn(C)cc2C)=O)C1 38877,C=CC1(CC(N2CCC(CCNC(C3CC3CF)=O)C2)=O)CCC1 38878,C(=O)(CC1CCOc2ccccc21)NCC1N(C(C2CC(OC)C2)=O)CC(F)C1 38879,c1(C(=O)NC(CC(C)NC(=O)C=CC=C(Cl)Cl)C)cc2n(n1)CC1(CC1)C2 38880,Cc1cc(Cl)cc2cc(C(=O)N(c3cnn(-c4ccccc4)n3)C)[nH]c12 38881,C1(NC(C(CC)OC)=O)CN(C(c2cc(Cl)c(C)cn2)=O)C(C)(C)C1 38882,C1(C(=O)NCc2cc(CC)no2)CC(NC(=O)C(=O)NC)C1(C)C 38883,c1(CCSCCC(N)C2CCC2)c(F)cccc1Cl 38884,CC1CC(NC(C2CC3CCC2O3)=O)CN(C(c2cccc(CO)c2)=O)C1 38885,c1(OC)cccc(C(=O)NC2CC(CNC(C3(CCO)CC3)=O)C23CCC3)c1O 38886,C1(N(C)C)CCCN(C(=O)C(CC2CC2)NC(=O)CCc2ncnn2C)CC1 38887,CC1(C)C2CCC1(C(N1CCC(NC(=O)Cn3cccn3)C(CO)C1)=O)C2 38888,N1(C(CC(C)(C)O)=O)CCC(NC(=O)CCN2C(=O)CCC2=O)C(F)C1 38889,N1(C(c2c(SCC)cccc2)=O)CC2CC(NC(=O)C(C)(C)N3CCCC3)C1C2 38890,c1(C(=O)OC)cc(=NCC(C)(C2CC2)NC(C2COC(C)C2)=O)[nH]c(Cl)n1 38891,c1(C(=O)OC)cccnc1N(C(C)CNC(=O)Cc1nnc(C)s1)C(C)C 38892,Cc1ccc(CC(N2CCCC2c2cnco2)=O)o1 38893,c1(SCC)ncccc1NC(=O)C(F)CC1CCN1C(=O)OC(C)(C)C 38894,C(c1cnccn1)=CC(=O)NC1C=CCN(C(=O)C(c2ccc(F)cc2)(F)F)C1 38895,c1(OC)ccc(N)c(C(=O)NC2CC(CNC(=O)C(C)c3ccsc3)C(O)C2)c1 38896,Cn1c(CC(=O)NCC2(CNC(=O)CC3CC(=O)NC3=O)CCC2)nnc1S 38897,C(=O)(C#CC1CCCCC1)N1C(C)(C(=O)NC2CC(CC)C2)CCC1 38898,O=C1CCC2(CN(C(=O)Cc3cc(Cl)ccc3Cl)C2)N1 38899,N1(C(c2[nH]ccc(=N)n2)=O)CC2CC1CC2NC(=O)CCNS(C)(=O)=O 38900,CCC(C)CCC(=O)N1CCCOC(C2CN(C(=O)C(CC3CCC3)OC)C2)C1 38901,CC(CC(N)=O)N(C(=O)CC1C(NC(c2nccs2)=O)CC1O)C 38902,CN1CCCCC1C(N1CCCC1CC(=O)NCCOC(F)(F)F)=O 38903,c1(CC(=O)NCC(C)N(C(c2ccc(COC)[nH]2)=O)C)cncc(C#N)c1 38904,CCC(CC(=O)NC1(c2nn[nH]n2)CCCN(C2C(COC)CCCC2)C1)C(C)(C)C 38905,C12(NC(CCC#C)=O)COC(C1)C(NC(=O)C(C)SCC)C2 38906,N1(C(CCOC)=O)CCC2C(CCN2C(c2cnc(F)cc2C)=O)C1 38907,N#Cc1csc(CNC(=O)CN(C(=O)C(O)C2CC2)C2CCC2)n1 38908,C1(COC)(NC(c2ccc(O)nc2)=O)CCCN(C(=O)C(O)P(C)(C)=O)C1 38909,c1(OC)cc(CNC2CN(C(=O)NC(C)C)CC2C)ccc1C 38910,C1(C(N2C(C=C)CCCC2)=O)CC2(CCN(C(=O)C(CC)N(C)C)C2)C1 38911,N1(C(c2c(SC)cn(C)n2)=O)CC(NC(C2CC(C)CCO2)=O)CC(O)C1 38912,C(=O)(C(F)(F)CCn1ccnn1)NC1C(NC(c2c(N)nccc2)=O)CCC1 38913,c1(NC(C)=O)ccc(Br)c(C(=O)NCCCNC(C2CC(C)=NO2)=O)c1 38914,c1(CCC)ncc(NC(C2CN(C(=O)CC(OCC)OCC)CC2F)=O)cn1 38915,c1(C(c2n(CC(=C)C)nnn2)NCCOC)snc(OC)c1Br 38916,N1(C(C2C(CC)CCCC2)=O)CC(C)N(C(=O)C(C)OCOC)CC1C 38917,C1(F)(CNC(C2CCN(CC(C)C)C2)=O)CCC(NC(=O)Cc2c[nH]nc2O)C1 38918,Cc1nn2c(c1CNC(=O)C(O)c1ccco1)CN(C(C1CCCSC1)=O)CC2 38919,c1(C(=O)OCC)cc(CNC(=O)NCCC2CCCC2O)cs1 38920,CCC(C(=O)NCCC1(C)CCN(C(=O)COc2ccsn2)CC1)C(F)(F)F 38921,N1(C(C2CN(C(C(C=C)OC)=O)CC2F)=O)CCCOCC1C 38922,c1(N2CCC(CC)C2)cc(=NCc2nc(=N)n(C)[nH]2)[nH]c(C(C)C)n1 38923,C1(C(N2C(CCNC(C(C(C)O)NC(C)=O)=O)CCCC2)=O)CCCC1C1CC1 38924,N1(C(CCSc2nc(C)[nH]n2)=O)CC2CN(C(=O)Cc3nccn3C)CC2C1 38925,Cc1cc(C(N2CCC(C)(NC(c3ncsc3C(C)C)=O)C2)=O)ccc1C(F)F 38926,N1(C(c2c(Cl)cnc(CC)n2)=O)CCC(C2CCN(C(C3CC3CC)=O)CC2)C1 38927,N1(c2n(CCC#N)c(C)nn2)CC2CS(=N)(=O)CC2C1.C1(C)CC1 38928,C1(OC(C)C(=O)NCC(C)(C)NC(=O)CC2CC3(CC3)C2)CCCCC1 38929,C1(C(=O)NCCC2CC(NC(C=CCOC)=O)C2)Cc2nccn2C1 38930,c1(C(=O)NC(C(C)NC(=O)CC2(CO)CC2)C)ccc(Br)c(F)c1F 38931,C1(CCNC(c2ncn(CC)n2)=O)CCN(C(=O)Cc2coc(C)n2)C(C)C1 38932,N1(C(C2(C)C(C)C2)=O)CC2CCN(C(=O)CCc3ccc(C(C)(C)C)cc3)C2C1 38933,C1(NC(c2c(C)cc(N)cn2)=O)CC2CCC1C(NC(C1CN(C)C(=O)N1)=O)C2 38934,c1(C(=O)NCC(C)(C)NC(=O)CC2(C)CC(F)(F)C2)c(Cl)ccc2c[nH]nc12 38935,C1(O)(C(=O)NC2CN(C(CNC(C3(C#N)CC3)=O)=O)C2)CCCCCC1 38936,C1(NC(c2c(NC)scn2)=O)CN(C(=O)C(CO)OC)C(C)(C)C1 38937,c1(C(=O)NC(C2(O)CCN(C(Cc3cnc(C)o3)=O)C2)C)c(F)ccnc1F 38938,C1(C(=O)OC2CN(C(CCc3ccc(OC)nc3)=O)C2)CCC(C)NC1=O 38939,CC1=CC(c2ccc(C(=O)NCC3(F)CCCCC3O)cc2)=C(C)S1=O 38940,C1(C(=O)NC(CC=CC)C(=O)NCC2(CCC)CC2)CCC2CC1CO2 38941,C(=O)(N=c1ccn(-c2ccnc(C#N)c2)[nH]1)c1c(C)cn(-c2c(C)ncs2)n1 38942,Cc1cc(C(N2CCN(C(C34CSC(C3)C4)=O)CC2)=O)c(N)c(F)c1 38943,C1(C(N2CCC(NC(c3c(SC)nccn3)=O)CC2C)=O)CCCCC12CCC2 38944,n1(CC(N2CCN(C(c3c(C)cno3)=O)CC2CCO)=O)ncc2ncccc12 38945,Cc1ncc2n1CCN(C(=O)NCCCCOc1ccc(Cl)cc1)C2 38946,C1(O)(CNC(C#CC(C)C)=O)CCCN(C(C2CCC3CC2CO3)=O)C1 38947,N1(C(CCC(=O)OC)=O)CC2(CC(NC(C3CCSC(C)C3)=O)CO2)C1 38948,O=S(=O)(c1ccc(Br)cc1Cl)NC1CC(NCc2c(F)ccc(F)c2O)C1 38949,c1(C(N2CC(C)(NC(CCn3ccc(C)n3)=O)C2)=O)ccc(C(C)=O)c(C)c1 38950,N1(C(C=C(C)Cl)=O)CCC2(CC1)CN(C(=O)Cc1cnn(C)c1)CC2CO 38951,c1(C(=O)NC2C(NC(CC3CC(=C)C3)=O)CCC2)cnncc1C 38952,C1(NC(c2nn[nH]c2Cl)=O)CC2(CCN(C(=O)Cn3cccc3)C2)C1 38953,C(=O)(C1=CC2(CCOC2)C1)N(C1CCN(C(c2ccoc2Br)=O)C1)C 38954,CCCC(C)(O)C(=O)NCC1CCCC1NC(=O)CC1COCC(C)(C)O1 38955,N1(C(CC2ON=C(C)C2)=O)CCCCC1C(N1CCN(C(=O)C(C)C)CC1)=O 38956,C1(C)(C(=O)NCC(C)NC(c2ccc(-n3ccnc3)nn2)=O)CC(C)OC(C)C1 38957,c1(CCNC(N2C(COC)C(C)(C)C2)=O)cnc2n1CCOC2 38958,c1(OCC(=O)NC2CCCCC2CNC(c2cnc(O)s2)=O)nc(O)nc(O)n1 38959,C#CCCC(O)C(=O)NCC1CCCN1C(c1ccccc1C(=O)OC)=O 38960,N1(C(CCC(=C)C)=O)CCCC(O)(CCNC(=O)C(O)C(C)CC)C1 38961,C(C)(C(=O)N(CC(C)(C)NC(=O)CC=C(C)CC1CCCCC1)C)(C1CC1)OC 38962,c1(C(=O)NC(C(=O)NCC(C#C)OC)CCC)nn(C)cc1C#C 38963,C1(CNC(=O)C(F)(F)C2CC2)CC2(CO1)CN(C(c1ccc3c(c1)CCC3)=O)C2 38964,C1(C(=O)NCC2(CC)CCOC2)CN(C(=O)CN2CCNC2=O)C(C)(C)C1 38965,CCC(C#N)C(=O)NCC1CCCC(NC(C2(C(F)(F)F)CCOCC2)=O)C1 38966,Cc1cn2c(n1)CC(C(=O)NC1CCN(C(c3cnn(C)n3)=O)CC1O)C2 38967,C1(C2CCN(C(=O)CN(C)C(=O)C3CC3)C2)(NC(CC(CCC)C)=O)CC1 38968,C1(C)(CNC(=O)NC2N(C(=O)OC(C)C)CCC2)CCC(=O)NC1 38969,c1(C(=O)NC2CC3CN(C(C(COC)NC(C)=O)=O)C2C3)ccsc1S(C)(=O)=O 38970,N1(C(C(C)C2CC2)=O)CCc2ccc(C(N3CC(C)(C#N)C3)=O)nc2C1 38971,c1(C(N2CC(O)(CN(C(=O)CO)C)C2)=O)ccc(-c2cscn2)nc1 38972,C1(C(N2C(C(NOCC=CC)=O)CC(O)C2)=O)CC2C(C1)C2(C)C 38973,N1(c2nnc(C)o2)CC2CC(NC(=O)CCCc3ccccn3)C2C1 38974,N1(C(Cc2[nH]c(=N)sc2)=O)CCC(C2(NC(c3ccn4nnnc4c3)=O)CC2)C1 38975,c1(C(=O)NCC(CC)NC(=O)C(c2cccs2)SC)cccc2oncc12 38976,O=C1CCCc2cc(C(=O)NC3CN(Cc4cc(F)cc(F)c4)CC3F)ccc21 38977,c1(C(N(C2C(C)CCN(C(=O)CO)C2)C)=O)ccc(S(C)(=O)=O)cc1 38978,c1(C(N2CCN(CCNC(CCC=C(C)C)=O)CC2)=O)ccc2nn[nH]c2c1O 38979,C1(N(C)C(=O)NC2C3CC4C(C3=O)C24)CC2CCC(C1)N2C 38980,S(=O)(=O)(c1cccnc1NCc1ccc(C)s1)NC(CC)C(O)C(C)C 38981,CCCC(CC(=O)NCC1CCC(C)CC1)NC(c1sc(C)nc1C)=O 38982,C1(C)(CNC(c2c(C)cns2)=O)CCCN(C(c2ccc(C(C)C)cc2F)=O)C1 38983,c1(CC)cccc(C)c1C(N1CCC(C(=O)OC)C1)C(=O)NCC(F)F 38984,C=C(C)C(C)(C)C(=O)NC(C1CCN(C(C2CSC3(C)CCC(=O)N23)=O)CC1)C 38985,C1(C(C)C)CCN(C(C2CCCO2)=O)C(CNC(=O)CC(=O)N(C)C)C1 38986,Cc1ccc(-n2ncc(NC(=O)CSc3ccc(C(C)(C)C)cc3)c2C)cc1 38987,N1(C(C(CC2CCC2)NC(C)=O)=O)CCCCC1C1C(C(=O)O)C1 38988,N1(C2CCCN(C)C2)CCC2(CC1)CC2C(N1CCCC(CCO)C1)=O 38989,c1(C(N2CC(O)(CCNC(CNC(=O)NC)=O)C2)=O)c(C)[nH]cc([N+](=O)[O-])c1=O 38990,C1(NC(C(c2cc(C)sc2)(F)F)=O)CN(C(=O)C2CC2)C2CCCCC12 38991,C(=O)(CC(C)F)NC1C(NC(C(C2CCCCC2)OC)=O)C1 38992,C1(NC(c2ccc(C#C)c(C)c2)=O)C2CCCN(C(=O)CC(F)(F)F)C2C1(C)C 38993,C1(C(=O)NCC2C(NC(C(C3CCC3)OCC)=O)CC2)CCC(C)(C)CC1 38994,C(=O)(n1ccc(SC(CN2CCCC2=O)C2COC2)n1)OC(C)(C)C 38995,C(=O)(CCCC(CC)CC)N1CCN(C(C(COCC)C)=O)C(C)C1 38996,C(=O)(C1=CCN(C(=O)CC(C)(C)COC)CC1)N1CCCC(CC=CC)C1 38997,c1(COC)ncccc1CNC(=O)COCC1(F)CC1 38998,C(C)(C(C(=O)O)NC(=O)Cc1ccc(C(C)(C)C)cc1)SC 38999,C(=O)(CC(C)(C)n1cccc1)N(CCCCNC(C(C)c1cccs1)=O)C 39000,N1(C(C2CC(C)(C(=O)OC)C2)=O)CC(NC(=O)C=CS(C)=O)C(F)C1 39001,CC1CCC(C(N2CC(CCCCNC(=O)C=CCN3CCOCC3)C2)=O)S1 39002,c1(C(=O)NCC(CNC(c2ncn(C)n2)=O)OC)ccc(C(C)C)c(F)c1 39003,N1(C(CCNC(=O)NC)=O)CC2C(CC(=O)NCc3cccc(CO)n3)C2C1 39004,c1(C(Cc2cccnc2-c2ccncc2)N)ccc(Cl)cn1.CC(C)(Cc1cn(CCO)nn1)CO 39005,c1(NC(c2cn(CC3(CF)CC3)nn2)=O)onc2ccccc12 39006,N1(C(=O)Nc2cc(C)cc(C)c2)Cc2cccn2CC(C(N2CCSCC2)=O)C1 39007,c1(OC(CC)C)cc(C(N2CCCC(CNC(c3ccncc3)=O)C2)=O)ccn1 39008,CCC(F)(F)CC(=O)N1CCC(F)CC1C(N1CCC(C(C)(C)O)C1)=O 39009,C1(C(N(Cc2cn(-c3cc(OC)nnc3OC)nn2)O)=O)CCN2CCCCC12 39010,N12CCCOC(C1)C2=O.Cn1cc(OC2(CNC(=O)CCCN(C)C)CC2)cn1 39011,C(C)(C)(CCCCC(=O)NC(C1CN(C(C2CCO2)=O)C1)C)OC 39012,CC(C)(CN1CCOCC1)C(=O)NCC1(NC(C2(c3ccno3)CC2)=O)CC1 39013,C(C(C)(C)C(=O)NCC1CCC(C)(CC)O1)NC(C(C=C)C)=O 39014,CC(C)(CCF)C(=O)NC1C=CCN(C(c2cc(CCO)on2)=O)C1 39015,C1(NC(CSCCOC)=O)CC(O)CN(C(c2ccn(C3CC3)n2)=O)C1 39016,N1(C(C23C(C)(C)OCC2C3)=O)CCCC2(C1)CN(C(c1ncc(F)cc1F)=O)C2 39017,c1(CC)ccc(CNC(C2CC2C(N2CC3CC2C3c2ccccc2)=O)=O)cc1 39018,c1(OCC(N2C(C(=O)NC3(C)CC=CCC3)CCC2)=O)ccccc1C#N 39019,c1(C(N2C(COC)(CNC(=O)C(C)C(C)O)CCC2)=O)cc2[nH]nc(C)c2cn1 39020,c1(OC)ccc(C(C)=O)cc1NC(=O)CC1CCC(C(=O)O)N(C)C1 39021,c1(C(C)C(N2CCC(N(C)C(C3(C)CCCO3)=O)CC2)=O)ccc(Cl)c(Cl)c1 39022,c1(C(N2C(C)C(C(=O)N3CCCO3)CC2)=O)cc(C#N)ccc1N 39023,Cc1ccc(CNC(=O)CN2CCC(CC(=O)N(C)Cc3ccccc3)C2)s1 39024,C#Cc1ccc(OCC(=O)NCCC2(NC(C3CCN(C)S3(=O)=O)=O)CC2)cc1 39025,c1(C(N2CC(NC(c3cccnc3)=O)C(C(F)F)C2)=O)cc(=O)n2nccc2[nH]1 39026,c1(C(=O)NC2C=CC(CNC(C(C)(C3CC3)OC)=O)C2)nc(Cl)oc1C 39027,N1(C(CC(CC)OC)=O)CCOCC(C)(CNC(c2ccc(C)cc2SC)=O)C1 39028,c1(C(=O)Nc2sc(C(=O)OC)c(Br)c2)ccc(S(=O)(=O)C2CCC2)cc1 39029,c1(C(=O)O)ccc2nc(O)n(CCOC3CCCC3)c2c1.c12ncccc1N2 39030,c1(CN(CC)CC)cc(C(C23CNCC2C3)=O)no1.C1(C(=O)OC)(CN)CC1 39031,C1(NC(c2n[nH]cc2I)=O)CC12CCN(C(c1c(Cl)cc(F)cc1Cl)=O)CC2 39032,N#Cc1c(NCC2CCC(NC(C3CC=CCO3)=O)C2)cccc1F 39033,c1(CC)cc(C(=O)NC2C=CCN(C(C3CC(=O)N(CC)C3)=O)C2)c(C)nn1 39034,C(=O)(C(C(C)(C)C)OCCN(C)C)NCC(=O)N(CC(N1CCCC1)C)C.C(C)O 39035,C1(C)(CC(=O)NCCOCCCCC)CCN1C(=O)COCCCN=[N+]=[N-] 39036,Cc1cnc(Cl)c(C(=O)NC2CC3CN(C(c4ccc([N+](=O)[O-])[nH]4)=O)CC23)c1 39037,C(=O)(CS(C)(=O)=O)N(CC(O)CN(C)C(c1cc[nH]c1C1CC1)=O)C 39038,N1(Cn2cccc(O)c2=O)CCCN(C(CCCS(C)(=O)=O)c2nn[nH]n2)CC1 39039,n1(CC(=O)N(CC(C)(C)NC(COCc2cc(C)on2)=O)C)nc(C)c(O)c1C 39040,c1(C2C3(CC3)C(C)N2)nnnn1C1COC1.c1(CO)cccs1 39041,c1(C(=O)NC2COCC2NC(c2ccnnc2O)=O)cccc(CCO)c1 39042,C(=O)(CCC(=O)N1CC(O)(CNC(C2C(Cl)(Cl)C23CC3)=O)C1)OC(C)(C)C 39043,C1(CN(C(=O)C2=CCC2)C)CCCCN1C(c1c[nH]c(-c2ccc(F)cc2)c1)=O 39044,c1(C(N2C(CNC(=O)COC3CCOC3)CC2)=O)ccnc(S)c1 39045,c1(C(=O)NC(CNC(c2nc(OCC)sn2)=O)(C)C)ccc(OC)c2ccsc12 39046,c1(C(C)C(=O)N2CC(CCNC(=O)C(C)C(F)(F)F)C2)cccc(C#N)c1 39047,C1(C(=O)NCCCOCCC=C)CCCCC1NC(c1cccc(OC)c1)=O 39048,N1(C(CCCC2C(C)C2)=O)CCC(C2CC2)C1C(=O)NOCCC(C)O 39049,c1(CNC(c2cccc(-n3c(C)c(C(=O)O)cn3)c2)=O)cn2cccc(C)c2n1 39050,N1(C(C2N(C(Cc3ccn(CC)n3)=O)CC2)=O)CC2CCC2(C)C1 39051,C(=O)(C(=O)N=c1cc(C)o[nH]1)NCC(CC)NC(c1ccc2c(O)n[nH]c2c1)=O 39052,C(C)(N=c1nc2c(ncn2C)c(NC(C)CS(N)(=O)=O)[nH]1)c1n(CC)ncc1 39053,c1(C(N(c2nc(OC)c(F)cn2)C2CCCNC2)=O)cc(O)ccc1[N+](=O)[O-] 39054,c1(C(=O)NC2CC(NC(c3c(C)nc(CC)o3)=O)CC2O)cc2n(n1)CCOC2 39055,c1(CC(N2CCN(C(CC(=C)C)=O)CC3(C2)CC3)=O)nc2nc(C)cc(C)n2n1 39056,c1(C(=O)NC2C(CNC(=O)CCC3CC3)CCC2)ccc(C(F)(F)F)nc1O 39057,c1(C(=O)NCCC(=C)CNC(C2(c3ccccc3)CC2)=O)ccc(C)c(O)c1 39058,C(=O)(C(C)(C)CCCO)NCC1CC2CN(C(c3cccc(OC)n3)=O)CC21 39059,N1(C(C2CN(C(COCCCC)=O)CC(C)(C)C2)=O)CCC(O)C12CCCC2 39060,C(=O)(C1=CC2CCC(C1)C2)N1CCC(C)CC1C(=O)NCCn1nccn1 39061,CCC(CC)C(=O)N1CCCCC1C(=O)N(CCN1CCCC1=O)CC 39062,C(CC(C)(C)CC(=O)NCCCCCN(C)C(c1cc(C2CCC2)[nH]n1)=O)OC 39063,Cc1ccnc(C)c1NC(C12CCC1CN(C(=O)Cc1c(C)nn(C)c1C)C2)=O 39064,C12(CCOCC1)C(=O)N2.c1(CNC(C2CCC2)=O)ccccc1C1CCNCC1 39065,CC1CN(C(c2cccnc2CO)=O)CCN1C(C1CCS(=O)(=O)CC1)=O 39066,c1(CC(=O)NC2C(CNC(=O)C=CC3CCC3)C2)nc([N+](=O)[O-])n[nH]1 39067,C(=O)(CCCCCCC=C)N1CC(CC#C)(C(=O)NC2CC(=O)N(CCC)C2)C1 39068,N1(C(c2ccc(CNC(N)=O)s2)=O)CC2CC1CCC2O 39069,CC(C)CN=C(NCc1nnnn1CC1CC1)NCC(c1ccnn1C)O 39070,Cc1cnc(C(=O)NC2COCCC2NC(=O)CCC(C)(C)F)c(C)c1 39071,Cc1scc(C(N2CC(NC(C3(C4CCCO4)CCCC3)=O)C(O)C2)=O)c1N 39072,c1(NC(=O)NCCC)ccc(C2CC2)cc1.C12CC(C1)C(=O)NC2 39073,CC(C)C1C(=O)N2CC3CC2C3C(=O)N1.C(=O)(C(N)=O)NCCSCOC(C)(C)C 39074,C1(NC(C(CCC)OC)=O)CC2CN(C(c3cn(C)c(=O)n3C)=O)CC2C1 39075,Cc1cnc(C#N)c(-c2c[nH]nc2C(=O)NCc2cc(F)c(F)cc2Br)c1 39076,CC1C(NC(C2COCCN2C)=O)CCCN1C(c1[nH]ncc1C#N)=O 39077,N1(C(C2(CC#C)CC2)=O)CCN(C2CCCN(C(c3c[nH]ccc3=O)=O)C2)CC1 39078,CC1(C(=O)NC(C2CCCC2)CNC(=O)Cc2ccc(Cl)nc2)CC=CCO1 39079,c1(C(C)C)ccc(C(N2CC(N(C(=O)CC3CC=CCC3)C)C2)=O)cc1 39080,C1(C)(COC(c2c(C)ccnc2C(C)C)=O)CC(C2CC2)=NO1 39081,c1(SC)ncccc1NC(=O)CCC1CCCN(C)C1 39082,C1(C(N2CC(=C)C2)=O)CCN(C(=O)CCCc2cccs2)C1 39083,c1(C(N2CCC(C)(CNC(C3CS(=O)(=O)C3)=O)C2)=O)c(F)ccc(Cl)c1N 39084,c1(C(N(CCCNC(C(C)SCC)=O)C2CC2)=O)cc(O)c2[nH]c(C)nc2c1 39085,C1(O)(CNC(CC2(CSC)CC2)=O)CCCN(C(c2csc(C#N)c2)=O)C1 39086,c1(C(C(N2CCC(C(F)F)(CNC(C)=O)C2)=O)C)ccccc1S(N)(=O)=O 39087,C1(NC(CCCC(=O)OC)=O)C2CC(CN(C(C3(CF)CC3(F)F)=O)C2)C1CO 39088,C1(OCC(=O)NC(CC(C)NC(CC(C)OC)=O)C)CCCCC1NS(C)(=O)=O 39089,c1(CNC(=O)CC(=O)NC2CC2)cc2n(n1)CCN(C(C1CC(C3CC3)C1)=O)C2 39090,N1(C(C2C=C(C)CS2)=O)C2CCC1CC(C(=O)NC(C)C(C)F)C2 39091,C1(CNC(C2ON=C(CC)C2)=O)CC2CCC1N2C(c1cc(C)ccc1C)=O 39092,N1(C(c2ncn(CC)c2)=O)CCC2(CCN(C(c3cnoc3CC(C)C)=O)C2)C1 39093,C1(OC(C(=O)NCCC2CC(NC(C(CSC)O)=O)C2)C)CCCCCC1 39094,c1(C(N2CCC(NC(c3c(C)onc3C(F)(F)F)=O)C2C)=O)ccc([N+](=O)[O-])[nH]1 39095,C1(C(=O)NC(C)(C)CNC(c2c(C(F)(F)F)ncn2O)=O)CC(=O)OC1(C)C 39096,c1(C(CC)(C)C)cn(CC2CC(NC(=O)C(F)OC(F)(F)F)C2)nn1 39097,C1(C(N2CC(C)N(C(C3CS(=O)(=O)CCO3)=O)CC2)=O)Cc2nccnc2C1 39098,CC1=NNC(=O)C1CC(N1CCCCC1CNC(C1(c2ncco2)CC1)=O)=O 39099,CS(=O)(=O)C1CCN(C(C(=O)NCc2ccccc2)C2COC2)C1 39100,C(=O)(CC(CC(C)C)NC(=O)C(CCC)=CCC)NC1(CC=C)CC1 39101,CC1CCN(C(=O)CC2CCCN(C(=O)NCc3ccc(Br)cn3)C2)CC1 39102,c1(C(=O)NC2C(C)CN(C(c3c[nH]nc3F)=O)C2)n[nH]c2c1CCCC2 39103,n1(CC(N2CC(NC(C(C)SCCCC)=O)C(C(F)F)C2)=O)ccc([N+](=O)[O-])n1 39104,c1(C(=O)OC)cccc(C(=O)NC(CO)C(C)NC(C2CCS(=O)(=O)N2)=O)c1 39105,C(=O)(CCS(=O)(=O)N(C)C)NC(CNC(c1ccc(OCC)nc1)=O)(C)C1CC1 39106,C1(C(=O)NCCCC(C)NC(c2sccc2C2CC2)=O)CC2CC1CC2O 39107,C1(CNC(c2c(C)cc(C)[nH]2)=O)(NC(c2c(C)ccn2C)=O)CC2CCC1CC2 39108,Cn1cc2c(C(=O)NCCC3=CCN(C(=O)CSCC(N)=O)CC3)cccc2n1 39109,CC(C)CC(CC(C)C)NC(=O)CCCC(C)NC(=O)Cc1ccc[nH]1 39110,C12(CNC(c3ccc(C)nn3)=O)CC(NC(c3nc(Br)c[nH]3)=O)(C1)C(C)O2 39111,Cc1cc(C(=O)NCCC2CN(C(=O)C=Cc3ccco3)C2)sc1C 39112,c1(C(N2CC3CCN(C(CSCC(C)C)=O)C3C2)=O)cc(=O)c2ccncc2o1 39113,c1(C(=O)NC)ccnc(CN(C(c2cocn2)=O)CC2C3CNC2C3)c1 39114,c1(N2CCN(C(C)(C)CO)CC2)nc2ccccc2nc1NCc1ccccn1 39115,C1(C(=O)NC2(CO)CN(C(CC3(C)CCC3)=O)C2)CNC(=O)CC1(C)C 39116,N1(CCC(=O)NCC(CC)(C)NC(c2cnc(C(C)O)s2)=O)CCCCC1=O 39117,C12(C(=O)NC(CCCC)C)CCCC1CN(C(C1(COC)CC(=O)C1)=O)C2 39118,C1(C(C=CC(=O)N(CC(CNC(=O)C=CCOC)O)C)=O)CCCN(CC)C1 39119,N1(C(C(Cn2ccnn2)NC(C2(CC)CC2)=O)=O)CCCN(C(C)=O)CC1 39120,Cc1cc(C(=O)NCC2CC2NC(=O)Cc2nc(C(C)C)c(C)s2)c(N)c(Cl)c1 39121,N1(C(Cc2cnc(C)[nH]2)=O)CCN2C(=O)C(NC(=O)CSCCC(C)C)CC2C1 39122,C1(N2C(=O)c3ccc(N)c(c3)C2=O)CC1C1CCOCC1.N1(CC)CCCC1 39123,Cc1cccc(C2CC2C(=O)NC(C)(C)CNC(c2ncccc2N)=O)c1Br 39124,Cc1nc(C)n(CCCC(=O)N(CC(C)NC(=O)Cc2sc(C)cc2C)C)n1 39125,c1(CCC(=O)NCCNC(c2c(C)noc2)=O)nc(O)c2c3c(sc2n1)CCC3 39126,C1(C)(C(N2C(C)(CC(=O)NCCc3n(C)cnn3)CC2)=O)CCNC1=O 39127,S(=O)(=O)(c1cccc(Br)c1)NCCC(=O)NC(Cc1c(F)ccc(Cl)c1F)CO 39128,CC1C(NC(=O)C=Cc2ccccc2)C(C)CCN1C(C1CCC=CO1)=O 39129,Cc1nc2ccc(-c3nc(C(F)F)nn3C(C)C(C)C)cc2n1C 39130,N1(C(C(C(=O)OCC)F)=O)CC2CCC(C1CO)N2C(=O)CCCc1ccsc1 39131,c1(C(N2CC(CC)N(C(=O)CCSC3CCCC3)CC2)=O)cc(O)cc(C#N)c1 39132,Cc1c(C(N2CCCC23CCN(C(C2CCCN2C)=O)C3)=O)nn2ccccc12 39133,N1(C(CCOCC)=O)CC2C(CN(C)C(C3(CF)CC(F)(F)C3)=O)C2C1 39134,N1(C(C(C(CC)C)O)=O)CCC2CN(C(=O)C(C)S)CCC12 39135,c1(C(=O)NCC2CN(C(CCCCSC)=O)CC2O)cc2cc(Cl)ccc2[nH]1 39136,C1(CNC(=O)C(=O)NC2CC2)CN(C(=O)CCC2OCCO2)CC12CCOCC2 39137,C(=O)(C(CC(F)F)NC(C1CN2CCC1C2)=O)NCC1(F)CCN(C)C1 39138,O=C1NC(=O)C(C2CC(C(=O)NCCCN3CCCC3)C2)N1 39139,N1(C(c2ccc(N)c(F)c2)=O)CC2ON=C(CNC(=O)CCc3nccs3)C2C1 39140,C1(C(C)C)C(=O)N1.N1(C2CN(NC(C)=O)C2)CCN(C(=O)CCC=C(C)C)CC1 39141,C12(C(=O)NCC3C(C)CCN(C(=O)COCCN(C)C)C3)CC(C)(C1)OC2(C)C 39142,C1(C2CCN(C(=O)C(=Cc3c[nH]cn3)F)C2)(NC(C2C3COCC23)=O)CC1 39143,Cc1scc(C(=O)NC(Cn2cccn2)C(=O)NCC2([Si](C)(C)C)CC2)c1C 39144,c1(C(=O)NC2C(NC(C3CCCC(C)(C)C3)=O)COC2)nc2cc(O)ccc2[nH]1 39145,CC1CCCc2ncc(C(=O)NC3CN(C(C4CC5CC4C5)=O)CC4(CC4)C3)n21 39146,N1(C(C(CC)C(C)C)=O)CCC(NC(=O)CNS(=O)(=O)CC)C(C)(C)C1 39147,Cc1ccc(C=CC(N2CCCC(NC(=O)CC3C=CCC3)C2C)=O)nc1 39148,C1(C)(C(=O)NC2CC(C(N(C)C)=O)C2)C=CCN1C(c1cc(C(F)F)no1)=O 39149,c1(C(N2CC(C(C(=O)NCC)OCC)C2)=O)sc(Br)cc1OC 39150,C1(C(=O)OC)CC(NCc2cc(Br)co2)C12CCC2 39151,N1(C(C(CC)CC)=O)CCC2(CC1)CN(C(C1CCCC13CC3)=O)CC(C)O2 39152,C1(NC(C)C)CC(NC(C2COCCN2C)=O)C12CCC2 39153,C1(C(N2CC=CC(C(N(CCC)C)=O)C2)=O)CC(C)(C)CN1C 39154,c1(OCCC(=O)N(CCN(C(CCC=CC(C)C)=O)C)C)c(F)cccc1Cl 39155,C1(CNC(C=CC(=O)OCCCC)=O)CN(C(=O)CC)C2CCN1C2 39156,C1(N(C)C)CCCC(N=c2[nH]c(=NC3CC(N4CCC4)C3)[nH]c3c2COC3)C1 39157,N1(C(=O)CC2CC(F)(F)C2)CCC2CCN(C(C3CC4CC3C4)=O)C2C1 39158,CC1CCC(NC(=O)CCC2(C#N)CCC2)CN1C(=O)CC1(N2CCCC2)CC1 39159,C1(NC(c2cc(C)nn2CCO)=O)CCC2CC1CN2C(=O)CCN(C)CCO 39160,c1(C(N(CC2CCN(C(c3c(CC)noc3)=O)CC2)CC)=O)cncc(Cl)c1C 39161,N1(C(c2ccc(C(C)C)c(Cl)c2)=O)CCN(C(c2cnncc2O)=O)C2(CC2)C1 39162,c1(OC)ccc(Cl)c(CC(=O)NC2CC(CCNC(=O)CCc3cc[nH]n3)C2)c1 39163,Cc1cc(=NCCCS(=O)(=O)C(F)F)[nH]c(N2CCC(C(C)C)C2)n1 39164,N1(C(CS(N)(=O)=O)=O)CCC2CCCN(C(=O)Cc3cccc4[nH]ncc34)C2C1 39165,C1(C(=O)NCCN(C(C(N2CCOCC2)C)=O)C2CCCC2)CC(F)(CF)C1 39166,C(=O)(C(C)S(=O)(=O)C1CCOCC1)NCC12N(C(C(C)NC(C)=O)=O)CC(C1)C2 39167,c1(C(=O)NCC(CC)NC(c2cn(CC)nn2)=O)cn(C)nc1CCC(F)(F)F 39168,c1(OC)noc(C2CC2)c1C(=O)NCC1CCCN1C(C1CC2CC2C1)=O 39169,c1(-c2cn(CC(COCC)(C)C)nn2)cc(C(=O)OC)ccc1NC(C)=O 39170,CCC(C)CCCC(=O)NCC(CNC(=O)Cc1cc(O)nnc1O)OC 39171,N1(C(C2OCCN(C(C3(C)ON=C(C)C3)=O)C2)=O)CCC2(CC1)CSC2 39172,c1(C(N2CCC(C)(NC(CN(C(C)=O)C)=O)C2)=O)nn(C)c(C)c1N 39173,c1(C(=O)NCc2c(C(=O)NCCC(CC)CO)n[nH]c2)cccc2ccoc12 39174,C(=O)(CC1=Cc2ccccc2C1)NCC(CC)(C)NC(=O)CCCc1cnn[nH]1 39175,Cc1nc2cc(C(N3CCCC3CCCNC(=O)C(C)N(C)C)=O)ccc2s1 39176,C1(NCc2c(C)c(Br)ccn2)CCCC2CN(C(=O)OC(C)(C)C)CC12 39177,C1(C(N(CC(C)OC)C)=O)COCCN1C(=O)C(CO)OC 39178,C1(NC(C(n2cc(C3(C(N)=O)CC3)nn2)C)=O)C(C)(C)C(N(C)C)C1(C)C 39179,N1(C(C=CCCC=C(C)C)=O)CCC2(CCCN2C(=O)Cc2ncc(F)cn2)C1 39180,c1(C(N2CCCC2CCC#N)C(=O)NC(CC)C)cnc(C2CCC2)s1 39181,C1(C(N(C2CCN(C(C3C(C)CCO3)=O)C2)C)=O)CCCN(C)C1 39182,CC1(C)CCN(C(=O)C2=NOCC2)CC1NC(=O)CCn1cc[nH]c(=O)c1=O 39183,N1(C(Cc2c(C#C)cccc2)=O)CC2(C1)CN(C(c1coc(C)c1)=O)CCO2 39184,c1(-c2cn(CCC(=O)NC(c3ccccc3)CC)nn2)cc[nH]c(=N)c1 39185,c1(C(N(CC(C)NC(=O)CNC(c2ncccc2O)=O)C)=O)nnc(O)cc1O 39186,C(=O)(CS(=O)(=O)c1ccccc1Cl)NC1CCC(F)(CNC(C(CC#C)O)=O)C1 39187,c1(C(N2CC(CCC)N(C(c3cncs3)=O)CC2)=O)ccc(Cl)c(F)c1O 39188,CC1(C)CN(C(c2csnc2Cl)=O)CC1C(=O)NCc1ccccc1Cl 39189,C1(C(N(CC(C)CNC(c2sc(Cl)cc2Cl)=O)C)=O)CCCC1C1CC1 39190,C1(CNC(C2(SC)CC2)=O)CCC(C)CN1C(c1ccc(C2CC2)o1)=O 39191,c1(C(=O)NCC(CO)NC(C2CCC(C(=O)OC)O2)=O)cnc(C2CC2)nc1O 39192,C(CCN=c1nc2scnc2c(NC(C2CC(F)(F)C2)C)[nH]1)N(C(C)C)C 39193,C(=O)(C(CC(C)C)NC(N)=O)NCC(C1CC1)NC(CC1C(C(=O)OC)C1)=O 39194,N1(C(CCC=C)=O)CC2C(C(F)(F)F)CC2(NC(c2ccc(C)c(C)c2O)=O)C1 39195,N1(C(C(=O)N(C2CCC2)Cc2ccc(Cl)s2)c2cnsc2)CCCCCC1 39196,c1(OCC(=O)NC2C(NC(c3cnc(C(C)C)[nH]3)=O)C2)ccc(F)c(Br)c1 39197,N1(C(COCCN(C)C)=O)CC(C)(CNC(C2CCCCCCC2)=O)CC1(C)C 39198,c1(C(=O)NCC2CN(C(=O)CCC3CCCC(O)C3)C2)cc(Cl)c(F)cc1Cl 39199,Cc1nc(C2CC2)nc(S)c1C(=O)NC1CCN(C(=O)CC2OCCOC2(C)C)C1 39200,N1(C(C2CCC(=O)N2)=O)CCC(C2CCN(C(C3CN4CCN3CC4)=O)CC2)C1 39201,C1(SC(CCNC2(C(=O)OCC)CC2)=O)CCC(F)(F)CC1 39202,C#CCC(C)(CC)C(=O)NCC1CN(C(c2ncsc2C2CC2)=O)CC1(C)C 39203,C1(N=c2[nH]n3cc(C)nc3s2)(CCNC(CCCC(CC)(C)C)=O)CCC1 39204,N1(C(C2=C(C)CC2)=O)CCC2(CC1)C(NC(c1cccc(F)c1C)=O)CS2(=O)=O 39205,CCCCCCC(C)CC(=O)NCCS(=O)(=O)Cc1cn(C2CCOC2)nn1 39206,CC1CC(C(=O)NC(C)(C)CCCNC(=O)Cc2cnc[nH]2)CCS1(=O)=O 39207,CC1CC(NC(C2(CF)CCC2)=O)CN(C(=O)CC2CCCCO2)C1 39208,CC(CF)CC(=O)N1CCCC(CN(C(=O)Cc2cccn2C)C)C1 39209,N1(C(CNC(CCCCC)=O)=O)CC2CN(C(C3(C(F)F)CCCO3)=O)CCC12 39210,C1(NC(c2cc(C(=O)OC)no2)=O)CC(F)(F)CC1NC(=O)Cc1scnc1C 39211,c1(OC)ccnc(O)c1C(N1CC(CNC(=O)C=Cc2ccnn2C)C1)=O 39212,N1(C(C(CC)O)=O)CCN(CC2CCN(C(=O)CCCc3ccsc3)CC2)CC1 39213,c1(C(=O)NCC#CCNC(CC2C(C)CCC2)=O)cnc(C(F)(F)F)c(F)c1 39214,N1(C(c2c(CC)nc(C)nc2)=O)CCCC2(C1)CN(C(=O)CC1=CCCCC1)C2 39215,C1(CC=C)(CNC(c2c(Br)ncn2C)C2CC2)CCN(C(=O)OC(C)(C)C)CC1 39216,C1(C(=O)NC(C(C)NC(C2CC3CC3C2)=O)CO)CC(C)(C)CO1 39217,C(c1cccc(C#N)c1)=CC(N1C(CNC(C(NOC)=O)=O)CN(C)CC1)=O 39218,N#Cc1cccc(Nc2nnc(Cc3ccc(Cl)cc3)n2Cc2ccsc2)c1 39219,C1(C(N(CC(C(C)C)OC)C)=O)C=CCN(C(C2CCC=CCC2)=O)C1 39220,C1(C(C(=O)N(CCC=C)CCOC)C)CCN(C(=O)CC2(OC)CCC2)C1 39221,CC(C)(CCNC(C1(CO)CCCO1)=O)NC(C1CCCO1)=O 39222,CC1CC(N(C)C(C2CC(O)CN2C(=O)C(F)CC2CCOC2)=O)CCO1 39223,C1(C(N2CC3C(C(N4CCCC(C(=O)OC)C4)=O)(C3)C2)=O)CC(C2CC2)=NO1 39224,c1(C(=O)O)ccc2c(C(N3CC(Oc4ccccc4)C(O)C3)=O)cnn2c1 39225,C(C(C)(C)C(=O)NC1CCCN(C(=O)CCNc2ccccc2C)C1)SC 39226,n1(CC)cccc1C(=O)NC(C1CCN(C(C2(F)CC=CC2)=O)C1)C 39227,C1(C(=O)NCCCCCCOC)CC2(CCC2)CN1C(C12CC(F)(C1)C2)=O 39228,C(=O)(C1=COCCO1)NCC(CN(C(c1ccc(C2CC2)cn1)=O)CC)(C)C 39229,c1(C(N2C(C(=O)NCC3CC(=O)NC3)CC(F)C2)=O)nccc2ccccc12 39230,N1(C(C(C)OCCOC)=O)CCN(C)C(C(=O)NC2CC(CO)(CO)C2)C1 39231,C1(CC=C)(C(=O)NC(C=C)C2CCC2)CCCN1C(=O)C(C)CSC 39232,Nc1cncc(C(=O)NC2CC(NC(c3cc[n+]([O-])cc3)=O)C(O)C2)c1 39233,S(=O)(=O)(c1cccc(Cl)c1)N(CC(N1CCN(C(C(CC)OC)=O)C(C)C1)=O)C 39234,N1(C(C(C(C)C)OC)=O)CC2(NC(=O)C(CO)NC(=O)C(C)C)CCC1CC2 39235,CC1CCCN1CC(=O)N(CC(=O)NC(c1cccnc1)CO)C1CCC1 39236,N1(C(C2CC(CC)C2)=O)CCN(C(=O)COc2ccc(C(N)=O)cn2)C(CO)C1 39237,C1(C(=O)NCC(C)NC(c2snc(OC)c2Br)=O)CCOC(=O)CC1 39238,N1(C(C(C=C=C)C)=O)CCCC(CC)(NC(c2cc(Cl)ccc2Cl)=O)C1 39239,C1(NC(C=C(C)C(C)C)=O)CCC(CNC(=O)CCc2ncc(F)cn2)CC1 39240,C1(C)(OC)CCCN(c2cc(NCc3nc(C)c(C)o3)nc(C(F)(F)F)n2)C1 39241,CC1CCN(C(c2n[nH]cc2Cl)=O)CCN1C(=O)CCCS(N)(=O)=O 39242,c1(N2CCC3(C(NC(C=C(C)C(=O)O)=O)CC3)CC2)ncc2c(Br)cccc2n1 39243,c1(NC(=O)CC2CC(NC(=O)Nc3cn[nH]c3)C2)ccc(-c2ccccn2)cc1 39244,c1(C(c2nn[nH]n2)NC(c2ccc(C(F)(F)F)s2)=O)cccc(F)c1 39245,C(=O)(C(C(C)(C)C)NC(C)=O)NCCN(C(CC1(OC)CCC1)=O)CC 39246,C(=O)(CS(=O)(=O)CCO)N1CCC(C)(CNC(C2C(CC(C)C)C2)=O)CC1 39247,N1(C(c2n(C)c(Cl)cn2)=O)CCCC2(CCN(C(=O)CC3CSCCS3)C2)C1 39248,C(=O)(C1=CCCCO1)NC(CCOC)C(=O)N1CC(C)=C(C)C1 39249,C1(C(=O)NCC2N(C(CN3C(C)CCC3)=O)CCC2)CC(S(C)(=O)=O)C1 39250,CC1CN(C(C2COC(C)(C)O2)=O)CC2(CCN(C(=O)CN3CCC3)C2)O1 39251,CC(C)CC(O)CC(=O)NCC(C(N1CC(CO)CC(C)C1)=O)N(C)C 39252,N1(C(c2cncc(C(F)(F)F)c2)=O)CCN(C(=O)CCn2ccnc2)C(CF)C1 39253,C1(C)(C(=O)NCC=CCNC(C=C(CC)C)=O)CCCC1O 39254,N1(C(c2c(CC)[nH]cc2)=O)CCC(NC(C2CN(C3CCOC3)C2)=O)C(F)C1 39255,N1(S(C2CCC(C(=O)OC)C2)(=O)=O)CCc2cc(C)ccc2C1C 39256,N1(C(c2cccc(F)c2Br)C(=O)NC)CCc2cc(F)cc(Cl)c2C1 39257,N1(C(=O)Cc2sccc2Cl)CCCC(N(CCO)C(C2CC(F)C(=O)N2)=O)C1 39258,c1(C(N2CC(OC)(CNC(C3CC4CC4C3)=O)C2)=O)cc2c(Cl)cc(F)cc2[nH]1 39259,N1(C(C(c2ccn(C)n2)C)=O)CC=CCC1C(=O)N(C)CC1(C)CC1 39260,CC(C)CCCC(C)C(=O)NC1(C2CCCN2C(c2cnc(C(C)C)o2)=O)CC1 39261,N1(C(c2c(CC)occ2C)=O)CC2CC(CNC(c3ccc(C#N)n3C)=O)C2C1 39262,C1(N(C(C)=O)C(C2CCN(Cc3nc(C(=O)O)co3)C2)=O)CCS(=O)(=O)C1 39263,C(=O)(C(C)(C(C)C)NC(C)=O)N(CCNC(C1(C(=O)OCC)CCC1)=O)C 39264,N(C1CCCn2ccnc21)C(C(C(C)(C)C)NC(CC(C)n1cccc1)=O)=O 39265,n1(C(C)C)ncc(C(N2CCC(CF)(NC(=O)CC3CCCC(=O)N3)C2)=O)c1Cl 39266,N=c1ccn(CCC(=O)NCCC2(CNC(=O)Cc3ccccc3)CC2)[nH]1 39267,c1(C(N2C(CNC(C3C(C)OCCO3)=O)CC2)=O)cc(=O)cc(Cl)[nH]1 39268,c1(C(=O)NCC(C)(C2CCC2)NC(c2cc(C3CC3)ncn2)=O)ccc(F)cc1 39269,N1(C(C2(CC)CCCC2O)=O)CCCN(C(c2oncc2C)=O)CC1 39270,C1(CNC(CCCOCCOC)=O)CCCN(C(c2ccc(F)c(N)c2)=O)CC1 39271,c1(C(N2CC(C)(C)C2Cn2cc(CCCOCCO)nn2)=O)cnn2ccsc12 39272,N1(C(CCOCCNC(C2C(=C)C2)=O)=O)CC(C)OC(C)(C)C1 39273,N1(C(C(C2CCCC2)OC)=O)CCC(NC(c2cc(C(C)C)on2)=O)CC(O)C1 39274,C(=O)(NNc1c(C#N)cc(C(F)(F)F)cc1[N+](=O)[O-])CCc1onc(C)n1 39275,CC1CCCC(N2CCN(C(c3ccoc3)=O)CC2)C1 39276,c1(CN2CCN(C(C3(CC(C)C)CC(=O)C3)=O)CC2)nc2ccccc2o1 39277,c1(C(=O)NCCC2N(C(C(C)OCC#C)=O)CCC2)ccc(OC(F)(F)F)cn1 39278,Cc1noc(C)c1NNC(=O)C(c1ccccc1Br)NC(=O)OC(C)(C)C 39279,c1(CN(C)C(C2(C)CC2)=O)cnn2c1CN(C(c1cc(F)ccc1F)=O)CC2 39280,C(=O)(C(O)C(F)(F)F)NC(CN1CCN(C(C(COC)(C)OC)=O)CC1)(C)C 39281,C(=O)(C1=CCC(C)(C)CC1)N1C(CNC(c2cc(C(C)=O)sc2)=O)CCC(C)C1 39282,c1(C(N2CCC(O)(CNC(CCCC=C)=O)C2)=O)ccc2c(c1)SCCN2 39283,C1(C(=O)NCC(CC)NC(=O)C(c2ccc(F)cc2)(C)C)CCCCN1N=O 39284,C(=O)(C(Cn1ccnn1)NC(c1cc(C2CC2)[nH]n1)=O)NC(CCOCC)C 39285,c1(CN2C3(c4cn(CC(C(CC)O)C)nn4)CC(C2)C3)csc2cc(C)ccc12 39286,c1(C(N2CC(CCO)(NC(c3ccn(C4CCC4)n3)=O)C2)=O)ccc([N+](=O)[O-])o1 39287,C1(O)(CC(N2CC(O)(CCNC(C(C=C)(C)O)=O)C2)=O)CCN(C)CC1 39288,C1(C(=O)NC(C(C)C)(C)CNC(=O)CC2CC3(CC3)CO2)CC2(C1)CC1(CCC1)C2 39289,C(c1ccc(N(C)C)cc1)=CC(=O)NC(CC=C)CNC(c1cc(C#N)cs1)=O 39290,C=C(C)CC(C(=O)N(CCC(=O)NC(CSC1CC1)C(=O)NC)OC)OC 39291,N1(C(c2ccc(OC)cc2O)=O)CCC(C)C(NC(=O)CSCC(N)=O)C1C 39292,N1(C(C(CCCNC(C2C(C(=O)OC)CC2)=O)O)=O)CCC12CCCCC2 39293,CCCCCCC(F)C(=O)N1CCC(C)(CNC(c2ccc(O)c(N)n2)=O)C1 39294,c1(C(N(CCOCCNC(C2C(C=C)C2)=O)C)=O)cccc(C(C)C)c1N 39295,Cc1scc(C(=O)NC2CCC(N(C(=O)C(c3cccnc3)C)C)CC2)c1N 39296,n1(CCC)nc(C)cc1C(=O)NCCOC1CN(C(=O)C(N2CCOCC2)C)C1 39297,c1(CC(=O)NC2CC(NC(c3c(COC)nn(C)c3)=O)C2)c(C)cccc1C 39298,c1(OC)cc(C=CC(=O)NCCN(C(C2(O)CCSC2)=O)C2CC2)ccc1OC 39299,Cc1cccc(CC(C)(C)S(C)(=O)=O)c1C(C)(C)C.c12nc(nn1-c1ccccc1)C2 39300,c1(N2CCCN(CC)CC2)nc(N(C)Cc2cncn2C)c2cnn(C)c2n1 39301,C1(C(=O)NCC(C)N(C(C(C(=O)OCC)CC)=O)C)CC2(C1)CC(F)(F)C2 39302,C(C(=O)NOCC(=O)OCC)=CCC.C1=CC(=O)NC1(C)C 39303,C(=O)C(CC(C)C)ONC(C1(C)CCSCC1)=O.c1(CN(C(C)=O)CC)ncc[nH]1 39304,C1(NC(c2c(OC)ccnc2)=O)CCCC2CN(C(C3(C)CCCC3C)=O)CC12 39305,n1(CCC(N2CCN(C(CSCCOC)=O)C(C)C2)=O)c(=O)oc2ccccc12 39306,c1(OC)nc(Br)ccc1NC(C1(F)CCN(C(c2ccccc2O)=O)C1)=O 39307,c1(C(c2n(CCC)nnn2)NCCCCOC)cccc2nccn12.C(CO)S 39308,Cc1cccc(OCC(N2CC(NC(C3(O)CCOCC3)=O)CCC2C)=O)c1C 39309,C(=O)(CCN=c1[nH]ccs1)NC1C(NC(C2C3CC(C)(C3)OC2)=O)CCCCC1 39310,n1(CC(=O)N(CCNC(C(N2C(=O)CCC2=O)CC)=O)C)cc(S(N)(=O)=O)cn1 39311,N1(C(Cc2ccc(C)cc2Br)=O)CC2COCCC2(NC(c2cn[nH]c2)=O)C1 39312,C(C)(CO)(C(=O)NC1CCN(C(c2ccccc2C(F)F)=O)CC1)NC(C)=O 39313,C(=O)(C(F)C(C)CNC(C1CC(=C2CCC2)C1)=O)NC(C(=O)NCC)(C)C 39314,C1(NC(C2(S(N)(=O)=O)CC2)=O)CN(C(C2CC3(CC3)CO2)=O)CCC1CO 39315,c1(OC)ncc(C(N2CC(C)(NC(C3CCC(OC)C3)=O)C2)=O)c(C(F)F)n1 39316,CC1(C)OCC2(CCN(C(c3coc(Cl)n3)C(=O)NC3COC3)C2)CO1 39317,C(=O)(CC1=CCCC1)NCC(=C)CCNC(=O)C(F)(F)c1ccccn1 39318,CC(C)S(=O)(=O)c1ccc(C(N2CC(C(C)NC(=O)C3=CC(C)(C)C3)C2)=O)cc1 39319,CC(C)CC(CC(=O)NC1CCC(=O)NC1=O)NC(c1cncnc1)=O 39320,N1(C(c2ccc(-n3cc(CC(C)(C)C)nn3)cc2)=O)CCC2NC(=O)OC2C1 39321,CCCC(CCC)CC(=O)N1CCCC1CNC(C1(CC)CC(C)(C)C1)=O 39322,c1(C(C)=O)ccc(C(=O)NC2CCC(CCC(=O)NCc3cnccn3)C2)o1 39323,C1(NC(Cc2cc(C)[nH]n2)=O)COCCN(C(=O)Cc2ccccc2F)C1 39324,C1(NC(C(CC)OCC)=O)CN(C(c2cn(C(C)(C)C)nc2C)=O)CC12CC2 39325,C1(C(=O)Nc2cccc(CC(=O)OC)c2)Nc2cc(C)ccc2S(=O)(=O)N1 39326,c1(C(=O)NC(C(C)C)CCN(C(=O)CCOCC2CC2)C)cccc(N)c1O 39327,CC1CN(C(C2(CF)CC2)=O)CC1CNC(=O)CNC=O 39328,N1(C(CC2CC(C)C2)=O)CC(CNC(c2ccc([N+](=O)[O-])s2)=O)C(C)(C)C1 39329,C1(=CC(=O)N(CCNC(Cc2cn(CC)nc2)=O)C2CC2)CCCCCC1(F)F 39330,C1(CNC(C2(CC=C)CC2)=O)CCC(C)CN1C(c1cc(SC)ccc1Cl)=O 39331,c1(CC)ccc(F)cc1C(N1CCC(NC(=O)CSC(F)F)C(CC)C1)=O 39332,n1(CCC)nc(C)cc1C(=O)NCC1CC1CC1CC1.C12CC1CC2=O 39333,N1(C(=O)CC(F)F)CCC2(CCCN(C(C3CC(c4ccc(Cl)cc4)C3)=O)C2)C1 39334,C1(NC(=O)OC(C)(C)C)C=CC(CCNC(=O)C(=O)NCCN2CCOC2=O)C1 39335,C1(C(N(CCC(F)(F)F)C)=O)CCC(C)(C)N(C(c2csc(=N)[nH]2)=O)C1 39336,c1(C(N(CCC(C)NC(=O)CC(C)c2cccnc2)C)=O)ncncc1Cl 39337,CCCCS(=O)(=O)NCC(N1CCC(CCNC(C2CCCCC2C)=O)CC1)=O 39338,c1(OCC=C)ccc(Cl)nc1C(N1CCC(C(C)CNC(=O)CCOC)CC1)=O 39339,N1(CCNC(C2(C)COC2)=O)CCN(C(=O)CCC(F)F)CC1 39340,N1(C(C2(CC=C)CCC2)=O)CCC2(C1)CN(C(=O)C(C)NC(=O)OC)CCO2 39341,C1(CCC)CN(C(c2cccnc2)=O)CC1C(=O)NOCC1CCC1 39342,C1(CC(N)=O)CC(N=c2[nH]c(=NCCC3(C(F)(F)F)CCC3)[nH]c3ccsc23)C1 39343,N1(C(c2ccc(SC)o2)=O)CC=C(CCNC(=O)C(C)COC2CCOC2)CC1 39344,C(=O)(C(CC)CC=C)NC1(CC=C)CN(C(C2(Cc3cnn[nH]3)CCC2)=O)C1 39345,n1(CC)ccc(C(N2CCC(CNC(=O)CCc3cncs3)C23CC3)=O)cc1=O 39346,CCCCC(C(=O)N=c1ccn(Cc2ccc(C(F)(F)F)cc2)[nH]1)C(C)C 39347,C1(C#N)(C(=O)NCC(CNC(c2ccc(N(C)C)cc2)=O)F)CCS(=O)(=O)CC1 39348,CCC(C)CC(C(=O)N(CC(N)=O)C)NC(=O)CCCCSC 39349,C1(NC(CC2CCN(C(C(CC)(C)O)=O)CC2)=O)CC12CCCCCC2 39350,C1(CC(=O)NCC(C)(C)OCCNC(CC(=O)NCC)=O)CCCCC1C 39351,C=CCC(CC=C)C(=O)NC1(CO)CCCN(C(=O)C(CO)C(C)(C)C)C1 39352,c1(C(=O)NCC2(CNC(c3c(C)scn3)=O)CC2)cnn(C2CCOCC2)c1C 39353,C1(C(=O)NCCCCC#C)(OC)CCN(C(c2cc(C)cc(F)c2)=O)CC1 39354,C(CC(O)C(=O)NC1CCOCC1F)NC(C(C)N(C)C)=O 39355,N1(C(c2c(CC)nc(C)[nH]2)=O)CC2(CCN(C(=O)CCCCF)C2)C1 39356,C(=O)(CCCCC(C)C)N(C(CCNC(C=Cc1n(CC)ncc1)=O)C)C 39357,C1(C(=O)NCC(C)(C)NC(=O)CCc2ccc(C#N)cc2)CCS(=O)(=O)C1(C)C 39358,C1(CNC(CCN(C)CC)=O)COC(C(F)(F)F)CN1C(=O)Cc1scnc1C 39359,c1(C(N2CCCC(CN(C)C)C2)=O)ccc(N=[N+]=[N-])cc1 39360,c1(OC)ccnc2c1CCCC2NC(=O)NCC(C)COC(C)C 39361,N1(C(CC(CC)NC(c2c(C#C)cnn2C)=O)=O)CCC2(C=CCO2)C1 39362,N1(C(CCC)=O)CCCCC1C(=O)NCC(O)CNC(c1oc(C)nc1CC)=O 39363,c1(OC)cc(CN2CCCC(C(=O)NC3CCOC3)C2)ccc1O 39364,O=C(C#CC1CCCOC1)NCC1CN(C(=O)Cc2ccc(Cl)cn2)C1 39365,C1(OC)CCCN(C(=O)NC2(c3cccnc3)CC2)C1 39366,c1(OC)cccc2cc(C(C)N(C(=O)NS(=O)(=O)CC(C)C)C(C)C)oc12 39367,CC1CCCCC1(C)NC(=O)C(c1cnn(C)c1)NC(=O)CC(=O)NC1CC1 39368,C(=O)(C(CCCO)c1ccccc1)N(CC=C)CCN(C(=O)COC)CC 39369,C1(NC(C=C(C)Cl)=O)CCCC1CNC(=O)CCCNC(=O)C1CC1 39370,C1(CN(CCCC)C)CCN(C(=O)Nc2ncc(CCC)cn2)CC1 39371,c1(C(=O)NC2CCCC(NC(C(CCSC)O)=O)C2)nccc2nn[nH]c12 39372,CCC(CC(=O)N1CC2CCN(C(c3cnccn3)=O)C(C2)C1)C(C)(C)C 39373,C(c1ccc(C)c(Cl)c1)=CC(=O)NC1C(NC(C(n2ccc(C)n2)C)=O)C1 39374,c1(COCCC)cn(C2CC3(C(=O)N(C(C)C(=O)OC)C4CC4)CC23)nn1 39375,c1(C(c2nnnn2C2CC(F)(F)C2)NC2CC(CC)C2)cncn1C1CC1 39376,C(C(COC)C(=O)N1CCCC1(C(N1CC(N(C)C)C1)=O)C(C)C)OC 39377,N1(C(c2ccc(OC)nc2)C(=O)NCCCC2CC2)CCC(O)CC1C 39378,c1(C(N2C(COC)(CNC(C3CC(C)CO3)=O)CCC2)=O)ccc([N+](=O)[O-])n1C 39379,C(C(C)(O)C(=O)N(CC(C)N(C(=O)CCn1cncn1)C)C)OC 39380,CC(O)C(C)C(=O)N1CCN(C2CCN(C(C34CC3C4)=O)C2)CC1 39381,c1(OCC=C)ccccc1C(=O)NCCC(C)CCNC(c1cc(Cl)n(C)n1)=O 39382,N1(C(C=COCC)=O)CC(CNC(=O)CC2CC(C)OC2C)OC(C)(C)C1 39383,N1(C(c2cc(C)c(C)o2)=O)CCC(C2CC2NC(C23CCCC2C3)=O)CC1 39384,c1(C(C)=O)ccc(CNC(=O)C(N)Cc2ccc(F)cc2)cc1C 39385,N1(C(=O)CN2CCN(C(c3cc(Cl)cs3)=O)CC2)CCC(C2CCOC2)C1 39386,N1(C(CSCCCC)=O)CC(NC(=O)C(CSC)c2ccccc2)CC12CCC2 39387,c1(C(N2CCSCC2C2CCC2)C(=O)NCCCF)cc2c(Cl)nccc2s1 39388,C1(CCCNC(CCOC)=O)CCCCN1C(=O)C(N1CCC(C)CC1)=O 39389,C1(C(N2CC(C3(NC(CC(C)F)=O)CC3)C2)=O)CN(CP(C)(C)=O)C1 39390,C1(CNC(C2(C(N)=O)CCC2)=O)CCN(C(c2cnn[nH]2)=O)C12CCC2 39391,N1(C(CCSC)=O)CCCC1C1CCCCN1C(=O)CN(C)CCO 39392,c1(N2CC3CC(NC(c4ccc(C(C)C)s4)=O)C3C2)c(Cl)cccc1[N+](=O)[O-] 39393,c1(CC)cc(OC)cc(OC)c1C(=O)NCC(C)(CC)NC(=O)C(F)C1CCC1 39394,CC(C)CCCCCC(=O)N(C)CC1(O)CCN(C(=O)C(O)C(C)(C)C)CC1 39395,C1(C(=O)NCC2(O)CN(Cc3onc(C(C)C)n3)C2)CCC=CCC1 39396,c1(C(N2CCC(NC(C(C)OCC=C)=O)CC2)=O)cc2n(n1)CCCC2 39397,c1(C(CC(=O)OC)NC(=O)CNC(N)=O)cccc(-c2cccnc2)c1 39398,CCC(C)CCC(=O)NCC(c1ccc(F)cc1)NC(=O)C=Cc1cc[nH]c1 39399,C1(NC(COCC#C)=O)CCOC(CNC(=O)CC2COCC2(C)C)C1 39400,C1(Cl)(C(=O)OC)CC1C(=O)NCCC(C)NC(C1(N(C)C)CC1)=O 39401,C1(CCC)CN(C(=O)C(C)CSC)CC1NC(c1ccc(C)nn1)=O 39402,N#CC1CCCC1NC(C1CCCCN1c1ncccn1)=O 39403,C1(NC(c2c(C)cnnc2)=O)CCCCC12CCN(C(c1ncc(F)cn1)=O)C2 39404,C(=O)(C(C)(C)CN(C)C)N1C(CN(C(CCNS(CC)(=O)=O)=O)C)CCC1 39405,C(C(C)(C)C(c1nnnn1C(C)C(=O)OC)NCc1sccc1C)OCC 39406,c1(CCC(=O)NC2C(NC(CCCNC(C)=O)=O)CCC2)cccc(F)c1F 39407,c1(CCC(=O)NCC(CNC(=O)C(C)C#N)OC)ccc(C(C)C)cc1 39408,CC(C(=O)N1CC(NC(=O)C(n2cc([N+](=O)[O-])cn2)(C)C)C1)C(C)(C)C 39409,Cc1ccc(F)cc1N(C(=O)C(C)NC(c1cc(Cl)cs1)=O)C 39410,Cc1cc(F)cnc1C(N1CC(NC(c2cccc(Cl)c2O)=O)CC(O)C1)=O 39411,c1(CCC(=O)N(CCCNC(C2N(C)CCOC2)=O)C2CC2)ccc(Cl)c(Cl)c1 39412,c1(C(=O)NCC2CN(C(C3C(C)(CC)C3)=O)C2)cnn(C(F)(F)F)c1 39413,c1(C(N(C(C)C)CCN(C(=O)COc2ccccc2Cl)C)=O)n[nH]c2c1CCC2 39414,O=C(CCC1CCN(C(c2ccn(-c3ccccc3)n2)=O)C1)NOCCO 39415,N1(C(CCOC)=O)CCC(NC(CNCC(=O)N(C)C)=O)C1 39416,CCC(CCC(=O)Nc1ccc(Cl)cc1)NC(C1CC(OC(C)C)C1)=O 39417,N(C(=NCCC(=O)N(C)C)NCC1CCN1C(C)(C)C)CC(CC)(C)C 39418,c1(C(OC)CC2CCCC2NC(c2sccc2-c2cccs2)=O)cn(CC)nn1 39419,CCC(C)(C(=O)NC(C1CCN(C(=O)C(C)(C)c2ccccn2)CC1)C)OC 39420,C1(C(=O)NC(C#CCC)(C)C)CCN(C(=O)Cn2ccnc2)O1 39421,C1(OC)CC(NC(c2cc(C)oc2C(C)C)=O)CN(C(C2(C#N)CC2(C)C)=O)C1 39422,c1(OC)ccc(Cl)cc1C(N1CCC(CCNC(C2(C)CCN(C)CC2)=O)C1)=O 39423,C(=O)(C(C)CCCC(C)=O)N1C(C(=O)NC(C(CC)CC)C)CCC1C1CC1 39424,N1(c2nc(=N)nc(N3CCC(C)(C(=O)NC)C3)[nH]2)CCc2nc(O)[nH]c2C1 39425,c1(SC)ncc(C(N2CCSC(C(=O)Nc3ccc(Br)nc3)C2)=O)c(Cl)n1 39426,Cc1nc(N(CC(C)NC(c2c([N+](=O)[O-])cnn2C)=O)C)c(C)c(Cl)n1 39427,Cc1noc(C2CC2)c1C(=O)NC(CNC(c1ccnc(C2CC2)c1)=O)C(C)C 39428,CC(C(C)NC(=O)CSc1nc[nH]n1)NC(c1csnn1)=O 39429,c1(OCCSCCN(CC)Cc2ccccn2)ccc(Cl)c(C)c1 39430,C1(C)(C(N2CCC(OC)CC2)=O)CCCN(c2cnc(C(N)=O)cn2)C1 39431,c1(NC2C3CN(C(C(CSC)(C)C)=O)CC32)ncnc2sc(C(C)C)cc12 39432,N#CC1CCCC(C(N2CCN(CC(=O)NCc3cnccn3)CC2)=O)C1 39433,C1(CCC)CCCN1C(C1CC1C(C)C)=O 39434,C1(=O)C(CC(C)(C)C)OCOCCC1OCC(=O)NCC(C(=O)OC)N(C)C 39435,C1(C(C)NC(CCCOCC=C)=O)CCCCN1C(=O)CCc1nccn1C 39436,c1(C(=O)NC(C(C)NC(COC(CC)CC)=O)C)cc(C)c(F)cn1 39437,c1(N(CC#C)C(=O)Nc2cccc(N3CCCC3=O)c2)cccnc1OC 39438,c1(N(c2ccc(-c3cccs3)o2)C(=O)CC2CCNC2)ccc2ncnn2c1.O=S 39439,C(=O)(CCCC)NC(C1CCN(C(=O)C(F)(F)c2ccccc2)C1)(C)C 39440,Cn1cc(C(N2CCCC2Cc2ccncc2)=O)c(C(F)F)n1 39441,c1(SC)cc(=NC(=O)C2CC(C)(C)CCN2C(=O)C(c2cnn(C)c2)C)[nH]n1C 39442,C(=O)(C(CC)CC(F)F)N1CC(NC(C(C(=C)C)(C)C)=O)CC1(C)C 39443,CN=c1[nH]cc(C(=O)NC2(COC)CN(C(C3CCCN3C)=O)C2)s1 39444,N1(C(C(CCOCC)NC(CCC#CC)=O)=O)CC(CC)CC(C)C1 39445,CCCCC(C(=O)NC1CCC1C(N1CCCC(C)C1CO)=O)NC(N)=O 39446,C1(C(=O)NCCc2n(C)c(=O)on2)C2CC3C(C2NC(=O)CC2CCC(=O)C2)C13 39447,C1(CC(=O)N(C(CC)C(=O)NCCC2C=CCC2)C)NC(=O)NC1=O 39448,c1(C(=O)NC(C2CCCN(C(=O)COC(F)(F)F)C2)C)ccnc2ccccc12 39449,C1(NC(C2(C)CC(=C)C2)=O)CCN(C(=O)Cc2nc(Br)sc2C)CC1C 39450,CC1(C)CCCC1NC(=O)C(N1CCCC(Cc2nc(C(F)(F)F)cs2)C1)=O 39451,c1(C(N2C3(CNC(CS(=O)(=O)NC)=O)CC(C2)C3)=O)c[nH]c2cc(N)ccc12 39452,N1(C(c2cc(COC)no2)=O)CC(F)CC1CC(N1CCC(O)(C(F)F)C1)=O 39453,N1(CC)CC2CN(C(=O)N=c3[nH]nc(N(C)C)s3)CC2C1 39454,N1(C(c2c(C)c[nH]n2)=O)CCCC2CN(CC(c3ccc(C#N)cc3)O)CC12 39455,Cc1cc2ccccc2cc1C(=O)NCC(O)CNC(c1cc(Cl)ccc1N)=O 39456,Cc1nc(CNC(c2nnsc2N)=O)oc1C(=O)N(C)CCOCCCO 39457,C=CC(C)(O)C(=O)N(CC(C)C(=O)NCCn1cccnc1=O)C 39458,c1(C(=O)NC(C(C)=O)C2CC2)n[nH]c2cc([N+](=O)[O-])ccc12 39459,Cc1cccc2c1CCN(CC(C1C3CCC1CN(C)C3)=O)C2 39460,Cc1ccc(-c2cn(-c3ccc(C(=O)N(C)C(c4nccs4)C)cc3)nn2)cn1 39461,S(=O)(=O)(c1ncc(F)cn1)Nc1c(CCCN)cc(F)cc1 39462,c1(CC)noc(C)c1CN=C(NC(C1CC1)C1CC1)NC1CC1(C)C(F)F 39463,C(C)(C)(C(C)NC(=O)CCCc1cc(C)no1)NC(CSCCC)=O 39464,C1(C(=O)NC(c2nc(SC)c(F)cn2)(C)C)CCC12CC(F)(F)C2 39465,c1(OC)c(C(N2CCC(O)(CNC(=O)C(C)OC)C2)=O)csc1C 39466,N1(C(C2CC(C#N)C2)=O)CCC(O)(CNC(C2CC(=O)N(CC(F)(F)F)C2)=O)C1 39467,c1(NC(C2(C)CN(c3ncncc3Br)C2)=O)cc(C#N)cn1C(C)(C)C 39468,Cc1ccc2nc(N3CC4CC3(CNC(=O)CC3C=CS(=O)(=O)C3)C4)sc2n1 39469,N1(C(C2C(O)CCN(C(CC3CCN(CC)CC3)=O)C2)=O)CCCC2CNCC12 39470,Cc1cc(C(F)(F)F)c2cc(C(=O)NC(C)CCN(C)C)oc2n1 39471,CCC(CC)C(O)CNC(=O)CC1CN(C(=O)CCc2ccco2)CC1C 39472,N1(C(C=CSC)=O)CC(N(C)C(c2cccc(-c3ccco3)c2)=O)C(C)(C)C1 39473,N1(C(c2cnc(C(C)O)s2)=O)CCC(C2CCCN(C(C3CCSC3)=O)C2)C1 39474,CON(C)C1CN(C(=O)CC2CN(C(=O)C(C)(C)C3CC3)CCC2C)C1 39475,c1(N(CCCCO)C)nc(=NCc2cc(F)ccc2Cl)[nH]c2c1COCC2 39476,Cn1nnc(Cn2nnnc2C(Cc2ccco2)NCCCOCC(F)(F)F)n1 39477,C1(C(N2CC(C)(C(N)=O)C2)=O)CCCN(C(=O)CC2CC3CCC2O3)C1 39478,C1(SC)CCC(N=c2nc(N(C)CC3CCCC3O)c3c([nH]2)CCCC3)CC1 39479,C(=O)(C(F)(F)C(O)C1CC1)N1CCC(N(C(C(C(C)C)NC(N)=O)=O)C)CC1 39480,c1(C(OC)OC)ccc(C(N2CCC(NC(=O)Cc3nccn3C)C2)=O)o1 39481,c1(OCC)cc(C(=O)NCC(C(C)C)NC(c2cocc2C)=O)ccc1OC 39482,N1(C(=O)OC(C)(C)C)CCN(C(c2cccc3oncc23)=O)CCCC1C(=O)O 39483,CC1CC(=O)CCC1C(=O)NCC=CC(=O)N(CCN1CCCCC1)C1CC1 39484,N(C)(S(N)(=O)=O)CC(=O)N(C1CC(NC(=O)CNC(c2ccco2)=O)C1)C 39485,C(=O)(C(O)CC(F)(F)F)NCc1c(C2CN(C(C(CC)OC)=O)C2)ocn1 39486,CC(CS(C)(=O)=O)C(=O)N1CC(O)(CN(C(=O)CCC(C)(F)F)C)C1 39487,C1(NC(COCC(=C)C)=O)(CO)CCN(C(c2ccc(CO)s2)=O)C1 39488,CC1(C(=O)NC2CCC(F)(CNC(=O)CCN3CCC3)C2)Cc2ccccc2N1 39489,c1(CCCCC)ccc(C(N2CC(O)(CN(C(=O)CC3CSC3)C)C2)=O)o1 39490,N1(C(CS(CCOC)(=O)=O)=O)CCOC2(C1)CN(C(c1ccc(N)c(F)c1)=O)C2 39491,c1(C(N2CCC3(C(C(=O)Nc4cnoc4)C3)CC2)=O)cc(F)c(Br)cc1[N+](=O)[O-] 39492,c1(C(N2CCC(NC(C(CC#C)(C)C)=O)C2)=O)cc2c(C)[nH]nc2s1 39493,c1(C(N2CC(CNC(CCSC)=O)C2)=O)ccncc1Cl 39494,C(=O)(C(O)CC(F)(F)F)NCCC1CCC(NC(C2CC3(CC(OC)C3)C2)=O)C1 39495,CCCC(C)(C)C(=O)NCC1CCC(C(N2CCC(CCN(C)C)C2)=O)CC1 39496,C1(C)(C(=O)NC)CCN(C(=O)C(=O)Nc2cnn(-c3nccs3)c2)CC1 39497,c1(CC)nc(=N)[nH]cc1C(=O)NC(C1CCCCN1C(=O)C=C1CCN(C)C1)C 39498,C1(NC(C2(CNC(=O)CC3CSC3)CCC2)=O)CC2CC2C1 39499,C12(C(N3C(C)CC(NC(C4CCCC(C)(C)C4)=O)C3)=O)CC=CCN1CCC2 39500,C1(C(=O)NC2CCN(C(c3nccc(SC)n3)=O)CC2F)Cc2ccccc2C1 39501,C1(NC(COCC)=O)CCCCC12CCN(C(c1cc(O)c(O)c(O)c1)=O)C2 39502,Cc1ccn2nc(C(N3CC4CCC3C(NC(c3nscc3N)=O)C4)=O)nc2n1 39503,c1(CC)cc(C(=O)NC2(CO)CN(C(C3CCCC3O)=O)C2)sc1C 39504,C(=O)(CC(C)CNC(C1CC(O)CN1C(=O)CP(C)(C)=O)=O)OC 39505,c1(CNC(=O)NC(c2ccc(OC)c(F)c2)C)c(C)cc(Cl)nc1Cl 39506,c1(OC)c(F)cc(C(=O)NCCC2CCN(C(=O)CC(C)SC)CC2)cc1Cl 39507,N1(C(CCCOC)=O)CCC2CCCC12CNC(c1cc(Cl)ccc1F)=O 39508,C(=O)(N=c1nc[nH]n2cccc12)C1C2(CN(C(c3ccc(C#N)cc3Cl)=O)C2)C1 39509,C(=O)(C(F)C(C)(C)O)NC1CC(C(C)NC(c2cncc(CC)c2)=O)C1 39510,C(=O)(C1CCCc2n[nH]cc21)N1C2C(NC(=O)CCn3cnnn3)(CCC2)CC1 39511,C1(C(N2CCC(C)(CNC(C3COCCO3)=O)C2)=O)(CC)CCC(O)CC1 39512,C1(CC(=O)NC2(C)CN(C(C(C)n3ccnc3)=O)C2)CCCC(C)(C)CC1 39513,c1(C(N(CC2N(C(C(CC#C)C3CC3)=O)CCC2)CC)=O)c(O)nnc2c1CCC2 39514,C(=O)(NNc1cc(C(C)C)ccc1F)c1onc(OC)c1I 39515,N1(C(C=C(CC)C)=O)CCC(N2CCN(C(C3CCOC(=O)N3)=O)CC2)CC1 39516,N1(C(CC(C)(C)C#N)=O)CC2CCCC1C2CNCC12CCCC(C1)OC2 39517,CC1(C)OC(=O)c2cc(C(=O)NC3CCC(c4ccc(F)cc4)C3)ccc21 39518,C(C)(C(CC(=O)N(C1CCC1C)C)NC(=O)COC1CC1)OC 39519,Cc1ncc(Cl)cc1C(=O)NCC1(C(F)F)CCN(C(=O)C(C)N2CCC2)C1 39520,N1(C(C2CC23CCC3)C(=O)NCCCOC)CC(C)OCC(C)(C)C1 39521,C1(C2CCC2)(C(=O)NCC2CN(C(C3(Cl)CC3)=O)CC2O)CC1(F)F 39522,C1(NC(C2N(CC)CCC2)=O)CCCC12CCN(C(=O)COC(C)(C)CC)CC2 39523,N1(C(N(CC(O)CN2CCCC2=O)C)=O)CCCCCC(S(C)(=O)=O)C1 39524,N1(C(C2C(C)CC=CC2)=O)CCC2C1CCCN2C(c1ncc[nH]c1=O)=O 39525,c1(C(=O)NC(C(C)NC(c2cc(CC(C)C)on2)=O)C)cc2c(nn1)CCOC2 39526,c1(C2(CN(CC(=O)OC)CC)CCC2)cc(C(F)(F)F)ncn1 39527,C1(NCCNC(CCN(C(=O)CSS(C)(=O)=O)C)=O)CC2(C1)CC21CC1 39528,C1(NC(CCSC)=O)C2CN(C(=O)CCn3cccnc3=O)CC12 39529,C=CC(CCC)CC(=O)N(C)CC1CCCC(NC(c2sc(CO)nc2C)=O)C1 39530,C(=O)(CC(F)(F)CC(=O)NCC1CCN(C(C2(C)CCCO2)=O)C1)OC 39531,C1(C(=O)NCC(C)N(C(=O)C(C2CCOC2)OC)C)(CC)CCOCC1 39532,C1(CCCNC(C2C(Cl)(Cl)C23CC3)=O)CCCCN1C(=O)Cn1nccn1 39533,N1(C(C2C(C=C)CC2)=O)CCN(C(c2cnn(C(C)(C)C)c2)=O)C(CO)C1 39534,N1(C(CCN(C(C(CC(C)(C)C)OC)=O)C2CC2)=O)CCN2CC(F)CC2C1 39535,Cc1cc(C(F)(F)C(=O)NC2CC(CNC(c3cc[nH]c3C3CC3)=O)C2)cs1 39536,c1(C(C(=O)NCC(C)(CO)NC(=O)CNC=O)O)ccc(F)cc1Br 39537,CCC(CC)C(C(=O)N1CC(OC)C(NC(=O)C(O)C2CCC2)C1)OC 39538,CCC(O)C(F)(F)C(=O)N(C)CC1CCCCN1C(=O)CN(C)C(N)=O 39539,C1(CNC(C=CCOC)=O)(NC(=O)C=Cc2cncn2C)CCCCCC1 39540,n1(C(C)(C)C)ccc(C(=O)NCCC2CCC(NC(=O)C=CCO)C2)n1 39541,Cc1nc(O)nc(C)c1C(N1CC2(C1)CN(C(c1cccc(S(C)=O)c1)=O)C2)=O 39542,C1(SC)CN(C(=O)CCn2cc(Cl)cn2)CC1NC(C1CCN(C)C1)=O 39543,C(C)(N=c1[nH]c(=NCc2ccc(N)cc2F)[nH]c2c1COC2)c1ccc(C)cn1 39544,c1(NC(C2CCCC(NC(C(C=C)(F)F)=O)C2)=O)cccc(F)c1C 39545,CC1CCOC(C(=O)O)CN1S(=O)(=O)CC(=O)NC(N)=O 39546,c1(C(=O)NC(CN(C(c2c[nH]c3nccc-3c2)=O)CC)C)sc2cncn2c1C 39547,c1(C(=O)NCC2(NC(CCCOC)=O)CCCCC2C)cnc2c(c1)COCC2 39548,N1(C(C2(n3cc(-c4c(OCC)nn(C)c4)nn3)CC2)=O)CCC(CO)C(O)CC1 39549,c1(CC(N2CCC(C(CNC(C3CC(SC)C3)=O)C)CC2)=O)c(F)cncc1Cl 39550,N1(C(c2cc(OCC)n[nH]2)=O)CCC2CN(C(=O)C(C)(C)C)CCC2C1 39551,c1(NC(CNC(C2(CC#C)CC=CCC2)=O)C2CC2)ncn(C)c(=O)c1Br 39552,c1(OC(C(N2C(CNC(c3cc(OCC)no3)=O)CC2)=O)C)ccc(Cl)cc1 39553,C1(C(=O)NCC(COCC)C)CCN(C(=O)CCc2cccs2)CCO1 39554,C1(CNC(c2n(C)cnc2)=O)CCCN(C(=O)Cc2ccn(CCF)n2)CC1 39555,C(CCCCC(=O)NCc1nc(C(=O)NCC2COC(C)(C)C2)co1)=CC 39556,C(=O)(CCCC(=O)N(C)C)NCC1(C(=O)NCC(C(=O)OC)(C)O)CC1 39557,C1(C(=O)NCC2(C)CCCN(C(CC3(C)OCCO3)=O)C2)OCCOC12CCC2 39558,c1(N(CC)CC)ccc(C(N2CCN(C(=O)NC3CC(=O)C3(C)C)CC2)=O)cc1 39559,Cc1cc(C)n2ncc(C(N3CC(n4cc(C(C)(C)CO)nn4)C(C)C3)=O)c2n1 39560,c1(C(=O)NCC2CC(OC)CN2C(c2scc(C)c2C)=O)ccc(N)cc1F 39561,N(C1CC(C)(C)CCc2ccccc21)C(NNc1ccc(C)cc1Br)=O 39562,N1(C(C(CC)O)=O)CCN(C(=O)Cc2cncc(F)c2)C(CC(F)F)C1 39563,Cc1cc(C(=O)NCC2(C)CCN(C(=O)C(C)(C)O)CC2)ccc1I 39564,CCCC(C(=O)N1CCC(NC(c2cn(Cc3cccnc3)nn2)=O)C1)C(C)C 39565,c1(C(N2CCCC(N(C(CC3N(C)CCC3)=O)C)CC2)=O)ccn2ccccc12 39566,N1(C(CC(c2ccc(C)cc2)(C)C)=O)CC(NC(c2cc[nH]n2)=O)CC(C)(C)C1 39567,C(C(C)CC(=O)NCc1ccc(CNn2cccn2)o1)NC(=O)OC(C)(C)C.C 39568,c1(OCC(=O)NCCCN(C(C(CC=C)C)=O)C)ccc(F)cc1F 39569,Cn1c(I)cc2c(N3CC(F)(C(=O)Nc4cnnc(Cl)c4)C3)ncnc12 39570,N1(C(c2cccc(C(N)=O)n2)=O)CCCC12CCN(C(=O)CN1CC=CC1)CC2 39571,C1(OCC)CCN(C(c2ccc(Cl)s2)C(=O)Nc2cccc(Cl)c2C)CC1C 39572,C12(C(=O)NCCOCCCNC(c3c(C)nc(C4CC4)[nH]3)=O)COC(CCO1)C2 39573,c1(CC(=O)NC2(CO)CCN(C(C=Cc3cn(C)nc3)=O)C2)cc(F)cc(Cl)c1 39574,CC1CC(CCNC(c2cnn(C)n2)=O)CCN1C(=O)CCNC(=O)C=CCl 39575,N1(C(=O)OC(C)(C)C)CCC(C(=O)OC2(C(F)(F)F)CCCCC2)CC12CCCC2 39576,c1(OCCOC)cc(C(=O)N(C)CC2CN(C(c3cnn[nH]3)=O)C2)ccn1 39577,N1(C(C(CC)O)=O)CC(C2CN(C(c3ccc(C)c(O)n3)=O)C2)C1 39578,C(=O)(C(C)(O)CCc1ccccc1)N(CCC(C)NC(CCCOC)=O)C 39579,c1(COC)ccc(Br)cc1Cl.c12ocnc1C(C)(C)NC2=O 39580,C1(NC(CCC#C)=O)CC(CNC(=O)CCc2nc(-c3ccoc3)no2)C(O)C1 39581,N1(C(CCOCCOC)=O)CCC(F)(F)C(CNC(c2scnc2COC)=O)C1 39582,N1(C(CC2CCC(C)(C)O2)=O)CCCC(CC(=O)NC2COCC(C)(C)C2)CC1 39583,C1(C(N(C2CCC(NC(=O)OC(C)(C)C)CC2)C)=O)CCC2CC2CC1 39584,c1(OC)ccc(C(=O)NCCCC(C)(C)NC(c2onc(OC)c2Br)=O)cc1 39585,C1(C(=O)NC2CN(c3ncco3)C2)CCCCN(C(=O)C2CC2)C1 39586,N1(C(C2C(C)(Br)C2)=O)Cc2ccccc2CC1CNC(C1CC(F)(F)C1)=O 39587,N1(C(C(C2CCN(C(C3(C4CC4)CC3)=O)C2)C)=O)CCC2CN(C)CC2C1 39588,c1(N2CC3C(CNC(C(C=C=C)C)=O)C3C2)ncc(Cl)c(C(=O)NCCOC)n1 39589,Cc1nc2c(s1)CCCC2C(=O)NC1CCOCC1NC(=O)Cn1cncn1 39590,C1(NC(C2(C(C)(C)OC)CC2)=O)CC2CC1N(C(C1(C(F)F)CCCO1)=O)C2 39591,CC(C)(CCCCNC(C1CC=CC(O)C1)=O)NC(C1CC1(F)F)=O 39592,C(=O)(C(CCN(C)C)N(C)C)NCCOCCNC(C(C)N1CCC1)=O 39593,c1(OC)ccc(-c2cn(CC3CCN(C(C4CCCCS4)=O)CC3)nn2)cc1F 39594,CC1(C(=O)NCC2CC(O)CN2C(C2COCCN2C=O)=O)CCCNC1=O 39595,N1(C(C(=O)NCC)=O)CCC(C)C(NC(=O)CCc2ccc(OCC)c(Cl)c2)C1 39596,C1(C(=O)NCC2(OC)CCN(C(c3nnn(CC)c3C)=O)C2)CN2CCC1CC2 39597,C1(O)(C(COC(C)C(=O)NCC2CC2)(C)C)CN(C(c2csc(C(F)F)n2)=O)C1 39598,C(C1CN(C(=O)C2=CCCCC2)CC1C(=O)NCC(C)(C)CC)=CC 39599,N1(C(Cc2cccc(C)c2)=O)CCC2CCC12CNC(=O)C=Cc1cncs1 39600,C1(NC(c2c(CC)cno2)=O)COC2C(NC(=O)Cc3nn(C)cc3Cl)COC12 39601,CC1CCCc2ncc(C(N3CCCC(C)(NC(=O)C4=C(Cl)CCC4)C3)=O)n21 39602,CCCCCCC(C(=O)NCC1CN(C(c2scnc2Cl)=O)CC1O)NC(C)=O 39603,c1(C(=O)OCC)cc(=NCC(C2CC2)N(C)C(C2(C3CCC3)CC2)=O)[nH]c(C)n1 39604,C(=O)(C(CC1CC1)OC)NC1(CNC(CCNC(COC)=O)=O)CCC1 39605,N1(C(CCC=CC)=O)CCc2ccccc2C1CNC(=O)CCC1(C)CC1 39606,C(=O)(C(CNC(c1ncsc1NC)=O)CC(C)C)N(C12CC(C1)C2)CC 39607,C1(NC(c2c(CC)cns2)=O)C2CCC(C2)C1C(=O)NC1CC2CC3C(C2)C13 39608,c1(OC)cc(C)ccc1CNC(=O)NCCC(C(=O)NC(C)(C)C)OC 39609,CCC(C)(CCC(C)C)C(=O)N(CC(C)(C)NC(c1n[nH]c2c1CC1CC21)=O)C 39610,Cc1cn2c(n1)CC(C(=O)NCCC1CCCN1C(c1ccncc1Cl)=O)CC2 39611,c1(C(=O)NC(CN(C(=O)CC(C)F)CC)C)c(C)c(O)nc2ccccc12 39612,C1(C)(C(=O)OC)CN(C(C2CCC2)=O)C1.C12(CC1)C(=O)N2 39613,C(=O)(C(=O)CCC(C)C)NC1CC(C(=O)NC2C=C(C)CCC2)OCC1 39614,c1(C(N2CCC(O)(C(=O)Nc3c(OC)nccn3)C2)=O)cccc2c1CCC2 39615,N1(C(C(COC)C)=O)CCC2(CCCN2C(=O)CCN2CCCCC2)CC1 39616,c1(CC(N2CCC(O)(C(=O)NC(C)(C)C)CC2)=O)cccc([N+](=O)[O-])c1.CCO 39617,C1(C)(CNC(C=NOC)=O)CC(F)(F)CN1C(c1ccc(C)nn1)=O 39618,C#Cc1cccc(CC(=O)NC2COCCN(C(=O)COC(C)(C)CC)C2)c1 39619,Cc1nc(=NN2CCC(C#N)CC2)n(-c2ccccc2C(F)(F)F)[nH]1 39620,c1(OC)ccc2c(CC(=O)NCC34CC(CN3C(=O)CC3CC3)C4)coc2c1C 39621,c1(NC(C2CC2C(=O)NC2CCC(CO)CC2)=O)n[nH]cc1[N+](=O)[O-] 39622,c1(OC)nn(C)cc1C(=O)NC1CC(CNC(=O)CC2CCN2C(C)=O)C1 39623,c1(N(CC(=O)NCC2C(NC(c3c(C)scn3)=O)CC2)C)ccc(Cl)cc1 39624,C(=O)(C(C)(C)C(C)NC(=O)CC(=O)N(C)C)NC(CCC=C)CO 39625,c1(CC(N2CC(CNC(C=CSC)=O)CC(C)(C)C2)=O)nccc2ccccc12 39626,C1(N(C)C(C2CNC(=O)C2)=O)CCCN(C(c2ccnc(O)c2)=O)CC1 39627,C1(C(C)C)(C(N2CCCCC2)=O)CCN(C(=O)C=CC2CCCC2)C1 39628,Cc1cc(Cl)ncc1NC(C1C=CC(NC(=O)Cc2cccs2)C1)=O 39629,C#CC1COCCN1C(c1ccc(OC(C)C)cc1)C(=O)NC(C)C(=O)OC 39630,CCCCCCC(F)C(=O)NC1CC2CCC(C1)N2C(c1ccc(Cl)o1)=O 39631,NC(=O)CCCC(=O)NC1CCCCCC1NC(=O)CNC(=O)C(F)(F)F 39632,CN1CC2CC2(NC(=O)C(Cn2cncn2)NC(C2CCC=CCC2)=O)C1 39633,C1(C(=O)NC2C(NC(C(c3cccc(C)c3)F)=O)COCC2)CC2CCC1CC2 39634,C=Cn1nccc1C(=O)NC(Cn1cncn1)C(=O)NC1(CC)CCOC1 39635,c1(OC)ccc(C(O)C(N2CCC(NC(c3nc(C(C)(F)F)cs3)=O)C2)=O)cc1 39636,C1(C(=O)NC2C(CNC(c3coc(-c4ccccn4)n3)=O)COC2)CCCCO1 39637,C1(C(=O)NCC(C(C)C)NC(C2CCN(CC(F)(F)F)CC2)=O)C2CCN1CC2 39638,Cc1cccc(-n2nc(CCN(C)C)nc2-c2cnn3ccsc23)c1C 39639,C1(NC(C2(OC)CCCOC2)=O)CCCN(C(=O)C=Cc2ccn(C)c2)C1C 39640,c1(NCCOCCO)nccc(=NC(C)Cc2ccco2)[nH]1.N12CC(CC1=O)C2C 39641,C1(C(N(C2CC(C)C2)C)=O)(NC(C2CCCC(=O)C2)=O)CCCC1C 39642,CC1(C)CCCC(NC(=O)CSCCNC(=O)CC2CC=CCC2)C1 39643,C(=O)(C#CC1CCOCC1)N1CC(C)C(CNC(=O)CCCCC2CC2)C1 39644,c1(NCC(=O)NC2(COC)CN(C(=O)Cc3ccccc3O)C2)ccc(O)cc1 39645,N1(C(C23OCC(C)(C2)C3)=O)CCC(C2CC2)(CNC(=O)CCCC2CCC2)C1 39646,N1(C(C2(CC#C)CCCO2)=O)C2CCC(C2)C1C(=O)NC1C(O)CC1O 39647,c1(-c2nc(Cc3scc(CF)n3)on2)cc(F)cc(F)c1 39648,Cc1cncc(CC(=O)N(C(C)CN(C(=O)CC2CCCC(=O)C2)C)C)c1 39649,C1(CC(=O)N(CC(CNC(C(COCC)C)=O)C)C)CCCCC1(C)C 39650,c1(C(=O)OCC)ccc(NC(C2CCN2Cc2coc(C)n2)=O)cc1F 39651,C12(C(=O)NC(c3ccccc3)CNC(CN(C)C(N)=O)=O)CC(C)(C1)OC2(C)C 39652,N1(C(c2c(C(=O)OC)nccc2)=O)CC2CC1CCN2C(C1(F)CCCCC1)=O 39653,C1(NC(CCC2CCN(C(c3ccc(CC)nc3)=O)C2)=O)CNC(=O)C1(C)C 39654,C1(NC(C2(CC)CCOCC2)=O)CCN(C(=O)C=CCOCCOC)CC1OC 39655,C1(F)(CNC(c2scnc2Cl)=O)COCCN(C(C2OCCCO2)=O)C1 39656,CCCC(C)(O)CC(=O)N1CC(NC(c2cnc(C(C)C)s2)=O)C(CC2CC2)C1 39657,c1(OCC)ccc(C(=O)NCCCCCCN(C(=O)CN2CCC2C)C)cn1 39658,c1(CC(=O)NCC2CCCOC2)cn2cc(-c3ccncc3F)ccc2n1 39659,CC(O)C(F)(F)C(=O)NCCC(C)(C)CNC(=O)CCOCc1ccncc1 39660,N1(CCNC(c2cc(CNC(c3cocc3C(N)=O)=O)[nH]n2)=O)CCCOCC1 39661,C12(NC(c3c(CC)c[nH]c3)=O)CCN(C(C3(CC4CC4)CC3)=O)CC1C2 39662,C1(C(=O)NC(c2ccccc2)C(C)C)CCC1(F)F 39663,N1(C(Cc2cc(C(C)C)no2)=O)CCC(NC(=O)C(F)C(C)(C)O)C(CO)CC1 39664,C=CCC(F)(F)C(=O)NC1CC2CC1CC2C(=O)NCCc1nc[nH]n1 39665,C(=O)(C(F)CC(C)(C)NC(C1CC(=O)CC12CCC2)=O)NCC(=O)NCCC 39666,C(=O)(C(F)CC(C)(C)NC(C1(C)CCCCC1)=O)N(C)CCc1ccccn1 39667,c1(C(C)=O)c[nH]c(C)cc1=NC1CCc2ncc(C(F)(F)F)cc2C1 39668,c1(OC)ccc(CNC(=O)C(N)Cc2cc(Cl)ccc2Cl)c(F)c1F 39669,CCC(CC(=O)N1CCC(CF)(NC(c2c[nH]nc2C)=O)C1)C(C)(C)C 39670,O=C(CCCCC(F)F)NCCC1CSCCN1C(=O)C(O)CC1CCCCC1 39671,C1(NC(=O)Nc2c(SCC)cccc2)CCN(C(=O)CCc2ccc[nH]2)CC1F 39672,N1(C(c2cnc(N(C)C)o2)=O)CCC12CCN(Cc1cccc(C(=O)O)c1C)CC2 39673,c1(C(C)C)cc(Cl)nc(NC(=O)C(N2CCCC(Cn3cncn3)C2CO)=O)n1 39674,C(CNC(=O)CC1(C)CCOC1)(CCNC(c1[nH]cnc1C)=O)OC 39675,C1(NC(c2c(Cl)cc(C)s2)=O)CCC12CN(C(c1ccnc(OC(F)F)c1)=O)C2 39676,N1(C2CCN(Cc3cc(C(=O)OCC)n[nH]3)C2)CCN(C(=O)CC(C)CF)CC1 39677,C(c1cncc(O)c1)=CC(=O)NCC1N(C)CCN1C(=O)CCC(N)=O 39678,N#CC1CC2(CC(NC(=O)CCC3CCCN(C(c4sccc4CO)=O)C3)C2)C1 39679,c1(CC)cc[nH]c1C(=O)NCCOCC(c1ccccc1)N1CCOCC1.OC 39680,CCCC(O)(CCC)CC(=O)N1CCN(C(=O)C=CC2CCOC2)C2(CCC2)C1 39681,CC1CCN(C(=O)CSC2CC2)CC1CNC(c1cccc(F)c1OC(F)F)=O 39682,C1(NC(C(C)NC(=O)C2CC2)=O)C2CC3C(C2)C13C(=O)N(CCC[Si](C)(C)C)C1CC1 39683,C1(NC(c2cncc(OCC)c2)=O)CC2CN(C(=O)COC3CCCOC3)CC12 39684,N1(CC)CCC(NC(=O)C(c2ccoc2)NC(=O)C=CC(C)(C)C)C1 39685,CC(C(=O)NC(CNC(=O)C(=O)NCC(F)F)CO)c1ccco1 39686,N1(C(c2c(C)c[nH]n2)=O)CC2(C1)C(NC(=O)C1Cc3ccccc31)CCS2(=O)=O 39687,Cn1nc2c(c1C(N1CCN(C(C3(Cl)CC3(C)C)=O)CC1)=O)CCC2 39688,C1(N(C(=O)C(C)COCC)CC)CCCN(C(C2CC3CC2C3)=O)C1 39689,C1(N(C(C(=O)NC)C)Cc2ccccc2)CCCN(C(c2ncnn2CC)=O)C1 39690,c1(CSCC(=O)NCC(C)N(C)C)ccccc1.C12CCN1C(C)C(=O)N2 39691,c1(OC)cnnc(C(=O)NC(C)CCCNC(=O)C(C)OCC2CC2)c1 39692,C1(CNC(c2c(C(C)C)c[nH]n2)=O)C2CC1N(C(=O)Cn1ccc(C3CC3)n1)C2 39693,C(CCCCC(=O)N1CCC(C(=O)NCC2CC2(Cl)Cl)C1(C)C)OC 39694,Cc1ncc(C=CC(=O)NC2(CN(C)C(C3CC(C)(CO)C3)=O)CC2)s1 39695,c1(C(C(=O)NC2CC(CCNC(c3cnc(CC)s3)=O)C2)(F)F)ccccc1F 39696,C1(CNC(CCNC(N)=O)=O)CCCCC1NC(C12CC(CF)(CO1)C2)=O 39697,Cc1[nH]c2ccccc2c1C(N1CCCCC(CNC(c2cnns2)=O)C1)=O 39698,N1(C(c2cc(C)c(C)s2)C(=O)NC2CCOC2)CCC(C)(N2CCOCC2)CC1 39699,C1(CNC(C(=O)N(C)C)=O)COC(C)(C)CN1C(C1CC2CC1C2)=O 39700,N1(C(c2nnn(C)c2C(F)F)=O)CCC2CCN(C(c3cccc(Cl)c3)=O)CC12 39701,c1(C(=O)NCC2(CCCNC(C(C(C)C)O)=O)CCCC2)nc(O)nc(O)c1N 39702,N1(C(CC(C)C)=O)CCC2(CCCCN(C(C3CN4CCN3CC4C)=O)C2)C1 39703,N1(C(C2(CCC)CC2)=O)CC(C)(C)C(NC(=O)CC(C)(C)CN(C)C)C(C)(C)C1 39704,C12(CNC(C=CC(C)(C)C)=O)CN(C(=O)Cc3ccccn3)CC1(C(F)(F)F)C2 39705,C1(CCC)CN(C(=O)CC2CCSC2)CC1C(N1CCC(C(=O)OCC)C1)=O 39706,c1(OC)cnccc1C(=O)NCCC1CCCCN1C(c1ncn(C(C)C)n1)=O 39707,c1(C(=O)NCCNC(CCCC2CCC(C)C2(C)C)=O)c2ccccc2nn1C 39708,C#Cc1cc(F)c(C(N2CC3CC3(NC(C3COC3)=O)C2)=O)cc1F 39709,O=C1COc2cc(C(N3C4CCC3CN(C(C3CCC5CC35)=O)C4)=O)ncc2N1 39710,N1(C(CC(=O)OC)=O)CCC2(CCC2NC(C23COC(CF)(C2)C3)=O)CC1 39711,C1(C(=O)NCC23CC(NC(=O)CCOCC4CC4)(C2)C3)CCC(F)CC1 39712,c1(C(=O)NCC(CCC)C(=O)N(CCC(F)(F)F)C)ncn2ccccc12 39713,CC(C)CCCC(C)C(=O)N1CCC(CCNC(c2cc3occc3[nH]2)=O)C1 39714,C1(CNC(c2c(C)occ2C(F)(F)F)=O)CC(F)(F)CN1C(c1ccno1)=O 39715,c1(CC)nc(C(=O)NCc2ccnc(C(=O)NCc3[nH]c(C)nc3C)c2)c(C)o1 39716,c1(C(N2CC(N(C(=O)CSC(F)(F)F)C)C2)=O)occc1CN1CCOCC1 39717,C1(C)(CC)CCN(C(c2cccc(I)c2)C(=O)NCCCC2CC2)C1 39718,C1(NC(C2C(NC(Cc3c(C)cnn3C)=O)COC2)=O)Cc2cscc2C1 39719,C1(C(=O)NCCOC2CCCC2)CCN(C(C2CC(F)C2)=O)C1 39720,C(c1cc(C)ccc1OC)=CC(=O)N(CCCCNC(CC(COC)C)=O)C 39721,N1(C(C(C(C)C)SC)=O)CCCCC(NC(=O)COc2cc(C)on2)C1 39722,Cc1ccc(C(N2CCCC2CCC(=O)N(CC(C)C)C2CC2)=O)nc1 39723,c1(OC)ccccc1OC(F)(F)F.c1ccccc1C1CCCNC1 39724,c1(C(=O)OCC(N2CCCC(N3CCN(C)CC3)C2)=O)cc(F)cc2[nH]ncc12 39725,c1(C(N2CCN(CC(C)(C)O)CC2)C(=O)NCC)cnn(C)c1CC1CC1 39726,c1(C(=O)OC)cn(C)nc1C(=O)NCC1CCC(NC(=O)C(C)(C)SC)C1 39727,Brc1c(-c2nc(-c3cccs3)nn2C2CSC2)nc2n1CCS2 39728,N1(c2cc(C)nc(C3CCC3)n2)CCC(C)C(NC(=O)CC2CC=CCC2)C1C 39729,C1(O)(CNC(CCCC)=O)CCCN(C(=O)CC(O)C(C)C)C1 39730,c1(CC(=O)NC(CC)CNC(C2(NC(N)=O)CC2)=O)cncc(C)c1 39731,CCCCCS(=O)(=O)CC(=O)NCC1(OC)CN(C(=O)C(C2CC2)N(C)C)C1 39732,c1(CCC)c(NC(N2CCCC(CF)C2)=O)nnn1Cc1ccccc1Cl 39733,c1(C(=O)NC2(C)CCN(C(c3cn4ccsc4n3)=O)C2)ccc(Cl)nc1O 39734,c1(CCNC(C2N(C(CS(C)(=O)=O)=O)CCC(O)C2)=O)ccc(S(=O)(=O)F)cc1 39735,C(C1=CCN(C)CC1)NC(C1C(CC)CN(C(=O)CC2CC2CC)C1)=O 39736,N1(C(c2c(Cl)cn(CC)n2)=O)CCC(C)C(CNC(=O)C(C)(C)C(N)=O)C1 39737,N1(C(C)=O)CC(O)CC1C(=O)N(CC(F)F)Cc1ccccn1 39738,c1(C(N(C2CCCC(NC(=O)CCF)C2)C)=O)ccc(P(C)(C)=O)s1 39739,c1(NC)ccc2c(c1)OCCN2C(=O)NCCN1CCCCC1=O 39740,n1(C(C(=O)N(CCNC(=O)CN(CC(C)(C)C)C)CC)C)ccc(C)n1 39741,c1(OCC)ccccc1N(C(c1cccnc1OC)C(=O)NCCC1CC1)C 39742,C(=O)(C1=C(C#N)CCC1)NCC1CC(C)(C)CN1C(C1COCC1(C)C)=O 39743,C1(C(N2CCC(n3cc(C(N4CCCC4)C)nn3)C2)=O)CCc2nncn2CC1 39744,Cc1ccn(C)c1C(=O)NCC1CC(F)(CNC(C2(F)CC=CC2)=O)C1 39745,C1(C(=O)NC(C=C)C)CC12CC(NC(c1c[nH]nc1C1CC1)=O)C2 39746,CC(C)CC(C(=O)NC1CC2C1CCN2C(=O)CC1CN2CCC1CC2)C(N)=O 39747,c1(OC)cccc(NC(=O)NCC2(CNc3cc(Cl)ccn3)CC2)c1 39748,C1(CNC(CSc2n(C)ccn2)=O)CCCCN1C(c1cn(C2CC2)cn1)=O 39749,N1(C(C2NC(=O)OCC2)=O)C2CCC1(CNC(c1cnn(CCO)c1)=O)CC2 39750,c1(C(CCC)NCCc2ccncc2)nnnn1Cc1nnn(C)n1 39751,N1(C(c2cccc(Cl)c2)C(C2CCCCC2)OC)CCC2(CSC2)C1 39752,Cc1ccc(F)c(O)c1C(=O)NC1CCCCN(C(=O)CCc2cscn2)C1 39753,N1(C(C=CC)=O)CCC(C)(C)C(CNC(=O)C(C(C)CC)N(C)C)C1 39754,C1(NC(C(C)=CC2CC2)=O)CN(C(=O)Cc2c(C)noc2Cl)CC12CC2 39755,C1(CNC(C2(C)CCC2)=O)CCCN1C(=O)CC1CCOC1=O 39756,Cc1cc(C(C)NCC(C)CCCO)ccc1[N+](=O)[O-] 39757,c1(OCC(=O)NC(C(C)NC(=O)CC2CCCCC2)CO)cccc(F)c1 39758,C1(C(C(=O)NC(CC=C)CNC(c2nncs2)=O)C)CCCCCC1 39759,C1(CC(N2CC(CC=C)(NC(CCCC#C)=O)C2)=O)NC(=O)CN(C)C1=O 39760,C1(CN(C(C2(CCNC(CCN(CCC)C)=O)CC2)=O)C)CC2CCC1O2 39761,C(CCCCC(=O)N(C1CC(C#N)C1)CC(=O)NCC(C#N)CC)=CC 39762,C(=O)(C(C)(C)CCC#N)NCCC(C)N(C)C(C1OCCN(C)C1=O)=O 39763,C(C)(CCCCNC(=O)COCC1CCOC1)NC(C=C(C)CF)=O 39764,Cc1cc(C2CC2)ccc1C(=O)N(CC(O)CNC(=O)CCN(C)CCO)C 39765,c1(C(=O)NC2CN(C(C(CO)NC(N)=O)=O)C2)cc(Cl)c(Cl)cc1N 39766,C=CCCCCCC(=O)NC1CCOCC1C(=O)NC1CC(C)CCC1O 39767,Cc1ccc2ccccc2c1CNC(N1CCCN(Cc2ccccc2)CC1)=O 39768,N1(C(C2CCC2)=O)CCCC2C1CCN2C(c1sccc1F)=O 39769,N1(C(C(CC=C)NC(C)=O)=O)CCC(C(=O)NCc2nccs2)C1(C)C 39770,C1(F)(C(=O)NCCC2(CNC(C(C)C3CCOC3)=O)CC2)C(C)(C)C1(C)C 39771,CC1CCCC(OCC(=O)N(C)CC2CN(C(C3CCCC4CC34)=O)C2)C1 39772,c1(C(=O)NS(CCC(C)(C)C)(=O)=O)cc2cc(F)ccc2cn1 39773,C12(COC)CN(C(=O)C3=CCC3)C(CNC(c3ccc(C)s3)=O)(C1)C2 39774,CC1OC(C)C(C(=O)N(C)CC2CN(C(C3(CC(C)=O)CCCC3)=O)C2)C1C 39775,Cc1cc(N(C2CCN(C(=O)C(C3(O)CCOCC3)(F)F)C2)C)c(C#N)cn1 39776,C(=O)(C(F)CC(C)(C)C)N1C(CC(=O)NC(C(=O)OC)C2CCC2)CCC1 39777,c1(C(N2CCC(CN(C(CCc3c(C)noc3)=O)C)C2)=O)cc(Cl)nn1C 39778,C(=O)(C1=NN(C)C(=O)CC1)NCCC1N(C(Cn2nnc(C)n2)=O)CCOC1 39779,c1(OC)c(C(=O)NCC2(C)COC(C)(C)O2)ccc([N+](=O)[O-])c1F 39780,N1(C(c2c(OC)nsc2)=O)CCC(C=CC(=O)NCCC(O)C(F)(F)F)CC1 39781,Cc1cc(C(=O)NC(CNC(=O)CNC(c2ccsc2)=O)C(C)C)ns1 39782,c1(CN2CC3C(C(N4C(CC(=O)OC)CCC4)=O)(C3)C2)cncc(Cl)c1Cl 39783,O=C(NN1CCCC1C(=O)NCc1ncsn1)C1CC(CC2CC2)C1 39784,N1(C(C2CCC(CC)CC2)=O)CCCCC12CC(NC(=O)Cc1ccn(C)n1)C2 39785,c1(C(=O)OC)cc(C(N2CCN(C3CCOC3)CC2)C(=O)NCCCF)nn1C 39786,C#CC(CC1CCOC1)NC(=O)CCC 39787,c1(C(C)C)cc(C(F)(F)F)nc(NC2(CNC(=O)C(F)=CC3CC3)CC2)n1 39788,C1(C(=O)NCCCNC(C(C)c2ccon2)=O)CSc2ccccc2O1 39789,N1(C(c2ccc(CCC)[nH]2)=O)CC(NC(c2cc(O)nn2C)=O)C(C)C1 39790,C(=O)(C(F)(F)C(F)F)N1CC(C(C(=O)NCC(C)CN2CCCC2)O)C1 39791,C(=O)(C(F)CC(C)(C)NC(C1CCN1C)=O)NC(C)CC1CCC1 39792,CN1CCN(C(=O)CC2(O)CCCOC2)C(C(=O)NCC2=CCCCC2)C1 39793,C1(C(=O)NC(CC)C(N)=O)CCCCC1CNC(c1ccc(CC#N)cc1)=O 39794,C1CCC(=O)NCC2CC(CO2)CNC1=O.C1(C)(SC)CCCC1 39795,c1(CC)cc(-c2ncccc2C(=O)Nc2cccc(C)c2C)ccc1O 39796,c1(OC)cc(C=CC(=O)NC2CC(NC(=O)C(O)C3CCC3)C2)ccc1O 39797,C=C=CCCC(=O)NCC(=O)NC1CCCC1.c12noc-1n2 39798,c1(CC)[nH]nc(C(=O)NC2(C(=O)NCCCN(C)OC)CCCC2C)c1C 39799,N1(CC(=O)NCC2CCC3(CCC3)O2)CCC2(C=CCO2)CC1 39800,c1(CC(=O)OC(c2ccccc2)C)c(F)cccc1F 39801,c1(CCC(=O)NC(CCCNC(c2c(C)n[nH]c2C)=O)C)ccc(Cl)cc1Cl 39802,n1(CC(=O)NC2(C3CN(C(CNC(C)=O)=O)C3)CC2)ncc2ccccc12 39803,C1(C(=O)NC2CON(CC)C2=O)CN(C(C2C3CC(=O)CC23)=O)CC1(C)C 39804,N1(C(c2cc(C)n(CCO)n2)=O)CC(CNC(c2n[nH]cc2Cl)=O)OC(C)(C)C1 39805,NS(=O)(=O)C1(C(=O)NCC2CC3CCC2N3C(=O)C2=CCCO2)CCCC1 39806,c1(C(=O)O)cc2oc(=O)n(-c3ccccc3Br)c2cc1CCCN1CC=C(Br)CC1 39807,Cc1cccc(C(=O)NCC2CCCC2NC(c2c(F)cccc2F)=O)c1C 39808,c1(NC(C23CC(NC(c4cc(C(C)(C)C)[nH]c4)=O)(C2)C3)=O)cnc(Br)c(I)c1 39809,C(=O)(C(C)(C)CS(C)(=O)=O)NCC(CN(C(=O)CCCc1cncs1)C)C(F)(F)F 39810,n1(CCOCCNC(C(c2cccnc2)C)=O)cc(C2CC23CC3)nn1 39811,Cc1ccn2c(C(=O)N(CC(C)(C)CNC(=O)CC(=O)NC3CC3)C)cnc2c1 39812,c1(C(=O)NCC2(O)CN(C(c3cn(CCOC)nc3)=O)C2)cccc(Cl)c1Cl 39813,c1(NCc2ccc(OCC(=O)NCC)c(OC)c2)cc2c(s1)CCOC2 39814,C1(C(=O)NC(CC(=O)NC)C2CC2)C=CCCN1C(=O)CCCCOC 39815,C1(NC(C2(C#C)CCCC2)=O)CC2CC1N(C(=O)C(CC)=CC)C2 39816,C(CN=C(NCC(c1ccc(F)c(F)c1)O)NCC1CCCO1)c1ncc(C)s1 39817,C1(c2n(C)cnc2)CN(C(=O)CSC2CC2)CC1NC(=O)CSC(F)(F)F 39818,Cc1nc(O)ccc1C(=O)NCCc1cc(C(=O)N(C2CCC2C)C)no1 39819,Cc1cc(NC(=O)Nc2c[nH]nc2C2CC2)n2ncnc2n1 39820,N1(C(C2N(C(C)=O)CSC2)=O)CC2(CC(NC(=O)C=C(C)C(C)C)CO2)C1 39821,N#Cc1cc(F)ccc1C(=O)NC1CC(=O)N(C2CCCCC2)C1 39822,C1(C(=O)NC2(C)CC(NC(C3(N(C)C)CCCSC3)=O)C2)CCCCC(=O)C1 39823,c1(C(=O)NCC=CCNC(C2C(C)C2)=O)ccc(N2CCC(C)CC2)nc1 39824,c1(C(=O)NC)ccncc1C1CC1.C1(C(=O)NCCO)CN(C(c2cnns2)=O)C1 39825,Cc1cccc(C)c1CNC1(c2nnnn2C2CC2)CC(C(C)C)C1.C1(=O)CO1 39826,C(C1CCN(C(C2CCCC(C)(C)C2)=O)CC1)=CC(=O)N(C(CC)C1CC1)C 39827,N1(C(C(C2CCC2)OC)=O)CC(NC(c2cc(Cl)c(F)cc2F)=O)C(N=[N+]=[N-])C1 39828,N1(C(CCCOC)=O)CCCC(CO)(CNC(c2ccon2)=O)C1 39829,c1(C(=O)NC2CC(CNC(C3CCN(C)CC3)=O)C2)cc(F)ccc1N 39830,N1(C(c2[nH]cc(CC)c2)=O)CCC(N(C(c2ccc(CN(C)C)s2)=O)CC)CC1 39831,C(=O)(CCC(C)(C)O)NC(C1CN(C(=O)C2=CCCCC2)C1)C 39832,c1(OCC)ccc(F)cc1C(=O)NCCNC(C1COCCC1c1ccccc1)=O 39833,N1(C(c2cncc(N)c2)=O)CCN(C(c2cc3c[nH]nc3s2)=O)C2CC12 39834,C(=O)(C(=O)CC(C)CC)N1CCCCC1.C(=O)(CS(=O)CC)N(NCC)CC 39835,c1(C(=O)NC2CCC(NC(c3c(CC)nns3)=O)CC2)cc2c[nH]cnc-2n1 39836,n1(CC)c(=O)c(C)nc2cc(C(=O)NCC3CC3NC(=O)COC(F)F)ccc12 39837,Cc1cc(CCCC(=O)N(CCCCCNC(C2CCC2F)=O)C)c(C)s1 39838,CC1(C)CCC2(CN(c3nccc(N4CC5C(C4)C5(F)F)n3)CCO2)C1 39839,C(=O)(C1OCCc2ccccc21)N1CCC(C)C(NC(=O)C(C)(F)C(C)(C)F)C1 39840,S(=O)(=O)(c1[nH]c(=NC(C)Cn2ccnc2C)ccc1Br)NCc1c(C)cccc1 39841,c1(C(N2C(CNC(C(C)(C)Br)=O)CCC2)=O)cccc2cc[nH]c12 39842,CCC(C)(C#N)C(=O)NCc1nnc(C2CCN(C(=O)C3=CCC3)CC2)s1 39843,C(=O)(C(C(C)C)n1cnnc1)N(CCN(C(=O)C(=Cc1cnc[nH]1)C)CC)CC 39844,c1(SC)c(C(=O)NC2CCCC2NC(c2conc2C(C)(C)C)=O)cnn1C 39845,C1(C2CCOCC2)(C(N2CCN(CCCNC(CCC3C(C)C3)=O)CC2)=O)CC1 39846,C1(NC(C=CC=CC)=O)CC(O)CN(C(=O)C(C)(C)CC#N)C1 39847,C1(C(N(CCNC(C(C)NS(CC)(=O)=O)=O)CC2CC2)=O)CCCSC1 39848,N1(C(C(C)O)=O)CCC2(CCCN2C(C2CCc3cn(C)nc3C2)=O)CC1 39849,c1(C(=O)NC(C2CCN(C(C(CC)OCC)=O)C2)(C)C)cc2n(n1)CCO2 39850,C1(NC(C2N(C(C)=O)CCC2)=O)CC2(C1)CN(C(=O)CC1C(=O)N(C)N=C1C)C2 39851,C(=O)(C(F)C(=O)NCCN(C(c1cc(=O)n(-c2ccccc2)[nH]1)=O)CC)OCC 39852,Cc1ccc(C2CC(C(=O)N(C)C)OC2)cn1.C12(CCOCC1)CNC(=O)NC2 39853,N1(C(c2ccnc(OC)n2)=O)CCC2(CNC(=O)C(C)=C3CCC3)CCCCC12 39854,C1(C(N(CCNC(C2CCCC(C)(C)C2)=O)CC)=O)CC12CCCCCC2 39855,C(=O)(CCCCC(F)F)N1CC2C(NC(c3ccc(N)cc3F)=O)C(C2)C1 39856,n1(CC)cc(Br)cc1C(=O)NCCOCCNC(C1(CF)CC(F)(F)C1)=O 39857,C1(CNC(c2cscc2F)=O)CCCCC1NC(C1CCC(O)C1)=O 39858,C=C=CCCNC(=O)C(C)NC(=O)C(C)c1cccs1 39859,Cc1cc(CNCc2cnc(N3CCOCC3)s2)c(O)c(Br)c1 39860,c1(C(=O)NCCOCC(=C)C)cccnc1CNC(=O)CN1CCCCCC1 39861,c1(N(C(CC(=O)NC2C(CC)CCCC2)=O)CC)ccc2nc(N(C)C)sc2c1 39862,C1(N(C(Cc2c(C)scc2)=O)C)CCCC(NC(=O)C=CBr)C1 39863,c1(C(=O)NCCC2CCN(C(CN3C(C)CCC3)=O)C2)cc(N)c(F)cn1 39864,C(=O)(CC(F)(F)F)NCC(C(=O)NCC(=O)NCC=C)C 39865,CC1=C(C(=O)N(C)CC2CCCN2C(C2OCCC2C(C)C)=O)CCO1 39866,C1(NC(CCn2c(C)ncc2)=O)CCCN(C(C2CSCN2S(C)(=O)=O)=O)CC1 39867,N1(C(CC(=O)OC)=O)CCOC2CN(C(c3n[nH]c4cc(C)ccc34)=O)CC12 39868,c1(C(N2C(C)CCC(CNC(CC(CC)OC)=O)C2)=O)cccc2ccsc12 39869,N1(C(=O)Nc2ccc(-c3nc(C(F)F)no3)c(Cl)c2)CCc2[nH]ccc2C1 39870,C(=O)(C(CC1CC1)NC(=O)CC=CC(C)(C)C)N1CC(CCC#C)C1 39871,c1(OC)ncc(C(N2CC(N(C(=O)CN(C)C3CC3)C)C(O)C2)=O)cc1F 39872,c1(OC(c2nc(-c3cc(O)cc(C#N)c3)no2)C)nc2ccccc2s1 39873,N1(C(c2c(C)nc(C)[nH]2)=O)CCN2CCOCC2(CNC(=O)CC(C)F)C1 39874,c1(C(=O)NCCC(C)N(C)C(C2(C)CCOC2)=O)sc2ncccc2c1N 39875,C1(CC)CN(C(C2CCCC(C#N)C2)=O)CCN1C(=O)CCCc1ccccc1 39876,c1(C(=O)NC2C(NC(CC(COC)C)=O)C2)cccc(=O)n1C 39877,Cn1cnc2ccc(C(=O)N(CCNC(=O)COCCF)C3CC3)cc12 39878,N1(C(C2(C)C=CCN2C(=O)CN2CCSCC2)=O)CC2CC1CC2CF 39879,N1(c2cc(C)ncn2)CCCC12CCN(C(c1cccc3c1ncn3C)=O)C2 39880,C1(C(N2CC(c3n(C)ccn3)C(NC(=O)C3=CCC3)C2)=O)Cc2cscc2C1 39881,N1(C(c2occ(C)c2)=O)Cc2ccccc2C(NC(c2ccc(N)c(O)c2)=O)C1 39882,C(c1ccccc1F)=CC(=O)NC(C)CC(C)NC(=O)C1=C(Cl)CC1 39883,C1(NC(CCC=CCC=C)=O)CCN(C(c2cnoc2C)=O)C12CC2 39884,CC1CCC(=CC(=O)NC(C)CNC(=O)C(C)N2CC(C)C2)CC1 39885,C1(C(N2CCOC(CCNC(c3cccc(Cl)c3)=O)C2)=O)(CSC)CCOCC1 39886,N1(C(c2nc(C(C)(C)C)sc2)=O)CC2(C1)CN(C(=O)CC1(C)CC1(Cl)Cl)C2 39887,C1(C(=O)NCCCNC(C2(CO)CCCCC2)=O)CCC2(CCC2)OC1 39888,CCC(C)C(O)C(C)C(=O)NCCn1cc(C(=O)NCC2(SC)CCC2)nn1 39889,C1(NC(c2ncn(C(C)C)c2)=O)CN(C(C2(O)CCOC2)=O)CC1C 39890,N1(C(c2c(C)cno2)=O)CC(NC(c2c(C)ncn2O)=O)CC12CCCCC2 39891,CC(C)(C(=O)NCC1CCCC1NC(=O)Cn1cc(CO)nn1)C1CCOCC1 39892,c1(OC)c(C(=O)NC2CCN(C(c3c(N)cccc3Cl)=O)C2)oc2ccccc12 39893,C1(CC)C(C(=O)NCc2ccc(C)cc2)CCN1C(=O)C(C)O 39894,N1(C(CC(=O)OCC)=O)CCC(C2CC2)C1CNC(c1cnc(C)c(C#N)c1)=O 39895,c1(OC)ccc(C#N)cc1-c1nc(CCO)nn1C(C)C(C)C 39896,N1(C(c2cccc(CNC(CCCCC#C)=O)n2)=O)CCC2C(CCN2C)C1 39897,c1(C(=O)NCCN(C(c2cncc(NC)c2)=O)CC2CC2)nc[nH]c2ncnc1-2 39898,c1(C(C)(C)NCCc2ccncc2)ccnc(Cl)c1F 39899,C(=O)(C1CCc2cccc(F)c21)N1CC(COC)OC(C)C1 39900,C(CC1=CCOCC1)NC(C(CC)N(C)C(c1cn(C)c(=O)cn1)=O)=O 39901,C1(NC(c2cc(Cl)no2)=O)CCC12CCN(C(=O)CCC1CC1)CC2 39902,N1(C(Cc2nc(C)sc2C)=O)CCCN(C(=O)CC(C)c2ccco2)C(CO)C1 39903,N(C(=NCCC)N1CCCC(CCC)C1)CCSCC=C 39904,C1(C(N2CCC(CC(=O)NCC(C(C)C)(F)F)C2)=O)CCC2(CCOCC2)C1 39905,Cc1ccc(CC(=O)NCC(C(C)(C)C)NC(=O)CC2(O)CCOCC2)c(C)c1 39906,N1(C(Cc2scc(C)c2)=O)CC(C)CN(C(=O)C(N2CCCCC2)C)C(C)C1 39907,C(C)(C)(CC(=O)NC(c1cn(C)nn1)C)NC(C=CCCC)=O 39908,c1(C(=O)NC2C(CNC(C3(C)CCC(=O)NC3)=O)CC2)cc2cc(Cl)ccc2o1 39909,C(=O)(CC(C)C(C)(C)NC(c1cnc(NC)cn1)=O)N1CCC(C)(CCC)C1 39910,c1(C(=O)OC)csc2cc(C(=O)NC3CN(C(=O)CSC(F)F)C4CC34)[nH]c12 39911,c1(C(=O)NC(C2CCN(C(c3csc(C)c3N)=O)CC2)C)ccn2nnnc2c1 39912,c1(C(=O)NC2CCN(C(C(COC)(C)OC)=O)CC2CO)cn2cnnc2cn1 39913,C1(NC(c2ccn(CC(C)C)n2)=O)CCN(C(=O)CC2CCC2)C1C1CC1 39914,CCC(C(=O)NCC(C)(CO)NC(=O)C(=O)N(C)C)C(C)(C)CC 39915,C(=O)(CCC(C)(F)F)NCCN(CCC)C(c1c(Cl)cncc1Br)=O 39916,CC1Cc2ccccc2N1C(=O)CC1CN(C(c2cnn(C)n2)=O)CCC1C 39917,CC(C)(CC(=O)NC1CCC(CNC(C2CCCC3CCCN23)=O)C1)C(F)F 39918,C1(C#N)(C(=O)NCC2CCC(NC(c3scc(C)c3Cl)=O)CC2)CC12CCCC2 39919,C1(C(N2CCC(OCC(N)=O)C2)=O)CCC(C)(C)N(C(C2CC2(Cl)Cl)=O)C1 39920,c1(CC(=O)N(C)CC2CCCN2C(C23CC(F)C2C3)=O)cc(Cl)sc1Cl 39921,CC(Cl)(Cl)C(=O)N1CCC(C2CCCN2C(c2csc(-c3ccco3)n2)=O)C1 39922,N1(C(C(CC#C)C)=O)CCN(C(c2cnn(-c3cccc(Cl)c3)c2)=O)CC1CO 39923,C1(OC)(CNC(C2C3CCCOC23)=O)CCN(C(=O)Cn2nnc(=N)[nH]2)C1 39924,C#CCCC(C(=O)NCC(c1ccco1)O)NC(=O)C=C1CCC(C)CC1 39925,c1(CNc2c(C(=O)NCc3ccsc3)scc2)cn2ccccc2n1 39926,c1(OC)ccc(C#N)cc1NC(=O)C(F)C1CC(C(=O)OC(C)(C)C)C1 39927,C(=O)(C(F)C(F)(F)F)NCC(C)(C)OCCNC(C(C)Cc1ccccc1)=O 39928,C1(C(=O)NCCC2(CNC(c3ccc(C#N)o3)=O)CC2)C2(CCC2)C12CCC2 39929,N1(C(C(C(COC)C)C)=O)CCCC2(NC(=O)CC3CCCCC3C)CCCC12 39930,O=C(C1=C(Cl)CCOC1)NC1CC(NC(c2cc(C(F)(F)F)nn2C2CC2)=O)C1 39931,c1(CC=C)ccccc1C(N1CC(C(C)NC(C2CCOC2=O)=O)C1)=O 39932,N1(C(COCC(C)(C)C)=O)CCC(F)(CNC(=O)CSCC2CCCO2)C1 39933,N1(C(Cc2c(C)scc2)=O)CC2CN(C(=O)C(=O)NC(C)C)CCC2(CO)C1 39934,C(=O)(C1CCCc2ncnn21)NC1CCCN(Cc2cccc(OC)c2)C1 39935,C12(C(=O)NC(COC)(C)C)CCC1CN(C(=O)CCN1CCN(C)CC1)C2 39936,C(=O)(C(C)S(N)(=O)=O)N1C(CN(C(C(C)C2CCC2)=O)C)CC(F)C1 39937,C1(C#CC(=O)NCC2CN(C(C34CC5CC3C4C5O)=O)CC2(C)C)(CC)CC1 39938,C(CC)(C(=O)NC1(C(=O)NC(C)C(F)F)CC1(C)C)=CC 39939,O=C(CC1=CCCCC1)N1CCC2(CC2C(N2CCCC2CCO)=O)C1 39940,Cc1ccc(C(O)C(=O)NCC2CCN2C(=O)C(C2CCCCC2)C)cc1 39941,N1(C(c2ccc(C)s2)=O)CC2CCCCC2(NC(c2occ(C)c2C)=O)C1 39942,C1(O)(CNC(c2cc(-c3ccco3)no2)=O)CCCN(C(C2SCCS2)=O)CC1 39943,C1(=O)C(F)(C(C)C)CN1CC(C)(C)C.C1(C(C(=O)OC)=O)CCCCC1 39944,N1(C(C2CC(C)OC2)=O)CC2CN(C(c3ccc4nccn4c3)=O)CC(C1)O2 39945,N1(C(Cc2nc(COC)sc2)=O)CC2CC1CN2C(c1sccc1F)=O 39946,C1(C(=O)Nc2cn(CC)nc2)CC12CCN(C(=O)COC(C)=O)CC2 39947,C1(CNC(C2(C)ON=C(C)C2)=O)Cc2ccccc2CN1C(=O)Cc1ccns1 39948,N1(C(C(C)(C)c2ccccn2)=O)CC2CN(C(=O)CC3CCCCC3(F)F)C2C1 39949,Cc1ccnc(O)c1C(=O)NCC1(CNC(C2C3COCC23)=O)CC(F)(F)C1 39950,c1(OC)ccc(CN(C)CC2CCN(C(=O)COc3sncc3C)C2)cc1 39951,CC1CCCN(C(C)CNC(=O)NC2CN(Cc3ncccc3C(F)(F)F)C2)C1 39952,C12(C(=O)NC3C(NC(c4n(C)cc(C#N)c4)=O)CCC3)CC3CC(CC(C3)O1)C2 39953,c1(C(N(CC(C)NC(CCN(CCC)C)=O)C)=O)noc2c1CCCCC2 39954,C1(C)(C(N2CC(O)(CN(C(=O)CNC(c3cscn3)=O)C)C2)=O)C=CCCC1 39955,C(=O)(CCCNC(C1CCC1)=O)NC(CN(C(C1(C#C)CC1)=O)C)(C)C 39956,c1(C(C)C(N2CC(NC(c3nn(C)cc3Cl)=O)C3(CC3)C2)=O)c[nH]c2ccccc12 39957,C1(NC(CCC(C)C)=O)CCCC12CN(C(C1(C)CCN(C)C1=O)=O)C2 39958,C1(C)(CNC(c2c(C)cno2)=O)CCCN1C(=O)CCSCC(N)=O 39959,Cc1noc(C)c1COc1ccc(C(=O)NCCC2CCN2C2CCCC2)cc1 39960,Cc1ccc(C(F)(F)F)c2c1N(Cc1cncc(N(C)CCO)c1)CC(C)C2 39961,C(C)(CN=c1nc(C(=O)OC)[nH]cc1OC)NC(c1ncc(OCC)nc1)=O 39962,C1(C(=O)NC2(C(N3CC(N4CCCC4)C3)=O)CCN(C)C2)CCC2(CCC2)O1 39963,C1(CNC(=O)C(F)(F)C2CCCO2)CC2CCC(C1)N2c1ncc(Cl)cn1 39964,N1(C(C(CCSC)O)=O)CC(C)N(C(c2ccc(CO)cn2)=O)CC1C 39965,C(C(O)C(=O)N1CC(O)(C2CCCN2C(=O)CCc2nc(=N)[nH][nH]2)C1)SC 39966,N(C1CCCc2c(F)cc(F)cc21)C(C1CCCO1)=O 39967,N1(C(C(C)NC(CC)=O)=O)CC(CO)C2(C1)CN(C(=O)CC(C)(C)CCOC)C2 39968,N1(C(C2C(CC)OCC2)=O)CC(N(C)C(c2cc(C)c(C)[nH]2)=O)C(C)(C)C1 39969,N1(C(C(C2CCC2)OC)=O)CCC2CN(C(=O)Cc3cc[nH]n3)C(C)C12 39970,N1(C(=O)C2=CCCOC2)CCC2(CCCN(CCOc3ccc(Cl)cc3)C2)C1 39971,C1(CNC(c2n(C(C)C)cnc2)=O)CC(NC(=O)C(C2CCC2)N(C)C)CCO1 39972,Cc1c(C(N2CC3C(C(N)=O)C3C2)=O)cc(Br)cc1F.c1nc2cccnc2s1 39973,S(=O)(=O)(c1cccs1)NCCC(=O)NCC1(O)CN(C(C2(C)CC3(CC3)C2)=O)C1 39974,c1(C(=O)NCCNC(c2ccc(C3C(C)C3)o2)=O)ccc(CNS(C)(=O)=O)cc1 39975,Cc1ccc(C(=O)NCC2(NC(c3ccn(C4CC4)c3C)=O)CC2)nc1O 39976,c1(C(CN(C2CC(C)(C)C2)C(c2ccccc2)=O)O)ccc(F)cc1 39977,N1(C(C2CCN(C(C)=O)CC2)=O)CC2CCN(C(=O)Cc3cnccn3)C2C1.CC=O 39978,N1(CCNCC2(CCCC)CCC2)C(=O)c2ccccc2C1=O 39979,N1(C(C2=C(C)OCC2)=O)CC2CC(NC(c3nccc4n[nH]cc34)=O)C(C2)C1 39980,c1(C(=O)NC2C(CNC(C(CCC)OCC)=O)C2)cc(OCC)ccc1C 39981,C1(P(C)(C)=O)(C(N2CC(CCNC(=O)C(CN(C)C)N(C)C)(OC)C2)=O)CC1 39982,c1(OCCCC)ccc(C(=O)NC2CCCC2NC(c2n[nH]cc2Cl)=O)c(O)c1 39983,C1(C(N2CC(CC)(CC)C2)=O)CCN(C(c2cc(C3CC3)no2)=O)C(C)(C)C1 39984,c1(C(=O)OC)sc(C(N2CCC(NC(C3(CC(F)F)CCC3)=O)CC2)=O)cc1N 39985,O=C1NCC2CN(C(c3ccccc3OC(F)(F)F)=O)CC12 39986,c1(NC(CC2C(CNC(CCSC)=O)C2)=O)cnc2[nH]cnc2c1 39987,Cc1ccc([N+](=O)[O-])c(C)c1C(N1CCC1CNC(c1cnc(C2CC2)s1)=O)=O 39988,N1(C(c2noc(CC)c2C)=O)CC(NC(c2ccc(C#N)[nH]2)=O)CC(O)C1 39989,C12(NC(CC)=O)CCOCC1CN(C(c1ccccc1NC)=O)C2 39990,c1(NC(C2CC(O)CN2C(c2ccc(S)cc2)=O)=O)cccc(C(F)(F)F)c1 39991,C1(C(=O)NCC2(C)CCCC2O)C2CCC(C2)C1NC(C1(C)COCCO1)=O 39992,c1(OCCC)ccc(C=CC(N2CCN(CC3CC3)C(C)C2)=O)cc1 39993,Cc1ccccc1C1(C(N2CCC(NC(C3CC(OC(F)F)C3)=O)C2)=O)CC1 39994,c1(CNC(C2C(OC)CCC2)=O)ccc(CNC(c2c[nH]c(C)c2)=O)cc1 39995,C1(NC(CSc2c(C)cccc2)=O)CN(C(=O)CCCC(C)N(C)C)CC1(C)C 39996,CC(CC(=O)NC1(C(N2CCCCCC2)=O)CCSC1)C(F)(F)F 39997,c1(C(N2CC(CNC(C(c3ccccc3)OC)=O)C2)=O)c2c(nn1C)CCSC2 39998,c1(C(=O)NC(C)CCCNC(c2csc(=N)[nH]2)=O)nccn2nccc12 39999,N1(C(c2cc(C)on2)=O)CC(C)(C)OC2(C1)CN(C(C1C3(CC3)C13CC3)=O)C2 40000,CC1=NS(=O)(=O)NC=C1C(=O)N1CC(NC(c2c[nH]cc2C)=O)CCC1C 40001,C1(N(C(CSCC#C)=O)C)CN(C(C2CCCCN2S(C)(=O)=O)=O)CC1(C)C 40002,O=S(=O)(c1ccc(NC2CC(C)(C)C2)cc1Br)NCC1CCCC(O)C1 40003,CCCC(CC(C)C)C(=O)N1CC(COC)(NC(=O)CCC(=O)NCCC)C1 40004,C(=O)(CCC(C)(F)F)NC1C(OC)CN(C(=O)CC2CCCCC2)C1 40005,N1(C(CS(C)(=O)=O)=O)CC(C2(NC(=O)COCc3ccncc3)CC2)C1 40006,CCCCCC(C)(CC)C(=O)N1CC2CCC(C1)N2c1ccncn1 40007,c1(C(=O)Nc2scc(C(C)NC(C3CC3C(N)=O)=O)n2)ccc(F)c(Cl)c1 40008,N1(C(c2c(CC)nns2)=O)CC2CC2(CNC(=O)CCOCC(=O)OC)C1 40009,c1(C(=O)NCC(C)(C)NC(C2(O)CC3(CCOCC3)C2)=O)cnc2cc[nH]c2c1 40010,N1(C(CCNC(c2ccncc2)=O)=O)CCCC2CCN(C(C3(O)CC3)=O)CC12 40011,N1(C(C2C(NC(c3ccc(F)c(C)c3F)=O)CCC2)=O)CC2CCN(C)C(=O)C2C1 40012,c1(C(=O)NCC2(F)CCC(NC(C(CCOC)C)=O)C2)cc(OC)c(O)c(N)c1 40013,N1(C(C2C(C(C)(C)C)CC2)=O)CCC2CN(C(=O)C(C)N3CCCC3)C2C1 40014,S(=O)(=O)(c1ccc(NCC2(C(C)C)CCOC2)c(Cl)c1)N1C(C)CC2(CCC2)C1 40015,C1(CNC(c2cn(CCC)nn2)=O)C(C)CCCN1C(C1CCCS(=O)(=O)C1)=O 40016,CCC(C)CCC(=O)NCC(C(C)C)NC(c1c[nH]c(=N)s1)=O 40017,c1(C(=O)NC2CC3(C(=O)NC(CO)CCCO)COC2C3)c[nH]c2ccncc12 40018,C1(NC(c2cc(COC)oc2C)=O)(CO)CCN(C(=O)C(C)CC(F)F)CC1 40019,C1(NC(CCSC)=O)CC12CCN(C(=O)CC1CCCN(C)C1)C2 40020,N12C(C3CC(O)C1C3)C2=O.C1(NC(C2CN(C(C)C)C2)=O)CCCC1CN(C)C 40021,N1(C(N2CC(OCC)C2)=O)CCC(NC(=O)COCCC(C)C)C1 40022,C(C)(C1CCCc2ccccc21)NC(=NCC)NCCc1ccc(Cl)cc1F 40023,c1(NCC(C)N(C(c2ccc(C)nc2)=O)C)ncnc2sc(C)nc12 40024,C1(C(=O)NCC(CNC(C2CC3(CCCC3)CO2)=O)O)C2Cc3ccccc3C12 40025,CCCCC(CNC(C1C=C(C)CS1)=O)NC(=O)C(C)OCc1ccccc1 40026,c1(-n2cc(CC3CCN(C(C4CC45CCC5)=O)CC3)nn2)ccc(Br)cc1F 40027,c1(C(C(N2CCCC(N(C(CC(=C)C)=O)CCO)C2)=O)C)c[nH]c2ccccc12 40028,C(CC(C)C)(C(=O)N1CCCC(CNC(c2c(C)noc2C)=O)C1)OC 40029,n1(CC(=O)N(CC)CC)cccc(NC(=O)C(O)CN2CCCC2)c1=O 40030,C=C(C)C(O)CC(=O)NCCC1CN(C(c2cnn(CC3CCOC3)c2)=O)C1 40031,C12(CC(=O)NCc3cccc(C)n3)CCC1CN(C(C1CCCCNC1=O)=O)C2 40032,CC(C#N)CCC(=O)N1CCOC(CNC(=O)Cn2cnc(C(F)(F)F)n2)C1 40033,C(C(C)C)(C(O)C(=O)N1CCCC(CO)(CNC(=O)COCCCF)C1)OC 40034,C1(c2cn(-c3cccnc3)nn2)(N(C)C)CCN(C(c2cnn(C)c2F)=O)C1 40035,N1(C(CCSC)=O)CCC(C(=O)NC2(CF)CCC2)(OC)C1 40036,C1(NC(c2ccc(C)nc2)=O)CN(C(c2ccc(SC(F)(F)F)s2)=O)CCC1C 40037,C=CCC(C)(C(F)F)NC(=O)CC(C)CNC(c1ccncc1OC)=O 40038,Cc1nc(C)c(CC(=O)NCCCC2(NC(=O)CN(C)C(C)C)CC2)c(O)n1 40039,CCCC(C(=O)NCCCCCN1CCN(C(C2COC(=O)C2)=O)CC1)N(C)C 40040,C12(CNC(C3CC4(CSC4)C3)=O)CCN(C1)C2=O.C1(CO)CCCC12CC2 40041,C1(C(=O)NCC(C)(C)NC(c2ncoc2Br)=O)CCOCC1(C)C 40042,C(=O)(C(F)CC(C)(C)C)N(CC(=O)Nc1c(C)ncc(Cl)c1)C1CCC1 40043,c1(C(=O)NCCCN(C(C(C)C2CCCC2)=O)C)cc(F)cc(S(N)(=O)=O)c1 40044,C(CCC(C)CC(=O)N1CC(O)(CCNC(C2CCCOC2)=O)C1)=C(C)C 40045,N1(C(c2cc(C)c(=N)[nH]c2)=O)C2CCC(C(=O)NC3(CC(C)C)CC3)C1CC2 40046,C1(C(CNC(c2cc(C(=O)OC)on2)=O)=O)CCCN(C(=O)C(F)(F)C2CC2C)C1 40047,c1(C(N(CC(C)NC(c2c(OC)cccn2)=O)C)=O)cc(Br)cnc1C 40048,N1(C(CC2C(C)(C)C2)=O)CCCCC12CN(C(C1SC3C=CC1CC3)=O)C2 40049,C1(C(C)NC(C)CCc2ccccc2)CCC(=O)N1 40050,C1(OC)(CNC(C2CCC(O)C2)C(=O)NC2CC2)CCN(C(C)(C)C)C1 40051,C1(CNC(C(C)NS(CC)(=O)=O)=O)CN(C(=O)Cc2c(C)noc2Cl)C(C)(C)C1 40052,CS(=O)(=O)c1cc(C(N2CCC3CN(S(=O)(=O)C4CC4)CCC23)=O)ccc1F 40053,C1(CCOC)(NC(Cc2n(C)ncc2)=O)CCN(C(=O)CSc2nncn2C)C1 40054,Cc1cc(Cl)c(C(N2CC(C)(C)C2Cn2cc(C3CCCCO3)nn2)=O)s1 40055,C1(C(N(CC(N2CCCCC2)=O)C(C2CC(C(C)C)C2)=O)=O)CCS(=O)(=O)C1 40056,C(=O)(C1=NOC(C)C1)NCCN(C(C1C(C=C)OCC1)=O)C 40057,C1(NC(CC(=O)OC)=O)CC(O)CN(C(=O)Cc2ccc(OC(F)(F)F)cc2)C1 40058,C(CCCCC(=O)N1CC2CC1(CNC(=O)Cc1cc(C)cs1)C2)OCC 40059,c1(C(=O)NC2CCCN(C(C3C4COCC34)=O)C2)cc2oc(Br)cc2s1 40060,c1(CC(=O)NC2(COC)CN(C(c3cc(C#N)cs3)=O)C2)cnccc1Cl 40061,C(=O)(C(C)(CC)CC)NC(C1CCCCC1)CNC(C(C)=C(CC)C)=O 40062,C1(CC)CCCN(C(=O)CC2CC(F)C2)C1C(=O)NCCCCc1ncc[nH]1 40063,c1(CNC(c2ccc(CC)cc2)c2n(CCC)nnn2)csc2sc(C)cc12 40064,O=S(=O)(c1cccnc1NCCC1CCC2CC12)NCc1cc(C(F)F)on1 40065,c1(C(=O)NC2C(C)N(C(=O)CCc3cnoc3)CC2)nccc2[nH]ccc12 40066,Cc1c(C(N2CCN(C(=O)C(C)(C)CO)CC2CS(C)(=O)=O)=O)cccc1C#N 40067,C(C(CC(C)C)C(=O)NC1CC(CCNC(=O)C(C2CCCC2)OC)C1)OC 40068,C(C(C)(F)F)N(C(C=CC(C)NC(C1(C(N)=O)CC1)=O)=O)C 40069,N1(C(C2CCSCC2)=O)CC2CCC(C(N3CCC(N4CCCC4)C3)=O)(C2)C1 40070,c1(C(C)NC(=O)CSC(C)(C)C)ccc(CNC(C2(F)CC2)=O)cc1 40071,N1(CC(N2CCCN(C(CCC#CC)=O)C(C)C2)=O)CCSC2CCCCC12 40072,C1(NC(c2c(C)nn(C3CCOC3)c2)=O)C2CCCC1CC2 40073,N1(C(c2cccc(CC)c2)=O)CCC2(CC1)CC2NC(C1(C)CC(C)=NO1)=O 40074,N1(C(c2ccc(OC)s2)=O)CCC2CN(C(c3cc(N)cc(O)c3)=O)CC12 40075,CC1OC2(CO)CC1(C(N1CC3CC1CN3C(=O)C(F)CC1CC1)=O)C2 40076,C1(C(F)F)(CNC(CC(=O)NCC)=O)CCN(C(c2cnn(C)c2OC)=O)C1 40077,c1(CC)nc[nH]c1C(N1CCCC1CN(C(=O)CC1CCSCC1)C)=O 40078,C1(C)(C(=O)NCCC(C)N(C(=O)CCCCN2CCOCC2)C)CCC12CCC2 40079,c1(C(=O)NCCOCCN(C(CC2CCCC(OC)C2)=O)C)cc(Cl)ccc1N 40080,C1(C(N(C(C)CN(C)C(c2ccc(-c3cccs3)[nH]2)=O)C)=O)Cc2nccn2C1 40081,N1(C(Cc2ncn(C)c2)=O)CC2CC(C1)N(C(=O)CCC(C)(C)F)C2 40082,C1(NC(Cc2cnc(C)s2)=O)CC(N=c2[nH]c3cccc(F)c3s2)C1 40083,C1(N(C(C(C)OCC(F)(F)F)=O)C)CN(C(=O)CCc2nccs2)CC1(C)C 40084,c1(C2C(C(=O)NCCN(C(=O)Cc3cnn(C(C)C)c3)CC)C2)ccccc1Cl 40085,C1(NC(C=CCNC(CC(C)(C)C)=O)=O)CN2CCC1(C)CC2 40086,c1(C(=O)NC(CN(C(=O)CC2CC(C)(C)CO2)C)(C)C)ccc(Cl)c(N)c1Cl 40087,N1(C(c2c(C)nsc2C)=O)CC(NC(=O)CC(O)CN(C)C)CC2(CC2)C1 40088,C(C)(CCN=c1cc(C2CCCCC2)nc[nH]1)NC(c1ccn(CC(C)C)n1)=O 40089,c1(-n2cc(C3(F)CN(C(C4(CSC)CC4)=O)C3)nn2)ccc(C)cc1C 40090,C1(C(=O)NC(COCC)C)CN(C(C2(CC)CCCC2O)=O)CC1(F)F 40091,c1(C(N(C(CNC(CC(C)OC)=O)C2CC2)C)=O)cnc2ncnn2c1C(C)C 40092,C1(CNC(CCC=CCC=C)=O)CC(NC(c2coc(Br)n2)=O)C12CCC2 40093,C1(CC#C)(C(=O)NCC(C)(CNC(=O)C=CCN(C)C)OC)CCOC1 40094,c1(C(=O)NCC(C)(C)OCCNC(C(CC=C)C)=O)c(C)cc(C)nc1O 40095,CCC(C(=O)NC(c1cnc(C)s1)C)N(C(=O)CNC(=O)CNC(C)=O)C 40096,N1(C(C(C(C)(C)C)NC(=O)C(F)OC(F)(F)F)=O)CC2C3CCC(O3)C2C1 40097,C(C(C(=O)N1CCN(C(C)C)C(=O)C1)C(C)(C)C)NC(CC=C)=O 40098,CN(C1CCCc2n[nH]cc21)C(C1COCCC1C1CC1)=O 40099,c1(C(N)=O)cc(C(=O)NCC2OCCC2C(=O)NCC2(F)CC(O)C2)n[nH]1 40100,Cc1cc(C(=O)NC2CC(O)(c3cccnc3)C2)c2c(c1)CCC2 40101,c1(OCC)cccnc1C(N1CC(CCO)(NC(c2ccncn2)=O)C1)=O 40102,C=C(C)CC(C(=O)NC1CC(C(=O)NCC#CC(F)(F)F)CC1O)OC 40103,N1(C(c2ncn(CC)c2)=O)CCC(NC(=O)CNC=O)C1C 40104,c1(SC(CN(C(C)=O)C(C2CC(F)(CO)C2)=O)(C)CO)nnnn1CC(F)(F)F 40105,N1(C(C(=O)NCC)=O)CCOC2(CCN(C(=O)C(O)CC3CCOCC3)C2)C1 40106,c1(C(N2C(CNC(C=CC(N)=O)=O)CCCCC2)=O)noc2cc(F)ccc12 40107,O=C(N=c1[nH]c(Cl)nc2ccc(Br)cc12)C1CN(C(c2cocn2)=O)CCN1 40108,C1(N=[N+]=[N-])(C(=O)NC(C(C(=O)OC)C)C)CCN(C(C2CCCC2C(C)C)=O)C1 40109,N1(C(CC(C)N2CCCC2=O)=O)CCC(C(F)F)(CNC(C2(Cl)CC2)=O)C1 40110,c1(C(=O)NN2C(CNC(c3scc(COC)c3)=O)CC2)cccn2nncc12 40111,C#CC1CCN(C(=O)C(COC(C)C)NC(c2cccn(C)c2=O)=O)CC1 40112,c1(C(=O)NCC2CN(C(CC(C)(C)C)=O)CC2O)c(N)c(F)cc(F)c1F 40113,CCC(Cc1ccccc1)C(=O)NC(C)CNC(c1cc(C(F)(F)F)no1)=O 40114,S(=O)(=O)(c1cc(C(=O)O)c(Cl)cc1Cl)N(C1CC(C(N)=O)C1)C 40115,Cc1cc(C(N2CCOCC2)=O)ccc1NC(C)C(C)S(C)(=O)=O 40116,C=C(C)C(CC(=O)NC1CCCN(CC(=O)N(C2CCOC(C)C2)C)C1)OCC 40117,c1(C(N2CCC(O)(C(C)CNC(=O)C(O)C3CCC3)C2)=O)ncc2ccccn12 40118,C1(NC(c2n(CC)ncc2)=O)CCC(C(=O)NCC2CC3C=CC2O3)CC1 40119,N1(C(CC)=O)CCC(C(=O)NC2(CCO)CN(C(C3SCCCS3)=O)C2)C1 40120,c1(C(=O)NCC2(O)CCCN(C(COC)=O)CC2)cc(C)c(C)c2ncccc12 40121,N1(CCC(=O)Nc2cn(-c3ccc(OC)cc3)nc2)CCCOC(NC(C)=O)C1 40122,N1(C(CCC2(C)N=N2)=O)CCC(CCC(=O)NCCc2cnnn2C)C1 40123,S(=O)(=O)(c1cnc(NC(c2cccc(Cl)c2C)C)c(Cl)c1)NC(COC)C1CC1 40124,n1(CC)nc(C)c(C(=O)N(C)CC2CCN(C(=O)CC(C)OC)C2)c1Cl 40125,C1(Cl)(C(=O)OCC)CC12CCN(Cc1cnn(Cc3ccncc3)c1)CC2 40126,CCC(O)C(C)C(=O)N1CC(C(F)Cn2cc(-c3ccc(C)cc3C)nn2)C1 40127,C(=O)(C(O)CCCNC(=O)C=CC(=O)N(C)C)NCCC(CC)C 40128,C(C(CNC(=O)CCc1cnoc1)NC(=O)CC1CC(C(C)(C)C)C1)OC 40129,CC1(C)C(NC(c2cc(C3CC3)no2)=O)CCN1C(=O)Cc1cnoc1 40130,C=CC(CCC)CC(=O)NC(CC1CC1)C(=O)NOCC(O)CO 40131,N1(C(C2CC(=C)C2)=O)CC2CCC1C1CN(C(c3ccsc3S(N)(=O)=O)=O)CC21 40132,C(=O)(CCN(OC)C(=O)C(C)(F)CCCC)NCC(C#C)CC 40133,C1(S(C)(=O)=O)(C(=O)NCC2C(NC(CSC)=O)CC2)CC(O)C1 40134,C1(NC(Cc2cncc(C)c2)=O)CC2CCC(C1F)N2C(c1csc(S)n1)=O 40135,N1(C(CCN(C(c2ncn(C)n2)=O)C2CC2)=O)CCOCC(CO)C1 40136,C(=O)(C(O)CC(N)=O)N1C(C(N(CC)Cc2ccoc2)=O)CC=CC1 40137,c1(C(=O)NC(CN(C(=O)COC2CC(F)(F)C2)CC)C)cccc(OC)c1F 40138,N1(C(CC)=O)Cc2ccccc2CC1CNC(C1CCC2CC2C1)=O 40139,N1(C(CCOc2ccc(C)cc2)=O)CCN(C(C2CCCCN2C)=O)CC1C 40140,c1(C(=O)NCC2CCCC(C)C2)cccc(S(C)=O)c1 40141,c1(C(=O)NCCN(C(c2c(OC)c[nH]n2)=O)C)ccc2c(c1)NC(=O)CCC2 40142,c1(C(=O)NC(C(C)NC(c2c(CCC)nco2)=O)CO)cc2cccc(C)n2n1 40143,CC1CN(C(C)C(=O)N(CC(=O)NC(C(N)=O)C2CCCC2)C2CC2)C1 40144,C1(NC(c2csc(-c3ccco3)n2)=O)CC(O)CN(C(C2CC(O)C2)=O)C1 40145,C(C(CC(=O)N1COC(C)C1)NC(=O)OC(C)(C)C)NC(C)=O 40146,C(=O)(CCC(=O)NN(C)C)NCC(C)(C)OCCNC(C1C(COC)C1)=O 40147,c1(CC(=O)NC2CCC(NC(C3C(C(N)=O)C3)=O)CC2)cc(Br)ccc1Cl 40148,c1(SC)cc(C(N2CCC(C3CCCN3C(c3ccc(O)nn3)=O)C2)=O)c(C)o1 40149,C1(CC)CN(C(=O)C=C(C)c2cccs2)CC1NC(C1(C(C)(F)F)CC1)=O 40150,c1(C(=O)NC(CC)CNC(=O)CCc2cncc(C)c2)cc(N)cnc1C 40151,CC1(O)CCN(C(=O)C(c2cn(C)nn2)NC(C2(F)CCCCC2)=O)CC1 40152,N1(C(c2c(C)c(F)ccc2)=O)CCC2CCCN(C(c3cnco3)=O)C2C1 40153,C1(C(=O)NC(C)CN=[N+]=[N-])CN(C(C2CC(=C3CCC3)C2)=O)CCC1(C)C 40154,c1(CNC(c2n(CCCSC)nnn2)(C)COC(C)C)cc(Cl)cc(C)c1OC 40155,c1(CN(C(Cc2cc(C)no2)=O)C)cccc(CNC(C2CCCC(O)C2)=O)c1 40156,C1(C(=O)Nc2cncc(C(=O)OC)c2)CC12CCN(C(=O)COC1CCCC1)C2 40157,N1(C(c2c(C(N)=O)cccc2)=O)CCC(F)C(NC(C2CCC(=O)C2)=O)C1 40158,c1(NC(C2(F)CN(C(c3c(CC)cccc3)=O)C2)=O)cc([N+](=O)[O-])ccc1I 40159,CC1OCCC1(F)C(=O)NC1CC(C(=O)N(C)CCC2CCCCC2)C1 40160,C12(CNC(COCC(=C)C)=O)CCC(C1)N(C(=O)C=C(C)C(C)C)C2 40161,c1(C(=O)NC2C(CNC(c3ccc(C4CC4)o3)=O)C2)cc2c(s1)CCCC2 40162,C(=O)(C(CCC(C)C)NC(c1cc(C)oc1C)=O)NC1CCN(C(C)=O)C1 40163,n1(CCC(C)N(C)C)nccc1-c1ccc(=N)[nH]c1 40164,C1(C2CCCN(C(=O)Cc3ccc4n[nH]cc4c3)C2)(NC(C=CSC)=O)CC1 40165,C1(C(N2CCN(C(CC3(C)CC3(F)F)=O)C3(C2)CC3)=O)CC2(CCOCC2)CO1 40166,C1(OC(C(C(C)C)C)=O)CC2(COC(C)C2)C1 40167,N1(C(c2c(C)onc2)=O)CCN(C(=O)C(C)Cc2cnc[nH]2)C2(CCC2)C1 40168,c1(CC(=O)NC(CCNC(CCCOCC)=O)C)cccc(Br)c1 40169,c1(CN(C(=O)NC2CCC(NC)CC2)C)ccc(C(C)C)nc1O 40170,C(=O)(C(O)CC[S+](C)C)NCC1(F)CCN(C(C2(COC)CC2)=O)C1 40171,c1(OC)nccc(C(=O)NC2CCN(C(=O)C(C)(C)Br)CC2O)c1Cl 40172,[N-]=[N+]=NCCC(=O)NCCC(O)C(=O)N1CCOC(C2CCC2)C1 40173,C(=O)(C(F)C(CC)CC)N1C(CNC(CN(CCCCCC)C)=O)CC(OC)C1 40174,N1(C(=O)CCCn2cccc2)CC2(CCCCN2C(=O)CCN2CCC(F)C2)C1 40175,Cc1ncc(C#N)c(N(C(c2cccc(Cl)c2O)=O)CC2CCNC2)n1 40176,C(CN=c1ccnc(N(CCS(N)(=O)=O)C)[nH]1)N1CCCC(C)C1 40177,c1(C(=O)NC(CCNC(Cc2ccn(CC)n2)=O)C)cc(C)cc(O)c1 40178,c1(C(=O)NC2CC(C)(C)CN(C(=O)C(O)C(F)F)C2)c[nH]c2ccncc2c1=O 40179,C1(NC(CCNC(CC(C)C)=O)=O)CN(C(=O)C(C)(C)C(F)F)CCC1O 40180,CC(C)C(C)CC(=O)N1CCC(CC(F)C(=O)NOCC=CCl)C1 40181,c1(C(=O)NC2C3CN(C(C4CCC(=O)N4)=O)C2C3)c[nH]nc1[N+](=O)[O-] 40182,N1(C(C(C(C)C)CO)=O)CC=C(CCNC(c2cc(F)c(CO)c(F)c2)=O)CC1 40183,c1(C(=O)NCC(CC=C)NC(CCC#C)=O)ccc(OCC(F)(F)F)nn1 40184,C1(C(N(C(CCNC(c2c(C)ncnc2)=O)C)C)=O)COc2ccc(F)cc2C1 40185,c1(NC2CC(C)N(C(=O)CCCc3ccsc3)CC2)ncc([N+](=O)[O-])cc1Cl 40186,O=C1CN(CC(=O)NCc2nc(CNC(C3(C4CCC4)CC3)=O)cs2)C(=O)N1 40187,c1(C(=O)NCC2C=CC(NC(C(CC)SC)=O)C2)c(Cl)ccc2c1OCO2 40188,c1(C(N2C(CC(=O)NCC3CC(C)(F)C3)CCCC2)=O)cccn2cncc12 40189,C12(C(=O)NCc3ccnc(C)n3)CCC1CN(C(C1CCCC1F)=O)C2 40190,C(=O)(CC(C(C)OC)NC(=O)CCc1cn(C)cn1)NC1C(OC)COCC1 40191,c1(OCC)nc2ccc(C(=O)NC3CC(N(C(=O)CC4CC4)C)C3)cc2[nH]1 40192,c1(C(N(C(C)CCNC(=O)CC2CCC(F)(F)C2)C)=O)cccc2c1CCC2=O 40193,C(C(CC(=O)NCCOCC(F)F)NC(=O)C(O)CN1CCCC1)OCC 40194,C#Cc1c[nH]nc1C(N1CCSCC1CCNC(c1scnc1CC)=O)=O 40195,C1(NC(C2(COC)CCCC2)=O)COCCN(C(=O)Cn2cc(Cl)cn2)C1 40196,C(=O)(C1=CCCCO1)N(C(C)C(=O)NCC1CC(=O)NC(C)C1)CC 40197,C1(NC(c2cnc(CC)s2)=O)(CF)CCN(C(=O)C(c2cscn2)N(C)C)C1 40198,c1(C(N2CC(OC)C(NC(=O)CSC)C2)=O)cnc(O)c(Cl)c1 40199,c1(OC)ccc(Cl)cc1CC(=O)NCC(C)(C1CC1)NC(=O)CCc1ccsc1 40200,N1(C(c2nc(CNC(C(C)C3CCCC3)=O)oc2)=O)CC(C2CCCCC2)C1 40201,C12(C(N(C3CCCN(C(c4c(CC)c[nH]n4)=O)CC3)C)=O)CC3CC(CC1C3)C2 40202,C12(NC(c3c(C)ncs3)=O)CCC(CN(C(c3ccc(F)cc3Cl)=O)C1)C2 40203,C(C1CN(C(C2(C)CCCCCC2)=O)CC1C(=O)NCC(C)(COC)CC)=CC 40204,C1(C(=O)NC2CC(NC(CC(C=C)(C)C)=O)C2)COc2ccc(OC)cc2C1 40205,Cc1nc(=N)[nH]cc1C(N1CCN(C(=O)Cn2ccnn2)CC1C1CC1)=O 40206,C1(CCC(=O)NCCC(C)NC(=O)C(c2ccc(F)cc2)(F)F)CCCCN1C 40207,C1(C(=O)NCC(C(C)C)(C)NC(=O)C2=COCCO2)CNC(=O)CC1C(F)(F)F 40208,C#Cc1cc(=NCC(c2ccncc2)OC)cc[nH]1 40209,Cc1nn(C)cc1C(=O)NCCOC1CCN(C(c2ccccc2Cl)=O)C1 40210,c1(CN(c2ccnc(N3CCOC(CO)C3)c2)C)cc2c(cc1O)CCCC2 40211,CC(C)CC(O)C(=O)NC(C)CNC(c1cc(C(F)(F)F)cc(N)c1)=O 40212,C(=O)(C1CCCn2ccnc21)NCC(C)(C)NC(C1N(CCCC)CCOC1)=O 40213,N1(C(C=CCNC(C2CC(C)(O)C2)=O)=O)CCc2ncccc2C1 40214,C1(C(=O)NCC(=O)NCCC)(CC)C=CCN1C(=O)COCCCN=[N+]=[N-] 40215,C(C(COC)CC(=O)NC1CCC(NC(=O)CC=C(Cl)Cl)CC1)OC 40216,c1(NC(CNC(=O)Nc2ccn(CCOC)n2)=O)ccc2ncsc2c1Br 40217,Nc1ccc(C(=O)NCC2CC3CCC2N3C(=O)C=C2CCC2)c2cccnc12 40218,N1(C(c2n[nH]c(CC)c2C)=O)CC(C(=O)NCCC2CC2C)OC(C)C1 40219,C12(CC)CC1CN(C(C1CCCCC1CNC(=O)C(C)c1cc[nH]n1)=O)C2 40220,c1(C(=O)NC(C2CN(C(C(=O)NCC)=O)C2)C)ccc2nnc(O)n2c1 40221,c1(C(=O)NC(CCOCC)C(=O)N2CC(c3ncc[nH]3)C2)cccc(=O)n1C 40222,c1(C(C(N2CC(C)N(C(=O)COC3CC=CC3)CC2)=O)O)cccc([N+](=O)[O-])c1 40223,Cc1ccc(CN2CCOCC2)cc1CC(NC(=N)N(C1CCCCC1)C)=O 40224,O=C(C(O)Cn1cncn1)NC1CN(C(C2CC2(Cl)Cl)=O)C1 40225,Cc1nc(C#N)c(NC(C2(O)CCN(C(c3ccccc3C(F)(F)F)=O)C2)=O)o1 40226,C1(C(=O)NC2C(NC(CC=CC=C)=O)CC2)CCc2ncsc2C1 40227,c1(C(=O)NC(C)CC(C)NC(=O)Cc2ccc(C#N)cc2)cnc2[nH]ccc2n1 40228,Cn1nc(C2CC2)nc1CNC(=O)COC(C1CCCCC1)=O 40229,N1(C(c2cnc(C)s2)=O)CCC(NC(c2cc(=O)n(C)o2)=O)CC1C 40230,C1(c2n(C(C)C(F)(F)F)nc(-c3ccc(Cl)cc3)n2)CC12CCOCC2 40231,c1(C(=O)NC23CN(C(C4(OCC)CCCC4)=O)C(C2)C3)ccc2n[nH]cc2c1 40232,c1(C(=O)NC(CNC(CC(C)C2CCCO2)=O)C)cccc(P(C)(C)=O)c1 40233,c1(C(N(CCNC(C2(O)CCSC2)=O)CC)=O)ccc(S(=O)(=O)NC(C)C)cc1 40234,Cc1ccsc1-c1cn(C(C)C(=O)N(C2CC2)C2CC2)nn1 40235,CCCC(CC(C)C)C(=O)NCC(C)CNC(c1cc(N)cc2c1OCCC2)=O 40236,NS(=O)(=O)C1CN(C(=O)Cn2nnc(-c3ccc(Cl)cc3)n2)C2(CCCC2)C1 40237,c1(CC(=O)NCc2c(CCNC(C(C)(C)C3CC3)=O)ocn2)ccc2c(c1)CC2 40238,c1(C(N2CC3C(CNC(C(CCC)N(C)C)=O)C3C2)=O)cn(C)c(C)cc1=O 40239,CC1(C)C(C(=O)NC(CCO)c2ccco2)CCN1C(=O)CCCn1cncn1 40240,Cc1nc(C2CC2)ncc1C(=O)N(CCCNC(c1ccco1)=O)C(C)C 40241,CC(CNC(C1COCCC1C)=O)C(F)C(=O)NC1(CC2CCC2)CC1 40242,n1(CC=C)c(SCC2NCCC2C)nc2sc3c(c2c1=O)CCC3 40243,C=CCC(F)(F)C(=O)NCC1(C)CCC(NC(=O)CCSCC)C1 40244,N1(C(C=C(C)Cl)=O)CCCN(C(=O)CCOC2CCC2)C(c2ccccc2)C1 40245,CC(C)C(O)C(F)(F)C(=O)NCC1C(C)CCCN1C(=O)CCc1cnc[nH]1 40246,c1(C(=O)NC(CNC(C2C(=C)CC2)=O)CCOC)c(C)cc(C)oc1=O 40247,C1(C(N2CC(OC)CC2(C)CNC(=O)CS(C)(=O)=O)=O)CC2(C1)CC(C)(C)C2 40248,C1(N(CCOC)C)CCN(C(c2cn(C)cn2)C(=O)NCC(C)C)CC1 40249,CCCCCC(C)CC(=O)NCCC(O)CNC(c1ncoc1C1CC1)=O 40250,CC(C)CC(C(=O)N(C)CC1(CO)CC1)NC(C1CCC(=O)N(C)C1)=O 40251,C(CCSC)(C(=O)NCCSCc1cn(Cc2ccccn2)nn1)SC 40252,C1(C(=O)NC(CCCOC)(C)C)CCC(O)CN1C(=O)CCCn1cccc1 40253,C1(C(N2CCC(F)C2)=O)CC2OCCC2N(C(C2Cc3ccccc3C2)=O)C1 40254,c1(C(=O)NC2C(NC(=O)C=Cc3cocn3)C2)cc2c(s1)CCCC2 40255,CCCC(CCC)C(=O)Nc1cccc(CC)c1.n12cnc(c1)C(=O)NOCC2 40256,Cc1nc(N2CCOC(C(=O)Nc3nc4c(s3)CCC4)C2)c2c(n1)CCC2 40257,Cc1cc2sc(C(=O)NCCC(C(C)C)NC(=O)C(c3ccccc3)O)cc2s1 40258,C(=O)(C(C)(C)C(=O)NCC(C1CC1)NC(C1CC2CC1CC2O)=O)N(C)C 40259,N1(C(CCS(C)(=O)=O)=O)CCC(C2CCN(C(C3CCSC3)=O)C2)CC1 40260,c12ncccc1C(=O)NC2.CC1CC(CCC(=O)N2CC(CF)C2)C1 40261,N1(C(C(CCCNC(C2(OC)CCCOC2)=O)O)=O)CC2(CNC(=O)OC2)C1 40262,C1(NC(C(CC)N(C)C)=O)(CO)CCCN(C(C2(Cc3cnn[nH]3)CCC2)=O)C1 40263,c1(C(=O)NCCC2CC(NC(C3CC3Cl)=O)C2)cc2c[nH]cnc-2n1 40264,Cc1ccc(F)c(C(N2CCCC(C)(CNC(c3c[nH]c(C#N)c3)=O)C2)=O)c1F 40265,O=C1CCC2(C(=O)Nc3cccc(-c4nncn4C4CC4)c3)CC3(CC3)CN12 40266,C1(OC)CN(C(c2c(C)noc2N)=O)CC1C(N1CCOCC1CO)=O 40267,N1(C(c2cc(C)ncc2)=O)CC(C(=O)NCC2CC(=O)N(C)C2)CC(F)C1 40268,c1(C(N(C2CCCN(C(c3csnc3Cl)=O)C2)CCO)=O)ccc2[nH]ccc2c1 40269,c1(C(C(=O)O)N(C)C(c2nnn(C3CC3)c2C(F)(F)F)=O)c(F)cccc1F 40270,n1(C(C)C)cc(C(=O)NCC2COC(CN)C2)c(O)nc1=O 40271,N1(C(c2sc(C)c(C)c2C)=O)CCCC(C2CN(C(=O)C3=CCCOC3)C2)C1 40272,N1(C(C(C)=CC(C)(C)C)=O)CCC2CC2(C(=O)N(c2cccc(CO)c2)C)CC1 40273,CC(CCNC(=O)C=Cc1ccco1)CCNC(C1COCCN1C)=O 40274,c1(C(N2CC(C(C)NC(c3c(C)scc3)=O)C2)=O)cnc2ccccn12 40275,C1(OC2(CC(=O)N(CC(=O)OC(C)(C)C)C)CCC2)CCCCCC1 40276,c1(C(N2C3C(CNC(CC=CC=C)=O)C(CCC3)C2)=O)nc2n(c1Cl)CCCC2 40277,N1(C(C(CCC)OCC)=O)CCc2nc(CNC(=O)Cc3cnc[nH]3)sc2C1 40278,C=C(C)CCCC(=O)NCC(CCOC)NC(c1nc(OC)cc(OC)n1)=O 40279,c1(C(C)C)ccc(C2CCCN(C(=O)C(C)n3cncn3)C2)cc1 40280,C12(CC(=O)Nc3ccc(CO)cc3)CCC1CN(C(c1ccncc1O)=O)C2 40281,C(=O)(C(C#N)CC)N1CC(N(C(=O)CCN(N2CCOCC2)C)CC#C)C1 40282,C1(CC=C)(Nc2cccc3cncn23)CC2CCC(C1)N2C(=O)OC(C)(C)C 40283,c1(-c2c(CCC(C)OC)cccc2)cc(F)ccc1F 40284,CC(C)(C)CC(C)(C)C(=O)NCC1CCN1C(c1ccc(O)c(Cl)n1)=O 40285,C1(O)(C(=O)Nc2cn[nH]c2)CC(C)(C)C1.C12COCCC1C(=O)N(C)CC(=O)N2 40286,N1(C(C2=CCN(C)C2)=O)CC(CNC(C2C=CCCC2)=O)CC(C)(C)C1 40287,c1(CCNCc2cc(C)n(C)n2)ccc2ccccc2c1.C1(C)C(=O)N1 40288,c1(N(CCC)C)ccc(C(=O)NC23CC2CN(C(=O)C(C)n2cccc2)C3)cc1 40289,CCC(C)C(O)CC(=O)NCC(C)(C)OCCNC(c1cnc2ccccn12)=O 40290,C1(NC(c2cnoc2)=O)CN(C(=O)COC2CCCCC2)CC(F)(F)C1 40291,c1(CCC(=O)NC2CCN(Cc3c(COC)noc3)C2)ccc(Cl)c(Cl)c1 40292,N1(C(COCCCCC)=O)CCC(CCC(=O)NCc2scnc2C)C1 40293,c1(C(=O)NC(CNC(CC=CC)=O)CC)csc(-c2nc[nH]n2)n1 40294,Cn1ccc2cccc(C(N3CCC(C)(NC(C4CCCS4(=O)=O)=O)C3)=O)c12 40295,N1(C(C(CC)OC)=O)CC2CCC(C1)N2CCCn1ccccc1=O 40296,c1(C(C(=O)NC2CCCC2)N(CCC)CC)cnc2n1CCC2 40297,N1(C(CCSC)=O)CC2=C(C1)CN(C(c1cnc(C(F)F)c(C)c1)=O)C2 40298,c1(C(N(C2CN(C(C(CC)(F)F)=O)CC2O)C)=O)cc(F)c(C(C)C)cc1F 40299,c1(C(=O)NCCC2(C(=O)NCC3CN(C)C3)CC2)ccc2nccn2c1 40300,c1(C(=O)NCC(C)N(C(=O)Cc2cc(Cl)ccc2O)C)cccc2c[nH]nc12 40301,C(=O)(C1=CCC(C)(C)CC1)NCC1(F)CCCN(C(CSCC=C)=O)C1 40302,c1(OCC)nc(C(=O)N(CC(C)NC(c2cc(Cl)c[nH]2)=O)CC)co1 40303,C(CC(C)C(=O)NC1CCCN(C(C2CN(CC(F)(F)F)C2)=O)C1)=CCC 40304,CC(C)C(C)C(=O)N(C)CC1(O)CCN(C(c2ccc(CC#N)cc2)=O)C1 40305,C(=O)(CN1C(=O)CCc2ccccc21)NCC1C(NC(CC2CN(C)C2)=O)CC1 40306,c1(NC(C=CCN2CCC(NC(CC(CC)C)=O)CC2)=O)ccc(Br)cc1F 40307,CC1(C)COCCC1NC(C1CC(NC(=O)Cc2ccc(O)nc2)C1)=O 40308,C1(C(N(CCN(CCC)C)CCOC)=O)CCC1C(=O)OCC 40309,N1(C(Cc2c(C)cnn2C)=O)CCN(C(=O)Cc2ccsc2)CC(O)C1 40310,C(=O)(C(C)C(O)CCCC)NC(C(=O)NCCCCC(=C)C)c1ccoc1 40311,c1(-n2c(C(C)CCC3CC3)nc(CN3CCOCC3)n2)ccnc2ccccc12 40312,N1(C(C(C)(C)F)=O)CCC2(CCN(C(c3coc(-c4ccc(F)cc4)n3)=O)C2)C1 40313,N1(C(C2N(C(CC(C)(C)C(F)F)=O)CCCCC2)=O)CCC2(CCCCO2)C1 40314,c1(C(=O)NC2CC(CS(N)(=O)=O)C2)cccc(C(=O)O)c1 40315,Cc1ncc(C(=O)NCc2ccc(C(=O)NC(C)(CO)C(F)(F)F)o2)c(C)n1 40316,C1(NC(Cn2c(C)nnn2)=O)CC(C)N(C(c2ccc(CO)nc2)=O)C1 40317,N1(C(C(C)(C)OCC)=O)CCN(C)C(CNC(C2CN(C)CC2OC)=O)C1 40318,C1(NC(C2(C)CCCS2)=O)CCC2(CC1)CCN(C(C1CCCC1(F)F)=O)CC2 40319,C1(NC(=O)C(CC(F)F)N2CCOCC2)CCN(C(=O)C(Cl)=CCl)CCC1(F)F 40320,Cc1csc2ncnc(NC(C)CC(C)NC(c3ccc4nccn4c3)=O)c12 40321,c1(C(N2C(C)(NCCC(CCO)c3nn[nH]n3)C=CC2)=O)cccn2nccc12 40322,c1(SC)nc(N2CCSCC2CCNC(C2(C)CNC(=O)C2)=O)cc(C)n1 40323,N1(CC(=O)NCC(CCC)OCC)CCN(C(=O)CC2CC3CCC2O3)CC1 40324,c1(N2CCCC(NC(c3c(C)nn[nH]3)=O)CC2)cc2ncnn2cn1 40325,c1(C(=O)NCCCN(C(C2C(C=C)C2)=O)CCO)ccc2c(c1)OCC2 40326,Cc1no[nH]c1=NC(=O)C1(C)CCN(C(=O)Cc2ccccc2I)C1 40327,c1(C(N2CC(C(=O)OC)CC(CC)C2)=O)ccc2c(Br)cnn2c1 40328,N1(C(C(C=C)OC)=O)CC(CC(=O)NCC(C)(O)CCC)C2(CC2)C1 40329,CN1CCN(C(C2(C)CCNC2=O)=O)CC1=O.c12conc1CNC2=O 40330,C1(C(=O)NC2CN(C(c3ccc(CC(C)(C)C)cc3)=O)C2)CCC(N=[N+]=[N-])CC1 40331,c1(OCCCC(=O)NCCC2CC(NC(CC=CC=C)=O)C2)ccc(F)c(F)c1 40332,c1(C2CN(C(C=C(C)C(C)C)=O)C2)ccc(F)c(F)c1 40333,CCCCC(COC)NC(=O)CCN(C(=O)CC(OC)OC)C1CC1 40334,N1(C(C2(C(=O)NC)CC2)=O)CCN(C(c2cn(C)nn2)=O)CC(CO)C1 40335,CC1CCC(Cl)=C(C(=O)NC2CC(NC(C3(n4cncn4)CC3)=O)C2)C1 40336,c1(OC(C(=O)NCC(CNC(C(C)(C)OC(C)C)=O)C)C)ccc(Cl)cc1 40337,C1(CCC)CN(C(c2cc(Cl)ccc2F)=O)CCN1C(=O)CC(O)C1CCCC1 40338,Cc1[nH]nc2ncnc(N(C(C)CCNC(c3ccc([N+](=O)[O-])[nH]3)=O)C)c12 40339,C=CC1CN(C(=O)C(CN(C)C)NC(=O)CCSCC)CCO1 40340,c1(C(=O)NC2CC(C)N(C(C3CCC(=O)NC3)=O)C2)cc(F)cnc1Cl 40341,C(=O)(CCCCC(C)CC)NCC1C(OCC)CN(C(c2cnc(O)n2C)=O)C1 40342,C1(CNC(c2cn(C)nc2C(C)(C)C)=O)CC2COCC2N1C(=O)C(C)(C)CO 40343,C(=O)(N=c1nn[nH]n1CCC(C)C)NC(c1ccc(Cl)cc1)CCC 40344,C(=O)(C(C)(C)C(=O)N(C)C)N1CCC(CC(C)NC(C(CC)F)=O)CC1 40345,C12(C(=O)NC(C3CCCOC3)COC)C3C4C1C1C2C3C41CN(C)C 40346,c1(CC)cc(NCC(C2CC2)NC(C2CCC(CC)CC2)=O)ncn1 40347,C(C(=O)N1CCCC1C1CCCC(C)(C)C1)(C(C)(C)C)n1cc(C(=O)OC)nn1 40348,c1(C(=O)NCCN(C(C2C(C)C2C)=O)C)csc(Cl)c1Cl.n12cc(cn1)C2 40349,c1(OCC)ccc(Br)c(C(N2CC(c3cn(CC(C)(C)COC)nn3)C2)=O)c1F 40350,c1(C(=O)NCCC2N(C(C(CCSC)O)=O)CCC2)cn(C)c(=O)n(C)c1=O 40351,c1(C(N(CC(CNC(Cc2c(C)noc2)=O)O)C)=O)cncc(-n2cccn2)n1 40352,N1(C(c2cc(C(=O)O)c(F)cc2)=O)CCC2CCCN(Cc3ccncc3)C2C1 40353,C1(C2CCN(C(COCC(c3ccncc3)C)=O)C2)CCCCN1C(=O)C(N)=O 40354,C(CCCCCCC(=O)NC(CNC(=O)CC(C)C(C)C)C1CC1)SC 40355,c1(OC)ncc(C(=O)NC2CN(C(=O)COCC3CCCO3)C2)nc1C 40356,CC(O)(CCNC(N1CC2(CCC2)C1CO)=O)C(F)(F)F 40357,c1(C(N(CCN(C(=O)C(c2cncn2C)O)C)C)=O)ccc(N)c(N)c1 40358,N1(C(CCOC(C)=O)=O)CC(C2CC2C(=O)N(C2CCOCC2C)C)C1 40359,N1(C(C(C2(O)CCCCC2)CC)=O)CCN(C(c2cnc(O)n2C)=O)CC1C 40360,C1(NC(Cn2c(C)c(Cl)cn2)=O)CC2CCC1N2C(C1(C)CC=CC1)=O 40361,CC1=C(C(=O)NC2CCC(NC(c3cn(C)nc3Cl)=O)C2)C=C2CCCN=C2N1 40362,CCCCCCOC(C)C(=O)NCC(CC)NC(c1ccnn1C1CCCC1)=O 40363,C1(C)(C(=O)NCC2CCN(C(COCC)=O)C2)CNC(=O)C1 40364,N1(C(C(CC)=CC)=O)CCC(O)(Cn2cc(C3CCN(C)C3=O)nn2)CC1.C1CO1 40365,N1(C(C2(CC=C)CCN(C(=O)C=CCN3CCC3)C2)=O)CCCCC(OC)C1 40366,C1(C2CCN(C(C3CC4CC3C4)=O)CC2)(NC(CCC(CCCC)C)=O)CCC1 40367,C(c1ccc(C(F)(F)F)cc1C)=CC(N1C(CCOC)(C(=O)OC)CCC1)=O 40368,C1(C(=O)OC)CC=CCN1C(C1CC2CCCC12)C(=O)NC(C)C 40369,C1(CNC(C(CC#C)C2CC2)=O)(NC(c2nccnc2C)=O)CC2CCC1CC2 40370,C1(CNC(=O)CCNC(C2CC23CCC3)=O)CCCCN1C(c1csnc1Cl)=O 40371,n1(C(C)C)cccc1C(=O)NCC1CC(F)(CNC(C2(c3ncco3)CC2)=O)C1 40372,C(C(C)C(=O)NC1CC1NC(c1cc(C2(C)COC2)no1)=O)OCC 40373,N1(C(c2c(CN(C(=O)COCC(F)F)C)cc[nH]2)=O)CC(CO)C1(C)C 40374,C1(C#N)(C(=O)NC2CC(C)(NC(CCC=CCC=C)=O)C2)CC2CC2C1 40375,Cc1[nH][nH]c(=N)c1C(=O)NCCCCCCN(C)C(c1coc(C(F)(F)F)c1)=O 40376,C1(C(=O)NC2C(N(C)C(c3n[nH]cc3C3CC3)=O)CCCC2)CCC(C)(C)OC1 40377,CC1CN(C(=O)CN2CCC2)CCC1NC(=O)C(C)(C)C1(O)CCOC1 40378,C=CCCCC(C(=O)Nc1cccc(NC=O)c1)NC(=O)CCC(=O)CC 40379,n1(CC(=O)NC2C(NC(C(F)=CCC)=O)CC2)cc(Cl)c(C)n1 40380,N1(C(c2ccc(C)c(F)c2)=O)CCN(C(c2cncc(F)c2)=O)CC2(CC2)C1 40381,C(c1cnn(C)c1)=CC(=O)NC(CC=CC(=O)N(C1C(C)CCC1)C)(C)C 40382,C1(NC(CCC(C)OC)=O)CCCC12CN(C(=O)Cc1nc(C)sc1C)C2 40383,C1(C(N(C(CC)C)CCO)=O)COCCN(C(C2(C#N)CC2)=O)C1 40384,C(CCCCC(=O)N(CCO)CCN(C)C)NC(C1(N(C)C)CC1)=O 40385,CC1(C)CCC(C(C2CCSCC2)NC(=O)C(=O)NC2CC(C(=O)O)C2)OC1 40386,C#CC1(C(N2CC(OCCC(N3CC(C)(CCO)C3)=O)C2)=O)CC(=O)C1 40387,CCCC(C(O)C(=O)NC12CCCC1C2)NC(=O)CN(C)C(C)=O 40388,N1(C(C=C(C)C2CC2)=O)CC(C(=O)NCC(n2ccnn2)C)C(C)(C)C1 40389,C(=O)(CC(c1ccccc1)NC(N)=O)N(CCCNC(CC=C)=O)C1CC1 40390,N1(C(C2(CC=C)CC=CC2)=O)CC2(CCC2NC(=O)CSS(C)(=O)=O)C1 40391,C1(C(=O)OC)CN(C(=O)OC(C)(C)C)CC1C.C12CC(C)N1C2 40392,C1(CNC(C(N2C(=O)CCC2=O)CC)=O)CC(C)(C)CN1C(=O)CCOC1CC1 40393,C1(NC(CSCC=C)=O)CC(C)CN(C(c2c(C)coc2C2CC2)=O)C1 40394,C(CCCC(=O)NCC(c1ccco1)O)NC(c1cc(OC)n[nH]1)=O 40395,C(C(C)(C)CNC(c1ncn(C)n1)=O)N(C(C1(CCC=C)CC1)=O)C 40396,Cc1nc(Cc2ccccc2)ccc1C(=O)OCC1CCCC(C(=O)O)CC1 40397,N1(C(COCCCC)=O)CCC(C)(C)C(NC(=O)CCN(CC(F)(F)F)C)C1 40398,C1(CNC(C=NOC)=O)COC2(COCCN(C(=O)C(C)Br)C2)C1 40399,C1(CNC(c2ncn(CC)c2)=O)CC(C)N(C(C2CCC(=O)N2C)=O)C1 40400,Cc1ccccc1C(=O)NCC(C)CNC(=O)CCCc1cncs1 40401,C(C(CNC(=O)OC(C)(C)C)CO)NC(C1N(C(C2(OCC)CC2)=O)CC1)=O 40402,c1(N2CCN(CC(C)(F)F)CC2)nc(N2CCC(CC#N)CC2)nc2scnc12 40403,c1(OC(C)C)ccc2cc(C(=O)NC3CCN(C(=O)CC#N)C3(C)C)[nH]c2c1 40404,C1(NC(Cc2nc(=N)[nH][nH]2)=O)CCC2CCN(C(c3csc(Cl)c3)=O)C12 40405,c1(OC)cccnc1C(N1CCCCC1C1CCN(C(c2ccc[nH]2)=O)CC1)=O 40406,N1(C(Cc2c(C)con2)=O)CCC(C)(C)C(CNC(=O)Cn2cc(CO)nn2)C1 40407,C1(C2CCOCC2)(NC(CN(C(=O)C(COC)OC)CC)=O)CC1 40408,c1(C(N(C(c2ccccc2)CNC(C2CCNC2=O)=O)C)=O)cc(Cl)ncc1N 40409,C1(NC(c2cccnc2O)=O)C2CC3CN(C(C4C5CCCC45)=O)C1C3C2 40410,N1(C(c2c[nH]c(=N)s2)=O)CCC2(CNC(C3Cc4cccnc4C3)=O)CCCC12 40411,C1(C2CN(C(c3cc(Br)c[nH]3)=O)C2)(NC(c2cnn(CC)c2Cl)=O)CC1 40412,c1(C(=O)NC(CCOC)CNC(=O)CC(C)CF)ccc(S(N)(=O)=O)c(F)c1 40413,C(=O)(C1SCc2cccnc21)NCCCN(C(c1c(C)coc1C)=O)C 40414,N1(C(c2cc(CC)no2)=O)CC(NC(C2CC2c2ccccc2)=O)CC(F)(F)C1 40415,C12(C(N3CCN(C(c4ccc(C)c(C)c4)=O)C(C)C3)=O)CCCC1CC(=O)C2 40416,CC1(C)CCC(CNC(=O)C(C2CCCCC2)O)N(C(=O)CN2CCSCC2)C1 40417,c1(C(=O)NC2C(C)CN(C(c3ccoc3)=O)C2)cccc(C(N)=O)c1N 40418,N1(C(COCCCC#C)=O)CC2CCN(C(c3nnccc3C)=O)CC2C1 40419,N1(C(c2n[nH]c(C)c2O)=O)CCC(C(=O)NC(c2nncn2C)C)C12CC2 40420,C1(C(=O)NC(C2CCCCC2)CNC(c2csc(Cl)n2)=O)(OC)CS(=O)(=O)C1 40421,C1(C(=O)NCC2CCC(CNC(CNC(C)=O)=O)CC2)CCCCC1(F)F 40422,c1(CC(N2CCC(CN(c3snc(C(=O)OC)n3)C)C2)=O)cc(C#N)ccc1F 40423,C1(C(=O)NCCC(C)(C)F)C2CCN(C(c3cccc(O)n3)=O)CC12 40424,CCC(C)(CCC(C)C)C(=O)NC1CCC(C(N2CCC(O)C(O)C2)=O)CC1 40425,c1(-c2cc(C)[nH]c2C)csc(=Nc2cccc(F)n2)n1CCC1CCSC1 40426,C(c1cccc(Cl)c1)=C(C(=O)NC1(CC=C)CN(C(=O)C(C)OCCOC)C1)C 40427,C=CC1CN(C(C2(c3ccccc3Cl)CCOCC2)=O)CC1NC(=O)CCF 40428,C=CCC(CC(=O)N(CCC(F)(F)F)CC)NC(=O)C(COC)CC 40429,c1(NC2(c3nnnn3C(C)(C)C)CC(COC)C2)nc2cc(Cl)cnc2[nH]1 40430,C(=O)(C(C)(C)C1=CCN(C(C2CCCC2C)=O)C1)NC1CC(CC)C1 40431,N1(C(C2(OC)CC(C)C2)=O)CC(C2(NC(C3COCC(C)(C)O3)=O)CC2)C1 40432,c1(OC)ncc(C(=O)NCC2(O)CCN(C(c3n[nH]cc3C)=O)C2)c(C)n1 40433,c1(NC2CCN(C(C3CC34CC(O)C4)=O)C2)ncc2ccsc2n1 40434,C12(C(N(CC(C3CCCC3)O)C)=O)COCC1CN(C(=O)CCc1cscn1)C2 40435,C(=O)(CC(C)CC(C)C)NCC(CCC)C(=O)N1CCC1C(=O)OC 40436,c1(C(=O)NC2CC(N(C(=O)CNC(N)=O)C)C2)c(F)ccc2[nH]ccc12 40437,c1(CNC(c2n(CC)ccc2)=O)ccc(F)c(CC(=O)OC)c1 40438,N1(C(CCCCN(C)C)=O)CC2(CCCC2)C1C(N1CCC2(CC(F)C2)C1)=O 40439,Cc1cn2cc(CC(=O)NCC(C)CNC(=O)CC(C)CF)nc2s1 40440,c1(N(CC(C)O)C(C)CSc2ccccc2)nccc(NC(=O)OC(C)(C)C)n1 40441,n1(C(C)C(=O)NCC(=O)Nc2ccc[nH]2)cc(CCCNC(=O)C(F)(F)F)nn1 40442,C1(NC(CCc2c(C)noc2)=O)CC=C(C(=O)N2CCC(CF)C2)C1 40443,c1(C(=O)NC(c2ncc[nH]2)CC)ccc(CNC(=O)COc2ccsc2)s1 40444,CC1=C(C(=O)N2CCC(O)(C(C)NC(=O)C(C)NC=O)C2)CCO1 40445,Cc1ccc([N+](=O)[O-])cc1C(N1CCC(F)(F)C(NCc2cnn(C)c2C)C1)=O 40446,N1(S(C(C)C#N)(=O)=O)CCC2(COCCN2C(C2CC2(F)Cl)=O)C1 40447,C1(C(=O)NCC2CCCC(CC)C2)C2CCC(C2)C1NC(C1(Cl)CCC1)=O 40448,c1(CC)sc(C(N2CCC(C(C)NC(c3cc[nH]c(=N)n3)=O)C2)=O)cc1C 40449,C(CCCC(=O)N1CC(C(=O)NC2CC(C(F)F)C2)OC(C)C1)(OC)OC 40450,CCCCC(CC)C(=O)N1CC(C(=O)NCCN2CCC2)CC1(C)C 40451,C1(C(=O)NCC(CNC(c2ccn(CCCC)n2)=O)(C)C)C2CCC(=O)C12 40452,c1(C(=O)NCCC(C)N(C(C(C)c2ccon2)=O)C)cnc2[nH]nnc2c1 40453,N1(C(c2cc3nnn(C)c3s2)=O)CCC2CCC(C1)N2C(=O)CNC(=O)C1CC1 40454,c1(NC(c2cncc(CC)c2)=O)ccc(NC(c2cnc(O)cc2C)=O)c(C)c1 40455,CC1(NC(c2ccc(F)cn2)=O)CCN(C(=O)C=CBr)C1 40456,Cc1occc1C(=O)NC(C1CCCN1C(c1cc(C(F)F)on1)=O)(C)C 40457,C#Cc1cncc(C(=O)N(CC(C)(C)CNC(=O)Cc2ccc(Br)cc2)CC)c1 40458,c1(C(=O)NCc2cc(OC)nn2C)[nH]c(C)c(C(N2CCN(CC)CC2)=O)c1C 40459,C(=O)(C(Cc1ccco1)NC(=O)CC1CNC(=O)O1)N(CCCC)CCCO 40460,Cc1c(C(=O)NCC(c2ccccc2)N(C(=O)CSC(C)C)C)nc2sccn12 40461,C1(C(=O)OCC)OCCNCC1N(c1c(CO)cccc1C)C(C1(C)COC1)=O 40462,CCC(CC(=O)NC1CCC(C)(NC(c2cnn(C)c(=O)c2)=O)CC1)CC(C)C 40463,c1(C2(C(=O)NCC(C3CCC3)NC(c3c(C)cco3)=O)CC2)ccc(F)c(Cl)c1 40464,CCCCC(CC)C(=O)NC1CC(C)(C(=O)NCCn2cc(CO)nn2)C1 40465,C(=O)(C1=CC2(CN(C(=O)C(O)CN3CCCC3)C2)OC1)NCC(COC)(C)CO 40466,c1(C(N2CC(C)NC(=O)C2)=O)ccc2c(n1)CCN(C(=O)Cc1ccccc1)C2 40467,CCCCCC(C(=O)NC1CCC(NC(=O)Cc2cn(C)nc2Cl)CC1)C(C)C 40468,c1(C(=O)NCC(CNC(COC)=O)C)oc2ccccc2c1CSC 40469,c1(CNC(C2(NC(CCC=CC(C)C)=O)CC2C)=O)ccc(F)c(F)c1 40470,C1(C(N(C2CCN(C(=O)C(C)(C)O)CC2)CC)=O)C2CCC1(c1ccccc1)C2 40471,N1(C(CN(C)CC)=O)CCCC1(C)Cn1cc(C2CCC(CO)CC2)nn1 40472,C1(C(N2CC(CNC(c3cncc(C)n3)=O)OCC2)=O)CCCCC1(C)C 40473,C(C(F)(F)C(N)=O)NC(C1(CCC=C)CN(C(=O)CN2CCC(C)C2)C1)=O 40474,Nc1cc2c(cc1C(=O)NC1CCC(NC(C3CC3(Cl)Cl)=O)CC1)CCC2 40475,C(=O)(CCCC(F)(F)CO)N1CC(C(C)NC(C23CCC(CC2)CC3)=O)C1 40476,C1(F)(CNC(C(SC)SC)=O)CCN(C(=O)C(=Cc2cn(C)cn2)F)CC1 40477,c1(CC)ccc(NC(=O)C(C2CCN(C)CC2)C)cc1S(C)(=O)=O 40478,Cc1nc(C=CC(=O)N(C2CCC(NC(=O)Cc3ccco3)C2)C)cs1 40479,c1(SC)ccc(NC(=O)NCCOc2cccc(F)n2)cc1C#N 40480,N1(C(c2ccn(CCC)n2)=O)CCC(C)(C)C1CNC(=O)C(C)(CC)CO 40481,c1(C2(COC(CN(C(CC)(C)C)C3CC3)=O)CCC2)ccc(Cl)c(Cl)c1 40482,c1(C(N2CC(C(=O)Nc3ccc(O)nc3)OCC2)=O)cn2ccc(Cl)cc2n1 40483,c1(OC)cc([N+](=O)[O-])c(NC(C2CCCCN2C(=O)C=CCBr)=O)cc1F 40484,C1(O)(C(N(C)CC2CN(c3cc(CC)ncn3)C2)=O)CC2CCC1C2 40485,N1(C(CCC)=O)CCCN(C(c2cc(C)n(C3CCCOC3)c2C)=O)CC1CO 40486,C(=O)(CCCCc1ccc(Cl)cc1)NCC(CNC(Cc1cc(C)sc1)=O)O 40487,C(C)(CN1CCOCC1)(C(C)C)N(c1cccc(C(C)C)c1)CC(C)C.CCO 40488,C1(NC(CSCC(=O)OC)=O)CCN(C(c2cnn(CC(F)(F)F)c2)=O)CC1C 40489,Cc1cc(N2Cc3ncsc3C2)nc(=NCCCc2nncn2C)[nH]1 40490,N1(C(c2c(C)nco2)=O)CCC2(CC(NC(=O)C(F)(F)c3ccnn3C)CO2)C1 40491,c1(C2CN(C(=O)OC(C)(C)C)C2)nnc(S)n1C.N12CCC1(C)C2=O 40492,C#CCCCCC(=O)N1CCCC(C)(CNC(=O)C(CCC)OC)C1 40493,C1(C(N2C(C#C)CCC2)=O)CN(C(=O)Cc2cnnn2C)CCC1(C)C 40494,N1(C(c2cc(OC)no2)=O)CC2CC(NC(=O)CC3CC(=O)NC3=O)CC1C2 40495,Cc1cc(F)c(C(N2CCC(C)(CNC(=O)C=Cc3cncs3)C2)=O)c(F)c1 40496,Cc1cc(C(c2ccc(C(=O)NC3(C)CCCCC3)cc2)N(C)C)cnc1C 40497,CC1CN(C(c2ccncc2F)=O)CC1CC(=O)NCCCCC1CC1C 40498,CC1CC(C(N2CC3(CC(CNC(c4ccc(=O)n(C)c4)=O)C3)C2)=O)CC(C)C1 40499,N1(C(C(c2cccc(F)c2)C)=O)CCC(C2(NC(c3cc(Cl)n(C)n3)=O)CC2)C1 40500,C1(NC(C(C)OC)=O)CCC(NC(c2cnn(C)c2C)=O)CC1 40501,c1(C(=O)NC(CC(C)NC(CCN(C)CC)=O)C)cccc(Cl)c1C 40502,N(C)(S(=O)(=O)N(C)C)CC(=O)NC(C)CNC(c1cn(C2CCCC2)nn1)=O 40503,C1(C(=O)NCC2(OC)CN(C(c3cocc3C(N)=O)=O)C2)CCC(C)(C(C)C)C1 40504,C=C(C)CC(C(=O)NCC(O)C(=O)NC(C)CCCCCO)OC 40505,C1(C#N)(C=O)C(C#N)C1(C)C.Cn1cc(C#N)cc1.N12CC3CC1CN23 40506,N1(C(C(CCC2CC2)NC(C(CC(C)C)N(C)C)=O)=O)CCOC(C)(C)C1C 40507,c1(OC(C(=O)N(CC(CNC(C2N(C(C)=O)CSC2)=O)O)C)C)ccc(C)cc1 40508,N1(C(c2c(CC)n(CC)nc2)=O)CCCN(C(C2CCOC2=O)=O)C(C)C1 40509,c1(C(N2CCN(C(COC3(C)CCC3)=O)CC2C2CC2)=O)cc(F)c(N)cc1F 40510,c1(OC)cc(NC(c2cccc(N3CCNC(=O)C3)c2)=O)ccc1O 40511,N1(C(c2c(CC)cccn2)=O)CCCC12CCN(C(C1CC=CCC1)=O)C2 40512,c1(CC(=O)N(CCC2N(C(C(C(C)C)OC)=O)CCCC2)C)cc(F)ccc1Cl 40513,c1(C(=O)NCC(CC)NC(=O)C(C)(C)C(N)=O)ccc([N+](=O)[O-])cc1 40514,N1(C(c2c(COC)cc[nH]2)=O)CC(CNC(=O)C=C2CCN(C)C2)CC1(C)C 40515,Cc1nc(C(=O)NC2(CNC(C3(C)CC=CCO3)=O)CC2)ccc1C#N 40516,Cc1occ(C(F)(F)F)c1C(=O)NC1CN(C(=O)C(c2ccccc2)F)CC1O 40517,CCCC(C(=O)N1CCC1Cn1cc(-c2cnn(C(C)C)c2)nn1)OC 40518,C1(CSc2nnc(N(c3ccccc3)C)s2)CCOC(c2cccc(F)c2)C1 40519,C(=O)(C=CCNC(=O)COC(C)=O)N(CC=C)CCO 40520,N1(CC2(O)CCN(c3c(OC)cccn3)CC2)CCC2(CCCC2)C1 40521,C1(C(N(C(C)CNC(=O)C2CC2)C)=O)(NC(=O)OC(C)(C)C)CC=CC1 40522,c1(CC(=O)NC(CC)CNC(C23CCC2C3)=O)nnn(-c2cccc(Cl)c2)c1C 40523,C1(C(N(C2CCCN(C(CC3CC(=C)C3)=O)CC2)C)=O)CNC(=O)CC1(C)C 40524,N1(C(c2c(C)cns2)=O)CCOCCC1C(=O)NCCc1cncs1 40525,C1(C2CCN(C(C3CCC(C)S3)=O)CC2)(NC(c2n(CCC)ccc2)=O)CCC1 40526,C(=O)(C(C)(C)CCF)N1CCCC(N2CCN(C(CC=C(C)C)=O)CC2)C1 40527,c1(C(=O)NC(C(C(C)C)C)CNC(c2cccnc2S)=O)noc2c1CCCC2 40528,CC1(C)CCC(C(N2CC=CC2CNC(c2ccon2)=O)=O)C1 40529,N1(C(=O)C=Cc2cccs2)CCC(C2CCN(C(C3(F)CCCCC3)=O)CC2)C1 40530,C1(NC(c2cc(CCC)on2)=O)CCCN(C(=O)C=C(CC)CC)C1C 40531,C1(O)(CNC(C(C)N2CCC2)=O)CCN(C(c2ccc(C#N)cc2)=O)CC1 40532,c1(C(N2CC(CNC(CCC3CC(C)C3)=O)OCC2)=O)ccc(F)c(Cl)c1N 40533,Cc1c(Br)csc1C(N1CC(CC(C)NC(=O)C(C)C2CCC2)C1)=O 40534,C(C(=O)N1CC(O)C(O)CO1)C1N(C(c2ncc(CC)cn2)=O)CCC1(C)C 40535,C1(C(=O)NC2C(OC)CN(C(C3(C4CCC4)CC3)=O)C2)CCC(C)(O)CC1 40536,C1(CNC(C2CCCC(NC(CC(C)F)=O)C2)=O)CC12CCOCC2 40537,C1(C)(CCC(=O)NC(CC)CN(C(=O)COC2CCC2)C)CCC(=O)N1 40538,C(=O)(C(C)CC(C)(C)C)N1CCC(N(C(Cn2ncc(CC)c2)=O)C)C1 40539,c1(NCC2(CC)CCCCO2)ncc(S(=O)(=O)NC2CC(CF)C2)cc1Cl 40540,CCCCCCC(C)C(=O)N1CCCC1C(C1CC1)NC(C1CCCCN1N=O)=O 40541,N1(CC(N2CC(NC(=O)CSc3ccncc3)C2)=O)CCCCCCC1=O 40542,C(=O)(C1=CCOCC1)NC1(CO)CN(C(c2c(C(C)C)n(C)nc2)=O)C1 40543,Cc1cc(NC(=O)C(=O)NCCc2ccc(Br)s2)ncn1 40544,C(c1ccncn1)=CC(=O)NC(C(=O)NCC(=O)NC1CC1)C1CCCO1 40545,Cc1cccc([N+](=O)[O-])c1C(N1CC(N(C(=O)CC2OCCC2C)C)C1)=O 40546,c1(CC(=O)NCC(C)(CO)NC(C2CCN(C)C2=O)=O)c[nH]c2cccc(Cl)c12 40547,C(=O)(CS(=O)C(F)(F)F)NC1C(CO)CCN(C(C(C)N(C(C)=O)C)=O)C1 40548,CC1CCc2ncc(C(N3CCC(NC(c4cnc(C(C)(F)F)s4)=O)C3)=O)n2C1 40549,N1(C(C23CCC(OC)C2C3)=O)CCCN(C(c2cccc3c[nH]nc23)=O)C(C)C1 40550,N1(C(C2CC(N(C)C)C2)=O)CCC(C)(CNC(C2CC3C=CC2C3)=O)CC1 40551,N1(C(c2oc(C)c(CO)c2)=O)CCN(C(C2CCC(=O)N2C)=O)CC1CF 40552,N1(C(c2cc(C)c(C)s2)C(=O)NCCCSC)CC(C2CC2)OC(C)C1 40553,N1(C(c2c(N)nccc2)=O)CCC=C(CNC(=O)CCN2CCCC2)C1 40554,CCCCC(C)C(=O)N1CC(C(=O)N(CC)CC2CCOC2)C(F)C1 40555,c1(C(N2CC(C#N)OCC2)=O)cc(-c2cccc(OC(F)F)c2)c2[nH]ccc2c1 40556,C[S+](C)CCC(O)C(=O)N1CC(O)(CCNC(=O)COCC2CCOC2)C1 40557,c1(C(=O)NC(CNC(=O)CN2CSCC2=O)C2CC2)cc(C2CC2)nc(O)c1 40558,c1(C(C(=O)NC)N(C2CCC(F)(F)CC2)C)ccc2c(c1F)CCC2 40559,c1(C(=O)NCC(CNC(C(CC)(C)OC)=O)CO)ccnc2ncccc12 40560,c1(C(N2CCC(CNC(C(C(=C)C)(C)O)=O)CC2)=O)ccc2c(C)nn(C)c2n1 40561,N1(C(c2c(CC)ncs2)=O)CC2CN(C(c3cnc(C(C)(C)C)o3)=O)CC(C1)O2 40562,c1(N2CCN(CC)CC2)cc(C)c(S(=O)(=O)NC(C)C(C)NC(=O)OCC)cn1 40563,C12(C(=O)NC3C(C)NC(=O)CC3)CCN(C(=O)CCC(C)(C)F)CCC1C2 40564,Cc1ccc(CN2CCCC2CCC(=O)Nc2ccnc(OC(C)C)c2)cn1 40565,c1(C(N2CCC3CCN(C(CC=C)=O)C3C2)=O)cnc2c(c1)OCC(=O)N2 40566,N1(C(Cc2c(C)nc[nH]2)=O)C(C)C2CC1C2NC(c1cccnc1O)=O 40567,N1(C(COCC#C)=O)CCC(NC(=O)CCc2cccs2)C1C1CC1 40568,c1(OC)cc(N)ccc1C(=O)NC1CCCC1CNC(=O)CN1CCCS1(=O)=O 40569,C1(C(=O)OC)(Nc2c(CS(=O)(=O)N(CCCC)C)cccc2)CCC(C)(C)C1 40570,C(N=c1ccc(CC(F)F)c[nH]1)N(C(C)C)CCN 40571,c1(C(N(C(C)CNC(=O)C(C)(C)COC2CC2)C)=O)cccc2nsnc12 40572,c1(NC(C2N(Cc3ccn(CC)n3)CC(O)C2)=O)cc(F)c(C)c(F)c1 40573,c1(C(=O)NCC(CN(C(c2c(COC)ccs2)=O)C)C)cc(S(N)(=O)=O)ccn1 40574,N#Cc1cc(C(=O)NCC2CC2NC(c2c(Cl)ccc(F)c2F)=O)c(N)nc1O 40575,C1(NC(C2CC(C)(C)OCC2)=O)CCC2CCN(C(C3(F)CCOC3)=O)C1C2 40576,c1(NC(c2cc(-c3ccc(C)o3)[nH]n2)=O)nccnc1C(=O)Nc1ccccc1 40577,CC1CCCCC1(CNC(c1ccc(O)c(O)c1)=O)NC(c1c[nH]ccc1=O)=O 40578,Cc1cccc([N+](=O)[O-])c1C(=O)NC1CC2CC(C1)N(C(=O)Cc1cccs1)C2 40579,C1(CNC(c2scc(C)c2)=O)CC(NC(c2coc(N(C)C)n2)=O)C12CCC2 40580,C(=O)(C(O)CCN(C)C)N(CCC(=O)NC1COCC1n1ccnn1)C(C)C 40581,C1(CNC(c2c(CC)cncc2)=O)N(C(=O)CCNS(C)(=O)=O)CCCC1(C)C 40582,C(=O)(CCCNC(=O)C(C)Cn1ccnc1)N(CCC(=O)OC)CC=C 40583,c1(CC)nc(C)[nH]c1C(=O)NC1CC(CCNC(=O)Cc2[nH]cnc2C)C1 40584,CC1(CNC(C2CC2F)=O)CCCN(C(=O)Cc2c(Cl)cccc2Cl)C1 40585,c1(C(CC)NC(=O)COC2CN(C(=O)C(C)C3CCCC3)C2)ccc(Cl)s1 40586,C1(C(C)C)N(C(c2cncn2C)=O)CC12CCN(C(C1CC1F)=O)CC2 40587,N1(C(c2c(Cl)nc(OC)s2)C(=O)NCC(F)F)CCCCNC(=O)C(F)(F)C1 40588,CC(C)(C)C(CC(=O)NCC1CCN(C(=O)CN2CSCCSC2)C1)C(F)F 40589,c1(C(=O)NC2(COC)CN(C(C3CC3c3ccccc3)=O)C2)ccc(CF)cc1 40590,CN1CCOCC1C(=O)NCC1(C(N2CC=CC2CF)=O)CC1 40591,Cc1c(C(=O)NC(C)CNC(=O)CCc2ccon2)ccn1C 40592,c1(CSC(C)(C)C)cc([N+](=O)[O-])ccc1C(=O)Nc1nc(=N)[nH][nH]1 40593,C(=O)(C1=NOC2(CCN(C(C3(CN)CC3)=O)C2)C1)Nc1cnc(C)c(Cl)c1Cl 40594,N12CCC3(CCCCN(C3)C(=O)c3coc(n3)SCCC1=O)C2.CCSC.COC 40595,C12(CNC(C=CCC)=O)CCCC(CN(C(c3cccc4nsnc34)=O)C1)C2 40596,Cc1cc(C(=O)OCC(c2c[nH]nc2C)=O)no1 40597,c1(N2CC(NC(C3C(C)(Br)C3)=O)(CO)C2)ncncc1Br 40598,N1(C(C2C(C)(C)CC2)=O)CCCCC1C1CCN(C(c2cc(Br)no2)=O)CC1 40599,N1(C(CC(C)OC)=O)CCCC(CN(C)C(c2sc(NC3CC3)nc2C)=O)C1 40600,N1(C(C(C2CCN(C(=O)C(N3CCOCC3)C)C2)C)=O)CCC(O)C(C)C1 40601,C1(C(N2CCC(OC)C2(C)C)=O)CC2C=CC1N(C(=O)C(C)n1ccnn1)C2 40602,Cc1sc(C)c(C(N2CC3(CC(NC(=O)C(C)CC(N)=O)CO3)C2)=O)c1C#N 40603,C1(C(N2CC(F)(C(=O)NC3CN(C4CCC4)C3)C2)=O)CC2CCC2C1 40604,CC(c1ccccc1)=CC(=O)NCC1CCC1NC(C1(CCN(C)C)CC1)=O 40605,N1(C(C(C)CC(F)(F)F)=O)CCCC2(NC(=O)CN3CCC3)CCCC12 40606,C1(CC(=O)NCC(C(C)C)(C)C)C2CCC(C2)N1C(=O)CCCn1cncn1 40607,c1(C(N2C(CNC(COC3(C)CCC3)=O)CC2)=O)ccc(Cl)cc1Br 40608,N1(C(COCC#C)=O)CCN(C)CC1CNC(=O)CSc1n[nH]c(C)n1 40609,c1(C(C(=O)NC2CC(O)(Cn3cc(-c4cccnc4)nn3)C2)O)ccc(O)cc1 40610,N1(C(C=C(C)C)=O)CCC2(NC(=O)COc3cccc(C)c3)CCCC12 40611,Cc1ccsc1C(=O)N(CCC(=O)NC(C)(C)CO)C 40612,C(=O)(CCCS(=O)(=O)N1CCCC1)NC(CN(C(COCCC#C)=O)C)C 40613,c1(OC)cccc(Cl)c1C(=O)NC1CCN(C(C2(CCF)CC2)=O)C(C)C1 40614,c1(C(=O)NCC(CNC(CNC(=O)OCC=C)=O)C)ccnc(O)c1 40615,N1(C(CC(C)C)=O)CC2CCCC1CN(C(=O)Cc1ccc3nc(O)[nH]c3c1)C2 40616,C(=O)(CCCC(C)(C)C)NCc1cn(CC(=O)NC(CC(C)C)C(N)=O)nn1 40617,N1(C(C(C)S(N)(=O)=O)=O)CCC2(CCCC2NC(c2cc(Cl)cn2C)=O)CC1 40618,C(CCCC(=O)NCC1(O)CN(C(c2cn(C(C)(C)C)nc2C)=O)C1)NC(C)=O 40619,N1(C(c2ncc(NC)nc2)=O)CCC(C(=O)N(C)CC2CCN(C)C2)=C(F)C1 40620,O=C(C1=CC2CCCC12)NCC1CC(NC(c2ncnc(O)c2Br)=O)C1 40621,CCC(C)C(O)C(=O)NCC(CO)NC(c1ccc(F)c(C(F)(F)F)c1)=O 40622,CCC(C)(CO)C(=O)NCC1(CNC(=O)CCn2ccc(C)n2)CC1 40623,C#CC1(C(=O)NCCN2CCOC(C)C2)CCN(C(=O)CC2CSC2)CC1 40624,c1(C(=O)NCC2CC(NC(c3c(OC)nn(C)c3)=O)C2)ccc(F)c(Cl)c1 40625,c1(C(N2CC(CNC(c3ccco3)=O)C(C(F)(F)F)C2)=O)cnc(F)c(F)c1 40626,Cc1[nH][nH]c(=N)c1C(=O)NCC1(O)CCN(C(=O)CCC2CNC(=O)N2)C1 40627,C1(CCNC(=O)CNC(c2cccs2)=O)CCN(C(C2CCO2)=O)CC1(F)F 40628,c1(C2C(C)N(C(c3ccccc3)=O)CCC2)ncnc2c1ncn2CC(O)CO 40629,c1(C(N(C2CCCN(C(CC(C)F)=O)C2)C)=O)ccc2oc(S)nc2c1 40630,C1(C(=O)NCCN(C)CC)CCCN(C(=O)CC2(OC)CCC2)C1C 40631,C1(CN(C(CCCNC(C2CCC(C(=O)OC)C2)=O)=O)C)CCCC2CC12 40632,N1(C(CS(CCC)(=O)=O)=O)CCC2(CCOCC2)C(NC(c2ccon2)=O)C1 40633,N1(C(CC=C=C)=O)CCC(NC(c2ccn(-c3ccccc3)n2)=O)C1C(C)C 40634,c1(C(=O)NN2CC(C)(C(=O)Nc3cc(C(C)C)no3)C2)cc(N(C)C)ccc1F 40635,c1(CC)cc(C(=O)NCC(C)CN(C(=O)COCC2CC2)C)oc1CSC 40636,c1(C(=O)NCC(CC)NC(c2cnn(CCO)c2C)=O)cccc(F)c1OC 40637,C(=O)(C1=CC2CCC(C1)C2)NC1CC(NC(CSCC)=O)CC1O 40638,C1(NC(=O)CS(=O)(=O)NC2CC2)CN(C(=O)C=CBr)CC2(CC2)C1 40639,N12CC3(CC3)CC1C2=O.c1(CNC(c2c(C)ocn2)=O)cc(CO)n(C)n1 40640,C=C(F)C1(CC(=O)NCCC2CCC(NC(c3ncn(C)c3C)=O)C2)CCC1 40641,c1(NC(N(CC(C(C)C)OC)C)=O)c2c(c(Br)c3c1CCC3)CCC2 40642,O=C(N=c1[nH]ccc2cc(Cl)ccc12)C1CCN(Cc2c(Cl)cc(F)cc2Cl)C1 40643,C(=O)(C1=C(C)CCOC1)NC(CC#C)CC(=O)NCC(O)C1CC1 40644,C1(C(=O)NCC2C(=O)CC2)CCCN1NC(=O)c1cn2c(n1)CCC2 40645,N1(C(c2ccc(OCC)nc2)=O)CCN(C(=O)CCF)C2CCCCC2C1 40646,c1(C(N2CCCC(N(C(C3CC=C(C)CC3)=O)CCF)C2)=O)cc2n(n1)CCC2 40647,c1(-c2ccc(Cn3ncc(-c4ccc(C)cc4)c3)nn2)cccc(F)c1O 40648,C12(CNC(C(CC#C)O)=O)CCC(C1)N(C(=O)CNC(c1ccncc1)=O)C2 40649,C1(OC)CN(C(=O)CCN(CC(F)(F)F)C)CC1NC(=O)Cc1cccn1C 40650,Cc1ncnc(C)c1CC(=O)NCC(O)CNC(C1(C)COC1)=O 40651,CC1CCN(C(C2CC(=O)NC(=O)C2)=O)CCN1C(=O)C=CC=C(Cl)Cl 40652,C1(C)(CC)CCN(C(=O)CC2(NC(=O)COC)CCC2)CC1 40653,C1(C(=O)NCC2COCCN2C(=O)Cc2ncc(Cl)s2)CC2CCC(C1)C2 40654,C1(CNC(c2c(C)c[nH]n2)=O)CN(C(c2ccc(F)cn2)=O)CC1C(F)(F)F 40655,Cc1cnnc(O)c1C(=O)NC1CC(CNC(=O)C(N2CCOCC2)C)C1 40656,C#CC1CC2(CC2)CN1C(C1CCN(C(C2CCCCC2OC)=O)CC1(C)C)=O 40657,c1(CC(=O)NCCC(=C)CNC(=O)CCCc2ccsc2)nn(C)cc1Br 40658,C(=O)(C(Cc1cnc[nH]1)NC(=O)COC1CC=CC1)N(C(C(C)SC)C)C 40659,c1(OC)cccc2c1OCCC2NC(c1c(Br)ccc(C(F)(F)F)c1F)=O 40660,N1(C(=O)C(c2ccccc2)Oc2ccc(F)cc2)CCC(O)C(O)CC1 40661,N1(C(c2nc(OC)oc2)=O)CC2=C(C1)CN(C(=O)CC1COCC3(CCC3)O1)C2 40662,C(=O)(C1CC(C)(C)Oc2ccccc21)N(CCCCNC(C1CC1(C)C(F)F)=O)C 40663,C1(C(=O)NCCCc2nccs2)CCN(C(=O)C=CC2CCOCC2)CC1 40664,c1(C(=O)NCC2N(C(C(C)S(N)(=O)=O)=O)CC3(CC3)C2)coc2ccc(O)cc12 40665,N1(C(=O)C=C2CCC2)CCCC(C2CCCN2C2CC2c2ccccc2Cl)C1 40666,N1(C(C=C(C)CNC(c2nn(C)cc2Cl)=O)=O)CC(C)CCC(C)C1 40667,CN1CC2(CCN(C(NC3CCCc4ccoc43)=O)CC2)c2ccccc21 40668,N1(C(C2C(C(=O)OC)C=C2)=O)C(C(=O)NCc2cnn(C)c2OC)CC2CC12 40669,c1(C(=O)OC)cc(C)ccc1Cn1cc(-c2cncnc2NC2CC2)nn1 40670,c1(NC2(CCNC(C3(C)CC(C)OCC3)=O)CCC2)ncc2c(ncn2C)n1 40671,C1(CC(=O)NC)SC(=Nc2ccccc2CO)N(Cc2cc(Br)ccc2Cl)C1=O 40672,N1(C(c2cn(C(C)C)nc2)=O)CCC(C)(CNC(c2[nH]nnc2C2CC2)=O)CC1 40673,CC1(NC(C2C(N(CC(F)(F)F)CC(=O)NCC(F)(F)F)COC2)=O)CCOCC1 40674,c1(C(N(CCCCCCNC(C(C)=C(C)C)=O)C)=O)cc(=O)n(C)cc1Br 40675,CCC(CC(=O)N(C(C)C(=O)NC1(CCO)CCCCC1)CC)OC 40676,C1(C(=O)NC(C)CCNC(c2cc(Cl)c(N)cc2F)=O)CCc2nc(O)[nH]c2C1 40677,C1(CC(=O)NCC(CNC(CCOCC#C)=O)(C)C)CCC(=O)N1CC 40678,C(C)(C)(C(=O)N1CCCCO1)C1CCN(C(c2ccn(CCC)n2)=O)C1 40679,Cc1ccsc1CC(N1CCC(CNC(c2cnc(-c3ccccc3)o2)=O)C1)=O 40680,C=CCC(C)(C)CC(=O)NCC(O)CCNC(C1(CC)CC1)=O 40681,c1(CCCC)nc(C)c(CC(=O)NC2(COC)CN(C(c3nccn3C)=O)C2)s1 40682,N1(C(C2C3COCC23)=O)CCC2(CCCN2C(=O)C2=CCCC2)C1 40683,c1(NC(C2N(c3ncc(C)c(C)n3)CC(O)C2)=O)cc(F)c(C#N)cc1F 40684,N1(C(C2C(CC)CCCN2C(=O)OC(C)(C)C)=O)CC2CCC1CN2C(=O)CC 40685,C1(C(N2C(CCNC(C(C)(Cl)Cl)=O)CCCC2)=O)CCC2CCC1O2 40686,CCC(O)C(C)(C)C(=O)N1CC2CCCC2(NC(c2ccoc2C2CC2)=O)C1 40687,C(=O)(CCC(F)(F)Cn1cc(CC(O)COC)nn1)N1CCCC(CC)(OC)C1 40688,N1(C(c2c(OC)cncc2)=O)CCC(C)(C)C1C(=O)NCCCSCCO 40689,c1(OC)cc(Cl)c(C(N2CCCN(Cc3nc(C4CC4)no3)CC2)C)cc1OC 40690,c1(NC(c2n(CCOCC)nnn2)CCOc2ccccc2)ccc(Cl)cc1 40691,C1(NC(C(c2ccco2)OC)=O)CCC(C)(C)C1.n12cnc(c1)C(=O)NCC2 40692,C(=O)(C=C1SCC(=O)N1C)N1C2CC(NC(C(COC)(F)F)=O)CC1CC2 40693,CCC(C)(C)C(=O)NCc1nc(C(=O)Nc2ccc(C(N)=O)cc2)c(C)o1 40694,c1(OC)ccc(CC(=O)NC2C3CN(C(=O)C(F)=CC4CC4)CC23)cc1 40695,C1(CNC(CC2ON=C(C)C2)=O)CC12CCN(C(c1cnc(N)c(N)c1)=O)CC2 40696,Cn1nnc(C(=O)NCc2csc(-c3ccco3)n2)n1 40697,C1(C(=O)NC(COC)C(N2CC(C(N)=O)C3(CC3)C2)=O)Cc2nccn2C1 40698,n1(CC)c(C(=O)NCCC(F)Cn2cc(C3(C)CCCC3O)nn2)cnc1O 40699,c1(C(=O)NC2C(SC)CN(C(C3ON=C(C)C3C)=O)C2)cnc2c(c1)nnn2C 40700,N1(C(C(CC=C)CNC(=O)CNC(C)=O)=O)CC(C)CCCC1C 40701,c1(C(=O)NCC2N(Cc3ccc(OC)nc3Br)CCC2)cccc2cn(C)nc12 40702,C1(CC=C)(NC(=O)Cc2ccsc2)CCN(C(=O)C(C)(C)COC(C)C)C1 40703,S(=O)(=O)(c1ccc(=NCc2cnn(C(C)(C)C)c2)[nH]c1)N(C1C(C)CCCC1)C 40704,c1(OC)ccc(COCCCC(=O)NC2(C)CN(C(=O)C3CC3)C2)cc1 40705,CC1(OC(C2CCOCO2)=O)CN(C)C1.C(C)(C)(C)O 40706,C(C1CCCN1C(=O)CC1(c2ccon2)CC1)=CC(=O)NCCN1CC=CCC1 40707,c1(OC(C)C)ccc(F)cc1C(=O)NCC1CCC1NC(C1(O)COC1)=O 40708,C#Cc1cncc(C(=O)NC2CCCCC2CNC(=O)C(F)C(C)(F)F)c1 40709,C1(C(N2C(COC)CCCC2)=O)CN(C(=O)C(C)c2cc[nH]n2)CC1(C)C 40710,c1(C(N2C(C(=O)NCCNC(=O)OC)COCC2)=O)cc(C)c(F)cn1 40711,CN1CC(F)CC1C(=O)NC12CC1CN(C(c1cccc(CCO)c1)=O)C2 40712,N1(C(CC(CC)C)=O)CCCCCC(NC(C2OCCC2(C)C)=O)C1 40713,c1(C(=O)NC2CCN(C(c3c(C)nn[nH]3)=O)CC2C)cc2c(s1)CCSC2 40714,Cc1cc(F)c(Cl)cc1C(=O)NCC(F)CNC(=O)CC(O)C(C)C 40715,C1(NC(COC(CC)CC)=O)C2CCC1CN(C(c1cc(O)n(C)n1)=O)C2 40716,C(=O)(CC1=CCCCC1)NCC1CCCN(C(CCCOC(C)=O)=O)C1 40717,c1(CCC(=O)NCC(C)NC(c2n(CC(C)C)ncc2)=O)ccc(Cl)c(Cl)c1 40718,CCC(C(C)O)NC(C1(CNC(c2c[nH]nc2C(C)C)=O)CCC1)=O 40719,C1(CNCC2CCN(C(C)=O)C2)CCCCC12CCN(c1cc(=O)n(C)cn1)C2 40720,c1(C(C)C)cc(C(=O)N(C(C)C(=O)N(CC(O)CO)CCO)C2CC2)n[nH]1 40721,C=CCC(CC(=O)N1CCCC(N(C)C)CC1)NC(c1ccc(C)c(C)c1)=O 40722,C(CCN(C)C(C1CCC(O)CN1C)=O)(C(C)(C)C)NC(C(CSC)OC)=O 40723,c1(C(N2CC(NC(c3ccc(C)cn3)=O)C3C2C3)=O)cnc(C2CC2)nc1C 40724,CC(C)CC(C)(C)C(=O)NC1CCOCC1NC(C1CN(CC(F)(F)F)C1)=O 40725,Cc1nn(C)c(C)c1CNC(=O)C(C(C)O)NC(=O)OC(C)(C)C 40726,C(=O)(C1=Cc2ccccc2OC1)NCC(CN(C)C(C1CCCC1(C)C)=O)(C)C 40727,c1(C(N2CC(C)(NC(=O)CC3CCCO3)C2)=O)cccc(Cl)c1Cl 40728,C(C)(C)(C(C)NC(=O)C(C)=C(C)C)NC(C1(CCOC)CCC1)=O 40729,C(=O)(C(C)C(O)C(C)C)N1CCC(C(C)NC(C(Br)=C(C)C)=O)CC1 40730,C1(CC(=O)NCC(C)N(C)C(c2csc(C3CCCCC3)n2)=O)CC=CCC1 40731,C1(C)(CC(N2CC(O)(CC=C)C2)=O)CCN(C(=O)CNC(=O)NC)C1 40732,c1(C(N(CCCCCNC(CC(CCC)C)=O)C)=O)ccc(=O)n2c1COCC2 40733,c1(C(=O)NCC2CCN(C(=O)Cc3ccnc(Br)c3)C2)cc2n(n1)CCO2 40734,CCC(CCC(=O)N(CCOCCCO)CC)NC(=O)CCCC(=O)NC 40735,C(=O)(C(C)(F)C(C)(C)F)NCCCC1(NC(CCc2cccc(OC)c2)=O)CC1 40736,C1(NC(C(CSC)C)=O)CC2CCC1N2C(=O)Cn1nc(O)ccc1=O 40737,c1(C(=O)NCC(COC)(C)OC)cc2c(cc1O)CCCC2 40738,C1(CC2CCC2)C(=O)OCCOCC(=O)N1.C(C)(CC)(C1CC1)NCC 40739,N1(C(Cc2ccc(CC)cc2)=O)CCC(C(C)C)CC1CNC(=O)C(C)SC 40740,C1(NC(=O)CSc2cccc(F)c2)CC(O)CN(C(c2ccc[n+]([O-])c2)=O)C1 40741,C1(NC(C(C)(N(C(=O)COCCCN(C)C)C)C2CC2)=O)C2CCCC1CC2 40742,CC1=C(C)CC(C(N2CCCC2C2CCN(C(=O)CC3CCOC3)C2)=O)CC1 40743,c1(CC(=O)N(C2CCN(C(C3(C)CCCC3C)=O)C2)CC)ccccc1O 40744,C1(NC(c2ccc(OC)nc2C)=O)CCN(C(=O)CC(C)N(C)C)CC1(C)C 40745,C=CC(C)(CCOC)C(=O)NC1CCC(C)N(CC(=O)NC2CC2)C1 40746,C1(N(C(C)=O)Cc2c(C(=O)OC)occ2)COc2cc(Cl)ccc2O1 40747,CC1(CNC(=O)C(c2ccoc2)NC(=O)CCc2nc(O)n[nH]2)CC2(CCC2)C1 40748,C1(C(N(C)CC2(CNC(c3cnns3)=O)CC2)=O)C2Cc3c(Cl)cccc3C12 40749,c1(N2C(CC)CC(C(=O)O)CC2)nc2ccc(C(F)(F)F)cc2s1 40750,C1(NC(C2C(CC)C2)=O)(CNC(C2CC3CCCC3C2)=O)CC2CCC1CC2 40751,c1(C(N2CCC(N(C(C(C(C)C)F)=O)C)C2)=O)cccn2nccc12 40752,c1(CC#N)ccc(NC(C2COCCN2S(=O)(=O)Cc2ccc(F)cc2)=O)cc1 40753,c1(C(N2CCCN(C(C3CCC(C(N)=O)O3)=O)CC2)=O)cccc2c1CCO2 40754,N1(C(C2C(NC(=O)COc3ccc(F)cc3)CCC2)=O)CCN2CCC1CC2 40755,C(=O)(C(C)(O)C(C)C)NCC#CCNC(c1c(C)[nH]nc1C(F)(F)F)=O 40756,N1(C(=O)NCCN2C(C)CCCC2C)Cc2cnnn2Cc2ccccc21 40757,C1(C(N2CC(CNC(C(C)N(C)Cc3ccccc3)=O)C2)=O)CCS1(=O)=O 40758,C12(CNC(c3ccn(CCOC)n3)=O)CCC(CC1)N2C(C1(F)CCCCC1)=O 40759,C1(C2CCC(=O)NC2)(C(=O)NC(C2(O)CN(C(=O)CN=S(C)(C)=O)C2)C)CCC1 40760,C1(NC(c2cc(C)c(C)nc2)=O)CN(C(=O)CCC2CCCCC2)CC1N=[N+]=[N-] 40761,C1(NC(CC2CCC(C)O2)=O)(CNC(c2ccc(F)o2)=O)CCOCC1 40762,c1(CC)ccc2c(c1)cc(C)n2C.n12nnnc1C2NC1CCN(C(=O)CC)C1 40763,Cc1ncc(CC(=O)NC(C(=O)NCCCF)c2ccoc2)s1 40764,C1(C(N2CC=CC(NC(C3CCC(C)(CC)O3)=O)C2)=O)CCC(F)(F)C1O 40765,c1(C(N(C(CNC(CC2(C(=O)OC)CC2)=O)C2CC2)C)=O)nc(C)ncc1Cl 40766,CC#CCCC(=O)N1CCC(N2CCN(C(c3cnn(C)c3N)=O)CC2)CC1 40767,N1(C(C(C)COc2ccccc2)=O)CCC2CC1CN(C(C1(Cl)CC1)=O)C2 40768,c1(Cn2cc(C34N(C(CC56CC(C)(C5)C6)=O)CC(C3)C4)nn2)cc(O)cc(=O)o1 40769,c1(CN(C)C)cccc(NC(c2nnnn2CCCF)C2(Br)CC2)c1 40770,C1(C)(C(=O)NCC(CC=C)NC(=O)COc2cc(C)on2)CCCCNC1=O 40771,C(C)(N=c1[nH]c(=N)[nH]c(=NC2CCC(=O)N(C)C2)[nH]1)c1nc(C(CC)C)[nH]n1 40772,N1(C(c2cnn(C3CCC3)c2)C(=O)NCCCSC)CC2CCC1C(O)C2.C1CC1 40773,CC(CC(F)(F)F)C(=O)N1CC(CC(=O)NCCP(C)(C)=O)CC1(C)C 40774,c1(C(N(CCNC(CCN(C(C)=O)C)=O)C2CC2)=O)c(Br)ccc2n[nH]cc12 40775,C(=O)(CC(C)OC(C)C)NCCCOCCCNC(C1C(F)(C(=O)OC)C1)=O 40776,C1(C(N(CCN(C(c2c(C)noc2C)=O)C(C)C)C)=O)CC(C(C)C)=NO1 40777,O=C(C1=C2CCCN=C2NN1)C1N(C(c2ccc3c(c2)CNC3=O)=O)CCOC1 40778,C1(NC(c2cc(C)sn2)=O)CCC2(CC1)CCN(C(=O)CCc1cnn[nH]1)CC2 40779,C(=O)(CCC(=O)NC1CCC(CCNC(c2ccn(C(C)(C)C)c2)=O)C1)N(C)C 40780,C1(COC)(NC(C2CC(n3cc(C4(C)CSC4)nn3)C2)=O)CCCC1 40781,c1(NC)snc(C)c1C(N1CC(CNC(c2cncn2C(C)C)=O)C(O)C1)=O 40782,C1(NC(Cc2cccc(C(C)C)c2)=O)CN(C(=O)C(C)n2cncn2)CC1(C)C 40783,CC1CN(C(C2CCN(C)CC2)=O)CC(C)N1C(c1cnn2ccncc12)=O 40784,C1(N(C(C(C2CCC(=O)N2)C)=O)C2CC2)CCCCCC1C.C12CCCC(C1)NC2C 40785,c1(C(C(=O)NCC)N(C)C(c2ccco2)C)cc2n(n1)CC(C)(C)CO2 40786,C1(CNC(c2n(C3CC(F)(F)C3)nnn2)CCCCl)C(F)(F)C12CC2 40787,C1(COC)CC(C)(C)CCC1NC(c1ccccc1-n1cc(C=CC(C)C)nn1)=O 40788,C1(NC(CSC)=O)CCC2CN(C(C3CCCCNC3=O)=O)CC2C1 40789,c1(C(=O)NCCC(C)NC(c2cc(C)nnc2O)=O)c2c(nn1C)CCC2 40790,C=C(F)C1(CC(=O)NCC=CCC(=O)NCC2CC(CC)=NO2)CCC1 40791,CC1(C)COCC(NC(=O)C(C2(C)CC2)NC(=O)Cc2cnns2)C1 40792,C1(C(=O)NC(C2CCOCC2)C#C)(CC)CCN(C(=O)C(CO)N(C)C)CC1 40793,c1(C(c2n(CC)nnn2)NC2CN(c3nncs3)C2)cc(C)nnc1C 40794,C1(NC(c2c(F)ncc(OC)c2)=O)CC2CN(C(C3CC=CCC3)=O)CC2C1 40795,N1(C(C(CC=CCC)C)=O)CC2CC(NC(=O)C3=C(C)CCC3)C1C2 40796,C1(C(N2CCN(C(=O)CN(C(=O)CNC(=O)NC)C)CC2)=O)CCC2CC2CC1 40797,c1(C(CC(=O)NCC(CCNC(C=CCCC)=O)O)C)ccccc1OC 40798,C#Cc1cn(C)nc1C(=O)NCC1CC(NC(=O)C2=COCCO2)CC1O 40799,Cc1nc(CN=C(NCC2CCCO2)NC2CCC(=O)NC2)c(C)o1 40800,CC(C)C(CCNC(C1(C(F)(F)F)CCCCC1)=O)NC(=O)CC1CCOC1C 40801,N1(C(CC(CCC)O)=O)CC(CNC(c2cc(OCC)no2)=O)OC2(CCC2)C1 40802,CC(C)(C)C1=CCN(C(=O)COC2CCN(C(c3ccc(C(N)=O)[nH]3)=O)C2)CC1 40803,c1(C(=O)NC2CC(NC(=O)C(F)(F)C3CC3)C(O)C2)n[nH]c2c1CCCC2 40804,N1(C(CCCCC#C)=O)CCN(C(=O)CCCC(F)(F)F)CC(CO)C1 40805,C1(NC(C(CNC(C2(COC)CC(=O)C2)=O)C)=O)C(O)C2CCOC12 40806,C(=O)(C1=COCCO1)N1C(C(C)NC(C2(C)CC2C(F)(F)F)=O)CCC1 40807,c1(OC)ccc(C(N2CC(OC)CC2CNC(=O)CC2(C)CC2)=O)c(F)c1Cl 40808,c1(CC)c(C(=O)NC(C)C=CC(=O)NCC(C)OCCO)ccn1C 40809,C1(CN(C(CNC(C(CC)C)=O)=O)C)CCN(C(c2cc(F)c[nH]2)=O)CC1 40810,c1(CCNC(C=C(C)CNC(=O)C(C)CN(C)C)=O)ccc(C)s1 40811,N1(C(C2CCN(C(C)=O)C2)=O)CCCC2(NC(C3COCCN3C)=O)CCCC12 40812,c1(C(=O)OC)cc(F)c(F)cc1NC(C1CC(O)CCN1C(c1nc[nH]n1)=O)=O 40813,C(C)(C)(CN=c1nc(N2CCN(CC(C)F)CC2)c2c(ncn2C)[nH]1)OC 40814,CC(Cc1ccccc1)C(=O)NNC(=O)c1cc2c(s1)CCCCC2 40815,c1(CCCC(=O)NCCC)ccc(C#N)cc1.C(=O)(C(C)=CC(C)(C)C)N(CCC#N)C 40816,C(=O)(CCCC(F)(F)F)N1C(C)CC(NC(=O)CCC2(O)CCC2)C1 40817,N1(C(c2cc(N)c(F)cc2)=O)C2CCC1CN(C(c1cn(C3CCC3)nn1)=O)C2 40818,n1(CCNC(=O)NC(c2ccc(F)cc2)C(=O)OC)c(=O)oc2ccccc12 40819,N1(C(C2CC(C)=C(C)CC2)=O)CC2CN(C(C3(CCF)CC3)=O)CC2(C)C1 40820,c1(CC)ncc(C(=O)NC2(CCCNC(c3ccc(CC)s3)=O)CC2)[nH]1 40821,c1(C(N2CC(O)(CN(C)C(c3nsnc3O)=O)C2)=O)ccc(Cl)c2c1OCCO2 40822,c1(C(=O)NCCN(C(C2CN(C)C(=O)N2)=O)C)cccc(C#CCO)c1 40823,N1(C(C(C)n2ccnc2)=O)CCSCC1CCNC(C1NC(=O)CC1C)=O 40824,CC1CC(N(C)CC2CCC3CC3C2)CCN1Cc1ccccc1 40825,C1(CNC(=O)C=CC2CC2)CC2COCC2N1C(=O)Cn1ccc([N+](=O)[O-])n1 40826,N1(C(c2csc(Cl)n2)C(=O)NCCC)CCC(C2(C)CC2)CC1 40827,CCCCCCC(C)(c1nnnn1CCC)NC1CCn2cncc2C1 40828,C(CNC(C1CSCN1C(C1CCC1)=O)=O)(CO)(CO)N(C(C=CC)=O)C.C(C)(=O)O 40829,c1(C(N2CCC(N(C(=O)C(F)F)CC#C)CC2)=O)noc2c1COCC2 40830,C#Cc1cccc(CC(N2CCC3(NC(c4nn(C)cc4C)=O)CC3C2)=O)c1 40831,C1(C)(C(=O)NC(C2CN(C(c3cc(O)ncn3)=O)CCO2)C)COC(=O)N1 40832,C1(NC(c2occ(C)c2C)=O)CCC(C)N(C(=O)CCc2ccc(F)cc2Cl)C1 40833,C=C(C)C1CN(C(=O)CC(C)(C)NC(c2ccncc2)=O)CCO1 40834,N1(C(C(C(=O)OC)C)=O)CCOC2CCN(C(c3ccc(C(N)=O)[nH]3)=O)CC12 40835,c1(C(=O)OC)cc(C(=O)CN2C(=O)NC3(CCC3)C2C)no1.C1(OC)CC1 40836,n1(CC)cc(-c2ccc(N3CCN(C(=O)C=CC)CC3)cn2)ccc1=O 40837,C1(C(=O)NCC2(CC)CCC(=O)N2)CCCCCCN1C(C1CC=CC1)=O 40838,C1(C(=O)NCc2nccc(C)c2)COC2(C1)CN(C(=O)CC1CC1(C)C)C2 40839,c1(C(C)COC(=O)COC(=O)Cc2cccs2)ccncc1Br 40840,C(=O)(C1=NNC(C(F)(F)F)C1)NC(C1CN(C(=O)C(C)(C)O)C1)C 40841,c1(C(N(C(C)CN(C)C(c2csc(Cl)c2)=O)C)=O)ccc(F)c(Br)c1 40842,N1(C(CCCCC)=O)CCC(NC(c2cccnc2O)=O)C(CO)C1 40843,C(CNC(C1(c2cccc(F)c2)CC1)=O)(C(C)C(C)C)NC(CNC(CC)=O)=O 40844,N1(C(C2C(C(C)NC(c3cccc(C)n3)=O)C2)=O)C2CCC1CN(C)C2 40845,C1(C(=O)NC2(c3cn(C(CC)C)nn3)CCC2)CCc2ncc(C)n2C1 40846,CN1CCC(O)(CNC2(N3CCNC3=O)CC2)C1.C12C(CC1O)NC(=O)C2O 40847,C(C(CN=c1cc(NC(c2ccc(Br)cc2)CF)nc[nH]1)OC)OC 40848,C1(C(=O)NCC(c2cc(OC)c(Cl)cc2)F)CC2COCC(C1)C2(F)F 40849,C1(CNC(Cc2ccn(C(C)C)n2)=O)CC(C)(C)CN1C(C1CC(C)C1)=O 40850,C1(NC(c2ccc(C)s2)=O)CN(C(=O)CC2CC=CCN2C)CC1C 40851,N1(C(C(c2cn(C)nc2)=O)=O)CCCC(CNC(C2CCCN2C2CC2)=O)CC1 40852,Cc1cc(C(=O)NC2CCCC(NC(=O)C3=NOCC3)C2)cc2c1NCCC2 40853,c1(C(N(C(C(=O)N(C(CCCC)C)C)CC)C)=O)cc([N+](=O)[O-])n[nH]1 40854,c1(C(=O)NC(CCC)C(=O)NC2CCC(C)(C)CC2)n[nH]c2c1CCC2 40855,c1(CC(=O)N(C(CNC(C2C=CC(C(=O)OC)C2)=O)C)C)ccnnc1O 40856,CC1CCOC(C(=O)NCCc2n[nH]cc2C(N2CC=CC2)=O)C1 40857,CCC(C(=O)NC(C1CCN(Cc2nc(C3CC3)no2)CC1)C)C(C)C 40858,N1(C(N2CCN(C(COC)C)CC2)=O)CCCc2cc(C)cc(F)c21 40859,c1(CC(=O)NCCCN(C(CCC2CCN(C)C2)=O)C2CC2)cccc(Cl)c1 40860,C1(OC)(NCCC(=O)NCCC(=O)OC)CCC(C)(C)C1 40861,C1(C(=O)NC(CC)CN(C)C(C2(OC)CCCC2)=O)CCCCC1C(C)(C)C 40862,c1(CC)nn(C)cc1C(=O)NCC(C)NC(c1onc(Br)c1C)=O 40863,C(=O)(C1=NN(CC)C(=O)CC1)N(C)CC1N(C(c2nc(CC)oc2)=O)CCCC1 40864,c1(C2(CNC(c3nc(C)c(C)o3)(c3n(CCSC)nnn3)C)CC2)ccccc1C 40865,C1(NC(c2cccc(CNC(CC3CC(SC)C3)=O)n2)=O)CCC12CCCC2 40866,N1(C(CS(C)(=O)=O)=O)CCCC(O)(CNC(C2OCCC2c2ccccc2)=O)C1 40867,c1(NC(N2CC(C(C#C)C)C2)=O)cc(C(=O)OCC)cc([N+](=O)[O-])c1 40868,Cc1ccc(C)c(C(=O)NCC2C(C)CCN2C(=O)CNc2ccccn2)c1C 40869,c1(C(=O)NC(C2CN(C(c3onc(CC)n3)=O)C2)C)nc(C)sc1C 40870,C1(C(=O)NC(C2CCCN(C(=O)CCC3CC3)C2)C)(NC(C)=O)CCCCC1 40871,C(=O)(C1=CCCSC1)NCC=CCC(=O)N(C)Cc1cc(=O)cc[nH]1 40872,Cc1ccc2cc(C(N3CCC(C(C)NC(C4CCCC4F)=O)CC3)=O)cn2c1 40873,c1(C(N2CCN(C)CC2CNC(=O)CCCCO)=O)cnc2n1CCOC2 40874,C1(C(=O)N(C)Cc2ncc[nH]2)(COC)CCCN1C(=O)CC(O)CN(C)C 40875,C(C(CC(F)(F)F)NC(=O)CCOC)NC(c1ccc(N(C(C)=O)C)cc1)=O 40876,c1(C(=O)NCC2C(CNC(c3ncn(C(C)(C)C)c3)=O)C2)cc2scnc2[nH]1 40877,CN1CCN(C(C2CCCC2(F)F)=O)C(CNC(c2cc[nH]c2)=O)C1 40878,c1(C(=O)NC(CCC)c2ccco2)oc(CNC(C2(Cl)CCCCC2)=O)nc1C 40879,N1(C(C(C#C)(C)C)=O)CC2(CCN(C(C3(c4ccsc4)CC3)=O)CC2)C1 40880,N1(CCOCCOC)CCC2(CCN(C(c3c(C)cc(C)nc3Cl)=O)C2)C1 40881,C#CC1(C(=O)NC(COC)CO)CN(C(c2cnnn2C=C)=O)C1 40882,N1(C(c2cn(C)nc2)C(=O)NC2CCOC2)CCOC(c2cccc(Cl)c2)C1 40883,c1(C(=O)NCCNC(=O)CCC2CCC2)cccc(F)c1 40884,N1(C(C(C)=C(CC)C)=O)CC2CC(C1)C2NC(=O)CN1CC(C)C1 40885,CC1CC2CC(C(=O)NCCC3CCCN(C(=O)C4=COCCO4)C3)(C2)O1 40886,c1(C(C)NCC2(NC(=O)OC(C)(C)C)CCCCC2)ccc(Cl)c(F)c1 40887,N1(C(C2C(C(=O)OC)CC2)=O)CCC(C(=O)NC(c2nc(C)no2)C)C12CC2 40888,C1(NC(C2(C(=O)OC(C)(C)C)CCC2)=O)CCOC(c2ccc(F)cc2)C1 40889,n1(CC(=O)NC2CN(C(CC3(OC)CCCCC3)=O)CC2O)cc(F)ccc1=O 40890,CC1Oc2ccccc2OC1C(N1CCCC(NC(C2(C)CC2)=O)C1C)=O 40891,N1(C(C2CC(SC)C2)=O)CC2CN(C(C3CCCS3(=O)=O)=O)CC2(C)C1 40892,CCCC(CCC)CC(=O)N1CCN(C(=O)CN(CC)CC)C(CS(C)(=O)=O)C1 40893,C1(C(=O)NC(CNC(C(C(C)C)NC(=O)C(C)(C)C)=O)(C)C)CCC(F)(F)CO1 40894,C(=O)(C(C)(C#N)CC)NCc1c(CNC(c2c(CC)nn(C)c2)=O)cccc1 40895,N1(C(c2cc(C)c(Cl)cn2)=O)CCCC(C2CCN(C(=O)CCCC#N)C2)C1 40896,C(c1cncnc1O)=CC(=O)NCC1(NC(Cc2nn(C)c(Cl)c2)=O)CCOC1 40897,CC(C1CCCCC1)=CC(=O)NCC(C)NC(=O)Cc1cc(C)n(C)n1 40898,NC(=O)CC(C(=O)N1CCCC(C(F)F)C1)NC(c1ccc(O)cn1)=O 40899,CCC(C(=O)NCCC1CCN(C(=O)C(N2CCC(C)CC2)=O)CC1)C(C)O 40900,c1(C(N2CCC(NC(C(C(C)C)OCC)=O)C2)=O)cnc(C)nc1C1CC1 40901,N1(C(CC(C)F)=O)CCC(CNC(=O)CN(S(C)(=O)=O)C)C(F)(F)CC1 40902,N1(Cc2cccc(OC)c2)CCCC(CO)(NC(=O)CC2(OCCC)CC2)C1 40903,CC(C)(C)CCCCC(=O)NCCC1CCN(C(c2cc(F)c(F)cc2O)=O)C1 40904,C(C)(C)(C(=O)NCCCN(C(=O)CC1(C)CCCC1)CCO)OC 40905,N1(C(COC(CC)C)=O)CCCC(C(=O)N(C)CCC2CCCC2)CC1 40906,CCCC(C)(C)C(=O)N1CC(C(=O)Nc2ccc(Cl)cc2O)CC(C)C1 40907,O=C(C1CNc2ccccc21)N1CCN(Cc2ccc(Cl)cc2)C(=O)C1 40908,C=CCC(CC=C)C(=O)NCC1CC(C(=O)CCC)N(CCCO)CC1CCCO 40909,CS(=O)(=O)c1coc(C(=O)NCC2CCCCN2C(C2CC3CCC(C2)O3)=O)c1 40910,Cc1c(C(=O)NCCCOCCCNC(=O)CC2CCC(O)C2)ncn1C 40911,Cc1nc(Cl)[nH]c(=NC(C)CC(C)NC(c2ccc(C(C)C)c(Cl)c2)=O)c1F 40912,CCCCC(CNC(=O)C1=CCCC1)NC(=O)CCc1cnc(C2(C)CC2)o1 40913,C1(C(N2CCC(C(CC)CC)C2)=O)C2CC3C(C2NC(=O)C(C)(O)CCOC)C13 40914,N1(C(C(CC#C)C2CC2)=O)CCN(C(=O)C(C)(F)F)CC1C1CC1 40915,c1(C(N(CC(C)NC(c2n[nH]cc2Br)=O)C)=O)cc2c(cc1O)CCC2 40916,C1(CNC(CCCc2onc(CC)n2)=O)CCN(C(C2CCCSC2)=O)CC1 40917,c1(C(N2CCC(C)(NC(CCOCCOC)=O)CC2)=O)ccc2occc2n1 40918,CN1CC(C(N2CC(C3CC3C(=O)NC3(CC(N)=O)CC3)C2)=O)CCC1=O 40919,c1(C(=O)NCC2CN(C(=O)CN3CCOCC3)C2)ncn2cc(Cl)ccc12 40920,c1(C(C)NC(CC)C(C)C)cc(C(F)(F)F)ccc1F 40921,c1(C(=O)NC(CCNC(c2c(COC)nn[nH]2)=O)(C)C)cn2c(n1)CCCC2 40922,c1(C(C2CC3CC3C2)NC2(C)CC2)nnnn1CCNC(=O)C1CC1 40923,c1(C(=O)NCCN2CCN(C(C3C(C(=O)OC)C3)=O)CC2)ccc2ncsc2c1 40924,c1(C(=O)NC(CNC(C=NOC)=O)CO)cc(Br)c([N+](=O)[O-])[nH]1 40925,C1(NC(C2(N(C)C)CC2)=O)CCCC(N=c2[nH]c(Cl)nc3ncn(C)c23)C1 40926,C(C1c2ccccc2CN1C(c1ncoc1C)=O)NC(CCC(CC)C)=O 40927,c1(C(=O)NCC(CNC(C(c2cc(C)sc2)(C)C)=O)F)c(C)coc1C 40928,CC(C)(C)C(C)(O)C(=O)NCC1(NC(=O)C2=CCCCCC2)CCCC1 40929,N1(C(CNC(CC)=O)=O)CC(NC(=O)C(C2CC2)OCC)CC2(CCC2)C1 40930,c1(C(N2CCCC(CCNC(CC(=O)N(C)C)=O)C2)=O)cc(Cl)ncc1N 40931,CC1(C)CCC(C(=O)NC2(CNC(C3(C(F)F)CC3)=O)CCOC2)C1 40932,C1(C(=O)OCC)CC(C)CN(C(=O)C(=O)NC(c2c(NC)cccc2Cl)C)C1 40933,CCN=C(NCCOCC1CCOC1)NCC.C12CCCC1N2 40934,C1(CC(=O)NCCCCN(CCCNC(C(CCC)C)=O)C)COC(C)(C)CO1 40935,C(=O)(CC1OCCc2ccccc21)NC1CC(NC(C2COCC(C)(C)O2)=O)C1 40936,C12(NC(Cc3nc(CC)sc3)=O)CCN(C(=O)COC3(C)CCC3)CC1C2 40937,C12(C(N3CCN(C(c4c(C)onc4C4CC4)=O)CC3)=O)CCC(CC1)C(C)O2 40938,C1(C(N2C(CNC(C(CCSC)O)=O)CC3CC32)=O)CCC(=O)N(C2CC2)C1 40939,CCC(C)CC(C(=O)NCc1c(C)coc1C)NC(C1CN(C)C(=O)N1)=O 40940,N1(CC(=O)NC(c2ccc(C)cc2)=O)CCCN(Cc2cscc2C)CC1 40941,C1(F)(CNC(CC2(CSC)CC2)=O)CC(NC(=O)C(C)(C)C2CCCCO2)C1 40942,c1(C(N2CC(C(C)NC(Cc3c(C)noc3)=O)OCC2)=O)ccn2nnnc2c1 40943,N1(C(C#C)(C)C)CCN(C2CCCN(C(C3CC3c3ccccn3)=O)C2)C(=O)C1 40944,c1(C(N2CC3(C(NC(c4ccc(F)s4)=O)CC3)C2)=O)coc2ccccc12 40945,c1(C(N2CCC(C)(CCNC(CN3C(C)CC3)=O)C2)=O)cnc2[nH]cnc2c1 40946,CC(CN(C)C(=O)NC(CCCC(=O)OC(C)(C)C)c1ccccc1)S(C)(=O)=O 40947,c1(C(=O)NCCOCCNC(CC(COC)(C)C)=O)cc(N)c2ncccc2c1 40948,c1(CCC(=O)NCCOCCNC(C(C)(C)F)=O)ccc(F)cc1F 40949,C(C(CC(C)C)NC(=O)C(O)C(F)F)NC(CCCN(C(=O)OC)C)=O 40950,N1(C(CCSC)=O)CCC2C(C1)NC(=O)N2C1CCN(C(=O)CC(C)(C)C)CC1 40951,C=CCCC(C1CC1)NC(=O)C#CCNC(c1csc(=N)[nH]1)=O 40952,C1(NC(C2C(C)C2)=O)CCOCC1C(=O)NCC(=O)NC1CC1 40953,CC(C)CC(O)C(=O)NCC1OCCC1C(=O)NC1(CO)CC(F)(F)C1 40954,c1(C(=O)NC(C(CO)NC(COc2cccc(OC)c2)=O)C)ccc(C)nc1O 40955,C(=O)(C1=NN(C)C(=O)CC1)N1C(C)CCC(NC(C2(CCO)CC2)=O)C1 40956,N1(C(CC(=O)N(C)C)=O)CC(C2(NC(=O)CCc3ccoc3)CC2)C1 40957,CC1CN(C(=O)CN2CCC(=O)CC2)CCC1NC(=O)CCC1CCN(C)CC1 40958,c1(C(=O)NCC(C)N(C)C(c2ccc(F)cc2Cl)=O)ccc2cnsc2c1 40959,CC(C)C(O)C(=O)N1CCC(C(C)NC(C2C(c3ccccc3)C2C)=O)CC1 40960,c1(C(N2CCCC(C3Cc4ccccc4O3)C2)=O)n[nH]c2c1CCCCC2 40961,CC#CC1CN(C(C2CCN(C(c3cn[nH]c3)=O)CC2)=O)C1 40962,N1(C(CCN(C(c2noc(C)n2)CC)CC#C)=O)CCC(C=C)(C(=O)OC)CC1 40963,Cc1cc(C)n(CCCNCc2ccccc2-c2ccc(F)cc2)n1 40964,C(c1cc(Cl)ccc1Cl)=CC(=O)NCCCNC(CCc1ccc(C)s1)=O 40965,C1(N)CCc2ccccc2C1.C1(c2ccn(C)n2)CCN(C(=O)C(N2CCCC2)N)CC1 40966,N1(C(C2(O)CCN(CC3CCOC3)CC2)=O)CCc2cccc(O)c21 40967,CCCC(CNC(=O)CSC(F)F)NC(=O)CCOCC 40968,c1(C(=O)NC2(CF)CCN(C(Cc3c(C)nc(C)s3)=O)C2)cc(C)c(F)cc1F 40969,C1(NC(c2cc(OC)c(F)cc2)=O)CCN(C(C2CC2(Cl)Cl)=O)CCC1CO 40970,Cc1c(C(=O)NCC(C2CCCCN2C(c2cnc[nH]2)=O)(C)C)cnn1C(C)C 40971,N(C1C(=O)N(C)CCc2ccccc21)CCN1C(C)CCC1 40972,N1(C(COC(C)C)=O)CC(NC(=O)CC2(C)CC2)C2CC12 40973,N1(C(CC2CN(C)C2)=O)Cc2ccccc2CC1CNC(C1CC2C=CC1C2)=O 40974,N1(C(Cc2cnc(C)[nH]2)=O)CCOCC(C)(CNC(=O)C(C)NC(=O)C2CC2)C1 40975,CC1(C)C=C(C(=O)N2CCN(C(c3cn(C4CC4)nn3)=O)C(C3CCC3)C2)C1 40976,N1(C(CC2(C)CCC2)=O)CC2CC(C1)N2C(=O)CN1CCN(C2CC2)C1=O 40977,N1(C(C(CC#C)C2CC2)=O)CCC2CN(C(c3cc4sc(C)cc4s3)=O)CC12 40978,c1(C(N2CC(N(C(CCSC)=O)C)C(F)C2)=O)cc(Cl)cc(Cl)c1[N+](=O)[O-] 40979,CC(C)(CS(N)(=O)=O)C(=O)NCC1CN(C(C2(O)CCC2)=O)CC12CC2 40980,CN1CCC(C(=O)NC2(C)CCN(C(=O)CC3CCSCC3)C2)S1(=O)=O 40981,C1(C(=O)NCC2CCC(C(=O)NCc3cnc(CC)s3)O2)CC2CCC1O2 40982,CC(c1cccnc1)=CC(N1CC(NC(c2nccc(C)c2N)=O)C2(CC2)C1)=O 40983,Cc1cc(NC(=O)C(Cc2ccoc2)NC(C2COCCC2C)=O)cc(CO)c1 40984,CCC(CC=C)NC(=O)CC1(OC)CN(C(=O)CC2CCC(=O)C2)C1 40985,Cc1nc(F)ccc1NC(c1ccc(NCCC(C)C)cc1Cl)=O 40986,c1(NC(C2(NC(c3ccc(C)cn3)=O)CCCCC2)=O)ccc2occc2c1 40987,c1(-c2nc(COC)nn2CC(C)C2CC2)c[nH]c2c(OC)cc(F)cc2c1=O 40988,C(=O)(CC(C)CC(C)C)NC(CC=CC)C(=O)NCCc1cccnc1F 40989,c1(C(=O)NC2CC(NC(C(C3CCCCC3)OC)=O)C2)cccc(C(F)(F)F)n1 40990,CN1CCc2[nH]nc(NC(N3CCOCC3CC(c3ccco3)O)=O)c2C1 40991,O=C(C1=Cc2cc(F)ccc2OC1)NCC1CC(NC(c2ccno2)=O)C1 40992,c1(OC)cc(NC(C2CCCN(C(=O)C(=O)c3ccco3)C2)=O)ccc1Cl 40993,C12(C(NOCCCC#C)=O)CCN(C(=O)CCOCCOCC)CCC1C2 40994,c1(C(=O)OCC(CC)C)cccnc1-c1ccccc1 40995,CC1CCCC(C)C1NC(=O)CCOCCCNC(c1ccc(CC#N)cc1)=O 40996,c1(NCC(CC)(C)OCC)[nH]cnc1C#N 40997,C=CC(CC)C(=O)NC1(CC(=O)NCC(C)COC)CC1 40998,N1(C(C(C=COCC)O)=O)CC2C(CO)C2C1.c1(C(N(CC(=O)N)C)=O)ccccc1 40999,Cc1ccc(F)cc1CN1CCC(OCc2cnc(C)n2C)C1 41000,c1(C(=O)NCCCCC(C)NC(=O)C(F)(F)C(F)F)cnc2c[nH]nc2c1 41001,C1(CC(=O)N(C(C)CCNC(=O)C2=COCCC2)C)COc2ccccc2O1 41002,N1(C(C2=C(C#N)CCC2)=O)CCC2(CCC2)C(CNC(c2ccoc2Cl)=O)C1 41003,C1(CNC(c2cc(C(C)=O)sc2)=O)CN(C(c2ccc(O)nn2)=O)CC1C 41004,Cc1nc(C(=O)NC2CN(C(C3CCCN3C=O)=O)CC2C)c2ccccn12 41005,N1(C(CN(CC#C)C(c2cn(C)nc2CC)=O)=O)CCCC(CN(C)C)CC1 41006,N1(C(CCC2CC(NC(=O)CC3(CO)CCC3)C2)=O)CCC2(CC1)CC(O)C2 41007,C=Cn1nncc1C(=O)NCCCCCNC(c1c(Br)n[nH]c1C)=O 41008,C(=O)(CC(CC(C)C)NC(c1ncccc1CC)=O)N(C(C=C)C)C 41009,C(C)(CC(=O)N(C1CCN(C(C2(N(C)C)CC2)=O)C1)C)=C(C)C 41010,C(=O)(C(CCNC(c1nn(C)cc1N)=O)OC)N(CCOC)CC1CC1 41011,c1(C(=O)NC2C(NC(CCN(CC(F)(F)F)C)=O)CC2)cccc(N)c1 41012,c1(CC(=O)N(CCCCCNC(C2(C#C)CCC2)=O)C)cccc(F)c1F 41013,C12(C(=O)NCCCCC(C)NC(C=CC)=O)C3C(=O)C4C5CC(C14)C2C35 41014,N1(C(Cn2cc(C(=O)OC)nn2)=O)CC2CC3CC2C1C3NC(=O)CSC(C)C 41015,Cc1cc(C#N)c[nH]c1=NC(C)CC(C)NC(=O)Cc1cnsc1 41016,c1(C(N2CCC3C(NC(CC(CCC)C)=O)C32)=O)cc(N)c(Br)c(F)c1 41017,c1(C(=O)NC(C2CN(C(=O)CC3CCC(=O)N3C)C2)C)ccc2nc(O)[nH]c2n1 41018,Cc1[nH]nc2ccc(C(N3CC4(C)CN(C(=O)C(=O)N(C)C)CC4(C)C3)=O)cc12 41019,S(=O)(=O)(c1ccc(=NCCCSCCO)[nH]c1)NC(C1CCCCC1)(C)C 41020,C1(CC)(NC(=O)COC2CCOC2)CCN(C(c2noc(C3CC3)c2C)=O)CC1 41021,C1(C)(C(=O)NCC2CN(C)C2)CN(C(=O)CCN2CCOCC2)C1 41022,c1(C(C(=O)NC(C(CO)NC(C(CC)C)=O)C)(C)C)cccc(F)c1 41023,c1(C(=O)NCC(CC=C)NC(C2CC2c2ccccc2)=O)nccnc1SC 41024,C1(CC)CN(C(c2cnn(C)c2CC(C)C)=O)CCN1C(=O)CS(=O)(=O)N(C)C 41025,c1(CC)oc(C)cc1C(=O)NCCC(C)N(C(=O)Cc1cc(C)cs1)C 41026,CC(C)CC(O)C(=O)NC1CCCN(C(c2cccc(C3(F)COC3)c2)=O)C1 41027,N1(C(C(=O)NC2CCCC(F)(F)C2)=O)CCC2(CCc3ccccc32)C1 41028,C1(N(C(C(C)CC2CC2)=O)C)CCCN(C(=O)Cc2cncc(Br)c2)C1 41029,N1(C(C2C(NC(=O)CC3CSCCO3)COC2)=O)CCC2(CC1)CC(O)C2 41030,c1(CC(C)C)ccccc1CNC(=O)NC(CCc1ccc(Cl)cc1)C(C)C 41031,c1(C(N2CC(N(C)CCO)C2)=O)cc(CCNC(c2c[nH]c(=N)o2)=O)on1 41032,C1(NC(c2c(C)n(C3CC3)nc2)=O)CC2(CCN(C(C3(C)C=CCC3)=O)C2)C1 41033,C1(NC(C2CCC(=O)OCC2)=O)CC2CCC1C(NC(C1(F)CCC1)=O)C2 41034,c1(OC(C)C)ccc(CNC(=O)CC2CCCCN2C)nc1 41035,Cc1ccc(OCCCC(N2CC(NC(=O)C(C)N(C)C)C(C)C2)=O)cc1 41036,N1(c2ncc(C)c(O)n2)CC(CNC(C2(C)CCCCO2)=O)OC(C)(C)C1 41037,N1(C(=O)COCC2CCCO2)CCC2C(C1)CN2C(c1cc(CC(=O)O)c[nH]1)=O 41038,c1(OC)nccc(CNC(=O)CC2(OC)CN(C(C3CCOC3C)=O)C2)n1 41039,N1(C(C(C#C)NC(=NCc2ccco2)NCC(C)(C)C)(C)C)CCCC1(C)C 41040,c1(CNC(C2CC(CC)C2)=O)nnn(C)c1C(N1CCC(OCC)C1)=O 41041,Cc1cc(F)c(C(N2CCC(N(C)C(c3nc(C)c(C)s3)=O)C(C)C2)=O)cc1F 41042,C1(C#N)(C(=O)NCCCCCCNC(CC2C(C)CCO2)=O)CCCCCC1 41043,CCC(C)CCCCC(=O)N(C)CC1C2CN(C(=O)C=C(C)C(F)F)CC12 41044,c1(C(=O)NC2C(NC(c3cc(C)cc(Cl)c3)=O)CC2)cccc2nn(C)cc12 41045,C1(CC(=O)N(C(CC#C)C)C)CN(C(=O)CC2CCC(=O)C2)CC12CC2 41046,c1(C(C)C)ncc(C(N2CC(C(C)(C)O)(CNC(C3C(C)C3C)=O)C2)=O)s1 41047,c1(C(=O)NC(C2CCCN(C(c3n(CC)ncc3)=O)C2)C)cc2n(c1)CCSC2 41048,c1(C(=O)NC2C(NC(c3cc(C4CCC4)on3)=O)CCC2)ccn2ccsc12 41049,c1(C(=O)NC2C(CNC(CC(COC)C)=O)CCC2)cnc(O)c([N+](=O)[O-])c1 41050,c1(C(N(CC(CNC(C2(SC)CCC2)=O)(C)C)C)=O)ccnnc1C 41051,C=C(CNC(=O)C(CCC1CC1)NC(C1CC(=O)CS1)=O)C(F)(F)F 41052,Cc1ccccc1C1(C(=O)NCC2CC(NC(c3n[nH]cc3Cl)=O)C2)CC1 41053,C1(CNC(COCCCC)=O)CN(C)CCN1C(c1cc(C2CC2)nc(O)c1)=O 41054,N1(C(CCC2CCN(C(c3cc(C)no3)=O)C2)=O)CC2CCC2(C)C1 41055,c1(C(=O)NCC2C3CN(C(C4(C)CCCS4)=O)CC32)ccc2scnc2c1 41056,N#Cc1ccc(S(=O)(=O)N2Cc3ccc(O)nc3C2)nc1 41057,c1(C(=O)NCC2(F)CC(CNC(=O)CC3CCC4CC34)C2)cccn2nncc12 41058,Cc1[nH]c(C#N)cc1C(N1CCC(C)(CC(=O)NCCN2CCNC(=O)C2)C1)=O 41059,C1(CC)CN(C(C2CCC3CC3C2)=O)CCC1Nc1nc(C)cc(C)n1 41060,C(CN=c1[nH]c(C)cc(=NCc2ncc(Br)cn2)[nH]1)c1ccc(OC)cc1 41061,c1(C(N(CC(CN(C(CCOC(C)C)=O)C)O)C)=O)cn(C)cc1C(F)(F)F 41062,c1(NC(C(CCC(=O)N2CCCCCC2)F)=O)cccc2c1OCCC2 41063,c1(C(=O)NCCC2(C(=O)NCc3c(C)occ3)CCC2)cn(C)c(C)n1 41064,c1(C(=O)NCCCCNC(C(C)(C)OC(C)=O)=O)snc(Cl)c1Cl 41065,C1(NC(c2cncc(SC)c2)=O)CCCN(C(C2(S(C)(=O)=O)CC2)=O)CC1 41066,C(=O)(N=c1[nH]nc(-c2ccc(OC)cc2)s1)N1C(CC(C(=O)OC)F)CC1 41067,N1(C(C(Cc2ccoc2)NC(C2CN(C)C2)=O)=O)CC2CC1CO2 41068,O=C(CCCn1cncn1)NCCCc1cn(C2CCCC2O)nn1 41069,C(CC1=CCCCCC1)NC(C1C(CNC(C(C)(CO)OC)=O)CCO1)=O 41070,C1(NCC2(C(C)N)CC2)CCN(c2ccc(SC3CC3)cc2)C1=O 41071,Cc1nc(C(=O)NCC2(C)CCC(NC(=O)CCC(=O)N(C)C)C2)c(C)n1C 41072,C1(O)(CNC(C2CC(CCC)C2)=O)CCCN(C(=O)COC(=O)CO)CC1 41073,CC1(C(=O)NC2CCC(C(=O)NC3CCOCC3F)C2)CC2C=CC1C2 41074,C#CC1CCCCN1C(=O)C(F)CC1CN(C(=O)COc2ccsn2)C1 41075,C1(CC)(NC(=O)C(C)SC(F)(F)F)CCCN(C(C2CN(S(=O)(=O)CC)C2)=O)C1 41076,C1(NC(CCCCNC(C(c2ccn(C)n2)C)=O)=O)CCN2CCCCC12 41077,C(CCC(C)NC(c1cscc1OCC)=O)NC(CN(S(CC)(=O)=O)C)=O 41078,N1(C(C(N2CCC(CC)CC2)=O)=O)CCC2(CC1)CC2C#N 41079,N1(C(COC(C)C)=O)CCN(C(=O)CSc2cccs2)C(C)CC1C 41080,c1(NC(=O)N(C)C2CC2)cc(Cl)ccc1CNC1OCCC(CSC)C1 41081,c1(C(=O)NC2C(C)CN(C(=O)C(C)(C)CN(C)C)C2)c[nH]c2nc(F)ccc12 41082,c1(OC)ccccc1-c1nc(CN(C)C(=O)N(C2CC2)Cc2cscn2)cs1 41083,C1(NC(c2c(C)oc(C(C)C)c2)=O)CCCN(C(c2[nH]nnc2C2CC2)=O)C1C 41084,CC(C)(C)C(CCc1cccc(F)c1)C(=O)NC1(C)CCCN(C(=O)C(F)F)C1 41085,Cc1cc(C)cc(C=CC(=O)NCC(CNC(C2C(C#N)C2(C)C)=O)CO)c1 41086,C(=O)(C1=CCCC1P(C)(C)=O)N1CC(C)C(NC(=O)Cc2cnccn2)C1 41087,c1(C(N(CC(C)N(C)C(C2CCN(C)C2)=O)C)=O)cnc2ncc(Br)cc2c1 41088,N1(C(C2CN(CCCC)C(=O)C2)=O)CC(NC(=O)CCOC2CCC2)CCC1C 41089,CC(C)(C)C(CO)C(=O)NCc1cccc(NC(C2CCn3ncnc3C2)=O)c1 41090,N1(C(c2c(C)ccn2C)=O)CCC2(CC1)CN(C(=O)C1=CCCCC1C)C2 41091,C1(CC(N)=O)CCN(N2CCC(Cc3ccccc3F)CC2)CC1(F)F 41092,c1(OC)cc(Cl)ccc1C(N1CC2(NC(=O)C(C3CCCC3)OC)CCC1C2)=O 41093,c1(C(N(CC#C)C)=O)cc(CNC(C2(Cl)CC2)=O)no1 41094,CCC(C)CC(=O)C(=O)NCC(C(=O)N(C)CC1CCCN1CC)C(C)C 41095,C(c1ccccc1C#N)=CC(=O)NC1(C)CC(NC(c2ccc(Cl)o2)=O)C1 41096,N1(C(c2c(CCC)[nH]cc2)=O)CCCC12CCN(C(=O)C(C)CC(C)(C)C)C2 41097,c1(C(N2C(CNC(c3cc(C(=O)OC)on3)=O)CC(O)C2)=O)ccc([N+](=O)[O-])[nH]1 41098,C1(n2cc(N(C(c3c(OCC=C)cccc3)=O)CC)nn2)CCCC1S(C)(=O)=O 41099,c1(Cn2ncc(C(N(CCN(C)C(C3CC3Cl)=O)C)=O)c2)ccccc1Cl 41100,CC1CCN(C(C2CCCN(C(N)=O)C2)=O)CC1NC(=O)C(F)n1cccn1 41101,N1(C(C(CC)=O)=O)CCC(O)(c2cn(C(c3ccccc3F)C)nn2)CC1 41102,c1(NCCC(N2CC3C(NC(C=C(C)C)=O)(C3)C2)=O)oc(C)nc1C#N 41103,C1(NC(c2c(OC)ccs2)=O)CCOC(C(=O)NCCNC(N)=O)C1 41104,N1(C(CC(c2cccc(OC)c2)C)=O)CCCC(N=c2nc[nH]s2)C1 41105,c1(C(=O)NC2COCCC2NC(C2(C3CCCO3)CC2)=O)cc2n(c1)CCCC2 41106,CC(Cn1ccnc1)C(=O)NCC1(C(=O)NCC2(CO)CC2)CCCO1 41107,CC(C(=O)N1CC(F)CC1C(=O)Nc1ccc2c(c1)CCO2)C(F)(F)C(F)F 41108,C(=O)(C1CS(=O)(=O)c2ccccc21)NC1(C)CCN(C(C2(CC3CC3)CC2)=O)C1 41109,c1(C(C(=O)N(CC(C)C#N)C)NC(=O)C(F)C2CCC2)cn(C)nn1 41110,C1(C(N2CC(COC)(NC(=O)CC#N)C2)=O)CC2CCC1CC2(F)F 41111,N1(C(CN2N(C)C(=O)C2)=O)CC(O)(C2(CNC(=O)CNc3ccccn3)CC2)C1 41112,C1(CNC(CSC)=O)CCC2(CN(C(c3csc(-c4ccoc4)n3)=O)C2)O1 41113,c1(C(N2C(C)C(NC(c3cnsc3)=O)CC2)=O)cc(C(F)(F)F)ccc1N 41114,Cc1ccc2c(c1)CCC2C(=O)NCC(O)CCNC(=O)CCOCC(C)C 41115,C(CC(C)C)(C(=O)Nc1ccc(C#N)cc1)NC(C)=O.C1C(=O)NNC(=O)N1 41116,c1(C(=O)NCC(C(C(=O)NCc2ccc(C)c(C)n2)F)C)ccc2nccn2c1 41117,C1(COC)(CNC(=O)C(C)O)CCCN1C(=O)CC1CSCCS1.c1(C)ccccc1 41118,c1(CC)nc(C)n(C)c1C(=O)NCC1CN(C(=O)C=CSc2nc[nH]n2)CCO1 41119,c1(-c2ccc(OCC)c(CN3CC(O)CN3CC)c2)cc(OC)c(CC)cc1OC 41120,n1(CC)ncc(C(=O)NC2(OCCO)CCN(C(=O)Cc3cncnc3)C2)c1C 41121,C=CC1(C(=O)NC(c2cccc(O)c2)C)CCN(C(c2[nH]ccc(=O)c2C)=O)C1 41122,c1(OC)nc(C)ncc1C(=O)NCC(C)NC(C1CCC2CC2CC1)=O 41123,C1(CNC(=O)CC2CC=CC2)C2CCC1CN(C(C1CCC(O)CC1)=O)C2 41124,C1(OC)CCCCC1CC(=O)NCCC1CN(C(c2cncnc2C(C)C)=O)C1 41125,N1(C(c2cncc(OC)c2)=O)CC2CCC1C2NC(=O)CS(=O)(=O)N(C)C 41126,Cc1cc(F)cc(NC(C2CC2NC(=O)CCCn2ccnc2)=O)c1Br 41127,C1(NC(c2c(CC)scc2)=O)CN(C(c2ccc(C)cc2)=O)CC1N=[N+]=[N-].C1CC1 41128,C(=O)(CCC(=O)NCC1CN(C(=O)Cc2nccn2C)CC1OC)OCC 41129,C1(NC(C23C(C)(C)OCC2C3)=O)CCCC12CN(C(c1coc(C(F)F)n1)=O)C2 41130,c1(N(C)C)ccc(F)c(C(=O)NC2CN(C(=O)CCC3CC3(C)C)C(C)(C)C2)c1 41131,CCCC(CC1CCCC1)C(=O)NCC(C(C)(C)C)NC(=O)CSCC(N)=O 41132,Cc1ocnc1C(=O)N(CC(C)N(C)C(C1CC(CF)C1)=O)C 41133,C1(C(=O)NC(C)C=CC(=O)NCCC2CCCOC2)CCSCC1 41134,C1(C(C(=O)N(CCOC(C)=O)C)C)CCN(C(c2c(C)noc2C(C)C)=O)CC1 41135,CC1(C)CN(C(=O)CCc2ccc(Cl)cc2)CCC1NC(C1CC1CF)=O 41136,C#Cc1cnc(C(=O)NCC(O)CNC(C23CCCCN2CCC3)=O)c(C)c1 41137,C1(c2cn(C3CCN(C(C(C)OCC4CCCO4)=O)C3)nn2)COC(C)(C)O1 41138,Cn1ncc2nc(Cl)nc(NCC3CN(C(C4CCC4)=O)CC3C(F)(F)F)c12 41139,C1(CNC(C2C(C#N)C2)=O)CCN(C(=O)CSCc2cccnc2)CC1 41140,C(CN=c1[nH]c2c(c(=NC3CCCc4ccc(F)cc43)[nH]1)SCC2)NC(=O)NC 41141,C(CC(C)(C)C(=O)NCCC(C)CCNC(c1cncc(N(C)C)c1)=O)SC 41142,Cc1[nH]nc(C(=O)NCC2CC(CNC(c3ncccn3)=O)C2)c1C 41143,Cc1ncnc(C(=O)NCc2ccc(CNC(=O)C(C)C(C)(C)C)c(F)c2)c1C 41144,c1(CCC(=O)NC23CN(C(C4CCN(C)C4)=O)C(C2)C3)ccc(Cl)cc1Cl 41145,N1(C(C(c2ccc(F)cc2F)N(CCCCC)CCC)=O)CCC2COCC2C1 41146,N1(C(c2cnc(CCC)s2)=O)CCCC(CCC)(NC(c2nccn2C)=O)C1 41147,N1(C(C(=O)Nc2ncc[nH]2)=O)CCOC2(CCC(N=c3[nH]ncs3)CC2)C1 41148,C1(C(N2CC(N(C(c3c(C)nc(CC)s3)=O)C)C2)=O)CCCCC12CC2(F)F 41149,N1(C(C(c2ccc(Cl)s2)C)=O)CCN(C(=O)COCC2CC2)C(CC(C)(C)C)C1 41150,C1(C(=O)NC(CC)(C)CNC(c2cc([N+](=O)[O-])n[nH]2)=O)CC2CC1CC2(F)F 41151,C1(N(C(C)=O)CCNC(C)CCCCCC=O)CCc2ccccc2C1 41152,C(CN=c1[nH]c(=NCCOC(F)F)[nH]c2c1COC2)(c1ccccc1Cl)N(C)C 41153,CC1CNC(=O)CN1C(C1(NC(c2coc(C(N)=O)c2)=O)CC(F)(F)C1)=O 41154,C1(CN(C)C(C2(C3CC3)CC2)=O)CCN(C(=O)CCCC2OCCO2)C1 41155,C1(C(=O)NC2(C)CCN(C(C=CCOC)=O)C2)CN(C)C(=O)CCO1 41156,C1(CCC)CN(C(c2ccnc(S)c2)=O)CC1NC(c1cn(C)c(C)n1)=O 41157,CCC(CC)(CCNC(=O)C(F)C(C)C)NC(c1ccc(C2CCC2)cc1)=O 41158,Cc1ccnc(O)c1C(=O)NCCCC1CN(C(C2CCNC(=O)C2)=O)CCO1 41159,C1(C(=O)NCC(n2cc(C(c3ccccc3)O)nn2)C)CCCN1CC1CC1 41160,Cc1ncc(CCC(=O)N(CC(C)(C)CNC(C2CC2F)=O)C)s1 41161,Cc1coc(C)c1C=CC=O.C(=O)(CCCSC(C)(C)C)N(C)NC.C12(CC1)CC2 41162,C1(N(C(C2CC(CC)C2)=O)C)CCCN(C(=O)CCC2CCC(=O)NC2)CC1 41163,Cn1nccc1CN1CSCC1C(=O)NOCC(=O)OCC1CCCC1 41164,c1(C(N2CC(NC(C(C)NC(C)=O)=O)(CO)C2)=O)cc(N)c(C)cc1C 41165,CCC(C)C(C(=O)NC1CCCC1CNC(=O)CCCOC)N(C)C 41166,CN1CCC(C(N2CCN(C(=O)C=Cc3cnccn3)C(C3CC3)C2)=O)CC1=O 41167,C1(NC(C(C)=CC)=O)COC2C(NC(c3cnn(C)c3C(C)C)=O)COC12 41168,Cc1c(C(=O)NCC2CC(CNC(=O)CCc3cscn3)CO2)cnn1C 41169,CCCC(C)(C)CC(=O)NCC1CCN(C(C2C3CCCOC23)=O)C1(C)C 41170,c1(C(=O)NCC2C(CNC(c3c(SCC)nccn3)=O)C2)c(O)nnc(C)c1C 41171,CC1(C)CCC(C(N2CC(C(N)=O)(CNC(=O)CCC3CCCCO3)C2)=O)OC1 41172,c1(C(=O)NCC(N(C(C(CC)(C)O)=O)C)C2CC2)cc(Br)ccc1C1CC1 41173,C(=O)(CC1=CCCCC1)N1C(C(C)NC(=O)C2=CSCS2)CCCC1 41174,c1(C(=O)NC(C2CCCC2)CNC(c2nnc(C)s2)=O)cc(Cl)cc(F)c1F 41175,CC1C(NC(=O)Cc2csc(Cl)c2)CCN1C(=O)CCc1cccs1 41176,c1(CC)ncc(C(N2CCC(CCN(C)C(c3ncccn3)=O)CC2)=O)c(C)n1 41177,C1(CNC(C2CC2c2cccs2)=O)CC2(CCN(C(=O)C=C(Cl)Cl)CC2)CO1 41178,C(=O)(C(COCC)NC(=O)CCc1nc[nH]n1)NC1CC1.C1(=O)CN1CC 41179,N1(C(CN(C2CC2)CC)=O)CCC(C)(NC(c2nc(Cl)oc2C)=O)C1 41180,c1(N2CCCC(N(C)C(C3CC4CCC(C3)S4)=O)CC2)ncc(Br)cc1[N+](=O)[O-] 41181,c1(N(CC(C)OC)C)nnc(-c2ccccc2)n1CC(C)(C)c1cccs1 41182,C1(C(N2C(CNC(C=C(COC)C)=O)CC(C)(C)C2)=O)CC(C)(C)SC(C)(C)C1 41183,C(=O)(CCCC(=O)OC(C)(C)C)NCCC(C)CCNC(C1CC(=O)N(O)C1)=O 41184,C(=O)(C1=C(Cl)CC1)NC1(C)CN(C(C(C)CC2CC2)=O)C1 41185,C1(C(=O)NCCC(C)(C)NC(=O)C=C(Cl)Cl)CC(C(C)(C)C)=NO1 41186,c1(N2CCC(CC)C2)nc(=NCCc2c(C)noc2C)[nH]c2c1SCC2 41187,C1(C(C)C)N(C(=O)N(c2ccncc2Br)C)CC12CCC2 41188,c1(CNC2N(C(C=COCC)=O)CCC2)ccc(F)cc1O 41189,CC1CC(=O)NC1C(=O)NCCCNC(=O)CCOc1cccc(Cl)c1 41190,c1(C(=O)NCC2CCN(C(C3(C)ON=C(C)C3)=O)CC2O)cc(F)c(F)cc1O 41191,c1(OC)cc(C(=O)NCC2(OC)CN(C(c3cnccc3OC)=O)C2)cc(C)n1 41192,C12(C(=O)NCC(CNC(CCCOC(C)C)=O)F)CC3CC(F)(C1)CC(F)(C3)C2 41193,C(=O)(C1=C(C)OCC1)N1C(C(N(CC(CC)C)C)=O)(COC)C=CC1 41194,CC1CCCC(CN2CCC(NC(N3CCN(C(c4cccs4)=O)CC3)=O)C2)C1 41195,N1(C(C(C2CC2)OC)=O)CC(O)(CNC(C2(CO)CCC2)=O)C1 41196,c1(CC)n[nH]c(CC)c1NC(N1CCCC(c2n[nH]c(C3CCCCC3)n2)C1)=O 41197,Cn1ncc([N+](=O)[O-])c1-c1nc2ccccc2n1CCCCC(=O)O 41198,C1(C(=O)NCCN(C(=O)CN(c2ccc(Br)cn2)C)CC)COCC(C)(C)O1 41199,C1(NC(c2cn(CCNC(C3(CF)CC3)=O)nn2)=O)CCCC(F)C1 41200,N1(C(c2cc(C)c(F)cc2F)=O)CCC2C(CCN2C(C2COCCO2)=O)C1 41201,C1(NC(CCCc2cc(C)no2)=O)CC(N2CCOCC2)C1(C)C 41202,c1(CS(N)(=O)=O)ccc(CC(N)=O)cc1.c12cncn1CCNC2 41203,N1(C(c2c(C)con2)=O)CC2COCC2(C(=O)NC(C)CC2CCC2)C1 41204,C(=O)(CCCCCS(N)(=O)=O)N1C(C(C)(C)NC(C(C)O)=O)CCC1 41205,c1(C(=O)NCC2(C)CC(NC(C(CC)SC)=O)C2)oc2c(C)ccc(C)c2c1C 41206,C(CC(O)C(=O)Nc1cccc(NC(C2CCC(=O)N2C(C)C)=O)c1)SC 41207,CC(C)CC(C)(CNC(c1nccn1C)=O)NC(C1CCC(=O)N(C2CC2)C1)=O 41208,C1(C(=O)NC(CNC(c2cn(CC=C)nn2)=O)C(C)(C)C)CC2(C)CC1CO2 41209,c1(OC)ccc(CCC(=O)NC2CCC2NC(=O)COc2ccc(F)cc2)cn1 41210,N1(C(c2nn(CC)c(=O)cc2)=O)CCOC2CCN(C(C3(O)CC3(C)C)=O)CC12 41211,N1(C(C2(C)CCCCC2)=O)CC2(CNC(C3CC(F)(F)C3)=O)CC1CO2 41212,CC1C(=O)CCC1CC(=O)NC1(CCNC(c2coc(C3CC3)n2)=O)CCC1 41213,N1(C(C=CCN(CC(F)(F)F)C)=O)CC(F)(c2ccncc2)C1 41214,C1(CNC(CC2(CC(=O)OC)CCCC2)=O)CC(F)CN1C(=O)Cc1cc[nH]n1 41215,C1(C(N2CCCC(C)(NC(c3cc[nH]n3)=O)C2)=O)CC2(C1)CC21CCC1 41216,C1(NC(c2ccc(C(F)(F)F)cn2)=O)CC(CNC(C2CC(O)C2)=O)C(O)C1 41217,c1(C(=O)NC2CC(NC(c3c(C)nsc3)=O)C(O)C2)c[nH]c2c(C#N)cccc12 41218,c1(-c2nc(C(C)C3CC3)n(-c3cccc(Cl)c3)n2)ccc(Cl)cc1O 41219,Cc1cc(=NC(=O)c2cc(CNC(=O)C(C3CCCCC3)O)no2)[nH]n1C 41220,N1(C(CCOCCC)=O)CCN(C(C2OCCCC2(C)C)=O)C(CO)C1 41221,c1(CC)cc(F)ccc1CC(=O)N(CC(O)CNC(=O)C1=COCCO1)C 41222,Nc1cc(C(=O)NCC(CO)NC(=O)CC2CC3CC3C2)cc(C(F)(F)F)c1 41223,CCC1=C(C(=O)N2CCCCC2CCCNC(=O)CCCOC(C)=O)CCCO1 41224,C(C(CC1CC1)C(=O)Nc1cscc1C1CC1)NC(C(C)Cn1ccnc1)=O 41225,CCC(CC)C(C)C(=O)NCCOC1CCN(C(c2csc(C(=O)OC)c2)=O)C1 41226,N1(C(C(C)=C(CC)C)=O)CC2(NC(=O)CCc3cccc(Cl)c3)CC1C2 41227,Cn1ccc2ccc(C(N3CCC4(CCCC4NC(=O)C=C4CCC4)C3)=O)cc12 41228,c1(NC(CC2N(C(c3c(C)ncnc3)=O)CCC2)=O)cnc(Cl)c(Br)c1C 41229,C1(NC(C2C(C)(CC)C2)=O)CCC2CN(C(C3CC3(F)F)=O)CC2C1 41230,N1(C(C(C(C)C)S)=O)CCCC2(C1)CN(c1ccnc(Br)n1)CCO2 41231,C(=O)(C(C)S(=O)(=O)CCC)NC1C2CN(C(C3CC(C#C)(O)C3)=O)C(C2)CC1 41232,CC(=O)CCCCCCC(=O)OCC1CCCC(F)C1 41233,c1(NC(Cc2n(C)nnc2)=O)cccc(C2(NC(C34COCC3C4)=O)CC2)c1 41234,CC1(C)C(NC(=O)C2=C(Cl)CCC2)CCN1C(=O)CCC1CCCO1 41235,N=c1[nH]c2c(s1)CCCC2C(=O)N1CCCC(F)(CNC(=O)C(N)=O)CC1 41236,c1(-c2cc(C(=O)OCC)n[nH]2)ccc(NC(c2ccnn2C(C)C)=O)nc1 41237,C1(NC(C(C)NC(=O)OC)=O)CC=C(C(=O)Nc2cnc(C(C)C)nc2)C1 41238,C1(C(N(CC(CC)NC(C2(CCCC)CC2)=O)C)=O)CCCC2(CCC2)C1 41239,C#Cc1cccc(NC(C2CC23CN(S(=O)(=O)CCOC)C3)=O)c1 41240,CC1CN(C(c2cn(CCNC(C3CNC(=O)N3)=O)cn2)=O)CCO1 41241,C1(CC(C)NCc2cn(C)nc2Br)CCCN(C(=O)OC(C)(C)C)C1 41242,c1(C(N2CCCC(O)(CNC(=O)CC3(O)CCCC3)C2)=O)cc2n(n1)CCOC2 41243,Cn1cc2cccc(NC(C3CCC4(CN(C(=O)CCC(N)=O)C4)O3)=O)c2n1 41244,n1(C(C)F)cc(-c2noc(C3CCCN3C(=O)OC(C)(C)C)n2)cn1 41245,C(=O)(C(C)(C)CC(C)C)N1C2C(NC(c3c(Cl)ccc(OC)n3)=O)C(CC2)C1 41246,c1(C(=O)NCCC2(CNC(=O)CC3CCOC3=O)CC2)cnc2ncnn2c1O 41247,N1(C2CCN(C(c3c(C)n[nH]c3)=O)C2)CCN(C(c2cccnn2)=O)CC1 41248,C1(C)(SC)CCCO1.C(C(C)C)N(C(C)=O)CCN(C)C 41249,N1(c2c(OC)c(Cl)ncn2)CCC(C2CC2)(CNC(c2cnoc2C(C)C)=O)C1 41250,C1(OC)CCC2(C(=O)NC(C)(C)C(=O)NC(CO)CCC3CC3)CC12 41251,N1(C(c2ccc(C)o2)=O)CCN(C(c2c(Cl)cccc2I)=O)C(C#N)C1 41252,N1(C(COC(C)=O)=O)CC2(CCC(CNC(c3cccc(Cl)c3C(F)F)=O)O2)C1 41253,N1(C(c2c(C)c(N)cnc2)=O)CC2CC(NC(=O)CC3(N(C)C)CCC3)C(C2)C1 41254,c1(NC(C(=O)NC(c2ccc(OC)cc2)CC#N)=O)cc(C)ccc1C 41255,c1(C(=O)NC2CN(C(C(C(C)C)OC)=O)CC2SC)cncc2c(O)nccc12 41256,C1(N(C(=O)CSCC2CCCCO2)CC)CCCN(C(=O)C(C)(C)O)CC1 41257,N1(C(CS(N)(=O)=O)=O)CCC(SCN2CCCC2=O)CC12CC2 41258,C1(O)(C(=O)NCC2C(C(=O)NC(C)Cc3ccccn3)C2)CCOCC1 41259,c1(C(N2CC(C)(C(=O)OC)OCC2)=O)ccc2ccccc2n1 41260,N(C(=NCCN1CCCC1)NCC1CCCC1C)Cc1c(OCF)ccc(Cl)c1 41261,N1(C(CCOCC#C)=O)CCC2(CCN(C(C3(n4cc(Cl)cn4)CC3)=O)C2)C1 41262,C1(CNC(C(=O)N(C)Cc2ccc(CO)cc2)=O)CCC(C)(C)CC1 41263,CC1CCN(C(c2sccc2C2CC2)=O)C(CNC(c2cc(=O)cc(Cl)[nH]2)=O)C1 41264,C1(C(N2C3CC(NC(C(C)(C)N(C)C)=O)CC2CC3)=O)Cc2ccc(F)cc2O1 41265,c1(C(N(C)CC2N(C(CCCCOCC)=O)CCCC2)=O)nc2c(s1)COCC2 41266,c1(CCC=C)ccc(C(N2CC(CC=C)(C(=O)NCC3CNC(=O)C3)C2)=O)cc1 41267,C(=O)(C1=CC2CCCCCC12)N(CCNC(CS(C(C)(C)C)(=O)=O)=O)C1CC1 41268,c1(C(=O)OCC)sc(NC(C23CC(NC(=O)CCCOC)(C2)C3)=O)c(C#N)c1C 41269,Cc1cc(C(=O)NC2CCC(N3CCOCC3)C2)nc(C)c1 41270,N1(c2cc(Br)ncn2)CCN(Cc2cc3cccnc3[nH]2)CC12CC2 41271,c1(OC)ncc(-c2nc(C)c(NC(c3nccc(Cl)c3Cl)=O)s2)cc1C 41272,C1(C(=O)NC2CC(NC(CN3CCC(C)CC3)=O)CC2O)SC2C=CC1CC2 41273,N1(Cc2cn(CC(CC)O)nn2)CCOC(C)(CCO)C1 41274,C(=O)(N=c1[nH][nH]c2cc(C#N)ccc12)C1CC(N(C)Cc2ccnc(Cl)c2Cl)C1 41275,c1(NC(C23C(CN(C(c4ccccc4C(F)(F)F)=O)C2)C3)=O)cc(Br)cnc1Br 41276,C12(NC(C(CSC)C)=O)CC1CN(C(=O)Cc1ccnn1C)C2 41277,N1(C(c2ccc(SCC=C)cc2)=O)CCN(C(=O)C(N)=O)CC1C1CCC1 41278,c1(C(=O)NC2C(CNC(=O)CCC3CCCC(=O)N3)C2)cccc2[nH]nc(O)c12 41279,C(CCC(=O)N1CCCC1C(C)(C)NC(C1C=CCCC1)=O)N(C(=O)OCC)C 41280,CCC(CCC(=O)NC1CC12CC(OC)C2)NC(c1cncn(C)c1=O)=O 41281,C(c1cc2ccccc2o1)=CC(N1CC(CCNC(C(C=C)(C)C)=O)C(C)C1)=O 41282,C(CCCC(CO)NC(C1(N2CCCC2)CC1)=O)NC(CC(CC)SC)=O 41283,CCCCCC(F)C(=O)N(CCC(C)(C)NC(c1ccsc1SC)=O)C 41284,C=CCC(C)(C)C(=O)N1CCCOC(CNC(C2CC2C(C)O)=O)C1 41285,C1(C(N(CCC(=O)NC(C)CCN(C)C)CC)=O)CCCSC1 41286,c1(CC)sc(C(=O)NC(C)CCNC(c2nnsc2C)=O)cc1Br 41287,C1(C(=O)NCC(C23CCC(CC2)C3)NC(C(C(C)C)F)=O)CN2CCN1CC2C 41288,CC1(CNC(=O)Cc2cc(Br)cs2)CC(NC(=O)Cc2ccon2)C1 41289,N1(C(C(C)CC(N)=O)=O)CC2CC(NC(=O)C=Cc3cnn(C)c3)CC1C2 41290,C(CSC)(C(=O)NCc1cc(C(=O)NCC(C(C)C)OC)no1)OC 41291,C1(C(N(CCCCNC(c2cc(C)c(O)nn2)=O)C)=O)CCc2ncsc2C1 41292,C(=O)(CS(=O)CCC(F)(F)F)NCCc1c(CNC(CCC(N)=O)=O)nco1 41293,C=CCCCCC(C(=O)NCc1cccc(Br)c1)N1CCC(O)C(C)(O)C1 41294,O(NC(=O)CC(CC=C)NC(=O)CC1CCOCC1)CC(=O)OCC#C 41295,c1(CCNC(C(C)(C2CC2)OC)(C)c2nnnn2C)ccc(S(N)(=O)=O)cc1 41296,CC1CN(C(=O)CCOc2ccc(F)cc2)CCCN1C(=O)C(N)=O 41297,c1(C(=O)NC(CC)CN(C)C(c2ccsc2S(N)(=O)=O)=O)cnn2cccnc12 41298,C1(CC(=O)OCC)NC(=O)N(CC(C)OC(F)F)C1=O 41299,C12(CNC(C3N(C)CCCC3)=O)CCC(CC1)CN2C(c1cc(Cl)cnn1)=O 41300,C(=O)(C1=C(Cl)CCOC1)NC1CCN(C(CCC2C(C)=NOC2=O)=O)C(C)C1 41301,CC(C)C(C(=O)NCC1CN(C(C23CCC(C2)OC3)=O)C1)n1cccc1 41302,C1(C(N(C(CCC)C)C)=O)OCCC1NC(C1CN(C(N)=O)C1)=O 41303,C1(NC(CSC)=O)CCN(C(c2ccc(CC#N)cc2)=O)C1C 41304,N1(C(=O)OC(C)(C)C)CC2CCC1C2C(N1CC(CNC(=O)C(N)=O)C(C)C1)=O 41305,C1(C(N(C)CCc2cc[nH]n2)=O)CC2CC1CN(C(=O)Cn1cnnc1)C2 41306,C=CCCC(C(=O)OC)NC(C1CN(C(c2cnc(O)cc2C)=O)CC1CC)=O 41307,C1(CNC(CN(C)C)=O)CN(C(c2ncc3ccccn23)=O)CCC12CCOC2 41308,CC1(C)CC(NC(=O)C(N)=O)CCN(C(c2ccnc(F)c2O)=O)C1 41309,C1(C(=O)NCCCC(C)NC(C2CC(=O)CC23CCC3)=O)CC2(CCCC2)CO1 41310,C(=O)(C1CCCc2c[nH]nc21)NC(C)CNC(=O)CNC(=O)C(F)(F)F 41311,N1(C(c2ccn(C)n2)=O)CC(Nc2ncc3ccsc3n2)CC(C)(C)C1 41312,CC1(CCC(=O)NCC2CCC2NC(=O)CCCc2csc(=N)[nH]2)CCC(=O)N1 41313,CC1(NC(C2(C3CC3)CCC2)=O)CCCN(C(=O)CSc2ccc(Cl)cc2)C1 41314,c1(C(N2CCCC(n3cc(C(C)OC)nn3)C2)=O)cc(O)nc(Cl)c1 41315,C=CCC(CNC(C1CCSCC1)=O)NC(=O)C(C1CC1)SC 41316,C1(CNC(CN2C(C)CC2)=O)CN(C(=O)Cc2ccnc(C(F)(F)F)c2)CC1C 41317,C(=O)(N1CC(n2cc(CC3(O)CCC3)nn2)CO1)C1N(C)CSC1 41318,c1(OC)cccc(C(=O)OCC2CC(NC(=O)OCc3ccccc3)C2)c1C 41319,N1(c2nccc(C(=O)OC)n2)CCC(C)(C)C(CNC(=O)CCC2CCCO2)C1 41320,CC1(C)Cc2cccc(S(=O)(=O)NCCn3ccc(O)nc3=O)c2O1 41321,C1(O)(C(C)NC(=O)CCOC2CC2)CCN(C(C2(c3nccn3C)CC2)=O)C1 41322,CN=c1[nH]c(C(=O)NCC2CN(C(=O)CC3CC(CF)C3)CC2C)cs1 41323,c1(C(C(=O)NC(C)C(CO)NC(=O)C=CCN2CCCC2)O)ccccc1F 41324,N1(Cc2c3ccc(OC)cc3ccc2)CCC(N=c2[nH]cnc3cc(I)sc23)C1 41325,c1(CN(C(C=CC(=O)NC(C2CCCC2)C)=O)C)ccccn1 41326,C(=O)(C1=CC2(CCOC2)C1)N1C(CNC(Cc2cc(C)[nH]n2)=O)C(C2CC2)CC1 41327,c1(C(N2CC(F)(C(=O)NC3(c4nc[nH]n4)CC3)C2)=O)ncccc1F 41328,C1(CNC(CC2(C)CC2(F)Cl)=O)CCC(CNC(C2(F)CCCCC2)=O)CC1 41329,c1(CC)cc(Cl)ccc1C(=O)NCC1(CNC(=O)C(C(C)C)NC)CCCC1 41330,C(c1ccc(OC)cc1OC)=CC(=O)NCCNC(CCCOCCOC)=O 41331,C(=O)(C(CC(C)C)N(C)C(c1cc(CO)on1)=O)N1CCC(C(CC)CC)C1 41332,Cc1cc(C(=O)NC2CN(C(=O)CC3CCCN3C)CC2F)c(O)nn1 41333,N1(C(C(C)OCC=C)=O)CC2CC(O)C1C2NC(c1cc(C)sn1)=O 41334,C1(NC(c2scc(C(=O)OC)c2)=O)CCC(CNC(C2(C3CC3)CC2)=O)CC1 41335,C12(CNC(CCOCC)=O)CCC(C1)N(C(c1ccc(C(F)F)nc1O)=O)C2 41336,N1(C(c2ccc(OC)c(O)c2)=O)CC2OCCN(C(=O)COC3CC3)C2C1 41337,c1(CC(N2CC(C(=O)Nc3n(C)nc(C)c3Cl)NCC2)=O)ccc2c(c1)CCO2 41338,c1(SC)ccc(C(N2CC3CC2C3C(=O)NCCS(C)(=O)=O)=O)cc1 41339,C1(C)(NC(C2C(NC(CCCNC(C)=O)=O)COC2)=O)C=CCCC1 41340,N1(C(CC(=O)NCC)=O)CCC=C(CNC(=O)C(C)CC2CCC2)C1 41341,N1(C(c2c(C)n[nH]c2)=O)CC2CCCCN2CC1CNC(c1cc(O)ncn1)=O 41342,C1(CC(=O)NCc2nc(C(N3CC(n4ccnc4)C3)=O)co2)COCCOC1 41343,C1(CNC(CN(C(C)=O)C)=O)CCC(C)(C)CN1C(C1CCOC1)=O 41344,C(C)(C(=O)NC1COCCN(C(c2cc(F)ccc2Cl)=O)C1)(C(C)C)OC 41345,N1(C(c2cc(C)ncc2)=O)CCN(C(=O)C(C2CCCCC2)O)C(CC2CC2)C1 41346,c1(N2CC(C(=O)Nc3c(C(=O)OCC)nc[nH]3)C2)ncc2cc(Br)cnc2n1.CCO 41347,c1(C(=O)NC(CNC(=O)C=Cc2cn[nH]c2)C2CCC2)c(F)cccc1F 41348,c1(CNC(C(=O)OC)(C)Cc2ccccc2F)ccc(S(C)(=O)=O)cc1 41349,N1(C(C#CC(C)C)=O)CC2(C1)CN(C(C1CCSC1)=O)CCO2 41350,CC(CCC(=O)NCC(c1cccnc1)O)NC(C1(C)CCC1)=O 41351,N1(C(C2CC(NC(C)=O)C2)=O)CC(NC(=O)Cc2ccon2)CC(O)C1 41352,C(=O)(CCS(=O)(=O)C(F)(F)F)NC1CCN(C(c2cn(CCC)nc2)=O)C1 41353,c1(C(=O)NC2C(NC(C3(C(C)=O)CC3)=O)CCCC2)ccc(F)c(C#N)c1 41354,C1(Cl)(C(=O)NCCN(C2CCCC2)C(C2C(CCC)C2)=O)CC12CCOCC2 41355,CC(C(C)C(=O)N(C)CC1CN(C(C23CCC(CC2)C3(C)C)=O)C1)S(C)(=O)=O 41356,O=C1Nc2ccc(C(N3CCCC3(C)CNC(=O)CC3CC=CC3)=O)cc2CO1 41357,C(CCN=c1[nH]c(N2CCOCC3(CC3)C2)nc2ccccc12)SC 41358,CN1CCN(C(C2CC2NC(=O)CC2CCN(C3CC3)CC2)=O)CC1CCO 41359,c1(C(=O)NC2C(NC(c3n(OC)cnc3C)=O)COC2)cnc(O)n(C)c1=O 41360,c1(CCCC)cc(F)c(CC(=O)NCC2(N)CC(OCC)C2)cc1Br 41361,C1(CC=C)(C(=O)NCC2(F)CC(NC(c3coc(C(F)F)n3)=O)C2)CC=CC1 41362,c1(C(N2CC3C(CNC(c4cn(CC)nn4)=O)(C3)C2)=O)ncc(F)cc1F 41363,N1(C(c2cnn(C)c2Cl)=O)CC2=C(C1)CN(C(=O)CP(C)(C)=O)C2 41364,C1(NC(c2c(C)nc(C)o2)=O)CCN(C(=O)Cc2cc[nH]n2)C12CCC2 41365,C1(OC)CC(NC(=O)CNC(=O)OC(C)(C)C)CN(C(=O)CC2(C)CCCO2)C1 41366,C1(NC(COCCC)=O)CC2CCCC(C1)N2C(C1CC12CC2)=O 41367,N1(C(c2c(C)cc(OC)c(OC)c2)=O)CCN(C(=O)C(N)=O)CC(CO)C1 41368,Cc1cc(CC(=O)NC(C)(C)CNC(C2CCCC(C)(C)O2)=O)ccc1O 41369,c1(OC)cc(F)ccc1CC(=O)N(CC(C)NC(c1nccnc1C(N)=O)=O)C 41370,c1(C(N2CCC(NC(C(C)c3ccsn3)=O)C2)=O)c(N)cc(F)cc1Cl 41371,C1(CC(=O)NCCOCCN(C(Cc2cn(CC)nn2)=O)C)CCCCC1F 41372,c1(C(N2CC(CC)C(OC)CC2)=O)ccc2cnn(CCOC)c2c1 41373,C(=O)(C1CC(=O)Nc2ncccc21)N1CCCC(CNC(c2c(C)c[nH]n2)=O)C1 41374,N1(C(C=CSC)=O)CCOC(C)(CNC(=O)Cc2cccc(C(C)=O)c2Cl)C1 41375,N1(C(c2c(CC)c[nH]n2)=O)CCN(C(=O)C(C(C)O)N(C)C)C2(CC2)C1 41376,c1(OC)cccc(Br)c1C(=O)NC12CC1CN(C(=O)C(=O)NCC(F)F)C2 41377,CC1C(=O)CCC(C(=O)NC2(c3ccc(F)cc3)CNC2)C1(C)C 41378,C=C1CC(CC(=O)NCC(C)(C2CC2)NC(=O)Cc2ccsn2)C1 41379,N1(C(=O)CSc2ccccc2)CCC2CC(CNC(C34CC(C3)C4)=O)CCC2C1 41380,C#CCCC(C(=O)NCC1(O)CCC(C)(C)C1)NC(C1CCO1)=O 41381,c1(C(N2CC(OCCNC(C3(C)CC=CC3)=O)C2)=O)ccc2c(c1)C(=O)CCN2 41382,c1(C(=O)Nc2nccc(N3CCC(OC)C3C)c2)ccccc1I 41383,CCC(C)C(O)C(=O)N1CCCC1C1CCN(C(c2c[nH]c(=NC)s2)=O)CC1 41384,c1(CNC(=O)NC(C)CC#N)ccccc1OCc1cccnc1 41385,c1(C(N2CCC(CNC(C(C)SCC)=O)C2)=O)[nH]c2c(c1C)C(=O)CC(C)(C)C2 41386,CC(C)CC(C(=O)NCc1ccc(C(=O)NCC(=O)N(C)C)cc1)C(N)=O 41387,CCCC(C(=O)NCC1(NC(=O)C(C)NC(N)=O)CCCC1)OCC 41388,Cc1c(Cl)ccc(C(N2CCOCC2c2cn(C3CCCC=C3Br)nn2)=O)c1N 41389,N1(C(c2cccc(NC)n2)=O)CCC2CCN(C(=O)Cc3sccc3Cl)C2C1 41390,CCCC(CNC(=O)Cn1cc(CNCC2(OC)CC2)nn1)OC 41391,C(=O)(CC(F)(F)C(F)F)NCCN(C(C(CC#C)O)=O)C(C)C 41392,C12(C=O)CC(NC(=O)C)(C1)C2.C1(O)(CC(=O)NC2C(C(C)(F)F)C2)CCOC1 41393,C1(NC(CCSCCC)=O)CC2CC1CN(C(c1ccnn(C)c1=O)=O)C2 41394,C1(CNC(CCCCC)C2CC2)CC2(CCC2)C(=O)O1 41395,c1(C(=O)NC2CN(C(C3(O)C(C)(C)C3)=O)CC(F)C2)cc(F)c(F)cc1F 41396,C1(NC(=O)COc2cccc(C(F)(F)F)c2)CC2CCC1N(C(C1CC(O)C1)=O)C2 41397,C12(C(N3CC(=CC)C3)=O)CC(CN(C(C3CCC(C)=C(C)C3)=O)C1)C2 41398,CC(C)CC(C(=O)NC(c1cccnc1O)C)NC(C1CCCC1C1CC1)=O 41399,C(=O)(CC(O)CNC(=O)COC1CCC1)N(C(C1(C)CC1)C)C 41400,CC1CC(C(N2CCC(C(=O)NCCC(=O)N(C)C)CC2)=O)CCO1 41401,C1(C(N(CCCNC(C(CC=CCC)C)=O)CC2CCCC2)=O)CCC(C)=C(C)C1 41402,C12(CC(N3CC(NC(c4c(C)nn(C5CCOC5)c4)=O)C3)=O)CCC(CC1)CC2 41403,N1(C(C(C)=CC)=O)CCN(C(C2CC3CCC2O3)=O)C(c2ccc(F)c(F)c2)C1 41404,C=C=CC(C)C(=O)NC1CC1CNC(=O)Cc1cc(Cl)sc1Cl 41405,C1(NC(CSCC#C)=O)CCC(N(C)C(c2cnc(-c3cnn(C)c3)s2)=O)C1 41406,c1(COC(C)C(=O)NC2(CN(C)C(C3CS(=O)C3)=O)CC2)ccccc1 41407,S(=O)(=O)(c1ccc(NC2CCN2C2CCCCCC2)c(F)c1)N(C)CCC1CC1 41408,C(=O)(C1=NOC2(CCCN(C(=O)C(=O)NCCc3cccc(Cl)c3)C2)C1)OC 41409,Cc1cccc(NC(C2OCCC2NC(c2cnsc2C)=O)=O)c1C 41410,C(=O)(C1CCc2cccnc21)N1CCCC(NC(C(CCC)(C)CC)=O)(CO)C1 41411,c1(C(N2CC3C(N(C(C4C(C)CCO4)=O)C)C3C2)=O)cccc2c1OC(C)(C)C2 41412,c1(OC)cc(Br)ccc1C(=O)N(CC(C)NC(c1cc(F)ccc1C)=O)C 41413,CCCCC(CNC(c1c(C2CCC2)noc1C)=O)NC(=O)C(C)OCC1CC1 41414,Cc1cc(=NCCCc2nnc3ccccn23)[nH]c(=NCc2cccs2)[nH]1 41415,c1(OC)cc(N)ccc1C(=O)NC1CC(C)(NC(C2CCCCC2O)=O)C1 41416,N1(C(C(C)C2CC(NC(C3(c4ccccc4)CC3)=O)C2)=O)CCCCC1CN(C)C 41417,C#Cc1ccc(F)c(C(=O)NCC2CC(OC)CN2C(c2cnn(C)c2N)=O)c1 41418,CCC(CCOC)C(=O)NC1C=CCN(C(=O)CC(C)(F)F)C1 41419,C1(C(N2CCC(NC(CCc3nc(C)sc3)=O)C2C)=O)CCc2nc[nH]c2C1 41420,c1(CCN(CCCNC(=O)OC(C)(C)C)C(N)=O)ccccc1.C1(=O)C(=O)NN1 41421,N1(C(c2cc(C)c(F)nc2)=O)CCc2ccccc2C1CNC(=O)C1=COCC1 41422,C1(C(N2CC(NC(CCCN(C(C)=O)C)=O)C(C)C2)=O)CCCCCS1(=O)=O 41423,CC1(C)CCN(C(C2CCC(F)C2)=O)CC1CNC(c1cc(C2CCC2)on1)=O 41424,c12c(nnn1C)CCC(=O)NN(CC(C)O)C2=O.C(C)(=O)NCC 41425,c1(C(=O)NCC(CC)(C)NC(=O)COCC2CCOC2)ccc(CO)c(Cl)c1 41426,N1(C(C(C)(c2ccccc2)N(C)C)=O)CCC2(CCC(=O)NC2)C1 41427,Cc1ccc(F)c(CN(C2CC(C)(C)C2CC(C)C)C(=O)OC(C)(C)C)c1 41428,C(=O)(C1OCCc2c(O)cccc21)N1CC2N(C(C=C(CCC)C)=O)CC(CC2)C1 41429,C1(CC)CCN(C(=O)C(CC)N(C2CCCC2)C(c2ccc(C(=O)OC)[nH]2)=O)CC1 41430,C#CC1(NC2CCn3nccc3C2)CC2(CCCC2)C1 41431,c1(NC(CCSCCCC)=O)cccc(NC(c2cc(Br)sn2)=O)c1 41432,Cc1ncc2n1CCN(C(C1CCCC1CNC(C1(C3CC3)CC(=O)C1)=O)=O)C2 41433,C(=O)(CC(C)(C)CC(F)F)N1CC(NC(Cc2c(C)cc(C)nc2O)=O)C(F)C1 41434,C1(C(=O)NCC2N(C(c3c(C)nc(C4CCC4)o3)=O)CCC2)CCN(C)S1(=O)=O 41435,N1(C(C2(CC)CCC2)=O)CCCC(C2CC2NC(c2ccccc2O)=O)C1 41436,CN1CC=C(CC(=O)N2CCC(CN(C)C(C3Cc4ccncc4N3)=O)C2)CC1 41437,C12(C(=O)NC3C(OC)CN(C(=O)CCS(C)=O)C3)CCC(C(F)(F)F)(CC1)CC2 41438,N1(C(c2cnn(C(CC)C)c2C2CC2)=O)CCN(C(C2CC23CCC3)=O)CC1C 41439,C(CCCCC(C)C)NC(N(CC)CC1CCCCN1C(C)=O)=O 41440,Cc1cc(C)c(C(=O)NCC2(C(C)NC(c3cocc3C)=O)CC2)c(O)n1 41441,C1(NC(CC)=O)CC2CCC(C1C)N2C(c1cnn(C)c1C(F)F)=O 41442,C1(NC(c2cc(CNC(CC3C(C)(C)C3)=O)on2)=O)CCC(C#N)CC1 41443,Cc1ccc(F)c(CC(N2CC(CNC(c3nnsc3C)=O)C3(CC3)C2)=O)c1 41444,N1(C(=O)OC(C)(C)C)CCC(n2cc(CCNC(C(N)=O)c3ccc[nH]3)nn2)C1 41445,C1(CNC(=NC)NCCCCOC)CC2(CCOCC2)O1 41446,CC(N=[N+]=[N-])C(=O)NC1(CNC(C2COCCOC2)=O)CCCC1 41447,CCCCCCC(CC)(CC)C(=O)NC1CC(NC(C2CC3(CCCO3)C2)=O)C1 41448,C1(CC(=O)NCCC(C)NC(c2cscc2C2CC2)=O)COC(C)(C)C1 41449,CCC(CNC(c1ccncc1Br)=O)(CC)NC(=O)COCc1nc[nH]n1 41450,N1(C(C(CC)c2ccccc2)=O)CCCC2(CCCCN2C(C2CCOC2C)=O)C1 41451,Cc1ncc(C(=O)NOC(CC(C)C)C(=O)NCCN(C2CCCC2)C)c(=N)[nH]1 41452,C12(CNC(C3(C)CC3)=O)CC1CN(C(=O)CCCCc1cnn[nH]1)C2 41453,c1(C(N2C(C(N3CCC=C(F)C3)=O)CCC2)=O)cccc2cc[nH]c12 41454,C1(CNC(C2(CCCC)CCCC2)=O)CC(OC)CN1C(=O)Cc1cccs1 41455,c1(NC(c2c(CCC)occ2)=O)cccc(NC(=O)C(C(=O)OC)OC)c1 41456,N1(C(C(CC#C)O)=O)CC2CCC(CNC(c3nc(C4CC4)cs3)=O)(C2)C1 41457,C1(NC(CC(CN(C)C)O)=O)CN(C(=O)COCc2ccccn2)CC12CCC2 41458,CC1C(C(=O)N2CCC(C)(C)C2C(=O)NC2CC(C(C)(C)C)C2)=NOC1C 41459,C1(C(=O)NCC(CC)(CC)NC(C2C3COCC23)=O)CC12CCCCCC2 41460,CCC(CC)C(=O)NN(C(=O)COc1ccccc1C(C)C)C.C12(CC1)CN2 41461,c1(CNC(C(=O)N(CCCN)CC)=O)cccc(NS(C)(=O)=O)c1 41462,Cc1cc(N)c(C(=O)NCC2(CNC(c3cnc(N(C)C)o3)=O)CC2)cc1F 41463,C(=O)(CC(CCCC(C)C)NC(C1(NC)CC2(C1)CC1(CC(F)(F)C1)C2)=O)OCC 41464,CC1(NC(=O)CCCNC(C2(C(F)(F)F)CC2)=O)CCCOC1 41465,N1(C(C=CC)=O)CCC(NC(c2cccn(C)c2=O)=O)C(c2ccccc2)CC1 41466,c1(CCC)nc(C)c(C(=O)NCC2CC(NC(C3CCOC3(C)C)=O)C2)o1 41467,CCCCC(C)C(=O)N1CCC(C(=O)Nc2ccc(Cl)cc2O)C1C 41468,N1(CC)CCN(C(C23CC(CO)(CN2C(C2(C)CC(C)=NO2)=O)C3)=O)C(C)C1 41469,N1(C(C=CCC)=O)CC(C)N(C(c2cc(CC(C)C)c[nH]2)=O)CC1C 41470,C1(C(=O)OCC)CN(C(=O)CC2COCCN2CC(F)(F)F)C2(CCC2)CO1 41471,N1(C(CCc2cccc(C)n2)=O)CCC2COC(CC(=O)N(C)CCN(C)C)C2C1 41472,N1(C(C)=O)CCCC1C(=O)N(C1CC1)CC1CCCN1C(c1csnn1)=O 41473,C(=O)(C(O)CC(C)(C)C)NCCC(C(=O)NC1(COCCN(C)C)CC1)OC 41474,N1(C(c2nc(NC)nc(O)c2)=O)CCOC2CN(C(C3CC=CCN3C)=O)CC12 41475,c1(CC)ccc(C(=O)NC2CCN(C(=O)C#CC3CC3)C23CC3)cc1OC 41476,C(=O)(C(C)(O)Cn1ccccc1=O)NC1C(NC(c2ccc(OC)s2)=O)C1 41477,C=C(Br)CC(C)(C)C(=O)ON1C(Cc2cn(Cc3noc(C)c3C#N)nn2)CC1 41478,C1(O)(CNC(CC(C)F)=O)CC2CCC(C1)N2C(c1cc(F)ccc1N)=O 41479,C1(NC(C(C)NC(CC)(C)C)=O)C=CCN(C(=O)CCC2CC2(F)F)C1 41480,C(=O)(C(C)NC(C1CC(=O)C1)=O)NCCN(CCC)CCC 41481,n1(C2CCC(C(C)C3CC3)C2)cnc2c(N3CCC(S(N)(=O)=O)CC3)ncnc12 41482,Cn1cc(NC(c2nnnn2-c2ccccc2)C=CC2CCCC2)c(C#N)n1 41483,c1(C(=O)NCC2COCCN2C(=O)C(F)CC2CC2)nc[nH]c2nccc1-2 41484,C1(CC(=O)OC(c2ccccc2Cl)c2nc(C)on2)COCCN1C 41485,C1(CN2C(C(=O)O)CC(CC)C2)CC2CC(=O)C1C2 41486,C1(C(=O)NCc2snnc2C2CC2)CSCCN1C(=O)CCCCC1CC1 41487,CC1CC(NC(=O)COc2ccccc2)CN1C(c1cc(F)c[nH]1)=O 41488,c1(C(=O)NCC(CN(C(c2cnc(C)n2C)=O)C)(C)C)cnc2ccc(F)cn12 41489,c1(NC(c2c(Br)cc(C)s2)c2nnnn2CCCF)cc(Cl)cc(Cl)c1[N+](=O)[O-] 41490,C(=O)(CCCCC1CC1)N(CCC(=O)N)C.C(CCCC1CCCC1)C(C1CC1)O 41491,CC1=CCC(C(=O)NC2CC(C)(NC(=O)CC(C)(C)O)C2)CC1 41492,c1(C(c2cn(CCC(=O)NCC(C)(C)[N+](=O)[O-])nn2)O)c(Br)cncc1Br 41493,c12ccnc(c1)C(=O)NC2.C1(CNC(C2(OC)CCOC2)=O)CCOC(C)C1 41494,C(C)(CN=c1ccnc(NCc2nnc(O)n2C)[nH]1)(C1CC1)OC 41495,Cn1ccc(=NC(=O)C2CC(O)CN2C(c2ccn(C(C)(C)C)n2)=O)[nH]1 41496,C1(CNC(=O)Cn2cnnc2O)CN(C(c2cccc(F)c2F)=O)CC12CC2 41497,c1(OC)ccc(F)c(F)c1C(N1CCN(Cc2cc(C(N)=O)nn2C)CC1C)=O 41498,C(=O)(CCCCC(=O)N(c1ccc(CNC(=O)CCCC(C)(F)F)cc1)C)OC 41499,Cn1cc(C(N2CCC3(CC(NC(=O)OC(C)(C)C)C3)C2)=O)c(=O)[nH]c1=O 41500,c1(C(=O)NCC(CO)NC(C2CC23CCC3)=O)nnc2c(F)cccc2c1O 41501,C(=O)(C(C)(O)COC)N(C)CC1N(C(CC(=O)NC)=O)CCC1 41502,CCCCC(O)CCC(=O)NCC(C)(C1CC1)NC(C1CCCCN1N=O)=O 41503,C1(C)(C(=O)NCC2C(NC(CCC(C)(C)C)=O)CCC2)CC2CCC(C1)S2(=O)=O 41504,Cc1cc(C(C)C)ccc1NC(c1cc(O)cs1)=O 41505,C(=O)(CC1=CCN(C)CC1)N1C(CNC(C2(C(=O)NC(C)C)CC2)=O)COCC1 41506,C1(C#N)(C(=O)NCCCOCCCNC(c2ccc(CC)cn2)=O)CCCCC1 41507,C1(NC(=O)C=CC=C(Cl)Cl)CC2C(NC(c3ccc(Br)s3)=O)C2C1 41508,C1(CC(=O)NCC2OCCN(C(c3c(C)cn(C)c3)=O)C2)COCC(C)(C)O1 41509,CCCC(C)C(=O)N1CCC(C(C)(O)CNC(=O)C=Cc2ccc(SC)s2)CC1 41510,N1(C(CNC(C)=O)=O)CC2CS(=O)(=O)CC2(CNC(c2cc(Cl)cs2)=O)C1 41511,C1(NC(COCC)=O)CCCN(C(=O)CC(CC#N)c2ccccc2)CC1 41512,C1(c2nnnn2C)(NC2CCC(C)C2)CC2CCC(C1)S2(=O)=O 41513,C1(CC)(CNC(=O)C(CO)NC(N)=O)CCN(C(c2cccn2C(C)C)=O)CC1 41514,c1(OC)ccc(C(c2coc(C)n2)O)cc1.N12CCC(CC1)C2 41515,c1(CC)ccsc1C(=O)NCC(C)(C1CC1)NC(=O)CSc1ccccc1 41516,c1(NC(c2n(CCCOC)nnn2)C2CC2)cccc(COC(=N)O)c1 41517,C=CC1CCCCN1C(C12CC1CN(C(=O)CC(C)(C)CC1CC1)C2)=O 41518,c1(NC(C(N2CCC(c3cn(C)nc3)C(C)(C)C2)=O)=O)cccc2c1CC(=O)N2 41519,C12(NC(=O)CC3CC(F)C3)CCCC1N(C(c1cnc(Cl)s1)=O)CCC2 41520,c1(C(=O)NC2C(NC(Cc3c(C)ccs3)=O)CC2)cnn(C(C)C(C)C)c1C 41521,n1(CCOC)cc(C(=O)NCC2COC(CNC(c3nn[nH]c3Cl)=O)C2)c(C)n1 41522,S(=O)(=O)(c1c(Cl)ccc(I)c1F)N(CCSc1cccc(Br)c1)CC 41523,CC1(F)CC2(CN(C(C3(NC(c4cc5n(n4)CCO5)=O)CC(F)(F)C3)=O)C2)C1 41524,C1(C(=O)NC(C)C(=O)NCc2ccccn2)CC(=O)CCO1 41525,CCC(CC(=O)NCC(C)(C(C)C)NC(c1ccc(CC(N)=O)cc1)=O)C1CC1 41526,CC1CC(C(=O)N(C)CCNC(C2(CF)CC(F)(F)C2)=O)CCO1 41527,C#CCC(C)C(=O)NCC(C)(C)CN(C(=O)C(c1ccccc1)SC)C 41528,C1(CC(=O)NCC2ON=C(C)C2)CCC(NC(C2CS(=O)(=O)C2)=O)CC1 41529,CC(CCCc1cn(Cc2nc(C(=O)O)cs2)nn1)C(=O)NC1CCNC1=O 41530,c1(CN(C(=O)COC2CCN(C(=O)C=C3CCN(C)C3)C2)C)cccnc1 41531,CCC(C(=O)NC1CCN(C(=O)CCn2cnc(C)c2C)C1CC)C(F)(F)F 41532,CC1(C)CCN(CCNC(=O)C(O)C2CN(C(=O)C=CCF)C2)C1 41533,c1(C(C)NC(N2CC(C(O)CO)C2)=O)cc2c(s1)CCC(C)(C)C2 41534,c1(C(=O)NCCCC(C)NC(c2cncc(SCC)n2)=O)ccc(N)c(C)c1 41535,Cc1ccc(F)cc1C(N1CC(CNC(c2nc(C3CC3)cs2)=O)C(O)C1)=O 41536,N1(CCC(=O)Nc2c(C)nc(CC)s2)CC(CN)C(C2CC2)C1 41537,c1(CC)nnc2c(C(N3CCC(NC(C4(O)CC4)=O)CC3C)=O)cccn12 41538,C(=O)(C(C)(C)C(C)O)NCCC1(OC)CN(C(=O)Cc2c(Cl)c(CC)nn2C)C1 41539,c1(N(C)C)ncnc(N2CCOC(C3CN(C(=O)CC(F)(F)F)C3)C2)c1[N+](=O)[O-] 41540,C1(CC)(NC(=O)CN2CCOCC2=O)CCCN(C(=O)C(CC)n2ccnc2)C1 41541,N1(C(c2ccc(F)c(C#N)n2)c2n(C)nnn2)Cc2ccccc2OC2(CCOC2)C1 41542,C(=O)(CCCCC1CC1)NCC(C=C)O.C12(CC1)C(=O)N2 41543,c1(C(N2CC3CN(C(c4ccon4)=O)CC32)=O)cn2cccc(Br)c2n1 41544,C12(CNC(c3ccc(CC)s3)=O)CCC(NC(C3COC(=O)O3)=O)(CO1)C2 41545,n1(CC)cc(NC(C2CN(C(=O)C(C)(C)N(C)C)CC23CC3)=O)ccc1=O 41546,N1(C(CN(C(=O)NC2CC2)CC)=O)CC2CC(NC(=O)COC)C1C2 41547,c1(NCC)ccc(C)cc1C(=O)NCCCNC(c1cccc(C(=O)NC)c1)=O 41548,CCC(C)C(O)C(=O)NC1(CC(=O)N(C(C)CO)C)CC1 41549,N1(C(C2(C)C=CCC2)=O)CCCCCC(NC(=O)C(c2ccc(O)cc2)=O)C1 41550,N1(C(C(C)CBr)=O)CCC2(CCN(C(c3cc(C4CC4)nn3C)=O)C2)C1 41551,c1(NC(C)=O)c(C(=O)OC(C)(C)C)cccc1F.C1(=O)CC(=O)ONCCN1 41552,CC12CC(NC(C3CC4CC4C3)=O)(C1)C1(CCN(C(c3sccc3Cl)=O)CC1)O2 41553,N1(C(c2c(Cl)ccc(OC)c2)=O)CC2CCC1C(CNC(C1CCOCC1)=O)C2 41554,N1(C(c2cccc(CC)c2)=O)CC2CN(C(C3(O)CCCCC3)=O)C2C1 41555,c1(-c2cc(C(=O)NCC(C)N(C(C(C)=C(CC)C)=O)CC)no2)ccc(Cl)cc1 41556,CC1(CNC(C2CCOC(=O)N2)=O)CCCN(C(c2cn(CCO)nn2)=O)C1 41557,c1(CC(N2C(C(N3CCCOCC3)=O)CC(=C)C2)=O)cccc(Cl)c1F 41558,CC1(CNC(c2ncn3c2CCC3)=O)CN(C(c2cccc(Cl)c2Cl)=O)CCO1 41559,C1CCCC(N=c2[nH]c(=NCC3CCSC3)c3ccccc3[nH]2)C1 41560,c1(CC)ccc(C(=O)NCC2(Nc3cc(Cl)nc(C)n3)CCCCCC2)c(F)c1 41561,N1(C(C=C(C)c2cccs2)=O)CCCC1C1CCCN1C(=O)CCCN=[N+]=[N-] 41562,c1(C(C(=O)NCCCC2CC2)N(CCOCC=C)C)csc(Cl)c1 41563,N1(CC(N2C(CCC)CCC2)=O)CCN(C(C2(C(N)=O)CCC2)=O)CC1 41564,C(c1ccc(C(=O)NC2(CCNC(=O)CC(C)F)CC2)cc1)=CC(=O)OC 41565,C1(C(=O)NC2(CC=C)CC2)CCN(C(=O)CCOCC(F)F)O1 41566,Cc1[nH]c(C)c(C(=O)NC2CC(C)(NC(c3ccnn3CCF)=O)C2)c1C 41567,CN1CC(NC(c2occc2CNC(C2C3CCCC23)=O)=O)C(F)(F)C1 41568,C12(C(N3CC(C)C(NC(C4(F)CCCCC4)=O)CC3)=O)C3CC(CC13)C2(F)F 41569,N(C(=NCCOc1ccc(Cl)cn1)NCC1CCC(F)CC1)CC(COC)C 41570,N1(C(C2C3CN(C(C(CSC)O)=O)C2C3)=O)CC2C(C1)C2(F)F 41571,C1(CNC(CSCC#C)=O)CN(C(C2CCN(C(C)=O)CC2)=O)CC1(F)F 41572,c1(C(=O)NC2CCC(CCC(=O)NCCOCC=C)C2)nc(C)ccc1C 41573,C1(NC(=O)COc2cccnc2)CN(C(=O)Cc2ccc(Cl)cc2)CC1F 41574,C1(OC)(CNC(c2cncc(C(F)F)c2)=O)CCN(C(C23CC(CO)(C2)C3)=O)C1 41575,C1(C#N)(C(N2CC(CC(CNC(C3N(C)CCCC3)=O)(C)C)C2)=O)CCOCC1 41576,c1(CC(=O)NC2COCC2NC(C2CC3CCC3C2)=O)cc(Cl)ccc1Cl 41577,c1(C(N)=O)cc(CC(=O)NCC2(O)CN(C(C3(n4nccn4)CC3)=O)C2)on1 41578,c1(CC)c(C(=O)NCC2C(C)CCCN2C(=O)CC2CCC2OC)cccc1C 41579,CCCC(C)CC(=O)NCC1CCCN(C(c2cc(CC)ccc2C)=O)C1 41580,CCCC(C)C(=O)N1CCC(C(=O)NCC(F)(F)COC)(CO)C1 41581,c1(OCC)ccc(C)cc1C(=O)N(CCNC(=O)CC1CC(C)=NO1)C1CC1 41582,C12(C(=O)OC)CCN(N3C(COC(C)(C)C)C(C(F)(F)F)C3)C1C2CCC 41583,C1(C(N(CC(=O)NC(C2CC=CCC2)CO)CC#C)=O)C(C(C)=O)C1(C)C 41584,c1(CC)[nH]nc(C(=O)NCCOCCNC(=O)C(O)CC2CC2)c1Cl 41585,C=CCC(C)C(=O)N1CCC(n2cc(CNC(C3CC(C(=O)OC)C3)=O)nn2)C1 41586,N1(C(CC(CC)C2CC2)=O)CCC2(C=C(C(=O)N3CCCN(C)CC3)C2)C1 41587,c1(C(=O)NC2CN(Cc3ccc(Br)nc3Br)C2)cc2cccnn2n1 41588,C(=O)(C(CC(C)C)NC1(CCF)CC1)N(CC(COC)O)C 41589,C1(C)(COC)CC(NC(=O)Cc2c[nH]nc2C)CN1C(c1cc(C)ccc1C)=O 41590,N1(C(C)=O)CC2CCC1CN2C(C1(C#N)CC(n2cc(CCO)nn2)C1)=O 41591,c1(C(=O)NCC23CC(NC(C4CC(C)OC4)=O)(C2)C3)ccc(C(F)(F)F)c(N)c1 41592,N1(C(C(CC)=CC)=O)CCCC12CCN(C(C1CCN(C3CC3)C1=O)=O)C2 41593,CN1N=C(CC(=O)N2CCC=C(CNC(=O)C(C)(C)C3CCCO3)C2)CC1=O 41594,N1(C(C2(CC)CC2(F)F)=O)CCC(CO)(NC(c2ncoc2-c2cccs2)=O)C1 41595,N1(CCOC)CCN(C(=O)Cn2cc(CCC3(OC)CCC3)nn2)CC1 41596,CCCC(C)(O)CC(=O)NC1CCCC1NC(c1cnc(C)c(N)c1)=O 41597,C(CN=C(NCCSc1cccs1)N(C)Cn1ncc(O)nc1=O)c1cnc(C)s1 41598,c1(NC(N2CCCC(NCC=C)C2)=O)c(-c2ccccc2)c(C)nn1C 41599,c1(NCC(COC(C(C)SCCCC)=O)C)c([N+](=O)[O-])c(C)nn1CC 41600,CC1(C)CCCC(CC(N2CC(CNC(c3cncc(N)c3)=O)C2)=O)O1 41601,CC1CC(N(C(=O)COC2CCN(C(C3(C)CCCCCC3)=O)C2)C)CC(C)C1 41602,C(CO)(CC(C)(C)C)NC(C(CC=C)NC(c1ccc(F)cn1)=O)=O 41603,CC1CN(C(=O)C(N2CCOCC2)C)CC1CNC(c1cnn(C)c1C(F)F)=O 41604,c1(C2CCN(CCC)C2)nc(-c2ccc(OC)cc2)nn1-c1ccn(C(C)C)n1 41605,Cn1c(C(=O)NC2CN(C(=O)CCC3CCCCO3)CCC2F)cc(Cl)c1Cl 41606,N1(C(C(C)CC2CCC2)=O)CCOCC(C(=O)NC2CN(C)CC2(F)F)C1 41607,c1(N(CC)CC)ccc(SC)c(NS(C)(=O)=O)c1.c12cccc(c1)NC(=O)N2 41608,CC(C)CC(O)C(C)C(=O)NC(CC1CC1)C(N1CCCC(C=C)C1)=O 41609,C1(C(=O)NCC2(F)CC(CNC(C3N(C(C)C)CCC3)=O)C2)C2CCCCCC12 41610,N1(C(c2nn(C)c(Cl)c2)=O)CCC2CN(C(=O)C(O)CC3CCOCC3)CC12 41611,Cn1ncnc1C(N1CCCC1C(=O)NCc1ccccc1)C(=O)NC1CCC1 41612,CC#CCC(C(=O)NCC(C)(C)C1(O)CCC1)NC(C1CN2CCC1C2)=O 41613,N1(C(CCCCC)=O)CC2(C1)SCCC2NC(c1ccccc1OC)=O 41614,c1(SC)nc(N(c2ccc(N3CCCCC3)cc2)C)nc(N)n1 41615,c1(C(=O)NC(c2c(C(=O)NCCCC=CC)con2)C)cc(CC)oc1C 41616,N1(C(COCc2cc(C)no2)=O)CC(NC(c2ccc(=O)oc2)=O)C(O)C1 41617,C1(O)(CNC(=O)CCn2cccc2)CCCN(C(c2nc(Cl)cs2)=O)C1 41618,C1(NC(C=COCC)=O)CS(=O)(=O)CC1NC(c1cc(Br)sn1)=O 41619,C1(C(N(CCC(=O)OC)CC=C)=O)CCN(C(=O)CC2CCCC2)C1C 41620,C(CN=c1nc(CC2CC2)[nH]s1)CC1CCCN(C(c2cc(OC)n[nH]2)=O)C1 41621,C1(N(C(=O)COc2cn[nH]c2)C)CCCCN(C(=O)C=Cc2cccc(O)c2)C1 41622,c1(CC)cccc(CNC(=O)NC(=O)CN2CCC(C)CC2)n1 41623,N1(C(C(CC(=C)C)OC)=O)CCC2CN(C(=O)CN3C(=O)CCC3=O)C(C)C12 41624,CCC(C)(CNC(=O)CCc1ccccc1Br)C(N)=O 41625,c1(COC)nn(C)cc1C(=O)NCC(C)(CO)NC(=O)Cc1cncc(O)c1 41626,C1(C(=O)NCC2C(CNC(=O)CCCn3cccn3)C2(F)F)CC2C=CC1O2 41627,C(=O)(C(C(=O)NCC1CCN1C(c1cc(O)n(CC)n1)=O)C(C)C)OCC 41628,C(=O)(CC(C)C(C)(C)CC)NCCCOCCN(C(CCC=CC)=O)C 41629,Cn1c(C(N2C3CN(C(=O)Cc4cccnc4Cl)CC23)=O)cc2ccccc12 41630,Cc1ccc2oc(C(=O)NC3C4CCN(C(C5(C)CCCOCC5)=O)C34)cc2n1 41631,c1(C(=O)NCc2scc(CNC(c3ccc(C)s3)=O)n2)ccn2nncc2c1 41632,c1(CC(=O)NCC(CN(C(C(C)SC)=O)C)C)cncc(C)c1 41633,c1(CC(=O)NCC(CC)(C)NC(C2CCCCC2C)=O)cn(C)c2ccccc12 41634,C1(F)(C(N(c2ccccc2)CCC=C)=O)CCN(C(=O)CCNC(=O)OC)C1 41635,CC(=O)CCCC(=O)NC1C2CN(C(c3cc(C)c(C)s3)=O)CC12 41636,C(=O)(C(F)(F)CCC=C)NCCN(CC#C)C.C(=O)(C(C)OC1CO1)NOC(C)=O 41637,CC(C(=O)NCc1ccc(C(F)(F)F)cn1)N1C(=O)COc2ccccc21 41638,Cc1cccc(SC(C)CC(F)(F)F)c1.c1(-c2n(CC=O)nnn2)ccccc1F 41639,CC(C)(C)CC(O)C(=O)NC(Cc1cc[nH]n1)C(N1CCCCCC1)=O 41640,c1(C(C)NC(c2nnnn2C)(COC(C)=O)C)cn(-c2ccncc2)nc1C 41641,CCC(CC(=O)N(CCC(C)NC(=O)COC1(C(F)(F)F)COC1)C)OC 41642,c1(CNCC2N(C(c3nc(CC)oc3)=O)CCCC2)n[nH]c2ccccc12 41643,C1(C)(C(N(CCNC(=O)C=C(C)C)CC)=O)CCC(=O)NC1 41644,N1(C(C(C)OCC#C)=O)CC(NC(c2sccc2OCC)=O)C2CCCCC12 41645,C1(CCOC)(NC(=O)C=CC2CCCN2C)CCN(C(=O)C(C)(C)C2CCC2)C1 41646,C(=O)(CC(C)(F)F)N(CC(C)O)CCNC(C1C(C)C1C)=O 41647,C=CCCCC(C(=O)N1CCC(n2ccnn2)C1)NC(c1cn(C)cn1)=O 41648,N1(C(C2CC(C#N)C2)=O)CCC2(NC(c3ncccc3Cl)=O)CCCC12 41649,c1(NC(C(CC=CC)NC(=O)Cc2ncoc2C)=O)cc(C)ccc1CO 41650,c1(C(=O)NCC2C(OCC)CN(C(=O)C(C)(C)SC)C2)cccc2ccnn12 41651,CCC(C)CCNC(=O)CC1(CNC(C2CC(OC)C2)=O)CC1 41652,N1(C(C(CC)Cl)=O)CC(NC(C2CCCC2C)=O)C2(COC2)C1 41653,n1(CC(=O)NC2CCCC(C(=O)NCc3cncs3)C2)cc2ccccc2n1 41654,C(=O)(C(CC)CC(C)C)NCCCC(C)NC(c1c(CC)c(F)ccc1)=O 41655,C1(C(=O)NCC(CNC(CN(CC#C)C)=O)C)CCCN(Cc2ccccc2)C1 41656,N1(C(c2c(C)cccc2F)=O)C2CCC1CN(C(C1CCC3(CC1)CC3)=O)C2 41657,Cc1nn(C)c(Cl)c1CNCCC(N1CCOCC(C(=O)NC(C)(C)C)C1)=O 41658,CCC(CNC(=O)C=Cc1cnc(C)s1)N=c1[nH]nc(C2CC2)o1 41659,c1(C(=O)NC(CC)CNC(c2ncccc2Cl)=O)cc(Cl)sc1S(N)(=O)=O 41660,c1(C(=O)NC(CCN(C(C(C)NC(CC)(C)C)=O)C)C)nccc2nn[nH]c12 41661,Cc1nc(C(C(=O)NCC(C)C)N(C2CCN(c3ccncc3)CC2)C)sc1C 41662,CCN=C(NCc1cc(COC)no1)NCc1ccc(-n2ccnn2)cc1 41663,CC(O)(C(=O)NC12CC(CNC(=O)CSC3CCCCO3)(C1)C2)C1CCC1 41664,C1(NC(Cc2c(OC)cccc2)=O)CCSC12CN(C(C1CCCOC1)=O)C2 41665,C1(OCC)COCCC1CC(=O)NCC(=C1CN(C(c2ccoc2)=O)C1)F 41666,CC(C)CC(CNC(=O)CCN1CCCCC1)NC(C1COC(=O)N1C)=O 41667,C12(CNC(c3c(OC)nsc3)=O)CCC1CN(C(C1CC(O)CN1C)=O)C2 41668,CS(=O)(=O)C1CCCN(C(=O)CC2CCN(C(=O)CCc3ccco3)C2)C1 41669,N1(C(COCCCC#C)=O)CCCC(O)(CCNC(c2c(Cl)csc2Cl)=O)C1 41670,Cc1c[nH]cc(C(=O)NC2CC(F)(CNC(c3cnns3)=O)C2)c1=O 41671,c1(NC(C(c2c(C)nccc2)C)=O)ncc2c(n1)COCC2 41672,C(=O)(C(C)(C)C(N)=O)NCCCCN(C(=O)C(C#N)C1CC1)C 41673,N1(C(C=C(CC)CC)=O)CCC(O)(CN(C(=O)Cc2cnn(C)c2)C)C1 41674,O=C1CC(CC(=O)NCCC2CCCN2C(c2cc(Cl)no2)=O)CCCN1 41675,c1(C(=O)NC2CCN(C(C3COCC4(CCC4)O3)=O)C2)cc2cc(F)ccc2s1 41676,CC1(C(=O)Nc2cncnc2)CCCN1C(c1nc(Cl)sc1Cl)=O 41677,CC1CCCC=C1C(=O)N(C(C)CNC(c1cc2ncccc2[nH]1)=O)C 41678,C(=O)(CCCC(C)(F)F)NC(C1OCCN(C(c2c(C)csc2)=O)C1)C 41679,C1(NC(C(Cn2ccnn2)NC(=O)CC2C=CCC2)=O)CC2CCCC2C1 41680,N1(C(CN(C(C)C)C)=O)CCOC2CN(C(c3ccsc3C(F)F)=O)CC12 41681,C1(CC(=O)NCc2cc(C)on2)COCCN1C(C1CC1C(N)=O)=O 41682,Cc1ncc(Cl)c(C(N2CCC(O)(CNC(C3CCCC34CCC4)=O)CC2)=O)n1 41683,N1(C(COC)=O)CC(C)(C)CC1CNC(=O)C(O)C(Cc1ccccc1)OC 41684,N1(C(C(N2C(C)CCCC2C)=O)C)CCC2(CC1)CC(C)N(C(C1CC1C)=O)C2 41685,N1(C(C2(N(C(CSCC#C)=O)C)CC2)=O)CC(O)(CO)C1 41686,N1(C(Cc2cn(C)nn2)=O)CCCC(n2cc(CN3CCCCCC3)nn2)C1 41687,N1(C(C(CC)Nc2ccccn2)=O)C2CCC1CN(C(=O)C(C)OC)C2 41688,CC(C)CCC(C)NC(C1(C2CC2)CCCN1C(=O)CCC(=O)N(C)C)=O 41689,C1(CNC(CCOc2ccc(OC)cc2)=O)CN(C(=O)C2=CSCS2)CCC1C 41690,C1(CNC(C(C=C)O)=O)CCN(C(=O)CNC(=O)OC)C12CC2 41691,C(=O)(C(C)(CC(C)C)NC(=O)Cc1cc(C(F)(F)F)c(O)nn1)OC 41692,N1(CC(C)O)CCC(C2CCCN(C(c3cnc(C4CC4)o3)=O)C2)C1 41693,c1(CCNC(C2C=CCN2C(c2ccnnc2)=O)=O)ccc(F)cc1 41694,c1(C(N2CC3C(CNC(c4cnc(CCC)s4)=O)C3C2)=O)cc2nc[nH]c2cn1 41695,C1(COC)OC(c2nc(Cc3ccoc3)no2)CC1C 41696,C1(CC)CN(C(C2COCCOC2)=O)CCN1C(C12CCCC1(C(N)=O)C2)=O 41697,c1(C(=O)NCC(CNC(C(CCCC)N(C)C)=O)F)oc2ccccc2c1CO 41698,c1(CC(=O)NCCC(=C)CNC(=O)C(O)C(C)CC)ccc(Cl)c(OC)c1 41699,C1(C(=O)NC2CC(C)(NC(Cc3ccc(C)nc3)=O)C2)CCCCNC1=O 41700,c1(C(=O)NC2(CNC(C(CC)CC3CCCC3)=O)CCC2)cc2cccnn2n1 41701,N1(C(c2ncc(C(C)=O)[nH]2)=O)CCN(C(C2(c3ccc(Cl)cc3)CC2)=O)CC1C 41702,N1(C(c2c(C)oc(Cl)n2)=O)CC2CCOCC2(NC(c2cc(Cl)no2)=O)C1 41703,C1(NC(=O)C2=CCSC2)CC2CN(C(c3c[nH]cc3Br)=O)CC2C1 41704,c1(-c2c(N(CC(N3CCCC3)=O)C)c[nH]c2)ccc(-c2ccncn2)cc1 41705,CN1CCC(F)(C(=O)NCCC(O)CNC(c2ccccn2)=O)CC1 41706,CCC(C)(CNC(C1(F)CCN(C(c2ccc(CO)cn2)=O)C1)=O)C(N)=O 41707,C(=O)(C(C)C(CC)CC)N1CCCC(n2cc(C(C3CC3)OC)nn2)C1 41708,c1(C(C)(C)C(N)=O)ccc(NC(C2CC2c2cncc(Br)c2)=O)cc1 41709,C(=O)(C1=CC(O)C(O)C(O)C1)Nc1ccc(NC(c2cccc(Br)c2)=O)cc1Cl 41710,C(=O)(CC(F)(F)CS(C)(=O)=O)NCCCC1N(C(c2c(C)nccn2)=O)CCC1 41711,C(CCC(=O)NC(c1nocc1C(N1CC(C)(C)C1)=O)C)OCC 41712,c1(OC)ccnc(C(C(=O)NC2CCOC2)N(C2CCCCC2C)C)c1C 41713,N1(C(C2N(CC)CCC2)=O)CCC(C(=O)NC(CC2CC2)C(=O)NC)C1(C)C 41714,c1(OC)cc(SC)ccc1C(N1CC(O)(C(C)NC(c2nccnc2C)=O)C1)=O 41715,C1(C(N(C2CCCN(C(c3sc(C)nc3C)=O)C2)CC)=O)CC2(CCC2)CO1 41716,Cc1cccc(CN(C(=O)C(c2cccs2)NC(=O)C(C)n2ccnn2)C)c1 41717,c1(C(=O)NCCN(C(C2CC2c2ccnn2C)=O)CC)ccn(C(C)C)c1 41718,c1(C(=O)O)nc2ccc(F)cn2n1.C(=O)(C(O)CC(C)C)N(C1CC2(CNC2)C1)CC 41719,C1(N)CCn2nccc2C1.c1(SC(C(N2CC(CCC(=O)OC)C2)=O)=O)nnnn1C 41720,C1(C(=O)NC(CC2CCC2)CO)CCN1C(=O)C=C1CCC1 41721,C1(CNC(c2nc(COC)sc2)=O)CCCC(CNC(=O)C=CC=C(C)C)C1 41722,C(=O)(CCCC(=O)NC1CC1CNC(C1CCN(C2COC2)C1)=O)OCC 41723,C1(NC(C2(CC#C)CCC2)=O)CCCC(NC(c2cc(C)n(C)c2)=O)C1 41724,Cc1nc2cc(C(=O)NCCCNC(=O)C(C)c3cccs3)ccc2n1C 41725,c1(C(N(C2CCN(C(CCC(C)SC)=O)CC2)C)=O)ccc(F)c(F)c1F 41726,C1(CC)CCC(C(=O)NC23CC(C(=O)NCC(F)(F)CO)(C2)C3)CC1 41727,C1(CCNC(C(C2CCOC2)OC)=O)CN(c2nc(C(C)C)ns2)CCS1(=O)=O 41728,c1(OCC=C)ccc([N+](=O)[O-])c(C(=O)NCC2CC2NC(=O)C(C)=CCC)c1 41729,c1(C(=O)NC2(CNC(C(C(CC)(C)C)O)=O)CCC2)ccc(C=NOC)cc1 41730,C1(N(C(C(C(C)O)NC(c2cc(CC)on2)=O)=O)C)CCOC(C)(C)C1 41731,C1(C(=O)NC(C)CC(C)NC(c2cnn(C3CC3(F)F)c2)=O)CC(C2CC2)=NO1 41732,C(CNC(=O)Cc1ccc(C)o1)(C(C)(C)C)NC(c1nc(OCC)oc1)=O 41733,c1(C(=O)NCC2C(C)CCN2C(=O)CCN2CCCC2=O)cnn2c1OCC2 41734,CCC(CC)CC(=O)NC(C)CCCNC(c1ccc(Cn2cccc2)cc1)=O 41735,N1(C(C(CC)C)=O)CCCC(C(N2CCCC2Cc2ccccc2)=O)C1 41736,N1(C(CCc2n(C)ccn2)=O)Cc2n[nH]cc2C1C(=O)NC1CNC(=O)C1 41737,C=CCCCCCC(=O)N(C(C)C(=O)NC1CCCC(CC)C1)C 41738,C1(C(=O)NCCC(C)N(CCC)C)COCCN(C(=O)OC(C)(C)C)C1 41739,N1(C(CC2(C)CCC2)=O)CC2C(NC(c3ccc(CO)cn3)=O)C2C1 41740,CCCCCC(F)C(=O)N(C)CC.N1(C(C)=O)c2ncnn2CCC1 41741,n1(CC)ncc(=NC(=O)C(CC2CC2)CC2CC2)[nH]1 41742,c1(NS(C)(=O)=O)cccc(C(=O)NC2CCCCC2CNC(C2CCCC2)=O)c1 41743,CC1(C)Cc2occc2CN(C(=O)CCc2cnc[nH]2)C1 41744,c1(CNC(C2CN(C(C3(CC)CC3)=O)CCC2(F)F)=O)ccc(S(N)(=O)=O)cc1 41745,C1(C(=O)NC2CC(NC(C(C3CCC3)OCC)=O)C2)CC2(C1)CC21CCC1 41746,c1(CCC(=O)NC(C2(O)CCN(C(CCOC(C)=O)=O)C2)C)c(F)cccc1F 41747,C1(CC)CCCC(C(=O)NCCn2cc(SCCSC(C)(C)C)nn2)CC1 41748,C(=O)(C1=NNC(=O)CC1)N(C1CCCC(NC(c2ccoc2Cl)=O)C1)C 41749,C(=O)(C(C)N(OC)C(=O)C=CCN(C(=O)C(C)SC(C)C)C)N(C)CC 41750,N1(C(CCn2c(C)cc(C)n2)=O)CC(C)(C)CC1CNC(c1cc(Cl)sc1Cl)=O 41751,N1(C(C2(CC)CN(C(C(C=CC)O)=O)C2)=O)CCC(O)(COC)C1 41752,c1(C(=O)NCC(C)NC(CC)=O)cc(-c2ccccc2)n[nH]1 41753,C(=O)(CS(=O)(=O)CCC(F)(F)F)N1C(C(C)NC(c2c(C)occ2)=O)CCCC1 41754,Cc1nc(C)c(C(N2CSCC2C(=O)NC(C2CCC2)C)=O)o1 41755,C1(C(=O)NCCC2N(C(c3c(CC)nn[nH]3)=O)CCC2)(COC)CCOCC1 41756,Cc1ncncc1C(N1CCC(=CC(=O)Nc2ccc(F)nc2)CC1)=O 41757,C1(NC(CONC(=O)CC2(O)CCCC2)=O)CCCN(CCO)C1 41758,C#Cc1ccc(OC)c(C(=O)NCC2(C)CC2C)c1 41759,C1(=O)C(CCSCC)OC2CC(C2)N1C.c1(C(=O)NC)ccoc1 41760,N1(C(C2(NC(C=Cc3ccc(C)o3)=O)CC(F)C2)=O)CC(C)OC2(CCC2)C1 41761,N1(C(C2C(CNC(C=C3CCC(C)CC3)=O)CCO2)=O)CC(C)C(O)C(C)C1 41762,CC1(CCNC(=O)Cn2cnnn2)CCN(C(c2ncncc2F)=O)CC1 41763,CC1CC(CO)CN(C(=O)C(C)NC(c2ncccc2Cl)=O)C1 41764,C(=O)(C(C)CC(N)=O)N1CCC(N(C(CCCCC)=O)CCOC)CC1 41765,CCN=c1ccc(C(=O)NC2COCC2CNC(c2cccc(F)c2F)=O)c[nH]1 41766,c1(N(C(=O)NC(C)CCF)C)ccc2cnccc2c1 41767,CC1CN(C)CC(C(N2CCOCC(C(=O)NC(C)C(O)C(F)F)C2)=O)O1 41768,c1(C(=O)NCCSCC(=O)NCCC(C)N(CCC)C)coc(CO)c1 41769,Cc1nn(C)c2ccc(C(=O)NCC3CN(C(=O)Cc4ccco4)CC3O)cc12 41770,c1(C(N(CCCCNC(C(CC)O)=O)C)=O)c(C)sc(C)c1C#N 41771,c1(C(=O)NCCN(C(C(c2cccnc2)OC)=O)C(C)C)cnn2ccccc12 41772,c1(C(N(CCCCNC(c2ccc(C(N)=O)cc2)=O)C)=O)cccc2c1NCC2 41773,N1(C(c2ccc(CCC)cc2)=O)CC(C)(C)OC2(C1)CN(C(C1(O)CCC1)=O)C2 41774,Cc1cncc(CC(=O)NCCC2CCCN2C(C2COCCO2)=O)c1 41775,N1(C(c2cccc(C(N)=O)c2)=O)CC2CN(C(=O)C(N)=O)CC2C1 41776,CC(C)CC(CNC(C1Cc2nccn2C1)=O)C(=O)NCCC(C)C(F)F 41777,C(=O)(C(CNC(=O)Cc1cnsc1)(CC)CC)NC(c1ccccc1)C=C 41778,CCC(C)C(C)CNC(C1CC=CC(NC(=O)Cc2cnn(C)c2)C1)=O 41779,C(=O)(C#CC1CC1)NC(CN(C(c1nc(SC)sc1)=O)C)(C)C 41780,C1(NC(C2C(C)=C2)=O)CC12CC(NC(C1(c3ccc(C)cc3)CCCC1)=O)C2 41781,N1(C(C=C(C)C(C)C)=O)CCC(C)C1CNC(c1cn(CC(F)(F)F)nn1)=O 41782,C1(CC(=O)NC)CN(C(c2sccc2C(F)F)=O)CCN1C(=O)C(CCO)OC 41783,C1(NC(C(COC)N(C)C)=O)CC(OC)CN(C(=O)CSC(F)(F)F)C1 41784,c1(OC)cccc2c(CC(=O)NCC(O)CCNC(=O)CO)c[nH]c12 41785,c1(-c2cc(C(=O)NC3(CNC)CCCC3C)no2)cc(OC)cc(OC)c1 41786,C1(NC(c2c(CC)nccn2)=O)CN(C(c2cc(CO)ccn2)=O)CC1N=[N+]=[N-] 41787,N1(C(c2nnn(CCOC)n2)=O)CC2(CCC2NC(=O)C(C)(C)CSC)C1 41788,N1(C(CSCCC)=O)CC(CN(C)C(c2cccc(N(C)CC)c2)=O)C2(CC2)C1 41789,c1(C(C(C)NC(=O)Cc2cc[nH]n2)NC(=O)C(F)F)ccccc1 41790,c1(C(=O)NCCCC(C)NC(=O)C2=NNC(=O)C2)cc2cc(Cl)cnc2o1 41791,N1(C(c2c(C)[nH]nc2CO)=O)CCC2(CC1)CCN(CCC1CCCC1)C2 41792,C1(C(N(C2CCN(C(c3nn[nH]n3)=O)CC2)CC(C)C)=O)(CN)CC2C=CC1C2 41793,CC1OC2(CNC(C3CC3F)=O)CC1(NC(c1nccc(F)c1Cl)=O)C2 41794,N1(C(C2C(C3C(C)C3)C2)=O)CC2CN(CCOC3CCC3)CC2C1 41795,N1(C(CCC(CC)C)=O)CC(CNC(C2CC(=C3CC3)C2)=O)C2CCCCC12 41796,C1(NC(CC2C(C)OC(C)C2)=O)CCC2CN(C(=O)CCCCC3CC3)CC2C1 41797,CC1=NOC(CC(=O)N(C2(C(=O)Nc3csc(C)c3)CC(O)C2)C2CCC2)C1 41798,Cc1csc(C(N2CCCC2C(C)(C)NC(=O)CCn2ccnc2C)=O)c1 41799,c1(C(N2CC3CC2CS3=O)C(=O)NCCN2CCOCC2)noc2c(Cl)cccc12 41800,C(CN=c1[nH]c(=NC2CCC=CCC2)[nH]c2cc[nH]c12)N1C(=O)OCC1 41801,C(=O)(C(C#N)(CC)CC)N(CCNC(C1CC(C(C)C)=NO1)=O)CC 41802,C1(C(N(CC(C)N(C(=O)C(C2CC2)C2CC2)C)C)=O)CC(CC(F)F)C1 41803,CC1CCCC(C)N(C(C2CC3CCC(C2)N3C(c2ccncc2Cl)=O)=O)C1 41804,C(=O)(C#CC1CCOC1)N1CC(CNC(CCc2cc(C)cc(C)c2)=O)C1 41805,C1(NC(C(C)(C2CC2)OC)=O)CCCCC1C(=O)NC1(c2ccsc2)CC1 41806,Cc1ccc2occ(C(=O)N(C)CC3(O)CN(C(C4CC4C)=O)C3)c2c1 41807,Cc1nc(C)c(C(=O)N(C2CCN(C(c3cc(-c4ccccc4)cs3)=O)C2)C)s1 41808,C(=O)(C(C(C)(C)C)C1CCC1)NCC(C)NC(=O)C(C)S(C)(=O)=O 41809,N1(C(C(c2cnn(C)c2)OC)=O)CCCC(O)(CCNC(=O)CC(F)(F)Cl)C1 41810,O=C(N=c1[nH]oc2cc(Cl)ccc12)C1CC(F)CN1Cc1cnco1 41811,Cc1c(Cl)ccnc1C(N1CCCCC1CNC(C1(S(N)(=O)=O)CC1)=O)=O 41812,C1(N(C(CCN(CCCCC)C(C)C)=O)C)CCN(C(=O)C(F)C(C)C)CC1 41813,Cc1cccnc1C(=O)NC1CC(F)(CNC(=O)C=Cc2cscn2)C1 41814,C1(NC(Cc2cccc(C(N)=O)c2)=O)CS(=O)(=O)C2CN(C(=O)CC3CC3)CC12 41815,c1(C(=O)NCc2c(C)cc(OC)cc2C)cc2c([N+](=O)[O-])cccc2s1 41816,CCC(C)C(O)C(=O)NNC(=O)c1ccc(OC(CC)C(=O)OC)nc1 41817,C(=O)(CCCCC(=O)c1ccccc1)NC(C1OCCN(C(C(C)OC)=O)C1)C 41818,C#CC1CCCCN1C(C1CN(C(=O)CCC(=O)NCCC)CC1CCC)=O 41819,c1(CNC2CC(C(N3CCCC(CO)C3)=O)C2)cc(Br)ccc1Cl 41820,CCCCCCCC(=O)NC(CCCOC)C(=O)NCc1cn(C(C)C)nn1 41821,CCCCC(C)CCC(=O)N1C(C(=O)NCCOC2CC2)CCC1C(C)C 41822,c1(C(C(=O)NCCCOCCNC(C2(C(C)(F)F)CCC2)=O)OC)cnn(C)c1 41823,N1(C(C(CC=C)(C)C)=O)CC2CC(NC(=O)CCc3cnc(C)nc3O)CC1C2 41824,C1(CNC(N(c2ccc(F)c(Br)c2)CC)=O)CCC2(CC1)NC(=O)N(C)C2=O 41825,c1(SCC)ccc(CC(=O)NC(CCNC(c2ccsc2SC)=O)C(C)C)cc1 41826,c1(C(N2CCCC(C(CNC(CCC=C)=O)(F)F)C2)=O)ccc(F)c(C(C)C)c1 41827,C(c1ccc(Cl)s1)=CC(=O)NC(CN(C(c1c[nH]nc1OC)=O)CC)C 41828,N1(C(c2ccnn2CCOC)C(=O)NC)CC2CC(O)C(O)CC2C1 41829,N1(C(C=CC(C)(C)C)=O)CCC(C)(NC(=O)Cc2cc[nH]n2)CC1 41830,CC(F)(F)C(C)(C)C(=O)N1CC(NC(=O)Cc2cnsc2)C(N=[N+]=[N-])C1 41831,c1(CSC)ccc(C(N2CC(O)(C(C)NC(C3CC(C)(C)CO3)=O)C2)=O)cc1 41832,N1(C(C(C)Cc2ccc(O)cc2)=O)CCC2(CC1)CN(C(C1(C)CCCO1)=O)C2 41833,C(=O)(C(C)C(C)C)OCCOCCOC(CC)(C)C.C(C)=O 41834,N1(C2CCN(C(C(C)C#N)=O)CC2)CCN(S(N)(=O)=O)CC1 41835,N1(CCCNC(C(=O)NC)C)CCOC(C)C1 41836,C1(C(N2CC(N3CCCC3)C2)=O)CCCCCCN1C(C1CCCOC1)=O 41837,c1(C(=O)NCC2C(NC(CCCCOC)=O)CCCC2)ncnc(O)c1Cl 41838,C#CCC(CC(F)F)NC(C1CC12CCN(C(C1(C)CC=CCC1)=O)C2)=O 41839,C1(C(=O)OC)CCC(CN(C(CC2(C)CCOC2)C(=O)NCc2ccccc2)C)O1 41840,N1(C(CSCC=C)=O)CC(CNC(=O)COC(F)F)OC2(CCC2)C1 41841,c1(C(=O)NC(c2nc(C)[nH]n2)C(C)C)nsc2cc(Br)ccc12 41842,C12(C(N(C)Cc3cnccn3)=O)CCC1CN(C(C1CCNC(=O)C1)=O)C2 41843,Cc1cccc(C(C)C(=O)N2CC(C)C2)c1.C(C(F)(F)F)NC.C1(=O)C=CCN1C 41844,c1(C(N2C(CNC(CCCCOCCC=C)=O)CC2)=O)ccnc(C)c1O 41845,N1(C(C2(SCC)CCC2)=O)CC2CC(N(C(=O)CCCc3ncc(C)o3)C)C1C2 41846,c1(C(N2CCCN(CCNC(C(CC)F)=O)CC2)=O)cccc2c1CCCN2 41847,CC1CN(C(C2CNC(=O)N2)=O)CC1(C)C(=O)NC1CCNC(=O)CC1 41848,Cc1scc(C(=O)NCC(O)CNC(c2csc(CC(F)F)n2)=O)c1C 41849,C1(C(=O)NCCN(C(=O)Cc2csnc2C)CCC)CC12CCC(C)(C)CC2 41850,CC1(NC(C2CC3(CCC3)CO2)=O)CCN(C(=O)COc2ccon2)CC1 41851,N1(C(C(COCC)C)=O)CCC(CNC(=O)Cc2n[nH]c(=N)s2)(COC)CC1 41852,C(=O)(CCCCC(N)=O)NC1CCC(C)(CNC(C2(CF)CC(F)(F)C2)=O)CC1 41853,CCCC(CC(C)C)C(=O)N(CCNC(c1cc(N(C)C)ccn1)=O)CC1CC1 41854,N1(C(C(CC)=CCCC)=O)CCC2(C=C(C(=O)NC(C)C(=O)OC(C)C)C2)C1 41855,C#CC1(C(=O)NCC2(C)CCCN(C(C3(O)CCC3)=O)C2)CCOCC1 41856,N1(C(Cc2scc(N(C(C)=O)C(c3ccccc3)C)n2)=O)CC2C3CCC(C3)C12 41857,N1(C(C(CC)N(C)C)=O)CC2CN(C(=O)C(C)CO)CC2C1 41858,Cc1cc(C(N2CCCC(NC(=O)C(C)(C)NS(C)(=O)=O)CC2)=O)c(F)cc1F 41859,CCC(C)CC(C)C(=O)NCC1(CNC(=O)CCCCC(C)C)CCCC1 41860,N1(C(C=C(C)C(C)(C)C)=O)CCOC(C)(CNC(c2cc3sccc3s2)=O)C1 41861,C(CCCC(C)(C)C(=O)NNC(=O)C1(F)CC1)NC(C(CC)CC)=O 41862,Cc1cnnc(O)c1C(=O)NCc1nc(C(N2CCCC2CC2CC2)=O)co1 41863,Nc1cc(C(=O)NCC2CCN(C(C34CCCN3CCC4)=O)CC2)cc(O)c1Cl 41864,C1(NC(c2c(Cl)cn(CCC)n2)=O)CCN(CC=C(Cl)Cl)CC1C 41865,c1(C(C)(C)C(=O)NCCC2CCN(C(=O)CC3C=CCC3)C2)ccc(O)cc1 41866,Cc1cc(-n2nc(C3CCC3)nc2CC2CCOC(C)C2)cc(Br)c1 41867,c1(C(C(=O)NC(CNC(c2c(CC)con2)=O)C)(C)C)ccc(F)cc1F 41868,N1(C(c2nc(C)sc2)=O)CC2(CCCC(CNC(C3(F)CCCOC3)=O)O2)C1 41869,CC(C)CC(O)CNC(C1(C)CCCN1C(=O)C1CC1)=O 41870,C1(NC(COC2(C)CCC2)=O)CCCN(C(c2ccc([N+](=O)[O-])o2)=O)CC1 41871,C1(C(=O)NCC2C(C)CC2)CCN(C(C2CCCCS2)=O)C1 41872,N1(C(CCOCCOC(C)=O)=O)CCC2CN(C(c3ccc(C)nn3)=O)CC2C1 41873,C(=O)(C(F)C1=CCCCC1)NCCCN(C(CC(CC)O)=O)CC1CCCC1 41874,C12(COC)CCC(C(=O)NCC3C4CN(C(=O)C=C(C)Cl)CC34)(CC1)CO2 41875,c1(C(=O)OCC)c[nH]c(=NC2CN(C(C3CC(C(C)(C)C)=NO3)=O)CC2C)cn1 41876,c1(C(C(=O)N(CCN(C(=O)CC2CC=CCN2C)C)C)O)ccc(Br)cc1 41877,N1(C(CC(=O)OC)=O)CC2CC(C(N3CC(C)(N(C)C)C3)=O)CC2C1 41878,N1(C(C2CC(NC(C3C(C)(C)OCC3)=O)C(O)C2)=O)CCC2(CC1)CC2 41879,N1(C(C2C(C)C2C)=O)CC2CCCC(NC(c3ccc(C(N)=O)c(Cl)c3)=O)C2C1 41880,CC(C)C#CC(=O)NC(C)(CO)C(=O)N1CC(CO)C1(C)C 41881,C1(C(=O)NC2CC(CC(=O)NC3CC(C(C)O)C3)C2)CCCC12CCC2 41882,C1(NC(C2N(CC)CC2)=O)CCC(O)CN(C(c2cn(C)nc2OC)=O)C1 41883,N1(C(CC2(C=C)CCCCC2)=O)CCCC2(C1)CN(C(=O)Cc1ccn(C)n1)C2 41884,C1(C)(CNC(CN(C(=O)C(O)C2CCC2)CC)=O)CCCCO1 41885,N1(C(c2c(C)scc2)=O)CCCN(C(=O)CCC2CCN(C)C2)C(C)C1 41886,C1(C(=O)NC(C(=O)NCC)C)CC(C)CCN1C(C1CC2(CCC2O)C1)=O 41887,N1(C(c2cn(C)nn2)=O)CC2C(C(=O)N(C3CCCC3)Cc3ccccc3)C2C1 41888,c1(C(=O)NCC2(OC)CN(C(=O)COc3ccsn3)C2)cc2scnc2[nH]1 41889,C(=O)(C1CCc2cccnc21)NCC1(C)CCN(C(=O)COC2CCOCC2)C1 41890,CC(C)CC(F)C(=O)NC1COCC1CNC(c1coc(C(C)C)n1)=O 41891,N1(C(CC(C)N(C)C)=O)CC(C(=O)Nc2ccccc2C2CC2)CC2(CC2)C1 41892,CC(C)CCCC(=O)N1CCN(C(=O)C=CCO)CC1CO 41893,C1(CNC(C(C)(C)OCC)=O)CC(C)N(C(c2cccc(-n3cccc3)n2)=O)C1 41894,c1(OC)ccc(C(=O)OCC2CC23CCCCC3)c2ccccc12 41895,N1(C(=O)CCN2CCCCC2)CC2(CCN(C(C3CCCS3)=O)CC2)C1 41896,C1(C(N(CC(Cc2ccccc2)NC(CSC)=O)C)=O)CCC=CCC1 41897,C1(C(=O)NCCOCCCN(C)C(C2CN(C3COC3)C2)=O)CC2(CC2)CO1 41898,N1(C(c2cn(C)nc2)=O)CCC(C(=O)Nc2ncc(F)cc2F)C(O)C1 41899,C(C(=O)NC(C(=O)N(CC)CC1CCC1)c1ccco1)(C(C)C)OCC 41900,c1(C(N(C2CCN(C(=O)C=Cc3ncc[nH]3)C2)C)=O)ccc2cnnc(O)c2c1 41901,c1(C(=O)NCC2N(C(C(C(C)(C)O)F)=O)CCC2)cc2c(O)cccc2[nH]1 41902,C#CC(C)(C)C(=O)N1CC(=O)CC1C(N1CCC(CC)C1)=O 41903,c1(C(=O)NCCC(C)(C)OCC)ccc(S(=O)(=O)N2CCCC2C(=O)O)o1 41904,n1(CC=C)cc(C(=O)N(C2CCCC2)CCNC(=O)CSCCC(F)(F)F)nn1 41905,c1(C(N(CC(C)NC(c2c(SCC)cccn2)=O)C)=O)cn2c(n1)CCC(C)C2 41906,c1(CNC(CCC=C(C)C)=O)cccc(C)c1.C(=O)(C(O)Cc1cnc[nH]1)NC 41907,C1(NC(C=COCC)=O)CCC2CCN(C(=O)CC(C)C3CC3)C1C2 41908,N1(C(C=Cc2cnc(C)s2)=O)CC(NC(c2cc(C(N)=O)c[nH]2)=O)CC(O)C1 41909,c1(C(=O)NC(CNC(CCc2n(C)ccc2)=O)C2CC2)coc2ccccc12 41910,N1(C(C2(CC)CCNC2=O)=O)CC2(NC(c3ccc(Cl)nc3O)=O)CCC1CC2 41911,C12(C(N3CC=CC(NC(C4C(C(=O)OC)C4)=O)C3)=O)CC(C)(C1)OC2(C)C 41912,c1(OC)ccc(OCCC(=O)N2CC(C(C)NC(=O)CC=CC(C)(C)C)C2)cc1 41913,N1(C(CC=CC=C)=O)CCC(N(CCC)C(c2cc(N)c(C(=O)OC)s2)=O)CC1 41914,c1(C(N2CC(F)CC(NC(=O)CC3CC=CC3)C2)=O)cc2cc(Cl)ccc2o1 41915,C(=O)(C(CC(C)C)N(C(=O)Cc1sc(O)nc1O)C)NCCNC(=O)NCC 41916,N1(C(c2cc(C)nc(C)c2)=O)CCOC2(C1)CN(C(=O)C(C)OC1CCOC1)C2 41917,N1(C(CC(CCC)C)=O)CCC2(C1)CN(C(C1CCCN1c1cnccn1)=O)C2 41918,C1(C(N(CC(C(C)C)C)C)=O)C(C)OCCN1C(c1c[nH]c(=O)cn1)=O 41919,C1(NC(CC2C(C)CCO2)=O)(CNC(C2CC(N(C)C)C2)=O)CCCCC1 41920,c1(CC)nccnc1C(N1CCN(C2CCN(C(=O)C(O)C(C)SC)C2)CC1)=O 41921,C1(CC)CN(C(C2(CO)CCOCC2)=O)CCC1NC(c1ns[nH]c1=O)=O 41922,c1(C(=O)NC(c2ccccc2)CNC(C2(CF)COC2)=O)cccc2nc[nH]c12 41923,C(=O)(CC(C)CC(=O)N1CCCN(C(=O)Cc2ncc(Cl)s2)CC1C)OC 41924,c1(-c2ccc(OCCOCC)cc2)cncc(F)c1C(=O)NCCC#N 41925,c1(OC)c(C(=O)N(CC(C)CNC(c2nocc2C(C)C)=O)C)cc(Cl)cc1Cl 41926,N1(C(C2CC(NC(c3c(CC)ncs3)=O)C(O)C2)=O)CCS(=O)C(C)C1 41927,C1(NC(C2C(C=C)C2)=O)CC(F)CN(C(c2ccc(Cl)cc2NC(C)=O)=O)C1 41928,C1(NC(Cc2c(C)ocn2)=O)CN(C(C2CC3CCCCCC23)=O)CCC1(C)C 41929,N1(C(CC2OCCN(C(c3c(C)ccnn3)=O)C2)=O)CC(O)CC(C)(C)C1 41930,C1(NC(=O)Nc2cc(C)c(-n3cccn3)cc2)C2Cc3ccc(Br)cc3C12 41931,c1(OC)ncc(Br)cc1C(N1CCCC(CO)C1)C(=O)Nc1ccc(C)cc1OC 41932,c1(C(N2C(C(C)(C)NC(COC(C)C)=O)CCC2)=O)coc2c1C(=O)NCCC2 41933,N1(C(C(=CC2CCCC2)C)=O)CCC(NC(c2sccc2C2CC2)=O)C(CO)C1 41934,c1(CN2CC3C(C(=O)NCC)(CC3)C2)ccc(Br)c(OC)c1[N+](=O)[O-] 41935,C1(CC(N2CC(CNC(C(COCC)C)=O)OCC2)=O)CN2CCC1CC2 41936,N(C1CN(C(=O)Cn2cncn2)CCc2ccccc21)C(C1=CC(C)(C)C1)=O 41937,Cc1nc(=NCC2CCCC(NC(=O)C(C3CCOCC3)F)C2)[nH]cc1[N+](=O)[O-] 41938,CC(CC(=O)NCCC1CC(C(=O)NCc2nc(=O)o[nH]2)C1)CC(C)(C)C 41939,C1(NC(CCCC)=O)COCCN(C(=O)CNC(=O)CCC(C)C)C1 41940,N1(C(Cc2cn(CC)nc2)=O)CC(NC(c2nocc2C)=O)C2CCCCC12 41941,c1(C(=O)NCC2(C)CCCN(C(CCC(C)(C)F)=O)C2)ccc2nc(O)sc2c1 41942,C(C)(CNC(=O)COc1ccc(CCOC)cc1)(C(C)C)NC(C=C(CC)C)=O 41943,NS(=O)(=O)c1ccc(C(N2CC(CC(N3CCN(CCCO)CC3)=O)C2)=O)o1 41944,CC(C)CC(C)CN=c1[nH]c(N2CCC(C3CCN(C)C3)CC2)nc2c1CSC2 41945,C(=O)(CCC(C)(C)[N+](=O)[O-])N(CCC(C)C(F)F)C.C1(=O)C(C)(C)CN1CC 41946,CC1COC(CCO)N1C(=O)Nc1ccccc1-c1ccccc1 41947,N1(CCNc2c(F)cccc2)CCN(C2CC2)C(c2ccccc2F)C1 41948,N1(C(c2c(OC)n[nH]c2)=O)CCN(C)C(C(=O)NC2CCNC(=O)C2)C1 41949,C1(NC(C2C(C)(C)C2)=O)CCCN(C(c2cc(Cl)nnc2Cl)=O)CC1 41950,Cc1ccc2c(c1)CC(C(=O)NC(CNC(=O)CCc1cnoc1)C1CCC1)O2 41951,Cc1c(C(=O)NCC(C)(C)CN(C(=O)C(C)N(C)C)C)ccc(Br)c1F 41952,C1(N(C(=O)CSC(F)F)C)CCCCN(C(=O)C(C)(C)C2CCCC2)C1 41953,N1(C(Cc2nnc(C)o2)=O)C2CCC1CC(CNC(C1CC13CC3)=O)C2 41954,N1(C(C(C(C)C)NC=O)=O)CC2(CCN(C(C3CC3(C)Br)=O)CC2)C1 41955,c1(C(N(CCN(C(c2c[nH]nc2OC)=O)CC)CC)=O)cccc(Cl)c1OC 41956,C1(C(N2CC(CCNC(c3c(C)nc(CC)o3)=O)OCC2)=O)CS(=O)(=O)CCO1 41957,N1(C(c2ccc3c(c2)C(=O)NC3)=O)CCC2(CCN(C(=O)COCC(F)F)C2)C1 41958,c1(CC(N2CCC(CN(C)C(C3(C4CC4)CC3)=O)C2)=O)cnc2c(=O)[nH]ccn12 41959,C(CC)(C(=O)N1CC(N(C(=O)CCc2scnc2C)C)C1)=CC 41960,Cc1ccc(C(=O)NC2CC(C(=O)NCC(C)C(C)(F)F)C2(C)C)c(O)c1 41961,c1(C(=O)NC(C(C)O)C)ccc(NC(=O)CC2CCC(N(C)C)C2)cc1 41962,c1(CN(c2cc3ccccc3[nH]2)C)ccc2nccn2c1 41963,N1(C(CCC(=O)NCCC)=O)CCN(C(=O)C2=C(Cl)CC2)C(C2CC2)C1 41964,N1(CC)OCC(NC(=O)CCN(C(=O)CCCn2cccn2)CCCO)C1=O 41965,N1(C(COCC(=O)NC)=O)CC(C)(C)OCC1CNC(C1CCCCCCC1)=O 41966,N1(C(C(C)CN(C)C)=O)CCN(C(C2(n3cncn3)CC2)=O)CC1CCN(C)C 41967,C1(C(=O)NCC2CC2CNC(c2coc(C)n2)=O)(OC)CCCOC1 41968,Cc1cn2c(n1)CCC(NC(N1CCC(Nc3cc(O)ncn3)C(C)C1)=O)C2 41969,O=C(CS(=O)(=O)CCO)NCC1CCCC1NC(C1CNC(=O)O1)=O 41970,N1(C(C2C(NC(c3ccnc(SC)n3)=O)C2)=O)CC(F)(F)C(F)(F)C1 41971,c1(OC)ncc(C(=O)NC2C3CC2N(C(C2CCS(=O)CC2)=O)C3)c(C)n1 41972,CC(C)CC(C)CC(=O)N1CCC=C(CNC(c2cn(C(C)C)cn2)=O)C1 41973,N1(C(Cc2c(C)noc2C)=O)CC2(C1)CN(C(=O)C(C)(C)CCl)CCO2 41974,N1(C(CC2CCCC(C)C2)=O)CC2(CC(NC(=O)CC=CC(C)(C)C)C2)C1 41975,c1(OC)cc(N2CCC3CCC(C2)N3C(C2CCCO2)=O)ccc1[N+](=O)[O-] 41976,C(=O)(C1=CC2CC(C1)CC2O)NC(C)CNC(=O)CCn1cccn1 41977,N1(C(c2cnc(C(C)(C)C)nc2)C(=O)NCC)CCn2c(cnc2C(F)F)C1 41978,c1(NC(C2(C)CC2)=O)ncc(C)cc1C.CCC(=O)NC1CC1C(=O)O 41979,c1(COC)ccccc1Cl.Cc1nnc(C(N2C(CC(=O)N(C)C)CCC2)c2nn[nH]n2)s1 41980,C=CC(C)(CC)C(=O)NCC1(C)CCN(C(C2(Sc3ccccc3)CC2)=O)C1 41981,N1(C(C(CC)Oc2ccccc2)=O)CCC(NC(=O)C(C)(C)n2cnnn2)CC1 41982,C1(C#N)(C(N2CC(CNC(C3(C(=O)OC)CC3)=O)C2)=O)CC1C(F)(F)F 41983,C(=O)(C1=C(C)CCOC1)N(CC(C(=O)NC(c1cccnc1)CC)(C)C)C 41984,c1(C(=O)NCC(C)(C)NC(=O)CCc2ccsc2)cc(F)c2ccccc2c1 41985,CC1(C)CC(N=c2cc(C(F)(F)F)nc(Cl)[nH]2)CN(C(=O)CCC2CC2(F)F)C1 41986,c1(NC2CCN(C(C(C(C)(F)F)(C)C)=O)C2)nc(Cl)nc2c1CCOC2 41987,N1(C(COC(c2nccn2C)C)=O)CCC(C(C)NC(c2ccns2)=O)CC1 41988,C1(CNC(C2CCN(CCC)C2)=O)CC2CCC1N2C(=O)CCCCOC 41989,c1(C(CF)NC(=O)C(=O)Nc2ccccc2)ccc(Cl)cc1.C12CC1N2 41990,CC(C)(CCCNC(=O)C(CO)C(F)(F)F)C(=O)NCC12CCC(CC1)OC2 41991,c1(C(N2C(C)(CC(=O)NC3(C#C)CC3)CC2)=O)cc(C#N)[nH]c1C 41992,c1(N2CCCC(NC(N)=O)C2)nc2c(c(=NCc3ccc(Br)s3)[nH]1)COC2 41993,C1(O)(CC(=O)NCC#CC(=O)NCc2ncnn2CCCF)CCCOC1 41994,c1(CN(C(=O)C(=O)NCC2CC2)CCOC)c(C)nn(C)c1C 41995,N1(C(C(CC)N(CC)CC)=O)CCCC2CN(C(=O)COC3CCOC3)CCC12 41996,c1(C(C)(C)C)cccc(OCC(N2CC(CNC(=O)COc3cnsc3)C2)=O)c1 41997,c1(NC(C2CCC3(CCCN3)CC2)=O)ccnc2c(Br)cc(F)cc12 41998,c1(C(=O)NCC2C(C(=O)NCCC)C2)ccc(S(C)(=O)=O)s1 41999,CC1(C)CC(NC(=O)C=CS(C)(=O)=O)CN(C(c2cc(N)cc(O)c2)=O)C1 42000,N1(C(C(c2ccccc2)=O)=O)CC2CC(NC(C3(C4CCCO4)CC3)=O)CC1C2 42001,C(=O)(C(C)(C)C(=O)N(C)CC1CCN(C(c2ccccn2)=O)C1)NC 42002,c1(C(C)C)nnnn1CC(=O)NCC(=O)NCC1CCN1C(C1(C)CC1(C)C)=O 42003,C#CCC(CC#C)C(=O)N(C1CN(C(c2ccc(S(C)(=O)=O)o2)=O)CC1(C)C)C 42004,C1(NC(c2c(F)cncc2Br)=O)CC2(C1)CN(C(=O)C(O)C(F)F)C2 42005,n1(CC(=O)NC2C(CNC(C=C(CC)CC)=O)C2)cccc([N+](=O)[O-])c1=O 42006,CC1(C)CN(C(C2CCCCO2)=O)C1C1CCN(C(c2ccon2)=O)CC1 42007,N1(C(C2CCCN(C(C)=O)C2)=O)C2CCC1CC(C(=O)NC1CC1C(N)=O)C2 42008,c1(OC)ncc(Cl)cc1C(N1CC(CNC(C2CCC(C)(O)CC2)=O)C(C)C1)=O 42009,O=C(O)CCCCCCCCCNC(=O)CCOCCCO 42010,c1(C(=O)OCC)cc(N2CCC(C(=O)O)C2(C)C)n2nccc2n1 42011,CC1CN(C(c2ccnc(O)c2F)=O)CCC1N(C(=O)C=C(Cl)Cl)C 42012,c1(C(N2CC(CC=C)(NC(c3ccnnc3C)=O)C2)=O)nnc(O)cc1O 42013,c1(CC(N2CCOCC(NC(C(C(C)C)O)=O)C2)=O)ccc(C#N)cc1F 42014,c1(C(N(C)C2CC2)=O)cnc2c(-c3cncc4cc[nH]c34)cccc2c1 42015,C1(CC(=O)N(CC(C)CNC(c2csnc2C2CC2)=O)C)CCC(=O)NC1=O 42016,CCC(C)(CNC(=O)CCc1cccs1)NC(C1CC=CCC1)=O 42017,c1(C(=O)NC(C(=O)N(CCCC)CC)CO)cnncc1OC 42018,c1(C(N(CC(CC)NC(c2ccc(N)cc2Cl)=O)C)=O)cc(P(C)(C)=O)ccn1 42019,Nc1ccc(C(=O)NC2(C3CN(C(C4CCN4S(C)(=O)=O)=O)C3)CC2)cc1F 42020,Cc1n[nH]cc1CC(=O)NC1CC(C)(CNC(=O)C(C)OCOC)C1 42021,CC(C)(CN=c1nc(N2CCC(C(N)=O)C2)c2sccc2[nH]1)C(F)(F)F 42022,C1(CC(=O)NCCOC(C)(C)CNC(=O)CC2(CO)CC2)CS(=O)(=O)C1 42023,C1(OC)CCn2cc(C(=O)NC3CCCC(CNC(c4cscn4)=O)C3)nc2C1 42024,C1(C(N2CCCC(N(C(=O)COCC3(F)CC3)C)C2)=O)CCOCC12CCC2 42025,C(=O)(CC(C(F)F)n1ccnc1)NC(C(=O)OCC)Cc1ccccc1Br 42026,CCCS(=O)(=O)CC(=O)NCC1CN(C(c2sc(C)c(C)c2C)=O)CC1O 42027,Cc1cccc(C)c1C(=O)NCC(=O)NCC1COCCN1C(=O)CSC1CC1 42028,C1(CNC(=O)CC2CCOC2)CN(C(=O)Cc2ccc(O)c(Cl)c2)CCC1(F)F 42029,N1(C(C(C(C)C)O)=O)CC(C)OC2(CCN(C(c3ccc(F)cc3O)=O)C2)C1 42030,c1(C(=O)NCCCC#C)ccc2c(c1)CN(C(c1ccc([N+](=O)[O-])cc1O)=O)C2 42031,c1(C(N(C2CC3CN(C(CCCCOC)=O)C2C3)C)=O)noc2c1COCC2 42032,CC(C(C(=O)NC)N1CCCC(C(C)C)C1)=Cc1ccc(Br)s1 42033,N1(C(Cc2ccc(C)s2)=O)CCC(NC(c2cnoc2-c2cccs2)=O)C(F)C1 42034,c1(C(=O)NC(C)(C)CCNC(c2sccc2SC(F)F)=O)ccc2c(c1)CCN2 42035,C12(C(=O)NCC3(C#C)CCCC3)C(NC(c3cccc(C)c3F)=O)C3CC1C2C3 42036,C1(CC(=O)NC(c2c(C(=O)NCC#CCC)con2)C)CCCC12CC2 42037,c1(OC)nccc(C(N2CC(C(C(=O)NC3CCC(CO)C3)OC)C2)=O)n1 42038,CC1C(NC(=O)C#CC2CCCC2)C(C)CCN1C(=O)CNC(N1CCCC1)=O 42039,N1(CC(=O)N(Cc2c(C(=O)Nc3ccc(OC)s3)cco2)CC)CCC(F)CC1 42040,C1(O)(CCNC(c2c(C)cns2)=O)CCN(C(C2CCCC(O)C2)=O)C1 42041,C1(C2CCN(C(C3C(CC)(CC)C3)=O)C2)CCCCN1C(C1CCCC1(C)C)=O 42042,C1(C(N2CCC(O)(CN(C(C(C)=CC)=O)C)C2)=O)Cc2cncn2C(=O)N1 42043,C(=O)(C#CC1(CC)COC1)NCC(CC)NC(=O)C=Cc1ccccc1C 42044,C(=O)(C(CCC)NC(C)=O)NCC1(C(=O)NC(CC#C)CC)CC=CC1 42045,C1(NC(CCOC)=O)CCN(C(c2cnc(S)nc2)=O)CCC1(F)F 42046,c1(C(N(CC(CC)NC(=O)C=Cc2nccs2)C)=O)cnc(O)n1CC 42047,C1(C)(C(=O)NC2CC3(CN(C(c4c(C)cccc4C)=O)C3)C2)CC(C(C)C)=NO1 42048,CC1(C)CCC(C)(C)c2cc(C(N3CC4CCS(=O)(=O)CC4C3)=O)c(Br)cc21 42049,N1(C(Cc2ccc(C(=O)OC)s2)=O)CCC(CN(C)C(C2(C)CCCO2)=O)CC1 42050,C1(C(N(C)CC2CCN(C(=O)CC#N)C2)=O)C2CCC1(c1cncs1)C2 42051,C1(C(N(C(C(CC)C)C)C2CC2)=O)CCCC(NC(=O)C(C)=C(C)C)C1 42052,CCC(CC(=O)NCCc1cnc(C)cn1)N(C(=O)CCCCSC)C 42053,C(C)(C(C)N=c1cccc(S(=O)(=O)NC2CCCC2)[nH]1)n1ncc(C)c1 42054,c1(CN(c2c[nH]c(=NC)s2)CC)ccc(F)c(Oc2ccccc2)c1 42055,C1(F)(CNC(c2nc(OCC)sn2)=O)CCCN(C(C2CNC(=O)C2)=O)C1 42056,c1(CNC(=O)Nc2c(C#N)cc(CC)s2)ccc2ccccc2n1 42057,C12(C(=O)NC3CC(CC(C)(C)C)C3)CC(NC(=O)CSCC(N)=O)(C1)C2 42058,C1(CC(=O)NCCCCCNC(c2nc(C)n(C)n2)=O)(NC(C)=O)CCCCC1 42059,c1(OCCOC)cncc(C(=O)NC2CCC2CNC(C2CC(O)C2)=O)c1 42060,N1(C(C=CCOC)=O)CC(NC(=O)COc2cc(C)on2)CC(C)C1 42061,c1(C(=O)NC2(CC=C)CCC2)c(CNC(=O)C(C#N)CC)cnn1C 42062,C12(CNC(=O)COc3ccon3)CC(CN1C(=O)C=Cc1nccs1)C2 42063,CC1(C)CCC(C(N2CC(CNC(C3COCCO3)=O)C(O)C2)=O)C1 42064,C1(CNC(C(C)=CC2CC2)=O)C(C)CCCN1C(c1cccnc1)=O 42065,C=C(C)C1OCCC1C(N1CC(OCC(=O)NC2(C)CC(C)C2)C1)=O 42066,N1(C(CN(C)C2CC2)=O)CCC(CNC(c2csc(Cl)c2)=O)C1(C)C 42067,C1(F)(C(N(C2CCN(C(c3cnc(C(N)=O)s3)=O)CC2)CC#C)=O)CCOCC1 42068,C1(CC=C)(NC(=O)NCC)CCN(C(c2cccc(-n3nnnc3O)c2)=O)C1 42069,c1(C=O)nn(C)cc1C#C.C1(OCC#C)CC(CCC(=O)NC2CN(C3CCC3)C2)C1 42070,C(c1ccc(F)cc1)=C(C)C(N1CCC(C)(C)C1CNC(=O)C=CC1CCOC1)=O 42071,Cn1cncc1C(=O)NC1CCCC1C(=O)NCCN1CCNC1=O 42072,C1(C(N(C)Cc2scc(C)c2)=O)C=CCCN1C(C1CCSCC1)=O 42073,c1(CNC(c2c(C(C)NC(C(CSC)OC)=O)noc2)=O)ccnc(F)c1F 42074,c1(CC)c(C(=O)NC2CCCCC2CNC(C2(C)CC2)=O)ccn1C 42075,N1(C(CN(C(=O)CN2CCN(C)CC2)C)=O)CCC(C)(CC2CC(C(N)=O)C2)C1 42076,Cc1c(F)cc(CNC2(C(=O)Nc3cnn(-c4ccncc4)c3)CCC2)cc1Br 42077,c1(C(N2CCCC(N(C(=O)C#CC3(C)CC3)CC)C2)=O)nn2c(c1C)CCCC2 42078,CCC(C)(C(=O)Nc1cccc(NC(=O)C(N2C(=O)CCC2=O)C)c1)OC 42079,C1(CCC2N(C(C(=O)N(C)C)=O)CCC2)CCCCN1C(=O)C=Cc1cocn1 42080,C(=O)(C(C)(C)CF)NCC(CCOC)NC(C1(N2CCCC2)CCC1)=O 42081,Cn1ncnc1C(c1nnnn1C)NCC1(C2CC2)CCCO1 42082,C(=O)(CC(C)C(F)(F)F)N1C2(C(N(CC#C)CCF)=O)CC2CC1 42083,Cc1ccoc1C(=O)NC1CCC(C(=O)NCCC2CC=CCC2)C1 42084,c1(CC(=O)NCC(CC=C)NC(=O)CCCn2cc(CO)nn2)cnn(C)c1C 42085,CC1(C)CN(C(=O)Nc2cnn(C(C)(C)C)c2C(F)(F)F)CCS1(=O)=O 42086,c1(CCC(=O)OCC)nc2cc(-c3cc(CO)ccc3F)ccc2o1 42087,CC(C)C(C(C)NC(=O)C=CCF)NC(c1cc(C2(C)CC2)on1)=O 42088,O=C1CC(C(=O)NCC2(C3CC3)CCCO2)N(C(C2CCCCC2)=O)C1 42089,c1(C(=O)NCC(N(C(C2(CC#C)CC=CC2)=O)C)C2CC2)ccc(SCC)cc1 42090,C1(NC(C2(OC)CC2)=O)CC(NC(c2noc(C3CC3)c2C)=O)C(O)C1 42091,C1(C(=O)NCC2(C(C)C)CCCC2)CN(C(c2ccc[nH]2)=O)C2(CCC2)C1 42092,O=S(=O)(c1cccc(=NC2C=CCCC2)[nH]1)NC1(c2ccc(F)cc2)CCC1 42093,c1(CCC(=O)N(CC(C)O)CCNC(=O)CP(C)(C)=O)ccc(Cl)cc1F 42094,c1(CC(=O)NCCCN(C(CCC)=O)C2CCCC2)coc2cc(Cl)ccc12 42095,C=CC(C)CC(=O)N(C1(C(=O)NCc2ccc(Cl)cn2)CCC1)C1CC1 42096,C12(CNC(c3cccc[n+]3[O-])=O)CCCC(CN1C(C1CCCCC1)=O)C2 42097,C(C(CC(C)C)C(=O)N1CCCC(N2CCCCC2=O)C1)n1cc(OCC)nn1 42098,N1(C(CSCC#C)=O)CC(C2CC2C(N2CC(N3CC(O)C3)C2)=O)C1 42099,c1(C(=O)NC2(C)CCN(C(C(CCC)N(C)C)=O)C2)c[nH]c2ncccc12 42100,c1(C(=O)NCC(CNC(CC(C=C)c2ccccc2)=O)F)cc([N+](=O)[O-])oc1C 42101,C1(N(CCC)C(C2CC2(C)C(F)F)=O)CCN(C(c2scnc2C)=O)CC1 42102,c1(C(N(C)CC2CCN(C(CC3(COC)CC3)=O)C2)=O)cncc(OC)c1C 42103,C1(NC(C(C)NS(CCC)(=O)=O)=O)CC(NC(=O)CCNC(C)=O)CC1O 42104,C1(CC=C)(NC(c2cc(Cl)cnc2O)=O)CCCN(C(=O)CSCCC(C)C)C1 42105,c1(CC(=O)NCCC2N(C(C=C(C)C)=O)CCC2)ccc2c(c1)CCCC2 42106,N1(C(C(n2cc(C3(O)CCCC3)nn2)C)=O)CCC(CC2N=N2)C1C(C)(C)C 42107,C(=O)(C(O)CC(C)(C)C)NC1CCC(CNC(C2CC(C)OC(C)C2)=O)C1 42108,C1(C(=O)NC2COCCN(C(c3ccc(CC)[nH]3)=O)C2)CC2(CCOCC2)CO1 42109,N1(C(c2c(NC)snc2C)=O)CC(NC(=O)Cn2cnccc2=O)C2(CC2)C1 42110,c1(C(=O)NCC2CN(C(c3c(OC)n[nH]c3)=O)C(C)C2)nccc2[nH]ccc12 42111,c1(C(=O)NCC2C(NC(c3c(CC)scn3)=O)C2)c(C)nn2cccnc12 42112,Cc1ccc(Cl)c(C(N2CC(NC(=O)CN3C(=O)C=CC3=O)C(F)C2)=O)c1 42113,c1(CC(=O)N(C)CC2CCN(C(C3CC(C)(C(=O)OC)C3)=O)C2)cnn(C)c1C 42114,c1(CC)ccccc1C(=O)NC(CCF)C(=O)N(CCC1CC1)CC 42115,C1(CC(=O)NC2C(CNC(=O)CNC(=O)Cn3cncn3)C2)CN2CCN1CC2 42116,C1(CC(=O)NC(C)C(=O)NCCN(C)C(c2ccccc2)=O)CCCCC(=O)N1 42117,C(=O)(CCCCCCCNC(=O)CC(O)C(C)CC)N(CCCCC)CCO 42118,C=CC1(CC(=O)NCC(c2ccccc2)NC(=O)CC2(O)CC2)CCCCC1 42119,CCCCC(O)C(=O)NC1COCCN(C(C2CCCCN2C)=O)C1 42120,C1(NC(=O)CCCn2c(O)nnc2O)COCCN(C(c2ccsc2CO)=O)C1 42121,c1(Cn2c(C3(NCc4sccc4)CN4CCC3C4)nnn2)ccc2cccnc2n1 42122,N1(c2nc(OCC)c(C)cn2)CCC2(NC(c3ncccn3)=O)CCCCCC12 42123,Cc1ccc(C(=O)N(CCCCCC(=O)NCC2CCC(F)C2)C)nc1C 42124,N1(C(C=C(CC)C)=O)CCN(C(C2(C(C)(C)O)CC2)=O)CC12CC2 42125,O=C1NCc2ccc(NC(=O)CC3CCCC(C(F)(F)F)C3)cc21 42126,c1(C(N(C2CC(NC(c3cc(C)c(C)[nH]3)=O)C2)C)=O)coc2c(F)c(Cl)ccc12 42127,N1(C(CC2C(C)CN(C(=O)CN3CCNC(=O)C3)C2)=O)CCC2CCCC12 42128,C(=O)(C1=CCCCC1C)N1CC(N(C(CSc2cccc(OC)c2)=O)C)C(F)C1 42129,c1(C(N2C(CNC(Cc3cc(C)[nH]n3)=O)CC(F)C2)=O)c(F)c(F)cc(F)c1F 42130,C(C(CC=C)C(=O)NCc1ncsn1)NC(C(C)=CC=C)=O 42131,c1(CCN(C2CCNC2)CC(=O)NCc2nn[nH]n2)ccccc1 42132,C1(NC(=O)NCCOc2cccc(O)c2)CCC2(CC1)OCCO2 42133,c1(CC(=O)NC2CCN(C(c3cocc3C(N)=O)=O)CC2)ccccc1Cl 42134,CC1CCCCC1C(=O)NC(C1CN(C(C2(C)CCCCC2)=O)C1)C 42135,Cc1nc(CNC(=O)C(c2cn(C)nn2)NC(=O)CC2(C#N)CC2)cc(O)n1 42136,c1(SC(C)C)ncccc1C(=O)NC1CC(C)(NC(=O)CNC(=O)C(F)(F)F)C1 42137,N1(C(c2cccc(C)n2)C(=O)NC2CC2)CCC(F)(F)C2(CC1)NC(=O)NC2=O 42138,c1(C(N(C2CCC(NC(=O)Cn3cnc(Br)c3)CC2)C)=O)ccnnc1O 42139,c1(C(=O)NCCN(C(c2n(C=C)nnc2)=O)C(C)C)cc(Cl)cc(C)c1C 42140,c1(C(C)C)ccc2occ(-c3nc(CN4CCOCC4)nn3C3CCOC3)c2c1 42141,N1(C(c2c(C)csc2)=O)CC(NC(c2cc(C(C)(C)C)no2)=O)CCC(O)C1 42142,CC1(C(=O)NCc2ccccc2O)CC(C2CC2)=NO1.c12cccc(c1)NC2=O 42143,Cc1c(C(=O)OC(C)C(=O)Nc2ccccc2)c(=O)oc2ccc(Br)cc12 42144,C1(N(C)C)CN(C(C2CC23CC(NC(=O)CCCC2CCCO2)C3)=O)CC12CC2 42145,N1(C(c2c(CC)nn[nH]2)=O)CC(CNC(=O)Cc2c[nH]nc2O)CCC1C 42146,N1(C(C2OCC(C)(C)C2)=O)CC2(CC2)CC1CNC(c1cc2n(n1)CCC2)=O 42147,C1(NC(C2(C)CCC(=O)N2)=O)CCN(C(c2cnc(C3CC3)nc2)=O)CC(O)C1 42148,c1(C(N2C(CNC(C(C(C)(C)C)O)=O)C3CCC2C3)=O)sc2ncccc2c1N 42149,CC1(C)CNc2ccc(C(=O)NCC(F)CO)cc21 42150,C1(OC)CCCC(NCC(=O)Nc2cccc(I)c2)C1 42151,C1(NC(Cc2cc(C)on2)=O)CCOC(C(=O)NCc2ccc(Cl)cn2)C1 42152,CC(C)C(C(=O)NCC(C)CN(C)C(C1CN(C)C1)=O)C1CCC1 42153,C1(OC)CS(=O)(=O)CC1NC(=O)NC(c1ccc(Cl)nc1)C 42154,c1(C(=O)NC2CN(C(C3(CC#C)CCCCO3)=O)CC2F)cncc(C)c1Cl 42155,C(=O)(CC(C)(O)C(F)(F)F)NC1CCC(CNC(CCN(C)CCO)=O)C1 42156,N1(C(c2cc(C)nc(O)c2)=O)CC2CCC(C1CO)N2C(c1ccnc(O)c1)=O 42157,C(=O)(C1CC(=O)Nc2ccccc21)NC1C(NC(CN(C)C2CC2)=O)C1 42158,C1(NC(C2(CO)CCN(C(CN(C)C(N)=O)=O)C2)=O)CCCCC1C#N 42159,C(N=c1[nH]c(=NCC(C)C#N)[nH]c2c1SCC2)c1c(C)ccnc1C 42160,c1(OC)c(NC(=O)C=C2CCN(Cc3c(Cl)ccnc3Br)CC2)cccc1C#N 42161,C1(C)(C(=O)NCCC(C)(C)NC(=O)C(C2(O)CCCC2)F)CC(C(C)(C)C)=NO1 42162,C(c1ccccc1F)=CCC(=O)NC1CN(C(C2(CCCC)CCC2)=O)CC1F 42163,CCC(C)(C)C(=O)C(=O)N1CC(C(=O)NCC2(CO)CC2)C(F)(F)C1 42164,c1(C(=O)NCC(c2cc(OC)c(C)cc2)=O)cnc2onc(C(C)(C)C)c2c1 42165,c1(C(N2CC(O)(CN(C(CC=CC)=O)C)C2)=O)ccc2c(c1)CCCS2(=O)=O 42166,C1(OC)CC(NC(=O)C2=CCC2)C12CCN(C(=O)CC1(O)CCCCC1)CC2 42167,N1(C(C2(C(=O)OC)C=CCC2)=O)CC(C2(NC(=O)C=Cc3ccoc3)CC2)C1 42168,CON1CCC(NC(=O)C(c2cn(C)nn2)NC(c2ccc(Cl)cn2)=O)CC1 42169,C1(CNC(CSC)=O)(CNC(C2CNC(=O)O2)=O)CCOCC1 42170,C1(NC(c2cc(SC)oc2C)=O)CCN(C(=O)C(C)NC(=O)C(C)(C)C)CC1F 42171,Cc1c(C(=O)NCCC2CC(NC(=O)C(C)c3cccs3)C2)cnn1CC(F)F 42172,N1(C(N2C(c3n(CC)cnc3)CCCC2)=O)CCCc2ccc(F)cc21 42173,C1(C(NOC)=O)CC(C)N1C(c1cncn1C)=O 42174,N1(C(c2nc(CC)sc2)=O)CCC(C2CCCN(C(C3(O)CC3(C)C)=O)C2)CC1 42175,C(=O)(C(C)C(C)(C)C)N(C(C)CN(C)C(c1cn(C)nc1C(C)(F)F)=O)C 42176,N1(C2(C(=O)NCCC(C)NC(c3cc(C4CC4)n(C)n3)=O)CC2)CCCCC1=O 42177,Cc1cn2c(C(=O)NCC(C)CNC(=O)COc3cccc(C)c3F)cnc2s1 42178,c1(C(=O)Nc2nc(COCC)nc(O)c2)cc2cc(C)ccc2cn1 42179,c1(NC(C(C)N(C(C2(C#N)CC23CCC3)=O)C2CC2)=O)cnc2ncnn2c1 42180,C1(CC)CC(C(=O)NC(c2ccnn2C)C(N2CC(F)(F)C2)=O)CCO1 42181,N1(Cc2ccc(N3CCCC(C(C)=O)C3)o2)CCCc2ccccc21 42182,Cc1cc(CNC(C2CC(NC(C3(N(C)C)CCOCC3)=O)CCO2)=O)ncn1 42183,C1(CC)(CC)CNC(=O)C1NC(c1cc(OC)c(Br)s1)=O 42184,c1(OC)ccc(C(C)NCC2CC(F)(F)C2(F)F)c(OC)c1 42185,C(c1cc(C)ccc1OC)=CC(=O)NC1C(CNC(CC=CC)=O)COC1 42186,c1(C(=O)NC(c2cccc(Cl)c2)CNC(CN(C2CC2)CC)=O)nc(C)nn1C 42187,N1(C(c2cccc(CC)c2)=O)CCC(F)C(NC(C2CCCCC2CC)=O)C1 42188,CCCC(O)CC(=O)NC(CNC(C1CCCS1)=O)(CC)CC 42189,c1(CC(=O)OC)ccc(NC2C3COCC23)c(C)c1 42190,CC(C)CCCCC(=O)NC1(CNC(=O)C(C)C2CC2)CCCC1 42191,Nc1c(Cl)cc(C(=O)NCC2(F)CC(NC(C3CC3[N+](=O)[O-])=O)C2)cc1[N+](=O)[O-] 42192,N1(C(c2ccc(CC)cc2)=O)CCN(C(=O)CCc2cccnc2)CC1C#N 42193,Cc1nc(C)c(F)c(=NCC(C(C)(C)C)NC(c2cccc3c2C(=O)NC3)=O)[nH]1 42194,c1(C(N(CC(C)NC(=O)Cn2cc(CN)nn2)C)=O)csc(CO)n1 42195,C1(NC(C2(COC)CCCC2)=O)CC(NC(=O)C(C)(C)Cn2cccn2)C12CCC2 42196,C1(C(C(=O)NCC)N(C2CC(C)CC(C)C2)C)OCCOC1(C)C 42197,CN1CCOC(CNC(C2CCN2C(=O)CN2CCOCC2)=O)C1 42198,N1(C(CN(C)C(N)=O)=O)CC2CCC(NC(c3c(Cl)ccnc3F)=O)CC2C1 42199,c1(C(C(=O)NCC(O)CN(C(=O)CCOCC2CCC2)C)OC)cnn(C)c1 42200,N1(C(C2C(CC)N(C(=O)Cc3cscn3)CCC2)=O)Cc2cnn(C)c2C1 42201,C(=O)(C(C1CCC1)NC(=O)C=CC(F)F)NCCCOC 42202,n1(CC)cc(Cl)c(C(=O)N(CC(C)NC(=O)CC(c2ccccc2F)C)CC)n1 42203,C1(O)(CC=C)CCN(C(=O)C(C)(C)C(=O)NC2CCCC2)CC1 42204,C(CCCCCCCO)=CC(=O)NC1C(CNC(C(COC)(C)O)=O)CC1 42205,CC1C(NC(C2CCCC2)=O)CC2CCC1N2C(c1ccc(C(F)F)o1)=O 42206,c1(C(=O)NCC(CCC)NC(C2CCCC2F)=O)cc(C)c(C)o1 42207,CC1CCCN(C(C2COCCN2CC(F)F)=O)C1CNC(C1CCOC1)=O 42208,C(CC(C)C)(C(=O)NC1(C(=O)NCc2cccc(Cl)n2)CCC1)OC 42209,N1(C(C2C(CNC(CC(C=C)CCC)=O)OCC2)=O)CCc2cc(C)ccc21 42210,c1(CC)cccc(CNCC2CC2)n1.C12CCC(CC1)CC(=O)N2CCO 42211,C1(NC(c2c(C)nsc2C)=O)CC12CCN(C(c1cnn3ccn(C)c13)=O)CC2 42212,N1(C(CC2CCCN(C(C(CC)(C)COC)=O)C2)=O)CC(C)N(C)C(C)C1 42213,C(C(C)(C(=O)N(CC(C)(C)CO)C)NC(c1cc(=N)[nH][nH]1)=O)SC 42214,C1(C(N(C)Cc2cccnc2O)=O)CCCC(NC(=O)C=Cc2cscn2)CC1 42215,N1(C(C(C)NC(CC)=O)=O)CC2CC(NC(c3coc(C4CC4)n3)=O)CC1C2 42216,c1(C(N=c2[nH]nc(C(CC)CC)s2)=O)cc2c(cc1Cl)NC(=O)C2 42217,N12CC3CCCC3(C1)C2=O.CC1(C#N)CCN(C(=O)CNC(CC(F)F)=O)C1 42218,CCC(O)C(F)(F)C(=O)N1CC(CCNC(=O)C(CC)c2ccccc2)(OC)C1 42219,c1(NC(C(=O)NC(CC)CNC(=O)CCCn2cncn2)=O)c(C)cccc1C 42220,C1(O)(CNC(C(CC)(C)F)=O)CCCN(C(=O)CN2CCCCC2=O)CC1 42221,N1(C(CC2(C)CC2)=O)C2CCC1CC(CNC(=O)CCCC1CCCC(=O)N1)C2 42222,C(CNC(C1(Cl)CC1(F)F)=O)(CC(=O)NCCc1cnn(C)c1C)OC 42223,C1(CC)(NC(c2cc(OC)cs2)=O)CCN(C(C2CCCC23CC3)=O)CC1 42224,CCCC(C)(C)CC(=O)N1CCC(NC(=O)CCOCC2CCCO2)C(C)C1 42225,CCCCC(CC)CC(=O)N(C1CC(NC(c2csnn2)=O)C1)C 42226,CC1C(C)N(C(=O)C=Cc2ccco2)CCN1C(=O)C=Cc1ccc(C2CC2C)o1 42227,N1(C(c2c(CC)non2)=O)CC(NC(=O)Cc2ccc(C)cc2)C(C)C1 42228,C1(CCCC)(CC=C)CCCCC1.C1(C)C(CO)NC(=O)C2C(C2)C(=O)N1 42229,Nc1ccc(C(=O)NC(CNC(=O)C(O)C2CC2)CC(F)(F)F)c(Br)c1 42230,c1(N(C)C)ccc(Br)c(C(N2CCC(NC(=O)C(c3cnn(C)c3)O)C2)=O)n1 42231,CCC(CC)C(=O)NCCN(C)CCF.N12CCOCC1c1ccc(n1C)C2=O 42232,C12(CCNC(c3cncc(C)c3)=O)CCC1CN(C(C1CCCN1C(N)=O)=O)C2 42233,C12(C(N3CC(CC(=O)OC)C3)=O)CC1CCN2C(c1ccc(C(N)=O)o1)=O 42234,c1(C(=O)NC2C(NC(c3c(C4(C)CC4)cccc3)=O)C2)ccc2cc[nH]c2c1 42235,C(c1ccc(C)cc1)=CC(=O)NCC1C(C)C1.n1(CNC(C)=O)cc(CO)nn1 42236,N1(C(C2C(C)OCC2)=O)CCC(NC(c2c[nH]cc(Br)c2=N)=O)C(C)(C)C1 42237,c1(C(c2n(CCCOC)nnn2)NCC2CC2)ccc2c(c1)COC2(C)C 42238,CC(C)C(CCNC(C1(c2ccccc2)CC1(F)F)=O)NC(c1cncc(O)c1)=O 42239,Cc1cc(C(N2CCC(C)(CNC(c3cc(F)ccc3N)=O)C2)=O)c(F)cc1Cl 42240,C1(c2n(C(CC)C)nnn2)(NCc2ccns2)CCCN(Cc2ccccc2)C1 42241,c1(NC(C2C(C(=O)NCCc3ccccc3O)C2)=O)cc2ccccc2cc1O 42242,c1(C(=O)NC2(C)CC(NC(C3C(c4ccccc4)(C)C3)=O)C2)ncccc1CO 42243,C1(NC(c2n(CC)ccc2)=O)CCCN(C(=O)CCc2n[nH]c(=N)s2)CC1 42244,CC(CC(=O)N(C1CC(NC(c2sc(Br)cc2Cl)=O)C1)C)C(F)F 42245,C1(C(C(=O)N(CC(C)NC(=O)CSC(F)F)C)OC)CCOCC1 42246,C(C(=O)C(C)(C)CC=C)NC(C1(C#C)CN(C(=O)C(C)=CC(C)(C)C)C1)=O 42247,N1(C(c2c(COC)con2)=O)CCC2CN(C(C3(C(=O)OC)CC3)=O)CC2CC1 42248,C(CN=c1[nH]c(=NCC2CCOCC2)[nH]c2c1CSC2)c1c(F)ccc(Cl)c1 42249,c1(CC)cnc(CNC(=O)COC2CCN(C(c3cc(O)cs3)=O)C2)[nH]1 42250,c1(C(N2CC(CC=C)(NC(=O)Cc3nnc(C)s3)C2)=O)cnnc(SC)c1 42251,N1(C(c2cc(C)[nH]c2C)=O)CCN(C(C2(F)CCS(=O)(=O)C2)=O)CC1C1CC1 42252,c1(C(C(=O)NCC2CCCO2)N(C2(C#C)CC2)C)cc(Br)c(Cl)cc1OC 42253,Cc1ccnc(C)c1C(=O)OCCCOCC1CC1c1cnn(C2CC2)c1 42254,c1(C(=O)NC2C=CCN(C(C(C)OCCC=C)=O)C2)nc2c(s1)COCC2 42255,c1(C(C(=O)NC(COC)C)NC(=O)OC(C)(C)C)cnc(O)nc1O.C(C)(C)(C)O 42256,C(=O)(NNC(=O)Cc1cccnc1)c1cn(CC2C(C)CCCC2)nn1 42257,N1(C(CCCn2cc(CCN(C)C)nn2)=O)CCCC(n2ccnn2)CC1 42258,c1(CNC(C2CC(CCC)C2)=O)cn(C2CCN(C(c3cnc(Cl)s3)=O)C2)nn1 42259,C1(C(N(C(c2cc(C)on2)C)C)=O)CCN(C(=O)C2=CCCC2C)O1 42260,C1(C(N2CC(NC(C3C(C)(C)C3)=O)C(F)C2)=O)CC2(CCCO2)C1 42261,c1(C(=O)NCCC2(C)CCN(C(COC(C)=O)=O)C2)n[nH]c2ccccc12 42262,c1(C(C)C)noc(CCCC(=O)NCC(F)CNC(=O)CN2CC=CC2)n1 42263,C1(NC(c2ccc(CC(C)C)s2)=O)CC2(C1)CC2NC(=O)C(O)C(C)C 42264,CCC(C)C(C(=O)NCCN1CCCC1)NC(=O)NCC1CCCO1 42265,Cn1cc(OCC(N2CC(C)(NC(=O)CCc3cscn3)C2)=O)cn1 42266,CS(=O)(=O)C1CN(C(=O)C=Cc2cnccn2)CC1NC(=O)CN1CCCCC1 42267,c1(CN(C)C)ccc(C(N2CCCC(CNC(=O)C=CBr)C2)=O)cc1 42268,c1(OC)cnc(C(N2CC3C(CNC(=O)C=Cc4ccc(Cl)s4)C3C2)=O)c(F)c1 42269,c1(C(N2C(C(N3CCOCC3CC)=O)CC(=C)C2)=O)cc2cn[nH]c2cc1OC 42270,c1(C(N2C(CNC(c3c(OC)ccs3)=O)CC2)=O)cc(C(F)(F)F)cc(O)c1 42271,C(C1CN(C(=O)CN2CC3CC3C2)CC1C(=O)NC1C2CCCCCC12)=CC 42272,c1(C(=O)NCC2CC(COC)CN2C(=O)Cc2cncnc2)cccn(C)c1=O 42273,CCCCCCCCCCS(=O)(=O)N1CCCC(CN2CC(NS(C)(=O)=O)C2)CC1 42274,N1(C(C=C(C)C(F)F)=O)CC(NC(c2n[nH]c3c2CCC3)=O)CC12CCCCC2 42275,C1(=CC(=O)NC2(CCCNC(CC3C(CC)C3)=O)CC2)CCOCC1 42276,N1(C(c2cc(COC)[nH]n2)=O)CCCC1(C)CNC(=O)C#CC1CC1 42277,C1(C2CCC2)(C(N2CCC(OCCNC(CC3CCC(C)O3)=O)C2)=O)CC1 42278,N1(CC(C)(C)N(C)C)CCC(NC(C2(C(N(CC(=O)NC)C)=O)CC2)=O)CC1 42279,C1(C(C)NC(C2CCC(C(=O)OC)O2)=O)CCN(C(c2cncnc2C)=O)CC1 42280,c1(C(=O)NCCC2(C(N3C(C=C)CC3)=O)CCCC2)cnn(C)c1C 42281,C1(OCC(=O)NC(C2CCCN2C(=O)C=Cc2c[nH]cn2)C)CC(F)(F)C1 42282,N1(C(c2cc(C)c(Cl)cc2)=O)CC2CCC(C1)N(C(=O)CCC(F)(F)C(F)F)C2 42283,c1(CC(=O)NCC(CNC(=O)C=CC2CCCC2)OC)ccccc1CC#N 42284,Cc1c(-c2cn(CCOc3ccccc3)nn2)c(=O)oc2ccc(O)cc12 42285,C(=O)(CCCCCCN=[N+]=[N-])NC1C(C)CN(C(=O)CN2CC(C)(C)C2)CC1 42286,N1(C(C2C(O)CCN2C(c2cccc(O)c2)=O)=O)CCC2(CCCC2)C1 42287,c1(CCNC(C(=O)N(C(c2c(C)cccc2)C)C)=O)ccc2c(c1)CC(C)O2 42288,c1(SCCC(=O)NC2CN(C(CC3CC(=O)NCC3)=O)C2)ncnc2[nH]cnc12 42289,N(C(=NCCN1CCOCC1)NCC1CCC(F)C1)CC(c1ccccc1)OC 42290,C#CC1(NC(=O)C(O)CCNC(c2cccc(=O)o2)=O)CCOC1 42291,N1(C(C(CCC)(C)O)=O)CCN(C(=O)C(n2nccc2C)C)CC(C)(C)C1 42292,C1(CNC(c2scc(C(N)=O)c2)=O)CCCN(C(=O)C(=O)NCC(F)F)C1 42293,CC(C)(C)C(CNC(=O)C=Cc1nccs1)C(=O)NCCCCCCF 42294,c1(C(N2CCCN(C(C(C(C)C)F)=O)CC2)=O)coc2cc(F)ccc12 42295,C(=O)(C1=CC2CC=CCC12)N1CC(NC(c2n(C)ncc2C2CC2)=O)C1 42296,CCC(O)C(=O)NC1CC(C(=O)NCC2(c3ccccc3)COC2)C1 42297,Cc1ccc(F)cc1C(N1CC2(CNC(c3cc(Cl)c(Cl)n3C)=O)CCC1C2)=O 42298,C1(NC(C2C(CNC(C(CC)(C)C)=O)CCC2)=O)CCCOC12CCC2 42299,C1(C(=O)Nc2cc(Br)ccc2I)CC1N=c1[nH]c(C(F)(F)F)nc2ccccc12 42300,c1(NC(c2nnc3ccccn23)CCC)nccc(=NCCCNC(C)(C)C)[nH]1 42301,C1(C(N2CCC(N(C(CCCC)=O)CC3CCCO3)CC2)=O)CN(C)CC(C)O1 42302,CN1CC(O)CC1C(=O)NCCN(CCOCCO)C(C1C(CO)C1(F)F)=O 42303,C1(C2(O)CCN(C(=O)C(C)C#N)CC2)(NC(c2ccc3nnc(C)n3c2)=O)CC1 42304,C1(c2ncc(C)s2)CCCCN1CC#CC(C)(C)C 42305,C1(NC(c2c(C(C)C)c[nH]n2)=O)CN(C(=O)CCc2ccnn2C)CC2CC12 42306,c1(C(=O)NCCC2(O)CCCN(C(C(CC)(C)C)=O)C2)cc(O)cc(F)c1F 42307,N1(C(C(C)OCOC)=O)CCC(C(=O)N(C)Cc2cnnn2C)C(C)(C)C1 42308,N1(C(c2cc(F)c(F)cc2F)C(=O)NCCCF)CCc2cccc(Br)c2C1 42309,C1(C(=O)NCC2CCN2C(C2CCCC23OCCO3)=O)CCCC12CCOCC2 42310,C1(OCC(C)C)CCCN(C(C2CCCC(N(C)C)C2)=O)C1 42311,c1(C(N2CCC(NC(CC3C(C)C3)=O)C(C)(C)C2)=O)n[nH]c2ccc(F)cc12 42312,c1(NC(C2CCCC(NC(C3CC(O)C3)=O)C2)=O)ccc(Br)c(Cl)c1 42313,c1(CC)nn(C)cc1C(=O)NC(C)(C)CC(=O)NCC(O)C(F)(F)F 42314,CCC(C)(CCC(C)C)C(=O)N1CCC(CC(=O)NCC2CCNC(=O)C2)C1 42315,c1(C(=O)NC2CC(CNC(C3C(CC)OCC3)=O)C2)cc(C)cc2c[nH]nc12 42316,C1(NC(c2n(C(C)C)ncc2)=O)C2CCC1CN(C(c1ccc(F)cc1Br)=O)C2 42317,c1(C(N2C(CNC(CC(C)(C)OC)=O)CCCC2)=O)ccc2c(c1)C(=O)NC2=O 42318,Cc1cc(C(N2CCCC2CCNC(=O)CS(=O)(=O)N(C)C)=O)nc(O)n1 42319,CC(CC(=O)NC1CCCC1NC(C1(CF)CC1)=O)n1cccn1 42320,O=C(C#CC1CCC1)N1CCN(C(C2CC(CF)C2)=O)C(C2CCCC2)C1 42321,Cc1ccc(OCC(N2CCC(CNC(C34CC(CF)(CO3)C4)=O)C2)=O)c(C)c1 42322,Cc1cc2[nH]c(C(N3CC4(CC(NC(c5c[nH]c(=O)cn5)=O)CO4)C3)=O)cc2s1 42323,c1(N2CC(NC(C=C(C)Cl)=O)CC3(C2)CC3)nc2cc(F)ccc2o1 42324,c1(CSCCC)ccc(NC(=O)NC2(O)CCCSC2)cc1 42325,CCCC(CC)C(=O)NC1CCOC1C1CCN(C(C2C3CCCC23)=O)CC1 42326,C(=O)(C(F)C(F)(F)F)N(CC(CC)NC(C1(c2ccncc2)CC1)=O)C 42327,CC1(C)CC(NC(=O)C(C)(F)C(F)(F)F)CCN(C(c2ccns2)=O)C1 42328,Cc1nc(C(=O)NCC2(C)CCN(C(=O)Cc3cnc(C)s3)C2)c2ccnc-2[nH]1 42329,c1(N2CCN(C(=O)Nc3cccc(F)c3)C3C2C3)ncnc2sccc12 42330,C1(NC(C(COC)OC)=O)CN(C(c2ccccc2OC(F)(F)F)=O)CCC1O 42331,C12(CC(=O)NCC3(F)CC(CNC(c4ncccn4)=O)C3)CCC(CC1)OC2 42332,c1(C(=O)NC2CC(CNC(C(CCC)C)=O)C2)ccc2nc(O)cn2c1 42333,c1(C(N(C)CC2N(C(C(C)(CO)OC)=O)CCC2)=O)cc2c(cn1)COCC2 42334,c1(OC)cc(OC)c(CN2CC3CC(CN)C3C2)c(OC)c1 42335,C1(C(N(CCCNC(c2cn(C)nc2C(F)(F)F)=O)C)=O)CCOC(=O)CC1 42336,CC(C(=O)NCC1(F)CN(C(c2ccc(SC(F)(F)F)s2)=O)C1)S(N)(=O)=O 42337,c1(C(N2CCC(COC)(NC(=O)CC(C)SC)CC2)=O)cccc2c1COC2 42338,N1(C(CCC2(NC(C(C)CC3CC3)=O)CCCC2)=O)C2C=CCC1CC2 42339,c1(C(=O)NCCN(C(=O)CN2CCC(C)C2)CCOC)nccc(Br)c1C 42340,C1(NC(CNC(C(c2ccccc2)C)=O)=O)CC(C)(C)C12CC2 42341,CCCCC(O)CC(=O)N1CCCC(NC(=O)Cc2c(F)cccc2F)C1 42342,C1(CNC(CCC#C)=O)CC(F)(F)CN1C(=O)C=Cc1scnc1C 42343,Cn1oc(C(=O)NCCC2CCN(C(=O)COCC3CCC3)C2)cc1=O 42344,N1(C(C2CCC(CC)CC2)=O)CC(C)N(C(c2nnn3c2CSCC3)=O)CC1C 42345,C(=O)(C#CC1CCCCC1)NC1(C)CC(C(=O)NC(CC=C)CC=C)C1 42346,C1(NC(C(C=CC)O)=O)CCC12CN(C(C1(C(N3CCCC3)=O)CC1)=O)C2 42347,C1(C(=O)NCc2c(C(=O)NCCCn3cccn3)nco2)(CC)CCCC1O 42348,n1(CCOC)ccc(C(=O)NC2(C3CCCN3C(=O)C(N)=O)CC2)n1 42349,Cc1ccc(C(=O)NC2(C(=O)NCc3ccc(CO)o3)CCCC2)c(O)n1 42350,C1(NC(=O)C(=CC2CCCCC2)F)CCN(C(=O)C(F)OC(F)(F)F)C12CC2 42351,NS(=O)(=O)C1CN(C(=O)CSCc2cn(C3COCCC3O)nn2)C2(CCC2)C1 42352,CC1CC2CN(C(c3cnc4[nH]cncc3-4)=O)CC2N1C(=O)CCCCCCF 42353,C1(C)(C(c2n(CC(=C)C)nnn2)NCCc2cnoc2)CCCC(F)(F)C1 42354,c1(C(=O)NS(=O)(=O)CCC2CCCOC2)cccc(C(F)(F)F)c1 42355,c1(CC(=O)NC2CCN(Cc3cn(C(C)(C)CO)nn3)C2)c(F)cc(Br)cc1F 42356,c1(C(N2CC(O)(CNC(=O)C=Cc3cc[nH]c3)C2)=O)ccc2c(O)nncc2c1 42357,C(CC(=O)N1CCOC(CC)CC1)(C(F)(F)F)NC(C(CCCC)N(C)C)=O 42358,c1(OC)cccc(N(C)C)c1S(=O)(=O)Nc1csnn1.C12C3CN(CC13)C2=O 42359,C1(N(CC)CC)CCN(C(=O)C(=O)NC2CC2)CC1.c1(C2C(=O)N2)ccnn1C 42360,C(=O)(CCCC(F)(F)CO)NCCOCCCNC(C1C(C)OC(=O)N1)=O 42361,CCC(C)(C(=O)NCC1CC(NC(=O)CCc2cn(C)nn2)C1)OC 42362,c1(CC)cc(C(=O)NC2CC23CCN(C(=O)CCC2CC(OC)C2)C3)ccc1F 42363,Cc1ccc(C2(CC(N3CCN(CC4CCCS4(=O)=O)CC3)=O)CC2)cc1 42364,c1(OC)ccc(CN2CCN(C(C3CCCC(C)O3)=O)C(C)C2)nc1Cl 42365,c1(CC(=O)NCC2CC2CNC(c2cnoc2C2CC2)=O)cccc2ccoc12 42366,C1(CC(=O)NC2CC=C(C)CC2)N(C(c2csc(F)c2)=O)CCC1(C)C 42367,N1(C(c2c(C)n[nH]c2)=O)Cc2cccc(CNC(c3cc(F)ccc3Cl)=O)c2C1 42368,Cc1c(CN2CCC(SC(C)(C)C)C2)occc1=O 42369,C(=O)(C(CCO)c1ccccc1)NC(C)CN(C)C(c1ccc(CCF)cc1)=O 42370,N1(S(CCNC(C(C)C)=O)(=O)=O)CCCCCC1NC(=O)C(F)(F)F 42371,C1(NC(C2C(C)CCN2C(C2C3CCCC23)=O)=O)CC2(C1)CC(C)(C)C2 42372,C(C(F)(C(=O)NC(COC)COC)C(C)C)NC(c1c(CCC)nco1)=O 42373,c1(C(=O)NCC(C2CCC2)NC(c2c(C(C)(C)C)ncs2)=O)cc[n+]([O-])cc1 42374,N1(C(c2cnn(C(C)C)c2N)=O)CCC(NC(=O)CC2CNC(=O)C2)CC1C 42375,C12(CNC(C3(OCC)CC3)=O)COCC1CN(C(=O)C(C1CC1)OC)C2 42376,C(CCCCCN(C)C)NC(C(C1CCCO1)NC(c1c(C)occ1)=O)=O 42377,c1(C(=O)NCC(C2CCOC2)NC(c2ccon2)=O)snnc1-c1ccccc1 42378,C(=O)(C(C)(C)C(C)C)NC(c1sc(C(=O)NCC(CSC)OC)c(C)n1)C 42379,c1(C(N(C2CCN(C(C(Br)=C(C)C)=O)C2)CCO)=O)cnn2c(N)ccnc12 42380,C1(C(=O)NC2CCN(C(=O)NC)C2)CC1C1CCN1C(=O)CSc1nc[nH]n1 42381,C(=O)(C(O)CCCNC(c1cnnn1C1CC1)=O)N(CCO)CC 42382,N1(C(c2c(C)nc[nH]2)=O)CC(C)C(NC(=O)C2=CCC(C)CC2)C(C)C1 42383,N1(C(c2n(C)nc(O)c2)=O)CCCC(CNC(c2c[nH]c(=N)s2)=O)CC1 42384,c1(-c2nnc(N3CCC(OCC=C)C3)n2CC=C)cc(Cl)ccc1OC(F)(F)F 42385,Cc1c(C(N2CC3CC(C2)N(C(=O)C(C)C#N)C3)=O)cc(Br)cc1Cl 42386,N1(C(C(CCC#C)O)=O)CCCN(C(=O)CCCc2ccsc2)CC1CO 42387,C1(C(=O)NC2(COC)CC=CC2)(CC)CC=CCC1 42388,C(=O)(C1=CCCOCC1)N1CCCC(CC=C)(NC(=O)Cc2cnn(C)c2C)C1 42389,c1(OC)cc(C)sc1C(N1CCCCC1C(C)NC(=O)CC1(O)CCC1)=O 42390,C=CC1(CC(=O)N(CCO)CC2CC2)CN(C(=O)C(C)(C)n2cncn2)C1 42391,C1(CC)CN(C(c2cc(Cl)cnc2OC)=O)CCN1C(=O)Cc1csc(C)c1 42392,Cn1nc(C(F)F)cc1C(=O)Nc1cccc(NC(c2cc(C3CC3)no2)=O)c1 42393,CC(CC1CC1)C(=O)N(CCCOCCNC(C1(C2CCCO2)CCC1)=O)C 42394,N1(C(C(C)(N(C(=O)CCC(=O)C2CCCC2)C)C2CC2)=O)CCC12CCCC2 42395,N1(C(c2n(C)nc(O)c2)=O)CCC2(CCC2CNC(=O)COC2CCCC2)CC1 42396,C1(C(=O)OCc2n(CC)c(=O)sc2)Cc2ccccc2C1C 42397,Cc1cc(C)c2cc(C(N3CC(NC(=O)CC4CCC4)C4CC4C3)=O)sc2n1 42398,C=CC(C)(CCOC)C(=O)NCCC(C)NC(=O)C(C)C(=O)OC(C)(C)C 42399,c1(OC)cc(F)c(C(=O)NCC2CC(C)N(C(c3cc(CF)on3)=O)C2)cc1N 42400,C1(C)(C(N2CCCC(N(C(=O)CSC(C)C)CC)C2)=O)CCC(C)C1(C)C 42401,c1(C(=O)NC(CCC)CNC(=O)C(F)Cc2ccccc2)nccc(C)c1N 42402,C1(CC)CC(C)CN(C(C2(C)CCCN2C(=O)CCC(C)CC)=O)C1 42403,O=C1COc2ncc(C(=O)NCC3C4CN(C(c5cnc[nH]5)=O)CC34)cc2N1 42404,Cc1nc(O)nc(O)c1CCC(N1CCN(c2ccc(C#N)nn2)CC(O)C1)=O 42405,c1(CC)cc(C)c(C(=O)NC2CC(CCn3cc(CC4CCCOC4)nn3)C2)o1 42406,Cc1nocc1CC(=O)N(CCCNC(C1CCCN1C(=O)NC1CC1)=O)C(C)C 42407,Cc1c(C(N2CCC(CCCNC(=O)C(C)n3ccnn3)CC2)=O)nnn1C 42408,C(=O)(C(C(C)(C)C)n1ccnn1)NC1CCC(NC(c2nn(CC)nc2C)=O)C1 42409,C1(NC(C(C)=C(C)C)=O)CCN(C(=O)CCOCC2CC2)CC12CCC2 42410,S(=O)(=O)(c1cccnc1NCC1SCCc2ccccc21)NCC(CC(C)O)(C)C 42411,c1(CC)ccc(F)c(C(=O)NCC2CN(C(=O)CC3CCCC3)CCCO2)c1F 42412,C(c1ccccc1Br)=CC(N1CC2CC2(C(N2CCCCC2CCO)=O)C1)=O 42413,C(CC1=CCN(C(C23CCC(C(=O)OC)(C2)OC3)=O)CC1)NC(C(C(=C)Cl)(C)C)=O 42414,C(=O)(C(C)C(C)NC(=O)C(N)=O)N(CC=C)C 42415,C1(C)(C(N(CCN(C(CCc2onc(C(C)OCC)n2)=O)C)C)=O)CCC(=O)N1 42416,c1(C(N(CCN(C(c2nnn(C)n2)=O)CC)CC)=O)cc([N+](=O)[O-])n[nH]1 42417,C1(C(=O)NCC2CC(OC)CN2C(=O)COC2CCC2)C2CCC1(C)C2(C)C 42418,c1(C(N2CC(SC)C(NC(=O)C(O)Cc3cnc[nH]3)C2)=O)cc(C)cc(C)c1 42419,N1(C(CSCCC)=O)CC2CC(NC(C3(CC#N)COC3)=O)C(C2)C1 42420,N1(C(C(N2CCOC2=O)C)=O)CCOCC1CC(N1CCCC(F)C1)=O 42421,CCC(CC(=O)N1CCN(C)C(C(=O)NCC2(C)CC(C)C2)C1)C(C)(C)C 42422,c1(C(N2CCCC(Cn3cc(C(CC)O)nn3)C2)=O)c(C)[nH]c2ncccc12 42423,C1(NC(C(C=C)(F)F)=O)CC2CC1CN(C(=O)C(CO)OC)C2 42424,CC1CN(C(c2csc(F)c2)=O)C(C)CN1C(c1ccnn1CCF)=O 42425,CCCC(CNC(=O)C=CC1CCOCC1)C(=O)N1CCC(c2cnn[nH]2)C1 42426,C1(CNC(c2c(OC)cnnc2)=O)CC(C)CN(C(=O)Cn2nc(C)cc2C)C1 42427,N1(CC(=O)NC(C(=O)NCCC(=O)OC)(C)C)CCC(F)CC1 42428,CCC(C)(C)CCNC(=O)CCC1CCCN1C(=O)C(C)NC(=O)NC 42429,CN1CCCC(C(C)(C)C(=O)NC2CC(F)(CNC(C3CSCCS3)=O)C2)C1 42430,C(=O)(CCCCCCCSC)NC1C(NC(c2cccc(CC)n2)=O)CCC1 42431,N1(C(C2(CC#C)CCCC2)=O)Cc2occ(C(=O)NCCN3CCCCC3)c2C1 42432,c1(COCCC(=O)NC2(C)CC(NC(C3CCCCO3)=O)C2)cccc(CO)c1 42433,N1(C(c2c(=O)ccn(C)c2)=O)CC2CCC(C1)C2CNC(c1ccn(C)c1)=O 42434,c1(-n2cc(C3(C)CCN(C(c4ncn(C)n4)=O)C3)nn2)cc(F)ccc1C1CC1 42435,CC1(C)C(C(N2CC3CC(NC(=O)CC4CC=CC4)C2C3)=O)CCS1(=O)=O 42436,c1(C(=O)NC(C(C)NC(CCc2c(C)ncs2)=O)CO)ccn2ccccc12 42437,C1(C2(O)CN(C(c3ccc(F)c(F)c3)=O)C2)(CNC(c2n(C)c(S)nc2)=O)CC1 42438,C#Cc1cccc(CC(=O)NC(C)(CNC(C2COC(C(F)F)C2)=O)C2CC2)c1 42439,N1(C(c2c(C)nc(O)cc2)=O)CC2(C(=O)NC(C)C(F)F)CC1CCO2 42440,C1(C(N(C2CCN(CC)C2)C)=O)CC2CC2N1C(c1cc(O)n(CC)n1)=O 42441,N1(C(COCC)=O)CC(NC(=O)CN(CP(C)(C)=O)CC)CC1(C)COC 42442,CC#CCCC(=O)NC(c1ccccc1)CNC(c1[nH]cnc1C)=O 42443,C(=O)(C(C)C(O)CCCC)N(CCNC(c1cccc(C#C)c1C)=O)C(C)C 42444,n1(CC)nc(C)cc1C(N1CC2C(C1)N2C(=O)Cc1csc(C)n1)=O 42445,Cc1ccc(CC(=O)NCC(O)CCNC(C2(N3CCOCC3=O)CC2)=O)cc1 42446,C1(C(=O)NC(CC(=O)N(C2CCN(CC)CC2)C)(C)C)CC2(CCCO2)C1 42447,C1(C(=O)OC)C(F)(F)C12CC(C(=O)NC(C)(CNC(c1cc[nH]n1)=O)CO)C2 42448,c1(C(N(CC(CC)NC(c2n[nH]c(C)c2Cl)=O)CC)=O)ccc2nnnn2c1 42449,c1(-n2c(-c3csc(Cl)n3)nc(-c3scc(C)n3)n2)c(C)cc(C)cc1C 42450,C1(CC=C)CCCN(C(=O)CC(CNC(=O)C(C)C)OC)C1 42451,S(=O)(=O)(c1ccc(C#N)cc1Cl)N1CC(C)C(NC(c2cc(Br)c(Br)[nH]2)=O)C1 42452,C(=O)(C(CC)C(C)O)N1C(CO)CC(NC(CC(=C)C)=O)C1 42453,c1(C(c2nnnn2CCC)NCCC=CCCC)nn(C)c(C)c1Cl 42454,C1(C(=O)NCC2C(C)(C)COC2)CCC2(CC2)N1C(c1cc(C2CC2)no1)=O 42455,N1(C(C2N(S(C)(=O)=O)CC2)=O)CCC2(CCN(C(c3cc(Cl)c[nH]3)=O)C2)C1 42456,n1(CC)c(C(N2CC(C)C2C(=O)N(C2CN(C(C)C)C2)C)=O)cnc1O 42457,C1(C(=O)NC(C(=O)Nc2csc(Cl)c2)c2cccs2)CC1C1CCC1 42458,c1(NCCc2cn(CC)nc2)cc(=NC2CCCN(C)C2)[nH]c(C(C)C)n1 42459,N1(C(c2c(C)nccc2)=O)CCC(C)C(NC(=O)CC2CCCC(F)(F)C2)C1 42460,n1(CC(=O)NC2C(NC(C(C)OCCOC)=O)CCC2)ncccc1=O 42461,C(=O)(C#CC1CCCO1)N1CC(CNC(Cc2[nH]c(=N)sc2)=O)C(C(F)(F)F)C1 42462,Cc1ncn(C)c(=O)c1C(=O)NCCN(C(=O)CNC(C1CCC1)=O)C 42463,C(=O)(C(CC(C)(C)C)OC)N1C(C(=O)Nc2c(CC)n(C)nc2)CCC1 42464,N1(C(C(C)C(C)(C)C)=O)CC(NC(=O)CN2CCCNC2=O)C(S(C)(=O)=O)C1 42465,Cc1nn(C)cc1Cc1noc(C2C3CC(=O)CC23)n1 42466,c1(C(=O)NC2(CC)CN(C(CSCC)=O)C2)cc(NC)nc(Cl)c1 42467,c1(CNC(C(CNC(=O)CCC2CCCN2C)OC)=O)cnccc1Cl 42468,CCC(C)C(C)C(=O)NC1(C(=O)NCCC2CC2C)CCN(C)C1 42469,C(=O)(C(CNC(C1CCCN1C(C1(NC(N)=O)CC1)=O)=O)OC)NC 42470,C1(C(N2CC(NC(CCn3ccc(C)n3)=O)C(C)C2)=O)CC(C)(C)OC(C)(C)C1 42471,Cc1cnccc1C(C)C(=O)NCC(C)(O)CNC(=O)CCc1cccnc1 42472,CCN=C(NCC(C)(CO)c1ccccc1)N1CCOC(C(F)(F)F)C1 42473,C1(NC(COc2cn(C)nc2)=O)CCN(C(=O)C(C)(C)C2CCC2)CC1F 42474,C1(=O)C(CCSC)NC(=O)C2OCCC2N1.C1(C2CC2)(CC)CC1 42475,c1(-c2c(F)ccc(CN(C)C)c2)cccc2c(NC3CC3)cccc12 42476,N1(C(CSS(C)(=O)=O)=O)CCC2CN(C(=O)COCC3CCCO3)CC12 42477,c1(SC)nc(=N)[nH]c(=NC(C)C2CCCN(C(C3C(C4CC4)C3(F)F)=O)C2)[nH]1 42478,C#CC1CCCCN1C(C1(C#C)CCN(C(c2cnn3c2OCC3)=O)C1)=O 42479,C=C(Br)CN=C(N)NC1CC1.c1(C2CC2C)ccco1 42480,c1(CN(C)C)cccc(-c2cnc(NC(=O)NCc3nccn3C)nc2)c1 42481,C1(CCN(C(CCOCC)=O)C)CCCCN1C(c1csc(Cl)n1)=O 42482,c1(C(=O)NCC2(CNC(c3c(OC)c(=O)cco3)=O)CC2)nc[nH]c2ncnc1-2 42483,CC(=O)CCCCCCC(=O)N1CCN(C(C2CC3CC3C2)=O)CCC1C 42484,CC12CSCC1CN(C(=O)C(c1ccccc1)NC(c1cnc(O)o1)=O)C2 42485,N1(CC)C(=O)CCC1C(=O)N(C(C)CCNC(=O)CC1CCCCO1)C 42486,C1(CC)CN(C(=O)C(=Cc2ccncc2)C)CCN1C(c1cccc(=O)n1C)=O 42487,C1(NC(CCC=CC(C)C)=O)CC2C1CCN2C(=O)CC(C1CCC1)C1CCC1 42488,N1(C(C(CC)N(C)C)=O)CC2(CCN(C(=O)Cn3ncnn3)CC2)C2COCC12 42489,C1(C)(C(=O)NC(C(=O)NCc2snc(CC)n2)CC2CC2)CCC(O)CC1 42490,C1(NC(CN(S(C)(=O)=O)C)=O)CN(C(C2CC23CCSCC3)=O)CC1C1CC1 42491,Cc1nsc(C)c1C(=O)NCc1cc(C(N2CCCC2CC2CCC2)=O)n[nH]1 42492,C(c1cc(F)cc(F)c1)=CC(N1CCN(C(C2CC2F)=O)C(CC2CC2)C1)=O 42493,CN1CC(CCNC(=O)CN(C)C(c2ccc(C3CC3)o2)=O)CC1=O 42494,C1(C)(CNC(CCCC#C)=O)CN(C(=O)CCc2ncc(C)[nH]2)CCO1 42495,c1(C(=O)NCC(C)(C2CCC2)NC(CN(C(=O)OC)C)=O)cc2ccnn2cn1 42496,c1(OC)cc(CC2C(C(=O)NC(=O)C3CC3)C2)cc(F)c1OCCC(C)C 42497,N1(C(c2cc(C)[nH]n2)=O)CCCCC1CC(=O)NCCN(CCCF)C 42498,N12CCC3(CCC3N(c3ccccc3Cl)CC1=O)CC2.C(C1CCC1)=CC(=O)O 42499,C1(C(=O)NC(CCN(C(C2(NC(C)=O)CCCC2)=O)C)C)CCS(=O)(=O)C1 42500,C=C=CC(C)C(=O)NCCOCCOCCNC(C1(C#N)CC(C)C1)=O 42501,N1(CC(=O)N(CC(CC)NC(=O)Cc2nccs2)CC)CCCCCC1=O 42502,c1(C2(C)CC(OC(C(c3ccccc3F)OC)=O)C2)cccc(Cl)c1 42503,c1(-c2ncc(CN=C(NC(C)CF)NCC3CC3C(N)=O)s2)c(F)cccc1F 42504,C1(CC)CCCCC1OCC(=O)NC(C1CCN(C(=O)C(=O)NC)C1)C 42505,C12(NC(CCc3n(C)ccn3)=O)CCC1CN(C(=O)CSC1CCOC1=O)C2 42506,c1(C(N2C(C)C(NC(C3CN(C(N)=O)C3)=O)CC2)=O)cc(F)cnc1Cl 42507,C1(C(N2C(C(C)C)C(C(=O)NCc3ncc[nH]c3=O)CC2)=O)Cc2nccn2C1 42508,n1(CC(=O)Nc2c(C)cc(CCC(=O)O)cc2)nc(C(F)F)c2c1CCC2 42509,c1(C(=O)NCC2CCN2C(C23CC(CO2)C3)=O)nc(Br)c2ccccn12 42510,C1(NC(c2cccc(C#C)c2)=O)CN(C(=O)C(C)SC(F)(F)F)CC12CCC2 42511,c1(C(=O)NCCC(CNC(c2nc(OC)c(F)cn2)=O)O)c(F)cc(N)cc1F 42512,N1(C(C2(NC(C(COC)C)=O)CCC2)=O)CC(O)(C2CCC2)C1 42513,N1(C(c2c(OC)cccn2)=O)CCC(C2CC2NC(=O)C(C(C)C)SC)CC1 42514,C=C1CN2C(=O)CCC2(C(N2CC(CCNC(c3sccc3OC)=O)C2)=O)C1 42515,Cc1cccc2c(CC(N3CC4CC4(NC(c4c(Cl)cnn4C)=O)C3)=O)c[nH]c12 42516,N1(C(Cc2c(C)cnn2C)=O)CC2(CC(CC(N3CCCC(C(C)C)C3)=O)C2)C1 42517,c1(C(NOCC(=O)NC(CC#C)C(=O)OC)=O)cc(C)ccc1F 42518,c1(C(N2C(CNC(C(CC)(C)CO)=O)CCCCC2)=O)onc2ccccc12 42519,N1(C(CC(=O)N(CC#C)C)=O)CCC(CSc2nccn2CC)CC1 42520,C1(C(=O)NC2(CN(C(=O)C(C)(C)c3ccn(C)n3)C)CC2)CCCCCC1(F)F 42521,CCCC(CC1CCCC1)C(=O)N1CCC(O)(CNC(c2[nH]ncc2C#N)=O)CC1 42522,CC12CCN(CC1)CC2C(N1CC(F)(CNC(=O)Cc2c(F)cncc2Cl)C1)=O 42523,C1(S(C)(=O)=O)(C(=O)NC(CCCC)CNC(c2cc(C)nc(O)n2)=O)CC(O)C1 42524,N1(CC(=O)N(CCN(C(c2cncc(OC)c2)=O)CC)CC)CCCCS1(=O)=O 42525,N1(C(c2c(NC)nccc2)=O)CCC2CC2(NC(C2(N(C)C)CCCC2)=O)CC1 42526,c1(C(C)N(CCN2CCCC2)C2CC2)cccc(C2CCCC2)c1 42527,N1(C(COCCC=C)=O)CCC(C)(CCNC(c2ccc(OCCF)cc2)=O)C1 42528,C1(NC(CSCCC)=O)CCCN(C(=O)C(c2ccc(OCC)cc2)C)CC1 42529,C(=O)(CC(C(F)F)c1ccccc1F)NC(CC)CN(C(C1CC1(C)C)=O)CC 42530,c1(COC)nc(N2CCCC(N(C(=O)CC3(O)CCC3)C)CC2)cc(Cl)n1 42531,N1(C(C(F)=CC(C)C)=O)CC(C)CCC1CNC(=O)COC1(C)CCC1 42532,c1(CC(=O)NCC(C)NC(c2c(Cl)cncc2Cl)=O)cccc2nonc12 42533,c1(CN(CCN(C(C2(NC)CCSC2)=O)C(C)C)C)ccc(C)c2cccnc12 42534,c1(CC)cccc(F)c1C(=O)NC1(COC)CN(C(C2CCN2C)=O)C1 42535,c1(C(=O)NCC(C)(C)NC(C(C(=O)OCC)F)=O)ccc2c(c1)COCCN2 42536,C=CC1(C(N2CC(CCNC(C3(CCF)CC3)=O)C2)=O)CCCCC1 42537,COn1cnc(C)c1C(=O)NCCCN(C)C(c1sc(Br)cc1C)=O 42538,C1(CC(=O)N(CC(=O)NC(C)CN(C)C)C)(NC(C)=O)CC1 42539,c1(C(=O)NC(CC)(CNC(C2(CO)CC2(F)F)=O)CC)cnc2c[nH]nc2c1 42540,Cc1nc(C(C)(C)C)sc1CNCC1(CNC(=O)Cc2ccsc2)CC1.C1(C)CC1 42541,c1(CC(=O)C(=O)C2CC2)csc(SC)n1.C(=O)(C(O)C1CCC1)NCCCN 42542,N1(C(C2(C(N(C)C)=O)CC2)=O)C2CCC1CC(NC(C1CC13CC3)=O)C2 42543,C1(C(N(CCO)CC)=O)CCOC1CNC(C1C=C(C)CS1)=O 42544,Cc1ncc(C(=O)NCc2ncoc2C2CN(C(=O)C=CS(C)=O)C2)cc1N 42545,Cc1cc(C(=O)NC2CC(O)CN(C(=O)COc3cccnc3)C2)c(F)cc1N 42546,c1(C(=O)NC2C(CC)N(C(C3CCOCC3)=O)CCC2)cc(F)c(C)cc1N 42547,C12(CNC(c3ccc(CC)nc3)=O)CCCC1CN(C(C1CC(C3CC3)C1)=O)C2 42548,n1(CC(=O)NCC2N(C(CCCC=C)=O)CC(F)C2)nc2n(c1=O)CCCCC2 42549,C(C(=O)NCCNC(=O)C(C)Cc1ccc(F)cc1)(C(C)C)NC(C)=O 42550,C(=O)(C(C)(C)CC(C)C)NCC1C(CNC(C(CC)(O)c2ccccc2)=O)C1 42551,CC1(NC(C2CCC(P(C)(C)=O)C2)=O)CCCc2ccccc21 42552,c1(SCC)ccc(C(=O)NC2CCCCC2CNC(=O)C(C)C)cc1 42553,Cc1cc(O)cc(=O)n1CC(=O)NCC1CC(NC(=O)CCC2CCC(=O)N2)C1 42554,C(CC(=O)N(C)CC1CCOC1C)(CC(C)C)NC(C1C(CCC)C1)=O 42555,CCC(CC(=O)NCC(C(C)C)NC(=O)C(CO)C(C)(C)C)C(C)(C)C 42556,C1(OC)(OC)CC(C)(CNC(c2cnn(C(C)C)c2Cl)=O)C1 42557,N1(C(CN2CCN(C)CC2)=O)CCC2CN(C(=O)C(C)(O)C3CCCCC3)CC12 42558,c1(C(=O)OCC(c2c(C)n[nH]c2)=O)cccc2c(N)cccc12 42559,Cc1ccccc1COCC(=O)NC1C2CC1N(C(C1(C)CC(C)C1)=O)C2 42560,N1(C(C2(OC)CCC2)=O)CCC2C(CCN2C(c2cc(C)ncc2Cl)=O)C1 42561,Cc1cc(C(N2CC(C(=O)NCCSC(F)F)CCC2C)=O)nnc1C 42562,Cc1c(C(=O)NC2C=CCC(C(N3Cc4c[nH]nc4C3)=O)C2)cccc1F 42563,c1(SC)cc(N2CCC(C)(CNC(=O)Cc3c(C)noc3Cl)CC2)nc(SC)n1 42564,N1(C(C2(C)CCOCC2)=O)CCCC(NC(=O)CCC2(O)CCC2)CC1 42565,C(=O)(N=c1cc(C)n(CCC#N)[nH]1)N(c1ccncc1)CC=C 42566,c1(CN2CC3C(CNC(c4cc(C(F)(F)F)no4)=O)C3C2)ccc2ncnn2c1 42567,CCCCC(CNC(=O)C(CC)OC1CCCC1)NC(C1CC(F)C(=O)N1)=O 42568,c1(C(N2CC(O)(C(C)NC(C(CSC)C)=O)C2)=O)ccn2cccc2c1 42569,N(C1CN(C(=O)C(O)CC2CC2)Cc2ccccc21)C(c1c(C)nc[nH]1)=O 42570,C1(NC(C2CC(CCC)C2)=O)CCCC(C(N2CCSCC2)=O)CC1 42571,N1(C(C(N2CCC(N)CC2)C)=O)CCC2(CC1)CC(=O)NC(=O)C2 42572,C1(N(C(=O)C(F)F)CC#C)CCN(C(C2(C(C)(F)F)CC2)=O)CC1 42573,N(C1CN(C(=O)CC2(C)CC2)Cc2ccccc21)C(c1cc(C)no1)=O 42574,C1(c2cn(CCNC(c3ccncc3F)=O)nn2)CC2CCC1O2 42575,c1(C(=O)NCC(C)NC(CCC(=O)NCCC)=O)cc(C)c(C)nc1C 42576,c1(CC)c(C(=O)NCCCOCCNC(C2(CSC)CC2)=O)cccc1F 42577,CC1CN(C(c2cn[nH]c2)=O)CC1CNC(C1CCNC(=O)C1)=O 42578,C1(N(C(C=CC(CC)=CC)=O)CC)CCCN(C(c2ccncc2CC)=O)C1 42579,CC1CC(C)(C(N2CC(CC(C)NC(c3csc(Cl)c3Cl)=O)C2)=O)CC(C)O1 42580,CC(C)(C(=O)NCCC1CN(C(=O)COc2ccsc2Cl)C1)C(F)F 42581,c1(C(=O)NCC(=O)NCC(=O)NCc2nc(C)sc2)ccnnc1O 42582,c1(OC)ccc(C(N2CCC(CNC(=O)C(C)OC)(OC)C2)=O)cc1F 42583,c1(NC(CCOCC)=O)cccc(NC(c2snnc2C(C)C)=O)c1 42584,N1(C(CC(C)(C)OC)=O)C2CCC1CN(C(c1cnoc1C)=O)CC2 42585,C1(CNC(C(C2CCOCC2)OC)=O)CC(NC(c2coc(SC)c2)=O)C1(C)C 42586,C(=O)(C(C)CC(N)=O)NC(C1CCN(C(Cc2cccc(C)c2)=O)CC1)CO 42587,N1(C(C(C)C2CCCC2)=O)CC2CC1CC2CNC(=O)C(C)(C)c1cnn(C)c1 42588,c1(C(=O)NCC2(CNC(c3ccc(C)nc3)=O)CCCC2)cc(F)cnc1O 42589,N1(C(C2(Cl)C(C)(C)C2)=O)CC2CCOC2(CNC(=O)CCC2OCCO2)C1 42590,c1(OC)cc(C)nc(N(C)CC2CCN(C(=O)CC(C)SC)CC2)n1 42591,C1(CC)C(C(=O)NCc2nc(CO)n[nH]2)CCN1C(=O)C(c1cncnc1)C 42592,C1(c2n(CC(=C)C)nnn2)(NCc2cc(Br)no2)CCC2(CCOCC2)C1 42593,Cc1cccc2cc(C(=O)NC3(CNC(C45CC(F)(C4)C5)=O)CCOC3)nn12 42594,c1(C(=O)NCc2cc(OC)no2)n[nH]c2c1CCN(c1ccnc(SC)n1)C2 42595,c1(NC)ccccc1C(N1CCC(C)(CNC(=O)CCc2ccnc(Cl)c2)C1)=O 42596,CC(F)(F)CC(=O)N1CCN(C(c2cnnc(C)n2)=O)CC1 42597,c1(OC)nc(C(=O)N(C(C)CN(C(=O)C(C2CCCC2)OC)C)C)cc(O)n1 42598,CCC(C)C(O)C(=O)NC1CC(CCNC(=O)C(F)C(F)(F)F)C1 42599,C1(N(C2CC3CC2CN3)C(=O)COCCOC)CCNCCC1C 42600,S(=O)(=O)(c1ccc(N2CC(C)SC(C)C2)nc1)NCCc1cn(CC)nc1 42601,N1(C(C2(C)CCN(C)C2)=O)CC2CCC(C1)N2C(c1cnn2ccccc12)=O 42602,C1(C)(N(C(=O)COc2ccn(C)n2)C)CCN(C(=O)CCc2cccs2)C1 42603,c1(C(=O)NCC2CC(NC(C(CC#C)C)=O)C2)ccc2c(Br)n[nH]c2c1 42604,C#CC1(C(N2CCC2CC)=O)CCN(C(c2cccc(C)c2F)=O)CC1 42605,C1(CC(=O)NCCc2cc(C)ncc2)N(C(=O)C=Cc2ccco2)CCC1(C)C 42606,C1(NC(c2n(C)nnn2)c2ncc(-c3ccccc3)s2)C(=O)OC2CCCC12 42607,C(C)(C)(CC(C)NC(=O)CC1CN(C(=O)Cc2cccnc2F)CCO1)OC 42608,c1(C(N2C(C(C)NC(C(CC)(C)COC)=O)CCC2)=O)cccc2ccn(C)c12 42609,CCC1=C(C(=O)N2CCCC2CCNC(c2ccccc2)=O)SCCO1 42610,c1(-n2c(C)nnn2)ccc(C(=O)NC(C)CCNC(c2csc(C#N)c2)=O)cc1 42611,N1(C(c2ccn(CC)n2)=O)CCC2(C=C(C(=O)NOCCOC)C2)C1 42612,C(C(=O)N=c1ccn(CC2CC2)[nH]1)(C1CCCC1)NC(c1n(C)cc(C#N)c1)=O 42613,Cc1cnn(CC(N2CC(NC(=O)CC3CCC(C(F)(F)F)O3)C2)=O)c1 42614,C#Cc1cn(C)nc1C(=O)NC(C(=O)NCC(F)(F)C(N)=O)C(C)C 42615,N1(C(C=CCN(C)CC)=O)CCN(C(CNC(=O)C(F)C(C)C)C(F)F)CC1 42616,N1(C(c2nc(C(=O)OCC)sc2)=O)CCCC(C(=O)NCCCCO)C1 42617,c1(C(N2C(C)CN(C(=O)Cc3cnns3)CC2)=O)cc2c(nc1N)CCC2 42618,c1(-c2n(CC)nc(CCC(F)(F)F)n2)ccc2c(c1)C(C)(C)CO2 42619,Cc1ccc2oc(C(=O)NCC3(F)CC(CNC(=O)C(C)(O)C4CC4)C3)cc2n1 42620,C1(NC(c2cn(C)nn2)=O)CCOC12CCN(C(C1CC(CC3CC3)C1)=O)CC2 42621,C1(NC(Cc2n(C)ncc2)=O)CCC12CCN(C(c1ncc(F)cc1F)=O)CC2 42622,CC(C)(C)CC(=O)NCC(c1ccccc1)NC(c1ccc(C(C)(C)C)s1)=O 42623,C(=O)(CC(C)CCC=C(C)C)NCC1CC(NC(c2cncc(OC)n2)=O)C1 42624,N1(C(c2ncc(OC)cn2)=O)CCC(C2CC2)C1CNC(=O)C=C1CCOCC1 42625,N1(C(c2occc2Br)=O)CC(C2CCCCN(C(=O)C(F)OC(F)(F)F)C2)C1 42626,c1(NC(=O)CC2(O)CN(Cc3cc[nH]n3)C2)ccc(Cl)c(Br)c1 42627,Cc1cccnc1C(=O)N(C1CN(C(c2cnn(C(C)(C)C)c2)=O)CC1F)C 42628,c1(CCC(=O)NCCOCCNC(=O)CC(F)F)ccccc1OC(F)(F)F 42629,C1(NC(c2c(C)cccc2Cl)=O)COC2C(NC(C3CC(F)(CO)C3)=O)COC12 42630,c1(CN(C)CC2CCCN2C(C2(CC3COCCN3C)CC2)=O)ccc(F)cc1 42631,C(=O)(C1=NOC(C)(C)C1)NC1CN(C)NC1=O.C1(OC)CC2(C1)C(=O)N2 42632,CN1CC2(CCN(Cc3ccc(-c4ccc(O)cc4)s3)C2)OCC1=O 42633,N1(CC(N2CCC(C(=O)NCCC(=O)OCC)C2)=O)CCCCC1C 42634,C1(CCC)CC1N=c1[nH]c(N2CCC3(CCSCC3)C2)nc2c1CCC2 42635,CCC(CC(=O)N1CC2CCC(C(=O)Nc3cscc3C(N)=O)(C2)C1)C(C)C 42636,C1(C(=O)NCC(C)(C(C)C)NC(Cc2c(C)noc2C)=O)C(O)C(=O)N(C)C1C 42637,c1(C(N2CC(NC(C3C(C)(C(F)(F)F)C3)=O)C2)=O)c(C2CC2)nc2sccn12 42638,N1(C(c2c(CC)ccs2)=O)CC2=C(C1)CN(C(=O)C(c1ccccc1OC)O)C2 42639,Cc1c(N)ccc(C(=O)NC(C)C(C)NC(=O)Cn2c(C)ccc2C)c1Cl 42640,Cc1c(F)cc(C(N2CC3CN(Cc4ccc(O)c(I)c4)C3C2)=O)cc1Br 42641,c1(N(C)CC2CCCN2C(c2coc(Cl)c2)=O)ncnc2sc3c(c12)CCC3 42642,Cc1n[nH]c(C)c1C(C)CC(=O)NCC(F)CNC(=O)CCC(F)F 42643,S(=O)(=O)(CCC1CCc2ccccc21)N1C(C)CC2(CCC2)C1 42644,C(c1ccccc1C)=CC(N1C(C)(CNC(CCSCCC)=O)CCC1)=O 42645,C12(CNC(=O)OC(C)(C)C)CC(CO1)N(c1ncccn1)C2 42646,CC(CN(C)C)CCC(=O)NCC(C1CCC1)NC(=O)CSCCC#N 42647,CC1(C)CN(C(c2ccsc2Cl)=O)CCC1NC(=O)CCCC1CC1 42648,C1(C)(CNC(Cc2c(CC)con2)=O)CCCN(C(c2cc(OC)cs2)=O)C1 42649,CCCCC#CC(C)(C)NC(c1c(CNC(=O)CC2CC(C)C2)cnn1C)=O 42650,c1(CC2(C(=O)NCCCOCCCC)CN(CC(C)CC)C2)ccc(Cl)cc1 42651,C1(C(N2CC(C)(CNC(COCC#C)=O)OCC2)=O)CCc2ccccc2C1 42652,N1(C(=O)NCC(C2COC(C)(C)O2)O)CCC(=C(Br)Br)CC1 42653,Cc1cccc2[nH]c(C(N3CCC(NC(=O)CCCc4cccs4)C3C)=O)cc12 42654,C(=O)(C(C)(F)C(F)(F)F)N1CCC(CN(C(C2CN(C)C(=O)N2)=O)C)CC1 42655,N1(C(C2(CSC)CCC2)=O)CCCC(NC(c2nnc(O)cc2O)=O)CC1 42656,C(c1nc2ccccc2s1)=CC(N1CCN(C(CCCC=C)=O)CC1)=O 42657,CC1(F)CC(C(=O)NC(C(=O)NCc2nn[nH]c2C2CC2)c2ccoc2)C1 42658,N1(C(CS(=O)(=O)N(CC)CC)=O)CC(OC)CC(NC(c2cc[nH]n2)=O)C1 42659,c1(NCCCCCCSC)[nH]c(=NC2CCC(C(F)(F)F)CC2)nc2sccc12 42660,N1(C(C2C(OCC)C2)=O)CCN(C(=O)CN2CC(C)(C)C2)CC1CS(C)(=O)=O 42661,C(=O)(C(C(C)C)C(C)C)NC1CC2C(NC(C3CN(C(=O)NC)C3)=O)C2C1 42662,C1(COC)CCN(C(c2csc(CNC(c3ccc(Cl)s3)=O)c2)=O)CC1 42663,c1(OC)ccc(C(=O)NC(C)CCNC(C2CCN(C)C2=O)=O)c(F)c1F 42664,C(CC1=CCCCCC1)NC(C(C)N(C(=O)C(O)C(C)(C)c1ccccc1)CC)=O 42665,O=S(=O)(c1ccc2[nH]ccc2c1)NC1CCCNCC1F 42666,c1(C(=O)NC(CC=C)CNC(=O)CC(C)C)ccn2cnc(C)c2c1 42667,C(=O)(CCCCCn1cc(-c2ccnn2C2CC2(F)F)nn1)N(CCCC)CC 42668,C(=O)(C1=CCN(C(c2csc(CO)n2)=O)CC1)NC1(CC)CCCC1 42669,N1(CCC)CCCCC1C(=O)NC1CCC1NC(c1ccn(C2CC2)n1)=O 42670,C1(C(N(CC(C)NC(=O)Cc2ccon2)CC)=O)COc2cc(Cl)ccc2C1 42671,N1(C(C(C=C)(C)CC)=O)CCC2(CCCN2C(C2CC(F)(F)C2)=O)C1 42672,c1(C(=O)NC(CNC(CN(C)CC)=O)CC(C)C)cnc2n1CCS2 42673,c1(C(C=CC(=O)NCCN(C(=O)CNC(C2(O)CCCC2)=O)C)=O)ccccc1 42674,C1(C(=O)NC(CNC(c2cnc(C)[nH]2)=O)C2CCC2)CC2CCC1CC2 42675,C12(C(N3CC(CNC(C=C(C)Cl)=O)C(C(F)(F)F)C3)=O)CCN(CC1)S(=O)(=O)C2 42676,CC(C)(Cc1cnn[nH]1)C(=O)N1CCC(CCNC(c2ccc(CO)cc2)=O)C1 42677,n1(CC#C)cnnc1C(=O)NCCC1(NC(=O)C(C)OCC2CCCO2)CC1 42678,c1(-c2nc(C(C)Nc3nc(Cl)ccc3Cl)sc2)ccc2c(c1)OCCO2 42679,N1(C(C2N(CC)CCC2)=O)CCC=C(C(=O)NCCN2CCNC2=O)C1 42680,c1(NC2(c3n(CCC)nnn3)CCN(CCOC)CC2)cccc2c1nnn2C 42681,C(=O)(C1CCc2ccc(OC)cc21)N(C)CC1CN(C(C(CC)(C)O)=O)C1 42682,c1(N2CCC(Br)=C(C)C2)nc(NC2CCC3C(CC2)C3(F)F)c2ccsc2n1 42683,C1(C(=O)NCCC(C)NC(C2CCC3CC2C3(C)C)=O)CCC2CCCCC2C1 42684,c1(OC)ccc(C(N2CCN(C(=O)C=C(C)c3ccco3)CC2C)=O)c(OC)n1 42685,S(=O)(=O)(CCC(=O)N1CC(CNC(=O)CCc2ccc(CC(C)C)cc2)C1)NC 42686,C1(OC)CC(NC(c2cc(C)ns2)=O)C12CCN(C(=O)C(N)=O)CC2 42687,C(=O)(C(C)(C)C(C1CC1)NC(C(C)(C)CO)c1cccs1)OC 42688,C1(C(=O)NC2CN(C(C(=O)NCCOCCCC)=O)C(C)C2)CCCC(=O)N1C 42689,C1(NC(C2CC2C2CCC2)=O)CC2CC1CC2C(N1CC(C2CCCCC2)C1)=O 42690,CC(C)C1C(=O)N1.N1(C(CCOC(=O)C2CC2)C)CCOCC1 42691,N1(C(=O)CCCO)CCC(S(=O)(=O)N2CCCC2)CC1 42692,N1(C(C(C)N(C(C)=O)C)=O)CC(NC(C2CCC2)=O)C2(CCC2)C1 42693,c1(C(=O)NCCN(CCC)C(c2cnc(C(C)C)o2)=O)c(C)coc1C1CC1 42694,c1(C(C(=O)NC(CCC)CNC(=O)C(C)Cc2ccnn2C)O)cccc(C)c1 42695,c1(NC(C(CN(C)C)NC(=O)CC2CC3C=CC2C3)=O)ccc(Cl)cc1O 42696,N1(C(c2nnn3c2CSCC3)=O)CC2(CCN(C(C3CC(=C4CC4)C3)=O)CC2)C1 42697,C1(CC)(NC(C2CCC(=O)N2)=O)CCCN(C(=O)CCCN(C)C)C1 42698,Cc1nncc(C(=O)NC(CCN(C)C)C(=O)NCC(O)C2CCC2)c1C 42699,N1(C(C2ON=C(CC)C2)=O)CCN(C(=O)Cc2ccc3c(c2)CC3)C(C2CC2)C1 42700,C1(C(=O)OC)COC2(CCN(C(C)=O)C2)C1.c12ccc3c(n[nH]c3c1)C(=O)NC2 42701,c1(C(CC)NC(=O)CCN2CCC(F)(F)C2)ccc(Br)c(Cl)c1 42702,C1(C(N2CC(C)C(NC(=O)C(C)(C)CF)C2)=O)CCc2nn[nH]c2C1 42703,C1(C)(COC)CC(NC(c2c(C)cnn2C)=O)CN1C(c1scnc1Cl)=O 42704,c1(CC(=O)NCC2(F)CCN(C(C3(O)CCSC3)=O)C2)cnn2ccccc12 42705,CCCCCCCC(=O)N(C)CC1CN(C(=O)CC2CC(CC)C2)CCO1 42706,Cc1cocc1C(c1nnnn1CC)NCC1(CO)CCCC1.N1(C)CCOCC1 42707,c1(CC(C)C(=O)NCC2CCCC2NC(C2CCN(C)C2=O)=O)ccc(F)cc1 42708,N1(C(C(=O)NCCOC)C2CC2(Br)Br)CC2CCCC2(C(N)=O)C1 42709,C1(CCC(=O)NC(CNC(=O)Cn2ncc(Br)n2)CO)CC2CCC1C2 42710,c1(OC)ccc2c(C(=O)NCCOCCNC(=O)CCc3nccs3)cnn2c1 42711,C(C(C)CN(C(=O)CCNC(=O)C=CCl)C)OC(C)=O.C12CC1NC2=O 42712,C1(NC(=O)COc2ncccn2)CCCCC1Nc1cnco1 42713,c1(NC(c2c(COC)n(C)nc2)=O)nccc2[nH]ccc12.C(C(C)(C)CC1CC1)N 42714,c1(NCCCCOC(C)C)cc(=NCC2CS(=O)(=O)CCO2)[nH]cn1 42715,C1(C(N(C2CCCC2)CC=C)=O)CCC(C)(C)N(C(C2CC2(F)Cl)=O)C1 42716,C(=O)(C(C(C)(C)NC(C)=O)c1ccccc1)N1CCN(CCCOCC)CC1 42717,c1(NC(N(C(CC(=O)OCC)Cc2ccccc2)C)=O)ccc(F)cc1F 42718,CCCC(C)CN=c1cc(NCc2ccccc2CC)nc(COC)[nH]1 42719,c1(C(=O)NC2CN(C(c3cccc(OC)c3)=O)C(CO)C2)cccc2nn[nH]c12 42720,N1(C(CCCn2cc(-c3nc(C(=O)O)sc3)nn2)=O)CCC2C(C1)C2(Br)Br 42721,c1(C(=O)OC)cc(C(=O)NCC2(NC(c3cscc3F)=O)CC2)n2c1COCC2 42722,c1(C(N2C(CNC(C(C)Oc3ccccn3)=O)CC2)=O)cccc(C(N)=O)n1 42723,c1(C(CC)(C)O)cn(CCCNC(c2coc(C(C)C)n2)=O)nn1 42724,CC1(C)CC(O)CN(C(=O)C(=O)NC(C2CCCCC2)C2CCOCC2)C1 42725,CCC(C)(C)C(O)C(=O)N1CC(C(C)NC(c2cn3c(n2)CCC3)=O)C1 42726,c1(N2CCC(CCNC(C(C(C)C)(C)O)=O)CC2)ncc([N+](=O)[O-])cc1C(N)=O 42727,c1(C(=O)NC(C)C(C)NC(=O)C(C)(C)CS(N)(=O)=O)cc2c(cc1Cl)NC(=O)C2 42728,c1(CC)cc(=NC(=O)C2CCN(C(=O)CN3CCC(C)CC3)CC2O)[nH]n1C 42729,c1(NC(C)=O)ccc(C(N2CCCCC2C(N2CC3CC3C2)=O)=O)cc1 42730,Cc1n[nH]c(C)c1CC(N1CC2C(CNC(=O)C(C)(C)C)C2C1)=O 42731,C1(CNC(C(C)NC(C)=O)=O)CC(F)(F)CN1C(=O)COC1COC1 42732,N1(C(c2c(C)c(F)ccc2)=O)CCC2(CNC(c3cscc3F)=O)CCCCC12 42733,CC1CCC(CNC(=O)COC2(C)CCOCC2)CN1C(c1cncc(N)c1)=O 42734,c1(C(C(=O)O)NC(=O)NC(c2nc(C(F)(F)F)cs2)C)cccc(Cl)c1 42735,c1(SCC)ncc(Cl)cc1C(=O)OCC#CCOC1CC1 42736,C12CCN(CC1)CC=CC(=O)N2.C1(CC(=O)NCCSC)SC(=N)NC1=O.CO 42737,C12(NC(C(CC#C)CC#C)=O)CCCC1(F)CN(C(=O)C(C)COCC)C2 42738,Cc1nnc2c(C(=O)NCC(CC(C)C)NC(=O)C(CO)N(C)C)cccn12 42739,c1(C(c2nnnn2C2(C)CC2)NC(CC)C)cccc(CCC(=O)OC(C)C)c1 42740,n12cc(nn1)C2.C(=O)(CCCn1cc(C)cn1)CN(C(CC1(CSC)CC1)=O)C 42741,C1(CN(C)C)COCCN1C(=O)CC(C1CC1)NC(=O)C(C)(C)C1CCOC1 42742,C(=O)(C1=CC2CC(C1)CC2O)NCC(CNC(Cn1nc(C)oc1=O)=O)O 42743,S(=O)(=O)(c1ccc(F)cc1Cl)NCC(N1CCOCC2(COC2)C1)=O 42744,C1(C2CC2)(CNC(=O)CC2CC=CC2)CCN(C(=O)CN2CCCCCC2)C1 42745,c1(OCC)ccc(C(C)NC(=O)CCC2(C)CC2)cc1F 42746,CC(CC(F)(F)F)C(=O)NC1CCN(C(=O)C=C2CCSCC2)CC1O 42747,c1(C(=O)NC(C)CN2CCCCC2C)cnc(Br)c(Cl)c1 42748,CCCC(C)(CCC)C(=O)N1CCC(CNC(=O)CN(C)C)(OC)C1 42749,c1(NCC#CC)cc(=NCC(C(C)C)c2ccnn2C)[nH]cn1 42750,C1(C(N2CCC(OCC(=O)NCc3ccc(SC)o3)C2)=O)CCN(C)CC1 42751,c1(-c2cn(C(C)C(N3CCC(C(C)(C)C)C3)=O)nn2)ccc2[nH]ccc2c1 42752,CCC(CC1CC1)C(=O)N1CC(NC(=O)CCN(C)CCO)C(F)C1 42753,Cc1nc(CCCC(=O)NC2CC(NC(c3cscc3C(F)F)=O)C2)cs1 42754,C1(CC)C(C(NC[Si](C)(C)C)=O)CCCN1C(c1ccccc1F)=O 42755,N1(C(CN(CC)CC)=O)CCC2(CCCN2C(=O)CC(F)(F)c2ccccc2)CC1 42756,C1(NC(COCC)=O)CC2CC(NC(=O)CNC(=O)C3CC3)C1C2 42757,N1(C(c2n(C)cnc2)=O)CCc2sc(CNC(=O)CCc3cnc(O)[nH]3)nc2C1 42758,c1(C(N2CCC(NC(C(OC)OC)=O)(CO)C2)=O)cc2occc2n1C 42759,C1(CN(C(C2CC(C)C2)=O)C)CCCC1NC(=O)C(CN(C)C)c1ccccc1 42760,CC1CN(C(C2CC(CCO)C2)=O)CC(CCNC(c2nnn(C(C)(C)C)n2)=O)O1 42761,C1(CC)CC(C)CN(C(=O)CC(C)(C)N(C(=O)CCCN=[N+]=[N-])C)C1 42762,c1(C(=O)NCC(CC(=O)N(CC(=C)C)C)OC)cnn2c1OCC2 42763,C1(c2nnnn2-c2ccccc2)(NCC2COCC(C)(C)O2)CSC2CCCC12 42764,N1(C(CSS(C)(=O)=O)=O)CC(NC(=O)Cc2cc(-c3ccccc3)on2)C(F)C1 42765,c1(C(N(CC(C)NC(c2ccc(OC3CC3(F)F)cc2)=O)C)=O)ccc[n+]([O-])c1 42766,C1(C(N)=O)CN(C(=O)C(=O)NCc2cc(N3CCCC3)n[nH]2)c2ccccc2O1 42767,c1(C(N2CCC3(C(NC(COCC)=O)C3)C2)=O)scc2c1OCCO2 42768,C(=O)(CC(C(C)C)C(C)C)NC(CCNC(C1C(=C)CC1)=O)(C)C 42769,Cc1cnn(C)c1CC(N1CC(N(C)C(C2C3COCC23)=O)C1)=O 42770,C1(C(C)C)C(NC(=O)CNC(=O)CC(C)(C)C)CCN1C(=O)CC1CC(C)C1 42771,C1(CNC(CNC(CCC)=O)=O)CC(C)(C)CN1C(c1cc[n+]([O-])cc1)=O 42772,c1(OC)c[nH]c(C(N2CC(C)(C)CC2CNC(C2CC(C)(C)CO2)=O)=O)cc1=O 42773,CCC(C)C(O)C(C)C(=O)N1CC(NC(=O)CCCCCC(C)C)C(O)C1 42774,N1(C(c2n(COC)ncc2)=O)CC(NC(=O)C=CCCC(C)C)CC(C)C1 42775,CC12CC1CN(C(=O)C(N1CCC(c3cccc(Br)c3)CC1)=O)C2 42776,c1(C(=O)NC2CC(CNC(C(CC)O)=O)C2)ccc(C(C)C)cc1 42777,N1(C(C(CC)OCC)=O)CCC(CC(=O)NCC(C)(C)CC)C1(C)C 42778,C1(C)(CNC(CCc2c(C)nccc2)=O)CN(C(=O)Cc2cn[nH]c2)CCO1 42779,O=C(C1Cc2ccccc21)N1CCC2(CCCN2C(C2CC(F)(F)CS2)=O)C1 42780,C=C=CCCC(=O)NCCCOCCNC(=O)CCC1CC1(C)C.c1(C)ccccc1 42781,C(C(C(=O)N(C)CCN(C)C1CC1)C(C)C)NC(c1c(C)n(C)cn1)=O 42782,c1(C(=O)NC(C(=O)NCCc2n(CC)cnn2)C2CCOC2)nnc(S)n1C 42783,S(=O)(=O)(c1ccnn1C1CCOCC1)N1CCN(C(=O)Nc2ccccn2)CC1 42784,C(C(O)CS(C)(=O)=O)NC(=O)NCc1sc(C)c(-c2ccccc2)n1 42785,C(=O)(CC(C)(C)CCC)NCC(CC=C)C(=O)NC1COCC1O 42786,C(=O)(CCCC(C)=O)N1CC(NC(C(C)=CC)=O)C(c2nccn2C)C1 42787,C1(C(=O)NCCCN(C(c2cc(O)nn2C)=O)CC)OCCOC12CCC2 42788,N1(C(C(C)(C)NC(=O)OC)=O)CCC(CNC(c2cc(CO)n(C)n2)=O)CC1 42789,C1(C(=O)NC(C)CCNC(C2CC(F)(CO)C2)=O)COCCN1CC(F)(F)F 42790,C=CC(C)CC(=O)NC1CC(CNC(c2ccccc2CO)=O)C(O)C1 42791,O=C(C1=CCN(C(=O)COC(F)(F)F)CC1)NC1CC1C1CCCC1 42792,C(=O)(C(F)(F)C1=CCOCC1)N(C)CC1CCN(C(=O)C(F)(F)C(O)C2CC2)C1 42793,c12sc(cc1C)C(=O)NC2.C1(C(=O)NC2CC(CF)C2)CCN(OC(C)=O)CC1 42794,C1(C(=O)NC2C(C)CCN(C(C=C(C)C)=O)C2C)CCc2nc(O)[nH]c2C1 42795,c1(C(=O)NC2CC(CNC(=O)CC3CCCCC3O)C2)ncc(F)cc1F 42796,C1(CNC(=O)CC2(c3ccccc3)CC2)CCCCC1CNc1cc(Cl)ncn1 42797,C(=O)(C(F)(F)C(F)(F)OC(F)(F)F)N1CCN(C(C)=O)C(c2nccn2C)C1 42798,C1(C(N(C2CCN(C(=O)OCc3ccccc3)C2)C)=O)CCN(c2nn[nH]n2)C1 42799,c1(C(=O)NCCC2N(C(c3cnc(C#N)s3)=O)CCC2)cc2cc(Cl)cnc2[nH]1 42800,C(CCCC(=O)NCC1CCCCN1C(c1cccc(F)c1SC)=O)(OC)OC 42801,N1(C(C(CCSC)OC)=O)CC2CC3CC2C1C3NC(=O)C(c1ccc(Cl)s1)C 42802,c1(CN2CC(CNC(c3c(O)cccc3F)=O)OCC2)c(O)ccc(Cl)c1Cl 42803,N1(C(CSCC#C)=O)CCN(C(=O)Cc2ccc(F)cc2)C(c2nccn2C)C1 42804,c1(CNC(CCCC)c2nnnn2C)cc(C(C)C)n(C(C)(C)C)n1 42805,Cc1cc(C(N2CC3CC3(CNC(=O)OC(C)(C)C)C2)=O)cnc1C 42806,Cc1ccc(C(=O)NCC2COC(CNC(=O)Cc3csc(Cl)c3)C2)cc1CO 42807,C(C(C(=O)N1CCC(C)(NC(c2cccnc2)=O)C1)C(C)(C)C)OCC=C 42808,c1(C(=O)NCC(CNC(=O)C(CO)N(C)C)OC)ccc2c(c1)NC(=O)CC2 42809,C1(C)(CC(=O)NC2CN(C)C(C(=O)OC)C2)CCS(=O)(=O)N1 42810,C(=O)(C(C)(C)C(=O)OC(C)C)N1C(C)CC1C(=O)NC(C1CC1)C1CC1 42811,Cn1ncc2cc(C(N3CC(NC(C4C=CCC4)=O)CC(F)C3)=O)sc12 42812,CC(C1CC1)=C(F)C(=O)NC(C)C(C)NC(C1(CN(C)C)CC1)=O 42813,c1(OC)ccc(C(N2CC(CNC(c3cc(C#N)c[nH]3)=O)C3CC23)=O)cc1Cl 42814,CCS(=O)CC(=O)NC1CCC1NC(=O)CCc1cscn1 42815,C1(CC(=O)NCc2ccc(F)cc2)CCCN(C(c2cnn(C3CNC3)n2)=O)C1 42816,c1(C(CC)NC(C2CC2NCc2ccnc(Br)c2)=O)ccc(Br)cc1 42817,c1(CN2CCC(Oc3ccc(C)cc3)CC2)nc2ccccc2[nH]1 42818,N1(C(C2(OC)CCOC2)=O)CCC(NC(C23CC(CN2C2CC2)C3)=O)CC1 42819,N1(C(c2cc(OCC)ncc2)=O)CCCC(NC(c2ccncc2)=O)C(F)C1 42820,C1(C(N2C(CCC)CN(C(=O)CC(C)(C)C)CC2)=O)Cc2cncn2C(=O)N1 42821,C#Cc1c[nH]nc1C(=O)NC1CN(C(c2csnc2C2CC2)=O)CC1O 42822,c1(C(=O)NCC(CNC(c2cc(C)[nH]n2)=O)(C)C)cc2c(ncn2C)[nH]1 42823,N1(C(CN2CCC(C)(O)C2)=O)CC2CC(NC(=O)CN3CCNC(=O)C3)C(C2)C1 42824,C1(C(N(CC(CC)(C)OC)C)=O)CC(C2CCCCC2)CN1C 42825,C(=O)(CC(=O)NC1COCC1C(=O)NCC(C)(C)CC1CC1)NCC#C 42826,C(=O)(CCCC(C)(C)C#N)N1CC(C)C(CNC(c2cc(C(F)F)ncn2)=O)C1 42827,c1(C(N2CCN(C(CCS(C)=O)=O)CC2CO)=O)ccnc2cccnc12 42828,C1(C(=O)NCC2(COC)CCC2)CCN(C(c2cc(C)[nH]n2)=O)C1C 42829,C1(NC(CC2(C)CCN2C(C2CCC(=O)NC2)=O)=O)CC(F)(F)C1(C)C 42830,c1(C(=O)NC(CNC(C(CC#C)(C)CC)=O)(C)CO)ccc2ccccc2c1 42831,c1(N2CCC(C)C(NC(C3(C)CCCCO3)=O)C2)ncnc2c1c(Br)nn2C 42832,C#CCCC(C(=O)NC1CCCC(O)C1O)NC(C1COCC(C)O1)=O 42833,C(C(=O)N1CC(NC(=O)C(C)(C)C#N)C(c2ccnn2C)C1)(C(C)C)SCC 42834,CCC(C(=O)NCC1(C(N2CCC(C3(C)N=N3)C2)=O)CCCO1)NC(C)=O 42835,C=CC(C)(CC)C(=O)NC1CC(C)(NC(=O)Cc2ccc(CO)c(C)c2)C1 42836,c1(C(=O)NC(C2N(C(C(COC)OC)=O)CCC2)C)n[nH]c2ccc(OC)nc12 42837,C1(NC(C(C)n2cccn2)=O)(CF)CN(C(c2ccnn2C)=O)C1 42838,N1(C(C2CCC(C)S2)=O)CC2=C(C1)CN(C(C1(NC(C)C)CC1)=O)C2 42839,c1(C(=O)NCC2(O)CC(NC(CCS(C)=O)=O)C2)c(F)cccc1Cl 42840,c1(SC)ccc(N)cc1C(=O)NC(C)C(C)NC(=O)Cc1csc(C2CC2)n1 42841,C(=O)(C(C)C(O)C(C)CC)N1CCC(C(=O)NCC(C#C)OC)C12CC2 42842,n1(CC(=O)NC2CC(F)(CNC(COCCC(C)C)=O)C2)cc(C#N)cn1 42843,C1(O)(CNC(C(C=CC)O)=O)CCN(C(=O)Cc2ccccc2C)C1 42844,N1(C(C2CCC(C)(CC)O2)=O)CC2CCCC(C1)N2C(c1cc(C(F)F)cs1)=O 42845,c1(C(N(CC(=O)NCC2CC2)CC#C)=O)ccn(CC=C)c1.C1(C)C(=O)N1 42846,N1(C(CCNC(=O)OC)=O)CC(CCNC(c2ccncc2Br)=O)C(C)C1 42847,N1(C(Cc2c(C)nsc2)=O)CCN(C(c2ccn3nnnc3c2)=O)C2CCC12 42848,CC(C)S(=O)(=O)CC(=O)N(CCCNC(=O)CP(C)(C)=O)C 42849,N1(C(c2c(C)nsc2)=O)CCN(C(C2CC(C(F)(F)F)C2)=O)CC(CO)C1 42850,CC(c1ccccc1)=CC(N1CCC(C)(CNC(c2cc(C3CC3)on2)=O)C1)=O 42851,N1(C(CC2C(C)(C)OCCO2)=O)CCC2CN(C(=O)C=CC=C(Cl)Cl)CC2C1 42852,Cc1cc(C(=O)NCC(CC(C)C)NC(C2CCC(F)CC2)=O)cnn1 42853,c1(NC(C)=O)ccc(NC2CCN(C(=O)N(C3CCN(C)CC3)C)CC2)cc1Cl 42854,c1(NC(c2cccc(COC)c2)C(=O)OC(CCC)CCC)nn(C)c(C)c1Cl 42855,N1(C(c2cnn(C(C)C)c2F)C(=O)NCC)CC(C(C)C)c2ccccc21 42856,C1(C(=O)NCC(CC(C)C)NC(C2C=CCS2)=O)CC(C2CCCC2)C1 42857,C1(C)(C(=O)NCCNC(C(C)N(C)C)=O)CC(F)(F)C1.c12cn(nn1)C2 42858,C1(C(N2CCOCC2)=O)CCCCC1NC(CN(C(=O)C(O)C1CCCC1)CC)=O 42859,C1(CC(=O)NCC2C(C)(C)CCCN2)CCc2ccccc2N1 42860,N1(Cc2scc(C)n2)CCC(O)C(C(=O)N(C(C)C)CC2CC2)C1 42861,N1(C(C(COC)OC)=O)CCC(C)C(NC(c2cc(-c3cn(C)nn3)on2)=O)C1 42862,c1(C(C)NC(C23CC(NC(c4c(CC)c[nH]n4)=O)(C2)C3)=O)ccc(Cl)cc1 42863,CCCCCCC(CC)(CC)C(=O)NCC(CNC(=O)CNC(=O)C(C)C)CO 42864,C1(C(C(=O)NCC(O)CNC(c2coc(C(C)C)n2)=O)OC)CCC(F)(F)CC1 42865,C(C)(C(C)S(C)(=O)=O)N(C(C(=O)NC1CN(C(C)C)C(=O)C1)=O)C 42866,N1(C(=O)OC(C)(C)C)CCCC1C(C)(C)CO.c12cnc(o1)[nH]c2=O 42867,c1(CNC(Cc2c(C)nn(C)c2)=O)n[nH]c2c1CN(C(=O)C(C)S(N)(=O)=O)CC2 42868,c1(C(=O)NC2CCCN(C(C3(C#C)CCC3)=O)CC2F)ccc2ncccc2c1 42869,C1(CCCC(=O)NC(CCCC)C)N(C(=O)CCSC)CCC1(C)C 42870,c1(CCC(=O)NC2(C)CC(NC(=O)Cc3cnoc3)C2)cncc(F)c1 42871,c1(C(=O)NC2CC(F)(CNC(C3(C)CCN(C)C3)=O)C2)cccc2nc(O)[nH]c12 42872,c1(OCC)cc(C)[nH]c(=NCC2CC3CCC2N(C(c2csc(CO)n2)=O)C3)n1 42873,N12CCCC(O)(C1)NC2=O.c1(CC)ccc(C(N2CC(N(C)C(C)=O)C2)=O)cn1 42874,c1(C(=O)NC(C(=O)NCCc2ccc(C)s2)C2CC2)cnc(C)c(C)c1 42875,c1(C(N(CCOC)CCNC(c2c(F)cccc2Cl)=O)=O)ccc(O)c(F)c1F 42876,c1(C(=O)NC(C(C)NC(=O)C(=O)N(C)C)C)ccc(N2CCC(O)CC2)nc1 42877,N1(C(C2CCCCC2)=O)Cc2ccnn2CC(NC(C2CC23CCC3)=O)C1 42878,C(C(C)C(=O)NC1COCC1NC(c1cc(C(C)=O)c[nH]1)=O)OCC 42879,C1(CCC(=O)NCCCCN(C)C(C2(C)CCCN2C)=O)CCC(O)CC1 42880,c1(C(CC)C(=O)N(CC(O)CN(C)C(C2(OC)CC2)=O)C)ccc(F)cc1 42881,C12CCC1CN(C(=O)CCSCCCC)C2.C(CNC(C)=O)=CC 42882,Cc1cc(C(=O)NC(C)CCNC(=O)Cc2ccncc2Cl)c(Cl)cc1Cl 42883,c1(C(C)C)cccnc1NC(C1CCC(NC(=O)Cc2ccccn2)C1)=O 42884,c1(C(N2CC(C(C)CO)C2)=O)ccc2c(c1)CCCN2C 42885,c1(C(=O)NC2C(CNC(c3cc(C)sc3C)=O)C2)ccc2nc(Cl)nn2c1 42886,N1(C(c2cn(CC)nc2)=O)CCC2(CCC(CNC(c3csnn3)=O)OC2)CC1 42887,Nc1c(C(=O)NCCNC(=O)C(O)Cc2ccccc2Cl)cccc1F 42888,c1(-c2cc(Cc3n(C)ccn3)c(O)cc2)ccc2c(N)ncnn12 42889,c1(C(=O)NCCCC(C)NC(COCCC)=O)cc(Cl)c(F)cc1F 42890,c1(OCC(=O)NCCC(=O)NC2(C)CN(C(CCSC)=O)C2)ccc(C)cc1 42891,C1(NC(C2CC(C(F)F)C2)=O)CCOC(C(N2CC(O)(c3cc[nH]n3)C2)=O)C1 42892,C(C(=O)NCC12CCC(CC1)N2C(C1CCCOCC1)=O)(C(C)(C)C)SC 42893,c1(CCCC)nc(CNCc2cn(C3C(NC)CCCC3)nn2)c(Cl)[nH]1 42894,c1(SC)cc(C(=O)NCC2C(C)CCCN2C(=O)CC(=O)NC2CC2)ccc1F 42895,CC(C)(CNC(=O)COCC(=O)NC(=O)Cc1sccc1Br)CC1CC1 42896,CCC(C(=O)N1CC2C(NC(=O)Cc3scnc3-c3cccs3)C2C1)C(C)(F)F 42897,C(CCC(F)(F)F)N(C(CN(C(=O)C(=O)NC(C)C)CC)=O)C 42898,c1(C(N(CCCCCC)CCNC(=O)C(C)C#N)=O)ccc2nonc2c1 42899,CC(C)CC(C)(CNC(=O)C(C)(C)c1ccno1)NC(c1cc(C(C)C)on1)=O 42900,c1(C(N2CCC(n3cc(C(CC)O)nn3)C(F)(F)C2)=O)cnc2cccnc2c1 42901,Cc1ccc2oc(C(=O)NC(C)(C)CCCNC(C3(CO)CCC3)=O)cc2c1 42902,CC(C(=O)NCCOCC(=O)NCCCN(C)C(C)C)=CC1CC1 42903,c1(CC(=O)NC23CC(CNC(C4CCCSC4)=O)(C2)C3)ccccc1F 42904,C1(N(C(C(CNC(c2nc(C(C)C)oc2)=O)O)=O)C)CCCC1(C)O 42905,Cc1cc(Cl)cc(C(=O)NCCCNC(c2n[nH]c3c2CSCC3)=O)c1C 42906,CCC(CC)N(C(=O)CC=CCNC(C1CCCS1)=O)C 42907,c1(OCC)cccnc1C(N1CCCC1CNC(c1[nH]c(C2CC2)nc1C)=O)=O 42908,N1(C(C2C(C)(Br)C2)=O)CCCC(C2CC2NC(c2cnn(CC3CC3)c2)=O)C1 42909,c1(OC)cccc(C(N2CCC(=CCNC(C3CCCN3C(N)=O)=O)CC2)=O)n1 42910,Cn1nc2c(c1-c1cn(CCC(=O)Nc3ccc(I)cc3F)nn1)CCCC2 42911,C(=O)(C(C)CC(F)(F)F)NC(c1occ(C(N(CC(C)C)CC)=O)n1)C 42912,C(=O)(CCn1ccnc1)N(CC(C)O)CCNC(=O)CC1(C(F)(F)F)CC1 42913,c1(SC(C)C(N)=O)ccc(C(=O)NC2(C)CN(C(c3ccncc3)=O)C2)cc1 42914,c1(-c2n(-c3c(C)cccc3C)nc(C(C)C3CC3)n2)sc2cccc(F)c2c1C 42915,c1(C(N2CC(NC(=O)C(F)(F)CO)CC(C)C2)=O)nc2cccnc2s1 42916,CCCCC(CNC(C1CCCN1C)=O)NC(c1snc(Cl)c1Cl)=O 42917,N1(C(C(C2CC2)OC)=O)CCC(Cn2cc(CC(c3ccccc3)O)nn2)CC1 42918,CC1CC(N=c2cc[nH]cc2S(=O)(=O)NCCc2cncnc2)CC(C)N1 42919,N1(C(CC2C(C(C)(C)C)C2)=O)CCCC(CNC(=O)CCn2cnnn2)CC1 42920,C(=O)(CC(COC)COC)N1CCCC(N(C(=O)CC2CCNC(=O)C2)CC)C1 42921,c1(C(=O)NCCCN(c2nnco2)C(C)C)ccc2c(c1)NC(=O)CO2 42922,c1(OCC(N)=O)ccc(C(=O)NCC(C)NC(=O)C=CSc2ccccc2)cc1 42923,c1(C(=O)NC2(C(=O)NCc3ncccc3F)CC(CO)C2)ccc(O)cn1 42924,C1(NC(c2c(CC)c[nH]n2)=O)CCN(C(=O)CSc2cccc(F)c2)CC1(C)C 42925,C(=O)(C1COc2ccccc21)N1CC(C)(C)OC(CNC(C2CC=CCC2)=O)C1 42926,c1(N(CCOC)CCNC(C2CCC(=O)N2)=O)nc(C)cc(C)n1 42927,N1(C(=O)Nc2ccccc2N2CC(C(F)(F)F)OC2=O)Cc2ccc(Cl)cc2C1 42928,Cn1cc(C(=O)NC2CC2CNC(c2ccc(-n3cncn3)cn2)=O)n(C)c1=O 42929,N1(C(c2cncc(SCC)n2)=O)CCN(C(=O)CC=C(C)C)C(C)C1C 42930,c1(C(=O)NCC(CNC(C(CCCC)C)=O)F)ccc(S(N)(=O)=O)cc1Cl 42931,c1(C(=O)NC(C2(O)CN(C(CCC#C)=O)C2)C)cncc(C)c1Cl 42932,N1(C(C(CNC(C=CC(=O)NC(C)C)=O)N(C)C)=O)CCCC(N(C)C)CC1 42933,c1(C(=O)OC)nc(Br)cnc1NC(C1CCC(C)N1Cc1ncc(Cl)cc1C)=O 42934,Cc1c(NC(=O)Cc2ccccc2NCc2ccsc2)ccnc1Cl 42935,C1(C)(C(=O)NCCC(C)CCNC(=O)CCCc2ccccn2)CC2CCC1C2 42936,C1(C(=O)NCC2C(CNC(C(CCC)=CCC)=O)C2)COC2COCC2O1 42937,c1(C(N2CCC(C)(NC(c3nc(C)c(C)[nH]3)=O)C2)=O)ccc2[nH]c(=N)[nH]c2c1 42938,CCCN=C(NCCOCCSC)NCCCOc1ccccc1 42939,c1(CNC(C(C2CCOCC2)C)=O)cc(C(=O)NCC2CC(CO)CO2)on1 42940,C(=O)(C(C#N)C(C)(C)C)N1C(C(NOCC)=O)C2CCC1C2.C1(=O)CCCN1 42941,C(=O)(C1=C(Cl)CCCC1)N1CC(CC(N2CC(CCO)C2)=O)OCC1 42942,N1(C(c2cc(C)sc2)=O)CC(NC(C2(Cc3cnn[nH]3)CCC2)=O)C(C)C1 42943,c1(C(Cn2cc(CC(=O)ON3CCC(O)CC3)nn2)O)ccc(Br)cc1C(=O)O 42944,C(C)(C(F)(F)C(F)(F)F)=CC(=O)NC(CCNC(C(C)NC(CO)=O)=O)C(C)C 42945,N1(C(C2C(C)(Br)C2)=O)C(CNC(=O)Cn2cnnn2)CC2COCC12 42946,C1(NC(CC2(COC)CCCC2)=O)CCC(C)(C)CC1CNC(=O)C=CBr 42947,c1(OC)cc(C=CC(=O)NCc2ccc(CNC(c3cnn(C)c3)=O)cc2)sn1 42948,Cc1ccncc1C(=O)NCCC1CCC(NC(c2c(C)coc2C2CC2)=O)C1 42949,c1(NC(CNC(CC2N(OCC)CCOC2)=O)C(C)C)ccc(C)cc1[N+](=O)[O-] 42950,C(C(=O)NCC(C)(CO)NC(C1CN(C2CCC2)C1)=O)(C(C)C)OC(C)C 42951,N1(C(C(CC=C)C)=O)CCCCC(NC(C2(c3ccccc3)CC2)=O)C1 42952,c1(C(=O)NCC2C(C)CCN2C(C2(C(=O)N(C)C)CC2)=O)cc2ncccc2o1 42953,c1(NC(C2(CC)CN(C(C)CC(N)=O)C2)=O)cccc(OC)c1 42954,c1(C(N2C(CNC(C(CC#C)O)=O)CC(F)C2)=O)cnn2c1NCCC2 42955,c1(OC)cc(C)ncc1CSc1c(C(=O)OC(=O)C(C)C)sc(C)c1C 42956,c1(CNC(=O)NCC2CCN(C(=O)OC)CC2)ccc2cccnc2c1 42957,CC1CC(CNC(=O)C(=O)N(C)C)CN1C(c1ccc[n+]([O-])c1)=O 42958,CC1Cn2nc(C(=O)NC3COC3)cc2CN1C(=O)OC(C)(C)C 42959,C#CC1CN(C(=O)C(C(C)OC)NC(=O)C(O)CN2CCCC2)CCO1 42960,N1(C(C(C)CO)=O)CC(NC(c2cncc(F)c2)=O)CC12CCCC2 42961,C1(NC(c2ccc(C)nc2)=O)CC2(CCC(NC(C3C(C)CC3C)=O)CC2)C1 42962,N1(C(CC(C)OC)=O)CCCC(C)(NC(=O)Cc2ccc(O)cc2C(F)(F)F)C1 42963,N1(CC)CCc2occc2C1C(=O)N=c1ccn(CO)[nH]1 42964,Cc1ccc(O)c(CNC(=O)CC=CCNC(c2cn(C)cn2)=O)n1 42965,Cc1ccc([N+](=O)[O-])cc1C(=O)NCC(CO)NC(=O)CCCC1CCOCC1 42966,N1(C(CC2CN(C(C(C)NC(C)=O)=O)C(C)(C)C2)=O)CC2(C1)CC(C)(C)C2 42967,CC1(C(=O)NCCCCNC(=O)Cc2ccc(O)cc2Cl)CCC12CCC2 42968,Cc1ccc(CC(=O)NC2CC(NC(=O)C(CN(C)C)N(C)C)C(O)C2)c(Cl)n1 42969,C=CCC(CC=C)C(=O)N1CC(O)CC1(C)C(=O)NCCCCC 42970,Cc1cnc(C(N2CC(C(O)C(=O)NCCN3CCC(C)C3)C2)=O)cn1 42971,c1(OCC)nc(C)ccc1C(=O)NCC(O)CNC(=O)CCc1ccnc(C)n1 42972,c1(C(=O)NC(C)CN(C(=O)CO)C)ncccc1Br 42973,C1(C(=O)NC2C(C)N(C(c3ccc(CN=[N+]=[N-])cc3)=O)CC2)CCCC(F)(F)C1 42974,c1(C(C(=O)N(C2CN(C(C3CCCN3C)=O)C2)C)OC)ccc(F)cc1 42975,c1(CC(=O)NCC(C2CC2)NC(C2CNC(=O)C2)=O)cnccc1O 42976,CCCCC(O)C(=O)N1CC(NC(=O)CCCCCC)C(c2cccc(F)c2)C1 42977,C1(OC)CC(NC(c2ccnnc2C)=O)CN(C(=O)Cn2c(C)ccc2C)C1 42978,C1(C(=O)Cc2ccccc2)CN(C(=O)C(O)C(F)(F)F)CCN1C(=O)C(F)=CC1CC1 42979,c1(C(C)C)cnc(O)c(C(=O)NC2CCN(C(C3CC(C)(C)CO3)=O)C2)c1 42980,C1(NC(CCN(C)C)=O)CC(F)CN(C(c2ccc(O)cn2)=O)C1 42981,N1(C(C(CCC)N(C)C)=O)CCCC2(NC(c3ccoc3Cl)=O)CC2C1 42982,c1(NC(CC2(C)CN(C(=O)CN3CC4CC4C3)C2)=O)cccc(N2CCCC2)c1 42983,C(C(=O)N=S(C)(=O)N(C)C)NC(C(CC)Oc1ccccc1)=O 42984,c1(CC(N2CC(C)(C)OCC2CO)=O)cc(F)c(F)c(F)c1 42985,C1(C(C)C(=O)NCCNS(N)(=O)=O)CCN(C(C2CCN(C)CC2)=O)CC1 42986,N1(C(C2C(C(C)=O)COC2)=O)CC(C)C(C)(C(=O)NC2CCCCC2F)C1 42987,C#CC1CC2(CC2)CN1C(=O)CCC(C)NC(C1(C#N)CC1)=O 42988,c1(OC)ccc(CC(N)C(=O)NCCO)c(OC)c1.c12cccc(c1)OC2 42989,N1(C(C2(N=[N+]=[N-])CCN(C(c3cc(CC)sn3)=O)C2)=O)CC(C#N)C2(CCC2)C1 42990,N1(C(CC(C=C)C)=O)CCCN(C(=O)Cc2ccc(Cl)c(Cl)c2)C(CO)C1 42991,c1(OC)ccc(F)c(C(=O)NCCCN(C(=O)COCCF)C(C)C)c1 42992,C1(C(=O)NC(C=CC(=O)NC(C(C)F)C)C)OCC2CCCC12 42993,C1(c2noc(CC(=O)NC(C)CO)n2)(NC(C)=O)CCC(C)CC1 42994,N1(C(C(C)(C)OC)=O)C2CCC1C(CNC(c1nccnc1C(N)=O)=O)C2 42995,CC1=C(C(=O)NC2CCCC2C(=O)Nc2ccc(Br)nc2)CCO1 42996,c1(CNc2c(C)nc(-c3c(OC)cccc3)s2)c(C)nn(C)c1C 42997,c1(NC(C2N(Cc3ccc(SC)s3)CC(F)C2)=O)nc(Br)c(Br)cc1Br 42998,C1(NC(C(C)N(CC)CC)=O)CN(C(C2CCCO2)=O)Cc2nccn2C1 42999,C(=O)(CC(C=C)CC)N1CCC(N(C(=O)C(C=C)CC)CC#C)C1 43000,c1(CC(=O)NCCC2(O)CCCN(C(c3nocc3Cl)=O)C2)c(O)ncnc1O 43001,C1(OC)CC2CC(C(=O)NCCCC(C)(C)NC(=O)Cc3ccco3)CC12 43002,C1(NC(=O)CCC=CBr)C2CCC1N(C(c1ccc(CF)cc1)=O)C2 43003,c1(C(N(C)CC2CCN(C(c3ccc(F)cc3N)=O)C2)=O)cnc2[nH]ccc2n1 43004,C1(CC(N2CC(O)(CNC(C(CN(C)C)N(C)C)=O)C2)=O)COCC2(CCC2)O1 43005,CCCCC(O)C(=O)NCC(C)N(C(=O)CCC1CCCC1)C 43006,N1(C(C2(CC(C)C)CC2)=O)CC(O)(CCNC(C2(C(F)(F)F)CC(F)C2)=O)C1 43007,c1(C(c2n(CC)nnn2)NC(c2nccn2C)C)cc(Br)cc(Cl)c1F 43008,C(=O)(C1=CCCCC1C)N1CCC2C(C(=O)NC(COC)C)C2C1 43009,C(=O)(CCCC(=O)N1CCC(CO)C1)N(N1CCC(O)(C(F)(F)F)C1)C 43010,C1(NC(c2cc(Cl)ccn2)=O)COC2(C1)CN(C(=O)CC1CCC(C3CC3)O1)C2 43011,c1(C(=O)NCC2CC(NC(C(C)C3CCCO3)=O)C2)cc(F)c(N)c(F)c1 43012,N(C1CS(=O)(=O)Cc2ccccc21)C(=O)NCc1ccc(O)c(Br)c1 43013,C1(NC(CSCC=C)=O)CC2CC(NC(C3CCC4CC34)=O)C1C2 43014,C1(P(C)(C)=O)(C(=O)OCc2cnc(C)s2)CC1 43015,C1(CNC(C2(OC)CCCC2)=O)CC2(CC2)CN1C(c1cc[nH]c1)=O 43016,C(C)(CN=c1nc2ncccc2c[nH]1)NC(c1c(C)nc(C)s1)=O 43017,C(C(O)C(=O)NC1(c2noc(C)n2)CC1)NC(CC1CC(NC)C1)=O 43018,C1(NC(CCSC)=O)CCN(C(C2COCCN2C)=O)C1(C)C 43019,CC(C)CC(C(=O)N1CCCC(n2cc(CCCOCCO)nn2)C1)N(C)C 43020,C1(C(=O)NCCOCCN(C)C(C2(CO)CC2)=O)CC2CC(=O)C1O2 43021,C1(CCNC(C=CC=CC)=O)CCCN(C(=O)CC(=O)OCC)C1 43022,C12(CC=CCC1)C(=O)N2.O=C(C(=O)NCC(F)(F)F)NCCCOCCCO 43023,Cc1ncc(C(=O)NC2CC(OCC(=O)N(CC(C)(C)C)C(C)C)C2)c(=N)[nH]1 43024,Cc1noc(C)c1CSCCC(=O)NC1CCCN(C(c2cc(O)nn2C)=O)C1 43025,c1ccc(C2CC(NCc3cnc(C4CCC4)o3)CN2)cc1 43026,CC1CC(C(N2CC(O)(CNC(=O)CSCC(F)F)C2)=O)CN1C 43027,c1(NC(C)=O)ncc(S(=O)(=O)N2CCCC(c3ccc(C(F)(F)F)cc3)C2)s1 43028,Cc1ccc(C(C)C(=O)NCC2(F)CCC(CNC(c3cnc(O)o3)=O)C2)cc1 43029,c1(NCC(=O)NC2CC(CNC(C3CCC4CC34)=O)C2)ccccc1Cl 43030,C1(NCc2n(C)cc(Br)c2)CC2(CCCC2)C1 43031,C(C(CC(C)C)C(=O)NC12CC1CN(C(c1ccnc(C3CCC3)c1)=O)C2)OC 43032,CC1(C)C(=O)N(C(C2CCCC2N)=O)CCN1Cc1cccs1 43033,C1(CC)(NC(=O)CCCSC)CCN(C(=O)CC2CC3(CC3)C2)CC1 43034,C(C(CC(C)C)NC(=O)Cc1ccc(F)cn1)NC(C1CC(C)(CC)C1)=O 43035,C(C)(CC(C)NC(c1sccc1COC)=O)NC(CCN(C)CC)=O 43036,N1(C(CC(CC(=O)OC)C)=O)CCN(C(=O)CC2CC(=O)NC2=O)CC(C)(F)C1 43037,CC1CCN(c2nnc(C(F)(F)F)s2)C(C)C1NC(C1CSC1)=O 43038,C1(NC(CNC(N)=O)=O)CCC12CCN(C(C13CCCC1C3(F)F)=O)CC2 43039,c1(C(=O)NCC(CC(C)C)NC(=O)C=CS(C)(=O)=O)cc2cc(F)ccc2o1 43040,c1(C(N2CC(NC(c3nccc(C)n3)=O)C3C2C3)=O)cc2cccnc2s1 43041,C(=O)(C(=O)C(C)(C)CC)N(CC(N1CC(C)(OC)C1)=O)C1CCC1 43042,C#Cc1cc(C(=O)NCCC(C)NC(C2(C)CCCS2(=O)=O)=O)ccc1C 43043,c1(C(N2CCC3(CC3C(N3CCC(O)CC3)=O)C2)=O)cc(Cl)cc(Cl)c1O 43044,CCCC(CC)CC(=O)NCc1cccc(NC(c2c(N)cc(F)cc2F)=O)c1 43045,C1(NC(Cc2c(C)n[nH]c2)=O)COC2C(NC(=O)CCCC(F)F)COC12 43046,c1(C(C(=O)NCC=C)N(C)C(C2CCOCC2)C)c(Cl)nc2sccn12 43047,c1(Nc2nnc(C(C)OC)s2)nc(Cl)cc2cc(Br)ccc12 43048,Cc1cc(S(N)(=O)=O)sc1C(N1C(CNC(C2C=CC=CC=C2)=O)CC2CC12)=O 43049,N1(C(c2cccc(NC(N)=O)n2)=O)CCC(CO)(NC(=O)C(O)C(F)F)CC1 43050,Cc1nc(C(N2CC3(NC(c4ncoc4C)=O)CC2C3)=O)n(C)n1 43051,N1(CCC=C)CCC2(CC1)CC2N(C(C)=O)Cc1ccc(C(=O)OCC)nc1 43052,C12(NC(CC(C)C(F)F)=O)CCOCC1CN(C(=O)C(=O)NCCC(N)=O)C2 43053,C1(CNC2CC(C)S(=O)(=O)CC2)CCc2n[nH]cc2C1 43054,c1(NCC(=O)NCC(CN(C(C(CC)C)=O)C)O)ccc(Cl)cc1Cl 43055,O=c1cccnn1CC1CCC(c2ccccc2)CC1 43056,Cc1ccc2c(c1)CN=C(NCC(c1nc(C)on1)(C)C)N2C.C1CC1 43057,C1(NC(C(C(=O)OC)C)=O)CN(C(c2cc(C)ccc2Cl)=O)CCC1(F)F 43058,c1(C(N(CC(C)NC(C2CC3CC2CC3O)=O)C)=O)ccc(C#N)cc1F 43059,c1(C(=O)OC)cc(NC(=O)NCCCC(c2ccccc2)C2CC2)c(Br)cc1C 43060,C12(CNC(C3C(C)CCO3)=O)CCC(CN(C(=O)C=C3CCN(C)CC3)C1)C2 43061,N1(C(c2n(CCC)ncc2)=O)CCC(C(=O)NCC(C)C)C1(C)C 43062,N1(C(C(CCC#C)O)=O)C(CNC(c2cccc(C(C)C)c2)=O)CC2CCCC12 43063,CCCCC(CNC(c1cocc1C)=O)NC(C1CN(C(=O)NC)C1)=O 43064,CCCC(C(O)C(=O)NCC(F)(CC)CC)NC(=O)C(O)C(C)(C)C 43065,c1(C(N2CCN(C(CCP(C)(C)=O)=O)C(CO)C2)=O)ccc(N)c(Cl)c1O 43066,CC(N=c1[nH]c(=NC2CCN(c3ccncc3)C2)[nH]c2c1COCC2)C1CCC1 43067,C1(C(N2CCCC(OC)C2)=O)COCCN(C(C2CC2(C)C(F)F)=O)C1 43068,Cc1nc(N2CCCC2)nc(O)c1CC(N1CCN(C(=O)CO)CC1C1CC1)=O 43069,N1(C(CCCC(=C)C)=O)CC2COCCC2(NC(C2CC2C(N)=O)=O)C1 43070,Cc1cc(N)c(C(=O)NCC2CC(NC(C3CCCC3)=O)C2(C)C)cc1F 43071,C1(C(C)CN(C(C)C2CC2)Cc2cccnc2)CCC(C)(C)CC1 43072,CC(C)CC(C(=O)NC(C)CN(C)C(c1ccncc1Cl)=O)N1CCCCC1=O 43073,c1(C(N(CC(CN(C(C2CCN(CC)C2)=O)C)O)C)=O)cccc(F)c1 43074,c1(COCCN(C(C2CC(OC)C2)C(=O)Nc2ncn(C)n2)C)ccc(F)cc1 43075,C1(N(C(=O)CCc2ncco2)CC)CCCN(C(=O)CCC2CCCO2)CC1 43076,c1(CC)n[nH]c(CC)c1CC(N1CC(C)(NC(C2CCC2(C)C)=O)C1)=O 43077,Cc1ccc(CC(N2CCN(C3CCN(C(c4csnn4)=O)CC3)CC2)=O)cn1 43078,CC(C)S(=O)(=O)CC(=O)NC1CCCCCN(C(=O)CC2CCC(C)CO2)C1 43079,C(=O)(C(C#N)C(C)(C)C)NCC(CCC)NC(C1(CN(C)C)CC1)=O 43080,CCC(CC(=O)NC(c1ccc(C)cc1)C)NC(=O)C=CC1CCOCC1 43081,c1(C(=O)NC2C(CNC(c3cc(OC)ncc3)=O)CCC2)noc2c1COCC2 43082,N1(C(CC(C)C)=O)CCC(N(C)C(c2cc(-c3cccnc3)[nH]n2)=O)C(C)C1 43083,N1(C(c2c(C)cco2)=O)CCC2(NC(=O)Cc3cc(F)ncc3Br)CC2C1 43084,C12CCC3(CN(C3)C1=O)O2.Cc1cc(C(=O)NCCOCc2cccnc2)c[nH]1 43085,C1(CC(=O)NC2CC(F)(F)CC2NC(C2SCCCS2)=O)CN2CCC1CC2 43086,N1(C(Cc2c(C)cccc2Br)=O)CC2(CCN(C(C3C=CCCC3)=O)C2)C1 43087,c1(CC(C(=O)NCC2CNC(=O)O2)NC(C=C(C)C2CC2)=O)cnn(C)c1O 43088,c1(C(=O)NC(C2CCCC2)CNC(C2(C#C)CC2)=O)cnn2c1CC(F)(F)C2 43089,Cc1cccc(CN(C(C)=O)CC2CCN(C(C3CCCCO3)=O)CC2)c1 43090,N1(C(CCCC(C)C)=O)CCOC2(CCN(C(=O)CCc3ncco3)CC2)C1 43091,N1(C(c2c(C)scn2)=O)CCC(OCCNC(=O)CC2CCS(=O)(=O)C2)CC1 43092,CC1=CCC(C(=O)NCCCN(C(=O)CC(C)NC(=O)OC(C)(C)C)C)CC1 43093,CCCC(O)C(CO)NC(C1(N(C)C(C2(CC=C(C)C)CCC2)=O)CC1)=O 43094,N1(C(c2n(C)ncc2)=O)CC(C(N2CCCC3C(O)CC23)=O)CCC1(C)C 43095,C1(C(=O)NCC2CCCCC2)(CNC(C(c2cnn(C)c2)C)=O)CC(C)(C)C1 43096,N1(C(C(C)N2CCC2)=O)CCC(CNC(C2NC(=O)C3CCC23)=O)C(F)(F)CC1 43097,C(=O)(CC(O)CCCC)N(CCCCC(N1C(CC=CC)CCCC1)=O)C 43098,Cc1cc(CCC(=O)NCCC(O)CNC(C2(C)CCN(C)C2=O)=O)cc(C)c1 43099,C#Cc1cncc(C(=O)NCCC2CC(F)(F)CN2C(c2nocc2Cl)=O)c1 43100,CC1CN(C(c2cc(OCC3CC3)ncc2Cl)=O)CCN1C1CCCCC1 43101,C(CC(C)CC)(C(=O)N1C2COCC1C2)NC(CC=C=C)=O 43102,n1(CC(N2CCC(CNC(C(C(C)C)OC)=O)CC2C)=O)cc([N+](=O)[O-])nc1C 43103,N(C1CC(C)n2ncnc21)C(C1CCC(NC(C2(C=C)CCC2)=O)CC1)=O 43104,N1(C(c2ncn(-c3c(N)nc(Br)cc3)n2)=O)CCC2(C1)CN(CC(=O)O)C2 43105,N1(C(CC2(COC)CCCC2)=O)CCC(C)(C)C(NC(=O)C(C)OC)C1 43106,c1(CNC(C(C(C)C)F)=O)nnc2n1CCN(C(C1(C)CCOC1)=O)C2 43107,C1(NC(C2(CCCC)CCC2)=O)CN(C(C2CN(C)C2)=O)C2(CCOC2)C1 43108,C1(C(=O)NC(c2ccccc2)C(=O)NC(C)CCCCO)CC2(CC2)CN1C 43109,CCC(C)(C)CCCC(=O)NCCC(C)NC(c1nc(C)ncc1Br)=O 43110,CC(C)(CC(=O)N1CCC(O)(CNC(=O)CCCC(F)(F)CO)C1)CC(F)(F)F 43111,c1(C(=O)NCC#CCNC(=O)CCc2cnccn2)cc(Cl)c2c(c1)OCO2 43112,C(=O)(C(F)(CNC(C1(C#N)CCCC1)=O)C(C)C)NCC(CC1CC1)OC 43113,c1(C(N2CC(C)OC(c3ccc(F)cc3)C2)=O)cc(Br)cc(F)c1N 43114,N1(C(Cc2cc(C)[nH]n2)=O)CC(C)(C(=O)N(CC2=CCSC2)C)CC1(C)C 43115,C(=O)(CC(C)(C)C(F)F)N(CC(C)(C)CNC(=O)Cc1ccon1)C 43116,C1(CC)(NC(=O)C(C)Nc2nc(C)cs2)CCCN(C(C2CCSC(C)C2)=O)C1 43117,c1(NCCN(C)Cc2c(C)nc[nH]2)cnn2ccccc12 43118,C1(CC(N2CC(NC(C(C)OCC#C)=O)(CO)C2)=O)COCC(C)(C)O1 43119,N1(S(CC)(=O)=O)CCC(F)(F)C(CN(C(=O)CC(C)(C)C)C2CC2)C1 43120,N1(C(c2ccc(C(C)=O)[nH]2)=O)CC(C)(C)CC1CC(N1CCOC(CCO)C1)=O 43121,O(NC(=O)C(CNC(=O)CC1CC(O)C1(C)C)CC(C)C)Cc1ccc(C)cc1 43122,N1(C(C(C2CC2)SC)=O)CCC(C)(NC(=O)CC2(O)CCCCC2)CC1 43123,C1(NC(CCCCSC)=O)CCC2(CC1)CC2NC(=O)C(=O)N(C)C 43124,CC1CCN(C(c2cnc(N)c(Br)c2)=O)CC1NC(=O)C(C)(C)C1CC1 43125,N1(C(c2c[nH]c(=N)s2)=O)CCC(NC(C2CC(OC3CC3)C2)=O)C12CCC2 43126,C1(C(=O)NC2(CNC(C3C(C(=O)OC)CC3)=O)CC(OC)C2)CC(C2CC2)C1 43127,C(=O)(C(CCSC)NC(c1nnsc1N)=O)N1CCC(CC=C)C1 43128,c1(C(N(C(c2ccccc2)CNC(C2CC(=C)C2)=O)C)=O)ccn(O)c(=O)c1 43129,CC1CN(C(C2(O)CCCCCC2)=O)CCC1CNC(C1CC2CCC1CC2)=O 43130,c1(C(C(=O)NC2(C)CC2)N(C(c2ccccc2)C(=O)OC)C)c(SC)cccc1F 43131,C12(C(N(C(C=C)C)C)=O)CCC1CN(C(=O)C(CCC)=CCC)C2 43132,c1(C(N2CCC3CN(C(C4CC(SC)C4)=O)C3C2)=O)cnc2sc(C)cn2c1=O 43133,c1(C(=O)NC2CN(Cc3cnc(Cl)cn3)CC2F)cc(F)c(F)cc1F 43134,C1(NC(CC2N(C(c3c(CCC)n[nH]c3)=O)CC2)=O)CC2OC(=O)CC12 43135,C1(N(C)C(C2CC2C(N)=O)=O)CCC(NC(c2c[nH]nc2C(C)(C)C)=O)C1 43136,c1(CNCC2CCC(C)(C)O2)ccc(Br)nc1F 43137,C1(C(N)=O)Cc2c([nH]c3ccccc23)CN1C(=O)CNC(c1ccon1)=O.C(N)=O 43138,c1(SC)cc(F)ccc1OC(C)C(=O)Nc1ccc(OC(=O)C(C)(C)C)cc1 43139,c1(SCC(=O)NC2COCCN(C(CC(=O)OC)=O)C2)ccc2c(c1)CCC2 43140,N1(C(c2c(C)ncc(C)c2)=O)CCN(C(=O)CC(O)C(C)C)C2(CCC2)C1 43141,N1(C(C(CC)(C)OC)=O)CCCN(C(=O)CCNC(c2ccc(C)cc2)=O)CC1 43142,C1(C(=O)NCC(CC)NC(c2cccc(-c3nnc(C)o3)c2)=O)CN(C)CCO1 43143,N1(C(C=CCCC)=O)CC(CNC(=O)Cc2cc(-c3ccccc3)on2)C2CC12 43144,C#Cc1ccc(OCC(=O)Nc2conc2C2CN(C(=O)CNC=O)C2)cc1 43145,c1(C(N(CCN(C(C2C(C(=O)OC)C2)=O)C)C)=O)nnn2c1CSCC2 43146,C(CCCCC(=O)NC(C)CCC(=O)N(C)C(c1ccccc1)C)=CC 43147,C(C)(CCCN=c1nc(NC2COCC2CO)c2ncccc2[nH]1)OC 43148,C=CC(C)C(C)C(=O)NCC1(NC(=O)CC2CS(=O)(=O)C2)CCCC1 43149,c1(C(=O)Nc2cncc(C(=O)OCC)c2)cc(Br)cc2c1cnn2C1CCCC1 43150,CC1CN(C(C2CC2c2cccc(Cl)c2)=O)CC1NC(=O)C(C)(Cl)Cl 43151,c1(C(N2CCN(c3ncns3)CC2)C(=O)NC2(C)CC2)nccc2ccccc12 43152,C#Cc1cc(C(=O)NC2C3CC(NC(C4CCC(OC)C4)=O)CC23)ccc1C 43153,c1(C(N2CCC(NC(C3(CC)CCC3)=O)C2)=O)ccccc1NCc1ccoc1 43154,C(=O)(N=c1cc[nH]cc1SC)C1CCC2(CN(C(C(CCC)O)=O)C2)O1 43155,c1(OCC)cnc(N2CCN(C(c3cc(CNC)c[nH]3)=O)CC2)nc1 43156,N1(C(c2n(CC#C)ccc2)=O)CC(NC(=O)C(C)c2cc[nH]n2)CCC1C 43157,C(c1c(N)cnn1C)=CC(N1CC(C)C(CNC(c2ccc(F)cn2)=O)C1)=O 43158,c1(C(N2C(C(C)NC(C34CC(CCO3)C4)=O)CCC2)=O)nn(C)c2c1CCCC2 43159,Cc1oc(C(C)C)nc1C(=O)NCC(C)NC(=O)CC1CC(C(F)F)C1 43160,CC(C)C(C)CNC(=O)C(C)N(C(=O)CCCNC(N)=O)C 43161,c1(NC(CC)CNC(c2csc3cncn23)=O)ccc([N+](=O)[O-])cc1[N+](=O)[O-] 43162,CC(C)CC(O)C(C)C(=O)N(C)Cc1ccc2ccccc2c1 43163,N1(C(C2C(CC)OCC2)=O)CCC(CCNC(C2(OC(C)=O)CCCC2)=O)CC1 43164,c1(CC)cccnc1C(=O)NCCC1(O)CCN(C(=O)C(C)OCCC(C)C)C1 43165,c1(C(=O)NCC2N(C(c3c(C)ccnc3O)=O)CCC2)cccc(C#N)c1Br 43166,O=S1(=O)CCCC(N=c2nc3sccc3c(NCc3nc(Br)n[nH]3)[nH]2)C1 43167,c1(CC)nnc(C(c2cccnc2)C2CCC2)n1C1CCSc2ccc(Br)cc21 43168,c1(OC)cc(C(=O)NC2CCC(CNC(=O)Cc3nc[nH]n3)C2)sc1S(N)(=O)=O 43169,C(CNC(=O)CCc1nnc(S)n1C)(CC(F)(F)F)NC(C(C)SCC)=O 43170,c1(CN2CC3C(NCc4ccc(OC)nc4Br)C3C2)c(F)cc(Br)c(F)c1F 43171,CCC(C)C(O)CC(=O)N1CC(F)CC1CC(N1CCC(C(=O)N(C)C)C1)=O 43172,c1(C(N(C2CCN(C(C3=C(C)CCC3)=O)C2)CCO)=O)c(C)nn2c1CCCC2 43173,S(=O)(=O)(c1cccc(=NC(C)c2cc(F)cc(Br)c2)[nH]1)N(CC(C)C#N)C 43174,CCCN(OC)C(=O)c1cncc(CNC(c2csc(C)c2C)=O)c1 43175,C1(OC(CC)C)CN(C(=O)Cc2ccc(C(C)=O)cc2)CC1OCC 43176,N1(C(CSc2c(OC)cccc2)=O)CCc2cc(C(=O)NC(C)C)ccc2C1 43177,C1(C(N2C(CN(C(=O)CSc3n[nH]c(O)n3)C)CCCC2)=O)CCCCC(=O)C1 43178,c1(C(=O)NCC(CNC(=O)C=CC(=O)NC2CC2)F)ncoc1C1CCCO1 43179,C1(C(N(C)CCc2ccccc2)=O)CCC(n2cc(C3CC3)nn2)C1 43180,CCCC(C)CC(=O)NCCOCCCNC(=O)CC=C(Cl)Cl 43181,CC1CC(NC(=O)CNC(=O)C=Cc2ccncc2)c2nccn21 43182,N1(C(C2CC(NC(=O)CCc3cncnc3)C2)=O)CCC2CCCC12CO 43183,CC(C)C(C)CC(=O)NCC1(CCNC(=O)CC(C)CN(C)C)CC1 43184,C12(CNC(=O)Cn3nnnc3C3CC3)CCC1CN(C(C1C=CCCC1)=O)C2 43185,C(=O)(C(F)C(C)C(F)(F)F)NCC12CCC(CNC(CC=C)=O)(CC1)CO2 43186,Cc1cncc(C(=O)NCCN(CC(C)O)C(c2cn(C3CCOC3)cn2)=O)c1 43187,c1(C(N2CCCC(NC(c3cccc(Br)n3)=O)C2)=O)cc(Br)cc(Br)c1 43188,c1(C(=O)NC(CN(C)C)C(=O)NCC#CC(F)(F)F)ccc(C#N)n1C 43189,C1(NC(CN2C(C)CCC2)=O)C=CCN(C(c2ccc(O)nn2)=O)C1 43190,Cc1ncc(C(=O)NCC2C3CN(C(=O)C(O)CC(N)=O)CC23)c(C2CC2)n1 43191,c1(C(=O)NCC2N(C(C(CCOC)OC)=O)CC(OC)C2)scc2c1CCCC2 43192,C(C(C)(C)CNC(=O)COCC1CCC1)N(C(=O)COCc1ccncc1)C 43193,C1(C(=O)NCC#CC2CC2)(CC)CCN(C(=O)C(F)C2CCOC2)CC1 43194,C1(NC(c2c(CC)ncnc2)=O)CN(C(=O)Cc2cccc(F)c2)C2CCCC12 43195,C1(c2n(CCSC)nnn2)(NCC2CC2(C)C)CCOCCC1C 43196,N=c1[nH]c(=NCc2ccc(Br)cc2F)[nH]c(=NCc2ccc(F)c(Cl)c2)[nH]1 43197,c1(C(=O)NC(CN(C(=O)C(Cl)=CCl)C)(C)C)cc(N)c(Cl)cn1 43198,C1(CN(C2CC(C)CCO2)CC)CCCN(C(=O)CCCc2cnccn2)C1 43199,CC1CC(O)CCN(C(=O)CC(C2CC2)NC(c2cnn[nH]2)=O)C1 43200,C1(C(=O)Nc2cnn(CC)c2C)CC(C)(C)CN1C(=O)CC(C)COC 43201,c1(NC(C2(CNC(c3scc(Br)c3Br)=O)CC2)=O)cc(OC(F)F)ccc1O 43202,C1(CC(=O)OC)CCCCN1N1CCC(c2ccc(F)cc2)(NC(C)=O)CC1 43203,N1(C(c2c(CNC(C(N3CCNC3=O)C)=O)nnn2C)=O)CCC12CC(C)(CO)C2 43204,c1(C(=O)Nc2c(C#N)ncc(Br)c2)ccc2cccc(-c3cnoc3C)c2n1 43205,C12(CCN(C)C1)C(=O)N2.CC(C(=O)N(C1CC1C)C)NC=O 43206,Nc1ccc(C(N2CC=C(CNC(C3CC4CCC34)=O)CC2)=O)cc1OCCO 43207,c1(C(N2C(CCNC(c3ccc(C)s3)=O)CC(OC)C2)=O)cccn2cnnc12 43208,c1(C(=O)NCC=CCNC(CC)=O)ccc(=O)n(CCF)n1.C12(CO)CN(C1)C2 43209,C(=O)(CC(C)C(F)(F)F)NCCCC(C)NC(C(CC)C)=O 43210,C1(NC(C(C)OCC)=O)CS(=O)(=O)C12CCN(C(c1cc(Cl)nc(=N)[nH]1)=O)CC2 43211,N1(C(CCOCC)=O)CCC(C(C)NC(C23CCC2C3)=O)CC1 43212,C(=O)(CCC(=O)N1CC=CC1CNC(=O)C(O)CC1CCOCC1)OC 43213,C1(C(=O)NCCN(C(=O)C(C)n2cnnn2)CCOC)(OCC)CCOC1 43214,N1(C(CC(C)c2ccccc2)=O)CCN(C(=O)COCCOCCO)C2CCC12 43215,c1(C(N2CCC2Cn2cc(CC3CCOCC3)nn2)=O)cc2n(c1)CCCC2 43216,c1(NC(C2C3(c4n(C)ccn4)CC(C2)C3)=O)nc2ccc(C)cc2s1 43217,C1(C(=O)NCC(CC(=O)NC(c2cccnc2)CC)OC)NC(=O)OC1(C)C 43218,N1(C(c2cc(C)sn2)=O)CCC2(CC1)C(NC(C1CC3CCC1O3)=O)CS2(=O)=O 43219,Cc1cc(C(=O)NC2CC2NC(=O)C(C2CCCCC2)C)cnc1C 43220,c1(SC(C)C(N2CC=CC2CNC(C2CCCN2C)=O)=O)ccc(F)c(F)c1 43221,Cc1cc(C)c(C(=O)NC23CC2CN(C(=O)C=C2CCCCC2(C)C)C3)c(=O)o1 43222,c12cnn3c1CN(CC3)C2.N1(NC(C2(C(F)(F)F)CC2)=O)CCC1NS(C)(=O)=O 43223,c1(CC(C(=O)NC2C(NC(c3ccncc3O)=O)CC2)O)cccc(Cl)c1 43224,N1(C(C(N2C(CC)CCC2)=O)=O)CCOCC1CNC(=O)Cn1nc(C)cc1C 43225,c1(C(N2CC(NC(C(C)=C(CC)C)=O)C(C3CC3)C2)=O)cccc([N+](=O)[O-])c1Cl 43226,N1(C(C(C)(C)C2CCN(C(c3ccc(N)c(F)n3)=O)C2)=O)CCc2cnccc2C1 43227,c1(N2CCN(c3cc(NC(CC=C)C(=O)O)ncn3)CC2)c(F)ccc(Cl)c1F 43228,C(CS(=O)(=O)CC(=O)N1CC2(CC(NC(=O)CCCCC(C)C)C2)C1)OC 43229,c1(C(N2C(CN(C)C(C3CCS(=O)(=O)CC3)=O)CCC2)=O)ccc2ocnc2c1 43230,N1(C(CC=C)=O)Cc2[nH]nc(C(=O)NCC(COC)C(C)C)c2C1 43231,N1(C(c2c(C)n[nH]c2)=O)CCCC1C1CCCN1C(c1csc(C(C)(C)C)c1)=O 43232,Cc1c(NC(=O)CN(c2ccc(C#N)cn2)C)cc(F)cc1[N+](=O)[O-] 43233,N1(C(c2c(CC)csc2)=O)CCC2(CCN(C(=O)C(F)OC(F)(F)F)C2)C1 43234,C(=O)(C(C)(C)CC(C)(C)C)NC1CC(C)N(C(=O)C(c2cnn(C)c2)=O)CC1 43235,Cc1cc(C(=O)NC2C3CC2CN(C(=O)C(C)C(C)C)C3)c(N)c(C)c1 43236,c1(C(N2CC(CC)N(C(=O)C(O)CC(F)F)CC2)=O)ccc2ocnc2n1 43237,CC(C)CC(C)(O)C(=O)NCCC1(O)CN(C(C2CCCN(S(C)(=O)=O)C2)=O)C1 43238,C1(C(N(CCNC(C2(C(F)(F)F)CCN(C)C2)=O)CC)=O)CNC(=O)CC1(C)C 43239,c1(NC(C(CCN(C)C)NC(=O)C(O)C2CC2)=O)ccc2nccn2c1 43240,C1(CC)CN(C(=O)Cc2ccc(C(F)F)cc2)CCN1C(c1ncc(F)cn1)=O 43241,C1(OC(C2(F)CC3(CCC3)C2)=O)CCOC2(CCCCC2)C1 43242,C(CCC(C)(C)C(=O)NCc1nonc1C)NC(C(=Cc1ccco1)C)=O 43243,C=CCC(CC(=O)Nc1cnc(Cl)cc1C)NC(=O)CCC1OCCO1 43244,c1(C(=O)NC(C(N2C(C(CC)C)CCC2)=O)C2(O)CC2)cnn2c1CCC2 43245,N1(C(C(N2CCCCCC2)CC)=O)CCCC2CN(c3ncc(C)c(O)n3)CC12 43246,C1(C(NOC(CC)C)=O)CN(C(=O)C(C)(C)CC#N)CC1(C)C 43247,C#CCC(CC(=O)NC(c1nnc(C)o1)C)NC(C1CCCN1C(C)=O)=O 43248,c1(C(=O)NC(C(=O)NCC2N(C)CCOC2)CCF)cn(C)ccc1=O 43249,C(C(C)C(C)C(=O)NC1CC(CCNC(=O)COCc2ccnc(O)c2)C1)OC 43250,c1(CC(=O)NC2CCC2NC(c2ccc(O)nc2Cl)=O)n[nH]c2ccccc12 43251,N1(C(COC2(C)CN(N(c3ccc(C=O)o3)C)C2)=O)CCCC1(C)C1CC1 43252,C(=O)(NN1CCCC1C(=O)NCCSCCCO)c1c(CC)c[nH]n1 43253,Cc1sc(Cl)nc1C(N1CC(NC(=O)Cc2ccsc2)CC1CO)=O 43254,C1(C(=O)NCC(=O)NCC#C)N(C(=O)C(C)NS(C)(=O)=O)CCC1(C)C 43255,Cc1ncnc(C)c1NC(C1CCCCN(C(C23CC(F)(C2)C3)=O)C1)=O 43256,N1(C(C(C)CS(C)(=O)=O)=O)CCN(C(=O)CNC(n2cncn2)=O)C2(CCC2)C1 43257,N1(C(C=C(CC)CC)=O)CCC(O)(CCNC(c2csc(Cl)n2)=O)CC1 43258,c1(C(N2CCCC2CNC(C2COCCO2)=O)=O)ccc(C(F)(F)F)cn1 43259,c1(C(C(=O)NC)C(N2CCC2C2CCC2)=O)ccc(OC(F)(F)F)cc1 43260,c1(NC(C2CN(Cc3ccc(OC)c(Br)c3)C2)=O)ccc2c(ccn2C(C)=O)c1 43261,c1(C(=O)NC2CCC(C(N3CCCC(C)CC3)=O)CC2)c(F)cc(Cl)cc1F 43262,c1(C(=O)NC2CN(C(c3c(OC(C)C)cccc3)=O)CC2O)cc(Cl)ccc1Cl 43263,c1(C(N(C(CNC(C2(C(C)C)COC2)=O)C)C)=O)cc(C(N)=O)cs1 43264,C1(C(N2C(CC(=O)NC)CCCC2)=O)CN(C(=O)CC(F)(F)F)CCN1C 43265,c1(C(=O)NC2CCN(C(c3scnc3Cl)=O)CC2)cnc2c(c1)C(=O)CCC2 43266,Cc1cc(C)n2nc(C(=O)NCCCCCNC(c3cnc(Cl)[nH]3)=O)nc2n1 43267,N1(C(CC(C(C)C)OCC)=O)CCN(C(c2c(C)cccc2Cl)=O)CC(C)(C)C1 43268,C(=O)(CCC(C)(F)F)N(CCCCCC)CCNC(=O)C=CC(F)(F)F 43269,N1(C(C(C=C)(C)CC)=O)CC(C2CN(C(c3[nH]c(=N)ccc3C)=O)C2)C1 43270,c1(N2C3C(NC(=O)CC4CCOC4)(CCC3)CC2)ncnc2[nH]ccc12 43271,N1(C(Cn2ncc(C)c2)=O)CCCCC1c1cn(Cc2ccoc2C(=O)O)nn1 43272,C(CC)(CCCC(=O)NCc1cc(C#N)cs1)NC(C1(CC#C)CC1)=O 43273,C(CCC(=O)NOCC(C)(C)C)(C(C)C)NC(c1c(F)ccc(C)c1)=O 43274,CCCCC(CC)C(=O)NC(C)CCCNC(=O)C(c1ccc(OC)cc1)=O 43275,C1(C)(CNC(CCN(CC=C)C(c2cc(N)cc(F)c2)=O)=O)CCCCC1O 43276,C(CCC(C)C(=O)NCC1(C)CCN(C(C2(C)CC3CCC2O3)=O)CC1)OC 43277,C(=O)(C1Cc2ccccc21)N1CCCC(CCNC(Cc2ncc(C)[nH]2)=O)C1 43278,c1(C(=O)NC2(C)CCN(C(C3C(Cl)(Cl)C34CC4)=O)C2)cnc2cccnn12 43279,c1(CC(=O)Nc2c(C(=O)O)c(-c3ccccc3)cs2)csc2ccc(Cl)cc12 43280,Cc1nc(N2CCC(C)C2CNC(C2COCCN2CC(F)F)=O)[nH]c(=N)n1 43281,c1(C(=O)NCC=CCNC(C(C2CC2)SC)=O)cccc(CS(C)(=O)=O)c1 43282,C(=O)(C(C)(C)C1CCOCC1)NCCCN(C(c1ncoc1C1CCC1)=O)CC 43283,c1(C(N2CCC(C)C(NC(C3(C)CC(C#N)C3)=O)C2)=O)ccc(Cl)c2occc12 43284,n1(CC)cc(Cl)c(C(N2CCCC2C(C)(C)NC(=O)C(COC)N(C)C)=O)n1 43285,c1(C(N(C(CNC(CCOC(C)C)=O)C)C)=O)ccc(F)cc1 43286,C1(N(C(=O)COCC2CC2)CC#C)CCN(C(c2cc(O)cs2)=O)CC1 43287,c1(OCC)cccc(C(=O)OCc2ccc(OC)nc2F)c1CSc1ccccc1 43288,N1(C(C2(CC#C)CCCO2)=O)CCCC(N(C(=O)CCC2OCCO2)CCO)C1 43289,C(=O)(C(C)C(C)C(C)(C)C)NCCC1(CNC(c2c(C)cc(CC)o2)=O)CC1 43290,C(C)(C)(CC(=O)NCC(O)CC(=O)Nc1cnn(CCF)c1)OC 43291,N1(C(c2c(CC)n[nH]c2)=O)CC(C(N2CCC3C(OC)CC23)=O)C(F)(F)C1 43292,C(C(C)(C)C(=O)NC1CCN(C(=O)C(C)C(F)F)C1)NC(C)=O 43293,c1(NC(N2CCN(CC(O)CO)CC2)=O)ccc(C2CCOCC2)cc1 43294,C1(CNC(C(CC2CCC2)OC)=O)CCC(C)CN1C(=O)COC1CCC1 43295,Cc1cc(O)cc(C)c1CC(=O)NCC1(O)CC(NC(c2coc(CO)c2)=O)C1 43296,c1(C(N2CC(NC(C(COC)C)=O)C2)=O)ccc(N2CCOC2=O)cc1 43297,Cc1ccc(C(N2CCCC2C(C)(C)CNC(=O)C(C)(C)C(F)F)=O)c(O)n1 43298,c1(C(N2CCC(C(=O)NCC=C3CCSCC3)(OC)C2)=O)cc(C#N)oc1C 43299,C1(C(=O)NCCOCCN(C)C(c2cccs2)=O)CCCC1S(C)(=O)=O 43300,C1(CNC(c2ccc(=O)n(C3CC3)c2)=O)CC(F)(F)CN1C(c1scnc1Cl)=O 43301,N1(C(CCOC2CN(C(CC3CCC(C)CC3)=O)C2)=O)CCCNC(=O)C1C 43302,C1(C(=O)NC2C3CN(C(CN(C)C4CC4)=O)C2CC3)CCn2cnnc2C1 43303,C=CCC(C)C(=O)N1CCC(OC2CN(C(=O)C(N3CCNC3=O)C)C2)CC1 43304,c1(NC(N2CCCC(C(=O)OCCOc3cccc(F)c3)C2)=O)ccnc(O)c1 43305,N1(C(c2c(C(=O)OCC)con2)=O)CC(C2CCCN(C(=O)C(C)C(C)O)C2)C1 43306,C1(C)(CNC(Cn2c(C)c(Cl)cn2)=O)CN(C(c2cncnc2)=O)CCO1 43307,Cc1cccnc1C=CC(N1CCN(C(=O)CC(C)C(F)F)C(CO)C1)=O 43308,c1(C(N2CCCC(CCC)(NC(=O)C(O)C3CCC3)C2)=O)ccc2nncn2c1 43309,C1(F)(C(=O)NC(C(=O)NC(C)CCC2CCCC2)CNS(C)(=O)=O)CCCCC1 43310,C12(CNC(C(CC)c3ccccc3)=O)CC(NC(c3cc(C)[nH]n3)=O)(CCO1)C2 43311,c1(CCC(=O)NCC2(NC(c3ccnnc3)=O)CCCCC2)ccc(CO)nc1 43312,C1(CNC(C(C)(C)c2ccno2)=O)CN(C(C2CCCC2)=O)C2CCCC2O1 43313,c1(C(N2CC(NC(CCCSC)=O)C(O)C2)=O)c(C)ccc2n[nH]cc12 43314,c1(-n2cc(C(=O)NCC3CNCC(F)C3)nn2)c(F)cccc1Br 43315,c1(N2CCN(CC(C)C)CC2)nc(N2CCSC(C)(C)C2)nc2cccnc12 43316,C1(NC(c2c(C)cc(C)s2)=O)CN(C(C2CC3(C2)CC3F)=O)CC2(CCC2)C1 43317,c1(N(c2ccccc2)C(C2CCN(C(C)=O)C2)=O)nc(C)cc(O)n1 43318,C1(CNC(=O)C(C2CS(=O)(=O)C2)O)C2CN(C(c3cnccc3Cl)=O)CC12 43319,c1(CC)cc(N)ccc1C(N1CCC(CN(C(=O)CC23COCC(C2)C3)CC)C1)=O 43320,c1(C(N2CCOCC(NC(CC(C)(C)OC)=O)C2)=O)cc2cc(F)cc(F)c2[nH]1 43321,c1(C(N(C2CN(C(c3nc(C)sc3)=O)C2)C)=O)cc(Br)cn2ccnc12 43322,n1(CC(N2C(CN(C(C3C(=C)C3)=O)C)CCC2)=O)nc(C)cc1C(F)F 43323,C1(CNC(C(CC)(F)F)=O)CC2CCC1N(C(=O)C(COC)NC(C)=O)C2 43324,CC(C)(C#N)CC(=O)NCCC1CC(NC(=O)CNC(=O)NC2CC2)C1 43325,C(=O)(C1=C(C)CCCC1)NC1C(SC)CN(C(=O)C(=Cc2ccc(F)cc2)C)C1 43326,N1(C(C(C)C2(O)CCC2)=O)CC2(C=C(C(=O)NC3CCCN(C)C3=O)CO2)C1 43327,c1(OC)c(C(=O)NCC#CCNC(C2CNC(=O)CC2C)=O)oc2ccccc12 43328,c1(CC)cc(C(=O)NC(CC(=O)N(CC(=O)OC)C)C2CC2)n[nH]1 43329,c1(C(C(=O)NC(CC)C)N(CCCO)C(C)C)ccc(C2CCCC2)cc1 43330,n1(CC)nc(C(=O)NC(C)(CSC)C(=O)NCC(=O)OC(C)C)c(C)n1 43331,c1(OC)ccccc1CCNC(=O)C(=O)NC1CCCNCC1 43332,c1(C(=O)NC(C2(CO)CC2)C)ccc(C(C2CC2C)=O)cc1.C1CN1 43333,N1(C(C=CC(C)(C)C)=O)CCN(C(=O)CCc2ccc(Br)cc2)CC12CC2 43334,N(C(=NCCCN(S(CC)(=O)=O)C)NC(C1(O)CCOCC1)C)CCCOC 43335,CCC(O)(C(=O)N(CC(O)CNC(=O)CN(C)C1CC1)C)c1ccccc1 43336,C1(COC)CC(CNC(C2(C)CCNC2=O)=O)N(C(=O)CCOC2CC2)C1 43337,C1(C#N)(C(=O)NC23C(CN(C(COCc4ccc(C)cc4)=O)C2)C3)CC2CC2C1 43338,CC(C)(CCl)C(=O)N(C1CC2CC1CN2)CC1CCOCC1 43339,c1(OC)c(C(=O)NCc2ccc(I)cc2)cccc1Br.c12ccc(nc1)[nH]c2=O 43340,C1(CS(=O)(=O)Nc2ccc(C(=O)OCCSC)cn2)(OC)CCOCC1 43341,N1(C(c2ccn(CC)c(=O)c2)=O)CCCC2CN(C(C3(CC4CC4)CC3)=O)CC12 43342,c1(N(C(=O)CCCn2cccn2)Cc2ccc(Cl)cc2)cccc2c(I)n[nH]c12 43343,Cc1cccnc1CNC(C1CCN1C(C1CC(n2cccn2)C1)=O)=O 43344,C1(C(=O)NC(CCN(C(c2c(C)onc2)=O)C)C(C)C)CCC(=O)C(C)C1 43345,C12(C(=O)NC(CN(C(C(C)=CC3CC3)=O)C)(CO)CO)CC3CC1C2C3(F)F 43346,Cc1cc(C(F)F)nn1CC(N1CC2C(NC(C3COC(=O)O3)=O)C2C1)=O 43347,N1(C(c2cc(C)sn2)=O)CC23CCCC2(C1)CN(c1nnc(C(N)=O)s1)C3 43348,c1(C(=O)NC2C3(NC(c4ccncc4)=O)CCC(C2)C3)nnn2c1CCCC2 43349,Cc1cc(NC(C2CC(F)CN(C(c3cc(Cl)cnc3Br)=O)C2)=O)cnc1C#N 43350,Cc1c(CN=c2[nH]c(C(=O)NC(C)(C)C)cs2)cccc1C#N 43351,Cc1cccc(OCC(=O)N(C(C)CNC(C2(S(C)(=O)=O)CC2)=O)C)c1F 43352,Cc1c(N(CCCN(C2CCCC2)C)C)ncnc1N1CCOC(C(N)=O)CC1 43353,C12(NC(CCC(=C)Br)=O)CCC(C1)N(C(C1CC(C3CC3)=NO1)=O)C2 43354,N1(C(C(CC#C)CC(F)F)=O)CCCC2C1CCCN2C(=O)OC(C)(C)C 43355,c1(OC(CC)C)ccccc1C(=O)NC1CCN(C(=O)C(C)c2cccs2)CC1 43356,CC(C)CC(O)C(C)C(=O)N1CCC(CNC(c2coc(CO)c2)=O)CC1 43357,C1(C(=O)NC2C(NC(COC3(C#C)COC3)=O)C2)CN2CCCC2CO1 43358,CC(N=c1[nH]c(=NCC(CO)C(F)(F)F)c2[nH]ccc2[nH]1)c1c(F)cccc1Cl 43359,c1(OC)cc(C(N2CCC(C(N3CCOC(C#N)C3)=O)C(O)C2)=O)cc(OC)n1 43360,C1(CNC(=O)COc2ccccc2)CCN(C(=O)CSC(F)F)C12CC2 43361,c1(NC(C(N2C(C)CC(C(=O)NC3(CCOC)CC3)C2)=O)=O)ccc(C)c(C)c1 43362,CCCC(C(=O)N1CC(C(=O)NCC2CCC2C)C1)OC 43363,Cc1cc(C(=O)NCCN2CCC(NC(=O)CC3CCC(=O)N3C)CC2)nn1C 43364,C1(C(N(CCCCN(C(c2c(C)snc2)=O)C)C)=O)CNC(=O)CC12CCOC2 43365,c1(OC)ccccc1C1CC1C(=O)N(CC(C)(C)NC(c1nn(C)cc1C)=O)C 43366,N1(c2ncc(CC)c(C)n2)CCOC2CN(Cc3cc(Br)cc(C)c3O)CC12 43367,n1(C2CC(C)C2)nc(CC2CCCC2)nc1C1CC1(C)OC(C)(C)C 43368,c1(C(=O)OC)ccc(F)c(C(=O)NC2CCN(C(=O)C=CCN(C)C)CC2O)c1 43369,C1(C(N2CC(C)(NC(c3cc(OCC)n[nH]3)=O)C2)=O)(C(=O)OC)CC1S(C)(=O)=O 43370,c1(OC)cc2[nH]ncc2cc1C(N1CC2(CCC(C(=O)NC(C)CCO)O2)C1)=O 43371,C1(CNC(CN(C(COC)=O)C)=O)CC2CCC1N2C(C1CN(C)C(=O)N1)=O 43372,C1(C(N2CC3C(NC(Cc4c(C)cc(F)cc4)=O)(C3)C2)=O)CN(CP(C)(C)=O)C1 43373,n1(CCOC)cc(C(N2CC(NC(=O)Cc3cncs3)CC(C)C2)=O)ccc1=O 43374,C1(N(C(C(CCC)OCC)=O)C)CC2CCC(C1)N2C(=O)C(C)c1ccsc1 43375,C1(CNC(C(C)OCCCC)=O)CC2(CC(NC(=O)CS(=O)(=O)N(C)C)C2)C1 43376,c1(NC(C(CC(F)F)NC(CCCN=[N+]=[N-])=O)=O)ccc2c(c1)COC2 43377,N1(C(C2CCN(CC(C)C)CC2)=O)CC(NC(=O)Cc2cnns2)CC12CCC2 43378,Cc1cc(C(=O)NC2CC3CC2CC3C(N2CCC(F)(CF)CC2)=O)cnc1O 43379,c1(C(=O)NCC2N(C(C(C)C#N)=O)CC2)cnccc1C(F)(F)F 43380,c1(CC(N2CCCC(CN(C(=O)Cc3ccccc3)C)C2)=O)cccc(F)c1F 43381,C12(CC(=O)NCCCCNC(c3nccc(N(C)C)c3)=O)CCCCC1C2(F)F 43382,C1(CNC(COc2cccc(C(C)C)c2)=O)Cc2ccccc2CO1 43383,N1(C(C(C=C=C)C)=O)CCCC(C2CCN(C(=O)CCC(=O)OC)CC2)CC1 43384,c1(OC)cccc(C(=O)NC2CC(NC(C3CCC(C(F)(F)F)C3)=O)C(O)C2)c1 43385,Cc1cn(C)nc1C(N1CCCCC1CC(N1CCCC1(C)CO)=O)=O 43386,C1(NC(Cn2c(C)ncc2)=O)CCCN(C(c2ccc([N+](=O)[O-])cc2)=O)CC1F 43387,C(=O)(C(C)(C)CNC(=O)CCc1ccc[nH]1)NC1CC(CCOC)C1 43388,Cn1cnc2sc(C(=O)NCC(C3CC3)NC(C3CSCCS3)=O)cc12 43389,N1(C(CSCCC)=O)CCN(C)C(CNC(C2(c3ccccc3)CC(O)C2)=O)C1 43390,c1(NC(C(C2CC(NC(CCc3cc(C)[nH]n3)=O)C2)F)=O)ccc2c[nH]nc2c1 43391,C1(NC(C=CCCC(C)C)=O)CCCN(C(c2cnn(C3CC3)c2)=O)CC1 43392,c1(C(=O)NCc2cn(CC(CC)O)nn2)cc2c(C)cc(C)cc2[nH]1 43393,c1(C(=O)NC2C(NC(C(C)CN3CCCCC3)=O)CCC2)ccc(O)cc1 43394,CC(C)(CN=c1[nH]cnc2[nH]cc(C(F)(F)F)c12)N1CCOCC1 43395,N1(C(c2c(C)cn(C)n2)=O)CC(NC(C2COCC(C)O2)=O)C2(CCCC2)C1 43396,Cc1cc2c(C(=O)NC3COCC3NC(c3cc(CO)[nH]n3)=O)nccn2n1 43397,C1(NC(C2CN(C)C(=O)CC2)=O)CCC2CN(C(=O)COCC(F)(F)F)CC2C1 43398,CCCCC(C)CCC(=O)N1CCC(CNC(=O)C(C)NC(=O)NC)C12CCC2 43399,N1(C(C(C)C(F)F)=O)CC(CNC(C2(c3cccc(C#N)c3)CC2)=O)CC1(C)C 43400,N1(C(C=CC2COC(C)(C)O2)=O)CC(NC(=O)CC2CC2)CC2(CCC2)C1 43401,c1(C(N2CCCC(C(C)NC(c3ccc(Cl)cn3)=O)C2)=O)cc2n(c1)CCOC2 43402,c1(-c2cc(CNC(N3CCCC(CC(=O)OC)C3)=O)[nH]n2)ccc(F)c(C)c1 43403,C(=O)(C1=C(F)CN(C(c2csc(C)c2)=O)CC1)N1CC(C)CC(OC)C1 43404,C1(NC(=O)COC(F)(F)F)CCCCCCC1O.CC1CCC2CN1C2=O 43405,n1(C(C)C)cc(C(N2CCC3(CC3NC(=O)C(C)n3cncn3)C2)=O)ccc1=O 43406,c1(C(=O)NC2CCCC(NC(C3CC3F)=O)C2)cnc2[nH]ccc2n1 43407,Cc1cnc(S(C)(=O)=O)nc1N1CCC2(C(N3CC(CO)C(O)C3)=O)CC2C1 43408,N1(CCC)CCC(C(=O)NC2CN(C(=O)OC(C)(C)C)C2)C(O)C1 43409,CC1Cn2nc(C(=O)NCCCCCNC(=O)C(F)OC(F)(F)F)cc2C(=O)N1 43410,c1(CC(C)NC(=O)NCC2COCCN2)ccc(F)cc1Cl 43411,C(=O)(C(CCC(C)C)NC(=O)CCC1CCCCC1)Nc1ccc(OC)c(C)c1 43412,c1(N(C)C)ncnc(NC(C2COCCN2C(=O)OC(C)(C)C)=O)n1 43413,c1(N2CC(NC(C(C3CCOCC3)C)=O)C(C)(C)C2)ncc(Br)cc1C#N 43414,C(N=c1[nH]c(=NCCc2nccc(O)n2)c2[nH]ccc2[nH]1)c1c(C#N)cccc1 43415,O=C(CC1(C(=O)O)CCc2ccccc21)N(C1CCCO1)Cc1cc(Br)ccc1F 43416,CC(C)CC(O)CC(=O)NCCn1ccc(C(=O)N(CCCC(C)O)C)c1 43417,C(C1=Cc2cc(Cl)ccc2OC1)=CC(=O)NC1CCN(C(CN(C)CC)=O)C1C 43418,c1(OC)cc(C(N2CCC(N(C)C(c3cnc(Cl)cc3I)=O)C2)=O)ccc1O 43419,c1(OC)ccccc1NC(=O)C(C1CN(C(C2(SC)CCC2)=O)C1)OC 43420,C1(c2nnnn2C2CC2)(NCCC(=O)NC2CCCCC2)CCC(=O)NC1 43421,N1(C(c2nc(C)oc2C)=O)CCOC2CCN(C(C3CCC(F)CC3)=O)CC12 43422,N1(C(CCOCC#C)=O)C2CCC1CN(C(=O)Cc1ccccc1CC)C2 43423,C1(C(=O)Nc2c(C)cc(SC3CC3)cc2)CCc2ccnn2C1 43424,C1(C(N(CC(=O)NC)CC)=O)CC12CCN(C(=O)Cc1ccc(C)nc1)CC2 43425,C1(C(=O)NCC(CN(C(=O)CSCC(=O)NCC)CC)(C)C)CCCC2CCCN12 43426,C(=O)(CCCC(F)F)NC(CN1CCN(C(C2CCN(C(C)=O)C2)=O)CC1)C 43427,N1(C(CC=CCC)=O)CC2ON=C(CNC(C3CC(S(C)(=O)=O)C3)=O)C2C1 43428,N(C(=NCC)NCC1CCCN(C(C)=O)C1)CC(F)=CC 43429,Cn1ncc2c(C(=O)NC3CCC34CN(C(=O)CC3CC=CCC3)C4)ccnc12 43430,CC1(C)CC(C(N2CCCCC2C2CCCN(C(=O)COC(F)F)C2)=O)CO1 43431,CC12CN(C(=O)C3=COCC3)C(C(=O)NC(c3cscn3)CO)(C1)C2 43432,N1(C(c2c(C)n(C)cc2)=O)CCOCCC1C(N1CC(S(C)=O)C1)=O 43433,C1(C(=O)NC(C)(CC(=O)O)c2cccc(F)c2)CCn2nncc2C1 43434,C12(NC(CCCSC)=O)CCN(C(c3cc(O)nn3C)=O)CCC1C2 43435,Cc1cccc(C(O)C(=O)NCCC(C)NC(c2c(C)[nH][nH]c2=N)=O)c1 43436,C(C(S(C)(=O)=O)C1CC1)NC(c1ncccc1F)(c1n(CCSC)nnn1)C 43437,C1(C)(C(=O)NC2CC(C)N(C(c3ccon3)=O)C2)CCC(C)(C)CC1 43438,CCC(C)CC(C)C(=O)N1CCC(C)(NC(c2cc(=O)c(OC)cn2C)=O)C1 43439,N1(C(C(C)=C(C)C)=O)CCCC1C1(C(=O)N(C2CC=CC2)C2CC2)CC1 43440,N1(C(c2c(OCC#C)nccc2)=O)CCCC(C2CCN(CC=C)C2)C1 43441,N1(C(C(C)SC)=O)CCC(NC(=O)COc2ccc(F)cc2F)C(F)(F)CC1 43442,C1(NC(c2n[nH]c(CC)c2Cl)=O)CCN(C(=O)CSCC(=O)OC)CC1C 43443,Cc1ccccc1CN1CCCC1CN(C(=O)CCCOCCN(C)C)C 43444,N1(C(C2CC(O)(CNC(c3c(CC)nn(C)c3)=O)C2)=O)CCN(C)C(C(C)C)C1 43445,N1(C(CSc2c(C)n[nH]c2C)=O)CCC(NC(=O)CN2CCCNC2=O)CC1C 43446,N1(c2cc(OC)ncn2)CCC(CNc2ncnc3ccsc23)C(F)(F)CC1 43447,N1(c2n(CC(C)C)c(-c3cnc(O)nc3)nn2)CCC2CCCC12CO 43448,C1(O)(C(CNC(=O)C=CSc2nc[nH]n2)NC(C2CCC(O)C2)=O)CCCCC1 43449,CC1(CO)CCCN1C(=O)Cn1cc(I)nn1 43450,c1(C(N2CC(NC(c3cc(C)no3)=O)C(F)C2)=O)cc(F)c(C)cc1F 43451,C(C(CC(C)C)C(=O)N(C1CC1)Cc1ccoc1)NC(COCC(=O)NC)=O 43452,c1(C(=O)NC(CCN(C(C(COC)(C)OC)=O)C)C(C)C)c(C)cc(Cl)cc1N 43453,C(=O)(C(C)(F)C(F)(F)F)NCC1CCN(C(C=Cc2ccc(C)cc2)=O)C1(C)C 43454,C1(C)(CNC(c2c(C)nn(C)c2)=O)CN(C(=O)C=Cc2ccc(Cl)s2)CCO1 43455,C1(N(C(c2ccn(CCF)n2)=O)C2CC2)CCOC(C(N2CCOCC2)=O)C1 43456,C1(CC(=O)N(C)CC2CCN(C(=O)COCCCF)C2)CCCC2(CC2)C1 43457,C12(C(=O)NCC3(C(F)(F)F)CCN(C(CC#N)=O)C3)CC(CO)(C1)OC2(C)C 43458,CCCCCC(C(=O)N1CCC(C)(NC(c2onc(C)c2C)=O)CC1)C(C)C 43459,C(=O)(C(CCC(=O)OCC)N1CCCC(c2ccn(C)n2)C1)NCCC 43460,c1(C(=O)NCCCC(C)NC(c2cn(C)cn2)=O)nc(Cl)sc1Cl 43461,CC1(C)CCCC(CNC(C2CCC(CNC(C3SCCS3)=O)O2)=O)O1 43462,CC(C)(C(=O)N1CC(NC(=O)Cc2ccsn2)CC(O)C1)C(N)=O 43463,C12(NC(C(CC=CC)CC)=O)CCC(CN(C(c3ccc(OCC)nc3)=O)C1)C2 43464,Cc1cccc(C)c1CC(=O)NC1(CNC(=O)C(CO)NC(=O)CC(C)C)CC1 43465,C1(NC(C2(CC)COC2)=O)CC(NC(=O)C(C)OCC(C)C)CC1O 43466,C1(C(C)NC(C(C)CO)=O)CCN(C(c2cn(-c3ccccc3Cl)nn2)=O)CC1 43467,Cc1nc(C)c(C(=O)NCC2CC(F)(CNC(C3CCC(C)O3)=O)C2)nc1C 43468,CC1CC(Cc2ccccc2)CCN1C(C1CCCN1CN)=O 43469,C=C(CNC=O)CCNC(=O)OC(C)(C)C.C(CC(O)CSC)NC(=O)CNC 43470,c1(C(=O)NC2(COC)CN(C(C3CC3C)=O)C2)cn(C)c2ccc(Br)cc12 43471,C1(NC(C(C)C2CCC2)=O)C(C)CCN(C(c2ncc(C(F)(F)F)n2C)=O)C1C 43472,C1(C)(C(=O)NC2N(C)C(=O)CC2)CCCN(C(=O)Nc2cccc(Cl)c2F)C1 43473,C(CSC)(CN=c1nc(N(C)Cc2nc(-c3ccncc3)n[nH]2)cc(C)[nH]1)OC 43474,c1(C(=O)NC2C(C)CCN(C(c3cc(Cl)cnn3)=O)C2)ccc2nc(O)oc2c1 43475,C1(C(=O)NCCc2cc(C(=O)O)no2)(OC)CCS(=O)(=O)C1 43476,C1(C(N2CCCC(F)(C(=O)NCc3c(C)nc(C)[nH]3)C2)=O)CC(=O)CC12CCC2 43477,N1(C(C)=O)CC(O)CC1C(N1CC(C)(NC(=O)Cn2nc(C)nc2C)C1)=O 43478,c1(OCCOC)ncccc1C(=O)NCCC(C)NC(=O)CC1CCC(C)(C)C1 43479,N1(C(C(C)OCC=C)=O)CC2CC1C2CNC(=O)C(C)COC 43480,c1(OCCC(N2CCC(C(C)NC(CCC#C)=O)CC2)=O)cc(C)cc(C)c1 43481,C(=O)(CC(C)(C)C1CC1)N(C1CC1)CC1N(C(C(c2ccc(Cl)s2)C)=O)CCC1 43482,C1(CNC(C(C)SC)=O)CN(C(c2ccc(C(F)(F)F)cc2N)=O)CC1(F)F 43483,C1(C(C)NC(CCN(CCC)C)=O)CCCN1C(=O)CC1CCCO1 43484,c1(C(=O)NCC2C3N(C(c4c(C)cc[nH]4)=O)C(CC3)C2)cc2ncccc2o1 43485,C1(C(=O)NCC(C2CCCCC2)NC(C(C)n2ccnc2)=O)CCCC(C)(C)O1 43486,C(=O)(C(CO)C(F)(F)F)N(C)CC=CC(=O)NCC1CC(F)C1 43487,N1(C(c2c(C)nsc2)=O)CC(C)CN(C(=O)C(=O)Nc2ncc[nH]2)CC1C 43488,c1(N(CC(C)C)C)nc(=NCC2(CO)CC23CCC3)[nH]c2c1CC(C)CC2 43489,C1(C(N2CCN(C(C3CN(C(C(C)(C)O)=O)C3)=O)CC2)=O)CC2(C1)CC(C#N)C2 43490,N1(CCOC)CCN(C(c2ccccc2I)C(=O)NCC2CCOCC2)CC1=O 43491,C1(NC(c2c(C)nc(CCC)o2)=O)COCCN(C(c2ccc(C#N)s2)=O)C1 43492,O=C(N=c1ccn(C2CC2(F)F)[nH]1)C1=C2CCN=C2NC=C1 43493,C1(CC)CN(C(C2C=CCC2)=O)CCC1NC(c1ccc(=O)n(C)c1)=O 43494,C1(C(=O)NC(CC)(CSC)C2CC2)CN(C(=O)Nc2ccc(OC)s2)CC1C1CC1 43495,c1(NC(CC2CN(C(C3(Cl)C(C(C)=O)C3)=O)C2)=O)ccc(C2CC2)nn1 43496,C12(C(N(C)CC3(OC)CCC3)=O)CC(C)(CN1C(=O)Cn1cc(C#N)cn1)C2 43497,C(C(CCC)C(=O)NCC1COCCN1C)NC(CSCC#C)=O 43498,c1(C(N2CCC3CCCC23CNC(C2(CO)COC2)=O)=O)cn2cccnc2n1 43499,C12(NC(CCCC#C)=O)CCCCC1N(C(c1ncccc1F)=O)CC2 43500,Cc1cccnc1CC(=O)NC1(CCC(=O)NOCCC2CC2)CCCC1 43501,C1(C(N(CCCNC(=O)CCc2cccc(O)n2)C)=O)CCC2CCCCN12 43502,C(=O)(C(C)(C)CC1CCOC1)NC1C(NC(=O)NC)CCC1 43503,N1(CC2CN(C(C3(C)C(C)(C)C3)=O)C(=O)C2)CC2CCC(C1)O2 43504,N1(C(C2(C(C)C)CCCO2)=O)CCC(NC(=O)C(CCO)N(C)C)CC1 43505,CC(C)(CC(F)F)C(=O)N1C2CCC1CC(NC(c1ccc3cc[nH]c3n1)=O)C2 43506,CCC(CCCC(=O)NCC1(CF)CCC1)NC(c1cc(OC)n(C)n1)=O 43507,c1(CC(=O)NC2C(CNC(c3c(OC)scc3)=O)CC2)nn(C)c2ccccc12 43508,C1(NC(C=C(C)C)=O)CCN(C(c2ccc(Br)cc2C)=O)C2CC12 43509,N1(C(C(CC)N(C)C)=O)CCC(NC(C2CN3CCC2CC3)=O)C12CCCC2 43510,N1(C(CS(=O)(=O)NCC)=O)CCC(NC(c2ccn3ccsc23)=O)C(C(C)C)C1 43511,O=C1CCC(CNC(c2ccc(CNC(=O)CC3CCCO3)s2)=O)O1 43512,C1(NC(=O)CN2C(=O)C=CC2=O)CN(C(c2cccc(CO)c2F)=O)CC1(F)F 43513,N1(C2(C=O)CC2)CC(C)(CNC(C2(CCOC)CCC2)=O)CC1(C)C.C(F)(F)F 43514,c1(NC(C2CC(C(=O)NCCCC(OC)OC)C2)=O)c(Cl)nc(C)nc1Cl 43515,C1(C)(CNC(CN(CCC#C)C)=O)CCC(NC(C2CCN(C(C)C)CC2)=O)C1 43516,C1(CNC(C2CCCOC2)=O)CC12CCN(C(=O)CC1CC3CC(=O)C1C3)CC2 43517,N1(C(C(C)=C2CC2)=O)CC(C)CN(C(c2nc[nH]c3ncnc2-3)=O)C(C)C1 43518,c1(Nc2ccc(C(=O)OC)nc2I)c([N+](=O)[O-])cc(C(F)(F)F)cc1[N+](=O)[O-] 43519,n1(C(C)(C)C)cc(C(=O)NC23CC(NC(=O)C(Cl)=CCl)(C2)C3)cn1 43520,C(CCCC(F)(F)F)OC12C(CN(c3n(CC)c(C(C)F)nn3)C1)CC2 43521,C1(CC)(CC)CCN1C(=O)OC(C)(C)C 43522,CCCC(O)C(=O)N1CCC(N(C(=O)CC(C)SC)CC)C1 43523,c1(C(N2CC3(CCN3C(=O)C=Cc3cccnc3)C2)=O)c(F)ccc(F)c1F 43524,CC(C)(C)CCCNCCS(N1CCCC(CCC(=O)OC(C)(C)C)C1)(=O)=O 43525,C1(N(C(C(=O)NCC)c2cnsc2)C2CC2)CCS(=O)(=O)C1 43526,C(CCC(=O)N1CCN(CCO)C(C)C1)(C(C)C)NC(c1c(C)coc1)=O 43527,C12(NC(C(CC=C)NC(=O)C=Cc3ccccc3C)=O)CCC(C1)C(O)C2O 43528,C(=O)(CC(C)(C)CNC(=O)CC1CCCCC1O)N(C)CC 43529,Cc1ccccc1CC(=O)N(C1CN(C(c2cnn(C3CC3)c2)=O)CC1F)C 43530,N1(C(C=CC=CC)=O)CC(CNC(=O)Cc2cc(C(F)(F)F)co2)OC2CCCC12 43531,C1(C)(CNC(C2C=CC(NC(C(C)n3cccc3)=O)C2)=O)NC(=O)NC1=O 43532,c1(C(=O)NC2CCN(C(C(CCCC)CC)=O)C2)ccnc2c1CC(=O)N2 43533,N1(C(c2c(C)occ2)=O)CCC(NC(c2cnc(OCF)cn2)=O)C(O)C1 43534,CC(C)C(O)CC(=O)NCC1CC(F)CN1C(=O)C=Cc1cc[nH]c1 43535,C1(C(=O)NCc2cnco2)(NC(=O)Cc2ccsc2)CCCCC1 43536,CC(C(=O)NC1CN(C(c2ncccc2N)=O)CCC1c1ccccc1)C(C)(C)C 43537,C(=O)(C(F)C(F)(F)F)N(CCC)CCNC(C1CCC1C(C)(C)C)=O 43538,C(=O)(C1CCc2ccc(C)cc21)N1CC2C(CNC(C3(NC(C)=O)CC3)=O)(C2)C1 43539,N1(C(CCSCCC)=O)CC(CNC(c2cc(OC)cnn2)=O)CC1C 43540,c1(C(=O)NCC(c2nccn2Cc2ccccc2)O)cccc(Cl)c1Br 43541,c1(C(=O)Nc2ncc(-c3cccc(C(F)(F)F)c3)s2)cc(Br)cnc1O 43542,C1(C(N2C(C(C)(C)NC(c3[nH]cc(CC)c3)=O)CCC2)=O)CCCN(C)C1 43543,Cn1c(C(N2CCC(C)(CNC(=O)C(O)C(F)F)CC2)=O)c(Cl)c2ccccc12 43544,CCC(CC)C(=O)N1C(CNC(c2cc(CC(C)C)nn2C)=O)CC2CC12 43545,c1(C(N2CC(CNCC(=C)CCNC(=O)OC(C)(C)C)C2)=O)cc(C)ccc1Cl 43546,Nc1cc2ccccc2cc1C(=O)NC1CCN(C(c2ccc(F)c(F)c2)=O)C1 43547,C1(NC(C2=C(C)OCCC2)=O)C2CC(CN(C(=O)C(F)=CCCF)C2)C1CO 43548,C1(C(N(C2CCN(C(=O)CCCc3cnn[nH]3)C2)CC)=O)CCN(C2COC2)C1 43549,C(=O)(C1=NNC(=O)C1)NCC(C)(C)NC(C1CN(C2CCOC2)C1)=O 43550,C1(C(=O)NCC(CNC(CCCOCC)=O)C)CCCC12OCCO2 43551,N1(C(CC=CC=C)=O)CC(C)CN(C(c2ccc3c(c2)COCO3)=O)C(C)C1 43552,c1(CNC2CC(C(=O)NCCC(F)(F)F)C2)ccc(F)c(F)c1Br 43553,C1(C(N(CC(C)(C)CO)C)=O)C(C2CC2)CCN1C(c1ncccc1Cl)=O 43554,Cc1nc(C)c(C(N2CCC(OCCNC(c3cccc(F)n3)=O)C2)=O)[nH]1 43555,C1(NC(C(CC=CC)CC)=O)CCCCCN(C(c2ncsc2CC)=O)C1 43556,Cc1nn(CC(=O)NCCCN(C)C(C2CCC(C3CC3)C2)=O)c(=O)n1C 43557,c1(CN(C(=O)C(F)n2ccnc2)CCNC(CSC)=O)ncnn1C 43558,C1(CCNC(C(C)SCCCC)=O)(OC)CN(C(C2(c3ccnn3C)CC2)=O)C1 43559,c1(NCCCc2n(C)ncn2)[nH]c(=NCCc2ncc[nH]2)nc2c1cnn2C 43560,Cc1c(C(=O)NC(CNC(=O)CCc2cccn2C)CO)noc1C1CC1 43561,CCCCC(C(=O)NCCN(C)C(C1(NC(C)=O)CCC1)=O)ON=C(C)C 43562,c1(NC(CC)C)cc(N(C)CCn2cccn2)nc(C(F)(F)F)n1.C1C(=O)N1 43563,Cc1oc(C(C)(C)C)cc1C(=O)NCCC(C)NC(=O)C(C)(F)c1ccccc1 43564,c1(C(C(=O)N(CCOCCCNC(CCSCC(C)C)=O)C)O)ccnn1C 43565,Cc1cc(C(=O)NC(C)(C(=O)NCCc2cc(C)ns2)C2CCC2)ccc1C#N 43566,c1(C(=O)NCC23N(C(c4cc(C)c(C)o4)=O)CC(C2)C3)cccc(C=C(F)F)c1 43567,C1(C(N2CC(NC(C(C)Cn3cccn3)=O)C2)=O)C2C3CCC(C3)C12 43568,C1(CNC(C(C=C)(C)CC)=O)CN(C(C2CC(=O)CO2)=O)CCC1(F)F 43569,c1(C(N(CC(CC)NC(CCC)=O)CC)=O)ccc(=NC(=O)OC(C)(C)C)[nH]n1 43570,C1(NC(=O)Cc2ccc(O)cn2)CN(C(=O)C2=CCCSC2)C2(CCCOC2)C1 43571,N1(CC#C)CCN(C(C2CCN(C(C3CCCCO3)=O)C23CC3)=O)CC1=O 43572,c1(CCNC2CC(C)N(c3ccccc3)C2)cc(O)nc(O)n1 43573,Cc1ccnc(CC(=O)NC(C2CCCN2C(=O)CCc2ncc(F)cn2)C)n1 43574,c1(C(=O)OC)ncc(-c2cccc(NC(C)=O)c2)cc1O.N12CCCC(C1)C2=O 43575,CC(C(=O)N1CCN(CCNC(C2CCCN(C(=O)C(N)=O)C2)=O)CC1)C(F)F 43576,N1(C(C=C(C)C(F)F)=O)CC(NC(c2ccncc2C(F)F)=O)CC(O)C1 43577,C1(C)(C(=O)NCC2N(C(c3c(CC)nc(C)o3)=O)CCOC2)CCC12CCC2 43578,N1(C(=O)NC)CCC(C(=O)NC(CNC(c2cccn2C)=O)CO)CC1 43579,c1(NC)cnc(C(N2CC(CNC(c3n[nH]cc3Br)=O)C(C(F)(F)F)C2)=O)cn1 43580,Cn1cnc2cccc(C(N3CC(O)CC3CNC(C3CC3CF)=O)=O)c12 43581,C=CC(C)(C)CCCNC(C1CC(NC(c2cc(C)c[nH]2)=O)C12CCC2)=O 43582,Cn1c(=O)n(CC(N2CC3(C2)CN(C(=O)C2CC2)CC3CO)=O)c2ccccc12 43583,c1(C(=O)OC(C)(C)C)cc(CCNS(=O)(=O)Cc2csc(C(F)F)n2)no1 43584,CC1(C(N2CC(C#N)C2)=O)CCN(C(=O)CSc2nc[nH]n2)C1 43585,Cc1ccccc1C1(C(=O)NC2C3CC2N(C(=O)COCCN(C)C)C3)CC1 43586,C12(C(=O)OC)CCC(C(N3CCC(C)C(NC(=O)C(C)SC)C3C)=O)(CC1)CC2 43587,N1(C(c2cnc(Cl)s2)=O)CCC2CCCC12CNC(C1(C2CC2)CCOCC1)=O 43588,C1(C(N(CC(CNC(c2c(C)nc(O)[nH]2)=O)(C)C)C)=O)CC2CCCCC2O1 43589,C1(C(C)C)C(=O)NCCN1C(C1C2CCC(C2)N1C(c1cc(C#N)cs1)=O)=O 43590,n1(CCC)cc(C(=O)NCC(C)(C)NC(c2n[nH]cc2Br)=O)nn1 43591,N1(C(C=CCCC(C)C)=O)CCCC(NC(c2ccc(CC(C)(C)C)cc2)=O)C1 43592,c1(C(=O)NC(C)C(C)(C)NC(C2(C3CCCO3)CC2)=O)cc2sc(Cl)cc2s1 43593,N1(CCC)CC(NC2(CNC(=O)OC(C)(C)C)CCCC2)CC1=O 43594,N1(CCNC(CCCC2C(C)C2)=O)CCN(CCNc2nccc(OC)n2)CC1 43595,C1(C(=O)NCCc2nc(CC)[nH]n2)CCN(C(=O)c2cccnn2)O1 43596,c1(CCCC)cc(=NC(=O)Cc2csc(NC(=O)N(C(C)(C)C)CC)n2)[nH]n1C 43597,CN1CC(C)(C)CC1C(N1CC(NC(=O)C2=C(Cl)CC2)C(O)C1)=O 43598,C1(C(=O)NCC(CC(=O)NC(C)C(C)C)OC)CC2(CCC2O)C1 43599,c1(CC(=O)NCC2(NC(Cc3cc(C)[nH]n3)=O)CCCC2)c(C)noc1C 43600,N1(C(CC=C)=O)CC(NC(C2(C(=O)OCC)CCCO2)=O)C(c2cnn(C)c2)C1 43601,C1(NC(=O)CCn2cc(Br)ccc2=O)CCOC12CCS(=O)(=O)CC2 43602,N1(C(Cc2c(OC)cccc2)=O)C(C)C2CC1C2NC(=O)CCn1cc(C)cn1 43603,CS(=O)(=O)CCC(=O)NCC12CCC(CC1)N2C(c1cncc(OC2CC2)c1)=O 43604,C1(CNC(c2c(Cl)nsc2Cl)=O)CC(F)(F)CN1C(C1CCCC12CC2)=O 43605,c1(C(N2CCN(C(Cn3nnc(C)n3)=O)C3(C2)CC3)=O)cccc2[nH]c(C)cc12 43606,N1(C(=O)Nc2c(C(=O)NC3CC3)cccn2)CCOCC1C1CCCOC1 43607,CCCC(C)(O)CC(=O)N1CCCCC(CNC(=O)CCNC(C2CCC2)=O)C1 43608,c1(OC)cccc(C(=O)NC2CC(CCNC(C3CCC(=O)NC3)=O)C2)n1 43609,Cc1ncc(C)c(N2CCC(NC(c3cc(=O)cc(Cl)[nH]3)=O)C(O)C2)n1 43610,c1(OC)ccc(Cl)c(F)c1C(=O)NC(C1CCOC1)CNC(c1occc1C)=O 43611,c1(OC)cc(C(N2CC(C(C)NC(c3occc3C)=O)C2)=O)cc(N)c1O 43612,c1(CC)nc(C(=O)N(C)CC2(NC(=O)CC3(CO)CC3)CC2)cs1 43613,Cc1occc1S(C)(=O)=NC(=O)CC1(C)CC1 43614,C(c1ccc([N+](=O)[O-])s1)=CC(=O)NC1CCN(C(C(C)(CO)OC)=O)C1 43615,C(=O)(CC(C(F)(F)F)NC(c1ccc2ccoc2c1)=O)NC(CCC)C1CCC1 43616,N1(C(COC2(C)CCC2)=O)CCC2(CCN(C(C3CCCO3)=O)C2)C1 43617,C1(NC(COc2cncc(C)n2)=O)CCC(C)N(C(=O)C=CBr)C1 43618,C1(CC(=O)NCCN(CCC)CC)CCCCC1NC(=O)CC1CSC1 43619,N1(C(CC2CC(=C)C2)=O)CCC(N2CC(O)C2)C1(C)C.N12CCC(C1)C2=O 43620,CN1CCC(C(N2CCC2C2CCCCC2)=O)(NC(C2CC3(CC3)CO2)=O)C1 43621,Cc1cc2sc(C(N3CC(F)(CNC(=O)C(C)n4ccnc4)C3)=O)cc2s1 43622,N1(C(C2(C#C)CN(C(c3ccc(C4CC4)o3)=O)C2)=O)CCC(C2CCC2)C1 43623,c1(C(N2CCC(C3N(C(c4cc(C)no4)=O)CCC3)C2)=O)cn(C)c(=O)nc1O 43624,c1(C(C)C)cccc(C(=O)N(CC(C)(C)NC(=O)C=CC2CCCC2)C)c1F 43625,c1(C(=O)NCCCCCN(C(CC2(CC)CC2)=O)C)c(C(C)C)cccc1F 43626,c1(C(N(C)CC2(NC(C3CCCC3c3nc[nH]n3)=O)CC2)=O)cccc(=O)n1C 43627,CS(=O)(=O)C(CNC(=O)CC1CCCOCC1)CNC(C1CC(F)(F)CS1)=O 43628,C1(NC(c2cc(C(C)=O)sc2)=O)C2CC1CN(C(=O)CCN1CCCS1(=O)=O)C2 43629,C(=O)(CC(C(C)(C)C)NC(=O)Cc1cncs1)NCC(CN(C)C)O 43630,Cc1cncc(C(=O)NCC2CCN(C(=O)Cn3ccc(=N)[nH]3)C2)c1 43631,C1(C(=O)OC)CCc2cc(OC)ccc2N1C(C1(C)CC1(F)Cl)=O 43632,c1(OCCC(=O)NC2CN(C(=O)C(O)CC3CCCCC3)C2)c(F)cccc1Cl 43633,N1(C(C(C)C)=O)CCN(C(=O)CSc2nc(-c3ccccc3)no2)C(CF)C1 43634,C(=O)(C(CNC(=O)C(C)c1ccsc1)CC(C)C)Nc1cc(CC)c(C)nc1 43635,C(=O)(C(C)(C)C(C)NC(c1c[nH]c(C)cc1=O)=O)Nc1c(OC)cccc1 43636,c1(C(N(CCNC(C2(CC=C)CC2)=O)C)=O)cccc2ncnc(O)c12 43637,N1(C(C2CCCN(C(CCCCC=CC)=O)C2C)=O)CC(C)CCCC1C 43638,C1(NC(c2c(C)noc2)=O)CCN(C(c2cn(C3CCCC3)nn2)=O)CC1(C)C 43639,CS(C)(=O)=NC(=O)C(=O)NC1CN(C(C2CCCN2C(C2CCCC2)=O)=O)C1 43640,c1(C(=O)NCC(C)N(C(C(C)=C2CC2)=O)C)ccc(-c2cc[nH]n2)cc1 43641,N1(c2cc(CN3CCC(COCC)CC3)nc(C)n2)C2CCC1CC(N(C)C)C2 43642,CC1CC2(CCN(C(=O)CCN3CCCC3=O)CC2)CN1C(C1CCC1(C)C)=O 43643,c1(OC)ccc(O)cc1C(=O)NCC1(NC(c2nnn(C)c2C)=O)CCOC1 43644,N1(C(COC(C)=O)=O)CCCC12CCN(C(=O)Cn1cc3ccccc3n1)C2 43645,C1(SC)CN(C(=O)CCSCc2ccccc2)CC1N1CCOCC1 43646,C1(C)(C(N(CCC(=O)NC2C(C)CCCC2)CCCO)=O)C(C)(C)C1(C)C 43647,CC(C)C(F)C(=O)NC1CCCN(C(c2cc(C3CCC3)[nH]n2)=O)C1 43648,C1(C(=O)NCc2cccc(OC(F)F)n2)CCc2nc[nH]c2C1 43649,C=C(C)C(C)(O)C(=O)NCCN(C(c1cc(Br)ccn1)=O)CC 43650,C12(C(=O)OC(C(=O)NCC)C)CCC(CC1)C2(C)C 43651,C1(CCOC)OCCC1Nc1ncc(I)s1 43652,c1(C(=O)NCC2CCN(C(C(CCC)O)=O)C2(C)C)ccc2cc(Cl)ccc2n1 43653,c1(C(=O)NC(C2CCCN(C(C3CCOC3)=O)C2)C)cnc2sccn12 43654,c1(CC)cnc(Cl)[nH]c1=NC(CNC(c1ccc(C)c(Cl)c1)=O)c1ccccc1 43655,C1(CNC(C(CC)N(C)C)=O)CCCN(C(C2(C3CCCO3)CCC2)=O)CC1 43656,N1(C(c2c(N)ccc(Cl)n2)=O)CCN(C(c2ccc3[nH]ccc3n2)=O)CC(O)C1 43657,CC1C(C(=O)N(C(C)(C)CC(N2CC3C=CC2CC3)=O)C)=NOC1C 43658,c1(CNCc2ncc(F)cn2)cnn2ccccc12 43659,C#CCCC(O)CCNC(=O)CC1CC1CNC(=O)C(CC)(CC)OC 43660,N1(C(c2nccc(CC)c2)=O)CC2CCC2(NC(c2cnc(C3CC3)s2)=O)C1 43661,N1(C(C2CC(OC)CN2C(=O)Cc2cccc(O)c2)=O)CC(F)(F)CC1CO 43662,C1(CC(=O)N(CCCCN(C(c2cc(C)sc2)=O)C)C)CCOC(C(C)C)C1 43663,c1(C2(NC(c3occc3F)=O)CCC2)cccc(F)n1 43664,C(=O)(C(O)CC(C)C)N1CC(NC(C(=C(C)C2CC2)F)=O)C(C)C1 43665,CCCC(CC)C(=O)N1CCN(C(=O)CCCOc2ccc(F)c(F)c2)C(C)C1 43666,C(N=c1[nH]c2c(c(=NCCCn3cnnn3)[nH]1)SCC2)C1CC(C)CC(C)C1 43667,C(CC(CC)C(=O)N1CC(NC(=O)C=Cc2cn(C)cn2)C2(CC2)C1)=CC 43668,Cc1ncc(C(N2CC(C)(NC(=O)CCC3CC(C)C3)C2)=O)cc1C#N 43669,c1(C(N2CCN(C(C3C(C(N)=O)C3)=O)CC2)=O)ccc2c(c1)COCC2 43670,c1(CC)csc(CC(=O)NC2(CCNC(c3cc(C(C)(C)C)on3)=O)CC2)n1 43671,c1(NC(C2CC(=C)CN2Cc2cc(C)ccn2)=O)cc(Cl)c(F)cc1C 43672,c1(C(C)C)ccc(C(=O)NCC(C)(C)NC2(C(F)(F)F)CCCC2)nc1C(F)F 43673,C1(NC(c2cc(OC)ncc2)=O)CCN(c2ccnc(C(F)(F)F)n2)CC1C 43674,C(C(C)C)(C(O)C(=O)N(C)CC1CN(C(=O)COC(C)C)CCO1)OC 43675,C1(CC(=O)NCC(C)(C)CNC(C2(CCCF)CC2)=O)CC(C)(C)CO1 43676,C(C(C(C)C)NC(c1cn(CCNC(c2ccc(Cl)s2)=O)nn1)=O)OC 43677,N1(C(CCC(=O)NC)=O)CCC2(CC1)CC2(C)C(=O)NC(C)C(C)(C)C 43678,Cc1cc(C(=O)NCC2CC(NC(=O)C(C3CCC(C)CC3)(C)C)C2)cc(N)c1 43679,C1(NC(=O)CCc2cnc[nH]2)CC12CCN(C(=O)C=CC=C(Cl)Cl)C2 43680,C1(NC(CCOCCOCC)=O)CCN(C(=O)C(C)(CC)CC)CC1F 43681,N1(C(=O)Nc2cccc(C)c2C)CC(C2CN(C(C3CC3(F)F)=O)C2)C1 43682,c1(CC)c(C(=O)Nc2cccc(-n3cc(CCC(C)O)nn3)c2)cnn1C 43683,CC1CCN(C(c2ccc(Cl)c(N)c2)=O)CC1NC(=O)Cn1nccn1 43684,C1(C(N(C2CN(C(C3CCCCCC3)=O)C2)C)=O)CN(S(N)(=O)=O)C1 43685,C1(NC2(c3nnnn3CCCSC)C(CC)CC2)CCCCC1(C)C 43686,c1(C(=O)NCC2(O)CCCN(C(C(CC)(C)OC)=O)C2)ccccc1P(C)(C)=O 43687,N1(C(C(COC)C)=O)CC(C)CCC1C(=O)N(CCCC(=O)OC)C 43688,C1(c2n(C(C)C)nc(-c3ccccc3C(F)F)n2)CCc2nnc(O)cc2C1 43689,c1(CNC(C(N2CCCCC2)C)=O)cccc(C(=O)N(C)Cc2cccnc2)n1 43690,N12CCCN(C(=O)CCc3ncco3)CC1COCC2=O.CC(C)(C)C=O 43691,C1(C)(C(N2C(CN(C)C(C3CCCN3C)=O)CCC2)=O)CCOCC1 43692,C1(CNC(CCC(=C)C)=O)CC2COCC2N1C(C1CC2CCCC12)=O 43693,c1(C(=O)NCC(CNC(c2c[nH]c(=NC)o2)=O)F)ccc2nccnc2c1 43694,c1(CC(=O)NC(CNC(C2N(CC)CCCC2)=O)(C)C)ccc(OC)c(Cl)c1 43695,C1(CCC)CN(C(c2cc(C)[nH]n2)=O)CC1C(=O)NCCn1cncn1 43696,c1(C(=O)NC(CNC(C2(COC)C=CCC2)=O)C)nccnc1-n1ccnc1 43697,C#Cc1ccc(CCC(=O)NCC(C)NC(=O)CN2CCOCC2)cc1 43698,N1(C(CC)=O)CC(C(=O)NC(CCC)C(=O)NC)C2(CCC2)C1 43699,c1(C(C)C(=O)NC2CC(n3cc(CO)nn3)C2)ccc(N(C)C)cc1 43700,C1(C2CCCN(C(=O)C(C#N)C(C)(C)C)C2)(NC(COC)=O)CC1 43701,C1(CNC(CN)=O)CCCN1CC1(C(F)(F)F)CCC1 43702,N1(C(C(CCC)OC)=O)CC2(CNC(=O)CC(F)(F)F)CCC1C2.c1ccccn1 43703,Cc1ccnc(C)c1NC(C1CC2CC2N1C(c1cc(Br)cnc1Br)=O)=O 43704,c1(C(C(=O)NCCC2N(C(C(F)=C(C)C)=O)CCSC2)C)c(C)nn(C)c1C 43705,O=C1CCC(C(N2CCC(CNC(=O)C(O)CCc3ccccc3)C2)=O)CCO1 43706,c12cc[nH]c1NC2=O.C(CC(=O)NCC(CC)N(C)C(C)=O)OCCC 43707,c1(C(=O)NC2(CNC(C3CCCCO3)=O)CC2)cc(F)cc([N+](=O)[O-])c1 43708,C#Cc1cncc(C(=O)NC2CCC2NC(=O)Cc2ccc(F)c(Cl)c2)c1 43709,c1(N2CC(C)CC(OC)C2)ccc(S(=O)(=O)CCC(N2CCCCC2)=O)cn1 43710,n1(CC(=O)NCC(C)(C)CNC(=O)C(C)(C)CF)ccc2cc(F)ccc12 43711,C(c1ccc(F)c(Cl)c1)=CC(N1CC(NC(C2CN(OC)C(=O)C2)=O)C(O)C1)=O 43712,c1(C(=O)NC2C(CNC(C(n3cc(C)nc3)(C)C)=O)C2)cc2nc[nH]c2cn1 43713,Cc1ccc(C(=O)NCC2CC(F)(CNC(C3(C(C)(C)C)CCCC3)=O)C2)nc1 43714,c1(NC(C2CN(C(CNC(=O)OCC)=O)CC2F)=O)cc(Cl)cnc1C 43715,N1(C(CC2C(C)(C)CC2)=O)CC2(CCOCC2)CC1CNC(c1csc(S)n1)=O 43716,c1(C(N(CC(CNC(C2=C(C)OCC2)=O)(C)C)C)=O)cc(=O)c2ccccc2o1 43717,C1(C(=O)NC2CC(C(N(CC#C)CC3CCCO3)=O)C2)CC1C1(C)COC1 43718,c1(CC)cnccc1C(N1CCCC1C(=O)OC)C(=O)NC(C)CC 43719,C(=O)(CCCCC(F)F)NC1(C)CCCN(C(c2cccc(CCC)c2)=O)C1 43720,c1(CC(=O)N(CC(O)CN(C)C(C2CC2C(C)(F)F)=O)C)ccnn1C 43721,C(=O)(CCN=c1[nH]ccs1)NCC(CN(C(C1COCCC1(F)F)=O)CC)(C)C 43722,c1(C(=O)NCC(CNC(=O)CC2CCCC2O)CO)nccc2ccncc12 43723,N1(C(CNC(CC)=O)=O)CCN2CCN(C(=O)CC3CCCC(=O)N3)CC2C1 43724,C=CCC(C)(C(=O)NC1CC(NC(=O)CCc2cc(C)n(C)n2)C1)N(C)C 43725,C(=O)(C(CC(C)C)NC(c1ccc(C)n1C)=O)N1CCC(C(=O)NC)C1C 43726,C(CC(C)(C)C(=O)NCC1COCCN1C(=O)C=CC(=O)NC1CC1)OC 43727,C1(NC(C(CC=CCC)C)=O)CC2CCC(C1F)N2C(=O)C(C)(C)F 43728,C(=O)(C(C)S(C)(=O)=O)N1CCC(N(CC#C)C(c2cccs2)=O)C1 43729,C1(CCNC(C(C)n2cnnn2)=O)CCCN(C(c2cnoc2)=O)CC1 43730,c1(C(=O)NC2C(NC(CCOC(C)C)=O)CC2)cnc(Cl)c(N)c1 43731,C1(NC(CCCCC=CC)=O)CN(C(C2CC=CCO2)=O)CC2(CC2)C1 43732,C1(C(=O)NCCNC(CC2C(C)(C)C2)=O)CC=CC(O)C1 43733,N1(C(CC(=O)NCC)=O)CC2C(C(=O)NCc3[nH]nnc3C)C2C1 43734,C(CCC(O)C(=O)NCCCCn1ccnc1)NC(=O)CN1CC2CC2C1 43735,c1(C(=O)NC(CC)CNC(c2cnc(C)n2C)=O)cc2ccc(F)cc2nc1O 43736,c1(CNC(C(C(C)C)O)=O)nc(CNC(C2CCC(C)(C)C2)=O)cc(O)n1 43737,C1(CC)CCN(C(=O)C(C)=CC(C)(C)C)C1C(N1CC(OC(=O)N(C)C)C1)=O 43738,c1(C(CNC(C2(COC)CCOC2)=O)NC(c2cnnn2C)=O)ccccc1F 43739,c1(OC)ccc(CNC2CCC(C(=O)O)C2)c(O)c1 43740,CON=Cc1ccc(C(=O)NC2CCC(NC(=O)CC#N)C2)cc1.CC 43741,N1(C(C(c2cccnc2)N(C)C)=O)CCCCC1CNC(=O)CCNC(=O)CO 43742,Cc1cc2cc(C3=CCN(C(=O)CNC(=O)C(F)F)CC3)ccc2s1 43743,O=C(C(F)C(F)(F)F)NCC1CCCCC1C(=O)NCC1CC2CCC1O2 43744,C1(NC(c2ccc(CNC(C3C(C)C3C)=O)cc2)=O)CCC(=O)NC1C 43745,c1(-c2cn(CC3C(NC(c4ccc(SC)s4)=O)CCC3)nn2)c(C)cccc1C 43746,N1(C(c2cn(CC)nn2)=O)CC2CCCN(C(C3CC(OC)C(OC)C3)=O)C2C1 43747,C#CCCCC(C)C(=O)NC(c1nccs1)CC 43748,C1(NC(c2n(CCC)nc(C)c2)=O)CC2CN(C(=O)CCC(C)(C)F)CC2C1 43749,S(=O)(=O)(c1cc(C)c(Br)cc1F)NC(C(CCC)OCC)=O 43750,C1(NC(C2CCN(C(CC(C)(F)F)=O)CC2)=O)CCCCCC1O 43751,N1(CC(=O)NC(CC)C(C2CC2)C2CC2)CCC(N2CCC(C)(O)C2)CC1 43752,c1(C(=O)NC23CC(CNC(CCCSC)=O)(OCC2)C3)ccn2cnnc2c1 43753,N1(C(C2(C(=O)NC)CC2)=O)CCC(C2CC2)C1CNC(=O)CCCC(C)O 43754,C(=O)(CCCCCNC(C1COCCC1c1ccccc1)=O)NC 43755,C(c1cc(F)cc(F)c1)=CC(=O)NCC(C(C)C)NC(C(C1CC1)SC)=O 43756,N1(C(c2ccn(CCC)n2)=O)CCC2(CCN(C(c3cc(N)ccc3C)=O)C2)C1 43757,c1(-c2ccc(OC)cc2)c(C(=O)Nc2cccc3ccnn23)nc2ccccn12 43758,c1(NC2(CNC(CSc3c(C)cccc3)=O)CCCC2)c(Cl)cccc1[N+](=O)[O-] 43759,N1(C(CCC2CC(NC(c3c(C)n(C)nn3)=O)C2)=O)CCC(N(C)C)C(C)C1 43760,C(=O)(C(F)(F)CN)NCC(Cc1ccccc1)OCC 43761,c1(C(=O)NCC(C)(C)NC(C(CC)C(C)O)=O)ccc2c(O)nc(=O)n(C)c2n1 43762,c1(C(NOCC(=O)N(C)CC2CC(=C)C2)=O)ccc(F)cc1C 43763,c1(OC)ccc2c(c1)CC1(CCN(C(=O)NCc3ncc(C)o3)CC1)C2=O 43764,C1(CNC(C(C=CCCC)O)=O)(NC(c2cc(O)no2)=O)CCCCC1C 43765,N1(C(c2c(CC)cnn2C)C(=O)NCc2ccccc2)CC(COC)C2(CC2)C1 43766,N1(C(C(CNC(C(C(C)C)OC)=O)(C)C)=O)CC(=O)N2CCCC2C1 43767,C(=O)(CC(CNC(=O)C(n1ccc(C)n1)C)C1CCC1)NC(C#C)(C)C 43768,C=CCC(CNC(=O)C(=O)C1CC1)CC(C)C(C)(C)C 43769,Cc1ccc(O)cc1C(N1CCN(C(=O)Cc2ccon2)C(C)C1)=O 43770,CC1(C)CCN(C(=O)C(=O)NCCC(N)=O)CC1CNC(=O)CNC(=O)C1CC1 43771,C=CCCCCC(=O)N1CCC(CF)(NC(c2cnccc2Cl)=O)C1 43772,C1(CC(=O)N(CC(=O)NCC)CC)CN(C(=O)CC2CCCN(C)C2)CC1C 43773,c1(C(N2CC(CNC(CC=CCC)=O)C(F)(F)C2)=O)cccc2nc(Cl)cn12 43774,S(=O)(=O)(c1ccc(C(C)NC(c2ccc(-n3ccnc3)nc2)=O)cc1)NCC 43775,N1(C(c2cnc(CC)o2)=O)C(CC(=O)NC2C=CCCC2)C2CCCC12 43776,c1(C(C)=O)ccccc1C(=O)NCC1(CNC(=O)Cc2csnn2)CCC1 43777,c1(C(N2CC(NC(CS(=O)(=O)NCC)=O)(CO)C2)=O)ccc2c(c1)ncn2C 43778,c1(C(CNC(=O)NCc2c(C)nc(CC)o2)(C)C)cccc(Br)c1F 43779,c1(OC)nc(C(=O)NCC(N2CCN(C(c3cc[nH]c3C)=O)CC2)C)ncc1F 43780,C1(O)(CNC(CC=C=C)=O)CCN(C(=O)CC2(C)CCOCC2)C1 43781,C1(O)(C(=O)NCCN(C(=O)C(c2cccc(C(F)(F)F)c2)(C)C)CC)CC(F)(F)C1 43782,N1(C(CC#N)=O)CC(CNC(c2cc(Cl)c(C(F)F)cc2F)=O)OC2CCCC12 43783,N#Cc1ccc(F)c(C(N2CCC3CC3(NC(c3csnc3Cl)=O)CC2)=O)c1 43784,CC1CCN(CCn2ccc(C(F)(F)F)n2)CC1 43785,c1(C(=O)NC2(CNC(=O)CC3(C(F)F)CC3)CCOC2)cc(O)cc(Cl)c1 43786,c1(CC(=O)NC2CC(C)(NC(c3ccsc3Br)=O)C2)nc2ncccn2n1 43787,C1(CNC(COC(CC)(C)C)=O)CCCC1NC(=O)C=Cc1cncs1 43788,CC1CN(C(c2cncn(C)c2=O)=O)CCC1NC(c1cc(C2CCC2)[nH]n1)=O 43789,c1(OCC)nccc(C)c1NC(=O)CCC(C)NC(C1C=CCCC1)=O 43790,c1(C(N2CCC(Cc3ccn(C)n3)C2)C(=O)NCC)cccc2ccsc12 43791,C(CC(C)C(=O)N(C(C)CNC(C1(C)SCCCS1)=O)C)=CC 43792,C1(NC(C2CC(CCC)C2)=O)CCC2(CC1)CCN(C(c1cccnc1O)=O)C2 43793,c1(C(=O)NCC2(COC)CN(C(C3CCN3C)=O)C2)ccc(C)cc1C 43794,C(=O)(CC(C)C(F)F)N1CCCC(NC(c2nc(COC)sc2)=O)C1 43795,c1(CC(C)C)cc(C(=O)NC2CN(C(c3ccc(C4CC4)o3)=O)C3CC23)n(C)n1 43796,c1(C(N2C(C)(C(=O)NCc3ccc(O)c(O)c3)CCC2)=O)ccc2nn[nH]c2c1 43797,Cc1cccc2[nH]cc(C(=O)NCCC3(O)CN(C(=O)CCC4CC4(Cl)Cl)C3)c12 43798,N12CC3CC3(C1)C2=O.C(c1ccoc1)=CC(=O)NCCC(=O)NC(C)(C)C 43799,c1(N(C(CC)C(=O)NCC(=O)OC)C)nc(C(=O)OC)nc2ccccc12 43800,c1(CNC2CCN(C(c3c(C)n[nH]c3)=O)CC2F)c(F)cc(Br)cc1F 43801,C(CCO)(C(=O)O)Sc1ccc(C(=O)NCCCn2ccnc2)cc1 43802,n1(CC)cnc2c(NCC3CCCN(C(C)C)C3)nc(NC3CCN(C)C3)nc12 43803,C#CCCCC(C)C(=O)N1CC(C(N)=O)(CNC(c2ccc(Cl)c(F)c2)=O)C1 43804,Cc1cc(C(N2CCC(CN(C)C(C3CCN(C)C3)=O)C2)=O)cnc1C(F)(F)F 43805,C12(CC(=O)NC3CCCC(NC(C4CCC45CCC5)=O)C3)COC(CF)(C1)C2 43806,Cc1cc(Cl)c(C(=O)NCC2C=CCN2C(=O)CNS(C)(=O)=O)s1 43807,CC(N=c1ccnc(C2CCC2)[nH]1)C1CC(NC(c2cccc3nc[nH]c23)=O)C1 43808,CC1=NN(C)C(=O)C1CC(=O)N(C)CC1CN(C(c2ccnc(S)c2)=O)CCO1 43809,c1(C(N(C2CCN(C(=O)C(C)CCOC)CC2)CC)=O)cc(C)ccn1 43810,c1(C(C)NC(C(C)CN(C(=O)CCCC2CCCO2)C)=O)nccc(O)n1 43811,c1(C(N2CCC(COC)(NC(C3CC=CCC3)=O)C2)=O)ccc(OC)c(Cl)n1 43812,c1(CC(=O)NCC(CO)NC(C(CN(C)C)O)=O)ccccc1SCC#N 43813,N1(C(c2ncc(C)cc2F)=O)CC2CCC(N(C)C(c3occc3C)=O)C2C1 43814,C1(CNC(C2(OC)CCCCC2)=O)CC(C)(C)CN1C(c1scnc1Cl)=O 43815,C(=O)(CCS(C)=O)NC(c1ccccc1)CNC(C1C(OC(C)=O)C1)=O 43816,C1(NC(C2(NC(C(COC)C)=O)CC2(C)C)=O)CNC(=O)C1(C)C 43817,C(CCCCC(=O)N(C)CCOCCNC(C1CCC(C2CC2)C1)=O)SC 43818,c1(OCC)ccc(C)c(C(=O)NCC2CC2NC(c2nc(C3CC3)oc2C)=O)n1 43819,C(=O)(CC(C(F)F)c1cccc(F)c1)N(CC(C)N(C(C=C(C)Cl)=O)C)C 43820,CC1(C)C(CNC(=O)NCC2(c3nn[nH]n3)CC2)CC1O 43821,c1(NC(=O)NC2CCC(CC)CC2)cccc2c(OC)ccnc12 43822,N1(C(C(C(C)C)OCC)=O)CC2CCC1C(NC(=O)Cc1n[nH]c(C)n1)C2 43823,N1(C(c2c(C(C)C)onc2)=O)CCC2(CC(C(=O)NCCN(C)C)C2)C1 43824,C1(OCC(N2C(C3(NC(c4cc(F)c[nH]4)=O)CC3)CCC2)=O)CCCCCC1 43825,C1(NC(Cn2nnc(=N)[nH]2)=O)CCCCCN(C(C23CCN(CC2)CC3)=O)C1 43826,c1(OC)c(C(=O)NC2CC(NC(=O)C(C(C)C)OCC(C)C)C2)cc(Cl)cc1C 43827,N1(C(C2CC=C(C)CC2)=O)C2CCC1CC(NC(C13CC(C1)S(=O)(=O)C3)=O)C2 43828,c1(-c2n(C3CC(C)OC3C)ccn2)cc(F)c(O)c(F)c1 43829,CC1CN(C(=O)C(C)(CO)NC(=O)Cc2cn[nH]c2)CC(C)(C)O1 43830,C12(NCc3cc(OC)c(C)cc3)CCCC1CN(C(=O)CN1C(=O)CCC1=O)C2 43831,c1(NC(CN2CC(C)C2)=O)ccnc2c1cnn2C.C12CN(C1)C(=O)CO2 43832,N12CC3CC(C3C1)CN(C)C(CC)C(=O)N1CCCC1(C)C2=O.N(C)(C)CC 43833,N1(C(=O)Cc2cc(F)cc(Cl)c2)CCC2OCCN(C(=O)C=CCF)C2C1 43834,C1(C2CC2)(CNC(C2N(C(C)=O)CC(O)C2)=O)CCN(C(C2(C(N)=O)CC2)=O)C1 43835,C1(N(C(c2n(CC)ncn2)=O)C)CCN(C(=O)CCCOC(C)=O)CC1 43836,c1(C(N(CC(CNC(C2C(CCOC)C2)=O)(C)C)C)=O)cc(C(C)C)nn1C 43837,C1(C(=O)NC2CCCC(CNC(c3c(CC)c[nH]c3)=O)C2)OCCOC1(C)C 43838,CS(=N)(=O)CCNC(=O)C(Cc1cc[nH]n1)NC(=O)CC1CCCC1 43839,N1(C(C(C=C)O)=O)C2CCC1CN(C(c1sc(Cl)cc1Cl)=O)C2 43840,CC1CN(C(c2cc(O)nc(N(C)C)n2)=O)CCC1NC(C1CN(C(N)=O)C1)=O 43841,C(=O)(C(CCC)OCC)N1CCC(C(N2CC(CCC#C)C2)=O)C1 43842,C#CCC(C(=O)NCCCOC1CCC1)NC(C1CC=CCC1)=O 43843,C1(CC(=O)NC2C(NC(CSCC=C)=O)C2)OCCCC1(C)C 43844,c1(C(N2CCC(NC(C(C(C)O)C)=O)(CF)C2)=O)nc2cncnc2nc1O 43845,N1(C(C)=O)CC2CC1CN2C(C12CC1CCN2C(=O)C(N1CCCCC1)C)=O 43846,C1(C(=O)NCC#CCNC(c2cc(C)n(C)c2)=O)CC(c2cccc(F)c2)=NO1 43847,c1(C(N2CCC(CN(C)C(C3CC3CF)=O)C2)=O)cccc2nccn12 43848,c1(CC)ccc(C(=O)NCCC(O)CNC(c2cnc(O)cc2OC)=O)c(Cl)c1 43849,c1(C(=O)NC(c2ccccc2)CCC)ccc(N2CCC(N)CC2)cc1 43850,O(NC(=O)C(C)(C)S(C)(=O)=O)C(CC(C)C)C(=O)N1CCC(C(C)C#N)CC1 43851,n1(CC(=O)NCC2C(C(N3CC(OC(=O)OC)C3)=O)CC2)cnnc1O 43852,c1(OC)ccc(NC(=O)NC2CC2c2ccncc2)cc1Br 43853,N1(C(C)=O)CCCC2(CCN(C(=O)CNc3ncnc4[nH]cnc34)C2)C1 43854,C1(C(N(CC#C)C)=O)CC12CCN(C(=O)CN1CC(C)(C)C1)C2 43855,C(c1cccnc1)=C(C)C(=O)NC1C=CCCC1C(=O)NC12CC(C1)C2 43856,C1(NC(c2ccc[nH]2)=O)CN(C(C23CCC(CC2(F)F)C3)=O)Cc2nccn2C1 43857,CCCCCC(F)C(=O)N(CC(N1CC(O)CC1COC)=O)CC1CC1 43858,N1(C(C(C)C)=O)CC(n2cc(C(C)N(C(=O)OC(C)(C)C)C3CC3)nn2)CO1 43859,c1(CCC(=O)NC2C(NC(c3ccc(C)nc3)=O)CC2)ccc2ccn(C)c2c1 43860,C1(F)(CNC(C2C(CC(C)(C)C)C2)=O)CCN(C(=O)CS(N)(=O)=O)C1 43861,CC(C)(F)C(C)(F)C(=O)N1CC(NC(c2csc(Cl)n2)=O)C(CC(C)(C)C)C1 43862,Cc1nn(CC(N2CCC(C(O)CNC(c3ccoc3)=O)CC2)=O)cc1Cl 43863,N1(C(C=CC)=O)CCC2(CC1)CN(C(=O)C(C)n1cccn1)CC2CO 43864,c1(C(N2CCC(CNC(C3C(=C)C3)=O)CC2C)=O)ccc2nnc(O)n2c1 43865,C1(CNC(C2(C)CC(C)C2)=O)CN(C(c2ncc(F)cc2N)=O)CC(C)(C)C1 43866,C(=O)(C#CC1CC1)NC(CC)C(=O)NC1CC=CCC1 43867,C(=O)(C(S(C)(=O)=O)C1CC1)NCC(C)CNC(C1(C)CCSCC1)=O 43868,CC1COC2(CCC2)CN1C(C1CCN(C(c2cn3c(n2)CCC3)=O)CC1C)=O 43869,N1(C(=O)C=Cc2ccsc2)CCC2(C1)CN(C(=O)C(F)F)CCO2 43870,C(=O)(C(CC(C)C)NC(=O)OC)NCC(C1(OC)CCOCC1)(F)F 43871,C1(C(N2CC(CC(=O)NCCc3cc(C)n(C)n3)OCC2)=O)CN2CCN1CC2 43872,c1(C(N2C(C(=O)NCc3ccc(C(C)C)cc3)C(O)CC2)=O)ccc(Br)c(Cl)n1 43873,CCCC(C(=O)NC(C)(C)CNC(c1cccc(COC)c1)=O)S(N)(=O)=O 43874,c1(COC)nnc2cc(N3CCC(C4CCCN4C(=O)C(C)C(C)O)C3)ncn12 43875,C1(O)(CNC(c2ccc(OC)cc2C)=O)CC2CCC(C1)N2C(c1cnsn1)=O 43876,c1(C(C(=O)OCC2CCC(F)(F)C2)OC)cccc(CC(F)(F)F)c1 43877,C(=O)(C1=CC2CCC1C2)N(CCN(C)C(c1ccc(Br)cc1O)=O)C 43878,c1(CNCC(O)C(F)(F)F)c(O)ccc(F)c1F 43879,CCC(=O)CCC(=O)N1CCOCC(CNC(c2sccc2OCC)=O)C1 43880,Cn1cncc(C(=O)NCC2(NC(=O)C(O)CN3CCCC3)CCOCC2)c1=O 43881,C1(C(=O)NCCCCCn2cc(C(CC(C)C)O)nn2)CCN(C)C(=O)C1 43882,N1(c2cc(NCC(CC)N(C)C)ncn2)CCc2c(F)cc(F)cc2C1 43883,C1(C)(NC(CCCNC(C)=O)=O)CCC(NC(C2(O)CCSCC2)=O)CC1 43884,C(=O)(C1CC(=O)c2ccccc21)N1CC(N(C(=O)C2=CCOC2)C)C(O)C1 43885,CN1CCC(NC(C2N(C(=O)Cc3cncn3C)CCC2(C)C)=O)C(C#N)C1 43886,CCC(C)C(C(=O)NC1CCN(C)CC1C)N(C(=O)CCC1CCC1)C 43887,Cc1ccc(C)c2[nH]c(C(=O)NC3CC3CNC(C3CC(C)(C)C3)=O)cc12 43888,c1(C(=O)NCCCCNC(=O)CCc2cncnc2)c(Cl)ccc2c1OCO2 43889,C1(C(=O)NCCC2(NC(CC=C)=O)CCC2)CCCN(C(=O)NC2CC2)C1 43890,c1(C(=O)NC2(CC=C)CN(C(=O)C=CCC)C2)cc2c(s1)COCC2 43891,C1(C)(C(=O)OC)CC(C(=O)N(CC(O)CN(C)C(c2coc(Cl)c2)=O)C)C1 43892,c1(C(N2CC(N(C)C(C3(c4cccs4)CCC3)=O)C2)=O)cnn(C)c1N 43893,C1(CNC(C2C(C)=CCS2)=O)CN(C)CCN1C(=O)C1=CC(C)C1 43894,c1(OC)ccc(CN(C)CC2CCCN(C(C3CC(C)(C)C3)=O)C2)cc1C 43895,C1(C)(CC)CC(C(=O)NC(c2cccnc2)c2ccccn2)CCO1 43896,CCCCCC(F)C(=O)NCC(C1CCCCCC1)NC(c1cncn1C)=O 43897,c1(C(=O)NCc2cccc(CNC(C=CSC)=O)c2)ccc(C(C)(F)F)nc1O 43898,C1(C(=O)NCCC2(C)CCN(C(c3ccc(C)nn3)=O)C2)CCCC(C)(C)C1 43899,c1(C(=O)NC2C(CC)CN(C(c3cccnn3)=O)CC2)cccc2nccn12 43900,c1(C(=O)NCC)ccnnc1.C1(C(N2CC(n3cnnc3)C2)=O)(CO)CCC1 43901,c1(C(=O)NCCCN(C(c2ccc(N)cn2)=O)CC)cc2c(OC)cccc2[nH]1 43902,C1(O)(CS(=O)(=O)NC(C(C(C)C)NCCOC2CCCC2)=O)CCCCCC1 43903,c1(C(=O)OCC)cnc(N2CCS(=O)C(C)C2)cc1C 43904,C1(NC(C=CC(C)C)=O)CC(NC(=O)Cc2ccccc2)CC1O 43905,N1(C(CNC(CCC(C)C)=O)=O)CCC2(NC(=O)CC(=O)N(C)C)CC2C1 43906,C1(OC)CC(CCNC(c2nnc(C)s2)=O)N(C(C2CCCS2)=O)C1 43907,C1(n2c(C)ncc2)CCCN1N1CCCC1(C)Cc1cccc(Br)c1 43908,N1(CC(=O)N(C(CCNC(Cc2nnc(C)o2)=O)C)C)CCC(C(N)=O)CC1 43909,c1(OCCNC(=O)CN2CCCC2CF)cncc(Br)c1 43910,CC(C(=O)NC1(C(=O)NC2(CC3CC3)CC2)CSC1)S(N)(=O)=O 43911,c1(C(N(C2CC3CC2CN3)c2c(OC)csc2)=O)n[nH]c2ccc(Cl)cc12 43912,Cc1cnc2cccc(C(N3CC(NC(=O)C4=CCSC4)C(C)(C)C3)=O)n12 43913,C1(CN(C(=O)Cc2ncc(Cl)s2)C)COCCN1C(C1CC(=O)N(C2CC2)C1)=O 43914,C(=O)(C(C)(CO)CO)N1CCCC(C(=O)Nc2c(C(C)=O)cccn2)C1 43915,c1(C(=O)NC(C)CCNC(=O)CC(C)N(C)C)ccc2nccnc2n1 43916,C(CCO)(CC(C)C)N(C(C(c1c(C)cccc1Br)NC(CC(C)SC)=O)=O)CC 43917,Cc1ccc(C2(C(=O)NC3CC3NC(C3(C)COC3)=O)CC2)c2ccccc12 43918,C1(NCC2CC(OCC)C2)CCS(=O)(=O)C(C)(C)C1 43919,N1(C(COCC(=C)C)=O)CC(NC(C2CC(n3ccnn3)C2)=O)CCC1C 43920,N1(S(CC(=O)OCC)(=O)=O)CCC(O)(CN2CCCCC(N3CCCC3)C2)CC1 43921,c1(C(N2CCC(CNC(C=CC=CCC)=O)C(C)C2)=O)cc2c(cn1)CCCC2 43922,O=S(=O)(c1cnccc1N1CCCC(CCF)C1)NCC1(CC2CC2)CC1 43923,C1(F)(C(=O)NCC(C(C)C)OC)CCN(C(c2cscc2OC)=O)C1 43924,C1(c2n(C)cnc2)COCCN1C(=O)CCC1CCCCO1 43925,c1(C(N2CCN(CC3CN(C(C4C(C#C)C4)=O)C3)CC2)=O)cc(C)cc(C)c1N 43926,CC(CC(=O)NCC1CC12CC2(F)F)C(C)(C)NC(C12CC(F)(C1)C2)=O 43927,c1(C(=O)NCC(C)(C)NC(=O)Cc2ccoc2)ccc(-c2ccccc2)s1 43928,N1(C(c2cc(C(C)C)[nH]n2)=O)CCCCCCC1C(N1CCCC(N=[N+]=[N-])C1)=O 43929,c1(NC(C2C3CN(C(c4cc5cccnn5n4)=O)CC23)=O)ccc2nonc2c1 43930,c1(C(C)=O)ccc(C(=O)NCC2(CN3CCN(C)CC3)CC(F)(F)C2)cc1Cl 43931,CC1(C)C(CC(=O)NC2CCC(NC(c3coc(Cl)c3)=O)CC2)CC1O 43932,Cn1cc(S(=O)(=O)CCNC(=O)Cc2ccn(C)c2)cn1 43933,C(C(C)(C)C#CC(=O)NCC(c1cnc[nH]1)C)NC(CN1C(C)CCCC1)=O 43934,C=C(C)C1OCCC1C(N1CC(C(C)NC(=O)Cc2cnc(C)s2)C1)=O 43935,C1(C#CC(=O)NCC2CC2CNC(=O)CCCCN(C)C)(CC)CC1 43936,C1(C(=O)NCC(S(C)(=O)=O)CNC(C2CCCCC2O)=O)OCC2COCCC12 43937,C=CCCCC(C)(C)CN=c1[nH]c2c(c(=NCC3CC4(CC4)C3)[nH]1)CCCCC2 43938,C(=O)(C(F)C(=O)NCCNC(C1CSCN1C(=O)OC(C)(C)C)=O)OCC 43939,N(C(=NCCOCC)N1CCC2(CCCCCC2)C1)C(C#C)CC 43940,C1(NC(C2C(C(C)NC(=O)CCc3ccc[nH]3)C2)=O)CCCC(O)CC1 43941,c1(C(=O)NC2CN(C(COCCC)=O)C(C)(COCC)C2)n[nH]c(C)c1[N+](=O)[O-] 43942,c1(C(N(CC(=O)NC2CC2C(C)(C)C)C(C)C)=O)cnns1 43943,C(C(F)(C(=O)NCc1ccnc(Cl)c1)C(C)C)NC(c1c(C(C)C)c[nH]c1)=O 43944,C1(O)(C(C)CNC(=O)COC(F)F)CCN(C(c2c(Br)ncn2C)=O)C1 43945,Cc1cc(C(=O)NCC(C(C)(C)C)NC(c2cccc[n+]2[O-])=O)ccn1 43946,C(=O)(C1CCCc2c1ncn2C)N1CC(NC(c2c(C(C)C)occ2)=O)C(O)C1 43947,C1(C(N(CCN(C)C)CC)=O)C=CCN(C(=O)C(CSC)OC)C1 43948,C1(C(N2CCCC(C(F)F)C2)C(=O)NC(C(=O)OC)C)CCCOCC1 43949,N1(C(C)=O)CC(C)CN(C(=O)CCNC(C2(CC=C)CCCC2)(C)C)C(C)C1 43950,c1(CN2C(C(=O)NC(C3CCCCC3)CC)C(O)CC2)ccccc1[N+](=O)[O-] 43951,Cc1nscc1CC(=O)NC1(CCCC(=O)NC2CC(OC(F)F)C2)CCC1 43952,c1(C(N2CCN(C(c3ccn(COC)n3)=O)C3C2C3)=O)cn2c(C)cccc2n1 43953,C1(C(=O)NC2CC(CNC(CSC)=O)C2)CSc2ccccc2O1 43954,c1(C(=O)NC2(CNC(C(CC)(C)F)=O)CCCC2)ccc(Cl)cc1Cl 43955,c1(N2CCC(CCOC)(OC)C2)nc(Cl)nc(-c2ccccc2)c1C 43956,N1(C(C(C)CC#N)=O)CC2CCC(CN=c3nc[nH]s3)(C2)C1 43957,C1(c2cn(CCN(C(=O)CCC3CC4(CCC4)C3)C)nn2)CC2CCC1C2 43958,Cc1cccc(C(=O)NCC2CCC2C(=O)NC(C)(C)CNC(N)=O)c1 43959,C1(N(C(C=CC(=O)N(CC(C)NN(C)C)C)=O)C)CCCC1C 43960,CCC(C(=O)N(CCOC(c1cccs1)=O)Cc1cnccn1)Oc1ccccc1 43961,C1(CNC(C2(C)CC2(F)Cl)=O)C2CN(C(c3ccn(C4CC4(F)F)n3)=O)CC12 43962,C=Cc1ccc(C(N2CCCC(C)(CNC(c3c(Cl)noc3C)=O)C2)=O)cc1 43963,CC1(C)C2CC(C(N3CC(C(C)(C)O)(CNC(C4CCS(=O)CC4)=O)C3)=O)CC12 43964,CCC(C)C(=O)NCC(N1CCCC1C(=O)NCc1ccn(C2CCC2)n1)=O 43965,c1(C(=O)NC(CNC(c2c[nH]nc2C2CC2)=O)CO)cc(F)c(F)c(O)c1F 43966,CC(CNC(C1(F)CCC1)=O)C(F)C(=O)N(C)CCN1CCOCC1 43967,c1(N(C(C(C)Oc2ccccn2)=O)CC2CNCC2(F)F)ccnc(S(C)(=O)=O)n1 43968,C1(CNC(CCC=C)=O)CN(C(=O)C(CCC)OCC)CCCO1 43969,c1(C(=O)NCC2CN(C(c3c(C)coc3)=O)C(C)(C)C2)cc(P(C)(C)=O)cs1 43970,C(C(N=c1cnc(OC)c[nH]1)c1cc(C)cc(C)c1)OC 43971,N12CCC(C3CC3)C1CCn1cnnc1CCCCCC2=O.C1(SC)CC2(CCC2)C1 43972,C(C(CC(C)C)C(=O)NCCOC1CN(C(C2(OC(C)C)CCOC2)=O)C1)OC 43973,CS(=O)C1(CNC(=O)NCC2CNC(=O)C2)CCC1 43974,c1(C2CN(C(=O)NCc3nccc(C(F)(F)F)n3)C2)ccccc1Br 43975,C1(CC(=O)NCC(CC)N(C)C(c2cccc(CCO)c2)=O)CCCC(=O)C1 43976,c1(C(=O)NCC(CNC(c2n(C(C)C)cnc2)=O)O)ncc(F)cc1F 43977,C1(C(=O)NC2CC2NC(=O)C(F)(F)C2CCOCC2)(OC)CCSCC1 43978,c1(C(N(C2CCC(O)CC2)C(c2ccnnc2S)=O)=O)c(F)cccc1F 43979,c1(CC(=O)NC2CCN(C(COCCC)=O)C2)ccccc1CS(N)(=O)=O 43980,Cc1cc(C(N2CC3(CC(NC(c4cnn(C)c4Br)=O)C3)C2)=O)ccc1F 43981,C1(COC)CN(C(c2nccc(Br)c2C)=O)CCN1C(C1CC2CC2C1)=O 43982,c1(C(=O)NC2C(NC(c3c(C)cc(C(F)F)o3)=O)CC2)n[nH]c2c1COC2 43983,Cc1nc2ccccc2n1CCNC1CC(NC(C2CC(C)C2)=O)C12CCC2 43984,C1(CC#CC)NC(=O)N(C(c2nn(C)cc2O)C)C1=O 43985,C1(CC(=O)NCc2c(C)cncc2)C2CCCC2N1C(c1csc(=N)[nH]1)=O 43986,c1(C(=O)NCc2ccc(C(=O)NC(C=C)(C)CC)s2)cncc(Cl)c1 43987,CC1C(NC(=O)C(C)(Cl)Cl)CCCN1C(c1cnn(C(F)F)c1)=O 43988,C1(C(C)C)(C(N2CCC(C)(F)C2)=O)CCCN1C(=O)CCn1cccc1 43989,N1(CCC(=O)NC(CC)C)CCn2cnc(C(F)(F)F)c2C1 43990,c1(CSC)cc(C(=O)NCC=CCNC(C2CCN(CC(C)C)C2)=O)ccc1F 43991,N1(C(CCN(C(C(CC=C)CC)=O)C(C)C)=O)CC(C2CC2(F)F)C1 43992,C(CC1CCC1)(C(=O)N(CC(C)NC(=O)Cn1cnnc1O)C)NC(C)=O 43993,NS(=O)(=O)c1ccc(C(=O)NCC2CCCCC2NC(=O)CC2NC(=O)NC2=O)o1 43994,Fc1cc2ccc1C1CCCN21.c1(-n2c(OC(F)(F)F)nnn2)cccc(Br)c1 43995,C12(CNC(C(CNC(=O)C#CC(C)C)OC)=O)CCC(F)(CC1)C2 43996,C(=O)(C(C)P(C)(C)=O)NCC(CCOC)NC(c1ncccc1CSC)=O 43997,C1(NC(CCCOCCC)=O)CCCN(C(=O)CNC(=O)NC)C1CCC 43998,Cn1nc(C(N2CC=C(C(=O)NCc3ncsn3)C2)=O)ccc1=O 43999,c1(C(N2CC3N(C(c4c(C)nn(C)c4C)=O)C3C2)=O)cc([N+](=O)[O-])c(F)cc1Br 44000,C(CC1=CCN(C(c2cnc(NC3CC3)s2)=O)CC1)N(C(C)=O)C.c1cnn(C)n1 44001,C1(NC(C(C)(C)O)=O)CS(=O)(=O)CC1NC(=O)Cc1csc(C(F)(F)F)n1 44002,c1(C(N2C3CC(NC(c4nn(CC)nc4Br)=O)(C3)C2)=O)c(C)cnnc1O 44003,Cc1c(C(=O)NCCNC(C2OCCC2C(F)(F)F)=O)c(=O)oc2ccccc12 44004,Cc1cc(C(=O)NCCCOCCC(=O)N(C2CCCN(C)C2)C2CC2)c(C)n1C 44005,c1(CNC(C2CC23CN(C(=O)Cc2cccnc2Cl)C3)=O)cc(F)cc(Cl)c1 44006,N1(C(C(C)(C)NS(C)(=O)=O)=O)CC(CNC(c2cnc(Cl)cc2N)=O)C(C)(C)C1 44007,C12(CNC(=O)CC3CC=CCC3)CCCC1N(C(=O)C=Cc1cccnc1)CC2 44008,C1(NC(c2cc(C)on2)=O)CC1C1CCCN(C(=O)CN2CCN(C)CC2)C1 44009,N1(CC(=O)OC(C(c2ccc(CC)cc2)=O)C)C(=O)c2cccnc2C1=O 44010,N1(C(C2CC(C)=C(C)CC2)=O)CC2(CCCC(CNC(c3c[nH]nc3C)=O)O2)C1 44011,C1(CC(=O)N(C2CCCCC2)CCNC(CC(=O)NCC)=O)CCOC(CC)C1 44012,C1(N(CCN)C(c2ccn(C)c2)=O)CCCCCC1.C(CC(=O)OCC)OC 44013,c1(C(=O)NC(CNC(c2c(C)ccc(SC)c2)=O)C2CC2)ccc2c(c1)CCO2 44014,C1(C(C)C)CCN(C(=O)CNS(=O)(=O)NC)CC1.C12(CC1)C(=O)N(C)C2 44015,N1(C(=O)OCC)CCCN(C(CC2CCCC2)C(=O)NC)CC1 44016,C1(NC(C(C)=C(C)C)=O)CC(NC(c2cnn(C)c2N)=O)CC1O 44017,C1(CCN(C(=O)C(F)F)C)CCCCN1C(=O)CCOC1CC1 44018,C1(NC(c2cn(CCC)nn2)=O)CCN(C(=O)C(c2ccc(F)cc2)CC)CC1 44019,C(=O)(C1Cc2ccccc21)N(C1CCN(C(C2(C(F)F)CCCC2)=O)C1)C 44020,c1(C(C)NC(c2n(CCCOC)nnn2)c2cc(OC)ns2)cccc(OC)c1 44021,CC(C)(C)C(CNC(=O)CC1CCC(O)C1)NC(c1sccc1CO)=O 44022,C(=O)(CCC(=O)NC1CC(CNC(C2CSCN2C(C)=O)=O)C1)NCC 44023,C(=O)(C1=NN(C)C(=O)CC1)N1C(CNC(c2c(C)cccc2C)=O)C(C)OCC1 44024,C(C(=O)N1OC2C=CC1CC2)(C1CCOC1)NC(C1C=CCS1)=O 44025,c1(OC)ccc(CC(=O)NCCOCCNC(c2cc(Cl)ccn2)=O)nc1 44026,NC1C2CCC1N(C(c1ccnc(OCC(F)(F)F)c1)=O)C2 44027,c1(C(CNCC23OCC(C(C)C)(C2)C3)O)ccc(S(C)(=O)=O)cc1 44028,c1(C(=O)NCC(C)(C)NC(c2c(CC)n(C)cc2)=O)oc2ccc(C)cc2c1C 44029,c1(C(N(C2CN(C(c3ccc(N)c(Br)n3)=O)C2)C)=O)n[nH]c2c1CC1CC21 44030,C(=O)(C(CCc1ccc(F)cc1)C(C)(C)C)N(C)CCNC(=O)OC1CC1(F)F 44031,c1(SC)ccc(C(=O)NCC(C(C)(C)C)NC(C2CCCCC2)=O)c(Cl)c1 44032,c1(C(N2CC(CNC(COCCCC)=O)N(C)CC2)=O)ccc2ccoc2c1 44033,c1(C(N2CCOCC(CNC(C(C(=C)C)(C)C)=O)C2)=O)c([N+](=O)[O-])cnn1CC 44034,CC1=C(C)CC(C)(NC(C2CCN(C(C3(Br)CC3)=O)CC2)=O)CC1 44035,O=C(C1=CCCCC1)NCCCN(C(c1cccnc1)=O)C1CC1 44036,c1(CNC(C2C=CC(NC(C(CC)O)=O)C2)=O)cc(O)cc(F)c1 44037,C1(C)(C(=O)NCCCCNC(c2c(OC)c[nH]n2)=O)CCC(C(F)(F)F)CC1 44038,C=CC(C)CC(=O)NC1CC(CNC(c2ccsc2-n2cnnn2)=O)C1 44039,CC(C)C(CNC(c1cnn2c1OCC2)=O)C(=O)NCCCc1cnccn1 44040,n1(CC)nc(C)c(C(=O)N(CCCCNC(=O)COCc2cccnc2)C)c1Cl 44041,C1(NC(C2(CCCC)CCC2)=O)CCN(C(=O)C(C)(C)c2ccns2)CC1CO 44042,c1(C(N2CCC(c3ncc(C(=O)O)s3)CC2)=O)cnn2c1CCC2 44043,C1(C(N(CCC(=O)NC(C(C)SC)C)CCO)=O)CN(C)CC(C)O1 44044,N1(C(c2cc(C)sc2)=O)CCN(C2CCCN(C(=O)CCNC(N)=O)C2)C(=O)C1 44045,C1(C(=O)NC(CCOC)C)CCC2(CC2)N1C(=O)CC#N 44046,c1(OC)nn(C)cc1C(=O)NC1CCC(CN(C(=O)C(C)n2ccnc2)C)CC1 44047,C(=O)(C(C)C(C)NC(c1c[nH]cc1C)=O)NC1(COCC)CC1 44048,N1(C(C(CC=C)OC)=O)CCC2(CCC(NC(=O)Cc3ccccc3C)CC2)C1 44049,c1(NC(C2(C3N(C(C(CC)CC)=O)CCC3)CC2)=O)ccc(F)cc1SC 44050,c1(OC)cccc(C2CC2N(c2nnnn2Cc2cn(C)nc2C(F)(F)F)C)c1 44051,c1(C(=O)NC(C)CCNC(=O)C(O)c2cnc[nH]2)ccc(Cl)o1 44052,c1(C(=O)NCC(C)NC(c2ccn(C(CC)CC)n2)=O)cc(C)nn1CC 44053,N1(C(C(CCC#C)O)=O)Cc2ccccc2C(NC(c2ccc(Br)o2)=O)C1 44054,c1(C(C(N2CCC(O)(CNC(C3C(COC)C3)=O)C2)=O)(C)C)cccc(C#N)c1 44055,c1(NC(c2n(CCCOC)nnn2)(COC)C2CCCC2)ccc2nncn2c1 44056,c1(C(=O)NCC(C)N(C(CCC(C)c2ccccc2)=O)C)cnc2[nH]cnc2c1 44057,C(=O)(C1=C(Cl)CCOC1)NCCC(C(=O)Nc1c(OC)cc(F)cc1)(C)C 44058,C1(C(N2CC(COC)(NC(=O)Cc3cc(C(C)C)no3)C2)=O)CC=C(C)CC1 44059,N1(C(C(CCC)(C)C)=O)CCC2(CCN(C(=O)CC3CCCCC3(F)F)C2)C1 44060,N1(C(CC(C=C)(C)O)=O)CCC(C(=O)N2CCC23CCCCC3)=C(F)C1 44061,C(=O)(CC(C)CC(C)(C)C)NC1(C(N(CCC#C)C)=O)CCN(C)C1 44062,C1(C(=O)NCC(CN(C(c2c(C)cc(C)o2)=O)C)O)CCC(C2CC2)CC1 44063,Cc1nc(C(C)C)ccc1C(=O)NCC(O)CCNC(c1cc(F)cc(F)c1)=O 44064,CC1CCN(C(=O)C2=CCCCC2)CC1CNC(=O)C=Cc1ccoc1 44065,Cc1cc(N2CCn3cccc3C2)nc(=NCCCc2ccc(C)c(C)c2)[nH]1 44066,C#CCC(C)(C)C(=O)NCCCN(C)C(C1CC1C#N)=O 44067,N1(C(c2c(C)nns2)=O)CCCC(N(CCF)C(c2ccc(OCCO)cc2)=O)C1 44068,c1(C(=O)NCC(CNC(c2ccn(CCC)n2)=O)OC)nnn(CC)c1C 44069,c1(C(N2C(C)CCC(NC(=O)CCCC(N)=O)C2)=O)cc2c(cc1Cl)OCO2 44070,n1(CC)c2ccccc2c2cc(CN3CC(C)C3(C)C)ccc12 44071,Cn1ncc2nc(Cl)nc(N3CC(NC(=O)CC(C)(C)C(F)F)CC3(C)C)c12 44072,C1(O)(C(=O)NC2CC3(C(NC(c4c(C)c(N)ccc4)=O)C3)C2)CCCC(C)(C)C1 44073,C1(N=c2cc(Br)n(C)[nH]2)(c2n(C(C(=O)OC)C)nnn2)C(C)CCC1 44074,c1(C(=O)NCCSC)cc2cc(-c3cn(C)nc3C)ccc2oc1=O 44075,C1(NC(c2cccc(NC(C)=O)c2)=O)CC(C)CN(C(C2CCC(C)(C)O2)=O)C1 44076,C(=O)(C(C)C(=O)N1CCN(CCCNC(=O)C(C)(C)n2cnnn2)CC1)OC 44077,c1(C(=O)NCCC2N(C(c3c(C)con3)=O)CCOC2)c(Cl)cc(Cl)cc1Cl 44078,C1(C)(C(=O)NCCCN2CCN(C(CCSC)=O)CC2)C(C)(C)C1(C)C 44079,C1(C(N(CC(C)O)Cc2ccco2)=O)CCN(C2CCOC2C)CC1 44080,c1(C(=O)NC2CC(N(C(C(CC=C)OC)=O)C)C2)[nH]nc2ncccc12 44081,c1(CCC)n[nH]cc1C(=O)NCC(CNC(C1CCC(=O)C1)=O)CO 44082,CC1(C)CC(=O)N(CC(=O)NCC2CCCCN2C(=O)CCc2ccccn2)O1 44083,c1(CCC(=O)NCCCC(=O)NCC(CC=C)NC(N)=O)ccc(Cl)c(OC)c1 44084,C1(C(=O)NC2CC(C(C)C)OC2)C=CCN(C(=O)Cn2ccnc2)C1 44085,c1(C(N2CCC(CC)C2C(=O)NCCC2CC2C(=O)OC)=O)ncc(F)cc1C 44086,c1(C(=O)NCCCN(C(=O)CC2C=CCCC2)CC)cc(C(F)F)cs1 44087,Cc1nc2ccc(C(C)NS(=O)(=O)Cc3cc(Cl)ccc3Br)cc2o1 44088,N1(C(c2ncc[nH]2)=O)CCC(C2CCCN(c3nccn4nnnc34)C2)CC1 44089,C#CC1CC(NC(=O)CONC(=O)C=CC(C)(C)SC)C1 44090,C#CC1(C(N2CC(C(C)(C)C#N)C2)=O)CN(C(c2cc(OC)ccn2)=O)C1 44091,c1(C(=O)OC)ccncc1NC(C12CC(NC(C3COC(=O)N3C)=O)(C1)C2)=O 44092,N1(C(COC(C)=O)=O)CCC2C1CCCN2C(=O)C=Cc1c(C)coc1C 44093,c1(NC(C2CC(C)C(C)CC2)=O)cccc2c1CN(c1ccccn1)C2 44094,c1(C(C)C)ccc(C(O)C(=O)N(C2CC2)CC2CN(C)CCO2)cc1 44095,CCN=c1ccc(C(=O)NC2CN(C(c3cc(C(C)(C)C)c[nH]3)=O)C2)c[nH]1 44096,C1(C)(c2nc(CC)on2)CCN(N2CCC(C)(C(=O)OC)C2)C1 44097,C1(C(=O)NC(C2CCN(c3nnc(C(N)=O)o3)C2)C)CCOC2(CCC2)C1 44098,C(=O)(C1CCc2nccn21)N(CCC1CCN(C(C2CC(C)(CC)C2)=O)CC1)C 44099,C1(NC(=O)CCCF)CN(C(c2cccc(F)c2)=O)CC1C(F)F 44100,N1(C(Cc2c(C)n[nH]c2C)=O)CC(NC(c2cc(CO)ccc2O)=O)C(C#N)C1 44101,C(c1cccc(CO)c1)=CC(=O)NCCC1CSCCN1C(C1CC1F)=O 44102,N1(C(c2c(CC)ccc(F)c2)C(=O)NCCC2CC2)CCC2OC(C)(C)OC2C1 44103,c1(C(C)(C)C)noc(CCCN(C(=O)CCCN)C(=O)Cc2cccnc2)n1 44104,c1(C(=O)NC(C2CCCC2)CC)cc(CNC(C2CCC(F)CC2)=O)nn1C 44105,C1(C(N(C(C#C)C)C)=O)CN(C(=O)Cc2scnc2C)CCO1 44106,c1(C(=O)NCCCNC(C(C)C2CC2)=O)ccnn1-c1cccnc1 44107,C(=O)(CCCc1nccs1)C(C=CCNC(=O)OCC1(NC(C)(C)C)CCC1)=O 44108,CC1CC(C)N(C(c2oc(S(N)(=O)=O)cc2C#N)=O)CCN1C(C)(C)C 44109,C(=O)(CCCCCCNC(=N)N)N1CCCC(c2nnc(C)o2)C1 44110,n1(CCCNC(C2(CNC(C(C3CC3)OCC)=O)CCC2)=O)cc(C)cn1 44111,Cc1cc2ncnc(N3CCC4(CCN(C(c5ccc(F)c(F)c5)=O)C4)C3)c2[nH]1 44112,C12(COC(c3cc(N)c(N4CCOCC4)cc3)=O)CCCCC(=O)N1CCC2 44113,c1(OC)ccc(CN2CCC(C(N3CCOCC3C)=O)C(O)C2)c(Br)c1 44114,c1(C(=O)NC2C(CNC(=O)C3=CCC3)CC2)ccc2oc(=O)oc2c1 44115,C1(C(N2C(CCNC(=O)COc3cccc(F)c3)CCC2)=O)CCCC(F)(F)C1 44116,c1(NCCc2cccc(OC)c2)ncnc(NC2(C)CCC(C)CC2)c1C 44117,n1(C(C)C)cc2ncc(C(N3CCC4(CC3)CNC4C(=O)C3CC3)=O)cc2n1 44118,N1(C(C)=O)CCC2CCC(C1)N2C(=O)CCCCc1ccc(Cl)cc1 44119,CC(C)CC(F)C(=O)N1CC(CNC(=O)Cc2ccc(O)cn2)C(C)(C)C1 44120,C=Cc1ccc(C(=O)NC(CC(=C)Cl)C(=O)NC2(COC)CC2)cc1 44121,c1(NC(C2C(C(=O)OC)C2)=O)sc2c(c1C(N1CCC(O)C(F)C1)=O)CCC2 44122,N1(C(C2C(C(=O)OCC)CC2)=O)CCCC1CC(=O)NC(C(C)C)C1CC1 44123,C1(C(=O)NC(CC)(C)CNC(=O)C=Cc2ccc(C)s2)CC2(CCO1)CC2 44124,CC1CCN(C(c2ccn(-c3ccccc3)n2)=O)CC1N(C)C(C1CCCO1)=O 44125,N1(C(C(C(C)C)S)=O)CCn2ncc(CNC(=O)C(N3CCOCC3)O)c2C1 44126,c1(C(=O)NCCCCC(C)NC(c2cocc2C(N)=O)=O)nnc(O)cc1O 44127,C1(CNC(C2(CC=C)CCC2)=O)(NC(C2CCCNC2=O)=O)CCCCC1 44128,N1(C(=O)Nc2cnn(-c3ccncc3)c2)CCCC2(C1)CC(F)(F)C2 44129,CCC(C)(CNC(C1(C)CC1(F)F)=O)NC(=O)CCCn1cncn1 44130,C(CCCCC(=O)NCC1CCCC1NC(c1ccc(C(C)C)cn1)=O)=CC 44131,C12(N(c3cc(C(C)(C)C)c[nH]3)C(C(C)OC)=O)CCOCC1CN(C(=O)C(N)=O)C2 44132,C1(C)(OCC=C)CCN(C(=O)CC(CCC)NC2CCN(CC)C2)CC1 44133,C1(F)(CNC(CSCCC#N)=O)CN(C(C2CCCN2Cc2ccsc2)=O)C1 44134,N1(c2n(CC(C)C)c(CN3CCCC(C)C3)nn2)CCC(O)CC(C)(C)C1 44135,c1(C(N2CCC(C)(C(=O)NCC(CC)C)C2)=O)c(C)nn(C)c1C 44136,c1(SC)ccc2c(c1)C(NCC1CC(COc3ccccc3)CO1)CCO2 44137,c1(C(N2C(CN(C(CCSCCC)=O)C)COCC2)=O)ccc2c(n1)CCOC2 44138,C(=O)(CC(C(F)F)C(C)(C)C)NCC1CC(OC)CN1C(=O)CN1CCOCC1 44139,C1(CNC(C2(OC)CCCC2)=O)CC(NC(c2cncn2C)=O)CC1O 44140,C1(C(=O)N(CCCCCNC(=O)Cc2ccsc2)C)(OC)CS(=O)(=O)C1 44141,N1(C(CCCCCNC(N)=O)=O)CCc2sccc2C1CNC(c1ccoc1)=O 44142,C(=O)(C(C(C)(C)C)NC(C1(C)CC(=O)N(C)C1)=O)NCCOCCCC#C 44143,C(=O)(C(CC(C)C)C(N)=O)N(C)CC1(O)CCN(C(CC(CC=C)(C)C)=O)CC1 44144,c1(C(=O)OC)ccoc1C(=O)NC(C)CCNC(c1csc(C(F)F)c1)=O 44145,C(=O)(C(O)CCS(C)=O)N1CCC(N(C)C(C2(CN(C)C)CC2)=O)CC1 44146,N1(CC(=O)NCCCCOCC)C(=O)C2CCCCC2C1=O.C(=O)(C=CC(=O)OC)N 44147,C1(NC(CC2C(C)(C)OCC2)=O)CCCC12CN(C(C1CC3C(C1)C3(F)F)=O)C2 44148,O(N(C)C(=O)CNC(C(C)(C)C1CCCO1)c1nnnn1C1CC1)CC 44149,CCC(C)CCCC(=O)N1C2CCC(C(=O)NCC3Cc4nccn4C3)C1CC2 44150,c1(SCC(N2CCC(CCCC(=O)OC)CC2)=O)nc2ccccc2n1C 44151,N=c1nc(N2CC(CC(N)=O)C(CC(N)=O)C2)[nH]c(=NCC2CCCC(=O)N2)[nH]1 44152,c1(C(=O)OCC)cc(F)c(C(=O)NC(C(C)NC(=O)C=C(C)C)C(C)C)cc1F 44153,C1(NC(c2ccc(O)nc2)=O)CC2CN(C(c3ccc(S)cc3)=O)CC2C1 44154,C1(C(=O)NCCc2c(CNC(c3c(C)n(C)nc3)=O)nco2)CCC(O)CN1C 44155,c1(CC(=O)NCC2N(C(CC(C)SC)=O)CCCCC2)ccc2occc2c1 44156,C1(NC(CC(C)CF)=O)CCOC12CCN(C(c1cc3ccccc3[nH]1)=O)CC2 44157,C12(NC(CCC=C=C)=O)CCCCCC1N(C(=O)COCc1cccnc1)CC2 44158,c1(C(=O)NC(CC(C)NC(COC(C)=O)=O)C)cc(C)c(Br)o1 44159,N1(C(C(C=C)(C)CC)=O)CC(C)(C)C(NC(C2CC=C(C)CC2)=O)C(C)(C)C1 44160,CCC(CC(=O)N1CCC(OCCCNC(=O)CC2CCOC2C)CC1)SC 44161,N1(C(C(C)n2ccnc2)=O)CC=CC(NC(c2scc(Br)c2Cl)=O)C1 44162,C(=O)(CCCC(=O)N1CC(CNC(=O)CCCCCN(C)C)(OC)C1)OCC 44163,c1(C(N(CCN(C(C2N(C(C)=O)CCCC2)=O)C)C)=O)c(C)cn(C)c1C 44164,C(=O)(C1=CCC(C)CC1)NCCC(C)NC(C1(C(C)C)COC1)=O 44165,C(=O)(CCCCC(F)(F)F)NCC1CN(C(C(CC)C(C)(F)F)=O)CC1(C)C 44166,N1(C(C(CC)(C)C#N)=O)CC2CN(C(=O)C(C)c3ccsc3)CC2C1 44167,CC12CCC(C(=O)NCC3COC(CNC(C4(C5CCC5)CCC4)=O)C3)(CO1)C2 44168,N1(C(C2=C(C)CC2)=O)CC2(CC(NC(=O)C(c3ccnn3C)O)CO2)C1 44169,Cc1nccnc1C(=O)N(CC(C)(C)C(=O)NCC(C)(C)CN(C)C)C 44170,C(C)(CCC(=O)NCC(C)(C)OCCNC(=O)CCNS(C)(=O)=O)SC 44171,CN1CCOCC1c1n[nH]c(CNC(=O)NC(c2ccccc2)c2cccs2)n1 44172,C1(NC(C(CCC)c2ccccc2)=O)CN(C(c2ccc(Cl)cc2)C)CCC1C 44173,c1(C(=O)NCC(CCOC)NC(=O)CC2CSCCO2)cn2ccnc2s1 44174,N1(C(C(CCSC)(C)C)=O)CCC2(CCCN2C(c2ncc(Cl)cc2Cl)=O)C1 44175,N1(C(c2cc(Cl)ccn2)C(=O)NCC=C)CCOC2(CCSC2)C1 44176,C1(NC(C2(CCOC)CC=CC2)=O)CCN(C(=O)C(C)C2CCOC2)CC1C 44177,C(=O)(C#CC(C)(C)O)NCC1CC(COC)CN1C(C1CC2(CC2)CO1)=O 44178,c1(C(=O)NCC2(C(=O)NC(C(C)(C)O)CCO)CC2)ccn2cncc2c1 44179,N1(C(C(CC)NC(N)=O)=O)CC2(CCN(C(=O)C=C3CCC(C)C3)CC2)C1 44180,c1(OCC)ncc(C(=O)NC2CCC(NC(C3(C)CCCCO3)=O)CC2)cn1 44181,C(=O)(C(F)CC(C)(C)NC(=O)Cc1cnn(C)c1)N(CCCOCC)CC 44182,c1(C(=O)NCC(C)(C)NC(C2CCC(Cn3ccnc3)O2)=O)cc([N+](=O)[O-])n[nH]1 44183,c1(OC)cc(O)c(C(N2CCN(C(C3CCCC3(F)F)=O)C(C)C2)=O)cc1OC 44184,N1(CC)CCCC(C(=O)NCC2(CNC(=O)CN(C)CCO)CC23CCC3)C1 44185,C1(C(N2CCOC(C)(CNC(=O)CSC)C2)=O)(COC)CCCNS1(=O)=O 44186,N1(C(C2(O)CCC(C)CC2)=O)CCCC2(C1)CN(C(C1CCC(=O)C1)=O)CCO2 44187,c1(CC)ccc(CNC(C2CC2CNC(C2(C)CCOC2)=O)=O)cc1 44188,N1(C(C=CCOC)=O)CCC(C(=O)NCC2CN(C)CCO2)C1(C)C 44189,N1(C(c2c(C)c[nH]n2)=O)CC2CCCC2(NC(c2occ3c2CCC3)=O)C1 44190,C1(NC(CCNC(=O)CO)=O)CCN(C(=O)CCc2ccc(F)cc2Cl)CC1F 44191,CC(C)C(C)C(C)CC(=O)NC(C)(C)COCCCNC(c1cnc[nH]1)=O 44192,N1(C(C(CC)(C)C)=O)CC23CCCC2(C1)CN(C(c1cnc(OC)nc1)=O)C3 44193,C(=O)(C(CC)NC1(C)CN(CC)C1)OCC 44194,N1(C(c2ccc(CCC=C)cc2)=O)CC2CC(NC(c3snc(C)c3N)=O)C1C2 44195,Cc1nc2ccc(C(=O)NC(C)CN(C)C(c3cc(C4CC4)ncn3)=O)cn2n1 44196,c1(OCC(=O)N(C(C)CCNC(c2cnc(C(F)F)s2)=O)C)ccc(Cl)cc1F 44197,Cc1ccccc1C(=O)N(C1CCCC(N(C(=O)Cc2ccsn2)C)C1)C 44198,C(=O)(CC(O)CCCCC)NCC(CC=C)NC(=O)CN1CCN(CC)C(=O)C1=O 44199,c1(OC)cc(N)c(Cl)cc1C(N1CC(N(C)C(C23COCC2C3)=O)C2(CC2)C1)=O 44200,c1(C(=O)NC(CNC(C2(CCC)CCC2)=O)C)cc(C)c(Br)c(C)c1 44201,N1(C(C(CC)NC(C)=O)=O)CC(CNC(C2CCC(=O)N(C)C2)=O)CC(C)C1 44202,N1(C(c2cc(CNC(C(CCC)F)=O)on2)=O)CCC(O)C(F)C1 44203,c1(C(N2CCCN(C(C=CCOC)=O)CC2)=O)cc2nc(C)cc(C)n2n1 44204,C(C(O)C(=O)N1CC=CC1)NC(=O)CC1CCCO1 44205,c1(C(N2CC(CNC(COCCOC)=O)C(C)(C)C2)=O)cc2cc(Cl)ccn2n1 44206,N1(C(C2C(C(=O)OC)C2)=O)CCC(CNC(=O)Cc2cccs2)C(C)(C)C1 44207,c1(C(=O)NCCCCCN(C(c2c(C)snn2)=O)C(C)C)cncc(N)c1 44208,Cc1cccc(Br)c1-n1cc(CC2CCCN2C(=O)CCc2nc[nH]n2)nn1 44209,c1(CCC(=O)NC(C2CCN(C(C3C(=C)C3)=O)C2)(C)C)cn(C)c2ccccc12 44210,c1(NC(C2C(NC(CN3CCC(C)C3)=O)COC2)=O)cncc(C2CC2)c1 44211,O(C=CC(=O)N(CCC(C)NC(=O)CC1CC(C)(C)C1)C)CC 44212,CC(C)C(C(=O)NC1CCCN(C(=O)COC(C)(C)C)C1)c1cccnc1 44213,C(C)(CCC(=O)N(CC(O)CN(C(=O)CSc1nncs1)C)C)OC 44214,c1(CN2CCC(c3c(OC)cc(Cl)cc3)CC2)cn2cc(F)ccc2n1 44215,C1(C(N(CCC(=O)NC)C(C)C)=O)C2CN(C(=O)CCN3CCOCC3)CC12 44216,c1(C(N(C2CCCN(C(c3cnsn3)=O)CC2)CC)=O)ccc2c(c1)CCNC2=O 44217,N1(C(C(C)NC(C)=O)=O)CC(O)(CN(C(=O)CC2COCC2O)C)C1 44218,c1(NC(C(N2CC(CCC=C)(NC(C3(C(C)C)COC3)=O)C2)=O)=O)ccc(O)cc1 44219,c1(NC(C(=O)NCC(CC=C)NC(=O)C(C)(C)SC)C)ccc(C(F)(F)F)cn1 44220,N1(C(c2c(CNC(C3(C#N)CC3)=O)occ2)=O)CCC(O)(C(F)F)C1 44221,C1(CNC(c2c(OC)nsc2OC)=O)CCC(C)N(C(=O)CCC(C)OC)C1 44222,N1(C(C(C(C)C)O)=O)CC2CN(C(C34CSCC3C4)=O)CC2C1 44223,C1(C(=O)NCCC#C)CCN(C(=O)c2cccc(Cl)c2)O1 44224,CC1COc2c(C(=O)NC3C4CC3N(C(c3cc(=O)cc(Cl)[nH]3)=O)C4)cccc21 44225,C1(C)(C(=O)NC(CCC)CO)CN(C(=O)CC2(C)CCC2)CC1C 44226,c1(C(N2CCCC(N(C(C3(COC)CC3)=O)C)C2)=O)cc(C)c(C)nc1C 44227,Cc1nc2cccc(C(N3CCC4C3CCCN4C(c3ccn(C)c3)=O)=O)c2s1 44228,C1(NC(CC(=O)OC)=O)CC2CCC1CC2NC(C1(C)CC=C(C)CC1)=O 44229,CC1(C(=O)NCCC2CCN(C(=O)COC3CCC3)C2)CCOC1 44230,Cc1nc2cccc(C(=O)N(CC(C)NC(=O)C(F)n3cccn3)C)c2s1 44231,C12(C(=O)NCC(C)N(C(C3(c4cccc(C)c4)CCC3)=O)C)CCC(F)(CC1)C2 44232,C1(CN(C(C(C)C)=O)C)CN(C(C2CCS2(=O)=O)=O)CCO1 44233,c1(NC(C(c2ccccc2F)NC(C(C)=O)=O)=O)cccc2cncc(C)c12 44234,CCCCCC(CC)C(=O)NCC1CC2(CC(NC(C3(CCC)CCC3)=O)C2)C1 44235,Cc1cc(C(=O)NCC(C2CCCC2)NC(=O)C(C)(C)ON)n(C)n1 44236,c1(C(=O)NCC2(C(=O)NC(c3ccc(F)cn3)C)CC=CC2)ncncc1Cl 44237,C(c1cc[nH]n1)=CC(=O)NCC1CCC(NC(C2CCC(=O)N2)=O)C1 44238,Nc1cccc(F)c1C(=O)NCC1CCN1C(=O)CSc1ccncc1 44239,C(=O)(CCCC(C)(C)C)N1CC(CC)C(NC(c2cccc(NC(C)=O)c2)=O)C1 44240,CC(C(C)N(C(=O)CN)C1CC1)S(C)(=O)=O.C1CCC(=O)N1C 44241,c1(OC)cc(Cl)ccc1CC=O.N1(N2C(CNC)CCCC2)CCC2(CC1)CC2 44242,C1(NC(=O)NC2(CN(C)C(C3CSCCS3)=O)CC2)CCCC1c1nc[nH]n1 44243,N1(C(C(C(C)(C)C)N2CCCC2)=O)CCC2(CC1)CC2CNC(c1ccon1)=O 44244,C1(C(=O)NC2C(CNC(=O)CCC3CCCCO3)CCC2)CC2OC1C1CC21 44245,C(=O)(C1COc2ccc(Cl)cc21)NCCN(C(C1CCC1CF)=O)CC 44246,N1(C(CCC=C)=O)CCC2(CCCCN(C(=O)CC(=O)N(C)C)C2)C1 44247,C1(CC(=O)N(CCn2c(C)ncc2)C)CN(C(=O)Cc2nccn2C)CCC1C 44248,c1(CNC(C2(C)CN(C(=O)CC3CC4CCC3C4)C2)=O)cnc(C(F)F)nc1 44249,n1(CC)cc(Cl)c(C(=O)N(C(C)CCNC(=O)Cc2ncc(C)s2)C)n1 44250,N1(C(c2ccc(CC(C)C)s2)=O)CCCC(C)(NC(c2cc(F)cc(Cl)c2)=O)C1 44251,c1(OC)cncc(C(=O)NCC2CN(C(=O)CSCc3cccs3)CC2O)n1 44252,c1(C(=O)NCCCC(C)NC(C2(C)CC(C)C2)=O)cccc2c1COCCN2 44253,C(C(C)C)(C(O)C(=O)NCC(c1ccccn1)C)OC 44254,N1(C(C2CCCN(C(C)C)C2)=O)CCCC2CN(C(=O)CCc3nc[nH]n3)CC12 44255,c1(C(N2CC(CNC(C3(CC#C)CCC3)=O)C(C)C2)=O)cc2c([nH]1)CCCC2 44256,O(N(C)C(=O)CN=c1[nH]c(=NC(C)C(C)CC)[nH]c2c(F)cccc12)CC 44257,C=CCCCC(C(=O)NC1CCC(C(N)=O)C1)NC(=O)CC1(OC)CCC1 44258,[N-]=[N+]=NCCCCCCC(=O)NCC1CN(C(=O)CC23CCCC2C3)C1 44259,C1(C)(C(N(C)C)=O)CCCCO1.C1(C)COCC1NC(c1coc(CO)c1)=O 44260,N#Cc1ccc(C(=O)NCC(N2CCN(C(=O)C(F)(F)C(F)F)CC2CF)=O)cc1 44261,c1(NC(C2CCN(Cc3ccc(C)[nH]3)CC2O)=O)cccc2c1OCO2 44262,c1(N(C(C(n2c(CCCC)ncc2)C)=O)CC2CC2)ccc(F)cc1 44263,C(=O)(C1=C(Cl)CCCC1)NC1CN(C(Cc2c(C)scc2)=O)CC(F)C1 44264,C1(C(N2CCC(C(=O)NCCNC(=O)OC(C)(C)C)C2)=O)CCN(C)C1=O 44265,Cc1sc(Br)cc1S(=O)(=O)NC(c1c(F)cccc1F)C 44266,C(=O)(C(C)(O)COC)NCC1(OC)CN(C(=O)CCC(C)C)C1 44267,N1(C(CCS(=O)(=O)NC(C)=O)=O)CC2CC1CCC2NC(C1(C(F)F)CCC1)=O 44268,N1(C(CC(c2ccc(C)cc2)C)=O)CC2CC(NC(=O)CC3CC=CCC3)C2C1 44269,c1(CC(C(N)=O)NC(C2CCCN2C(c2ncccc2F)=O)=O)ccc(O)cc1 44270,CN1CCOCC1CC(=O)NCc1ocnc1Cn1cc(C2CC=CCC2)nn1 44271,C12(COC)COC(C(=O)NC3CCCCC3NC(c3c(C)coc3SC)=O)(C1)C2 44272,C1(C(N2CCC(O)(C(C)NC(C3CCC(C)(C)O3)=O)C2)=O)CCS(=O)(=O)CC1 44273,C1(NC(C2CCC(C)O2)=O)COCCN(C(c2cccc(Br)c2F)=O)C1 44274,N1(C(C(SC)SC)=O)CC(NC(=O)Cc2cc(C)on2)CC(C)C1 44275,C#CCC(C)(C)CNC(=O)C(CCOC)NC(c1[nH]ccc1C)=O 44276,c1(OCC(=O)NCCC2CCCN2C(=O)CC2COCC2O)ccc(F)cc1 44277,N1(C(C(N2CCSCC2)C)=O)CC2CCN(C(c3cccc(N)c3)=O)C2C1 44278,C1(C(=O)NCC23CC(NC(CC(C(=C)C)OCC)=O)(C2)C3)Cc2ccncc2C1 44279,C(=O)(CC(C)CF)N(CCOCCOCC#C)CC.C1C(=O)NCCCO1 44280,C(=O)(N=c1c(Br)c[nH]c(C)c1Br)C1CCCN(Cc2c(OC)ccc(C)c2)CC1 44281,C(N=c1[nH]c(=NCCC=CBr)[nH]c2c1CCCCCC2)C1(C)CCC(=O)N1 44282,c1(CNC(=O)CC2(O)CN(C(c3c[nH]nc3C3CCCO3)=O)C2)ccccc1 44283,N1(C(c2cc(C)no2)=O)CCC2CCC(C1)N2CC1CCC2CC2C1 44284,O=C1CCc2c(C(N3CCOC(C4CC(F)(F)C4)C3)=O)n[nH]c2C1 44285,c1(C(=O)O)ccnn1Cc1cn(CC(N2CCC(N3CCCC3=O)C2)=O)nn1 44286,C1(CCNC(Cn2ccc(C)n2)=O)CCCCN1C(=O)C=CCO 44287,C1(CCN(C)C(c2ccccc2OC2CCC2)=O)CCN(C(C2CC2F)=O)CC1 44288,C1(NC(C(C)C2CCC2)=O)CN(C(c2cc3cnccc3[nH]2)=O)CC2CCCC12 44289,C(=O)(C(CCC1CCC1)NC(c1c[nH]c(C)c1)=O)NCCOC 44290,C1(NC(c2ccn3nccc3n2)=O)CN(C(=O)CC2CCCC2O)CC2(CC2)C1 44291,C(=O)(CC1(O)CCOc2ccccc21)N1CC(C)(C)c2c1cccc2 44292,c1(CCC)cc(C(N2CCC(C(C)NC(C3(CC(C)C)CC3)=O)C2)=O)n(C)n1 44293,c1(OC)cc(C)c(C(N2CC=CC(NC(c3c(Cl)n[nH]c3C)=O)C2)=O)cc1Cl 44294,N1(C(C2(NC(C(CC=C)OC)=O)CCC2)=O)CCN(C2CC2)C(C)C1 44295,N1(C(C2C(c3c(C)cccc3)C2)=O)CC2CCCC(C1)N2C(C1CCCCC1)=O 44296,c1(C(=O)NCC(CCCC)NC(=O)C(CC(C)C)OC)cc(OC)cc(C)c1N 44297,N1(C(CC2(NC(c3cc(CO)on3)=O)CC2)=O)CC(O)(C(F)F)C1 44298,N1(C(c2cc(OCC)no2)=O)CCN(C(=O)CCC(C)OC)CC1C1CCC1 44299,C(CO)(C(=O)NCC1(C(=O)NCC2CCOCC2)CCCC1)NC(N)=O 44300,c1(C(=O)NCC2OCC(CNC(=O)C(Cl)=CCl)C2)cnn2ncccc12 44301,N#CC1CCCC(C(N2CC3CC2(C(=O)NCC2CC4C=CC2CC4)C3)=O)C1 44302,C12(NC(C34N(C(=O)CN5CCCC5=O)CCC3C4)=O)CCC(O)(CC1)CC2 44303,c1(C(N2CCCCC(NC(C(CC)(C)OC)=O)CC2)=O)c(F)cc(C#N)cc1F 44304,C1(C(N(CCn2ncc(C)c2)C)=O)CC(C)CN1C(c1ccc(O)cc1)=O 44305,C1(C(N2CCCC(NC(c3c(CC)noc3)=O)C2)=O)CN(S(N)(=O)=O)C1 44306,c1(C(=O)NCC2C(NC(C3C(CC)C3)=O)C2)cc(N(C)C)cc(C#N)c1 44307,Cc1ccc(NCC2CCN(c3ccc(F)cc3F)C2)cc1Br 44308,CN1CCN(C(C2(O)CCCCC2)=O)CC1C(=O)NCc1ccc(C(N)=O)o1 44309,Nc1cc([N+](=O)[O-])ccc1C(N1CC(NC(=O)Cc2cncs2)C2(CCC2)C1)=O 44310,c1(C(=O)NCC(C)(C2CCC2)NC(C2CC2F)=O)cc(Cc2ccccc2)c[nH]1 44311,C(C(=O)NC(CCSC)C(=O)NCC1C=CCC1)(C(C)C)OCC 44312,c1(Oc2c(-c3nc(C(CC)CC4CC4)n(CC)n3)nccn2)ccc(F)c(Cl)c1 44313,C=CCN=c1[nH]cc(C(=O)NC2COCCN(C(C3CCCCC3(C)C)=O)C2)s1 44314,C=C1CC2CCCC(C1)N2C(C1CC(NC(c2ccc(C)cc2F)=O)CCO1)=O 44315,N1(C(C23CC(C)C2C3)=O)CCC2(CC1)CC2CNC(c1cnn(C)c1Cl)=O 44316,c1(N(CCCC(F)(F)F)C)[nH]c(=NCc2nn(C)cc2Br)nc2c1ncn2C 44317,Cc1ccc(N2CCOC(C(=O)NCC3CCN3C(=O)OC(C)(C)C)C2)nc1Br 44318,C#CCC(C)(CC)C(=O)N1CCC(c2cccc(F)c2)(NC(=O)CC#N)C1 44319,c1(C(N(C2CN(C(N3CCCC(N(S(C)(=O)=O)C)C3)=O)C2)C)=O)cccnc1N 44320,CCC(C)(COC)C(=O)NC(CNC(=O)C1=COCCC1)C1CC1 44321,C12(CC)CN(C(=O)Cn3cnnn3)C(CNC(C3CCS(=O)(=O)N3)=O)(C1)C2 44322,C1(CC)(CC)CCN1C(=O)CC(C)N(C)C(c1cscc1C)=O 44323,c1(CCC(=O)NCCC(CNC(C=C(C)C)=O)O)cccc(C)c1Br 44324,O(NC(=O)C(C)(N(C(=O)CC(=O)N(C)C)C)C1CC1)Cc1cccc(C)n1 44325,N1(C(CCC2CCN(C(C(C)C3CCOC3)=O)CC2)=O)CCc2n[nH]cc2C1.CO 44326,CC1CN(C(c2csc([N+](=O)[O-])c2)=O)CCCN1C(C1CC(=O)N(O)C1)=O 44327,C1(NC(C(C)(C)OCC)=O)CN(C(=O)CCCCc2cnc[nH]2)CC1O 44328,C(C(=O)NCC(O)CCNC(=O)CCCc1cccnc1)(C(C)O)NC(C)=O 44329,c1(C(=O)NC2(C(N(CCCO)CC#C)=O)CC2(C)C)cnn(C)c1C#N 44330,C(=O)(CC(C)(C)CN(C)C)NC(C(C)C)CNC(c1ccnn1CC(F)(F)F)=O 44331,CC1(C)C(CC(=O)NCCCCCO)CCN1C(=O)C(O)CN1CCCC1 44332,Cc1nc(C(N2CC(NC(c3ncccc3Br)=O)C(O)C2)=O)n(C)n1 44333,CCC(C(=O)N(C(C)C(=O)NCC1CCCCO1)C1CC1)N(C)C 44334,C(=O)(C(F)(F)C(C)(C)O)N1CC(NC(COCP(C)(C)=O)=O)C(C(F)(F)F)CC1 44335,C1(C(=O)NCC=CCNC(CC2CC(CC)C2)=O)CC(=O)N(Cc2ccccc2)C1 44336,CCC(C)CCC(=O)N1CCCC1CCC1CCN(C(C2CC2(F)F)=O)CC1 44337,Cc1cc(=NC2CC(NC(c3c[nH]cc(F)c3=O)=O)C2(C)C)[nH]cc1C#N 44338,C1(NC(CCC(N)=O)=O)CN(C(c2cnn3c2OCC3)=O)C2CCCC12 44339,C(=O)(CCCCC(N)=O)NCC1(CNC(C2CC3(CC(=C)C3)C2)=O)CCC1 44340,C(=O)(C#CC1CCCOC1)NC1CC2CN(C(c3cc(C#N)on3)=O)CC21 44341,C1(NC(C2C(CCOC)C2)=O)COCCC1NC(c1nc(OC)c(C)s1)=O 44342,C(C1c2ccsc2CCN1C(c1[nH]ncc1C#N)=O)NC(C(CC(C)C)OC)=O 44343,N1(C(c2ccc(C3C(C)C3)o2)=O)CCN(C(=O)CCP(C)(C)=O)CC2(CC2)C1 44344,CC(C)C(CN(C1CC1)C1CC1)C(=O)NC1CCC(F)(F)CC1 44345,C1(C(N2CC(C(N3CC(C(=O)NC)OCC3)=O)OCC2)=O)CCOC(=O)CC1 44346,c1(C(N2CCC(CSc3ccccc3)C2)C(=O)NCC)ccn2nccc2c1 44347,c1(C(CC)CNC(N2CCCC(N(C)C)C2)=O)ccc(Cl)c(F)c1 44348,C#CC1(C(=O)NCC2CC2Cl)CN(C(=O)CC2CCCC2C)C1 44349,O=C(C1=CCCN(C(=O)Nc2cc(Cl)ncc2F)C1)Nc1ccccc1 44350,CC1CC(NC(=O)C(F)=CC2CC2)CN(C(=O)C(C)(O)c2ccccc2)C1 44351,c1(C(N(CC(C)CNC(=O)CCc2cnc[nH]2)C)=O)ns[nH]c1=O 44352,c1(OC)ccc(CC(=O)N(CC(C)NC(=O)Cc2c[nH]ccc2=O)C)c(C)c1 44353,N1(C(C2ON=C(C)C2)=O)CC(N=c2[nH]c3c(C)cccc3o2)C2(CCOCC2)C1 44354,C(=O)(CN=c1cc[nH]cc1)N1CC(NC(c2c(C)snc2)=O)CC12CCC2 44355,C1(CNC(C(CC)F)=O)CC2(CCN(C(=O)CCc3cc(Cl)no3)CC2)C1 44356,c1(C(=O)NCC(c2ccsc2)O)cc2cccc(Br)c2o1 44357,N1(C(COC(C)(C)C)=O)CCN(CC=CCNC(=O)CC2CC3COCC23)CC1 44358,C1(NC(c2c(C)[nH]nc2CO)=O)CN(C(C2(C)CNC(=O)C2)=O)CCC1CO 44359,C(C1=Nc2cccc(F)c2S(=O)(=O)N1)N1C(C)CC(O)CC1 44360,c1(OC)ccc(CNc2ncnc(NCCC(O)COC)c2C)c(OC(F)F)c1 44361,c1(C(=O)NC2CC(N)C23CCOCC3)nc(O)nc2ccccc12 44362,c1(C(N(C(CCNC(c2c(Cl)cn(CC)n2)=O)C)C)=O)ccc2cnccc2n1 44363,CC1=NNC(=O)C1CCC(N1CCOC(CNC(=O)CCC2CC2)C1)=O 44364,C1(C(=O)NCC(CN(C(C(CC#C)C)=O)CC)(C)C)Cc2cccc(Cl)c2C(=O)O1 44365,C1(NC(COCCOCCOC)=O)CN(C(=O)Cc2ccno2)C2(CCOC2)C1 44366,CCCC(O)C(CO)NC(=O)NC(Cc1ccccn1)CO 44367,c1(CC)ccc(OC)cc1C(N1CCCCC1CN(C)C(C1CCCN1C)=O)=O 44368,C1(CNC(C2C(CCC)C2)=O)CCC(CNC(C2CCC3(CC3)C2)=O)CC1 44369,C12(NC(C3CC(=C)C3)=O)CCC(CC1)N(C(=O)C(C)(C)NC(=O)OC(C)(C)C)C2 44370,C(CC1c2ccccc2CCN1C(=O)C(C)SC)NC(CCOCCOC)=O 44371,C12(C(N3CCCC(CNC(Cc4ccc(OC)cc4)=O)C3)=O)CCC(C)(C1)OC2 44372,c1(NCC2C(CC(C)C)C2)[nH]c(=NCCc2noc(C3CC3)n2)nc2ncn(C)c12 44373,N1(C(C(=O)Nc2c(C)n(C)nc2)=O)CCOC2(CC1)CCS(=O)(=O)C2 44374,C=C(C)c1ccccc1NC(C1CC12CN(C(c1cc(C(C)C)n(C)n1)=O)C2)=O 44375,C1(NC(c2c(CNC(C(CCOC)C)=O)cc[nH]2)=O)CCn2cncc2C1 44376,C1(C(=O)Nc2ccco2)CCCN(C(C2COCC2OCc2ccccc2)=O)C1 44377,c1(C(=O)NCC2CC(COC)CN2C(C2CC(C)(F)C2)=O)cc2cccnc2s1 44378,CC1(CNC(=O)CCN2CCOCC2)CCCN1C(=O)CC1(CO)CC1 44379,C1(CNC(C2C(CC)C2)=O)CN(C(c2ocnc2C)=O)CC12CC2 44380,c1(SC)cc(=NC(=O)C2CCN(C(C3CC=CCC3)=O)CC2C)[nH]n1C 44381,c1(C(C(=O)NCCCNC(C=CC(CC)C)=O)O)ccc(Cl)c(F)c1 44382,c1(OC)c(C(=O)Nc2cncc(-c3ccc(SC)cc3C)c2)ccc(Cl)c1Cl 44383,c1(C(=O)NC2C(C)N(C(=O)CCC3CCCCO3)CC2)cc(F)cc2ccoc12 44384,C=CCC(C)(C)CC(=O)N1CCN(C(=O)Cc2cc(OC)no2)CC1CF 44385,C12(C(=O)NC(c3c(C)cccc3)C)CC(C)(CN1C(c1cc(O)n(C)n1)=O)C2 44386,c1(NC(C(C)C)CNC(=O)CC2CCCOC2)ncncc1I 44387,c1(CN(C(c2csc(C)n2)C(=O)NCCOCC)C)cccc2c1OC(F)(F)O2 44388,N1(C(C(C)(C)NC(c2ccccc2)=O)=O)CC(OC(C)(C)C)CC(C(=O)O)C1 44389,C1(CCNC(C2(C=C)CC2)=O)CN(C(C2OCCC2C(F)(F)F)=O)CCS1(=O)=O 44390,c1(C(=O)NCC2N(C(C(COC)(C)COC)=O)CC2)cc2c(ncn2C)[nH]1 44391,Cc1ccc2c(c1)C(C(=O)NC1CC(NC(=O)Cc3nn(C)cc3Cl)C1)OCC2 44392,C(C(O)C(=O)N1CCC1c1cn(CC(n2cccn2)C2CC2(Cl)Cl)nn1)N(C)C 44393,Cc1cc(C)c(C(=O)N(C(C)C)Cc2cn(-c3ccc(CO)cc3)nn2)c(S)n1 44394,C1(NC(C(COC)(F)F)=O)CCC(C)N(C(c2ccc(-c3ccco3)[nH]2)=O)C1 44395,O(NC(=O)C(COC)NC(C12CC1CNC2=O)=O)CCOCC#C 44396,N1(C(C#CC2(CC)CC2)=O)CC(C)(CNC(=O)C#CC2CC2)CC1(C)C 44397,c1(NC(C2C(C(=O)Nc3ccc4sncc4c3)C2)=O)c(O)cccc1[N+](=O)[O-] 44398,N1(C(CCCNC(C)=O)=O)CCN(C(=O)C(c2ccc(Br)cc2)C)C(C)C1 44399,n1(CC=C)nnnc1C(c1ccc(-c2ccccn2)s1)NCc1ccc(CC)o1 44400,N1(C(C2(COCC)CCC2)=O)CC(C(C)(C)O)(CNC(=O)C=Cc2cn[nH]c2)C1 44401,C=CCC(CNC(C1C2CCC(C2)C1C)=O)C(=O)N(C1CCN(C(=O)CC)C1)C 44402,C1(CNC(C(C(C)C)C)=O)CN(C(=O)Cc2ccnn2C2CCC2)CC(C)(C)C1 44403,C1(NC(c2ccc(O)nn2)=O)(CO)CCCN(C(=O)Cc2ccc(O)cn2)C1 44404,Cn1cc([N+](=O)[O-])c(C(=O)NCC2(F)CCN(C(=O)CN3CSCC3=O)C2)n1 44405,c1(CC)oc(C(N2CC(CC(=O)N(CC(C)C(=O)OC)C)C(C)C2)=O)cc1C 44406,n1(CCC(=O)NC2CC(NC(c3c(C)oc(C(C)C)n3)=O)C2)ccc(O)nc1=O 44407,C1(C(N2CCOCC2)C)CCCCN(c2nc(=N)nc(N3CCC(N)C3)[nH]2)C1 44408,C1(NC(c2cc(C)ncn2)=O)CC2(C1)CC(C(=O)NCC(C)S(N)(=O)=O)C2 44409,C(=O)(C1=CCCC1C)NCC1CC(COC)CN1C(C1OCCC1C)=O 44410,C1(C(C)C)(C(=O)NCCC2CN(C(=O)C(O)C(F)F)C2)CNC(=O)C1 44411,c1(OC)ccc(NC(C2CC3CC3N2C(=O)Cc2ccccc2OC)=O)cc1C 44412,C(CCN(C)C)(C(=O)N1CCOCC1CC1CC1)NC(c1scc(C)c1)=O 44413,c1(CCC(=O)NC2CC2CNC(c2ccc(-c3cc[nH]n3)s2)=O)nc(O)n[nH]1 44414,c1(C(=O)NC(C2CC2C(=O)NCC2(CO)CC2)C)cnnn1C 44415,N1(C(C2(C#C)CC(=O)C2)=O)CCC2(CC1)CC2NC(=O)CCc1cc(C)n(C)n1 44416,C(C(=O)N1CCC(F)(C(=O)NCC2CC(OC)C2)C1)(C(C)(C)C)OC 44417,C1(C(=O)O)CC12CC(=CC(=O)NOCC1C3CNCC1C3)C2 44418,S(=O)(=O)(c1ccc(F)c(C(=O)NC2C3CC2N(C(=O)CC(C)SC)C3)c1)NCC 44419,C1(COC)(CNC(C2OCCC2C)=O)CCN(C(C2CC(OC)C2)=O)C1 44420,N1(C(C2(CC)CCCN2C(C2CCCCC2OC)=O)=O)CC(C)OC2(CCC2)C1 44421,C(=O)(C(CNC(=O)CCn1cnnc1)C(C)(C)C)NCc1cn(CC)nn1 44422,N1(C(c2c(C)cncc2)=O)CC2(C1)SCCC2NC(=O)CCCCN(C)C 44423,N1(C(COC(C)C)=O)CCC(C=CC(=O)NCC2CC(C)CO2)CC1 44424,N1(C(C2CC(C)OC2)=O)CCC2(CC1)CCN(C(c1cnc(N)c(Cl)c1)=O)C2 44425,c1(C(=O)NC(C2N(C(C(CC3CC3)OC)=O)CCC2)C)ncc(Cl)cc1F 44426,C(=O)(CC(C)P(C)(C)=O)NC(CCCC)CNC(=O)C(C)OC(C)(C)C 44427,Cc1cc(Cl)c(C(=O)NCC2(F)CCN(C(c3cnncc3O)=O)CC2)cc1C 44428,n1(CC(=O)N(C(COC)COC)C)cnc2cc(C)c(C)cc12 44429,C1(C(=O)NCC2CCN2C(c2cn(C3CCC3)nn2)=O)CCc2nn[nH]c2C1 44430,c1(C(N(CC)CC2CCCN2C(=O)CN(C)C)=O)ccc2c(c1)CCCCN2 44431,n1(COCC)nnc(C#N)c1NC(N1CC(CO)C(c2ccsc2)C1)=O 44432,CCCC(CC)C(=O)NC1(CC)CCCN(C(c2ccoc2)=O)C1 44433,c1(C(=O)NC(CN2CCN(C(C(CC)OC)=O)CC2)C)cc(C)ccc1F 44434,CCC(CC(=O)NC(C1CC1C(=O)NC(C)CC(F)(F)F)C)CC(C)C 44435,CC1(NC(=O)C(C2CCN(C(=O)Cc3csnn3)C2)F)CC2(CCC2)C1 44436,C12(CNC(c3c(C)nn[nH]3)=O)CCC(CC1)N2C(=O)C(c1ccc(F)c(F)c1)=O 44437,c1(COC)ccccc1C(N1CC(C)(NC(c2cc(Br)cn2C)=O)C1)=O 44438,Cc1cc(F)c(C(N2CCC3C(NC(=O)CC4C=CS(=O)(=O)C4)C23)=O)cc1F 44439,Cc1c(C(=O)NCC2(NC(C3CC(=O)CCO3)=O)CCC2)cncc1F 44440,c1(OC)cnc(C(=O)NCC(C)(C)OCC(=O)NCC(N)=O)cn1 44441,c1(C(N2C(CCNC(C(C)OCCCC)=O)CCCC2)=O)cc(F)c(C)cc1Cl 44442,CC1CCN(C(c2cccc3nsnc23)=O)C(C)C1NC(=O)CN1CCOCC1 44443,c1(CC)nnc(=NC2CCCC23CCN(C(=O)CC2CC24CC4)CC3)[nH]c1CC 44444,C1(C(=O)O)CC2(CCOCC2)CN1C(c1cc(N)c(O)c(F)c1)=O 44445,c1(OCC)cc(C(=O)NC(C2CN(C(=O)Cc3cn[nH]c3)C2)C)on1 44446,c1(N2CC3CN(CCCCC=C)CC32)ncnc2ccc(OC)cc12 44447,C1(CC(=O)NCCOC2CCN(CCO)C2)(CC)CNC(=O)C1.C(C(=O)NC)S 44448,C1(NC(C(=O)NCc2ccc(OCCCCOC)cc2)=O)CCC2OCCC2C1 44449,N1(CN(CCC#CC)C(=O)CCN2CCOCC2)CCc2[nH]nc(CO)c2C1 44450,c1(C(=O)NC2CN(C(c3cc(SC)oc3)=O)C(C)CC2)ccc(P(C)(C)=O)cc1 44451,N1(C(C2CC(OC)C(OC)C2)=O)CC(NC(=O)CSc2nccn2C)CC(O)C1 44452,c1(C(=O)NCC2C(NC(C(C)SC(C)C)=O)C2)cc(C(F)(F)F)ncc1Cl 44453,C12(C(c3cn(-c4c[nH]ccc4=O)nn3)O)CCC1CN(CC1=CCCCC1)C2 44454,N1(C(c2c(CC)csc2)=O)CC2CC(C(=O)NCCN3CCOC3=O)CC2C1 44455,c1(OCC(=C)C)ccccc1COC(C1(CF)CCNCC1)=O 44456,CC1CCCC(N(C)C(C2CC3(CC(NC(=O)Cn4ccnn4)C3)C2)=O)C1C 44457,C(c1cc(C)n(-c2ccc(C)cc2)c1C)=CC(=O)NCC.C1(=O)C(CC(C)C)O1 44458,C1(OC)CN(C(=NCCc2sccc2C)NCc2ccco2)CC1O 44459,C1(C(=O)NCCCNC(C(C)C)=O)CC(C)N1C(=O)C=Cc1ccoc1 44460,O=S(=O)(c1cccc2cccnc12)NCC1C2CNC1C2 44461,c1(C(=O)NC2CC(n3cc(-c4ccc(C(=O)O)o4)nn3)C2)ccc(F)cc1Cl 44462,N1(C(C(CC)N(C)C)=O)CC2C(NC(=O)CCc3cccnc3)CS(=O)(=O)C2C1 44463,C1(NC(C2SCCCS2)=O)CCC12CN(C(=O)CCn1cnnn1)C2 44464,c1(C(=O)OCC)ccc(O)nc1NCCCN(C1CCS(=O)(=O)C1)C 44465,c1(NC(CNC(c2ccc(COC)s2)=O)C)ncc(Br)cc1C#N 44466,c1(-c2nc(CCCC(=O)N(CC(CC)NC(C)=O)C)on2)c(C)n[nH]c1C 44467,C1(C(=O)NC(C(C)NC(c2ccnnc2)=O)CO)CCCC2(CCCCC2)C1 44468,c1(NC(=O)Nc2c(C)cc(Br)cc2F)c(C#N)oc2ccccc12 44469,N1(C(c2cc(C)n(C)c2C)=O)CCC(NC(=O)CCC2CC2(C)C)CC(C)(C)C1 44470,N1(C(CC2(CC(=O)OC)CC2)=O)CCC(N(C)C(C2CCC(O)CC2)=O)C2(CC2)C1 44471,C1(C(=O)NCc2ncco2)(CC)CCCN1C(=O)CCN(C)C 44472,N1(C(CCC(=O)NCCC)=O)CC2CCCN(C(=O)C=CCOC)C2C1 44473,C1(N(C)C(C2(CCNC(C3(C)CC(F)C3)=O)CC2)=O)CCCC1(F)F 44474,Cc1cnc2ccc(C(=O)NC3CCN(C(=O)CCS(C)(=O)=O)C3)cn12 44475,S(=O)(=O)(C1CCN(c2nnc(C(C)Cc3ccccc3)n2C)C1)NC 44476,Cc1ncncc1C(N1CCC(N2CCN(C(C3CCCCN3C)=O)CC2)C1)=O 44477,c1(C(N2CC(CNC(CN3CC(CC)C3)=O)OCC2)=O)cccc2ncc(C)n12 44478,N1(C(CC2CCC(=O)C2)=O)CC2(CCCC2NC(c2cccc(C3CC3)c2)=O)C1 44479,c1(C(=O)NCCCC(C)NC(c2ncc(OCC)nc2)=O)c[nH]c2nccc-2c1 44480,C1(CNC(C2CC23CCOCC3)=O)CC2(CO1)CN(C(=O)CC(F)(F)C(F)F)C2 44481,c1(C(=O)NC2CCCN(C(c3c(C#C)cn(C)n3)=O)C2C)cc2cn[nH]c2cn1 44482,C12(NC(N(C)CC3CC=CCC3)=O)CC(NC(=O)OC(C)(C)C)CC1C2 44483,c1(CC)ncnc(CC)c1C(=O)NCCN(C(=O)C(O)CC(N)=O)C 44484,CC(C(=O)NC(C)C(C)F)C(C)NC(=O)C=Cc1cscn1 44485,N1(C(c2ccn(CCOC)n2)=O)C2CC1CN(C(c1ccc(F)cc1I)=O)C2 44486,C1(C)(CC)CCN(C(C2CC2C2CN(C(C3(C)CCCN3C)=O)C2)=O)CC1 44487,N1(c2nc(CC)nc(=N)[nH]2)C2CCCC1CN(C(=O)C=C1CCCC1)C2 44488,c1(C(C(=O)NCC(CNC(c2cc(Cl)ccn2)=O)OC)=O)ccc(Cl)cc1 44489,Cc1cnn(CC(=O)NC2CN(C(c3coc(C4CC4)n3)=O)CC23CC3)c(=O)c1 44490,c1(C(N2CCN(C(COCC=C)=O)C(CO)C2)=O)cnn2cccc(Cl)c12 44491,c1(C(=O)NCC2(CNC(=O)CC(F)F)CCCC2)ccc(O)cc1F 44492,C(C)(C(=O)NC1CC(CC(=O)NCCCN(C(=O)COC)C)C1)NC(CC)=O 44493,c1(CC)cc(C(N2CCC(C3CCCN3C(C3OCCO3)=O)CC2)=O)cc(O)n1 44494,C1(C(=O)NC(c2nocc2C(=O)N(C2CCCCC2)C)C)CCC(C)(C)C1 44495,N1(C(c2ccc(CC)cn2)=O)CCCCC(CCC(=O)N(CCCO)CCCO)C1 44496,Cc1ncn(C)c(=O)c1C(=O)NCC1C(C)CCN1C(=O)C(F)=C1CCC1 44497,C1(CNC(c2csc(C(F)F)n2)=O)(CO)CCN(C(C2CC3(CC3)CO2)=O)C1 44498,c1(C(N2C(C)(CC(=O)N(C3CCOC3)C)CC2)=O)cnc(=N)[nH]c1 44499,CCC(C)C(C(=O)NOCc1nc[nH]n1)NC(c1ncc(F)cc1N)=O 44500,C1(CC=C)(NC(=O)C(COC)C(C2CC2)NC(=O)CC(=O)N(C)C)CCCC1 44501,C12(CC)CC(CNC(=O)CN(C)C(C)=O)(CO1)C2.C1(C)(CC)CC(C(=O)CC)C1.NC 44502,C1(C(=O)NCC2CC(NC(=O)CC3CCCC34CC4)C2)CC2(C1)CC1(CC1)C2 44503,N1(C(C(=O)NC2CC2)=O)CCc2c(C(N3CCNCC3)=O)cccc21 44504,c1(C(=O)NCC2CC(CC)C2)cc(CNC(c2cccnc2O)=O)ccn1 44505,Cc1cncc(C(=O)N(C)CCOCCCNC(C2CCC(N(C)C)CC2)=O)c1 44506,C(CN=c1cc(NCCc2cc[nH]n2)nc[nH]1)(c1cccc(F)c1)N(C)C 44507,c1(CC)ccnc(C(N2CCC(O)(COC)C2)=O)c1.C12(CC1)C(=O)NC2 44508,C1(C(N(CCN(C)C(c2cccnc2)=O)C)=O)CCCC2CCCN12 44509,c1(C(=O)NCCC2N(C(CC3CCN(C)C3)=O)CCC2)cn(C)ccc1=O 44510,N1(C(C(COC)(F)F)=O)CCC(C2(O)CN(C(C3CCCS(=O)(=O)C3)=O)C2)CC1 44511,CC1CN(C(c2ocnc2C2CC2)=O)CCN(C(=O)C(O)C(C)(C)C)C1 44512,c1(C(=O)NC2C3(CC(NC(CCC4(C)CC4(F)F)=O)C3)C2)ccc2nonc2c1 44513,C1(NC(c2cnn(CCC)c2C)=O)CC(C)CN(C(=O)CC2CCCC2(F)F)C1 44514,N1(C(C2(CC=C)CC2)=O)CCC2(CC1)CC2NC(=O)C(c1cc(C)cc(F)c1)C 44515,c1(SCC)ccc(Cl)cc1C(=O)NCCN(C)C(C1(O)CC2CCC1C2)=O 44516,C(=O)(CCS(=O)(=O)CC(C)C)N1CCCC(O)(CNC(C(CCC)OCC)=O)C1 44517,Cc1cccc(C(N2CCC(CN(C)C(C3CCS(=O)(=O)C3)=O)C2)=O)c1Cl 44518,c1(C(N2CCN(C(c3cc(S(C)(=O)=O)oc3)=O)CC2)=O)cccc2c1OCCO2 44519,C1(C(=O)NCCN(C(CC(=O)OC)=O)C2CCCC2)CC(O)C(F)C1 44520,c1(C(=O)NCc2c(CC)noc2C)coc2c1CN(C(c1ccc(C)s1)=O)C2 44521,C1(C(C(=O)NCC2CCN2C(c2cnc(C)cn2)=O)OC)CCC(F)(F)CC1 44522,N1(C(c2cccc(OC)n2)=O)CCc2ccc(C(=O)NCCCC(C)C)nc2C1 44523,CCC(CC)CCCC(=O)N1CC2CC2(NC(=O)Cc2nc(F)c(F)cc2F)C1 44524,c1(NC(CN(C)C)C(=O)N2CC(c3ccccc3F)(C)C2)cc(F)cc(F)c1 44525,C(=O)(C(CCOCCO)NC(C1CCO1)=O)N(CCOCC=C)C 44526,c1(C(=O)NC2C3CN(C(CSCCCC)=O)CC32)ncc([N+](=O)[O-])cc1C 44527,N1(C(C(CN(C)C)O)=O)CCC(NC(=O)CCc2cn[nH]c2)C2(CCC2)C1 44528,CC1COCC(CC(N2CCC(CN(C)C(c3cc(F)n(C)n3)=O)CC2)=O)O1 44529,c1(C(=O)Nc2cncc(C(N3CCC(CC(=O)OC)C3)=O)c2)cc(Cl)ncc1I 44530,c1(C(=O)NCC2CCCCN(C(C3(C(F)F)CCC3)=O)C2)ccc2nccn2c1 44531,c1(SC)nc(C)c(CCC(=O)NCC2CCN(C(=O)C=C(Cl)Cl)C2)c(O)n1 44532,c1(C(N2CC(O)(C(C)NC(c3cc(CC)c(C)s3)=O)C2)=O)cc2ncccc2o1 44533,C(=O)(CCS(N)(=O)=O)NC1CCN(C(CC(N2CCCCC2=O)C)=O)C1 44534,C(=O)(C(C)(F)C(C)(C)F)N1CC(C)C(CC(=O)NCC2CCC(=O)O2)C1 44535,C1(C(N(CC(CN(C(=O)CCc2nncn2C)C)O)C)=O)CCN(C2CC2)CC1 44536,N1(C(C2CC(C)(CC)C2)=O)CC2(CCCC2)C1C(N1CC(C)(C(F)(F)F)C1)=O 44537,C1(CNC(C(CC)(C)C)=O)CC2(CO1)CN(C(c1cccc(CO)c1C)=O)C2 44538,C(=O)(C(C)(C)C(F)F)N1C(CCNC(CC(C)NC(=O)OC(C)(C)C)=O)CCC1 44539,CCC(C)(CNC(C1CC(O)C(F)C1)=O)C(=O)NC(C)C1CC1 44540,C1(N(C(=O)CSc2nncn2C2CC2)C)CCCN(C(=O)CC2CCC2(C)C)C1 44541,C1(C(=O)NCCCC(CCC)Nc2ccc(COC)cn2)CC(C(C)(C)C)=NO1 44542,C1(CCNC(CN(C(C(C)C2CCC2)=O)C)=O)COC(C)(C)C1 44543,N1(C(CC=CC=C)=O)CCN(C(=O)Cc2ccc(C)c(OC)c2)CC1C(C)(C)C 44544,C12(C(N3CC(CNC(C4(C=C)CCCCC4)=O)C(C)C3)=O)C3CC(CC13)C2(F)F 44545,Cc1nccc(Cl)c1C(=O)NCCOCCN(C)C(C12COCC1C2)=O 44546,c1(C(N2CCCC(NC(C3C(C)CC(C)O3)=O)CC2)=O)ccc(F)c(Cl)c1F 44547,CC1CC(NC(=O)CN2CCCNC2=O)CCN1C(C1CC(=O)N(C)C1)=O 44548,CC1(C)OCC(CCNC(c2cccc(C(=O)NCN)c2)=O)O1 44549,N1(C(c2ccc(N(C)C)nc2)=O)CCC(NC(=O)C=CC2(C)COC2)C(C)(C)C1 44550,N1(C(c2cnc(CC)o2)=O)CCC=CC1C(=O)NCC(C#N)CC 44551,C(=O)(C1=CCC2CCC1N2C(=O)C(C#N)C(C)(C)C)NCC(C)CCO 44552,N1(C(C)C(=O)Nc2cc([N+](=O)[O-])ccc2F)CC(C)OC2(CCCCC2)C1 44553,C(=O)(CCCN=[N+]=[N-])NCC(C)(O)CNC(C1CCCN1S(C)(=O)=O)=O 44554,Cc1cc(Br)c(F)cc1NC(c1cncc(C(F)(F)CF)c1)=O 44555,c1(NC2CN(C3(c4ccccc4Br)C(CC)C3)C2)ccc(-c2nn[nH]n2)cc1 44556,C1(C(=O)OC)OC(C(=O)NC(CNC(=O)C=Cc2cnn(C)c2)C2CC2)CC1C 44557,C#CCCCCC(=O)NCc1nc(C(=O)NCCC)co1 44558,C(C#CC(=O)N(CCCCO)CC)NC(C1C(=C)C1)=O 44559,CC12CC(C(N3C4CCC3CN(C(C3C5CC(F)(F)CC35)=O)C4)=O)(C1)C1(CCC1)O2 44560,C(=O)(C1OCCc2c(O)cccc21)N1CC(CN(C(=O)CNC=O)C)OCC1 44561,C(=O)(C1COc2ccc([N+](=O)[O-])cc21)NC(CC=C)CNC(c1cnc(O)o1)=O 44562,C1(C(=O)NCC2(O)CCN(C(c3ccc(CC)s3)=O)CC2)CN2CCC1(C)CC2 44563,C(=O)(C1=CCC(C)CC1)NCCC(C(=O)NC(c1onc(C)n1)CO)(C)C 44564,c1(NC(=O)NC2CCC(C(=O)OC)C2)ccc(OC(C)(C)C)cc1 44565,C1(NC(C2C(OC(C)=O)C2)=O)CCC(C)N(C(C2CC(C)(C)C2)=O)C1 44566,C(=O)(C#CC(C)(C)C)N1CCC(C2N(C(c3cscc3Cl)C)CCC2)CC1 44567,c1(C(CNC(CCOCC#C)=O)NC(C2(Cl)CC2(F)F)=O)ccccc1F 44568,N1(C(c2c(Br)cn(CC)n2)=O)CCC2CC1CN(C(C1CCOC1)=O)C2 44569,C(N=c1[nH]c2ccc([N+](=O)[O-])cc2s1)C1(CCNC(C2CCC(C)(C)C2)=O)CC1 44570,c1(C(=O)NCC(CNC(C(C(C)OC)N(C)C)=O)CO)cc(C#N)cn1C 44571,N1(C(c2cccc(SCCC)c2)=O)CCN(C(=O)C(C)COC)C(CC)C1 44572,Cc1cc(Cl)ncc1NC(C1CCCCN1C(=O)Cn1ccc(C)n1)=O 44573,CCCCCC(=O)N1CCCC1(C)CNC(C1(F)CCN(C(C)(C)C)C1)=O 44574,CCC(C)(C)CCCC(=O)N1CCC2(NC(c3coc(Br)c3)=O)CC2C1 44575,c1(C(=O)NCC2C(NC(c3c[nH]cc3Br)=O)CCC2)cc2nn[nH]c2cc1F 44576,Cc1ccc(N2CCC(NC(=O)NCCC3CC3)C2=O)cc1 44577,N#Cc1cc(-c2ccc(CNC(c3ccc(OC(F)F)cc3F)=O)cn2)cc(F)c1 44578,C1(CC)CN(C(=O)C(=Cc2cccnc2)F)CCN1C(c1cc[nH]c1C(C)C)=O 44579,C1(C(=O)NCC2CCCCN2C(=O)C2=COCCC2)CCC2(CCC2)CO1 44580,c1(OCC)ccc(C(=O)NCC(C)CN(C(=O)COCCCF)C)cc1C 44581,C1(C(=O)NC(CC(C)C)c2cccs2)C(C=C(C)C)C1(C)C 44582,C(C)(C(C(=O)NCc1cc(O)ns1)NC(c1nonc1C)=O)OC 44583,c1(C(=O)NCC2(F)COCCN(C(C(CC)(C)O)=O)C2)cccc2nc(O)[nH]c12 44584,c1(C(=O)NC2C(CNC(CCCOC)=O)COC2)nccnc1C(N)=O 44585,C(=O)(C(=O)C(C)(C)C)N1CCC(C)C1C(N1CCC1(C)CCO)=O 44586,N(C1CCCc2n[nH]cc21)C(C1N(C(CN2CCC(OC)C2)=O)CC(O)C1)=O 44587,c1(C(=O)OC)ccnc(C(=O)NC2CN(Cc3ccnc(Br)c3)C2)c1 44588,c1(C(N2CC(C(C)NC(C(COC)O)=O)OCC2)=O)cncc(N=[N+]=[N-])c1 44589,c1(CC)cc(NC(=O)C(CNC(c2cnc(C)s2)=O)OC)cc(O)c1 44590,C1(CC(=O)OC)CCN(C(c2csc(NC(=O)C(C)COC)n2)=O)CC1 44591,c1(C(CNC(CC(=C)C)=O)NC(c2cccc(C3CC3)c2)=O)cc(F)cc(Cl)c1 44592,c1(C(=O)NCC(C)NC(C2C3CCC23)=O)ccc(NS(=O)(=O)CC)cc1 44593,C1(NC(C2C(NC(C=CC(=O)N(C)C)=O)C=CCC2)=O)CCCN(C)C1=O 44594,c1(C(=O)NCCC2N(C(CCOCC(C)C)=O)CCC2)ccc(NCCO)cc1 44595,CC1(C)OCCc2cc(C(N3CCS(=O)(=O)C4CCCCC34)=O)ccc21 44596,C1(C(N(CCCC)CCCC)=O)CCCCN1C(C1CCC2CC12)=O 44597,C1(C)(NC(CC(C)c2cccnc2)=O)CCCN(C(c2cnc(O)n2C)=O)C1 44598,C(=O)(C(C)(C)CC#N)NCC1(OC)CCN(C(c2ccnnc2)=O)C1 44599,n1(C(C)C)ncc(Cl)c1C(=O)NC1CCC(C)(CN)C1 44600,c1(OC)c(C(=O)NCC2(F)CC(CNC(=O)C3=CCCC3C)C2)cc(Cl)cc1Cl 44601,Cc1nc(C)c(C(N2CCC(C)(CNC(c3scnc3C3CC3)=O)C2)=O)[nH]1 44602,N1(C(C(C(C)C)SCC)=O)CCN(C(C2CC(C)CCO2)=O)CC1CC(F)F 44603,Cc1cc(C(N2CC=CC(NC(=O)CN(C3CCCC3)C)C2)=O)c2c(c1)CCC2 44604,C12(C(=O)NC3CC(C(F)C(=O)NCCCN4CCCC4=O)C3)CCC(CC1=O)C2 44605,N1(CCCCNC(c2cc(-c3cccnc3)no2)=O)CCC(C(=O)O)CC1 44606,C(=O)(C1=CC(O)C(NC(c2cnn(C3CC3)c2)=O)C1)N(C1CN(C)C1)C 44607,C1(C(N2C3CC(CNC(C(COC)C)=O)C2CC3)=O)Cc2ccccc2C(=O)O1 44608,N1(C(c2cn(SCC)nn2)=O)CC(C2CCN(C(C3(O)CC(C)(C)C3)=O)CC2)C1 44609,C1(NC(c2cccc(OC)n2)=O)CCCCN(c2cc(-n3ccnc3)ncn2)C1 44610,n1(CC(=O)NC2(C)CC(NC(c3n[nH]cc3Cl)=O)C2)ccc2ccc(F)cc12 44611,S(=O)(=O)(CC(C)C)NC(=O)NCC(C=CC)(O)CO 44612,C12(NC(c3ccc(CC)nc3)=O)CC(CNC(=O)Cc3[nH]cnc3C)(C1)OC2C 44613,CN1CC(O)CC1(C)C(=O)NCC(C)(C)NC(C1CC(S(C)(=O)=O)C1)=O 44614,N1(C(C2(C)CC3(CC3)C2)=O)CCN(C(=O)CNC(=O)C2CC2)C(CC(F)(F)F)C1 44615,c1(C(C(=O)NC2CC2)N(C)Cc2c(C)n(C3CC3)nc2)ccc2c(c1)C=CCC2 44616,N1(C(C2C(C(C)C)OCC2)=O)CC2C(NC(c3sccc3OC(F)F)=O)C2C1 44617,C1(C(C(=O)NCCC(=C)C)F)CCN(C(=O)C=CCCC)C1 44618,CC(C)(C)C(CO)C(=O)NC1CCC(NC(c2ccc(F)o2)=O)CC1 44619,c1(C(=O)NC2(CC=C)CN(C(C3NC(=O)CC3C)=O)C2)ccc(C(C)C)nc1C 44620,C1(NC(c2ccc(C(F)F)cc2)=O)CCN(C(=O)Cc2cccnc2)C12CCC2 44621,C#Cc1ccccc1.C(=O)CCCC=C.C(=O)CCCC 44622,C(CCCCC(=O)N(C)CCC1CCCN1C)NC(C1CC(C(C)C)C1)=O 44623,Cc1cc(C(N2CC(NC(C3(C)C=CCC3)=O)C(C)(C)C2)=O)ncc1C(F)F 44624,N1(C(c2n(C)cnc2)=O)CC(C(=O)Nc2cn(C)nc2C2CC2)CC12CCC2 44625,C1(O)(C(=O)NC2(C3CCNC3)CC2)CN2CCCC1C2 44626,C1(CNC(c2cccn2C2CC2)=O)CCN(C(c2cn3c(n2)CCC3)=O)CC1O 44627,N1(C(C2CCCC(C)CC2)=O)CCCC2(C1)CN(C(c1ccnc(S)c1)=O)C2 44628,C(=O)(CC(C)(C)CNC(C1CC(F)(F)C1)=O)NCC(C)(C)C(F)F 44629,C(CC(=O)NCc1ccc(F)nc1C)(C(C)(C)C)NC(C(C)N(C(C)=O)C)=O 44630,Cc1cc(S(N)(=O)=O)oc1C(N1CCN(C(=O)COC2CCOC2)C(C)C1)=O 44631,CC1CC(C)(C)N1C(C1CCN(CC(C2CC3CC3C2)=O)C1)=O 44632,C(=O)(C(C)(O)C1CCC1)NCC(C)CN(C)C(C1(Br)CC1)=O 44633,N1(C(CC2(OC)CCC2)=O)CCCCC1C(=O)NC1CC(C)(O)C1 44634,C1(NC(CCc2nnc(C)n2C)=O)CCCC(NC(c2cc(Cl)n(C)n2)=O)CC1 44635,CC1(C(=O)NCC#CC(=O)NCC2(CO)CCOC2)CCC(=O)C1 44636,N1(C(COc2cc(C)c(F)cc2)=O)CC2CCN(C(c3csnn3)=O)CC2C1 44637,C1(N(C(c2cc(C)n(C3CC3)n2)=O)C)CN(C(=O)C(C)c2cccs2)CC12CC2 44638,c1(-n2cc(CN3CCN(C(C4C(OC)C4)=O)CC3)nn2)cnnc(O)c1Br 44639,C(=O)(C(C(C)(C)C)n1cc(C(C)N(C)C)nn1)NC1C(OCC)C2C1CCC2 44640,c1(CC(=O)NCC#CCNC(=O)CCc2nncs2)c(F)cccc1Cl 44641,C1(CN(C(C2COC(=O)O2)=O)CC)CCCCN1C(C1CC(O)CN1C(C)=O)=O 44642,c1(C(N2CC(C(=O)NC3(C(=O)OC)CC(O)C3)C2)=O)cc(S(N)(=O)=O)sc1Cl 44643,C1(C(N(CC(=O)NCC2CCCC(F)C2)CC)=O)CC2(CSC2)C1 44644,N1(C(C=CC(C)(C)SC)=O)CCCC12CCN(C(C1CCN(CC(C)C)C1)=O)C2 44645,N1(C(C2CC(OC)C2)=O)CCN(C(c2ccc(SC)s2)=O)C(C)CC1C 44646,C=C(C)CCCC(=O)NC1(CNC(c2cc(F)ncc2OC)=O)CCCCCC1 44647,Cc1cc([N+](=O)[O-])cc(C(=O)NC2CN(C(=O)CCC3(C)CC3)CCC2F)c1Cl 44648,C(=O)(C1COc2ccc([N+](=O)[O-])cc21)N1CC(C)N(C(C2CCCCC2)=O)CC1 44649,c1(C(=O)NCc2c(C3CN(C(c4c(C)n[nH]c4)=O)C3)ocn2)coc(C#N)c1 44650,C(=O)(C#CC(C)(C)CNC(c1cnn(C(C)C)n1)=O)NC(C#C)CC1CC1 44651,c1(C(=O)OCC)ccc(NC(C(N2CC3(CC(NC)C3)C2)=O)C(C)C)nc1C 44652,C(=O)(C(C)(C=C)CC)NCCC(=O)NC(CC=C)C(=O)OCC 44653,c1(C(N2C(C)CC(CNC(=O)OC(C)(C)C)C2)=O)ncc(Cl)cc1F.NC 44654,C=C1COc2c(C(=O)NCCC(C)NC(C3(Br)CC3)=O)cnn2C1 44655,C1(C(N(CC(CN(C(CN(C(C)=O)C)=O)C)O)C)=O)CCCCCN1C 44656,CC1COc2ccc(C(=O)NC3CC(NC(=O)CO)C3)cc21 44657,C1(CC(=O)NC2(CC)CCCCC2)CCCN(C(=O)C(O)C2CC2)CC1 44658,C1(COC)(NC(C2C=CC=CC=C2)=O)CCN(C(=O)Cc2cn(C)nc2Cl)C1 44659,c1(C(=O)NC2C(C(N3C(C)(C(C)=O)CC3)=O)C2)ccc(Br)c2cccnc12 44660,C1(CC#C)(C(=O)NCC(O)CNC(c2conc2C2CCCC2)=O)CCCCO1 44661,Cc1cc(N)c(C)nc1C(=O)NCC(C)(C)NC(=O)COc1c(C)cccc1Cl 44662,c1(CC(=O)NCC(O)CCNC(c2sccc2F)=O)csc2c(F)cccc12 44663,c1(OC)cccc(C(=O)NCC2(F)CCN(C(=O)CC3C=CCC3)C2)c1F 44664,N1(C(CC(=O)OC(C)(C)C)=O)CCCC12CCCN(C(=O)C(F)(F)C1CC1)CC2 44665,c1(OC(CC)C)cc(CN2CCC(C(=O)N(C)C(C)C)CC2)ccc1OC 44666,C(=O)(C1CCCc2nncn21)NC(C)CCNC(c1cnc(O)c(Br)c1)=O 44667,Cc1c(CC(=O)NC(C)CNC(=O)C=Cc2cncs2)ccc(Cl)c1Cl 44668,C#Cc1ccc(C(=O)N(C(C)CCNC(C2CC(F)C2)=O)C)cc1C 44669,Cn1cc(C(C(=O)NC2CCC2(C)C)NC(=O)Cc2cn[nH]c2)nn1 44670,CS(=O)(=O)c1cnn(CC(N2CCCC2CCCNC(C2CCC3CC23)=O)=O)c1 44671,C1(C(=O)NCCCN(CCCNC(CCN(c2ccncc2)C)=O)C)CC2CC1C2 44672,N1(C(C2(COCC)CC2)=O)CCC2(CC1)CCN(C(C1(C)CCNC1=O)=O)C2 44673,c1(OC)cc(CCC(N2CC(NC(=O)C(N)=O)C(O)C2)=O)ccc1Cl 44674,Cc1cnc2nc(C(=O)NC3(C)CCN(C(c4cc(C)nnc4O)=O)C3)nn2c1 44675,Cc1cc(C)nc(SCC(=O)NC(C)C(CO)NC(C2(F)CC=CCC2)=O)n1 44676,C=CC1CN(C(C2CC3(CCC3)C2)=O)CC1NC(c1cn(CC)nc1C)=O 44677,C1(C(N(CC(C)C#N)C2CC2)=O)CCN(C(c2ccco2)=O)CC1 44678,n1(CC)cc([N+](=O)[O-])c(C(=O)N(CC(C)NC(=O)Cc2cc(C)cs2)C)n1 44679,C1(NC(COc2cc(C)on2)=O)CN(C(c2cnn(C(C)C)c2C)=O)CCC1F 44680,C#CCC(C)(C(=O)NC(c1nn(C)cc1O)C)NC(=O)C(C)=CC 44681,c1(C(=O)OCc2cccc(C(F)(F)F)c2F)nnn2c1COCC2 44682,Cc1ccc(CCC2CCN(C(=O)C(=O)N(C)CC3CC3)CC2)cc1C 44683,CN1C(=O)NCC1C(=O)NCCOCCNC(C1OC2CCC1C2)=O 44684,N1(C(C(CC)=CCCC)=O)CCN(C(C23CC(C)C2C3)=O)C(c2nccn2C)C1 44685,C1(C)(CCNC(C2CCC(C)O2)=O)CCN(C(c2cnccc2Cl)=O)CC1 44686,c1(CC(=O)OC2C(n3c(C)ccc3C)CCCC2)c(Br)ccc(F)c1F 44687,C(CCO)(CC(C)C)NC(c1cc(CNC(c2ccc(COC)o2)=O)nn1C)=O 44688,C1(CN(C(=O)CC2OCCO2)C)CCC(CNC(=O)Cc2csc(Cl)c2)CC1 44689,C(CCS(=O)(=O)c1ccccc1)OC(CC1CCCC(C(=O)OC)C1)=O 44690,c1(C(N2C(C)C(NC(C3CCC=CO3)=O)CCC2)=O)cc2ccccc2s1 44691,CCC1=C(C(=O)N2CCN(C(C3CCOC3CC)=O)C(C3CCC3)C2)CCCO1 44692,C1(C(=O)NCC(C)(C)CCNC(=O)C(O)C(F)(F)F)CCCC2(CCC2)O1 44693,C#CCCCC(C)C(=O)N1CCCC1(CNC(c1sccc1OC)=O)COC 44694,C(C(C)(F)C(C)(C)F)NC(C1CC(C)N1C(c1ncnc(O)c1F)=O)=O 44695,C(=O)(CC(Cc1cccc(Br)c1)NCc1cnc(-c2ccco2)s1)OC 44696,c1(OC)cc(CCNC(=O)C(C)Cc2ccc(Cl)c(Cl)c2)cc(Br)c1 44697,c1(C(N2C(C)C(NC(c3csc4cncn34)=O)CCC2)=O)cccc2oncc12 44698,S(=O)(=O)(c1ccc(C#N)c(N2CC=C(Br)CC2)c1)NCc1ncc(CC)s1 44699,Cc1cc(CCC(=O)NCCC(C)NC(=O)C(C(C)C)c2cccnc2)n(C)n1 44700,N1(C(C2CNC(=O)O2)=O)CC2CCCC1C2c1cn(Cc2c(F)cccc2Cl)nn1 44701,Cc1ccc(F)c(N)c1C(=O)NC(CCN(C(=O)C(C)n1ccnc1)C)C(C)C 44702,C(C(=O)N1CC(O)CC1CC(=O)NC1CC(CC(=O)OC)C1)(C(C)C)OCC 44703,N1(C(C)=O)C2CCC1CN(C(=O)Cc1ccccc1)C2.C(=O)(CNC(N)=O)N(C)C 44704,N1(C(C2C(OC)(OC)CC2)=O)CCN(C(=O)CCCOC(C)=O)CC1CF 44705,N1(C(=O)NC(=O)OC(C)(C)C)CC2(CCC2)CC1CO.C1CSC1 44706,C(C(CO)C(F)(F)F)NC(c1sc(Cl)cc1Br)c1n(CCOC)nnn1 44707,N1(C(=O)COCC2CCC2)CCOCC1CNC(C1(CO)CCCO1)=O 44708,N1(C(CC2CCC(=O)NC2)=O)CC2CCN(C(c3cnc(C4CC4)o3)=O)CC2C1 44709,N1(C(C(C=C)c2ccccc2)=O)CCC(CC)C1CNC(c1cnc(S)n1C)=O 44710,Cc1c(C(=O)NCC(C)NC(c2ccsc2C)=O)ccc2cncn12 44711,C12(C(N3CC(NC(C=CC4N(C)CCC4)=O)C(CO)C3)=O)CCCCC1CCC2 44712,c1(C(=O)NC(CN(C(=O)C(C)CC2CCCC2)CC)C)cccnc1C 44713,C(=O)(C1CCCc2c[nH]nc21)NC1C(CNC(CSCC(C)C)=O)COC1 44714,C1(NC(C(=O)NCCOC)=O)C=CCN(C(=O)C(O)Cc2ccc(OC)cc2)C1 44715,N1(C(CC(=O)OCC)=O)CC(NC(c2ccc(C(C)C)o2)=O)CC2(CCC2)C1 44716,C1(NC(c2c(C)nn[nH]2)=O)CN(C(=O)CCSC(F)(F)F)CCC1F 44717,Cc1nnc2n1CCC(NC(c1cccc(I)c1)c1nnnn1C1CC1)C2 44718,Cc1ccc(C(C)C)cc1C(=O)NCC1CCN(C(c2coc(C3CC3)n2)=O)C1 44719,C1(CNC(c2n(C=C)ncc2)=O)CC(C)(C)CN1C(c1cc(C#N)oc1C)=O 44720,C1(CCNC(C(c2nccs2)N(CCOc2ccccc2)CC)=O)CCCCC1 44721,C#CC1CN(C(c2sc(Br)cc2C)C(=O)NC(C)(C)CC)CC1O 44722,CC1CN(C(=O)C=Cc2cccnc2)CC(C)N(C(c2cscn2)=O)C1 44723,N1(C(C(C=CC)O)=O)CCC=C(C(=O)NC2CCCCCC2)C1 44724,c1(C(=O)NCC2(CNC(C3(C#N)CC3)=O)CCCCC2)ccc2nnn(O)c2c1 44725,N1(C(c2ccc(OC)s2)=O)CC2(CNC(c3snnc3C)=O)CCC1CC2 44726,c1(NC2C(NC(c3cc(C)n(C)n3)=O)CS(=O)(=O)C2)ncc(S(C)(=O)=O)cc1Cl 44727,C(C(=O)NCCC1CCN(C(=O)C(CC)N(C)C)C1)(C(C)C)NC(COC)=O 44728,C=CCC(F)(F)C(=O)N1CCCC1C(=O)NCC(O)Cn1cccn1 44729,Cc1cc(C(c2nnnn2C2CCOC2)NC2CCC(F)(F)CC2)cc(C)c1Br 44730,N1(Cc2c(C)nncc2)CC2CC1CN2C(=O)C(=O)N(c1ccccc1)C 44731,C1(NC(c2ccc(COC)cc2)=O)CCN(C(c2cc[nH]c2)=O)CC1CC1CCC1 44732,c1(C(N2CCN(C(C(CCC)=CCC)=O)CC2C2CC2)=O)ccc(C#N)cc1C 44733,O=C(C1=CC2CC=CCC12)NCC=CCNC(C1(O)CC(F)(F)C1)=O 44734,C1(F)(CNC(c2cc(C)[nH]n2)=O)CCC(NC(=O)C(C)Cc2ccccc2Cl)C1 44735,C1(NC(c2c(CC)cc(F)cc2)=O)COC2(CCN(C(=O)Cc3ccon3)C2)C1 44736,c1(CN2C(CC(=O)Nc3c(C#N)cc(Cl)cc3)CCCC2)cc2cc[nH]c2cn1 44737,CC1CCC(NC(c2cnnn2C)=O)CN1C(c1ccc(Cl)c(C(F)(F)F)c1)=O 44738,N1(C(C(F)=C(C)C)=O)CCCCC2(CCN(C(c3ccn(CCO)c3C)=O)C2)C1 44739,C1(C(=O)NCCCCCNC(C(C)OCCOCC)=O)CC2CC1CC2(F)F 44740,N1(c2nc(NCCC(C)F)c3c(n2)scn3)C2CCC1c1cncnc1C2 44741,c1(-c2c(CN(c3ncncc3Br)CC)cc(C(F)(F)F)nc2)c(C)cc(Br)cc1C 44742,N1(C(C2(C)CCNC2=O)=O)C2CCC(C2)C1C(N1CCC(OCC(N)=O)C1)=O 44743,N(C(=NCCN(C)C)NCC1CCS(=O)(=O)N1C)C(C1(C)CCCCC1)C 44744,C1(NC(COc2cc(C)on2)=O)CN(C(=O)C(C)C2CC2)CC1C(F)F 44745,CC1(C(=O)NC(CCCNC(=O)C=CCO)c2ccccc2)CCC(=O)N1 44746,CC(N=[N+]=[N-])C(=O)N1CCCC1C(C)NC(C1C2CCCOC12)=O 44747,CC(C)(C)CC(F)C(=O)NC1(C)CCCCC1C(=O)NCc1ncc(CO)[nH]1 44748,C1(NC(C(C)Cn2ccnc2)=O)CC2(CCN(C(=O)C3=CCCC3)CC2)C1 44749,C1(OC)CCC(NC(=O)C(c2ccoc2)NC(=O)CC2CCCO2)C1 44750,C1(OC)CCN(C(C2(CCNC(C3(C)CSC3)=O)CC2)=O)C1C 44751,C1(O)(CNC(c2cc(C(F)(F)F)cc(O)c2)=O)CCCN(C(=O)C=CBr)C1 44752,c1(OC)c(C(=O)NCCC2COCCN2C(=O)C(F)n2cccn2)csc1C 44753,C(=O)(CC1=NN(C)C(=O)C1)N1CCC2(C(C(=O)NC(CCOC)CO)C2)C1 44754,c1(N2CC3N(C(c4c(C(=O)N(C)C)cccc4)=O)C3C2)ncc2ccc(Br)cc2n1 44755,N1(CC2(C)CCC2)CCC(NC(=NCC2CCCO2)NC2CCCCC2)CC1 44756,N#CC1(CCC(=O)NCCn2cc(C3(CO)CC3)nn2)CCC1 44757,c1(OCC(=O)OC)ccc(S(=O)(=O)NC(C)(C)CCC(=O)O)cc1OC 44758,n1(CC)cc(Br)c(CC(=O)NC2CC2CNC(=O)Cc2cncs2)n1 44759,CC(C)(C)CC(CO)NC(=O)CCCNC(=O)CC1CC(C2CC2)C1 44760,c1(C(N2CCC(c3ccccc3F)C2)=O)ccc(-n2ccnc2)cc1[N+](=O)[O-] 44761,C1(C(=O)Nc2ccc(C)nc2)(CC)CCN(C(C2CC2(Cl)Cl)=O)CC1 44762,Cc1ccc(S(C)(=O)=O)cc1S(=O)(=O)NC(CO)CCO 44763,c1(NC(C2CC(NCc3cc(C(=O)O)cc(Br)c3)C2)=O)nccc(Cl)c1Cl 44764,O=C(CCS(=O)(=O)CC1CCC1)NCCOC1CCOC1 44765,N1(CC)CCCC1C(=O)NCCCN(C)C(c1cc(C(=O)OC)co1)=O 44766,c1(C(=O)NCC2CC(NC(CC3CCC(C)C3)=O)C2)csc(=NC2CC2)[nH]1 44767,c1(OC)cc(OC)cc(C(=O)NC(CNC(=O)CC2CC23CC3)CCOC)c1 44768,C1(C(NOC(CC)C)=O)CN(C(C2CC3CCCC3C2)=O)CCN1C 44769,N1(C(Cc2ccc(OCC)cc2)=O)CCC(NC(c2cc(F)n(C)n2)=O)C(F)C1 44770,S(=O)(=O)(c1ccc2[nH]c(=NCC(C)(C)C(F)F)sc2c1)NCc1c(OC)nsc1 44771,c1(C(=O)NC(C)CN(C(=O)Cc2c[nH]nc2O)C)ccc(O)cc1F 44772,n1(CC)c(C(=O)NC(C)C(C)NC(c2ccoc2Cl)=O)nc2ccccc12 44773,N1(CC(CC)Oc2cccc(F)c2)CC2CN(C(C3C4COCC34)=O)CC2C1 44774,c1(C(c2ccccc2)C(=O)OCc2cc(C3CCC3)[nH]n2)ccccc1F 44775,C1(CC(=O)N(C)Cc2nnc(CC)o2)CCCC(NC(c2cscc2C)=O)C1 44776,c1(C(=O)NCCCOCCNC(C=C(C)C)=O)cc([N+](=O)[O-])sn1 44777,C#CCC(C)(C(=O)C1C(CNC(=O)NC)C1)NC(=O)C(C)OCCN(C)C 44778,c1(C(=O)OC)cccc(CC(C)C)c1.CCC1CNC(=O)N1 44779,N1(C(C(C(COC)C)C)=O)CCCC2(C1)CN(C(=O)COc1cccc(F)n1)C2 44780,c1(SCC(=O)NCC2N(C(c3cn(CC)nn3)=O)CC2)ccc(C)cc1C 44781,c1(C(N2CCCC(CCNC(CC(C)SC)=O)C2)=O)cnn2c1S(=O)(=O)NCC2 44782,c1(C(N2CCC(C(C)NC(c3cc(C)n(C(C)C)n3)=O)C2)=O)cccc(N)c1C 44783,N1(C(C(CC)(F)F)=O)CCC(C2(NC(=O)C3=CCSC3)CCC2)CC1 44784,C1(C(N2C(C(=O)NCCCC(C)O)CCCC2)=O)CC2CC1CC2O 44785,N(C)(S(=O)(=O)N1CCC(C)(N)C1)CCCN(C)C 44786,N1(C(c2ncnc(C)c2C)=O)CCCC2(NC(C34CC(F)(C3)C4)=O)CC2C1 44787,N1(C(C)=O)CCc2cc(NC(=O)NCCCN(C)C(C3CCNC3=O)=O)ccc21 44788,C1(CNC(CNS(NC)(=O)=O)=O)CN(C(c2ccc(C)nn2)=O)C2CCCCC12 44789,C(=O)(CCCC(CC)NC(=O)CCc1ccoc1)NC(C#C)(C)C1CC1 44790,C(=O)(C(C)(C)C(=O)NCC1CCC1NC(c1occc1C(C)C)=O)NC 44791,N1(C(C(C)N(C)C)=O)CCCC1(C)CNC(C1CCCC2CC12)=O 44792,c1(CN(CCCC)C(C2CCC(C(=O)OC)CC2)=O)cccc(S(N)(=O)=O)c1 44793,c1(-c2nnn(CC(N3CCCC3C3CC3)=O)n2)ccc(Br)cc1 44794,N1(C(Cc2nn(C)c(Cl)c2)=O)CCC(C2CN(C(=O)CC(=O)NC3CC3)C2)CC1 44795,C1(CNC(c2ccc(C)o2)=O)N(C(c2ccc(F)c(Cl)c2)=O)CCC1(C)C 44796,Cc1nc2nccc(C(N3CC(C)CN(C(c4ccn(C)c4)=O)C(C)C3)=O)n2n1 44797,N1(C(c2nc(C(=O)OCC)sc2)=O)CCCCC(CNC(C2CCCO2)=O)C1 44798,N1(C(Cc2ccn(C)n2)=O)CCC(CO)(CNC(C2CCCC23CC3)=O)CC1 44799,S(=O)(=O)(c1ccc(NCCC(C)CC(C)(C)C)c(C#N)c1)N1CCC(CSC)C1 44800,c1(C(N(C2CCCC2)CCCNC(C(C)=C2CC2)=O)=O)cccc(C(C)(C)C)c1 44801,Cc1ccc(C(=O)NCc2nc(C(=O)N(C(C)(C)CO)C3CC3)c(C)o2)cn1 44802,c1(C(=O)NCC(C(C)C)NC(=O)C(F)C2CCCC2)cnn2cccnc12 44803,CCC(CC)C(C(=O)NCC(C(C)(C)C)NC(=O)C=Cc1cnccn1)OC 44804,CCC(C(=O)NC(C1(O)CN(C(c2cc(C)cs2)=O)C1)C)N(C)C 44805,N1(C(C2C(=C)C2)=O)CCC2(NC(=O)COc3ccccc3OCC)CC2C1 44806,CCC(CNC(=O)CNC(c1ccccn1)=O)(CC)NC(=O)C(C)C#N 44807,C(CCC(O)C(=O)N1CCCC(O)C1)NC(c1c(CC)ocn1)=O 44808,O=C(O)CC(C(=O)O)NC(C12CC(n3cc(-c4ncccn4)nn3)C1C2)=O 44809,c1(C(=O)NC2(C)CCCN(C(C(F)=CCC)=O)C2)ccc(C(C)C)c([N+](=O)[O-])c1 44810,Cn1nnc(C(=O)NCCCC(C)(C)NC(C2CC3(CC3)C2)=O)c1C(F)F 44811,C(=O)(C1=CCCSC1)NCc1cncc(C(=O)NC(CCCC)CC)c1 44812,O=C1C2CC(F)(F)CCN2C(=O)N1CCCn1cc2ccccc2n1 44813,Cc1cn2c(n1)CC(C(=O)NC(C)CC1CN(C(=O)CNC=O)C1)CC2 44814,n1(CC(=O)N(C2CCN(C(CC(C)(F)F)=O)CC2)CCO)ccc(O)nc1=O 44815,c1(-n2cc(COCC3CN(C(C4CCO4)=O)C3)nn2)cnccc1C(F)F 44816,C(=O)(CCCS(N)(=O)=O)NC(C1OCCN(C(c2ccc(CC)cc2O)=O)C1)C 44817,c1(C(=O)NCC(C(C)(C)C)NC(c2c(OC)cncc2)=O)n[nH]c2c1CCOC2 44818,Cn1nc(Br)cc1C(=O)NCC1CCC(NC(C2OCCO2)=O)CC1 44819,C1(C(C(=O)N(CCNC(c2ccc(C(C)O)cc2)=O)CCO)O)CCC(C)(C)CC1 44820,CC1CN(C(c2cncn(C)c2=O)=O)CCC1N(C)C(c1ccc([N+](=O)[O-])[nH]1)=O 44821,C(C)(CCC(=O)NCCOCCCNC(C1(c2ncccc2Cl)CC1)=O)OCC 44822,C1(F)(CNC(c2c(COC)cc[nH]2)=O)CCCN(C(C2CCCC3(CC3)C2)=O)C1 44823,N1(C(C(C)OCCCC)=O)CCCC(CCNC(C2(O)COC2)=O)C1 44824,C1(CN(C(CC2(OC)CCC2)=O)C)CN(C(=O)CC2(OC)CCC2)CC12CC2 44825,N1(C(Cc2cc(C)on2)=O)CCN(C(c2ccc(O)cc2C(F)F)=O)C2CC12 44826,N1(C(c2c(CNC(C(CCSC)O)=O)cnn2C)=O)CCN(C)C(=O)C1 44827,C(=O)(CCCC(F)(F)F)N(C)CCN(C(=O)C(C1CCCCCC1)F)C 44828,c1(CCC(=O)OC(C)=O)nc(O)c2c(C)c(C)sc2n1.C1(=O)C(C)N1CCCC 44829,C1(NC(C(CC=C)NC(C)=O)=O)CC2CCC1CN2C(=O)C(C)OCC(C)C 44830,C12(CNC(CC(C(C)C)C)=O)CCC(NC(=O)COC(F)F)(CC1)CO2 44831,N1(C(C2(NC(CCCNC(N)=O)=O)CCSC2)=O)CC(CO)C(C2CC2)C1 44832,C1(CC)(NC(=O)C2=COCC2)CCCN(C(C2(C)CCCCO2)=O)C1 44833,C1(NC(C(C(C)C)(C)C)=O)CCC(C)(C)CC1CNC(=O)Cc1nncn1C 44834,C12(CC(=O)NC3CC(N(C(C(CN(C)C)N(C)C)=O)C)C3)CCC(CC1)C2 44835,C(=O)(CCCCC(=O)N1CC(C)(C)CC1CNC(c1cnc(F)c(F)c1)=O)NC 44836,N1(C(=O)NCc2nc(=N)[nH][nH]2)CCNCC1c1cccc(Cl)c1 44837,c1(C(=O)OC)ccc(C(C)OC(=O)CCNc2ccc(C(C)(C)C)cc2)cc1 44838,N1(C(C(COC)(F)F)=O)CCCCC(N(C(=O)Cc2cnn(C)c2C)C)C1 44839,N1(C(CN2CCN(C)CC2)=O)Cc2nccn2CC(NC(C2CCSCC2)=O)C1 44840,c1(CNCCCC(=O)NCC(CO)NC(CSCC#C)=O)ccc(Cl)cc1 44841,C1(C(=O)Nc2cccc(CNC(C(C(=O)OC)OC)=O)c2)CCC2(CC1)CC2 44842,N1(C(C(C2CC2)OCC)=O)CCC(CC(N2CCCC2C(=O)OC)=O)C1(C)C 44843,N1(C(Cc2c(C)nc(C)s2)=O)CCCC(N(C)C(c2cnc(C3CC3)[nH]2)=O)CC1 44844,C(CCC(=O)NOC(Cn1c(C)nnn1)=O)C(C)C.N(C)C 44845,N1(C(c2ccc(CSC)cc2)=O)CC(NC(=O)COC(C)C)C2(CC2)C1 44846,C12(C(=O)NC3(CO)CCN(C(c4ccc(O)nn4)=O)C3)CCCN(CCC1)C2 44847,C(CC(C(=O)NCCN(C)CCF)NC(=O)CC(O)c1ccccc1)OC 44848,CCC(C)(CNC(=O)CCC1CCCCO1)C(=O)N(C)CC1(N(C)C)CCC1 44849,O=C(C1=CCOC1)NCC1CN(C(=O)COc2ccc(F)cc2)CC1O 44850,C(=O)(CCCC(=O)C1CC1)NC(C(=O)NCCc1nnc(C)s1)C 44851,c1(SC)cccnc1C(N1CCC(NC(c2cnc(O)o2)=O)CC1)=O 44852,N1(C(C(CC=CCC)C)=O)CCC2(CCC2NC(c2ccoc2C)=O)CC1 44853,N1(C(C(n2ccc(C)n2)C)=O)CCCCCCC1C(=O)NCc1cn(C)nc1C 44854,C(CC1CC1)(CC(=O)NCc1noc(C(N)=O)n1)NC(c1c(C)scc1)=O 44855,CCC(C)C(C(=O)NC1(CNC(C2CC(C(=O)OC)=NO2)=O)CCCC1)OC 44856,c1(C(=O)NCC23CC2CN(C(=O)Cc2nc[nH]n2)C3)cc2ccc(F)cc2[nH]1 44857,CC(CC(F)(F)F)C(=O)N(CCCCN(C(=O)C(CO)C(C)(C)C)C)C 44858,c1(-c2ccc(C(=O)NC(CCCNC(CS(CC)=O)=O)C)s2)c(C)cccc1C 44859,C1(C(=O)NC(c2ncccn2)CC)CCN(C(=O)CS(=O)CC)CC1C 44860,c1(CC(=O)NCC2N(C(C(CC)F)=O)CC=C2)cc(C)cc(Br)c1 44861,CCC(O)C(C)(C)C(=O)NC1CC(C(=O)NCC2(CO)CCN(C)C2)CC1O 44862,C(=O)(CS(=O)(=O)NC)NC12CC(C(=O)NCC(CCC)O)(C1)C2 44863,c1(CC2CC(c3ccc(-n4cc(C5C(OC)C5)nn4)cc3)C2)cc(F)ccc1F 44864,N1(C(C(C)C2CC2)=O)CCCC1CCNC(=O)CN1CC2CC2C1 44865,CC1CC(NC(=O)CCc2ccccc2O)CN1C(=O)C(N)=O 44866,N1(C(C2N(C(c3cc(COC)no3)=O)CC(C)C2)=O)CCC(O)C(C)C1 44867,CC1(CNC(=O)C(C2(O)CCC2)NC(=O)CCc2ccccn2)CCCOC1 44868,C1(NC(=O)CCc2cncs2)CC1C1CCCN(C(c2cc(Cl)cs2)=O)C1 44869,C1(C(N(C(CCSC)C)C)=O)C(CO)C1(F)F 44870,C1(CN(C(C(c2ccccc2)SC)=O)C)CCCN1C(C1CN(C(N)=O)C1)=O 44871,N1(C(c2ccc(CNC(C#CC(C)C)=O)nc2)=O)CC(C)(C)CC1C 44872,N1(C(C2(CC)N(C(c3cc(CC)no3)=O)CCC2)=O)CCCNC(=O)CC1 44873,O=C(C1=CC(O)C(NC(c2csc(F)c2)=O)C1)NCC1(O)CCC(O)CC1 44874,N1(C(C2C(C)(C)CNC2=O)=O)CC23CCCC2(C1)C(=O)NC3=O 44875,N1(C(CC(CNC(=O)CCC(CF)CF)OC)=O)CCCC2CNC(=O)C12 44876,C(CS(=O)(=O)CC(=O)NCC(=O)NC(C)(C)CC(C)(C)C)OC 44877,CC(CC(C)(F)F)C(=O)NCC=CCNC(=O)CCCc1nncn1C 44878,c1(OC)ccc(NS(=O)(=O)NC(=O)NC2CC(F)C2)cc1 44879,C(=O)(C(C)Cc1ccco1)OC(C)C(=O)NCc1nc(C(N)=O)co1 44880,C=CC(C)(C)CCN(CCc1ccnn1C)Cc1ccccc1C 44881,C1(NC(=O)C=Cc2ccc[nH]2)COC2(CNC(C3(F)CCOC3)=O)CC1C2 44882,C1(C(=O)NCc2cc(C3CCC3)no2)CCCN(C(=O)C(F)CC2CCOC2)C1 44883,Cc1ccc(C)c(C(=O)NC(C)CC(C)NC(=O)C=Cc2ccc(=N)[nH]c2)c1 44884,N1(C(c2c(C)cccn2)=O)CCCC(C2CC2NC(=O)CCC(F)F)C1 44885,N1(C(C(C)OCC)=O)CC(O)(C(F)C(=O)N(C(COC)CC)CC)C1 44886,c1(C(=O)OC)cc(F)cc(F)c1NCc1cnc(C(C)(C)C)s1 44887,C1(CC=C)(NC(c2ccc(OC)nn2)=O)CCCN(C(c2nsnc2O)=O)C1 44888,C=C1CC(N=c2[nH]c(=NCC(=O)NC3CC3)[nH]c3cc(OC)ccc23)C1 44889,C#Cc1cc(C(N2CC(NC(c3cc(Cl)nn3C)=O)CC(O)C2)=O)cc(F)c1 44890,N1(C(c2cncc(C)n2)=O)CCC(NC(c2ccc(Cl)nn2)=O)C1(C)C 44891,C12(NC(c3cnsc3)=O)CCCN(C(=O)Cc3nc(F)c(F)cc3F)CC1C2 44892,C1(C(=O)OC)CN(C(=O)NCc2cnc(O)cc2OC)CCC1C 44893,N1(C(c2ccc(C(N)=O)o2)=O)CC2(CNC(C34CCCCC3C4)=O)CCC1CC2 44894,C(N(C1CC1)N1CCCCC(F)(F)C1)c1ccc(OC(F)(F)F)cc1 44895,CCS(=O)(=O)c1ccc(S(=O)(=O)N2CCN(C(C3CC3C)=O)CC2)cc1 44896,C1(CC)CN(C(c2cc(C)ncn2)=O)CC1C(=O)NC(CC1CC1)C1CC1 44897,N1(C(COCCCC)=O)CC(CC(=O)N(CCC(N)=O)C2CC2)C2(CC2)C1 44898,c1(C(C(=O)N(CCCCNC(=O)C(O)CC2CC2)C)(C)N(C)C)ccc(F)cc1 44899,N1(C(CCCCOC)=O)CC2CCCC(CNC(=O)Cc3nnc(C)o3)C2C1 44900,c1(CC)cc(C(N2CCC(NC(c3cc(Cl)n[nH]3)=O)C(F)C2)=O)ccc1OC 44901,C(c1ccccc1F)=CCC(N1CCC(NC(c2cc(C#N)no2)=O)(CO)C1)=O 44902,C(=O)(C1OCCc2c(Br)cccc21)NCCCCN(C(C(CC)C)=O)C 44903,C(=O)(C#CC1CCCCC1)NCCCN(C(C1CCC(C)S1)=O)CC 44904,c1(CNC(C2(COC)C=CCN2C(C2CC(F)C(=O)N2)=O)=O)cc(C)nc(O)c1 44905,CCCCCCC(=O)NC(C(C1CCCCC1)NC(c1ccnn1C)=O)C(C)C 44906,CC(=Cn1ccnn1)C(=O)N1CC2(CCN(C(c3cc4n(n3)CCO4)=O)C2)C1 44907,CCCCC(CC)CC(=O)NCC(CNC(=O)C(=Cc1cccc(F)c1)F)CO 44908,C1(CNC(CCC)(CC)c2nnnn2C2CCCCCC2)CCN(C)C(=O)C1 44909,c1(C(C)C)cc(S(=O)(=O)NC2CCC(CC(=O)O)C2)c(Cl)cc1Cl 44910,c1(CC)cc(OCC(N2CCCC2CNC(=O)CCCC#N)=O)ccc1Cl 44911,c1(OC)cc(C)ccc1OCC(=O)NC(CNC(c1cn(C)cn1)=O)C(C)(C)C 44912,c1(C(N2CC(NC(c3cccc(C(F)F)n3)=O)C3C2C3)=O)c(F)cc(F)cc1Cl 44913,O=S(=O)(c1ccc(NC2CC(=O)OC2Oc2ccccc2)nc1)N1CCCC1 44914,c1(OC)ncc(C(=O)Oc2ccncc2-c2cnc(OC)cc2OC)cc1F 44915,C1(CNC(c2c(C)cns2)=O)CC2(CCN(C(C3COCCN3C)=O)CC2)CO1 44916,C1(C(N2CCCC(N(C(c3c(CC)scc3)=O)C)C2)=O)CCc2ncncc2C1 44917,c1(C(N(CC(C)N(C(C(C)n2cnnn2)=O)C)C)=O)c(O)nnc2c1COCC2 44918,C12(NC(c3c(C)nc(C4CC4)s3)=O)CCN(C(=O)C(C)(C)n3cccn3)CC1C2 44919,C1(NC(c2c(C3(C)COC3)noc2)=O)CCCN(C(=O)Nc2cncc(N)n2)C1 44920,C=CC(F)(F)C(=O)NC1CCCC1NC(=O)COc1ccc(C(F)(F)F)cc1 44921,N#CC1CC12CCN(C(=O)C(O)CCNC(c1cc(CO)[nH]n1)=O)CC2 44922,C12(CNC(CCC(=O)NC)=O)CCC(CNC(C3CC3(C)C(C)C)=O)(CC1)OC2 44923,c1(CC(=O)N(C)C)ccc(C(=O)NCCC(O)CNC(c2cccnn2)=O)cc1 44924,c1(C(C)=O)cncc(C(=O)NC(CNC(=O)Cc2c(C)noc2Cl)CO)c1 44925,N1(C(c2ccn(C(C)(C)C)n2)=O)C2CCC1C(NC(c1cc(Cl)cnc1O)=O)C2 44926,CC(C)(C)CCCC(=O)N1CC(O)(C(C)(C)CNC(C2CC23CCCOC3)=O)C1 44927,c1(C(C)NC(c2c(Br)cnn2C)c2n(CCOC)nnn2)ccc(F)cc1 44928,c1(OC)nccc(C(=O)NCC2CCCC2NC(C2C3CCCC23)=O)c1F 44929,CC(C)C(O)C(F)(F)C(=O)NC(C1CN(C(=O)C(C)O)C1)C 44930,C1(NC(c2cn3ccsc3n2)=O)CN(C(=O)C(Cl)=CCl)C2(CCCC2)C1 44931,C(CC)(C(=O)NCC(C)(F)F)NC(C(F)=CCC)=O 44932,Cc1cc(=NC(C)c2ccc(C)o2)[nH]c(=NCCC(=O)N(C)C)[nH]1 44933,C(C1=CCC2CC1C2(C)C)(c1nnnn1C)Nc1cccc(C(C)F)c1 44934,N1(C(Cc2c(C)noc2)=O)CCN(C(C23CC(CO)(C2)OC3C)=O)C(C2CC2)C1 44935,C1(CCC)(NC(C2CCS(=O)(=O)N2)=O)CCCN(C(c2cnsc2)=O)C1 44936,c1(C(=O)NC(CC=C)CNC(c2c(C)ncnc2O)=O)cnc2n1CCCC2C 44937,N1(CC(C)CSc2ccccc2)CC(C(=O)O)C(F)(F)C1 44938,c1(C(=O)NC2C(NC(C(CC)NC(N)=O)=O)CC2)ccccc1CCN(C)C 44939,c1(C(C)=O)c(C)[nH]c(C(N2CCC(O)C(NC(=O)CC=C(Cl)Cl)C2)=O)c1C 44940,c1(COC)ccccc1C(=O)NCCCN(C(=O)CCC(=O)OC)C(C)C 44941,c1(NCC2C(NC(c3c(CC)ocn3)=O)CCCC2)ncc2cccnc2n1 44942,C1(NC(CC2(CNC(Cn3ncc(CC)c3)=O)CC2)=O)CCCC1N=[N+]=[N-] 44943,n1(CCC)ncc(C(N2CC3C(NC(C4(C5CCCCO5)CCC4)=O)C3C2)=O)c1C 44944,c1(OCC)cccc(OC(=O)C(C2CCCCC2)NC(C2C3CCCC23)=O)c1 44945,N1(C(c2c(OC)cccc2C)=O)CC2CC3CC2C1C3NC(=O)C=C(Cl)Cl 44946,c1(OC(C(C)C)C(=O)NCCC2CCCN2C(=O)C2CC2)ccc(F)cc1F 44947,N1(CC)CCCC(C(N2CC(F)CC2CN(C)C(c2cc(C(N)=O)no2)=O)=O)C1 44948,c1(CC(=O)NC2C(NC(C3(COCC)CCC3)=O)CCC2)ccc(Br)nc1 44949,c1(C(N(CCC(C)NC(CCCOC(C)C)=O)C)=O)c(F)cc(O)cc1F 44950,CC(C)(C(=O)N1CC2CCC(NC(c3ncsc3Br)=O)(C2)C1)S(C)(=O)=O 44951,c1(C(N2CCC(CNC(c3occc3C3CC3)=O)C2)=O)ccc2c(c1)OCCC2 44952,C1(CNC(c2cn(C(C)(C)C)nn2)=O)CN(C(=O)Cn2[nH]cnc2=N)CCO1 44953,CCC(F)(CNC(=O)CC1CCCCN1C(=O)CCCOC(C)=O)CC 44954,N1(C(CSc2ccc(C)s2)=O)CCC(C)C1CNC(C1(C)CCC1)=O 44955,Cn1cnc(C=CC(=O)NC2CCC2NC(=O)C(c2ccccc2)OC(C)(C)C)c1 44956,C1(CNC(C2(C)CC2)=O)CCN(C(=O)C(c2ccc(Cl)cc2)(F)F)CC1O 44957,n1(CC)nccc1C=CC(N1CC(CNC(=O)Cn2ccccc2=O)C(C)C1)=O 44958,C(=O)(C1=COCCO1)NC1C(C2CCN(C(C(CC)=CC)=O)CC2)OCC1 44959,C1(CNC(c2cc(-c3ccoc3)[nH]n2)=O)CN(C(C2C3CCC2CC3)=O)CCO1 44960,c1(CC)c(C(N2CC(NC(=O)CN(C)C3CC3)CC2C)=O)csc1C 44961,Cc1nc(C(C)C)ccc1C(=O)NC1(C)CCN(C(C2(F)CCC(C)CC2)=O)C1 44962,Cc1[nH]nc2ncc(C(=O)NC3CN(C(C4CCC(=O)C4)=O)CC3O)cc12 44963,C1(C)(C(N(C(C)CNC(=O)CNc2ncccn2)C)=O)CCC(F)(F)C1 44964,c1(C(=O)NCC(C)N(C)Cc2ccc(N(C)C)nc2)c(F)c(F)c(F)c(F)c1F 44965,c1(C(CNC(C2CC=CCO2)=O)NC(C(C)(C)N(C)C)=O)ccccc1F 44966,c1(C(N(C)CC2(O)CCN(C(=O)CSCC(N)=O)C2)=O)oc2ccccc2c1Cl 44967,C1(C(=O)NC(CC)C(=O)NC)Cc2ccccc2CN1Cc1cncc(C)c1 44968,c1(C(=O)NC(C(C)C)CNC(=O)C(C)CF)cccc(N)c1N 44969,N1(C(c2cc(COC)no2)=O)CC(NC(=O)C(O)C2CCC2)CC12CCOCC2 44970,Cn1ncc2c(O)c(C(=O)NCC(C)(O)CNC(C3CC(=C(F)F)C3)=O)cnc12 44971,N1(C(CSCCNC(C2C3CC(=O)CC32)=O)=O)CCN2C(=O)NCC2C1 44972,c1(C(=O)NCCNC(C(C(C)C)CN(C)C)=O)cccc2ncnn12 44973,C12(C(=O)NCc3cc(Br)ncc3Cl)C3C4C1C1C2C3C41C(N1CCOC(O)C1)=O 44974,c1(C(=O)NCCN(C(c2n(CC)cnn2)=O)C2CC2)ccc(OC)c(F)c1Br 44975,n1(CCC(=O)NC(CNC(C2(F)CCCC2)=O)C2CCC2)ncc2c1CCCC2 44976,C1(OCCOC)CC(NC(C(=O)N(c2ccccn2)C2CC(C#N)C2)=O)C1(C)C 44977,N1(C(C(CC(C)C)OC)=O)CCC(C)(C)C(CNC(=O)C=CC2CC2)C1 44978,c1(C(N2CCCC(CO)C2)=O)cc2ccc(-c3ccc4occc4c3)nc2[nH]1 44979,CC1OC2(CO)CC1(C(=O)NC(C)CN(C)C(C1CC3CCC(C1)C3)=O)C2 44980,C(CCC1c2nnnn2C2CCC(C2)N1)OC.C1(C(=O)OC)(OC)CCCC1 44981,c1(CC)noc(C(=O)NCC(C2CCC2)NC(C2CC3C=CC2C3)=O)c1C 44982,C1(C2CCN(C(=O)CN3C(=O)CCC3=O)C2)(NC(=O)CCc2ccccn2)CC1 44983,C(=O)(C(CO)NC(C1CC(=C2CCC2)C1)=O)N(CC(C)OC)C 44984,C(CC(F)(F)F)N(C(c1cn(CCNC(c2n[nH]cc2Cl)=O)cn1)=O)CC 44985,N1(C(c2ccc(C(=O)OC)[nH]2)=O)CCN(C(c2cc(C)ns2)=O)CC(C)(C)C1 44986,CC(Cn1cccn1)C(=O)NC(C1CCCN1C(c1cc(C(F)(F)F)cs1)=O)C 44987,C1(NC(c2cc(Cl)cc(Cl)n2)=O)COC2(CCN(C(c3cccs3)=O)CC2)C1 44988,c1(C(=O)NC(C2CCOC2)C)coc2c1CN(C(c1[nH]ccc1C1CC1)=O)C2 44989,C(c1ccccc1)=CCOCCN(C(C(C1CC1)OC)=O)C.C1CC1 44990,C1(C(=O)NCC2CC(F)CN2C(=O)CC2CCOCC2)CC(O)C(F)C1 44991,N=c1[nH]c2ncc(C(=O)NC3CC(CNC(=O)C=C(Cl)Cl)C3)cc2s1 44992,Cc1occc1C(=O)NCCc1cc(C(=O)NCC(C)(C)C#N)no1 44993,C(=O)(C(CCSC)NC(c1cccnn1)=O)NCC(=O)NCC=C 44994,O=C1CCC(CCC(N2CCCC2CNC(=O)CC2CSC2)=O)N1 44995,C12CCOCCN1C2=O.c1(NCCN2CCN(C)CC2)cc(F)ccc1N 44996,C1(C(N2CCC(CC#C)C2)=O)(NC(=O)CC(C)(O)COC)CCC(C)(C)C1 44997,N12CC(C)CC1Cc1cnn(c1)CC2=O.C(C)(CSC(F)F)OCC 44998,c1(C(N(C(C)CNC(=O)CN2C(C)CCC2C)C)=O)ccc2ncc(=O)[nH]c2c1 44999,c1(C(N(CC(C)NC(=O)CC2CC3CC3C2)CC)=O)ccc(OC2CC2)cc1 45000,N1(C(C2C(C)C2)=O)CC2CCC1C(CNC(c1cc(-c3ccncc3)no1)=O)C2 45001,CCCCC(C(=O)NCCCC(C)(C)NC(c1cccc(CF)c1)=O)NC(N)=O 45002,C(CC(O)CNC(=O)CNC(=O)C(F)(F)F)NC(CCSCCC)=O 45003,c1(CC2N(Cc3n(COC)ncc3C)CCC2)ccc2c(c1)ncn2C 45004,C1(C)(C(N(CCn2cc(CCCS(N)(=O)=O)nn2)CC)=O)COCC(C)(C)O1 45005,N1(C(CC=C)=O)CCC(NC(=O)Cc2sc(C)nc2-c2cccs2)C(C2CC2)C1 45006,C(CC(C)(C)C)(C(=O)N(CC1CC1)CC1CC1)NC(C1C(CC(C)(C)C)C1)=O 45007,Cc1nc(C(N2CCC(OCCNC(c3ccnnc3)=O)C2)=O)n[nH]1 45008,C1(C(N2CC(COC)(NC(=O)CC(C)NC(C)=O)C2)=O)CC2CCC1CC2 45009,C1(O)(C(=O)NC2C(n3cc(C(COC)(C)O)nn3)CCCC2)CCCC(C)(C)C1 45010,C1(COC)(CONC(C2CC3CC3C2)=O)CCCO1 45011,C(C)(CCCC(=O)NC(CO)CCC1CC1)NC(c1n(CC)nnc1)=O 45012,Cc1ccc(CC(=O)NC(=S)NNC)c(C)c1.c1(N2CCC(C(F)(F)F)C2)cccc(C)n1 45013,c1(C(N(CCC(C)NC(C(C)OCCC=C)=O)C)=O)ccc(C(C)C)s1 45014,C1(C2CCN(C(=O)CC3CCSCC3)C2)(NC(c2cc(C)sn2)=O)CC1 45015,C1(N(C(c2ccc(CC)[nH]2)=O)C)CCCC2CN(C(C3(F)CCCCC3)=O)CC12 45016,CN1CCC(F)(F)C(CNC23C(NC(=O)OC(C)(C)C)C4CC2C3C4)C1 45017,C1(C(=O)NCC(C(N2CC3C(COC)C3C2)=O)(C)C)CCC(C)=C(C)C1 45018,CC(CCNC(=O)CCCCN(C(=O)CC(C)n1cccn1)C)CCO 45019,C=CCC(C(=O)NC(C)CCNC(c1cc2ncccc2s1)=O)C(C)C 45020,C1(NC(CC(C)CF)=O)CCCC12CCN(C(c1cnn[nH]1)=O)CC2 45021,N1(C(c2oc(C)c(CO)c2)=O)CCC(C2CC2)(CNC(=O)CN2CC(CF)C2)C1 45022,c1(C(N2C(C(N3CC(CF)OC(CF)C3)=O)CCCC2)=O)nc2ccccc2s1 45023,CC1CN(C(=O)CC(C)(C)C2CCCC2)CCC1NC(C1CCC2(CCC2)C1)=O 45024,Cc1ccc(CNC(c2cncc(NC(=O)CC(O)c3ccccc3)c2)=O)cn1 45025,C(=O)(C#CC1CCCCC1)N1CCC(NC(C(C)N(CC(F)(F)F)C)=O)C(O)C1 45026,Cc1cc(CC(=O)NCC23CC(CNC(=O)C(C(C)C)N(C)C)(C2)C3)cc(F)c1 45027,CC(C)CC(C)(CNC(C1(C#N)CC(C)C1)=O)NC(c1ccc(NC=O)cc1)=O 45028,N1(C(CC)=O)CCN(C(c2cccc(C3(OCCCC)COC3)c2)=O)CC(O)C1 45029,C(=O)(CC(C)(C)c1ccc(F)cc1)N(C1CC(NC(C2(CSC)CCC2)=O)C1)C 45030,N1(C(Cc2n(C)nnc2)=O)CCCC(C2CC2NC(=O)C=CCN2CCOCC2)C1 45031,c1(C(=O)NC2CC(NC(C3(CC)CC3)=O)C2)cc(=N)[nH]cc1Br 45032,C1(CCn2cc(CC(=O)O)nn2)CCN(C(c2cnc[nH]2)=O)CC1 45033,c1(C(=O)NC2(CNC(CCOCC)=O)CC2)cccc2nn[nH]c12 45034,c1(OC)ccc(CN2CCC2(C)C(=O)Nc2cccc(C)c2C#N)c(Cl)c1OC 45035,c1(C(=O)NC23CC(NC(C(c4cccc(C)c4)C)=O)(C2)C3)cc(F)c(N)cc1F 45036,c1(C(=O)OC)cc(NC(c2ccc3c(n2)OCCO3)=O)cc2[nH]ccc12 45037,C1(NC(C2CCC(C)(C)CO2)=O)CC2CCC1CC2NC(=O)CC1CCCOC1 45038,c1(C(=O)NC2CC(CNC(C3CC=CC3)=O)C(O)C2)ccc2oc(O)nc2n1 45039,C=C(C)C1OCCC1C(=O)NC1CN(C(=O)COc2cncc(Cl)n2)CC1OC 45040,c1(C(=O)NC2CC(CCNC(Cc3n(C)cnn3)=O)C2)cc(Cl)cc([N+](=O)[O-])c1 45041,C(C(C)(C(=O)N1CC(CC(N)=O)C(O)C1)OC)OC.C(CCC=O)NC 45042,c1(OC)ncnc(OC)c1CN1CCC(NC(=O)Cn2ccnn2)C1 45043,C1(NC(Cc2c(C)cccc2F)=O)CC1C1CCN(C(C2(C)COC2)=O)CC1 45044,CC1=NOC(CC(=O)N(C(C(=O)N(C2CCCCC2)C)C2CC2)C)C1 45045,C(c1ccc(C)cc1)=C(C(=O)N(C)CC1N(C(CC2(OC)CC2)=O)CCCC1)C 45046,C1(N(C(=O)Cc2cnoc2)CC)CCCN(C(C2CC(F)(F)C2)=O)CC1 45047,N1(C(c2nc(Br)cs2)C(=O)NCCCSC)CCC(CCO)CC1 45048,C(=O)(CC(O)CC(C)(C)C)N1CCN(C(CCCCN(C(C)=O)C)=O)C(C)C1 45049,C1(N=c2cncc(Cl)[nH]2)(CNC(=O)CN2CCSCC2)CCOCC1 45050,O=C1OCCC2CN(c3ncncc3-c3ccccc3)CC12 45051,n1(CCC(=O)N(CCF)CCc2ccccn2)cc(COc2ccccc2)nn1 45052,CCCCC(C(=O)NCc1ccnc(O)c1)NC(=O)CC1CC2CC2C1 45053,C1(CNC(C(C2CN(C(C(C(=O)OCC)F)=O)C2)O)=O)OC(=O)NC1(C)C 45054,CC(C)CCC=CC(=O)NC(C)C(=O)N(C1CCOC1)C1CC1 45055,N1(C(C(C)OCC(F)(F)F)=O)CCC(N(CCO)C(c2cncc(N)c2)=O)CC1 45056,N1(C(C(CC#C)O)=O)C2CCC1CN(C(=O)CC(O)CC(C)C)C2 45057,N1(C(C2CC(=O)NC(=O)C2)=O)CCC2(CCCN2C(C2CC3(CCCO3)C2)=O)C1 45058,Cc1cccc(Cl)c1OCC(=O)NC1CN(C(C2CC(C)(F)C2)=O)CC12CC2 45059,n1(CCc2ccsc2)cc(CNc2cc(Cl)on2)nn1 45060,Cc1cc(F)ncc1C(N1CCN(C(=O)CCCCCF)CC1C)=O 45061,N1(C(c2ccc(N(CCC)C)nc2)=O)CC(C)(C)CC1CNC(=O)C(C)N(C)C 45062,NS(=O)(=O)c1ccc(C(=O)NCCC2CSCCN2C(C2CCCOC2)=O)s1 45063,c1(CN2CC(F)(C(=O)Nc3cc(CC)cc(Br)c3)C2)cc(Cl)c(O)cc1F 45064,N1(C(C(C)=C(CC)C)=O)CCN(C(C2(S(C)(=O)=O)CCC2)=O)CC1CC(=O)NC 45065,CC1(C(=O)NC2CCCN(C(=O)C(C)(O)C(F)(F)F)CC2)CCC(F)(F)CC1 45066,CC1(C)CCC(C(CNC(=NCC2CCCCC2)N(C)Cc2ccccc2)O)CC1 45067,N1(C(C2(CCNC(c3n(CCC)ccc3)=O)CC2)=O)CC[Si](C)(C)CC1 45068,N1(CC#N)CCCC1C1CCCCN1C(c1cccc2nc(O)[nH]c12)=O 45069,C(CC1CCC1)(C(=O)N(C)CC1CCN(C(=O)Cc2cc(C(C)C)no2)C1)OC 45070,c1(N2CCC(CC=C)(NC(c3cc(C4(C)CC4)n[nH]3)=O)C2)ncnc(Cl)c1CC 45071,C1(C(=O)NC(C2C(C(=O)OC)C2)C)CC2(CCN(C(C3(C)CCC(=O)N3)=O)C2)C1 45072,N1(C(CCN(CC(C)(C)C)C2CC2)=O)CC(CO)C2(CCNCC2)C1 45073,c1(NC(C2CCC2F)=O)cc(C(F)(F)F)c(Cl)cc1F 45074,C1(NC(C(COCC)C)=O)CC2CC(NC(=O)CCC(C)C)C1C2 45075,N1(C(c2c(OC)nccc2)=O)C2CCC1C(C(=O)NC(c1ncccc1C)C)C2 45076,c1(C(=O)NC2CN(C(c3n(CC)nnc3)=O)C(CO)C2)ccc2nncn2c1 45077,C(=O)(C1=CS(=O)CCC1)N1CC=CC(NC(CCc2cn(C)nn2)=O)C1 45078,Cc1nn(C)c(-n2cncn2)c1C(=O)NC1CCCN(c2ccccc2F)C1 45079,N1(CC(N2CC(c3ncnn3C)(OC)C2)=O)CC2(COC2)C1 45080,C1(CN(C(=O)CCC2CCCO2)C)CN(C(c2cccc(O)n2)=O)CC12CC2 45081,c1(CC(N2CCN(C(C(C=C=C)C)=O)CC2C(C)C)=O)ccc(S(C)(=O)=O)cc1 45082,N1(C(C2(NC(C)=O)CCC2)=O)CCC2(CCCN2C(C2CCCC2C)=O)C1 45083,c1(NC(c2cncc(-c3ccc(SC)cc3)n2)=O)cc(C)c(I)cn1 45084,c1(CCNC(C(CCC)N2CCNCC2)=O)c(C)cccc1C 45085,c1(C(N(CCC(C)NC(C2CC23CCC3)=O)C)=O)c(Cl)cccc1Br 45086,CCCC(C)CCCC(=O)NC1CCC(C)N(C(=O)C=Cc2nccn2CC)C1 45087,C(=O)(C#CC1CCCOC1)N1C(C2(NC(Cc3ncc(C)s3)=O)CC2)CCCC1 45088,C#Cc1cncc(NC(C2CC=CCN2C(C2CCCN2CC)=O)=O)c1 45089,N1(C(C2C=CCN(C(c3oc(CC)c(C)c3)=O)C2)=O)CC2CCC(C1)O2 45090,N1(C(CNC(=O)OCC)=O)CCCC2(NC(c3ncccc3F)=O)CC12 45091,S(=O)(=O)(c1cccc(CBr)c1)N1CCC2CN(C(c3cc(Br)nc(Br)c3)=O)CC21 45092,C1(NC(c2[nH]cc(C(C)=O)c2)=O)CCC(NC(C2CC3(CC3)CO2)=O)CC1 45093,N1(C(C(C)OCC=C)=O)CCC2(CCCN(Cc3cc(C)ccc3O)C2)C1 45094,CC1CN(C(=O)CC2OCCC2(C)C)CC1NC(=O)Cc1n[nH]c(=N)s1 45095,c1(CC(=O)N(CC(C)N(C(c2cc(C)c(C)[nH]2)=O)C)C)ccc2sccc2c1 45096,c1(C(C)C)nc(C(=O)N(C2CN(C(=O)C(C)CN3CCCCC3)C2)C)cs1 45097,C1(NC(CC2N(C(CCC(C)=O)=O)CCCC2)=O)CC2(COCCO2)C1 45098,S(=O)(=O)(CCC(F)(F)F)N(c1ncc(C#N)s1)C1CC(C)(C)C1 45099,N1(C(c2nc(C)c(C)s2)=O)CCN(C(=O)C=CC2CCC2)CC1CC1CC1 45100,C1(CNC(=O)C2=C(Cl)CC2)C2CCCC1N(C(c1ccc(Cl)o1)=O)C2 45101,N1(C(c2[nH]cc(C#N)c2)=O)CC2(CCC2)CC1CNC(C1(N2CCCC2)CCC1)=O 45102,N1(C(CSc2c(C)n[nH]c2C)=O)CC2(CCC2)CC1CNC(C1(F)CCOC1)=O 45103,N1(c2c([N+](=O)[O-])ccc(OC)n2)C2CCCC1CN(C(C1CCC1)=O)CC2 45104,C(C(=O)N(CCCCN(C(=O)CC1C(=O)NN=C1C)C)C)(C(C)C)OCC 45105,C(C(CC)(CC)C(=O)NC(c1ccccc1)C)NC(C(CC=CC)C)=O 45106,c1(N2CC(C(C)NC(C3(C)CC(O)CN3C)=O)C2)ccc([N+](=O)[O-])cn1 45107,N1(C(COCC(=O)OC)=O)CCCC2CN(C(=O)C(C)CS(C)(=O)=O)CCC12 45108,C(C(=O)N1CC(=O)NC(C)C1)(C(C)(C)C)n1cc(-c2c(OC)ccnc2)nn1 45109,C(=O)(CCC(C)(C)NC(C1CCC(=O)C(C)C1)=O)NCCC(CCC)C 45110,c1(CC(=O)N(C2CCN(C(C3CCCN3S(C)(=O)=O)=O)C2)C)ncc(F)cc1F 45111,C(CC(C)C(=O)NC1CC(NC(C2CCOC2c2cccnc2)=O)C1)=CC 45112,C1(CC)(NC(=O)C(Cn2cncn2)NC(=O)Cn2nnc(C)n2)CCCC1 45113,c1(OCC)ncc(C(=O)NCC(CNC(C2CCCCNC2=O)=O)OC)cc1Cl 45114,C#CCC(CC(=O)N1CCCCC1CCO)NC(=O)C(C1CC1)OCC 45115,c1(C(=O)NCc2ccc(-c3ccc(CO)cc3)cc2)nc(Br)n2c1CCNCC2 45116,CC1(C)CC(CNC(C2CCN(C(=O)CS(C)(=O)=O)CC2)=O)CO1 45117,CCCC(CCCNC(=O)C(CC)C(C)C)NC(C1(c2ccccc2)CCC1)=O 45118,CCP1(=O)CCN(C(c2ccc(OCC(F)(F)F)nc2)C(=O)NC2CC2)CC1 45119,c1(C(C)CNC(C)Cn2cnc(-c3cccs3)n2)cccc(Cl)c1 45120,N1(C(CC(=O)NCC)=O)CC2CN(C(=O)CC(C)C(C)C)CC2(C)C1 45121,C1(CNC(CCC=C=C)=O)CC(C)CN(C(=O)CCC)C1 45122,C1(C(N2CC(C=C)C(NC(=O)C3=COCCO3)C2)=O)CC12CCCCCC2 45123,C1(NC)CCC(C(=O)NCC)O1.C1(C)(C)CO1.n1(CC(=O)N)cncn1.C1(=O)CN1 45124,c1(OC)ccnc(C(=O)N(CCCCNC(C2CCC(C(F)(F)F)O2)=O)C)c1F 45125,C(=O)(C(C)C(O)C(C)CC)N1CC(C(=O)NCC(CC)N(C)C)C(C)(C)CC1 45126,N1(C(C(CCNC(=O)CC2OCCO2)OC)=O)CCOC(C)(C)C1C 45127,C1(CNC(c2c[nH]cc(C)c2=O)=O)CCCCN(C(=O)Cc2c[nH]nc2O)CC1 45128,Cc1cc(F)cnc1C(=O)NCC1CN(C(=O)CCn2ccnc2)CC1O 45129,N1(C(COC)=O)CCOC(CNC(=O)CNC(c2ccnc(N(C)C)c2)=O)C1 45130,C(C)(C(C)C(=O)NCC(C)CC1CCC1)NC(c1cn(C(C)C)nc1)=O 45131,CCCCCC(C)(C)CNC(=O)C(C)N(C)C(C1CCN1CC)=O 45132,C1(C(N2C(CNC(C3N(C)CC4(CC4)C3)=O)CCC2)=O)CCC(C2CC2)CC1 45133,N1(C(C(F)=C(C)C)=O)CC(=O)CC1C(=O)NCCc1cc(O)ncn1 45134,c1(CC(C(=O)OC)NC(C2NCCCC2C(F)(F)F)=O)ccc(F)c(Cl)c1 45135,CC1(CCC(=O)NC23CC(CO)(C2)C3)CCCN1C(=O)CSc1ccnc(O)c1 45136,c1(C(=O)NCCCN(CCNC(c2ccc(OC)s2)=O)C)ccn2cccc2c1 45137,C(=O)(C(C)(C)CNC1(c2nnnn2CC2CCCO2)COC1)NC 45138,c1(C(=O)NCC2N(C(C(C)OCCCCCC)=O)CC2)nn(C)c2c1CCC2 45139,c1(C(=O)NC(c2nc[nH]n2)CC)ccoc1CNC(C1CC1(C)CC)=O 45140,N1(C(CC(CCC)(C)O)=O)CCC2C1CCCN2C(c1cn(C2CC2)nn1)=O 45141,c1(CC(=O)NC(C2CCOC2)CNC(C2(F)CC=CC2)=O)ccccc1Br 45142,CC(C(=O)N1CC(O)CC1CNC(c1ccc(N)c(C(F)(F)F)c1)=O)S(N)(=O)=O 45143,c1(C(=O)NCC2(F)COCCN(C(C=NOC)=O)C2)cnc2scc(C)n2c1=O 45144,C(CN=[N+]=[N-])(C(=O)NCCCc1ccccc1)NC(COCC=C)=O 45145,c1(C(=O)NC(C)CNC(=O)C(c2ccc(C#N)cc2)O)cnn2cccc(Cl)c12 45146,C(CC(=O)CCO)c1cn(CC2CCC(NC(=O)C=CC3CCCC3)C2)nn1 45147,c1(NCCCC)ccc(C(=O)NC2(C)CC(NC(=O)CC3CC3)C2)cc1[N+](=O)[O-] 45148,c1(C(C(=O)NC(CC)(C)C)N(CCC#N)C2CCC2)ccc(Br)c(F)c1OC 45149,N1(C(c2cc(C)nn2C)=O)CC2CCC1CC2NC(=O)C(O)CCC(C)C 45150,CC1(C)CCCCC1OC(F)(F)F.N12C(=O)NC(C1=O)CCCCC2C1COC1 45151,CC(C(=O)N(CCCNC(c1ccnc(C(C)(F)F)c1)=O)C)C(F)(F)C(F)F 45152,N1(C(C)(C)C)CCC(C(=O)NCc2[nH]nc3c2COC3)C(F)C1 45153,C1(C=O)CCN1N(CCNCC=CC(=O)C(=O)OC(C)(C)C)CCOC.CC=C 45154,C1(NC(=O)C(=C2CCCCC2)F)CCCC(CC(=O)NCc2cncs2)C1 45155,C1(NC(c2cc(OC)n(C)n2)=O)CN(C(C2CCC(=O)O2)=O)CC(F)(F)C1 45156,c1(C(=O)NC2(C)CCN(C(c3c(CC)c[nH]c3)=O)C2)ccc(N)c(C)c1Cl 45157,CCCCC(O)CNC(C1CN(C(c2nccn2C)=O)CC1C(C)C)=O 45158,c1(C(N2CC3C(C2)N3C(=O)Cc2ccc(Cl)cn2)=O)cncc2cnccc12 45159,C12C3CCN(CC13)C2=O.C12CN(CCO1)C(=O)C2.n1(CC)cc(C2CC2)cn1 45160,N(C(=NCc1cnc(C)cn1)NC(c1cccs1)C)Cc1nnc(SC)s1 45161,CN1CCN(C(=O)CC2(NC(=O)CC3CC4CC4C3)CC2)CC(O)C1 45162,c1(C(=O)NCCCOC)cc(-c2cc(OC(C)C)c(C)c(C)c2)c2cc[nH]c2c1 45163,c1(C(=O)NC2(CCNC(CCSC)=O)CC2)ccc(C(F)(F)F)cc1N 45164,c1(C(N2C(C(=O)NCCC(C)C)CC(F)C2)=O)ccc(Br)c(Cl)c1Cl 45165,Cn1cc(C(F)(F)F)cc1C(=O)NC1CCC1NC(=O)C1=NOCC1 45166,C(C(=O)N=c1cc(C)[nH][nH]1)c1cccc(NC(c2c(OCC)oc(C)n2)=O)c1 45167,C1(NC(=O)CC23CCCN2CCC3)CN(C(=O)Cn2cnnc2)CC1C1CC1 45168,N1(C(CN(C(C)C)C(c2cccc(C#N)c2)=O)=O)CC2(CC(F)C2)C1 45169,C(=O)(CCCOCC=C)NC(c1ccccc1)CNC(C(C)OCCC=C)=O 45170,N1(Cc2c(OC)ccc(Br)c2)CCC(F)(F)C(C(=O)Nc2ncc(F)cc2I)C1 45171,c1(OC)cc(C(N2CC(CNC(c3c(OC)noc3C)=O)C(C)C2)=O)ccc1F 45172,C1(O)(CNC(=O)CCCC2CCCC2)CCCN(C(C2COC(=O)O2)=O)C1 45173,C#CCCC(O)C(=O)NC1(CCC)CCCN(C(=O)Cc2ccnc(O)c2)C1 45174,N1(C(C2C(CCC)C2)=O)CCC(CN2CCOCC2)CC1.C12(CCC1)C(=O)N2CC 45175,C(=O)(C(CC1CC1)NC(C1(CCNC(=O)CCc2nc(O)n[nH]2)CCC1)=O)NC 45176,CC1(C)CC(CNC(c2cccnc2)=O)N(C(=O)CCc2cc(Cl)no2)C1 45177,c1(C(=O)NC2C(NC(C3C(C#N)CC3)=O)C2)ccc(C2CCCCC2)cc1 45178,c1(C(=O)NCCCCN(C(c2nc(=O)n(C)[nH]2)=O)CC)ccc(N(C)C(C)=O)nc1 45179,C(=O)(C(CNC(=O)CCCC1CCCC1)C(C)C)N(CCCOC)C 45180,Cc1c(CC(N2CCC(C(O)C(F)F)C2)=O)c(=O)oc2cc(N)ccc12 45181,Cc1cc(N2CCC3(CNC(=O)CC4CSC4)CCCCC23)n2nc(C)cc2n1 45182,C=CC1CN(C(C23CCOC(C)(C2)C3)=O)CC1NC(=O)CCc1csc(C)n1 45183,CCC(CC(=O)NC1COCC1CC(=O)NCc1ncn(CC)n1)C(F)F 45184,c1(C(=O)NC(CC=C)CNC(C2CC(C)=NO2)=O)ccc(Br)c(Cl)c1 45185,C1(CNC(C2=CC(C)(C)C2)=O)CC2COCC2N1C(=O)COc1cccc(Cl)c1 45186,N1(C(=O)NCCCC(=O)OC(C)(C)C)Cc2ncnc(O)c2C1 45187,c1(CC(C(=O)NC(CCCNC(c2occ(C)c2)=O)C)C)c(C)n[nH]c1C 45188,c1(C(=O)NCC(C)NC(CCn2ncc(C)c2)=O)ccc(Cl)cn1 45189,c1(CC)ccc(C(=O)NCC(C)(C(C)C)NC(=O)CCc2cnc(O)[nH]2)cn1 45190,C1(C(N(C2CCN(C(=O)CCc3csc(=N)[nH]3)C2)CC)=O)CC(C)(C)CCO1 45191,C1(N(C)C(c2cocn2)=O)CCN(C(C2CCCC(O)C2)=O)CC1 45192,Cc1cc(-c2nn(C)c(C(=O)OCCn3ccc(Br)n3)c2Cl)ccc1F 45193,c1(C(N(C2CCCN(C(CCCC#C)=O)C2)CC)=O)ccc(C)c(Cl)c1 45194,CC#CCC(C(=O)N1CCC1(C)CC)NC(c1cn[nH]c1)=O 45195,c1(C(=O)NC2CC(CNC(C(C)CC(C)(C)C)=O)C2)ccc2c(c1)CCCC2 45196,C1(C)(CNC(C(C(C)C)NC(N)=O)=O)COCCN(C(=O)C2=CCCCO2)C1 45197,C1(NC(C(CCOCC)NC(c2[nH]nnc2C)=O)=O)CC12CCCCC2 45198,c1(SC)cc(Br)ccc1C(N1CCCC(NC(c2ocnc2C)=O)C1)=O 45199,CC(O)C(C)C(=O)N(CC(C)NC(C1CCCN1Cc1ccccc1)=O)C 45200,c1(C(=O)NC(c2cccc(C)c2)CNC(C=COC)=O)nn2c(c1C)CCCC2 45201,Cc1cc(CC(N2CCC(c3nc(C(F)(F)F)cs3)CC2)=O)n(C)n1.C(CS)O 45202,C(C1CN(C(=O)CC2CC(=O)NC2=O)CC1C(=O)N1CC=CCO1)=CC 45203,c1(CC)ncc(C(=O)NC2CC(CCNC(c3nccn3CC)=O)C2)c(O)n1 45204,C=CC1CCCCN1C(C1OCCC1CNC(C1CC=C(C)CC1)=O)=O 45205,C(=O)(C(F)C(C)(C)O)N1C2C=CCC(C2)C1=O.c1(OC)c[nH]ccc1=O 45206,c1(NC(c2cc(F)ncc2NS(=O)(=O)CC2CC2)=O)cc(O)c(Cl)cc1Br 45207,N1(CC(=O)NC(CNC(c2cc(C3(C)CC3)n[nH]2)=O)(C)C)CCS(=O)(=O)CC1 45208,c1(SC)ccc(C(=O)NCC(C)(C2CC2)NC(=O)COC)cc1.C(=O)CO 45209,c1(CC)cc(CNCC2CSCCN2c2cc(N)ncn2)cc(CC)c1 45210,N1(C(c2[nH]cc(C)c2)=O)CCCOC(CNC(c2cc(C)ncc2Cl)=O)C1 45211,c1(NC(C2C3CN(C(C4(O)CC4)=O)CC23)=O)cc(O)nc(Cl)c1 45212,C(=O)(C(C)CC(C)C(C)=O)N(CCCNC(=O)CC1CC=CCN1C)CC 45213,c1(C(=O)NC(CN(C)C)C(=O)NCC(O)CC(F)(F)F)cc(F)cc(F)c1 45214,c1(C(N(CC(CN(C(C=CC(=O)OCCCC)=O)C)O)C)=O)nn[nH]c1Cl 45215,C#Cc1ccc(F)cc1C(=O)NCCOCCNC(c1cc2c(ccn2C)[nH]1)=O 45216,c1(C(=O)OC)cccc(C(CC(=O)NC(C)(C)C)C2CC2)c1.[nH]1cc(C=O)nn1 45217,CC1CCC(C)C(C)C1NC(c1ccncc1I)=O 45218,C1(C(=O)NC(CC)CN(C)C(c2ccsc2)=O)CCCCN1N1CCOCC1 45219,C(CC(C(=O)NCC1CCN(C(C)C)C1)NC(c1sccc1Cl)=O)OC 45220,c1(C(N2CC(OCCNC(=O)C(F)CC3CCCC3)C2)=O)ccc2sncc2c1 45221,C12(C(=O)NCC(CC#C)(C)C)CCCC1CCN2C(c1n[nH]cc1C)=O 45222,c1(C(C(=O)NCCC)N(C)CC2CC3CCC2C3)ccc2c(c1)NC(=O)CO2 45223,c1(C(N2CC(C)(C(=O)Nc3ccnc(F)c3)C2)=O)c(F)c(F)cc(F)c1F 45224,Cc1cc(C#N)nc(N2CC(C)(C)OCC2CNC(c2sc(F)cc2C)=O)n1 45225,CC(C)(C(F)(F)F)OCC(=O)NCCOCCNC(C1(F)CC=CCC1)=O 45226,c1(C(N2CCC(CNC(C=CCOC)=O)(OC)CC2)=O)ccc(C)c(C)c1O 45227,N1(c2nnc(C)s2)CC(CNC(C2(C)CC(C)(C)C2)=O)OC2(CCC2)C1 45228,C1(CNCCC(=O)OC)C2CN(C(=O)Cc3ccco3)CC12 45229,c1(C(=O)NC(CC(C)NC(c2cc(CO)[nH]n2)=O)C)cc(F)cc(Cl)c1 45230,C1(C(=O)NCCN(CCOC)C(c2nc(Cl)cs2)=O)CCCC1OC 45231,Cc1noc(C(F)(F)F)c1C(=O)NCC(F)CNC(C1(C2CC2)CC1)=O 45232,c1(CCC(N2C(CNC(c3ccc(COC)[nH]3)=O)CC2)=O)ccc(SC)cc1 45233,c1(N2CC(COC)C(SC)C2)cc(Br)ccc1S(=O)(=O)NCc1ccc(SC)o1 45234,C(=O)(C1COc2ccccc21)N1CCC(C2N(C(c3nccc(C)n3)=O)CCC2)C1 45235,Cc1cc(CC(=O)NCCCCNC(=O)CCC(=O)c2ccncc2)c(C)s1 45236,N1(C(c2c(C)nn[nH]2)=O)CCN(C2CCCN(C(=O)C(C(C)C)N(C)C)C2)CC1 45237,C1(C(=O)NC(C#C)CCC)CC(=O)CN1C(C1(C(=O)C2CC2)CC1)=O 45238,N1(C(c2c(C3C(C)C3)noc2)=O)CCC(C(=O)NCCNC(C2CCC2)=O)CC1 45239,n1(CC)ccc(=NC(=O)C2CN(C(c3ccccc3O)=O)CCC2(C)C)[nH]1 45240,N1(C(c2c(CC)c[nH]c2)=O)CCN(C(C2(C)CCC(=O)C2)=O)CC1CCOC 45241,C1(CNC(C2C=CCN2C(=O)C(O)C2CCCC2)=O)CC2(CCC2)C1 45242,c1(C(c2n(CC=C)nnn2)NCc2ccns2)ccc(C)cn1 45243,N1(C(Cc2ccc(C)s2)=O)CCCC(N(C)C(C2C(C)OC(C)C2C)=O)CC1 45244,C1(C(=O)NCC(C)C(=O)NC2C=CC(C)(C)CC2)CCC(C)(O)CC1 45245,c1(CNC(N(C(c2ccccc2)c2ccccn2)CC)=O)ccc(N(C)C)cc1 45246,CC(CS(C)=O)C(=O)N(CCCNC(=O)CNC(=O)CCCCO)C 45247,C(C(C)(C(=O)NCC=CCC(=O)N(CC(C)(C)O)C)OC)OC 45248,C(=O)(C1=CCS(=O)(=O)C1)NCC1(C)CCN(C(=O)Cc2cc(Cl)ccc2O)C1 45249,C(=O)(CS(=O)(=O)c1nccn1C)N1C(c2n(CC)ncc2)CCC1.C(C)(=O)O 45250,c1(NC)cnc(Cl)cc1C(=O)NCC1CCC(NC(C2COCCO2)=O)C1 45251,c1(NC(CN(C)Cc2cnc(CC)s2)=O)cc(Cl)c(OC)cc1CC 45252,C#CC(CNC(C1C=CCN1C(c1cnc(O)o1)=O)=O)CC1CC1 45253,c1(-c2cn(C)nc2)ccc(F)c(C(=O)NCc2cn(CC3C4CCCC34)nn2)c1 45254,c1(CNC(c2ccn(C)n2)c2nnnn2CCC2CC2)c(Cl)cncc1Br.C1CC1 45255,n1(CCCC)ncc(C(=O)NCC(O)CN(C)C(c2nnn(C)c2C)=O)c1CC 45256,N1(C(C)=O)CCCC1C(=O)NC(C)(CNC(c1cn(CC(N)=O)nn1)=O)CO 45257,C1(CNC(C(c2cnn(C)c2)C)=O)CCC(NC(=O)Cn2cncn2)CC1 45258,C(=O)(C1=CCCC1C)NC(CCOCC)C(=O)NCCNC(c1ccoc1)=O 45259,C1(CC(=O)N(C2CCC(NC(C(C=C)O)=O)CC2)C)CC(C)CC(C)(C)C1 45260,Cc1ncccc1C(N1CC=CC1CNC(C1C(F)(F)C12CC2)=O)=O 45261,c1(OC)ccnc(-c2cn(C3CCN(C(C4(C)C=CCCC4)=O)C3)nn2)c1 45262,c1(C(N(CCC(N2CC(C#C)C2)=O)C(C)C)=O)cnc2n1CCC2 45263,c1(OC)cccc2c1OCCCC2NC(=O)C(=O)NC1CCN(C2CC2)C1=O 45264,N1(C(=O)CCC2CCC2)CCC(C2CC2)C1C(N1CCn2ncnc2C1)=O 45265,N1(C(CCCOC)=O)CCCOC(CCNC(=O)C(C)OC2COC2)C1 45266,CC1(C(=O)NCCC2CN(C(c3cc(Br)co3)=O)CCO2)CCCNC1=O 45267,c1(CN(C(C2CCCSC2)C(=O)NCC)C2CC2)c(C)nn(C)c1C 45268,C1(NC(=O)Cc2ccon2)CC2CCC(C1F)N2C(c1nc(Cl)c(Cl)s1)=O 45269,C1(C(N2CCCN(C(c3cccc(O)c3C)=O)CC2)=O)(OC)CC(C)CC(C)C1 45270,CC1CCC(NC(=O)C(C)(C)C(=O)OC(C)(C)C)CN1C(=O)Cn1cccnc1=O 45271,N#CC1CC(C(=O)NCC(O)CNC(C2(CC3CCC3)CC2)=O)C1 45272,C12(C=O)CC(CN(N3CC(C(CC)CC)C3)C1)C2.n1(C(C(=O)N)C)ccnc1C 45273,CCCC(C)CC(=O)N1CCOC(CN(C(=O)CN(C)C2CC2)C)C1 45274,N(C(=NCCC)NCCC(C)Oc1cccc(C(F)(F)F)c1)CC=C 45275,N1(C(c2ccc(C)[nH]2)=O)CC(C(N2CCOCC(N(C)C)C2)=O)C(F)(F)C1 45276,N(C1CN(c2cc(Cl)ncn2)CCc2ccccc21)C(=O)CCc1cnc[nH]1 45277,C1(C(N2C(C)CC(CNC(c3cc(O)nn3C)=O)C2)=O)CCn2c(O)nnc2C1 45278,C12(CNC(C3C=CCC3)=O)CCCC(CN1C(=O)CSc1ccccc1)C2 45279,c1(C(=O)NC2CCN(Cc3c(C#C)cccc3)CC2O)ccc(O)c(O)c1Cl 45280,c1(C(=O)NC2CCCN(C(C3CC(OCC)C3)=O)C2)ccc2nccn2c1 45281,c1(CC(C)C)nc(C(=O)N(CC(=O)CC2CCC2)CCc2ccccc2)cs1 45282,c1(C(N2CC(CNC(C3(OC)CCC3)=O)(COC)C2)=O)ccc(C)c(S(N)(=O)=O)c1 45283,N1(C(C(CC)N(CC)CC)=O)CCC(C)CC1CNC(c1ccc(Cl)c(N)c1)=O 45284,c1(OC)ccccc1C(N1CC(N(C(=O)CCC(C)N(C)C)C)C(O)C1)=O 45285,Cc1[nH]c2c(C(N3CCC(CNC(=O)CC4CC4(Cl)Cl)C3)=O)cccc2c1C 45286,N1(C(C(C(C)(C)O)F)=O)CCC(C2(NC(c3ccnc(C4CC4)c3)=O)CC2)C1 45287,c1(OCC(N2CC(NC(=O)C(=O)NC3CC3)OCC2)=O)cc(F)ccc1F 45288,N1(C(CCN(C(C)=O)C)=O)CCOC2(C1)CN(C(=O)Cc1cnco1)C2 45289,c1(Cn2cc(CONC(c3cccc(C(CC)=O)c3)=O)nn2)cc(C)cc(C)c1Br 45290,C1(O)(CCNC(c2c(C)nc(CCC)s2)=O)CCN(C(=O)C(CC)OCC)CC1 45291,N1(C(=O)OCC)CSCC1C(=O)NCC(C(C)C)NC(=O)CN(C)C 45292,Cc1cc(N2CC(C)(C)CC2CNC(c2csc(CO)n2)=O)nc(C)n1 45293,c1(C(=O)NC2(C3CC3)CCN(C(C(CC)(C)C#N)=O)C2)cnc2ccncc2c1 45294,C(=O)C1=CCCNC1.c1(CC(NOCCC=C)=O)[nH]ccc(=O)c1C 45295,c1(C(=O)NC(C(C)NC(C2CC(=C)C2)=O)(C)C)cc(Cl)cc(F)c1N 45296,c1(C(N(CC(=O)N(C)CC2CCCS2)C2CC2)=O)occ2c1CCC2 45297,C1(NC(c2ccccc2Cl)(C)CO)CC2CCC(C1)C2N 45298,c1(C(=O)NC2(COC)CN(C(c3n(CC)c(O)nc3)=O)C2)cncc([N+](=O)[O-])c1 45299,C#CC1(NC(=O)CCC2(C)CN(C(=O)C(C)CCCC)C2)CCCCC1 45300,N1(C(CCC(=O)NCC)=O)CC(C)CC1(C)C 45301,N1(C(C(c2ccccc2)C)=O)CC(C)(CNC(C2(N(C)C)CCC2)=O)CC1(C)C 45302,CC(C)CCC(C)N(C(=O)C(C)N(C(C1CCC2CC12)=O)C1CC1)C 45303,c1(C(=O)NC2CC3CN(C(C(CC)CC)=O)CC3C2)ccc2cnnc(O)c2c1 45304,C(C1CCOCC1)=CC(N1CC(COC)(CNC(C2(C)CCOC2)=O)C1)=O 45305,c1(C(N2C(CNC(C=C(COC)C)=O)CC(F)C2)=O)cccc(OC)c1C 45306,c1(C(=O)NC(C)(CNC(=O)C(O)CN2CCCC2)CO)csc2nnsc12 45307,N1(C(COCC)=O)CC(C)(C)CC1CC(=O)NOCc1ccccc1 45308,N1(C(c2nnn(C(C)(C)C)n2)=O)CC(NC(c2ncccc2O)=O)CC(F)C1 45309,c1(C(N(C(C)CNC(c2ccnn2C(F)F)=O)C)=O)oc2ccccc2c1Cl 45310,C1(F)(CNC(COCCCOC)=O)CCCN(C(C2CCC=CCCC2)=O)C1 45311,C(CC(C(=O)NCCc1nncn1CC)NC(c1cnco1)=O)=CC 45312,N1(C(Cc2nc(C)oc2)=O)CCCC1(C)C(=O)NCC1(C)CCCC1O 45313,c1(OC)ccc(C(=O)NC2CCC2NC(C2CC2c2ccc(F)cc2)=O)c(F)n1 45314,Cc1ccc(F)c(C(=O)NCCC(O)Cn2cccn2)c1 45315,C1(NC(C(C)OCC#C)=O)CN(C(=O)CCc2cccs2)CC2(CCC2)C1 45316,c1(C(=O)NCCCN(C(C2C(OCC)CC2)=O)CC)ccnn1C1CCOCC1 45317,CC1CC(NC(=O)CCCNC(N)=O)CCN1C(=O)CSC(F)F 45318,c1(-c2onc(C(=O)NC3C(NC(c4nnn(C)n4)=O)CCC3)n2)cccc(Cl)c1 45319,N1(C(=O)Nc2ccc(C)c(C)c2)CC2C(C1C(N1C=CCSC1)=O)C2(C)C 45320,N1(C(C2C(C)CCO2)=O)CC=C(CC(=O)NCC(O)C(C)(C)C)CC1 45321,CC1(C)CCC=C1C(=O)N1CCC2CN(C(=O)C=Cc3ccccc3)C2C1 45322,C(=O)(CC(C=C)CCC)NC1CCN(C(c2cn(CC=C)nn2)=O)C12CC2 45323,N1(C(CC(C)(C)O)=O)CC2(C1)SCCC2NC(c1ccc(SC2CC2)cc1)=O 45324,C(=O)(C1=CC2(CCOC2)C1)N(C1CN(C(c2nn[nH]c2Cl)=O)CC1O)C 45325,C(=O)(C(C)CC(=O)OC)N(C1CCN(C(=O)CC(=O)NCC2CC2)C1)CC 45326,C1(NC(=O)CCc2cncs2)CC12CCN(C(C1CCCOC1)=O)C2 45327,Cc1nn(CC(=O)NCC(C)NC(c2nccnc2Cl)=O)c(=O)n1C 45328,N1(C(CC(C)C2CCCO2)=O)C2CCC1CC(CNC(c1ccc(=N)[nH]c1)=O)C2 45329,N1(C(C2N(C(C)=O)CC(O)C2)=O)CC(NC(c2ccnnc2)=O)C(C)(C)C1 45330,c1(C(C(=O)N2CC(CCNC(c3[nH]ccc3C)=O)C2)OC)c(F)cccc1F 45331,N1(C(c2cc3cccc(F)c3s2)=O)CCCC(C2CN(C(C3(F)CC3)=O)C2)C1 45332,c1(C(N(CC(O)CN(C)C(C23CC(CN2C2CC2)C3)=O)C)=O)cnn2cc[nH]c12 45333,C1(C(N(C(C=C)C)C)=O)CCC(CNC(=O)Cc2ccn(CC)n2)C1 45334,c1(CC(N2CCC(NC(C3C(CC)CCC3)=O)C23CC3)=O)n[nH]c2ccccc12 45335,C#CC(CC1CCC1)NC(=O)CC1(N(C(=O)CC=CCC)C)CC1 45336,C1(CS(=O)(=O)NCC2CC(C)(C)OC2)CCCC2(CCOC2)O1 45337,Cc1nc(CNC(=O)CC2(CNC(=O)C(C)C3CCOC3)CC2)n[nH]1 45338,C(=O)(C(C)(C)C(=O)N(C)C)NCC1(CNC(c2c(COC)noc2)=O)CCC1 45339,C1(C)(CCC(=O)NCC(C)CN(C(=O)CCOC2CCC2)C)CCC(=O)N1 45340,C1(C(=O)NC(C2CN(C(C(C)(C)OC(C)=O)=O)C2)C)CC1C1CCCC1 45341,c1(C(=O)NC(CC)CNC(C2(Cl)CC2(F)F)=O)cccc(-c2cscn2)c1 45342,C1(CNC(CC2CCCN(C)C2)=O)CN(C(=O)CCc2cn(C)nn2)C(C)(C)C1 45343,CCC(C)C(O)C(=O)NCC(C)(C)CN(C)C(c1ccccc1SC)=O 45344,C(=O)(C(CC(F)(F)F)c1ccc(F)cc1)NCCCCNC(CC(=C)Br)=O 45345,c1(CC)[nH]nc(C(N2CC(OCCNC(c3cccnc3C(F)F)=O)C2)=O)c1Cl 45346,N1(C(CC2CCN(C)CC2)=O)CC2CCN(C(c3ncc(F)cc3F)=O)C2C1 45347,C(=O)(C(O)CC(F)F)NCCCC1N(C(c2c(OC)n[nH]c2)=O)CCC1 45348,CC1(C)CN(C(=O)CCCC(F)(F)F)C(CNC(=O)CCn2cccc2)CO1 45349,CC1CC(NC(=O)NC(C)(C)C(F)(F)F)CN1Cc1ccccc1 45350,c1(C(=O)OC)cc(C(=O)NCC(CNC(c2cc(Cl)c[nH]2)=O)CO)no1 45351,C(=O)(C(C)(O)CCc1ccccc1)NC1CC(NC(C(CC=CC)C)=O)C1 45352,C1(C(=O)NCCC(CNC(CN2CC(C)C2)=O)O)CCCN1C=O 45353,C1(C(=O)NCC2C(CC)C2)CN(C(c2ccncc2N)=O)CC(C)(C)C1 45354,CC1CCC(NC(=O)C(=O)C=Cc2ccc(F)cc2)CN1C(C1CCCSC1)=O 45355,c1(OC)ccc(F)c(C(=O)NCC(O)CN(C(=O)CC2CCC(O)C2)C)c1F 45356,N12CCCCC(C1)CCC2=O.N1(C(Cc2n(C)ccn2)=O)CCOC(CO)C1 45357,N1(C(C(C(=O)Oc2ccc(C)cc2)(C)C)=O)CCc2c(CO)ccc(C)c2C1 45358,C1(NC(C2(C=C)CCOCC2)=O)C2CCN(C(C3(C#N)CCC3)=O)CCC12 45359,CC(C)(C)C(C(=O)NC1(CCOCc2ccccc2)CC1)C1CCCC1 45360,C1(C(=O)NCc2c(C)occ2)CCCN1NC(=O)CCCn1cncn1 45361,C1(N(C(c2c(COC)cco2)=O)C)CCCN(C(C2CCCOC2)=O)C1 45362,c1(C(C)(C)C)cc(C(=O)NC2CCCC(NC(C3(C)CC=CCC3)=O)C2)ccn1 45363,C1(CNC(=O)Cc2ccsn2)CCN(C(c2ccnn2C2CCCC2)=O)CC1O 45364,C1(C(=O)NC(C(=O)NCC(C2CC2)OC)C2(C)CC2)CC12CCCCC2 45365,N1(C(CN(C2CC2)CC)=O)CCCC1CC(=O)NCC1(C)CCCS1 45366,C1(NC(CCSC)=O)CCN(C(C2CNC(=O)N2C)=O)C12CCC2 45367,CCCCC(CNC(=O)CCCc1sccc1C)NC(C1(C)CC1(F)F)=O 45368,c1(C(N2C(CCCNC(c3c(OC)ccs3)=O)CCC2)=O)cccc2c1CCO2 45369,c1(C(=O)NC2CN(C(c3c(C)sc(Cl)n3)=O)CC2C)ccc2cnoc2c1 45370,c1(OC)c(Br)cc(CN2CCC(CC(N3CCCC(F)C3)=O)C2)cc1Br 45371,C(=O)(C(C)(C)c1ccn(C)n1)NC(C)CCNC(c1ncnn1C)=O 45372,Cc1nc2cc(C(=O)NCCCC(C)NC(=O)CC(C)C3CC3)cnc2[nH]1 45373,C1(CN(C(=O)C(c2cccnc2)O)C)CCCCN1C(=O)CC1C=CCC1 45374,N(C1CCSc2ccc(Cl)cc21)CC(=O)Nc1cccc(NC(C)=O)c1 45375,CC1CN(C(=O)CC2C3CCC(C3)N2C(=O)C(C)OC(C)(C)C)C(C)C(C)(C)O1 45376,c1(C(N2CC=C(CNC(C(C)OC)=O)CC2)=O)cnc2c(c1)COC2 45377,c1(C(=O)NC(CNC(CCCC)=O)C)ccc(OCC)cc1F 45378,N1(C(c2c(CC)ccs2)=O)CCN(C)C(C(=O)NCCc2ccccn2)C1 45379,C1(COC)(CNC(=O)CSc2cccs2)CCN(C(C2(C(C)C)CC2)=O)C1 45380,C(=O)(C(C(=O)OC(C)(C)C)C(C)(C)C)NCC1CN(C(C(C(CC)O)(F)F)=O)C1 45381,c1(SCC)ccc(C(N2CCOC(CCNC(C3(F)CCC3)=O)C2)=O)cn1 45382,Cn1cc(C(=O)NCCC2CCN(C(=O)CCCC#N)C2)c(=O)c(Br)c1 45383,NS(=O)(=O)c1ccc(F)c(C(N2CC3(C(=O)NCC(F)(F)F)CC2CO3)=O)c1 45384,CCC(C)CN=c1[nH]c2c(c(=NCc3ccc4nn[nH]c4c3)[nH]1)CCCCCC2 45385,N1(C(C2CC3(CC3)CO2)=O)CCCN(C(=O)C(F)(F)CO)CCC1 45386,C(=O)(CC(Cc1ccccc1)CC)NCCC(=C)CNC(c1cnc(C)[nH]1)=O 45387,C(C(C)(CCO)NC(=O)C(C)CNC(c1sccc1CO)=O)OC 45388,c1(C(N(CCC(C(C)(C)C)NC(C(CO)OC)=O)C)=O)ccc(F)c(F)c1F 45389,N1(C(C2CC(C(=O)OC(C)(C)C)C2)=O)CC2CCC2(NC(=O)C(Cl)=CCl)C1 45390,N1(C(c2n(CC)ccc2)=O)CCC(=CCNC(=O)Cc2cccc(SC)c2)CC1 45391,C1(C(N(C)CC)=O)CN(C(C2(CC=CCNC3CC3)COC2)=O)C1 45392,N1(C(CC(C)(C)C)=O)Cc2cccc(CNC(=O)CC3CCCCC(=O)N3)c2C1 45393,c1(CCC(N2CC(N(C(c3c(OC)ccs3)=O)C)C2)=O)cccc2ccccc12 45394,S(=O)(=O)(c1cccc(CNC(=O)COC(=O)CC2CCC2C2CC2)c1)N(C)C 45395,N1(C(c2nc(Cl)cs2)=O)CCOC2(CCN(C(C3CCn4nncc4C3)=O)C2)C1 45396,Cc1ccc2cc(C(=O)NCC3C=CC(NC(=O)C(C#N)C(C)C)C3)[nH]c2c1 45397,c1(CC)ncccc1NC(=O)CCCN(C(=O)COC1CCOC1)C 45398,C1(NC(CC2(C)CC2F)=O)CCC(NC(c2ccc(NC(N)=O)cc2)=O)CC1 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45467,c1(C(N2CC(C)(NC(C3CCC(CCC)C3)=O)C2)=O)ccc(C)cn1 45468,CC1C(NC(=O)Cn2cncn2)CCCN1C(=O)C(=O)Nc1cnn(C)c1 45469,C1(C(=O)Nc2ccccc2-n2cc(C3CC3)nn2)CCc2ccccc2C1 45470,N1(CC(c2ccc(SC)cc2)C)CCS(=O)C(C)C1C 45471,N1(CC(=O)NCCNC(C(CN(C)C)O)=O)CCC(Cc2cccs2)CC1 45472,N1(C(Cc2cc(C)no2)=O)CCCC(C2CC2NC(c2cncc(C)n2)=O)C1 45473,C(=O)(C1=CCCCC1P(C)(C)=O)NCCCCN(C)C(C1Cc2nccn2C1)=O 45474,c1(C(COC(C(C)(C)c2csc(C(F)(F)F)n2)=O)F)cccc(F)c1 45475,C1(CC(=O)NC(CC(=O)NC)(C)C)CN(C(=O)CC(C)(C)C)CC12CC2 45476,c1(C(=O)OC)ccc2[nH]nc(C(=O)NCCNC(=O)C(O)C(C)SC)c2c1 45477,C1(NC(c2c(CNC(C3(C)CC(C)OCC3)=O)nnn2C)=O)CC(C)N(C)CC1C 45478,C1(C(=O)NC2(OCc3ccccc3)CCC2)CCCN1C(C1CCCC1)=O 45479,Cc1cc(C(=O)NCC(C)NC(=O)Cc2cc[nH]c(=N)c2)c(C)cn1 45480,C1(C)(CCOC)CN(C(c2ccc(F)s2)C(=O)NCCC2(C)CC2)CCO1 45481,CC(CN(C(=O)CC(C)n1ccnc1)C)C(=O)NC1CC(NC(N)=O)C1 45482,N(C(=NCc1ccco1)NC1CN(C2CCOCC2)C1)Cc1nc(CC)on1 45483,C1(CC)CN(C(=O)Cn2cc(C)cn2)CCC1CNC(=O)CSC 45484,CC1C(NC(=O)C=Cc2cn(C)nn2)CCN1C(=O)CC1OCCO1 45485,Cc1ccc(C(=O)NCC2CN(C(=O)C(O)CC(C)C)CC(C)(C)C2)c(F)c1F 45486,c1(N2CCC(CC)CC2)nc(N2CCC3C(CCN3C)C2)nc2sccc12 45487,C1(NC(=O)CC2NC(=O)NC2=O)CC12CCN(C(=O)C1=CCOCC1)C2 45488,C=Cc1cncc(C(=O)NCCC2CN(C(=O)C3=C(C)OCC3)CC(C)O2)c1 45489,C(=O)(C(C(=O)OC)OC)N1C(C(C(=O)NCCC=CC)(C)C)CCC1 45490,C1(CC(=O)NC(CC=C)C)CCCN(C(=O)C(C)(CO)OC)CC1 45491,c1(CC)cc(C(=O)NCC2C(CNC(c3cc(CN(C)C)on3)=O)C2(F)F)no1 45492,C=C(C)C1CN(C(C2CCCN(C(c3n[nH]c(C)c3O)=O)CC2)=O)CCO1 45493,c1(CN2C(CNC(=O)C=Cc3cccnc3)CCC2)cc(Br)ncc1Br 45494,N1(C(CC(C)CF)=O)CCN(C(c2cccn2Cc2cccs2)=O)C(C)C1 45495,CCC(O)(CC(=O)NC1CCC1CNC(=O)C=CCO)c1ccccc1 45496,C1(CC(=O)NCCOCCOCCNC(=O)Cc2ccc[nH]2)CC(O)C12CCC2 45497,c1(NC(C(C(C)OC)NC(c2csc(=N)[nH]2)=O)=O)cnn2c1CCCC2 45498,C#CC1(C(N2CC(O)(CCNC(c3[nH]ccc3C)=O)C2)=O)CCCC1 45499,C(CC(C)C)(C(=O)NCCC1(OC)CN(C(=O)C(C)NC(=O)OC)C1)OC 45500,c1(C(=O)NC2CC(CNC(CCOC(C)=O)=O)C2)ccn2nnnc2c1 45501,N1(C(C2N(C)CC(C)(C)C2)=O)CCOC2(C1)CN(C(C1(C)CCNC(=O)C1)=O)C2 45502,C1(C(N(CC(CC)NC(C2(C)C(C)(C)C2(C)C)=O)CC)=O)CC2CCC(C1)C2O 45503,CC1CN(C(=O)CC(C)c2ccccc2)CC1NC(=O)CC(F)(F)Cl 45504,c1(CNCC23C(CN(C(C4CC(O)C4)=O)C2)C3)cccc(F)c1Cl 45505,O=C(C1CCCn2ccnc21)NCC1(F)CN(C(C2C3CCCCCC23)=O)C1 45506,N1(C(CNC(c2c(C)occ2)=O)=O)CCN(C(=O)CC2(C3CC3)CC2)C(C)C1C 45507,C(=O)(C1=CCC(F)(F)CC1)N1CC(CNC(=O)C=CC2CCCO2)OCC1 45508,CP(C)(=O)CCC(=O)NC(c1cccnc1)C(=O)NCC#CC#CCO 45509,C1(CC(=O)NC(CC)COCC2CC2)C2CN(C(=O)C=NOC)CC12 45510,C1(OC)CN(C(c2conc2C(C)(C)C)=O)CC1NC(=O)C=CSc1nc[nH]n1 45511,c1(C(N2CC(C)(NC(=O)Cc3cccnc3)C2)=O)cncc(N)c1 45512,N#CC1(C(=O)NCc2csc(C(=O)NCCC(O)C3CCCC3)c2)CCCC1 45513,C1(F)(CNC(=O)CCCN2CCCCC2)CCN(C(=O)CC2CCC(=O)N2)CC1 45514,C#CCC(C)(CC)C(=O)NCC(=O)NCc1nccn1C1CC1 45515,C1(CCNC(C(F)=C(C)C)=O)CN(C(=O)CCN2C(=O)CCC2=O)CC(C)O1 45516,c1(NC(c2n(CCCSCC)nnn2)c2nc(C)co2)ccc(Cl)c(N(C)C)c1 45517,N1(Cc2nc(C)sc2)CCCC(NC(=O)NCC2COCCO2)C1 45518,N1(C(CP(C)(C)=O)=O)CCN(C(=O)CCCn2cccn2)CC1c1cn[nH]c1 45519,C(C)(CCC(=O)N1CCN(CCCCCNC(=O)COCCC(C)C)CC1)SC 45520,c1(C(=O)NC(C)CCCNC(=O)C2CC2)cnccc1C(F)(F)F 45521,c1(CNC(C(C)OC2CCCCC2)=O)n[nH]c2c1CN(C(=O)C1=CCOC1)CC2 45522,N1(C(c2cc(OCC)cc(F)c2)=O)CCC2(CCCN(C(=O)C(C)(C)CF)C2)C1 45523,c1(NC(=O)OC(C)(C)C)ccc2c(c1)CC(C)N2C(c1c(OC)cccc1)=O 45524,Cc1ccc2oc(C(N3CC(NC(c4cn(C)c(=O)n4C)=O)C(F)C3)=O)cc2n1 45525,C12(CNC(c3c(C)sc(O)n3)=O)CCC(CNC(=O)Cc3csnn3)(CC1)OC2 45526,Cc1cc(C(=O)NCC(N2CCN(C(=O)CS(N)(=O)=O)CC2C)=O)ccc1[N+](=O)[O-] 45527,CC(CCNC(C1(CNC(=O)CC2CCOC2=O)CCCC1)=O)C(C)(C)C 45528,Cc1cccc(Cl)c1S(=O)(=O)N1CCN(Cc2cc[nH]n2)C2CC12 45529,C1(C(=O)NC(CNC(C(C)SCC)=O)CC(C)C)COC2COCC12 45530,C1(C(=O)NC2CCN(C(CC(C=C)(C)C)=O)C23CCC3)CCc2nnc(O)n2C1 45531,C1(C(=O)NC2CC(NC(C(CCC)NC(C)=O)=O)CC2O)CC2CCCC(C1)C2 45532,n1(CC)nc(C2CC2)cc1S(=O)(=O)NC1(CC2CCCC2)CCCC1 45533,N1(C(c2cnc(NC(C)=O)o2)=O)CC(NC(=O)C(C)(C)N2CCCCC2)C2CC12 45534,C1(C(N2CCOC(C(N)=O)C2)=O)CCOCCN1C(C1CC(=C2CCC2)C1)=O 45535,C1(c2nc(C(F)F)sc2)CCC(F)(F)CC1.c1(CC)ncno1 45536,N1(C(CC(CC)C)=O)CC(NC(C2CC3CCC2CC3)=O)CC(C)(C)C1 45537,c1(-c2scc(C(=O)NCCCCC#C)n2)cnn2c1CCCC2 45538,N1(C(C2C(CCC)C2)=O)CC2CC(NC(=O)CN3CC4CC4C3)CC(C2)C1 45539,CCC(C(=O)NC1CCSC12CN(C(=O)Cc1cnn(C)c1C)C2)C(C)(F)F 45540,C12(C(N3CCC(N(CC#C)C(C4CCC(C)O4)=O)CC3)=O)CCC(N=[N+]=[N-])C1C2 45541,C1(C(N(C(CN(C(c2c(C)nn(C)c2C)=O)C)C)C)=O)C2CC3CC(C2)CC1C3 45542,CS(=O)(=O)c1ccsc1C(=O)NC1C2CC1N(C(C1(C#N)CC13CCC3)=O)C2 45543,C(=O)(C(O)C(C)(C)C)NCCn1cc(C(N(CC#C)C)=O)nn1 45544,C1(CN(C)C(C2CCC(=O)NC2)=O)CCCN(C(C2CCC(F)(F)C2)=O)C1 45545,c1(C2C(C(N3CC(OC)C(NC(C4CC(O)C4)=O)C3)=O)C2)cc(Cl)ccc1Cl 45546,C(=O)(C1=COCCO1)N1CCC(CCCCCNC(C2CCCS2)=O)CC1 45547,c1(C(=O)NCC2N(C(C(C)(Cl)Cl)=O)CC2)cc(C2CC2)oc1C1CC1 45548,Cc1cccnc1C(C1CCCN(C(c2ccnn2C2CCCC2)=O)C1)O 45549,C1(C(=O)NCCCNC(C(C)Oc2ccc(F)cc2)=O)CCc2ncccc2C1 45550,C1(C(=O)OCc2nnnn2-c2ccccc2)CCc2cc(F)ccc2O1 45551,CCCC(C(=O)N1CCCC1(CCC)CO)NC(C1CCC(=O)N1)=O 45552,N1(C(c2c(C)ncs2)C(=O)NCCC2CC2)CCCCC1Cc1cccc(Cl)c1 45553,CC(C)(C)C(C)(C)C(=O)NC1CCC(NC(c2[nH]nnc2C2CC2)=O)CC1 45554,C1(C(=O)NCC=CCNC(C(c2c(F)cccc2F)C)=O)CC2CCCC(C1)C2 45555,c1(C(N(CCC)CCc2ccccc2)=O)nccc(OC(C2CCCC2)C)n1 45556,c1(CC)cncc(C(N2CC(CCNC(=O)C(CC)NC(N)=O)C(C)C2)=O)n1 45557,C1(C(=O)NC2CN(C(c3ccccc3Br)=O)CC2O)Cc2ccccc2CO1 45558,Cc1ccc(C=CC(N2CC=CC(C(=O)NCC3CCOC3C)C2)=O)cc1 45559,C(C1COC(C)(C)O1)=CC(=O)NC1CC(C)(NC(C(C=C=C)C)=O)C1 45560,c1(CC)cnc(Cl)nc1N(C)CCOCCN(C)C(C1CCC2CC2C1)=O 45561,CCCC(CCC)=CC(=O)NC1CN(C(=O)Cc2ncccc2C)C2CC12 45562,Cc1ccccc1SCC(=O)NCC1CCCCN1C(=O)CC(C)C1CC1 45563,c1(C(N2CCC(C(F)F)(CNC(C3CCO3)=O)C2)=O)c[nH]nc1[N+](=O)[O-] 45564,N1(C(CNC(CCC)=O)=O)CCC(NC(C2CC2c2c(F)cccc2F)=O)C(C)C1 45565,c1(CC(C(N2CC(n3cc(CN)nn3)(C(=O)OCC)C2)=O)C)ccc(O)c(F)c1 45566,Cc1ccc2nc(C(=O)NC3(CNC(c4nc(C)oc4C)=O)CC3)c(N)n2c1 45567,c1(C(=O)NCC2N(C(C(CC)n3cccn3)=O)CC2)ccccc1-n1cnnn1 45568,C=C(C)CC(C(=O)NC(c1cncs1)C)NC(C1CC2CC(=O)C1O2)=O 45569,C(N=c1[nH]c(=NCCc2csc(=N)[nH]2)[nH]c2cc[nH]c12)c1nccc(NC)c1 45570,C12(C(=O)NCCC(O)C(F)F)CCC(CC1)N(C(C1(CO)CCCCC1)=O)C2 45571,C(C(C(=O)N(C1(CO)CC1)C)SC)CCC1CCC1.C1(=O)CC2CC2N1 45572,c1(CC(=O)NC2C3CN(C(c4c(C)cc[nH]4)=O)C2C3)ccc2c(c1)CC(C)O2 45573,C1(C(=O)NC(CNC(c2cc(Cl)c(Cl)[nH]2)=O)CO)CCC2CC2CC1 45574,c1(C(=O)NC(CC=C)CNC(=O)C(c2ccc(Cl)cc2)O)c[nH]c2nccc-2c1 45575,c1(OC(C)C)cnc(C(=O)NC2CCC(CNC(c3cc(N)ccn3)=O)C2)cn1 45576,C(=O)(C1=CCN(C(=O)C(c2cnn(C)c2)=O)CC1)NC(CC(CC)C)C 45577,CCCC(CC(=O)NC1CCC(OC)CC1)NC(c1cc(C#N)oc1C)=O 45578,c1(OCC(=O)NCCCN(C(=O)CCc2ccncc2)CC)cnn(C)c1 45579,C(=O)(CS(F)(F)(F)(F)F)NCC1(C)CCN(C(C(C)OC)=O)C1 45580,CN1CCC(NC(=O)C=CCF)C12CCCN(C(=O)Cc1ccn(C)n1)C2 45581,Cc1c(C(N2CCOCC2CNC(c2cccc(Cl)c2)=O)=O)ccn1C 45582,c1(OCCOC)ccc(C(=O)NCc2cccnc2NC(=O)C(O)CSC)cn1 45583,Cc1ccnc2ccc(C(=O)NCCCOCCNC(C3CCC(=O)N3)=O)cc12 45584,c1(C(=O)NC2CC(C)(NC(=O)CCc3ccncc3)C2)ccc([N+](=O)[O-])cc1 45585,N1(C(CN(C(C(C)(C)OC(C)C)=O)C)=O)CCN(C(c2nc(Cl)cs2)=O)CC1 45586,C1(CC)CC2(CCN2C(c2cn(C)nc2Cl)C(=O)NC2CCCC2)C1 45587,C1(NC(CCC(C)SC)=O)CCN(C(c2cc(F)c(F)cc2Cl)=O)CC1(C)C 45588,N1(C(CC(C)O)=O)CC2CCC(N(C(=O)CCc3cnn(C)c3)C)C2C1 45589,CC(C)C(=O)NNC(=O)C1CCN(C(C2(C(N3CCCC3)=O)CC2)=O)CC1 45590,CCC(C(=O)NC(CNC(c1cccc2c1CCO2)=O)CO)C(C)(F)F 45591,c1(CC(=O)NCC=C2CCN(C(C3CN(C)C(=O)C3)=O)CC2)ccnc(Cl)c1F 45592,C1(C(N(C)CC2(NC(c3csc4nccn34)=O)CC2)=O)CCCCC12CCC2 45593,CCCCCCC(C)NC(=O)C(=O)Nc1cc(-c2ccccc2)nn1CC 45594,N1(C(c2cncc(NC)c2)=O)CCC(CCNC(c2coc(Cl)n2)=O)C(F)(F)C1 45595,Cc1c(C(=O)N(CCNC(C2(CO)COC2)=O)CC2CC2)sc2cccc(F)c12 45596,C=CCCCCC(=O)NCC=CCNC(=O)CCCSc1ccccc1 45597,CS(=O)c1ccc(CC(N2CCC(NC(C3CC(C)(O)C3)=O)C2)=O)cc1 45598,c1(C(=O)NCC2CC(OC)CN2C(=O)C(O)CCSC)cc(S(N)(=O)=O)oc1C 45599,N1(C2CCN(C(C(C)(C)OC)=O)C2)CCN(C(=O)CC2(C(F)(F)F)SCCS2)CC1 45600,c1(CC(=O)NCC(CC=C)NC(C2ON=C(C)C2C)=O)cccc(Cl)c1 45601,C1(C(=O)NCC2C=CC(NC(C(C)c3ccsc3)=O)C2)CC2(C1)CC2(F)F 45602,C1(C(=O)NCC2CCN(c3ncc(Br)cn3)C2)CCc2n[nH]cc2C1 45603,c1(CC)ccc(NC(c2c[nH]nc2CNC(c2cnc(C)nc2C)=O)=O)c(F)c1 45604,Cc1nccnc1C(=O)N(C)CCNC(=O)CC(C)Cc1cccc(F)c1 45605,N1(C(c2ccc(COC)o2)=O)C2CCC1(CNC(C1CC(SC)C1)=O)CC2 45606,C12(CC(=O)NCCC3CCN(C(=O)CCc4ccncc4)C3)CCC(CC1)OC2 45607,Cc1c(C(N2CCCC(N(C(=O)C#CC3CC3)C)C2)=O)cc(N)cc1O 45608,C(CC1CCCO1)N=c1[nH]c2ccc(S(=O)(=O)N3CCSCC3CCO)cc2[nH]1 45609,CC1(C)COC(C(=O)NCC2CCC(C(=O)NCCCN3CCCC3=O)CC2)C1 45610,C(=O)(C(C)(O)C1CC1)N(CC(C)NC(=O)Cc1n[nH]cc1Br)C 45611,N1(CCCc2ccc(C)cc2)C(=O)CN(CCc2ccc(F)cc2F)C1=O 45612,C1(F)(CNC(CCc2nc(C)c(C)[nH]2)=O)CCCN(C(=O)CCC(C)(F)F)CC1 45613,n1(CC)ncc(Cl)c1C(=O)NC1(C(=O)NCC2CCC(C)CC2)CC1.C(C)(=O)O 45614,N1(C(C(C)(C)n2cc(Cl)cn2)=O)CC2C(C(=O)NCCC3(C)CC3(F)F)C2C1 45615,C1(CC(=O)NC)CN(C(C2CN(C)C2)=O)CCN1C(C1CC=CCO1)=O 45616,c1(CC(=O)N(C(CNC(CSC)=O)C)CC)cc(Br)ccc1Cl 45617,c1(C(N(CCCOCCNC(c2ccc(SC)o2)=O)C)=O)nc(C)ccc1F 45618,C(CC(=O)NNS(=O)(=O)c1ccncc1)Sc1c(OC)cccc1 45619,C1(NC(C2C(C)CC2C)=O)(COc2ccccc2C(N)=O)CC2(C1)OCCO2 45620,c1(C(N2CCC(C(C)(C)C)(CNC(CS(CC)=O)=O)C2)=O)cccc(F)c1O 45621,c1(C2CCCN(C(c3ncc(I)s3)C(=O)NC(C)(C)C)C2)ccc(F)c(F)c1 45622,n1(CC)cnc2c(NCCCC(C)NC(=O)COc3ccccc3)nc(Cl)nc12 45623,CCCCS(=O)(=O)CC(=O)NC1CN(C(=O)COc2c(Cl)cccc2Cl)CC1C 45624,c1(CC)ncc(CNC(=NC)NCc2ccc(OCC(C)C)cc2)n1C 45625,C1(CNC(C2(SC)CC2)=O)CCCCN(C(c2ccc(N)cc2Cl)=O)C1 45626,CN=c1[nH]cc(C(=O)NC(CC)C(N2CC3C(C(N)=O)C3C2)=O)o1 45627,c1(C(=O)NCC2CC(C)(C)CN2C(c2cnccn2)=O)cc2ccccc2[nH]1 45628,c1(SCC(N2CC3C(NC(Cc4c(CC)con4)=O)(C3)C2)=O)cc(F)ccc1F 45629,Cn1ccc(C(=O)NCC2CCN(C(C3CC4CCC3O4)=O)C23CC3)cc1=O 45630,C1(NC(CC=C(C)C)=O)CS(=O)(=O)CC1NC(=O)CS(=O)(=O)NC(C)(C)C 45631,c1(OC)cc(C(N2CC3CC(NC(C4CCOC4)=O)C3C2)=O)ccc1C 45632,Cc1ccc(-n2cc(C(C)N(C)C(c3cccc(SCC#N)c3)=O)nn2)c(F)c1 45633,N1(C(c2ccc(C)cc2C)=O)CCCC(F)(CNC(=O)C(O)C(C)(C)C)CC1 45634,C1(C(=O)NCc2cc(C)c(C)s2)N(C(C2CCCC(CF)C2)=O)CCCC1(C)C 45635,N1(C(C(C2CC(NC(C(CC=C)OC)=O)C2)F)=O)CCC12CN(C)C2 45636,c1(CC)ccnc(C(=O)NC(CNC(C2CC23CC(OC)C3)=O)CC(C)C)c1 45637,C1(CNC(C23OC(C)C(C2)C3)=O)(CO)CCN(C(=O)C(O)CC(N)=O)CC1 45638,N1(C(CCC(=C)Br)=O)CC2CC(C1)CN(C(=O)CCC(CC)OC)C2 45639,CCCC(C)(C)C(=O)N1CCCCC(CNC(=O)C(O)CCSC)C1 45640,C1(NC(C(C2CCOCC2)C)=O)CC(C(=O)N(C2(C3CC3)CC2)C)=NO1 45641,c1(OC(C)C)ccc(C(=O)NC2CCCCC2CNC(c2ccnnc2O)=O)nn1 45642,C12(C(=O)NCCCN(C(C3CSC3)=O)C3CC3)CC3CC(F)(C1)CC(F)(C3)C2 45643,c1(C(=O)NC(c2ccc(-c3c(OC)cc(C)cc3)cc2)C)ccc2cncn2c1 45644,C(C)(CC(=O)NC(c1nocc1C(=O)N(C)Cc1ccn(C)n1)C)SC 45645,Cn1ncc([N+](=O)[O-])c1C(=O)NCC(=C1CN(C(c2cc(Cl)cc(Cl)n2)=O)C1)F 45646,CC12CC(CC1C(=O)N(CCCNC(C1(O)CCOCC1)=O)CC1CCCC1)C2 45647,n1(CC(=O)NCC(C)(C)NC(C2C(OCC)C2)=O)c(C)cc(O)cc1=O 45648,N1(C(c2c(F)ccc(C#C)c2)=O)CC(C)OC2(CCN(C(=O)CC3CCC3)C2)C1 45649,C(=O)(CCCS(N)(=O)=O)N1CC(NC(C2(C#C)CCC2)=O)C(C)C1 45650,c1(C(=O)NC(C(C)NC(Cc2c(C)noc2C)=O)C)ccc2nsnc2c1 45651,Cc1cnc(C(C)(C)NC(C2CS(=O)(=O)C2)=O)s1 45652,n1(CC)ccc(C(=O)N(CCCNC(c2cc(C)cs2)=O)CC2CCCC2)n1 45653,C1(CNc2cncc(C(C)NC(=O)OC(C)(C)C)c2)CCN(C)C(C)C1 45654,C(C(C)CC(=O)NCC1CCC(CN(C(=O)CCOC2CCC2)C)CC1)OC 45655,Cc1ccc(F)cc1C(=O)NCC(O)CCNC(c1csc(C(F)F)n1)=O 45656,C#CCC(CC)NC(=O)CCNC(C1(CO)CCCC1)=O 45657,C1(NC(CN2C(=O)NCC2)=O)CCN(C(C2CC3C=CC2C3)=O)C12CCC2 45658,C1(CN(C(C(n2c(C)ccn2)C)=O)C)CN(C(=O)CC2CC2(C)C)CC12CC2 45659,c1(C(=O)NC2CCCN(Cc3ncc(C)nc3)C2C)cnc2c(C)cccc2c1 45660,S(=O)(=O)(c1cccnc1N1CCS(=O)CC1)NCC(c1ccc(F)cc1)CC 45661,N1(C(C=C(CC)CC)=O)CCN(C(c2cc(N)c(Cl)cn2)=O)C2(CC2)C1 45662,N1(C(CC=C(C)C)=O)CC(F)(F)CC1CCNC(c1coc(Br)n1)=O 45663,C1(NC(C(=O)Nc2cnn(-c3ccc(C)cc3)c2C)=O)CCCCCC1C 45664,C1(OCCC)CN(N2CC(OCC)C2)C1.N(C)C 45665,C=C(Cl)CC(C(=O)N1CC(CO)C1)NC(=O)CNC(C)=O 45666,CCCCCCCCNC(=O)CC1CC(F)CN1C(c1cc(F)c[nH]1)=O 45667,c1(SC)cncc(C(=O)NCC=C2CCN(C(=O)CCn3cc(C)cn3)CC2)c1 45668,C#Cc1cc(OC)cc(C(=O)NC(C)(C)C(C)CCC)c1 45669,C1(NC(CCCOC(C)C)=O)CCC(CNC(c2csc(S)n2)=O)CC1 45670,c1(C(C(N2CCC(NC(C34CC(F)C3C4)=O)C2)=O)O)ccccc1Cl 45671,C1(C)(CNC(c2c(C)cc(=N)[nH]c2)=O)CN(C(=O)CC2CC2(C)C)C(C)(C)C1 45672,N1(C(c2c(C)cn(C)n2)=O)CCC(NC(=O)C=Cc2cccn2C)CC1C 45673,C1(NC(C2CC3CCC2CC3)=O)CN(C(=O)C(C2CCCCC2)O)CC2(CC2)C1 45674,C1(C(=O)NC2C(NC(C3C(c4cn(C)nc4)C3)=O)CCC2)CCCCNC1=O 45675,Cc1ccccc1C1(C(=O)NC2COCC2NC(=O)CN(C)C2CC2)CCOCC1 45676,C12(C(CNC(c3cn(C4CC4)cn3)=O)NC(N3CC4CC4C3)=O)CCC(CC1)C2 45677,c1(C(N2C(CNC(c3c(C)cn(C)c3)=O)CC2)=O)nn(C)c(Cl)c1Cn1cncn1 45678,N1(C(C(CCOC)OC)=O)CC2CC1CC2CNC(c1cc(C)nn1C1CC1)=O 45679,C(C)(C)(C(F)(F)F)OCC(=O)N(CC(C)NC(=O)Cn1cc(C2CC2)cn1)C 45680,N1(C(C=CC2C(C)C2(Cl)Cl)=O)CC2(CCN(C(c3cc(C(N)=O)no3)=O)C2)C1 45681,c1(OC)cc(NCC2CC(NC(C3CN(C)C(=O)N3)=O)C2)nc(OC)n1 45682,C=C1CCN(C(c2ccn(CCNC(=O)Cc3nocc3C)c2)=O)C1 45683,C12(C(=O)OC)CN(C(C)=O)C(CNS(=O)(=O)CC3CCCC(OC)C3)(C1)C2 45684,C1(NC(C2(C=C)CCC2)=O)CCN(C(c2c(SC)cnn2C)=O)CC1F 45685,Cc1c(CNC(=O)CCC2CCCN2C(=O)C(C)(O)C2CC2)nnn1C 45686,Cc1nn(C)cc1CCC(=O)NCCOC1CN(C(C2(C)CC=CCC2)=O)C1 45687,N1(C(C)=O)CC(O)CC1C(=O)NC1CC(CO)C(O)C1.c1(C(=O)N)ncccc1Cl 45688,C(=O)(C1=CCCCCC1)N1C(C)CC(CC(=O)NCC2COCCOC2)C1 45689,C1(NC(CCC(C)OCC)=O)CCN(C(=O)C(COC)COC)CC12CCC2 45690,C(=O)(C1=C(C)OCCS1)N1CCCC(C(=O)NC2(SC)CCC2)C1 45691,N1(C(C(=O)NCC(C)N(C(=O)C(N2CCC(C)C2)=O)C)C)CCOCC1 45692,C1(OC)CC(NC(=O)CCCCCc2ccccc2)CN(C(=O)CC(C)F)C1 45693,N1(C(C(CC)C(C)C)C(=O)NCC(F)F)CCC2(CC1)C(C)(C)C21CCC1 45694,CC#CCCC(=O)NCC(C)(O)CNC(C1COCCN1CC(F)(F)F)=O 45695,N1(Cc2c(OC)cccc2)CCc2sc(-c3cncc(F)c3)nc2C1 45696,C12(C(N(C)CC3CCN(C(=O)C(O)CF)C3)=O)CCC(C(F)F)(CC1)CC2 45697,CON(CCO)C(=O)C(CCOCCO)NC(c1ccc(C)cc1O)=O 45698,N#Cc1ccc(N)c(C(=O)NCC2(F)CCC(NC(=O)C(F)OC(F)(F)F)C2)c1 45699,C1(C(=O)OC)CC2CCC(C1)C2NC(C1OCCC1C)=O 45700,c1(C(N2C3CCC(NC(C=C(CCC)CCC)=O)(C3)C2)=O)cccc2ccnn12 45701,c1(C(=O)NCCC(C)N(C(c2[nH]cc(C)c2C)=O)C)onc2ccccc12 45702,c1(C(N2C(C(N3CCC(O)C3)=O)CC3CC32)=O)cccc(C(F)(F)F)c1F 45703,CC(C(=O)NCC1CN(C(=O)Cc2nnc(S)n2C)CCO1)S(N)(=O)=O 45704,C12(NC(C(C)Cc3ccc(Cl)cc3)=O)CCC(C1)N(C(=O)CCC1CCCC1)C2 45705,O=C(C#CC1CCC1)NCC1(CNC(c2ccc(C(F)F)o2)=O)CCC1 45706,Cc1cc(Cl)c(C(=O)NCC2CCC2NC(=O)C(c2ccncc2C)C)c(Cl)c1 45707,Cc1cn2c(CC(=O)NC(c3ccc(F)cc3)CNC(c3ccsn3)=O)csc2n1 45708,C(CC1=CCN(C(c2n[nH]c(C)c2N)=O)CC1)NC(C1(CC)CCOCC1)=O 45709,C1(NC(CC2CC(=C)C2)=O)CCN(C(C2CC3CC3CC2C)=O)CC1F 45710,C#Cc1cc(NC(=O)C(C)c2cccs2)cc(F)c1.C1CN1C(C)=O 45711,N1(C(C(C=C)O)=O)CC(NC(=O)CC2CCOC2)CC12CCOCC2 45712,C(=O)(CC(C)C(C)(C)NC(C1CC(=O)N(CC)C1)=O)N1CCC(C#C)C1 45713,N1(C(c2cn(C)nc2-c2ccncc2)=O)CC2CCCC1(CO)C2 45714,C1(C(C#N)NC)CCOCC1.CCC(C)SCC 45715,c1(CC(C(=O)NCC(CSC)(C)C)NC(C23CC(CO2)C3)=O)ccccc1Br 45716,c1(OC)ccnc(Nc2ccccc2-n2cc(CN(C)CCO)nn2)c1 45717,C1(CNC(C2CNC(=O)N2)=O)CCCN(C(C2CC3CC3C2)=O)C1 45718,Cc1nc(C(=O)NCC2CCN2C(C2CCN(C(=O)OC(C)(C)C)C2C)=O)c(C)[nH]1 45719,C(=O)(CCCC(C)(C)C)NC(CC#C)CC(=O)NC(CC1CC1)CC 45720,C1(CNC(C2(C(N)=O)CCC2)=O)CC2CN(C(C3(n4cccn4)CCC3)=O)CC12 45721,CC(CNC(=O)C(=O)NCC(F)F)(C1CC1)NC(=O)COC1CCOC1 45722,C1(CC#C)(C(N2CCCC2CNC(C2COCCO2)=O)=O)CCCCC1 45723,O=C1CC2(CCN(C(=O)CC3CN(Cc4cccnc4O)CCO3)CC2)C(=O)N1 45724,C12(CNC(c3c(OCC)nccc3)=O)CCCC1N(C(=O)CSC(F)F)CCC2 45725,N1(C(C2CC(=C3CCC3)C2)=O)CCN(C(C2CCn3cncc3C2)=O)C2COCC12 45726,c1(C(=O)NCC2CCN2C(=O)COc2ccsc2)ccncc1F 45727,C12(C(=O)NCC3OCCN(C(C4CN(CC)C(=O)N4)=O)C3)CC(C1)S(=O)(=O)C2 45728,c1(CC(=O)N(CC(C)(C)CNC(=O)CC2(COC)CC2)CC)cn2cc(C)sc2n1 45729,Cc1ccc(C(N2CC3CCC(C2)N3Cc2c(F)cncc2F)=O)c([N+](=O)[O-])c1 45730,c1(C(=O)NC2(CO)CN(C(c3ccnc(C)n3)=O)C2)cccc2nccn12 45731,C1(CNC(N(C(C)CN)C)=O)CC(OCC(F)(F)F)C1 45732,N1(C(C(C#C)(C)C)=O)CCC2C(CCCN2C(c2ccc3c(c2)CCOC3)=O)C1 45733,c1(C(N2CCN(C(CC)CC)CC2)C(=O)NCCOC)ccc(SC)cc1 45734,C1(C(=O)NCC2CN(C(c3cc(OC)n(C)n3)=O)C2)CCCC(C)(C)O1 45735,Cc1nn2ccccc2c1C(=O)N(C)Cc1cn(Cc2cccnc2Br)nn1 45736,CCC(CNC(C1CCN(C)C1C)=O)(CC)C(=O)NC1CC(C)N(C)CC1C 45737,Nc1nc(C(N2CC3CC(NC(c4cc(C(F)F)cs4)=O)C2C3)=O)ccc1O 45738,c1(CCC(=O)NC2CC(F)(CNC(c3nc(COC)sc3)=O)C2)ccc(Cl)nc1 45739,C1(CCOC)(NC(C2CC2(C)C)=O)CCN(C(=O)C(C)C2CCC2)C1 45740,Cc1c(NC(C2CC2NC(C2(C(=O)C3CC3)CC2)=O)=O)cnn1C 45741,C(CO)(C(=O)NC1(CCO)CN(C(C2CC2F)=O)C1)OC 45742,Cc1ccc(CNC2CC2C(=O)Nc2ccc(C(N)=O)nc2)c(Cl)c1Cl 45743,C=C(Br)CCC(=O)NC1CCC(CNC(=O)C=C(C)C)C1 45744,C1(C(=O)NC2(CN(C(C=CSC)=O)C)CC2)CCC2CC2CC1 45745,C(=O)(C(=O)C(C)CC)NCC(COC)NC(C(C=C)CC)=O 45746,c1(C(=O)NCCC(=O)NCCNC2CC2c2cscn2)ccoc1C1CC1 45747,C1(O)(CN(C(=O)CC2CC23CC3)C)CCN(C(=O)Cc2cccc(Cl)c2)C1 45748,C(=O)(CCC(=O)NCC1CN(C(=O)CN2C(C)CCC2C)CC1C)NC 45749,N1(C(Cc2ccc(C)s2)=O)CC(NC(c2cc(C(N)=O)n(C)n2)=O)CC(C)C1 45750,CC1CN(C(c2ccc(CN(C)C)o2)=O)CC1CNC(c1ccsc1C#N)=O 45751,CC1CC(C(N2CCC(NC(c3nsnc3O)=O)C(C)C2)=O)CC(C)O1 45752,S(=O)(=O)(CCC(=O)NC1CC(NC(=O)C(O)C(C)(C)C)C(O)C1)NC 45753,N1(C(COC(CC)C)=O)CCC1C(=O)NCCC1(CO)CC1 45754,c1(NC(C2CC(NC(c3nc(CC)oc3C)=O)C(O)C2)=O)ccc(O)c(CO)c1 45755,N1(C(c2c(SC)cccc2)=O)CC2CCN(C(=O)C(F)n3cccn3)CC2C1 45756,Cc1ccc2c(N3CCCC4(CC4)C3)nc(=NCC3CCOC(CO)C3)[nH]c2c1 45757,c1(C(=O)NC2CCCC(NC(C3N(CC)CCC3)=O)C2)cc(C#N)oc1C 45758,CC1CCc2ncc(C(N3CC4CC(C3)N(C(c3occc3Cl)=O)C4)=O)n2C1 45759,N1(C(c2nc(N(C)C)oc2)=O)CCCC1(C)CNC(=O)CCS(C)=O 45760,C1(CNC(C(CC)C)=O)CCN(C(=O)Cc2cccc(NS(C)(=O)=O)c2)C1(C)C 45761,C12(C(N(CCCCCCNC(=O)C3=CCCSC3)C)=O)CC(C)(C1)OC2(C)C 45762,C1(C(N2CC3C(NC(C(=O)NCCOC)=O)C3C2)=O)CC(C)(C)CCO1 45763,C1(C(=O)NCCC(C=C)(C)C)CN(C(C2CCC(=O)N(C)C2)=O)CCN1C 45764,Cc1ccc(CCC(N2CC3(C2)CN(C(c2cccc(=O)o2)=O)C3)=O)c(C)c1 45765,CC1CN(C(=O)CC2CN(C)C2)CCN1C(c1coc(C2CCC2)n1)=O 45766,Cc1ccc(C(=O)NCC2(O)CN(C(=O)C(C)N3CCC3)C2)o1 45767,c1(C(N(CCCCN(C(C(c2ccnn2C)C)=O)C)C)=O)cc(O)nn1C 45768,C1(N(C(CSCC)=O)C)CCC2(CC1)CCN(C(=O)CC1CCCC(C)(C)O1)C2 45769,c1(C(N2CCCC(NC(c3n[nH]cc3[N+](=O)[O-])=O)C2)=O)cc(F)cnc1O 45770,c1(-c2cn(CC(=O)NCCCN3CCCCCC3)nn2)ncc(Cl)cc1F 45771,N1(C(CC2CCN(C(CC(COC)(C)O)=O)C2)=O)CC2(COCC(=O)N2)C1 45772,c1(CN(C(=O)NC(c2c(Br)cn(CC)n2)C)C)cccc2cnccc12 45773,c1(OC)cc2cc(C(=O)NOC(C)C)sc2cc1NC1CCNCCC1C 45774,n1(CC)cc(Br)c(C)n1.c1(N2CC(=O)NCCC2)ccccc1.SC 45775,c1(CNC(N2CC(C)(CCc3ccccc3)C2)=O)ccc(Cl)cc1F 45776,c1(C(N(C2CCN(C(c3ccco3)=O)CC2)CC#C)=O)csc2c1CCCC2 45777,c1(OC)ccc(Cl)c(C(N2CCC(C)(CCNC(C3CC34CC4)=O)C2)=O)c1 45778,N1(C(C2N(C(C)=O)CCOC2)=O)CCCN(C(c2ccc(Cl)o2)=O)CC1C 45779,n1(C(COCC)C)cc(-c2ncc(C(=O)O)o2)nn1.C12CC(C1)NC2=O 45780,C1(NC(c2c(CCC)occ2)=O)CN(C(c2ccnc(S)c2)=O)C2(CCOC2)C1 45781,CN1CCOCC1CC(N1CCC(CCNC(=O)C(F)C2CC2)CC1)=O 45782,C1(NC(Cc2c(C)nc[nH]2)=O)CC12CCC(NC(=O)CCC1(C)CC1)CC2 45783,C1(F)(C(N2CCC(NC(c3cc(OC)nn3C)=O)C2)=O)CC2(CCC2)C1 45784,C=C=C(C)CC(=O)N(C1CN(C(c2cc(-c3ccn(C)c3)[nH]n2)=O)CC1O)C 45785,N1(Cc2ccc(C)[nH]2)CCC(C(=O)Nc2cccc(Cl)c2O)C(O)C1 45786,N1(C(C(c2cn(C)nc2)=O)=O)CCc2ccccc2C1CCNC(C1(Br)CC1)=O 45787,N1(C(c2nc3ccccc3[nH]2)=O)CCC2C(CCN2C(C2CC2F)=O)C1 45788,CCCCC(O)C(=O)NCCC1CCCN1C(c1csc(-c2coc(=N)[nH]2)n1)=O 45789,O=C(CS(=O)(=O)CCO)NC1CCC(CNC(c2ccc(F)cc2F)=O)C1 45790,n1(CC(=O)NCC(CC)NC(=O)Cc2ccn(C)n2)c(-c2cccs2)nnc1S 45791,C(=O)(C(C)C(F)(F)C(F)F)N(CCNC(C1CC(SC)C1)=O)CCOCCO 45792,Cc1ccc(NC(N2CC(NC(=O)C(C)C)C3(CC3)C2)=O)cc1F 45793,C1(NC(C=CC(C)NC(=O)Cn2ccnc2)=O)CCCCC1(C)C 45794,CC1CCc2ccccc2N1NC(C1CCCC(NCc2ccc(Cl)cc2)CC1)=O 45795,C1(OC)(CNC(c2nocc2C)=O)CCN(C(C2COCCC2C)=O)C1 45796,N1(C(c2c(N)cccn2)=O)CC2CC(NC(=O)CCSc3ccccc3F)C1C2 45797,Cc1ccnc(C(=O)NC2CC2CNC(c2ccc(Cn3cccc3)cc2)=O)c1 45798,c1(OC)cccc(NC(=O)CC(C=O)NC2(C)CC(C)=NO2)c1 45799,C1(NC(CCCCCC#C)=O)CCN(C(=O)CC(C(F)(F)F)OC)C12CCCC2 45800,c1(CCC)ccc(CC(N2CC=CC(NC(c3cnc[nH]3)=O)C2)=O)cc1 45801,C1(CNC(C=C(C)C)=O)(NC(C2CNC(=O)N2)=O)CCC(F)(F)CC1 45802,c1(CC(=O)NCC2(COC)CCCN2C(=O)C=C2CCC2)ccc(Cl)nc1C 45803,CCC(CC)C(F)C(=O)NCC1CN(C(C2CC3(CCC3=O)C2)=O)C1 45804,c1(N2CC(C)C(NC(c3cc[n+]([O-])cc3)=O)CC2)nc(Cl)nc2c1COCC2 45805,N1(C(Cc2c(CC)nccc2)=O)CCCC(COC)(NC(=O)C(O)COC)C1 45806,N1(C(c2cnn[nH]2)=O)CCSCC1C(N1CC(c2ncccn2)C1)=O 45807,N1(C(CC=C)=O)CCCC(C)(CC(=O)NCC2CC2c2ccc(F)c(F)c2)C1 45808,S(=O)(=O)(c1ccc(Br)cc1NCC(C)C#N)NCc1c(C)nc(C)c(C)n1 45809,CCC(CC)(CCNC(=O)C=CC=C(Cl)Cl)NC(=O)CN1CCCCC1C 45810,C1(NC(C(=O)NCc2ccc(OC)cc2)=O)CCc2cn(CCC#N)nc2C1 45811,c1(-c2scc(OCC)c2)cccc2cc(C(N3CCCC4CCCCC34)=O)sc12 45812,C1(C(=O)NCC(N(C(c2cc(C)sc2)=O)C)C2CC2)CC2CC1CC2O 45813,C(=O)(C(O)C(CCC)NC(C1CN(C(C)=O)C1)=O)N(CCCC=C)CC 45814,C1(NC(C(=Cc2cccs2)C)=O)CN(C(=O)Cc2ccc(Cl)c(F)c2)C(C)(C)C1 45815,c1(C(=O)NCCN(CC(C)O)C(c2c(C#C)cn(C)n2)=O)cn2cc(C)sc2n1 45816,c1(CC(=O)NC(CNC(C2CN(C(CC)CC)C(=O)C2)=O)C)cccc(F)c1O 45817,c1(NC)cc(C(=O)NC2CCN(C(c3cccc(F)n3)=O)CC2CO)cc(Cl)n1 45818,c1(NC(C2CCCCN2C(c2ccc(CO)c(F)c2)=O)C)nc(Cl)nc2sccc12 45819,C1(NC(c2c(NC(c3cnc(OC)nc3)=O)cn(C)n2)=O)CCC(C2CC2)C1 45820,c1(C(=O)NC2(CNC(=O)COC(F)(F)F)CCOCC2)ccc2n[nH]cc2c1 45821,c1(CC(=O)NCCCNC(c2ccsc2Cl)=O)cc(Cl)ccc1O 45822,C(=O)(CCOC(C1CN(C(C2CC2C(F)(F)F)=O)C1)=O)OC(C)(C)C 45823,N1(C(C23CCC(OC)C2C3)=O)CCN(C)CC1C(=O)NCC(C1CC1)SC 45824,N1(C(c2c(C)cc[nH]2)=O)CCCC2CCN(C(c3csc4c3CCCC4)=O)CC12 45825,C1(CCN(C)C(C2(C3CC3)CCCO2)=O)CCN(C(C2C(Cl)(Cl)C23CC3)=O)CC1 45826,C1(NC(C2CCCNS2(=O)=O)=O)CN(C(=O)COC(F)F)CCC1F 45827,Cc1ccc(C#N)cc1NC(C1CCN(C(C2CCOC2(C)C)=O)CC1(C)C)=O 45828,C(=O)(CC(C)CC(F)(F)F)N(C(C)C)N(C1CCCCC1)Cc1ccn(CC)n1 45829,Cc1ccc(C(=O)N(C2CC(C)(C)C2)CC(C)CN2CCNCC2)c(C(C)C)c1 45830,c1(C(c2n(CC=C)nnn2)NCC(CO)C(C)(C)C)ccc2c(c1)CCO2 45831,c1(CC(=O)NC2C(NC(CC(=C=C)C)=O)CCC2)c[nH]c2c(F)cccc12 45832,N1(C(CCCCC)=O)CCc2nc[nH]c2C12CCN(C(c1cccc(N)c1)=O)C2 45833,CC1(C)C2CCC1(C(=O)NCC1CC(F)(CNC(C3CC34CC4)=O)C1)CC2 45834,CC(C(=O)N(C)CCOCCCN(C)C(C1(C#N)CC1(C)C)=O)C(F)F 45835,Cc1ccc2[nH]cc(CCNC(=O)NCC(N3CCC(CON)CC3)(C)C)c2c1 45836,C1(CN)CN(C(C2CC23CCOCC3)=O)CCC1(F)NCC1CCCCC1 45837,c1(CN2CCC(NC3(CC(=O)OCc4ccccc4)CCC3)C2)ccccc1 45838,Cc1cc(F)cnc1C(=O)NCCCC(C)(C)NC(C1CC2CCC1C2)=O 45839,C1(N(C(CC(C)F)=O)C)CCCCC1N(C)C(c1cc(-c2ccccc2)cs1)=O 45840,c1(CC(=O)OC(CCC=C)C)cc(Cl)cc2ccccc12 45841,c1(C(N2CC(C)CC(CC)C2)C(=O)NC2CC2)ccc(F)c(F)c1Br 45842,c1(OC)cc(C(F)CNCC2(C)CCCCCC2)ccc1Cl 45843,Cc1ncsc1C(=O)N(C)Cc1cocn1 45844,c1(C(=O)NCC2(NC(C3C(C)(C(F)F)C3)=O)CCC2)ccnc(-n2cccn2)c1 45845,C(C(=O)NNC(=O)C(C)(C)CCCCNC(=O)C(O)C1CC1)OCC 45846,C(=O)(CCCCC1CC1)NC(C#C)CNC(=O)CCc1cccnc1 45847,C(=O)(C#CC1CCCOC1)NC1(COC)CN(C(c2ccnn2C2CCC2)=O)C1 45848,C1(O)(CCNC(=O)CSC2CCS(=O)(=O)C2)CCCN(C(C2(O)COC2)=O)C1 45849,c1(C(=O)NC2C(NC(=O)CSC3CCCCC3)C2)ccncc1.C1(=O)CN1 45850,C1(CC(=O)NCCCN(C(c2cccc(COC)c2)=O)C)OCCCC1(C)C 45851,N1(C(CCOC)=O)C2CCC1(CNC(=O)Cn1cc(C3(O)CCC3)nn1)CC2 45852,N1(C(c2nc(CCC)oc2)=O)CCN2C(=O)C(NC(C3(N(C)C)CC3)=O)CC2C1 45853,N1(C(=O)CC2CCCCC2)CCCC(C2CN(C(c3cc(F)ccc3Cl)=O)C2)C1 45854,c1(CNC(C2(SC)CN(C(=O)CC3(C)OCCO3)C2)=O)cc(F)ccc1O 45855,N1(C(c2cccc(C(C)(C)C)n2)=O)CC(C2CN(C(C3(C)CC(C#N)C3)=O)C2)C1 45856,C1(C2CC2)(CNC(C2C3(CC(OCC)C3)C2)=O)CCN(C(=O)CN=S(C)(C)=O)C1 45857,C1(NC(=O)CC2CCN2C(=O)C=Cc2nccs2)CC(=O)N(C2CCCCC2)C1 45858,C12(C(N3CCN(C(C4CC(C)OC4)=O)CC3)=O)CCC(CC1)OC2 45859,C(=O)(C1CSc2ccccc21)NCc1c(OCC#C)nccc1 45860,N1(C(CC(c2ccc(F)cc2)NC(C2CCCCO2)=O)=O)CC2OCCOC2C1 45861,N1(C(C2(OC(C)=O)CC2)=O)CCC(C(N2CCOC(CN(C)C)C2)=O)C(C)C1 45862,C(C(C)(C)CNC(=O)CC1(C)CCOC1)N(C(COCC(=O)NC)=O)CC 45863,C=C(C)CCCC(=O)N1CCC(C(C)(C)NC(=O)C(CC)c2cccnc2)C1 45864,C12(C(=O)NCC(C)NC(=O)Cn3ncnn3)CC3CC(C(=O)N1)C2C3 45865,C=CCC(CNC(=O)C(C)(C)C)C(=O)NCC(Cl)C(C)(F)F 45866,Cc1cccc([N+](=O)[O-])c1NC(C)CN(C)C(C1CC2(CSC2)C1)=O 45867,C=CCC(CC)C(=O)N1CCN(C(C2(SCC)CC2)=O)CC1c1cccc(F)c1 45868,N1(C(c2c(O)ccc(C)c2)=O)CCC(C(=O)NC(C)Cc2cnc[nH]2)CC1(C)C 45869,C1(N(C(c2c(C(C)C)ncs2)=O)C)CCN(C(C2(c3ccncc3)CC2)=O)CC1 45870,CCC(CNC(=O)CCCCNC(=O)CN1CCCCC1C)CCO 45871,C=C(Cl)CC(C(=O)NCCCOCC(F)F)NC(c1cc(C)ncn1)=O 45872,c1(CNC(C2(OCC)CCC2)=O)cccc(O)c1C(=O)NC.c12cc(cn1C)N2 45873,c1(C(=O)OC)nc(N2CC(OC)C(F)C2)cc(C)n1 45874,Cc1ccc(C)c(CC(N2CCC(CNC(=O)C=C3CC3)C(C)C2)=O)c1 45875,C1(NC(CCSCC)=O)CCC2(CC1)CC(NC(=O)C(c1ccccc1F)O)C2 45876,c1(C(N(CCNC(c2c(CC)n(CC)nc2)=O)C(C)C)=O)cccc(C)c1F 45877,C(=O)(C(F)CC(C)(C)NC(C1(CO)CCCC1)=O)NC1CC(CCN(C)C)C1 45878,CC(CC(F)(F)F)C(=O)N1CCC(CF)(NC(=O)C(F)C(C)(F)F)C1 45879,CC1CC(CNC(=O)CC2(C)CC2(Cl)Cl)CN1C(c1n[nH]c(=N)s1)=O 45880,c1(NC(C(=O)NCCNC(CC)(C)COC)=O)cnc(C)n1-c1ccccc1 45881,N1(C(C2(CCC)CCC2)=O)CC2CCCC2(NC(=O)C=C(Cl)Cl)C1 45882,N1(C(N2CCCC(CC(=O)OCC)C2)=O)CCCNC(=O)C1CC 45883,C1(NC(CC(=O)NCC)=O)CCN(C(C2(C)CCCC(F)(F)C2)=O)CC(O)C1 45884,c1(COC)ccc(C(=O)NCC(C2CCC2)NC(c2oncc2C)=O)cc1 45885,C1(NC(c2n(CC)ccc2)=O)CC2(C1)CC(NC(=O)CC(O)c1ccccc1)C2 45886,Nc1ccc(C(N2C(CNC(=O)CCc3ccc(O)nn3)CC3CC23)=O)cc1Cl 45887,C=CC1(C(N2CCC(O)(C(C)NC(c3scc(C)c3C)=O)C2)=O)CCCC1 45888,c1(C(N(C(c2n(CC)ccn2)C(=O)O)C)=O)cc(C)cc(O)c1 45889,N1(C(C(C)NC(CC)=O)=O)CCOC(CN(C(=O)CC2CN(C)C2)C)C1 45890,Cc1oc(C2CC2)nc1NS(=O)(=O)CC1CC1F 45891,C(CC1CC1)(C(=O)NCC1CCCOC1)NC(=O)Cc1ccsc1 45892,c1(C(N2CCC(CNC(C3CC4(CC4)C3)=O)C23CC3)=O)cc2c([nH]1)CCCC2=O 45893,C#Cc1ccc(CNc2cccnc2C(=O)NC2(c3ccccc3F)CCC2)s1 45894,N1(C(c2cc(C)cc(O)c2)=O)CCC(C2(NC(c3cnns3)=O)CC2)CC1 45895,Cc1cncc(C(N2CCC(O)(C(C)NC(=O)Cn3cncn3)C2)=O)c1 45896,C1(N(C(CCN(CCCCC)C)=O)C)CCC(NC(=O)C(O)CC)CC1 45897,c1(CNC(C(N(C(CN(CCC)C)=O)C)C2CC2)=O)cnc(C)cn1 45898,N1(C(=O)CO)CC2CCN(C(c3nn[nH]c3Cl)=O)CCC2C1 45899,c1(C(N2CC3C(NC(=O)Cc4ccnc(F)c4)(C3)C2)=O)cc2c(nn1)CCCC2 45900,c1(C(N2C(CNC(CC3C(C)=NNC3=O)=O)C=CC2)=O)cc(C)ccc1F 45901,c1(NC(=O)C(F)CC2CNC2)cnccc1C(F)F 45902,C1(CNC(C(C)OCC#C)=O)CCCN1C(c1c[nH]nc1-c1cccnc1)=O 45903,N1(Cc2ncc(C(=O)NC(c3nc(C)oc3)C)cn2)CCC(CN(C)C)CC1 45904,c1(NCC2OCCN(C(=O)C=Cc3ccccn3)C2)ncnc2c(Cl)cc(Cl)cc12 45905,N(C(=NCc1ccnn1C)N1CCC(CC2CC2)C1)Cc1[nH]nc(C(C)C)n1 45906,CC#CCCCCN=c1ccc2cc(S(=O)(=O)NC3CCOC(C)C3)ccc2[nH]1 45907,c1(C(N(C2CCCN(C(C3(Cl)CCCCC3)=O)CC2)CC)=O)ccc(C)c(O)n1 45908,C(=O)(C(C(C)(C)C)c1cc[nH]n1)N(CCNC(C(C(C)O)N(C)C)=O)C 45909,N1(C(c2n(C(CC)CC)nc(C)c2)=O)CCCC(NC(c2coc(C)n2)=O)CC1 45910,C1(NC(C2N(C(=O)NC(C)=O)CCCC2)=O)CCN(C)CC1 45911,C#CCC(C)(C(=O)NC1(C)CCSC1)NC(=O)CC(C)(O)COC 45912,C1(NC(c2occ(C)c2)=O)(CO)CCN(C(c2ccc(CC(C)(C)C)cc2)=O)C1 45913,N1(C(C2OCCN(C(C3(CC)CC3)=O)CC2)=O)C2CCC1CN(C)CC2 45914,c1(C(N(CCC)CCC)=O)cn2c(n1)CCN(c1ncnc3c1CCCC3)CC2 45915,C(=O)(C#CC1CCOCC1)N(C1CCN(C(C2CC(=O)N(CC(N)=O)C2)=O)C1)C 45916,c1(C(=O)NCC2C(NC(=O)Cc3cscn3)CC2)cc2ncccc2s1 45917,N1(C(C(C)NC(N)=O)=O)CC2(CC(NC(=O)C(C)(C)NS(C)(=O)=O)C2)C1 45918,CCCCC(CC)CC(=O)NC(C(C)N=c1[nH]ncs1)c1ccccc1 45919,C1(F)(CNC(C(C)=C(C)C)=O)CCCN(C(C2(C)CC(C)C2)=O)C1 45920,c1(C(N2C(CNC(=O)C=CC3CCCCC3)CC3CC32)=O)cc(=O)cc(Cl)[nH]1 45921,c1(CN(c2n(CC)c(CO)nn2)CC2(S(C)=O)CC2)c(O)cccc1Cl 45922,C(c1ccccc1)=CCC(N1CCC(CN(C(C(COCC)C)=O)C)C1)=O 45923,N1(C(c2c(CCC)onc2C(N)=O)=O)Cc2c(ccc(F)c2Br)C(C)(C)C1 45924,C(=O)(CCC(C(C)C)NC(c1c[nH]c(C)c1)=O)N1CCCC(OC)CC1 45925,N1(C(C)C)CC(C(=O)OCc2ccccc2C(F)(F)F)CC1=O.C1(C)C(=O)O1 45926,Cn1ncc(C(c2nnnn2CCNC2CC3CCCC3C2)CCO)c1S(N)(=O)=O 45927,C(CCCCC(=O)NCC1CN(C(=O)CC2(CO)CC2)C1)=CC 45928,c1(Cn2ncc(C(N3CCC(c4ncc(C)cn4)CC3)=O)c2)ccc(Cl)c(F)c1 45929,Cc1ccc(C2(C(=O)NCCCCN(C)C(c3snnc3C)=O)CC2)cc1 45930,CC1(C)CC(NC(=O)CC#N)CN1C(=O)COCc1cccc(Cl)c1 45931,C1(OCCCN(CC(=O)NC)Cc2ccccc2Cl)CCCC(C2CCN2)C1 45932,N1(C(=O)CCOC2CCCC2)CCC(C(F)F)(CNC(C23CC(F)C2C3)=O)C1 45933,CC1CC(CNC(=O)C(O)C2CCCC2)CN1c1nccc(C2CCCC2)n1 45934,N1(C(C(CCCC)C)=O)CCCC2CN(C(C3(CCOC)CCCC3)=O)CCC12 45935,C1(C)(C(N(CCC(C)(C)C)C)=O)CCCN1C(=O)CCc1ncnn1C 45936,C1(CC(=O)NCC2OCC(CNC(CC(=C)C)=O)C2)CCc2sccc2C1=O 45937,c1(CCNC(CCc2cc(C)on2)=O)c(C)n[nH]c1C 45938,N1(C(c2nccc(CC)c2)=O)CCN(C(C2CC(C)=NO2)=O)C(CC(=O)NC)C1 45939,N1(CCCCCNC(COC)=O)CCN(CC(O)COCc2cccs2)CC1 45940,Cc1ccc2nc(C)c(C(=O)N(C3CCN(C(C4CC(Cl)(Cl)C4)=O)C3)C)cc2c1 45941,C1(C(=O)NC2CN(C(c3c(O)ccc(CC)c3)=O)CC2O)CCc2cnnn2C1 45942,c1(N(C)C)ccc(C(=O)Nc2cccc(-c3nn(C)c(=O)n3C)c2)cc1[N+](=O)[O-] 45943,CCCCC(C)CCC(=O)N1CCC=C(C(=O)NCc2cnccc2Cl)C1 45944,C1(CNC(C(C=CC)O)=O)CC(C)CCN1C(=O)CNC(c1ccc(C)s1)=O 45945,c1(C(CC(=O)OC)NC(c2c[nH]cc2C)=O)cccc2ccccc12 45946,C1(NC(c2c(=O)ccn(C)c2)=O)CCC2(CC1)CNC2 45947,N1(C(C2CCCCC2)=O)CC2C(C(=O)NC(c3cccc(O)c3)C(=O)O)C2C1 45948,c1(C(N(C2CCC2N(C(=O)C(O)CN2CCCC2)CCCl)C)=O)ccnc(O)c1 45949,C1(NC(c2c(OC)nsc2)=O)CCC12CN(C(=O)CCc1csc(=N)[nH]1)C2 45950,N1(C(c2cncc(C(C)(F)F)c2)C(=O)NCCOC)CCN(C=O)CC1 45951,c1(CC(=O)NCC=CC(N2CCC(CF)CC2)=O)ccc2c(c1)CC2 45952,N1(C(C2(N(C)C)CCC2)=O)CCN(C(c2ccn3nccc3n2)=O)C2(CCC2)C1 45953,N1(C(C2(CCCC)CCC2)=O)CCC2(CCCN(C(=O)CNC(=O)OC)C2)C1 45954,C(=O)(C(C(C)C)ON(CCNC(=O)OC)CCl)NCCC#C 45955,Cc1cc(C(=O)NCCOc2ccccc2C(C)C)c(F)cc1Cl 45956,C1(CN(C)C(C2(C)CC=CCO2)=O)CCN(C(=O)CSc2n[nH]c(=N)s2)CC1 45957,C1(NC(C(N2CCSCC2)C)=O)(CO)CCCN(C(C2(O)CCSC2)=O)C1 45958,Cc1ccc(F)c(CC(=O)NC2CCC(NC(=O)C(F)C3CCC3)C2)c1 45959,C1(C(=O)NCC(O)CNC(C2CCC(c3ccccc3)C2)=O)(CC)CCCC1 45960,N1(C(C)=O)CCC2(CCOCC2)C(NC(c2coc3c2C(=O)NCCC3)=O)C1 45961,c1(CN(C)C(C2CC(NS(C)(=O)=O)C2)=O)ccccc1CNC(=O)C(C)(C)OC 45962,C1(C(N2CC(CC(C)NC(C3=C(C)OCC3)=O)C2)=O)CCc2nc(O)[nH]c2C1 45963,CCCC(C)CCCC(=O)N1CC2(CNC(=O)C#CC3CC3)CC1CO2 45964,c1(C(=O)NCC(CN(C(c2n[nH]c(C)c2C(F)(F)F)=O)C)O)ccnc(Cl)c1N 45965,CC1CCC(C(=O)N(C2CCCCCC2)CCNC(=O)CCOC2COC2)CC1 45966,C1(NC(CCCSC)=O)COC2(C1)CN(C(c1ncnc(O)c1F)=O)C2 45967,c1(C(N2CCC3CN(C(C4C(C=C)OCC4)=O)CC32)=O)cnc2ccccc2n1 45968,c1(OC)cc([N+](=O)[O-])ccc1CN=C(NCC(C)(C)C)NC1CCCCC1 45969,C(=O)(C1=CCC(NC(=O)CC2CCC2)C1)NCc1nccc(OC)n1 45970,CCC(Cc1ccccc1)C(=O)NC(c1nc(C(C)C)no1)C 45971,N1(C(C2(C)CCC(=O)C2)=O)C(CNC(=O)C=CCF)CC2COCC12 45972,c1(-c2cn(COC)nc2)ccc2ccc(C(=O)NC3CC3)nc2c1 45973,CC(C)CC(C)CC(=O)NCCC(C(C)C)NC(c1cnc(C2CC2)nc1O)=O 45974,CC(CN=c1[nH]c(=NC(C)c2ncc[nH]2)[nH]c2ccc(Cl)cc12)N1CCCC1 45975,N1(C(C(C)N(C)C)=O)CC(CO)C2(C1)CN(C(C1CCn3ncnc3C1)=O)C2 45976,C(=O)(C(C)CC(F)(F)F)NCC1CC(OC)CN1C(c1c[nH]nc1C)=O 45977,C(=O)(CS(=O)(=O)CC(=O)OC)N1C(CNC(C(CC)=CC)=O)C(C2CC2)CC1 45978,c1(C(=O)NC(CCCCNC(C)=O)C)cnc2c(C)cnn2c1 45979,C1(C)COCCC1CNC(=O)NC(C)(C)CC1CCOC1.c1(N)coc(CO)c1 45980,C1(C(=O)N(CC(C)(O)C2CC2)C)(CC)CCN(C(=O)C(C)CC)CC1 45981,c1(C(=O)NCc2ccc(-c3nn[nH]n3)nc2)cccc2[nH]ncc12 45982,c1(-c2cn(CCCCNC(c3c(C)coc3)=O)nn2)cccc(C(F)(F)F)n1 45983,N1(C(C2(F)C(C)C2)=O)CC2(CCCCN2C(=O)CCOCC(F)(F)C(F)F)C1 45984,c1(NCc2c(C)cn(C)n2)[nH]c(=NCC2CCCCN2C)nc2scnc12 45985,C1(NC(c2nccc(C)n2)=O)CCC2CCN(C(=O)C=Cc3ccc(C)o3)C12 45986,c1(NC(=O)CCC2CCC(=O)N2C(=O)O)ccc(S(=O)(=O)c2ccccc2)cc1 45987,N(C(=NCCC(C)(C)S(C)(=O)=O)NCC1CC(C(C)C)C1)CCOCC 45988,N1(C(C=CCOC)=O)CC(CNC(c2cnc(C3CC3)nc2O)=O)OC(C)(C)C1 45989,c1(OCC(=O)NC(C(C)NC(C2CCCCC2)=O)C)cccc(Br)c1 45990,CC1(C)CC(CC(=O)NC(CO)C2CCC2)CN1C(=O)CC1CC(=O)C1 45991,c1(NCCNC(N(CCCC)C2CC2)=O)ccc(Cl)c(Cl)c1OC 45992,c1(CC(C)C(N2CC3CN(C(C4(F)CC4)=O)CCC23)=O)cnc2ccccc2n1 45993,N1(C(CSCC)=O)CCSC(C(=O)NCCc2nc[nH]n2)C1 45994,C1(CC(=O)N(C2CC(CNC(=O)C=Cc3nccs3)C2)C)CCN(C)C1=O 45995,C1(NC(c2ncn(CC)c2)=O)CCN(C(c2ncsc2C(F)(F)F)=O)CC1(C)C 45996,c1(C(N2C(C)CN(C(=O)C(F)(F)CO)CC2)=O)cc2n(n1)CCCC2=O 45997,C1(C(=O)NCC2C(NC(=O)CCc3ccc(Cl)nc3)C2)CCOC(=O)CC1 45998,C1(CC(=O)NCCCNC(c2cncc(CSC)n2)=O)(OC)CCCCC1 45999,Cn1cnc2cc(C(=O)NC3C4CC3N(C(c3ccncc3Cl)=O)C4)ccc12 46000,C1(CNC(C(C)(C)CC(F)F)=O)CN(C(=O)C(O)C2CCC2)C2(CCOCC2)C1 46001,c1(OC)ccc2c(c1)C(NC1=NCCCN(C)C1)CCO2 46002,CN1CC(O)CCC1C(N1CC2(C1)CN(C(C1CN(C(N)=O)C1)=O)C2)=O 46003,C1(C(=O)OCC(N2CCOCC2)C)CNC2(CCOCC2)C1 46004,N1(C(c2ccc(OC)c(C)c2)=O)CC2CCN(S(=O)(=O)C3CC3)C2C1 46005,C1(CNC(c2ccc(O)nc2)=O)CC2(CCN(C(C3(CF)CC3)=O)CC2)CO1 46006,Cn1cnc2sc(C(=O)NCC3(O)CN(C(C4(O)CCCCC4)=O)C3)cc12 46007,c1(C(N2CCC(NC(C(C)(C)F)=O)C2)=O)cc2ccc(Cl)cc2c(=O)o1 46008,N1(C(C(=O)NC2COC2)c2nccs2)CCOCC1c1cccc(F)c1 46009,C1(C2CN(C(c3cc(F)cs3)=O)C2)(NC(C(C)CCc2cccc(F)c2)=O)CC1 46010,C1(CC=C)(NC(c2ncoc2C2CC2)=O)CN(C(c2cc(Br)c[nH]2)=O)C1 46011,C(=O)(C1CCCc2n[nH]cc21)NCC(C)NC(C1CC(C)(c2ccccc2)C1)=O 46012,CC1CCN(C(c2ccc[n+]([O-])c2)=O)CC1CNC(=O)CC1CCCCC1 46013,N1(C(c2c(C)csc2)=O)CC2CC(NC(=O)Cc3cc4ccccc4o3)C(C2)C1 46014,Cc1ccccc1N1CC(C(=O)N(CCCNC(=O)CC(C)F)CCO)CC1=O 46015,C=CCC(C(=O)NCCC(C)NC(c1cnn(C)c1CC(=O)OC)=O)C(C)(C)C 46016,CC1(C)CCN(C(c2ccc3sncc3c2)=O)CC1NC(=O)CCc1cncs1 46017,c1(C(C(=O)NCCNC(C(COC)COC)=O)C)ccc(S(C)(=O)=O)cc1 46018,CCC(=O)CCC(=O)N1CC(C)(CCC(N2CCC(N(C)C)(CC)C2)=O)C1 46019,CC(C)CC(O)CC(=O)Nc1sccc1C(=O)CN(C1(O)CC2CCC1CC2)C 46020,O=C1CCN(C(c2cccc(C3CC3)c2)C(=O)NCC2CCCO2)CCN1 46021,C(=O)(CCC(=O)NCC1CC(O)CN1C(c1cc(Cl)cn1CC)=O)NCC 46022,c1(C(=O)NCC2(NC(C3CC3F)=O)CCOC2)cc(Cl)cc(C(F)(F)F)n1 46023,c1(C(=O)NC(CC)(C)CNC(C2CS(=O)(=O)C2)=O)cc(F)c(F)cc1Br 46024,CC1(c2ccc(NC(C3CN(c4ncncc4I)C3)=O)cc2)NC(=O)NC1=O 46025,c1(C(N2CC(F)(CNC(C3CC34CC4)=O)C2)=O)ccccc1Cn1cncn1 46026,c1(C(=O)NC2CC(CCNC(C(C)n3cnnn3)=O)C2)cc(C#N)ccc1F 46027,C(CC(C(C)(C)C)NC(=O)C(F)F)N(C(=O)CC1(C)CCCCC1)C 46028,C(CCC(C)(C)C(=O)NCC(C)CCCO)NC(c1c(C)ncnc1)=O 46029,CCCS(=O)(=O)C(C)C(=O)NC1CN(C(=O)CCCCCN(C)C)C2(CCC2)C1 46030,C1(NC(c2oc(C)c(Br)c2)=O)CN(C(=O)CCCCCNC(N)=O)C2(CCC2)C1 46031,N1(C(C2(C(=O)NC)CC2)=O)CCC2(CCCN(C(c3ccn(C)n3)=O)C2)C1 46032,c1(C(N2C(CO)CC(NC(C3(C(N(C)C)=O)CC3)=O)C2)=O)ccc2nn[nH]c2c1 46033,c1(C(=O)NCC2(O)CN(C(c3ccc(CC4CC4)s3)=O)C2)ccnc(Cl)c1Cl 46034,C1(C(N(C2CCN(C(=O)Cc3cncc(C)c3)C2)SCC)=O)CCCC2(CC2)C1 46035,N1(C(C(C(C)C)NC(C)=O)=O)CCC12CN(C(=O)C(C)NC(=O)C1CC1)C2 46036,C1(NC(CCN(C(CC)CC)C)=O)CC2CC1N(C(=O)C(n1nccc1C)C)C2 46037,C12(C(N(CC(CC)O)CC)=O)CC(C)(CN1C(=O)Cc1cc(CC)no1)C2 46038,C(=O)(C1CCc2cc(Cl)ccc21)N(CCNC(c1c(CCC)n[nH]c1)=O)CCC 46039,C#Cc1ccc(C(=O)NC2CN(C(C3(C(=O)NC(N)=O)CC3)=O)C2)cc1F 46040,C1(C(=O)NC2(c3ccn(C)n3)CC2)(NC(CC=CCC)=O)CCN(C)C1 46041,c1(OC)ccc(CN(C(C2C3CCOCC23)C(=O)NC)C)c(OC)c1 46042,N1(C(C(C)NC(C2CCCC2)=O)=O)CC2(CCN(C(=O)CCCN(C)C)CC2)C1 46043,CC(C(=O)NO)NC(C1CC(C)N1C(=O)CCC1CCCCC1)=O 46044,N1(C(c2cc(C(N)=O)[nH]n2)=O)C2CCC1CN(C(C1CCC3(CCC3)C1)=O)C2 46045,C1(CNC(CCCCSC)=O)CCC2(CN(C(c3cccc(C)c3C#N)=O)C2)O1 46046,C1(C(=O)NCCCCCOC)C=CCCN1C(=O)C(C)C(=O)OC 46047,C1(C(=O)NCC(C)(CO)NC(c2ccc(C)cc2)=O)CCCC2(CCC2)O1 46048,N1(C(=O)C=Cc2ccc(C3CC3)cc2)CCOC2(C1)CN(C(c1cc[nH]n1)=O)C2 46049,CC(=O)CCCC(C)C(=O)NC1(C(N2CCC(C(=O)OC)C2)=O)CC(CO)C1 46050,c1(CNC(CCC2N(C(COCCSC)=O)CCC2)=O)cccc(O)n1 46051,C1(C(=O)NC(C(=O)NCCN(CCOC)C)CO)CC2(C1)CC2(F)F 46052,c1(OC)cccc2sc(NC(C3CC4CCCC4N3C(N)=O)=O)nc12 46053,C(CCCCC(=O)NC(C1(O)CCN(C(c2cc(CO)n(C)n2)=O)C1)C)OCC 46054,c1(C(=O)CCC(=O)NC2(CNC(=O)Cc3cnns3)CCC2)ccc(F)cc1F 46055,C1(NC(C2C(C)CC2)=O)CCC2(CCN(C(c3ccc4cc[nH]c4n3)=O)C2)C1 46056,C1(C(N2CCN(C(CC(=O)NCC)=O)C(C(C)C)C2)=O)CC2OC(C)(C)OC2C1 46057,O=C1CC(C(=O)NC2CC3(C2)CC3C(N2CCn3nccc32)=O)=NN1 46058,C1(NC(CC(C)c2cnn(C)c2)=O)CCCN(Cc2cccc(Br)c2)C1 46059,Cc1cc(CNCC2CCCCN2C(C2(O)CCSC2)=O)n(C)n1 46060,N1(C(C2(C)C(C)C2)=O)CCC(C2CC2)(CNC(c2ccc3[nH]ccc3n2)=O)C1 46061,C(=O)(C(F)CC(CC)CC)N1CCC(C(CC)NC(C23CCN(CC2)CC3)=O)CC1 46062,N1(C(c2c(CC)[nH]cc2)=O)CCC2CC2(C(=O)NCc2n[nH]c3c2CCC3)CC1 46063,c1(OC)cc(Br)ccc1C(CO)NC(=O)NCc1oc(C)cc1C 46064,NC(=O)CC(C(=O)NC1CCN1C(C)(C)C)NC(C1CCCCC12CC2)=O 46065,c1(C(N2CC(CNC(C3C(OCC)C3)=O)(OC)C2)=O)c(O)nnc2c1COCC2 46066,c1(C2(CNC(c3ccsc3)CO)CCC2)ccccc1Cl 46067,C1(NC(C2CCC(=C)CC2)=O)C(C)CCN(C(c2ccc(Cl)c(F)c2)=O)C1C 46068,C(=O)(C1=CCC(C)(C)CC1)NC(C(C)(C)NC(Cc1c(O)ccc(C)c1)=O)C 46069,c1(C(=O)NCC2C(C(=O)Nc3cnc(OC)nc3)C2)coc2c1COC2 46070,N1(C(C(C)OCCCC)=O)CC(F)(F)CC1c1cn(C)nn1.C1CO1.OC 46071,c1(OC(C)C)ccc(CC(=O)N(C2CCC(CNC(=O)CC(C)C)CC2)C)cc1 46072,c1(C(C(=O)NCCCSC)N(C2CCCO2)CC2CC2)ccc(-c2ccco2)cc1 46073,c1(CCOC)nc(=NC2CCCC(NC(C3(O)CCSCC3)=O)C2)s[nH]1 46074,Cc1cc([N+](=O)[O-])c(C)cc1C(N1CC2CN(C(c3c[nH]c(=N)s3)=O)C2C1)=O 46075,C(C(CNC(=O)C(C)Cn1ccnc1)S(C)(=O)=O)NC(C(COC)C)=O 46076,N1(C(c2c(C)[nH]cc2)=O)C(C(=O)N(C(C)C)Cc2ccco2)CCC1C 46077,O=C(C1CCCn2cnnc21)NCC1CC(O)CN1C(=O)CCc1ccncc1 46078,c1(N2CC(CC)OCC2)nc(N(C)CC2(CC)CC2)nc2cc(OC)ccc12 46079,C1(NC(c2cc(COC)no2)=O)CN(C(C2CCNC2=O)=O)C2(CCCCC2)C1 46080,c1(C(=O)NCC(C)CNC(c2ccc(C(F)F)o2)=O)c(F)cc(Cl)cc1F 46081,Cc1ncc(C(=O)N(CC(C)N(C(=O)CN2CC3CCC2C3)C)C)cc1N 46082,Cc1c(NC2CCN(CC(C)C)C2)ncnc1N(C)CCOC1CC1 46083,c1(N2CCC(N(C)C(c3ccc(O)nn3)=O)C2)nnccc1C#N 46084,C1(CC(=O)NCc2ccc(CNC(C3C=C(C)CS3)=O)cc2)CCCC(C)(C)O1 46085,c1(OC)ccc(CN2CCCC2CCCNC(C2CCCOC2)=O)cc1Cl 46086,C(=O)(CC(C)(O)C(F)(F)F)N1C(C(C)NC(c2ccc(CC)cc2C)=O)CCC1 46087,c1(-n2c(-c3cnc(F)c(C)c3)nc(C(C)OCC)n2)c(C)cc(C)cc1C 46088,c1(C(=O)NC(c2c(NCc3nccc(C)c3)cccn2)=O)ccc2nc[nH]c2c1 46089,c1(C(=O)NCC2CC(O)(CNC(C(OC)OC)=O)C2)nc(C)ccc1F 46090,C(=O)(C1CCCn2nccc21)N(CC(C)(C)CNC(=O)COC1CCOC1)C 46091,c1(NC(=O)NCc2ccc(CC)s2)cnccc1C(F)(F)F 46092,c1(C(=O)NC2CCC(CNC(C(N3CCNC3=O)C)=O)C2)ccc(F)cc1N 46093,n1(CC(=O)N(C(CNC(Cn2cc(C(C)=O)nn2)=O)C)C)ncccc1=O 46094,C#Cc1cnn(C)c1C(N1CCC(F)(CNC(c2cncn2C2CC2)=O)C1)=O 46095,CC1CC(NC(C2CC(O)C2)=O)CCN1C(=O)CC1CC1 46096,c1(C(=O)NCC(CC)(CC)Nc2cncc(C#N)n2)ccc2nc[nH]c2c1F 46097,c1(CC(C)C(=O)N2CCCC2CN(C)C(c2cc(F)c[nH]2)=O)ccc(F)cc1F 46098,C(=O)(CCC(C)SC)NC(CN(C(=O)CN1CCCC(C)C1)CC)C(=O)NC 46099,C1(NC(CCC(=O)NCCC)=O)CCCN(C(c2ccccc2SC)=O)CC1F 46100,c1(C(CC)C(=O)N(C(C)CN(C(=O)COCC(=O)NC)C)C)c(C)noc1C 46101,C123CC4CC(CC(C4)(C1)COC2=O)C3.CC1CC(C)OC1C(=O)OC(C)(C)C 46102,C1(NC(c2c(CC)noc2)=O)C=CCN(C(c2ccccc2OCC(N)=O)=O)C1 46103,c1(C2C3(CC3)NC(=O)N2)ccc2c(c1)CCCC2.CN1C(=O)CSC1=CC=O 46104,C1(CN(C(CC(C)O)=O)C)CCCCN(C(c2cccnn2)=O)C1 46105,N1(C(c2ccc(C)s2)=O)CCC(NC(=O)C(C)Cc2ccnn2C)C1C(C)(C)C 46106,c1(C(=O)NC(C(=O)OC)C2CC(C(=O)O)C2)ccc2[nH]cc(C=O)c2c1 46107,c1(C(=O)NC2CN(C(C=C(CCC)C)=O)C(C)C2)cc2c(OC)cccc2[nH]1 46108,O=C1COc2ccc(NC(=O)NC(COC(F)(F)F)Cc3ccccc3)cc2N1 46109,C1(CNC(C=C(C)Cl)=O)(CNC(=O)CC2CCC(=O)N2)CC12CCC2 46110,CCCC(C(=O)N1CCN(C(C23CCCN(CC2)C3)=O)CC1CO)C(C)C 46111,N1(C(c2cc(CSCC)on2)=O)CC(C)CCC1CC(=O)C(CC)(CC)OC 46112,c1(C(=O)NC(c2cnn(C)c2)C(=O)OC)ccc(-c2ccc(F)cc2F)cc1C 46113,CC1(C)CN(C(=O)CC2CC2(C)C)C1C1CCN(C(=O)COCCCF)CC1 46114,C(=O)(CS(=O)(=O)CC1CCCO1)NCC(CNC(CCC(C)C)=O)CO 46115,N1(C(c2c(CC)nccc2)=O)CC2(C1)OC1(COC)CC2(NC(=O)CCCF)C1 46116,CC(CCCNC(c1csc(F)c1)=O)NC(=O)C(c1ccccc1)F 46117,NC(CN1CCCC1)C(=O)N(c1nn[nH]n1)C1(c2ccccn2)CC1 46118,C1(CC)CCCN(C(C2CCCS2)=O)C1C(=O)N(C)CC1CCCS1 46119,C1(C(N)=O)CCCCN(C(C2CCN(C(=O)c3cc([N+](=O)[O-])n[nH]3)O2)=O)C1 46120,Cc1cccc(C(=O)N(C)Cc2cc[nH]c2)c1C 46121,C=CCCC(C(=O)NCC1CCC(=O)O1)NC(=O)CC(C)OC 46122,c1(C(N2CCCC(O)(CNC(c3c[nH]c(=N)o3)=O)C2)=O)cc(=O)n2nccc2[nH]1 46123,C1(CCNCC(C2CN(C(=O)OC(C)(C)C)C2)C)CCCCC1C#N 46124,C1(C(NOCCCOCC)=O)CCN(C(=O)Cc2c[nH]nc2C)C(C)C1 46125,N1(C(c2nc(C)oc2)=O)CCC(C)C(CC(N2CCCC(C)(C)C2)=O)C1 46126,CC1CCC(CC(=O)NCc2cnn(CC(N3CCC3(CO)CO)=O)c2)CC1 46127,C(CC(C(=O)NC1CCCN(C(c2csc(C(F)F)n2)=O)C1)OC)OC 46128,CC1(C)OC(=O)NC1C(=O)NCc1cccc(NC(=O)CCC(N)=O)c1 46129,c12c(cnn1C)CNC2=O.C1(C(C)C)CN(C(=O)CCc2nncs2)C1C(C)C 46130,C=C(C)CC(C(=O)NCC12CCCC1OCC2)NC(=O)C(CC)OCC 46131,N1(C(CCC2CCC(=O)C2)=O)CCC2(CC2NC(=O)C2=C(Cl)CCC2)C1 46132,N1(CCC(=O)N(C(C)CNC(C2(N(C)C)CCCCC2)=O)C)CCSC(C)(C)C1 46133,C1(C(=O)NCC(C)(C)Nc2nc(C3CCCC3)ns2)CCc2c[nH]nc2C1 46134,C(=O)(C(CCC1CC1)NC(c1nc(C)sc1C)=O)NCC(=O)N(C)CC 46135,C1(C)(C(=O)NCC2(C#C)CCC2)CCCN1C(=O)CCC1CCCCO1 46136,C=C(Cl)CC(C(=O)NC)NC(=O)CN(C(=O)C(C)CC)C1CC(C#N)C1 46137,C1(CN(C(c2cnn(-c3ccccc3)c2)(C)C)C(C)=O)CCCC(C2CC2)O1 46138,C1(C(=O)NCC(CC=C)NC(=O)C(c2ccc(F)cc2)CO)CCS(=O)(=O)CC1 46139,C1(CC(=O)N(CC=CC(=O)NCCCCC=C)CC)CCC(=O)C1 46140,C1(C(=O)NC2CCC(NC(c3cn(C)nc3Cl)=O)CC2)COC2(CCC2)CO1 46141,c1(CC)ccc2c(Cl)c(C(=O)NC(CNC(C3(C#N)CC(C)C3)=O)CO)sc2c1 46142,CN1CCCC(CC(N2CCC(CO)(NC(=O)COCc3ccccc3)C2)=O)C1 46143,c12cc(F)c(F)cc1NC2=O.C(=O)(C(C)(C)C)NCCNC(C=C(C)C(F)F)=O 46144,c1(C2(C(=O)NCCNC(C3C=CCN3)=O)CC2)cccnc1 46145,N1(C(C(CC#C)O)=O)CCC2CCC(C1)N2C(c1ccc(Cl)cc1Cl)=O 46146,C1(CCC)CN(C(C2(C)CCNC2=O)=O)CCN1C(c1nnn(C(C)C)c1N)=O 46147,C(=O)(C(CC(C)C)N(C1CC2CC2C1)C)N(CC=CC(=O)OC)C 46148,c1(C(C(C)C)O)cc(O)nc(NC(CCCC(=O)Nc2ccc(OC)cc2)=O)n1 46149,C1(NC(c2cc(Br)no2)=O)(CO)CN(C(c2ccnn2C2CC2(F)F)=O)C1 46150,N1(C(c2cccc(CC)c2)=O)CC(C)CN(C(c2cc(=O)cc(Cl)[nH]2)=O)CC1C 46151,CCCCCCCCC(C)CC(=O)N1CC(CO)(NC(=O)C=CCO)C1 46152,C1(CNC(c2cccc(COC)c2)=O)CC2CCC1N2C(=O)COCC(F)(F)F 46153,N1(C(C2C(=C)C2)=O)CC(NC(=O)CCc2cnccn2)C2(CCS(=O)(=O)CC2)C1 46154,N1(C(C2(COC)CC=CC2)=O)CC(CCNC(c2nn[nH]c2Cl)=O)OC(C)C1 46155,Cc1c(C(=O)N(C)CCNC(c2cn(CC3CCCO3)nn2)=O)cccc1Br 46156,C=CCC(C)(CC)C(=O)N1C2CCC(C2)C1CC(=O)NCCn1cnccc1=O 46157,C1(OC)(CNC(C2(CCl)CN(C(=O)CC(C)O)C2)=O)CCOC1 46158,C1(CC(=O)N(CC(N2CC(O)(CC=C)C2)=O)CC2CC2)CCC(=O)NC1 46159,c1(CN(C2(c3nnnn3C)C(C)COCC2)CC(F)(F)F)ccc(F)c(F)c1Br 46160,C1(NC(c2c(CC)nn(C)c2)=O)CCN(C(=O)CCC2CCCCO2)CC1CC 46161,C1(NC(c2ccc(SC)o2)=O)CCCCC1CNC(c1cc[nH]c(=N)c1)=O 46162,C1(CSC)CCCCN1C(C=Cc1ccccc1)C(=O)NCCC1CC1 46163,c1(CC(=O)NC2CC(NC(C3CC3C3CC3)=O)C2)c(F)cc([N+](=O)[O-])cc1F 46164,N1(C(=O)CCCn2cccc2)CCN(C(=O)Cc2cc(F)cc(Cl)c2)CC(O)C1 46165,C12(CNC(C(CC)=CCCC)=O)CC(NC(=O)C(C)=CCC)(C1)C(C)O2 46166,c1(NS(CC)(=O)=O)nc(N2C3CN(c4nccc(OC)n4)CC23)ncc1OC 46167,N1(C(CCC2CCC(C)O2)=O)CCC2CC(CNC(c3cnoc3)=O)CCC2C1 46168,c1(C(=O)NCC(CC)NC(=O)C(c2cccc(C)c2)C)c2c(nn1C)CCSC2 46169,C1(C(N2CCC(C(C)C)(C(=O)NC(C)CC(C)(C)O)C2)=O)CCC2(CC1)CC2 46170,CCCCC(C)(F)C(=O)NC1CC1CNC(=O)C=Cc1ccc(Br)s1 46171,Cc1ccc(OC(C)C(N2CC(CNC(C3(C#N)CCCC3)=O)C(C)C2)=O)cc1 46172,c1(NC(CNC(C(c2cc(C)sc2)(F)F)=O)C2CCC2)ncnc2cnn(C)c12 46173,CC(C)CC(C)CC(=O)NCc1cc(C(=O)Nc2cncc(C(C)C)c2)ccn1 46174,c1(OC)ccccc1S(=O)(=O)NC1CCCCC1C(=O)Nc1cc(C)cnc1C 46175,N1(Cc2n[nH]c(=N)s2)CCc2c(NC(=O)NCCCO)cccc2C1 46176,C1(C)(CNC(C(C=C=C)C)=O)CN(C(c2nc(O)nc(O)c2OC)=O)C(C)(C)C1 46177,CC(C)(C(=O)NCC1CC2CC2N1C(=O)CCP(C)(C)=O)S(C)(=O)=O 46178,CCCCCC(F)C(=O)NCC(CC1CCCC1)C(=O)NC1CC(C)(C)OC1=O 46179,c1(N(C)Cc2c(OC)cccc2)cc[nH]c(=NCCCc2cccs2)n1 46180,Cc1ccc(NC(=O)CC(=O)CN2CC(F)(c3nn[nH]n3)C2)cc1 46181,N1(C(CCOC)=O)CCC(O)(CNC(c2cnc(-c3ccccc3)s2)=O)CC1 46182,C(=O)(CS(=O)C(F)(F)F)N1C(CN(C)C(C23CCC(F)(CC2)CC3)=O)CCC1 46183,c1(CNC(c2nc(C)oc2)=O)nc(CNC(=O)CC(C)CF)cc(O)n1 46184,CCCC(C)C(=O)N1CC(Cc2conc2C(=O)O)(CNC(C2CCCC2)=O)C1 46185,N(C1COCc2ccccc21)C(C1CCCCN1C(c1ccc(Cl)c(Cl)c1)=O)=O 46186,C1(CC(=O)NCCC(C)(C)NC(C2C(C(=O)OC)CCO2)=O)CCCCC1(F)F 46187,c1(OC)cc(C(=O)NCC2CCC2NC(c2cscn2)=O)cc2c1OCC2 46188,N1(CCC(=O)NC(C)(CNC(=O)C=C(Cl)Cl)Cn2cccn2)CCC(O)CC1 46189,N1(C(CCCN(C(=O)OC)C)=O)CCC(NC(C2CCCC2C)=O)C2(CCC2)C1 46190,c1(NCCOC)cc(=NCC2CC(OCc3ccccc3)C2)[nH]c(C2CC2)n1 46191,CC1CC(C2CN(C(=O)C(CC(F)F)NC(c3c[nH]c(=S)cn3)=O)C2)=NO1 46192,N(C(=NCCSCc1ccsc1)N1CC(C)S(=O)(=O)C(C)C1)Cc1cc(C)on1 46193,CC1(C)C(CNC(=O)Cc2ccnc(F)c2F)CCN1C(C1CSC1)=O 46194,Cc1cc(=NC(=O)C(=O)NCC2(CNC(C3CC34CCCC4)=O)CCC2)[nH]o1 46195,c1(OC)cc(N)c(F)cc1C(N1C(CNC(=O)C=CC(C)(C)C)CC2CC12)=O 46196,c1(C(=O)NC(CNC(=O)CC2CCCC2)CO)csc2c(Cl)cccc12 46197,N1(C(C(C)(C)c2ccsc2)=O)CCN(C(=O)CSC2CCCCO2)CC(O)C1 46198,c1(-n2cc(CCNC(c3c(OC)nc(C)cc3)=O)nn2)ccc2c[nH]nc2c1 46199,C1(C(N2CC(C)(C#N)C2)=O)CN(C(C2CC3COCC3C2)=O)CC12CC2 46200,N1(C(C(CC=C)C)=O)CC2(C(=O)NC3CN(C)CC3C)CCC1CC2 46201,C(CCC1CCC1)(C(=O)NCc1ccco1)NC(C(C)n1ccnc1)=O 46202,Cc1cc(C(=O)NCC(C2CCCN2C(C2CC3C=CC2C3)=O)(C)C)c(C)o1 46203,Cc1nc(=N)[nH]c(=NCC2(NC(C3CCCC3(C)C)=O)CCOCC2)[nH]1 46204,Cn1cc(C(C)(C)C(=O)NC2CCC2NC(=O)CC2(c3ccon3)CC2)cn1 46205,c1(C(N2C(C3(O)CN(C(CC=CC=C)=O)C3)CCC2)=O)cnc(C)c(C)c1 46206,C(=O)(N=c1[nH]nc(S(=O)(=O)N2CCN(C(C)=O)C(C)(C)C2)s1)OC(C)(C)C 46207,N1(C(C2C(C)C2)=O)CC23CCCC2(C1)CN(C(=O)CC1(C#N)CCOCC1)C3 46208,C1(C(N2CC(NC(C3C4CS(=O)(=O)CC34)=O)C2)=O)CC2COCC(C1)C2 46209,c1(C(=O)NC2CCN(S(CCCC)(=O)=O)C2)cc(Br)c(O)c(Br)c1 46210,c1(C(N2C(C)CC(NC(c3c(CC)nccc3)=O)C2)=O)cccc2cccc(C)c12 46211,N1(C(CC(C)(C)C)=O)CCCOC(CNC(C2CC2c2c(F)cccc2F)=O)C1 46212,N1(C(C2N(CC)CC2)=O)CC=CC1(C)C(=O)NOCC1CC1 46213,C(CCN=C(NCc1ccc2c[nH]nc2c1)NCC1CCCC(C(F)F)C1)SC 46214,c1(CC(=O)NC2(CC)CCN(C(c3cnsc3C)=O)CC2)cnn2ccccc12 46215,C(=O)(C(C)(C)CS(C)(=O)=O)NC1C(C)CCN(C(c2ncnc3ccsc23)=O)C1 46216,c1(C(=O)NCC2N(C(C3(C(=O)OCC)CCO3)=O)CC2)c(C)cccc1Cl 46217,N1(C(c2ccc(C(=O)OCC)o2)C(=O)NCC2CC2)CC2C(C1)C2(C)C 46218,C1(N(C(CC2CCN(C)CC2)=O)C)CN(C(c2c(F)cncc2Cl)=O)CC1(C)C 46219,n1(CC)nnc(C)c1-n1c(S)nnn1.C1(C2(NCc3ccccc3)CC2)CCN(C)CC1 46220,Cc1ccc(C(=O)NC23CC2CN(C(C2(C)CC=CC2)=O)C3)c(Cl)c1 46221,c1(NC(C)C(N2CCN(CC=C(I)c3ccccc3)CC2)=O)ccc(C#N)cc1 46222,C1(NC(C(C)(Cl)Cl)=O)COC2(CCN(C(=O)COc3ccc(C#N)cc3)C2)C1 46223,c1(C(N2C(C)CCN(C(CC(C=C)(C)O)=O)CC2)=O)ccnc2ccc(Cl)cc12 46224,c1(C(=O)NCC2N(C(CNC(=O)OC)=O)CC(O)C2)cc(N)ccc1F 46225,C1(C(N2CCC(CN(C)C(c3cnc(N(C)C)s3)=O)C2)=O)CC12CCCCC2 46226,c1(C(=O)NCC(C)NC(c2cc(SCC)on2)=O)c(C)nn(C2CC2)c1Cl 46227,c1(C(=O)NC2CCN(C(C3(CCC)CC3)=O)CC2CO)n[nH]c2c1CCSC2 46228,C(=O)(CS(=O)C(F)(F)F)NCC(CCNC(C(CC)SC)=O)(C)C 46229,c1(CC)ccc(C(=O)NC2CCC(CNC(c3ccc([N+](=O)[O-])[nH]3)=O)C2)c(C)c1 46230,C1(NC(C(C)N(CCC)C(c2cc(CC)[nH]n2)=O)=O)CC2(CCOC2)C1 46231,Cc1noc2ncc(C(=O)NCC3CC3C(C)O)cc12 46232,Cn1cc(CC(O)C(=O)NC2(CNC(=O)CCC3(C#N)CCC3)CCC2)cn1 46233,N1(C(C(C)C2CCCC2)=O)CC(O)(CN(C(=O)CCCN(C)C)C)C1 46234,N1(C(CCSCC)=O)CC2CCN(C(c3ccc(OC)c(N)c3)=O)CC2C1 46235,N1(C(C(=O)NCCC)CC(C)CCC=C(C)C)CCC=C(c2ccco2)C1 46236,c1(C(=O)NCC2CC2CNC(C2CC3(CSC3)C2)=O)cc([N+](=O)[O-])c(Cl)cc1Cl 46237,CC1CCCN(C(C2CC23CCCC3)=O)C1CNC(c1cc(N)ccc1O)=O 46238,c1(OCC)ccc2[nH]cc(CN3C(=O)CCN(CCCCF)C3=O)c2c1 46239,c1(C(N2CC(NC(C(C)CC(C)(C)C)=O)C2)=O)cccc2c1C(=O)NC2 46240,C(=O)(CCCC(C)C)NCC(CCCC)NC(=O)CCc1cncnc1O 46241,c1(C(=O)NCC2C(NC(CCC(C)(C)OC)=O)CCCC2)cccc2ccnn12 46242,C1(NC(=O)CCSc2ccccc2)CC2CN(C(c3coc(C4CC4)n3)=O)CC12 46243,CC1=C(C)CC(C)(C(=O)NCC2(CNC(C3CC(=O)N(C)C3)=O)CC2)CC1 46244,CC1CCc2cc(C(=O)NCCN(C(=O)CC3(O)CCCCCC3)C)ccc2N1 46245,O=C(C1=CCN(C(C2CC2C2CCCC2)=O)C1)NCCN1CC2CC2C1 46246,c1(OCCOC)cc(OC)ccc1C(=O)NCC(C)(C)c1ccsc1 46247,N1(C(c2ccc(COC)o2)=O)CCN(C(C2CC(S(C)(=O)=O)C2)=O)CC1CO 46248,c1(NC(C)C)cnc(NC(=O)NOCCOCCO)cn1 46249,c1(CC)nc(C#N)cc(=NC(CC)CCN2CCCCC2)[nH]1 46250,c1(CCC#C)ccc(C(C)C(N2CCC(CN(C(=O)COC(F)F)C)C2)=O)cc1 46251,c1(C(=O)NCC2CCC(NC(C3(OCC)CCC3)=O)C2)cnc2c(C)cccn12 46252,CC1(C)CCC(F)(F)CC1C(=O)NC1CN(C(c2cc[nH]c2)=O)CCC1CO 46253,C1(CNC(C(=O)NCC)=O)C2CC1N(C(c1csc(-c3ccc(C)o3)n1)=O)C2 46254,C(C(C)(O)CC(=O)N1CCC(NC(=O)C(C(C)C)SC(C)C)C(C(N)=O)C1)OC 46255,N1(C(c2cc(SC)oc2C)=O)CCCC2(NC(c3cn[nH]c3)=O)CCCC12 46256,Cn1cc(CCNC(=O)NCCc2ccc(C(F)(F)F)nc2)c2ccccc12 46257,C(=O)(C(CC(C)(C)C)NC(=O)C=C(C)C(F)F)N1CCC(C)(NC(=O)NC)C1 46258,c1(C(=O)NC(CCCNC(c2c(OC)csc2)=O)C)cccc(OC)c1OC 46259,C1(NC(c2[nH]cc(COC)c2)=O)CCN(C(c2nc(C)c(C)s2)=O)CC1C(N)=O 46260,Cc1cc(C(N2CCC(OCCNC(=O)Cn3cccc3)C2)=O)nn1C(C)C 46261,c1(C(N(C2C(C)CCN(C(CSC)=O)C2)C)=O)cc2cccc(Cl)c2nc1C 46262,C1(C(=O)NC(CCCNC(C2(CC#C)CC2)=O)(C)C)Cc2cc(Br)cnc2C1 46263,C1(C(N(C2CCN(C(C3CC34CCOC4)=O)CC2)C)=O)CC(O)CN1C 46264,C1(CNC(CC(C)CF)=O)CCC(F)(CNC(c2cc(O)cc(F)c2)=O)CC1 46265,N1(C(C2(C)CCNC2=O)=O)CCCC(NC(=O)CNC(c2ccccc2)=O)CC1 46266,C1(NC(C(C2CCCN(C(c3nc(C)c(C)s3)=O)C2)(C)C)=O)Cc2cscc2C1 46267,c1(C(=O)NC2C(NC(CCNC(=O)NC)=O)CS(=O)(=O)C2)nc(C)c(C)[nH]c1=O 46268,c1(C(N2CCC(CC(=O)Nc3c(C#N)nc[nH]3)CC2)=O)cnn2ccccc12 46269,CCCCC(CN=c1[nH]nc(C(C)C)o1)NC(=O)CC(O)C(C)C 46270,c1(C(=O)NC2CCC(N(C(COC(CC)C)=O)C)CC2)cccc(Cl)c1O 46271,c1(C(N(CCN(C(=O)C(C)c2cc[nH]n2)CC)CC)=O)ncoc1C 46272,C(=O)(C1CCc2nccn21)NCC(=O)NCCCn1c(C)ncc1 46273,Cc1[nH]c2c(C(=O)NC3CC(NC(C4CCSC4)=O)C3)cccc2c1C 46274,C=C(C)CC(C(=O)NC1CCCN(C(C2CCCN2N=O)=O)C1C)NC(C)=O 46275,Cc1cccc(F)c1C(=O)NC1CCC(NC(C2(F)CC=CC2)=O)C1 46276,C(C(C(=O)NCCCCC1CCCC1)N(C)C)NC(C(C1CC1)OC)=O 46277,Cc1cnc(C(=O)NC(C)(C)CNC(=O)CCc2cnc(C)nc2O)c(Br)c1 46278,c1(NC(c2c(C(=O)NC3CCS(=O)(=O)C3)n[nH]c2)=O)n[nH]c2ccccc12 46279,C1(NC(CCOCC#C)=O)CN(C(c2c(C)noc2CC)=O)CCC1CO 46280,N1(C(C=C(CCN(C)C)Cl)=O)CCC(NC(=O)NC2CC(N3CCOCC3)C2)C1 46281,C1(CC(=O)NC2C3CC2N(C(c2csc(Cl)n2)=O)C3)(CO)CCOCC1 46282,C1(CNC(c2ncn(CC)n2)=O)CN(C(C23CCC(CC2O)C3)=O)CCN1C 46283,C(=O)(CC(CC(C)C)NC(C)=O)NC(CC)CN(C(=O)C1=CCCOC1)C 46284,C(=O)(CCCS(C)(=O)=O)N1CCCC(C)(NC(=O)CC(C)(C)c2ccccc2)C1 46285,n1(CC)nc(C(C)C)cc1C(=O)NCCN(C(c1cc(C(N)=O)n(C)n1)=O)CC 46286,C1(CN(C)C)CCCCN1C(C1CNCC1c1cncn1C)=O 46287,c1(C(N(CC(C)NC(c2ccn(COC)n2)=O)C)=O)cn(C)nc1Br 46288,C(=O)(C1=NOC(c2ccc(F)cc2)C1)NC1(C)CN(C(=O)Cn2cc(N)cn2)C1 46289,c1(C(=O)NCC2N(C(C(CC)SC)=O)CCC2)coc2c1CCCC2 46290,C(C(CC(C)C)NC(C1C(C)CCN1C(C)=O)=O)NC(c1nc(OCC)oc1)=O 46291,CC(C(CO)NC(C1CCO1)=O)NC(c1cc(Cl)ns1)=O 46292,c1(OC)cc(NC(=O)C(=O)NC(C)Cn2cnnc2)ccc1C(C)(C)C 46293,CCC(CC(=O)NC(C(=O)NCC(F)(F)C(N)=O)c1ccoc1)C1CCC1 46294,C1(C(=O)NCC2CCN(C(=O)CC34COCC(C3)C4)C2)C2CCCCCC12 46295,C1(CNC(CCNC(=O)Cc2nc[nH]n2)=O)CCCCN1C(C1CC2CC1C2)=O 46296,c1(C(N(CC(C)NC(c2ccn(CC(F)F)c(=O)c2)=O)C)=O)cc(O)cc(O)n1 46297,C(C)(c1ccco1)=NCC1(CC(=O)N)CC1.C12CCC(C1)CNC(=O)C21CC1.CO 46298,CCCCC(CC(=O)NC(CN(C)C)CCO)NC(=O)C=C1CCC(C)CC1 46299,C(=O)(CC1COCc2ccccc21)N(C)CC1CN(c2ncncc2Cl)CCO1 46300,C(=O)(CCCC(C)(C)C)N(C1CCN(C(=O)CN(c2ncccn2)C)CC1)CC 46301,N1(C(CCC=CCC=C)=O)CCCCC1C(C)NC(=O)Cn1cccc1 46302,N1(C(C(C=C)O)=O)CCCOC(CCNC(=O)CCCn2ccccc2=O)C1 46303,C1(CNC(c2n(CC=C)ccn2)=O)CCCCN1C(c1cn(C)nc1C)=O 46304,C(C(C(C)(C)C)NC(c1cc(Cl)c(Cl)[nH]1)=O)NC(C=C1CCC(C)C1)=O 46305,N1(c2nnc(CCc3cccc(OCC(C)C)c3)n2CCC)CCOCC(C)C1 46306,C(=O)(C(F)C(C)(C)O)N1CC(CCO)(NC(C2C(C(=O)OC)C2)=O)C1 46307,C1(CNC(C2N(CC)CC2)=O)CN(C(c2c(Cl)c(C)nn2C)=O)CCC1(F)F 46308,S(=O)(=O)(c1ccccn1)NC1CC(C(N2CCN(C(C)C)CC2C)=O)C1 46309,N1(C(CC(=C)Br)=O)CC(CCNC(c2cnc(C)cn2)=O)OC(C)C1 46310,c1(CC)ncncc1C(=O)N(CCNC(C1CCN1S(C)(=O)=O)=O)C1CC1 46311,C#Cc1ccccc1CN=C(NCC(F)F)NCC1(OCC)CCOC1 46312,N1(C(C2(CCOC)CC2)=O)CC=CC(NC(C23CCCC2(C(N)=O)C3)=O)C1 46313,C1(CNC(C2C(C)NCC2)=O)CC2(CC2)CO1 46314,CC(C)CCCC(=O)NCC1CC(F)(F)CN1C(c1cc(C2CC2)cc(F)c1)=O 46315,c1(CC(=O)N(C(C)CCNC(=O)Cc2cccnc2F)C)c(F)cccc1F 46316,C(=O)(CCCS(C)(=O)=O)NCC1C(C)(C)N(C(=O)C(=O)Cc2ccccc2)CC1 46317,N1(C(c2sc(C)c(C)c2C)C(=O)NCCOC)CC2CCC(C1)C2(F)F 46318,N1(C(c2cnc(C)o2)=O)CC(NC(=O)C(C)Cn2ccnc2)C2(CCCC2)C1 46319,NS(=O)(=O)c1ccc(CNCc2ccccc2C(=O)O)cc1 46320,C1(C2CCN(C(c3cc(Br)co3)=O)C2)(NC(C(=O)NCC2CC2)=O)CC1 46321,C1(C(=O)NCCCN(C(c2nccnc2N)=O)CC)C2CC3C(C2)C13 46322,N1(C(C(C)NC(C)=O)=O)CC2CCN(C(=O)CCN3CCOCC3)C2C1 46323,CCC(CC)(C(=O)NCC1CCC1C(=O)NC(COC)C1CC1)OC 46324,C(N=c1[nH]nc(CO)s1)C1(NC(c2cn(C(F)(F)F)cn2)=O)CCCC1 46325,c1(C(N(CC(CNC(C2(C(F)F)CC(=C)C2)=O)O)C)=O)nc2ccccc2n1CC 46326,c1(C(=O)NCC2CCCN(C(C(C(=O)OCC)F)=O)C2)ccnc2nc(C)nn12 46327,CCCC(C)C(=O)N1CCC(N(C(=O)CCC#N)CC2CC2)C1 46328,CCCCCCC(=O)N1CCC(O)C(C(=O)NC2(c3c(C)cccc3Cl)CC2)C1 46329,C1(NC(c2ccc(N(C)C)nc2)=O)(CO)CCCN(C(=O)Cc2ccsc2Cl)C1 46330,c1(CC)ncc(C(=O)NCC2(CN(C(=O)CN3CCCCC3)C)CC2)c(O)n1 46331,C1(C(=O)NC2CCCN(C(COCCCOC)=O)CC2)Cc2ccccc2S1 46332,c1(C2(C(=O)NC3CCC(CCNC(CCC#C)=O)C3)CC2)cccc(F)c1C 46333,c1(C(N(C(C)C)CCN(C)C(c2n[nH]c3c2COC3)=O)=O)nc(Cl)c(=O)[nH]c1N 46334,C(C)(C)(CN=c1[nH]c2cc(Br)ccc2o1)NC(Cc1c(C)noc1Cl)=O 46335,c1(CC(=O)NC2C(C)(C)C(CNC(C3(CO)CC3)=O)C2)ccc(F)c(Cl)c1 46336,O=C(N=c1[nH]ccnc1Cl)C1CCCN(C(=O)C(F)Oc2ccc(Br)cc2)C1 46337,CC(CN1CCCC1)C(=O)NNC(=O)C(F)(F)F.S(=O)(=O)(c1c(F)cccc1F)N 46338,C#Cc1cnc(C(=O)NCC2C=CCN2C(c2cc3nc[nH]c3cn2)=O)c(C)c1 46339,S(=O)(=O)(c1ccc(Cl)cc1F)NC(C)C(N1CCC(N2CCCC2)CC1)=O 46340,N1(C(C=CCNC(=O)C=Cc2ccco2)=O)CCOC(CC2CC2)C1 46341,C1(NC(CC(=C=C)C)=O)CN(C(c2ccc(NC)c(F)c2)=O)CC12CCOCC2 46342,C(=O)(C1=CN(C)S(=O)(=O)N=C1C)N1C(C)CCC(NC(c2ncn(CC)n2)=O)C1 46343,c1(N2CCCC(C)(CNC(c3n(CC)ccc3)=O)C2)ncnn2cccc12 46344,C1(CCNC(C2CC(=C)C2)=O)CCN(C(=O)CNS(=O)(=O)CCOC(C)C)C1 46345,C(c1ccc(S(=O)(=O)NCC)cc1)=CC(=O)NC1CN(C(CCOC)=O)C2C1C2 46346,Cc1nn(C)nc1C(=O)NCC1CC(C)N(C(=O)CN(C2CCCC2)C)C1 46347,CCCS(=O)(=O)NC(C)C(=O)NC(C)CNC(=O)CN(C(C1CCCCC1)=O)CC 46348,C1(CNC(CCSC)=O)CCN(C(C2(C3CCCCO3)CCC2)=O)CC1C 46349,c1(C(=O)NCC(C)C)ccc(F)c(NC(=O)CCc2ccccc2Br)c1 46350,N1(c2nnc(CCOC)s2)CCCCC(NC(c2cccc(=O)n2C)=O)C1 46351,N1(C(CCCNC(=O)OC)=O)CC2(C1)CN(C(C1CC(C)(C)CO1)=O)C2 46352,C1(NC(CCc2cnc(C)s2)=O)C=CCN(C(C2C(C)(C)C2(C)C)=O)C1 46353,c1(CNC(C2C(O)CCN(C(CCC=C)=O)C2)=O)ccc2nc[nH]c2c1 46354,N1(C(c2cnc(C)n2C)=O)CCC2(NC(=O)CCc3cncnc3)CCCC12 46355,N1(C(C(C)Oc2ccccc2)=O)CCC(C)(C(=O)Nc2nc3sccc3s2)CC1 46356,N1(CCN(C)C(=O)OC(C)(C)C)C(=O)CCN(CC2CCCSCC2)C1=O 46357,C1(C(=O)NC(CC)(C)C2CC2)C2CC1N(C(=O)C(=Cc1cn[nH]c1)C)C2 46358,C1(C(=O)NC(CCSCC)C)(CO)CCN(C(c2cc(O)ncn2)=O)C1 46359,c1(C(=O)NCC2CCCC(C#C)C2)coc2c1CN(C(=O)Cc1cncnc1)C2 46360,C1(CNC(C(=O)NCC2CC2)=O)CC12CCOC2.c12occc1C(=O)NC2 46361,C(=O)(C(C(=O)NC1(C)CC(NC(=O)C(c2ccc(F)cc2)OC)C1)OC)OCC 46362,C1(CC(N2CCC(Cc3cccc(Cl)c3)C2)=O)CCCCN1Cc1cscc1Br 46363,C1(C(N)=O)CN(C(C2CC3CC3N2C(=O)CCCN2CCCC2)=O)CCO1 46364,c1(CNC(N(C)Cc2nnc(-c3ccc(F)cc3)s2)=O)cc(S(N)(=O)=O)co1 46365,Cn1ccnc1Cn1cc(CN2CCC(CNS(C)(=O)=O)C2)nn1 46366,N1(C(CCc2ccc(C)o2)=O)CC(CNC(c2scc(C)c2Cl)=O)CC1C 46367,C1(NC(C2C3(CC(OCC)C3)C2)=O)CCN(C(c2ccncc2C)=O)C(C)C1 46368,C1(C(N2CC(C(C=O)O)C2)=O)CCC=CCC1.CC(C)C(O)C1(CO)CC1 46369,c1(CC(C)N(C(=O)NCCN2CC=CCC2)CC)cccc(C#N)c1 46370,c1(C(=O)NCC2CCN2C(c2cc[nH]c3nccc2-3)=O)cc(F)c(F)c(Cl)c1F 46371,c1(C(N(C2CN(C(C3CN(C(N)=O)C3)=O)CC23CC3)C)=O)n[nH]c2ccc(F)cc12 46372,C(N=c1[nH]c2cccc(F)c2s1)C1C(C)CN(C(c2cc3n(n2)CCCC3)=O)C1 46373,CCC(C)(C)CCCC(=O)NC1CN(C(=O)C(COC)N(C)C)CCC1(C)C 46374,CC1(COC(c2ccc3ncc(Br)n3c2)=O)COCC2CCCN12 46375,C(c1ccc(CC2CC2)cc1)=CC(C(CNC(=O)CC(=O)N(C)C)CN)=O.CO 46376,C1(c2cn(CC)nn2)(OCC)CCOC1.c1(CC=O)cnn(C(C)(C)C)c1 46377,C12(C(N(CCCN(C(C3(COC)CC3(F)F)=O)C)C)=O)CCC(COC)(CC1)C2 46378,N1(C(CCOCCOC)=O)CC2CCN(C(C3(C)CCCN3C)=O)CCC2C1 46379,c1(C(N2CCC(NCCO)CC2)=O)ccc(Cn2cc(C3CCOC3)nn2)cc1 46380,C(C)(C)(CC(C)NC(=O)CCN(C(c1ccc(C)s1)=O)CC1CC1)OC 46381,c1(C(N2C(C)CN(C(c3csc(C#N)c3)=O)C(C)C2)=O)ccc2c(c1)CCN2C 46382,C1(N(C(c2cncs2)=O)CC)CCCN(C(C2(C#N)CCOC2)=O)CC1 46383,C1(C)(NC(C(c2cccc(F)c2)C)=O)CCN(C(=O)C2=CCCC2)CC1 46384,c1(C(=O)NCC2(O)CCC(C)C2)ccc(O)c(N=[N+]=[N-])c1 46385,C1(O)(C(=O)NCCCN(C(c2cc3ccncc3o2)=O)CC)CCCC(C)CC1 46386,N1(C(C(C(C)C)F)=O)CC2CC(C)N(C(=O)CCCOc3ccccc3Cl)C2C1 46387,c1(C(N(C(C)C)CCN(C)Cc2nn(C)cc2Br)=O)c(F)cccc1Cl 46388,CCC(CC)(CO)C(=O)NCC(C)(F)CNC(c1ccc(N)cc1F)=O 46389,Cc1cc(C(N2CCN(C(=O)Cc3cnsc3)C3CC23)=O)c(C)nc1C 46390,C#CCC(C)(C)C(=O)NC1CCCCC1NC(=O)Cc1ccsc1C 46391,c1(CC)nn(C)c(CC)c1CNC(c1ccc(F)cc1)c1nnnn1C1CCC1 46392,N(C(=NCC1CCC(=O)N1C)NC1CCC1(C)C)C(COC)C 46393,C1(C(CNC(=O)C=CC2CCC2)C2CC2)CCN(C(C2C3CNC(=O)C23)=O)CC1 46394,Cc1cc(=NCC2CCOC2)[nH]cc1S(=O)(=O)N1CCCC1 46395,c1(C(=O)NCC2CCCCO2)ccc(CF)cc1.c12ccccc1OC2 46396,c1(C(=O)NCCCN(C(CSCC#C)=O)C)ncc(C)cn1 46397,C(CCCC(=O)N1CC(C(=O)NCCc2cccc(O)c2)CCC1C)(OC)OC 46398,Cc1cc(C(=O)NCc2nc(C(N3CC(OCC(N)=O)C3)=O)c(C)o2)c(O)nn1 46399,C1(C(N(CC(C)(C)CNC(=O)CC2CCCC2(F)F)C)=O)CCN(C)S1(=O)=O 46400,C(=O)(CCC1=CCCCC1)NCc1c(C(=O)NC2CN(C)CC2(F)F)[nH]cc1 46401,C1(N(S(c2c(C)onc2)(=O)=O)C)CCc2ccccc2C1 46402,C(=O)(C1OCCn2ccnc21)NCCCC(CCC)Nc1ncnc(CC)c1F 46403,CC(C)(CNC(=O)CC1CCCC(C2CC2)O1)CCNC(=O)Cc1ccns1 46404,N1(C(=O)NC2CC(COc3ccccc3)C2)CCCC2(CCCNC2=O)C1 46405,N(C(=NCCC12CC(CO1)C2)N(C)Cc1cccs1)C(COC)C 46406,N1(C(c2cc(C)no2)=O)CC(C)(C)CC1CNC(c1nnc(C)cc1O)=O 46407,C1(CNC(=O)CC(F)(F)F)CCN(C(C23CCCC2C3(F)F)=O)CC1O 46408,c1(C(=O)NC2C(C)(C)CN(C(C3CCCOCC3)=O)C2)cnn2cccnc12 46409,Cc1cccc2c(C(N3CCCC3C(=O)Nc3cccc(F)c3)=O)cnn12 46410,CC#CCCC(=O)NC1CC1NC(=O)C(C)CC1CCCCC1 46411,c1(NC(C2CSCCN2c2ccncn2)=O)cc(Br)cc2cn[nH]c12 46412,C12(NC(CC(C)NC(=O)C#CC3CC3)=O)CCC(CC1)C2(C)C 46413,C1(C(N2CC(OC)(CNC(=O)CCn3ccc(C)n3)C2)=O)CCOC(=O)N1 46414,C1(NC(C(=O)N(C2CC(CNC(C3CC3)=O)C2)C)=O)CC(C#N)C1 46415,Cc1c[nH]nc1C(=O)NC(CO)C(=O)N1CCCC1 46416,C(=O)(CCC1CCc2ccccc21)N1CCN(C(c2c(C)scc2)=O)CC1CF 46417,N1(CC)N=C(C(=O)N2CCCC2CN(C(=O)C(O)CC2CC2)C)CCC1=O 46418,C(=O)(C(CC1CCOCC1)NC(=O)C=CC1CCC1)NC(C(C)F)C 46419,Cc1cc(C(=O)NCCC2CCCN2C(=O)C=CC2CCOC2)c(Cl)cc1Cl 46420,c1(C(=O)NCCN(CCC)C(C2CCCCC2C(=O)OC)=O)cnn(C)c1CC 46421,CC(C)(C)S(=O)Cc1cccc(NC(=O)CCOC2CCCCC2)c1 46422,N#Cc1ccc(C(=O)NCC2(CNC(C34COCC3C4)=O)CC2(F)F)[nH]1 46423,c1(CNC(C=CC(CC)C)=O)cccc2c1CN(C(=O)CN(C1CC1)CC)C2 46424,CCC1CN(C(C23CC4(F)CC(F)(C2)CC(F)(C3)C4)=O)Cc2ccccc21 46425,CCC(CN(C)C)C(=O)N(CCCNC(c1sc(C)nc1CC(C)C)=O)CCO 46426,N1(c2nccc(Br)c2)CCC2CCCCC2C1 46427,CCC(C)CC(C(=O)Nc1cnc(SC)nc1)NC(=O)Cn1ccnc1C 46428,c1(C(=O)NCCNC(c2cnn[nH]2)=O)ccc(-c2ccccc2)cn1 46429,CC1CCCC(C(N2CCC(N3CCN(c4cc(=O)n(C)cn4)CC3)C2)=O)CC1 46430,C1(NC(c2cc(OC)no2)=O)CC(CC(=O)Nc2c[nH]ccc2=O)C1(C)C 46431,c1(OC(C)C)ccc(C(=O)NCC2CN(C(C3(O)CC(C)(C)C3)=O)CC2O)cc1 46432,CC1CCOC(c2ccccc2)CN1C(CCCCCS(C)(=O)=O)=O 46433,Cc1cc(C#N)cc(C)c1C(=O)NC1CCN(C(C2CCCC2)=O)CC1O 46434,c1(C(N2CCC(CC(N3C4CCC3COC4)=O)C2)=O)ccc(F)cc1O 46435,c1(OC)ccc(C(=O)N(CC)CC2CCCN2C(=O)C=C2CCN(C)C2)c(C)c1 46436,Cc1ccc(Br)c(NC(c2ccn(-c3cccc(NS(C)(=O)=O)c3)n2)=O)c1 46437,N1(C(C2CC2NCc2c[nH]nc2-c2ccccc2)=O)CCN2CCCCC2C1 46438,N1(C(c2cc(CC)oc2C)=O)CCC2(CCCN(C(=O)C(F)=C3CCCC3)C2)C1 46439,Cc1nn(C)c(C)c1C(N1CCC(N(CCO)C(C2CN(C)CC(C)O2)=O)C1)=O 46440,O=S(=O)(c1[nH]c(=NCC2C(F)(F)C23CCCC3)ccc1Br)NCC1CC=CCC1 46441,Cc1cc(C(=O)N(CCN(C)C(c2scnc2C2CCCC2)=O)C(C)C)no1 46442,C1(CC(=O)N(C(C(=O)N(C)C(C2(N(C)C)CC2)=O)C2CC2)C)CC1(C)C 46443,c1(C(N2CCC(CNC(C(CC3CC3)OC)=O)C2(C)C)=O)cccc2ccnn12 46444,c1(C(=O)NCC2C(C)CCN2C(=O)CSc2ccc(O)cc2)ccc(F)cc1Cl 46445,N(C)(S(C)(=O)=NS(=O)(=O)c1[nH]c2ccc(Cl)cc2c1Br)CC#C 46446,C1(NC(N(CCC)CCC)=O)(Cc2ccc(F)cc2)CCNCC1 46447,N1(C(C(C(C)O)(C)C)=O)C2CCC1CN(C(=O)CC13CCC(CC1)CC3)CC2 46448,C1(C(N2CC(CC(C)NC(=O)C=CCN3CCOCC3)C2)=O)CCC2CC1CO2 46449,CC(C)(C(O)C(F)F)NC(C1COCC1NC(C1CCCC12CCC2)=O)=O 46450,Cc1cc(=O)oc(C)c1C(N1CC(NC(C2COCCN2CC2CCC2)=O)C1)=O 46451,CCCC(CCC)C(=O)NCc1cc(C)c(C(N2CCC2C2CCCOC2)=O)o1 46452,c1(C(=O)NC2C(c3ccc(Br)cc3)(CC)C2)ccc(S(C)=O)c(F)c1 46453,C1(C(N2CCC(O)(CC)CC2)=O)CN(C(=O)Cc2cccc(F)c2)CCC1(C)C 46454,N1(CC(=O)NC(C(=O)N(CCOCC)CC)C2CCCO2)CCC(=O)CC1 46455,Cc1nc(C)n(Cc2cn(CC(C)NC(C3CCC3c3nc[nH]n3)=O)nn2)n1 46456,N1(C(c2ccn(CCC)n2)=O)CC(OC)CC1CNC(C1(C)CC1(Cl)Cl)=O 46457,N1(C(c2c(C)ccnc2O)=O)CCCCC(NC(c2cn(C)nn2)=O)CC1 46458,C(=O)(CC1CCOc2ccccc21)NCC1C(NC(CCN(C)CCO)=O)CC1 46459,N1(C(C(C)(O)c2ccccc2)=O)CC2CC1C2NC(c1ccnc(S)c1)=O 46460,CCC(CC(=O)N1CCC(CN=c2nc(-c3ccccc3)[nH]s2)(C)C1)C(F)F 46461,C1(CCC)(NC(=O)Cc2ccc(F)cc2)CCN(C(c2nnc(S)n2C)=O)CC1 46462,Cc1c(C(C(C)C)NC(N2CCOC(c3ccccc3)C2)=O)oc2ccccc12 46463,c1(C(=O)NC(C)CNC(=O)C(C)C2(O)CCC2)ccc(-c2cnn(C)c2)o1 46464,N(C1CC2(CN(C(c3ccnn3C)=O)C2)n2ccnc21)C(CC(=O)NCC#C)=O 46465,C(=O)(CC(O)C(C)C)NC1CCC(CC(=O)NCc2cc(C)ncn2)CC1 46466,c1(SCC(N2CC(CNC(C3C(CC)OCC3)=O)C2)=O)ccc([N+](=O)[O-])cc1 46467,Nc1ccnc(C(N2CCC(F)(CNC(=O)CC3CSCCS3)C2)=O)c1Cl 46468,CCCCC(C(=O)NOC(C)CC)NC(c1nonc1N)=O 46469,c1(C(N2CC(O)(CC(=O)Nc3nnc(C(C)(C)C)o3)C2)=O)c(Cl)cccc1Cl 46470,N1(C(c2c(C)cccc2)=O)C(C(N)=O)CCCC1C 46471,C(=O)(C1CCCc2scnc21)N1C(C)CN(C(C2CCC(SCC)CC2)=O)CC1.N(C)C 46472,c1(C(=O)NC)nccc(NC(c2cccc(F)c2)CNC(=O)OC(C)(C)C)n1 46473,c1(C(=O)NC2C(C=C)CN(C(=O)COCCC)C2)cc(S(N)(=O)=O)c(C)s1 46474,c1(C(N2CCC(F)(CNC(C3(F)CCOC3)=O)C2)=O)cc(O)nc(C2CC2)n1 46475,N1(C(C=C(C)CNC(C2CCC(C)(C)C2)=O)=O)CC=C(CO)CC1 46476,CCC(C)CCCCC(=O)NCC(CC1CC1)C(=O)N1CC(C)C(F)C1 46477,C(CC(C)C(C)C)NC(C(CN(C)C)NC(Cc1scc(C)c1)=O)=O 46478,c1(C(N2CC(NC(c3c(C)ccs3)=O)C(C3CC3)C2)=O)cc2nc(Cl)ccc2o1 46479,N1(C(c2c(C)nc[nH]2)=O)CCn2c(CNC(C3C(Cl)(Cl)C34CC4)=O)nnc2C1 46480,C1(CNC(c2c(C)con2)=O)CCN(C(C2CCOC2)=O)CC1C1CC1 46481,N1(C(C(C)N(C)C)=O)CCCN(C(c2cc(C(F)(F)F)ns2)=O)CC1C 46482,c1(CN2CC3(CCC(C(=O)Nc4ccnnc4)O3)C2)ccc2nc(O)[nH]c2c1 46483,CCP(=O)(CC)c1ccccc1NC(CC(N)=O)C(=O)O.c12ccccc1OC2 46484,C1(NC(C(C)c2cccs2)=O)C2CCN(C(=O)CC3CCCO3)CC12 46485,Cc1ncnc(C(=O)N(C)CC2(CNC(=O)C(C)CC3CCCCC3)CC2)c1C 46486,Cc1oc2ncnc(O)c2c1C(=O)NC1CCN(C(c2cc(Cl)no2)=O)CC1O 46487,n1(CCN(C)C(C2(C(F)(F)F)CCO2)=O)cc(C2CCCCO2)nn1 46488,c1(OC)cc(NC(=O)NCC2(O)CCOCC2)ccc1F 46489,n1(CCC(=O)N2CC(C3CCCO3)C2)cc(C2CCOC2)nn1.C1(C2CC2)CCCCO1 46490,c1(CC)nc(N2CCCC(NC(=O)C(C)Cc3c(C)n[nH]c3C)C2)cc(Cl)n1 46491,N1(C2CCN(C(=O)CC3COCCO3)CC2)CCN(C(c2cnns2)=O)CC1=O 46492,C1(NC(c2cc(C(=O)OC)oc2C)=O)CC2CC(C1)N(C(c1n[nH]c(O)n1)=O)C2 46493,C1(NC(c2c(C)noc2N)=O)CN(C(c2ccccc2)=O)C2(CCOC2)C1 46494,CC(C)CCCC(C)C(=O)NC1CCC(C)N(CC(=O)N(C)C)C1 46495,N1(C(=O)CCCn2cncn2)CC2CC2(C(=O)NC2CC23CCC3)C1 46496,C1(C(=O)NC2CCCCC2)(CC)CCCN1C(=O)CCSC1CC1 46497,CCC(C)C(C)CNC(C1CC(=O)CN1C(=O)CC1CCC(C)CO1)=O 46498,c1(C(N2CC(N(C)Cc3ccc(Cl)s3)C2)=O)cc(O)cc(Cl)c1 46499,c1(C(=O)NC2C(CNC(CNC(C(C)C)=O)=O)COC2)cnn2cccc(Cl)c12 46500,c1(C(=O)OCC(=O)Nc2c(C)cccn2)cccc2c1C(=O)OC2(C)C 46501,C(=O)(CC1=CCCCC1)NC1C(NC(=O)NCC(C(C(C)C)C)OC(C)(C)C)C1 46502,N1(C(C=CC=CC)=O)CCC2CCC12CNC(c1cn(CC)nc1C(C)C)=O 46503,c1(C(=O)NC2C(CNC(C=COCC)=O)COC2)cccnc1Sc1cccs1 46504,N1(c2nccc(SC)n2)C2CCC1CN(C(=O)C(C)Cn1ccc(C)n1)CC2 46505,n1(CC)c(=O)nc(O)c2c(C(=O)OCCCCCC(F)F)cc(C3CC3)nc12 46506,C12(C(N(C(CCNC(C(C=C=C)C)=O)C)C)=O)CC3CC1C2C3(F)F 46507,c1(C(=O)NC2C(C)N(C(=O)C(O)Cc3cnc[nH]3)CC2)ccc([N+](=O)[O-])c(O)c1 46508,C1(CC(=O)NCCS(N)(=O)=O)C2CCCC2N1C(=O)COC1CCC1 46509,c1(C(=O)OC)ccc(C(=O)NCCCC(C)(C)NC(C2CCS(=O)(=O)N2)=O)cc1 46510,C1(NC(C(C2CCC2)OC)=O)CC(O)(CNC(C2CCCN2C(N)=O)=O)C1 46511,C(=O)(C1=CC2CCCC12)NC1(CNC(COC(C)=O)=O)CCCC1 46512,C(C(C(C)C)NC(=O)CC1(OC)CN(C(=O)CC(C)n2cccc2)C1)OCC 46513,C(=O)(CC(C)(C)C(=O)NC1CN(C(c2cn(C(F)F)cn2)=O)C1)OC 46514,c1(NS(c2ccc(C)cc2)(=O)=O)ccc(C2=CCC(O)CC2)s1 46515,C1(COC)(CNC(=O)CCN(C)CCO)CCN(C(C2CCCC2C)=O)CC1 46516,CC(C)C(O)C(C)C(=O)NC1CCN(C(c2ccn3ccnc3n2)=O)CC1 46517,c1(N2CCC(NCC3(C(C)(C)O)CCCC3)CC2)cc(Cl)ccc1Cl 46518,c1(C(=O)OCC)cc(C(=O)NCc2c(CNC(=O)C(=O)NC)ccs2)oc1C 46519,c1(C(N2C(C)CC(C(F)(F)F)CC2)C(=O)NC2CC2)ccc(F)c2c1CCC2 46520,c1(C(N2CCC(NCc3cn(CC(=O)NC)nn3)CC2)C)ccc(F)cc1F 46521,C1(CC)(CC)CCCN(C(=O)CC2CCN2C(c2ccc(O)cn2)=O)C1 46522,CCCC(C)CCCC(=O)N1CCN(C(c2[nH]c(=N)ccc2Br)=O)CC(O)C1 46523,c1(C(N2CC(NC(C(CCCC)C)=O)C(SC)C2)=O)cc(N)cc(O)c1C 46524,c1(C(=O)NCC2CCCN(C(C(C)NC(C)(C)C)=O)C2)ncc(Br)cc1F 46525,CCC(C)(CC)C(=O)N1CC(OC)C(NC(=O)CCc2ccnc(C)n2)C1 46526,c1(OC)ncc(C(=O)NC2CCC(N(C)C(c3cnc(CC(C)(C)C)o3)=O)C2)s1 46527,c1(C(=O)NC2CC(O)(CNC(C(C)OCCC#C)=O)C2)cc(F)c(F)c(F)c1 46528,N1(C(C=C(C)C)=O)CC2CC(F)(F)CCC2(NC(c2cc(Cl)cnc2O)=O)C1 46529,c1(SC2CN(C(=O)C(O)C3CCCC3)C2)ccccc1 46530,N1(C(C)=O)CCN(C(=O)CCS(C)(=O)=O)C2CC12.C1CS1 46531,N1(C(C(C)(C)SC)=O)CC(NC(C2CN(C3COC3)C2)=O)C(n2ccnn2)C1 46532,c1(C(=O)O)cc2cc(CNc3ccc(C(F)(F)F)cc3F)sc2s1 46533,Cc1oc2c(F)c(F)c(F)c(F)c2c1C(=O)NC1CC1(C)C(F)F 46534,N1(C(COC2(C)CN(C(C3N(C)C(=O)OC3)=O)C2)=O)CCc2n[nH]cc2C1 46535,C1(CC(=O)NC)CN(C(=O)CC(C)(C)SC)CCN1C(=O)C(C1CC(F)(F)C1)O 46536,c1(CC)ncccc1NC(=O)CCC1(NC(=O)CCCF)CCC1 46537,C(=O)(C1CCCc2ncccc21)NCC1(F)CN(C(C2(C)CCCC2)=O)C1 46538,c1(C(=O)NC2C3(CCN(C(C(CCCC)O)=O)CC3)C2)c(C)nc2ncccn12 46539,CN1CC(C(N2CC(C(=O)NCCC(=O)NCC34CC(C#N)(C3)C4)C2)=O)CC1=O 46540,N1(C(CSSC)=O)CC2CC2(CNC(c2csc(C)c2)=O)C1 46541,CC1CCN(C(=O)CC(C)n2cccn2)C(C)C1NC(c1ccccc1F)=O 46542,c1(CCN2CCC(N(C(C(C)NC(CC)=O)=O)C)C2)ccccc1Cl 46543,c1(N2CCC(F)(C(=O)Nc3nccnc3Br)C2)ncnn2cc(Br)cc12 46544,C1(C)(CC(=O)N(CC(CNC(c2nccc(CC)c2)=O)O)C)CCS(=O)(=O)N1 46545,CCC(CC(=O)N(C(C)CCC)C)N(C(=O)CCCN(C)C(C)C)C 46546,N1(C(C2(CC)CCCN2C(=O)C(C2CCCCC2)C)=O)CC2CCCC(C2)C1 46547,C1(CO)CCC2C(CCN2C(c2cc3ccccc3n2CCBr)=O)C1 46548,C1(NC(c2nc(CNC(c3cc(OC)nn3C)=O)oc2C)=O)CCCCC1N=[N+]=[N-] 46549,c1(C(C)C)nc[nH]c(=NCCC2CC2(C)C)c1F 46550,C1(c2ccccc2)(C(=O)NC(CNC(CSC(C)(C)C)=O)CO)CCOC1 46551,CC1C(C(=O)NCC2(CNC(=O)CCc3nc(O)n[nH]3)CC2)=Cc2ccccc21 46552,c1(COC)cc(C(=O)NC2CC2CNC(c2cncnc2)=O)cs1 46553,c1(C(=O)NC2CC(NC(C(F)=C(C)C)=O)C23CCC3)c(F)ccc2nc[nH]c12 46554,C1(CNC(c2cnn(CC)c2C2CC2)=O)CCN(C(=O)C(OC)OC)CC1(F)F 46555,N1(C(C2CCC(CC)CC2)=O)CC(CC(=O)NCCc2cncn2C)CC1(C)C 46556,N1(C(C)=O)CCOC(C(N2CCC(NC(=O)C(F)(F)c3nccs3)C2)=O)C1 46557,c1(C(N(C2C(OC(=O)C=CCO)COC2)Cc2ccccc2)=O)ccnc(S)c1 46558,C1(CNC(CSCCC(C)C)=O)CCN(C(C23COC(CF)(C2)C3)=O)C1(C)C 46559,Cc1cc(CC(N2CCC(C)(CNC(C3CCS(=O)(=O)N3)=O)C2)=O)n(C)n1 46560,N1(C(C2(CCC)CCC2)=O)CCC2C(NC(=O)CCC3CC(F)(F)C3)C2C1 46561,C12(C)CCN(CC1)C2=O.C1(C(C)(C)C)CCCN(c2ncc(I)cn2)C1 46562,C(=O)(N1CCC(C(=O)NCC2CCN(C)C2)O1)c1n(CC)ncc1 46563,c1(C(C(=O)NCC2C(NC(c3c(SC)csc3)=O)CCC2)(C)C)cnccc1C 46564,N1(C(CCc2c(C)n[nH]c2C)=O)CCCN(C(=O)C(C)CC(C)C)C(C)C1 46565,S(=O)(=O)(c1c[nH]c2cc(F)ccc12)Nc1c(C)ccc(-n2cnnn2)c1 46566,c1(C(=O)NCC(C(C)C)NC(c2[nH]nc(OC)c2Cl)=O)c(S(C)(=O)=O)cnn1C 46567,n1(CC(=O)NCC2N(C(CCCCC=C)=O)C3C(C2)C3)ncn2nccc2c1=O 46568,C(=O)(C(O)CCSN1CC2CC2C1)N(C(C)CNC(C1(C(=O)N(C)C)CC1)=O)C 46569,c1(C(N2CCC(C(CNC(C(C)(C)F)=O)O)CC2)=O)c[nH]cc(Cl)c1=O 46570,c1(C(N(C(C)C(=O)NC2C3CCCC23)CC)=O)cc(C)nnc1C 46571,N1(C(CNC2(CC=C)CCOC2)=O)CC2CC(NC(=O)CCCCCC)C1C2 46572,c1(C(=O)NC2CC(C)(COC)N(C(c3[nH]nnc3C)=O)C2)ccn2ncnc2c1 46573,c1(N(CCCN2C3(CC3)C2=O)C)ccccc1.C(N)(=O)NCC#N 46574,N#Cc1ccccc1C1CCN(C(c2cc(CO)on2)C(=O)NCC(F)F)CC1 46575,Cc1cccc(CN2CCC(C(C)(C)O)C2)c1Cl.c12c[nH]nc1CNC2=O 46576,N12CC3CCCCC3(C1)C2.C(=O)(CC(C)(C)C(F)F)Nc1ccc(OC)cc1Br 46577,C(=O)(C(C)(CC)CO)NCCC1N(C(c2cnc(CC)s2)=O)CCOC1 46578,C(CS(=O)(=O)CC(=O)NCC1CCN1C(c1cn(C(C)C)cc1C)=O)OC 46579,N1(c2nccc(C#N)n2)CC2(CCCC2NC(=O)CN2CC3CCC2C3)C1 46580,CC(O)(C(=O)NCC1(NC(c2cnn(CC3CC3)c2)=O)CC1)C1CCC1 46581,C1(NC(c2n[nH]c(C)c2Cl)=O)CCC2(CC1)CCN(C(c1ccc(CO)s1)=O)C2 46582,c1(NCC2(C(N(CCCCC)CC(N)=O)=O)CCCC2)nc(=N)cc[nH]1 46583,c1(C(N(C(C)CNC(c2ccc(-c3cccs3)[nH]2)=O)C)=O)ncc(F)cc1N 46584,C1(C(N(C)CC2CCN(C(=O)CCc3ccccc3)C2)=O)CCC(F)(F)CO1 46585,c1(C(N2CC(NC(c3cncc(C)n3)=O)C(C)CC2)=O)c(C)nc2sc(C)nn12 46586,O=C(C1CCc2ccccc21)N1CC2CC1CN2C(c1cc(F)cc(F)c1F)=O 46587,C(CCCCCCCO)=CC(N1CCC(OC)(CNC(C2CCOCC2)=O)C1)=O 46588,N1(C(C(C)n2ccnc2)=O)CCC(O)CC1C(N1CCC(c2ncco2)C1)=O 46589,C1(C(=O)NCC2(NC(C(CCC)F)=O)CCOCC2)CN2CCC1CC2 46590,N1(CC(C)NC(c2c[nH]c(C(F)F)c2)=O)CCN(C(=O)Cc2ccncn2)CC1 46591,N1(C(COC2CC(NC(C(C)OC(C)(C)C)=O)C2)=O)CC2CN(C)CC2(C)C1 46592,CC(CNC(=O)CCc1cscn1)(CO)NC(=O)Cn1cccn1 46593,c1(C(=O)NCC(CNC(C(CC)N(C)C)=O)(C)O)cc(N)c(C)c([N+](=O)[O-])c1 46594,Cc1oc(C(N2CCOCC2CNC(=O)CC2=CCOCC2)=O)cc1S(N)(=O)=O 46595,c1(C(=O)Nc2c(C(=O)OC)nn(CC(F)(F)F)c2)c(C)cc(C)nc1C 46596,C=CCCCCC(=O)N1CCC(C(=O)NCc2sc(C)cc2C)(CC)C1 46597,Cc1cccc(CN2CC(CNC(C(C)NC(=O)CSC3CCS3(=O)=O)=O)C2)c1 46598,N1(Cc2cccc(OC(C)=O)c2)CCC(NC(C2CCCCC2)=O)C(F)C1 46599,c1(N(C)CC2(OC)CCOCC2)nc(=NCC#CCCO)[nH]c2cccc(F)c12 46600,NC(=O)CCC(C(=O)NC1(C2CS(=O)(=O)C2)CC1)n1cc(CN)nn1 46601,c1(C(N2CC(NC(C(COC)(C)OC)=O)(COC)C2)=O)cc2c(cc1N)OCO2 46602,C1(CSC)CCCN1CCNc1nocc1C(C)(C)C 46603,CCCCC(CNC(=O)CC1(CNC(=O)C(C)n2cccc2)CC1)CCC 46604,C(=O)(C1=Cc2ccccc2C1)NC1C2(CCN(C(COCCOC)=O)C2)CCC1 46605,CCCCCS(=O)(=O)CC(=O)NCC(C)(CO)NC(=O)C(C)NC(=O)CC 46606,N1(C(CSCC#C)=O)CCCC2(CCCCC2NC(c2cnn[nH]2)=O)C1 46607,C1(C(C(=O)OC)(C)C)CC1C1CCN(C(=O)C(C)CC(C)C(=O)O)CC1 46608,C1(Oc2ncc(C)cn2)CCN(N(Cc2cc(C(F)F)cs2)CC2CC2)CC1 46609,C(C(=O)N1CCCCCC1)(C(C)(C)C)N1C(C)CCC1 46610,C1(CC(=O)NC(C(C)NC(CCCn2c(C)ncc2)=O)CO)CC2C=CC1C2 46611,CP(C)(=O)C1(O)CCN(CC(=O)N(C2CCCCC2)Cc2ccccc2Cl)CC1 46612,C1(NC(C2C(=O)NCC2)=O)CC2CC1CN(C(=O)C1=CCOCC1)C2 46613,c1(C(CC)(C)N(C(=O)CCn2cc(-c3cc[nH]n3)nn2)C)ccccc1Cl 46614,C(C(CNC(=O)CN(C1CCC1)C)S(C)(=O)=O)NC(CCC)=O 46615,Cc1ccc(C)n1CC(N1CCCC1CCNC(c1cc(C(F)(F)F)cs1)=O)=O 46616,N1(C(=O)Cc2cccnc2)CC2(CCN(C(C3CCCN3C(=O)C3CC3)=O)C2)C1 46617,c1(C(C(=O)N(C)CCOCCNC(c2cocn2)=O)O)ccc2ccccc2c1 46618,C1(NC(C2COCCN(C(C3(OC)CCCC3)=O)C2)=O)CC(C)N(C)CC1C 46619,c1(OC)cccc(CNC(=O)C(O)C2CN(C(=O)C(C)(C)C#N)C2)c1 46620,N1(C(C(n2c(C)cc(C)n2)C)=O)CCC2C(C1)NC(=O)CN2C(=O)CC1CC1 46621,C1(C(=O)Nc2ccc(C(F)(F)C(F)(F)F)cn2)CC2(C1)C(C(=O)O)C2(F)F 46622,C1(CCC)(NC(=O)CC2C=CCC2)CCCN(C(c2ccccc2CO)=O)C1 46623,c1(N2C(C3CCN(C(C4(SC)CC4)=O)CC3)C(C)(C)C2)nc(C)nc(Cl)c1C 46624,C(=O)(C(C)(C)C(=O)N1CCCC(N(C(=O)CC2(C#N)CCC2)C)C1)N(C)C 46625,C1(N(C(=O)Cn2cccn2)Cc2cc(Cl)ccc2F)CCC12CCNCC2 46626,CC1CC(NC(=O)Cn2cnc(=N)[nH]2)CN(C(=O)COCCN(C)C)C1 46627,N1(C(CNC(C(CC)C)=O)=O)CCCC(CO)(NC(C2CCC2(C)C)=O)C1 46628,N1(C(CN2C(C)CCC2)=O)CC(O)CC1CNC(C1COC1)=O 46629,C(=O)(C(F)C(C)(C)O)NCC(C)CC(=O)Nc1cccc(C2CC2)c1 46630,c1(C(=O)NC(CNC(CC2(OCC)CC2)=O)CC(F)(F)F)ncnc2sccc12 46631,Cc1cnc(Cl)[nH]c1=NC(=O)c1cnc2ccc(-c3ccnc(F)c3F)cn12 46632,c1(C(=O)NC2CC(CNC(C(C)(C)CF)=O)OCC2)cc(Cl)c2n[nH]cc2c1 46633,C(C(C)C)(C(O)C(=O)NCC1(O)CCCN(C(c2cnn(C3CC3)c2)=O)C1)OC 46634,C(CC(C)C(=O)NCC(c1ccccc1F)NC(C1CCC1(F)F)=O)=CCC 46635,CCC(C)(O)CCNC(=O)C(C(C)OC)NC(=O)CN1CCC(=O)CC1 46636,c1(N(C(CCNC(C(CC)NC(N)=O)=O)C)C)cc(Cl)nc(CS(C)(=O)=O)n1 46637,C1(NC(c2ccc(OC)s2)=O)CN(C(=O)CC(C2CC2)C2CC2)CC2(CCC2)C1 46638,CC(C(=O)Nc1cnoc1C1CCC1)C(C)O 46639,N1(C(c2csc(C)c2N)=O)CC(C)CN(C(c2sc([N+](=O)[O-])cc2Cl)=O)CC1C 46640,c1(SC(C)C(=O)NC2CCCCC2CNC(=O)CCNC(N)=O)ccc(F)cc1 46641,C1(C(=O)NC2CCC(F)(F)C2)CC(F)(F)CN1S(=O)(=O)CCBr 46642,c1(C(=O)NCC2CC2NC(c2sc(Cl)cc2Cl)=O)cn2c(n1)CCC2 46643,Cc1nc2ccnn2c(C)c1C(=O)NCC1COCC1NC(=O)CCC(F)F 46644,N(C(=NCCc1ccc2occc2c1)N1CCN(CC2CCCO2)CC1)CC=C 46645,c1(CC(N2C(C)CC(NC(c3cnc(S)[nH]3)=O)C2)=O)cnc2c(=O)[nH]ccn12 46646,N1(C(C(CCC)NC(N)=O)=O)CCOC2(CCCN(C(=O)C(O)C(C)(C)C)C2)C1 46647,C(C(C)CC(=O)N(C(C)CN(C(=O)CN1CC(F)(F)C1)C)C)OC 46648,N1(C(c2n(C)nc(Br)c2)=O)CC(NC(=O)C2CC2)C2(CC2)C1 46649,CC(CCc1ccccc1F)C(=O)NCC1CCCN1C(c1c[nH]nc1Cl)=O 46650,N1(C(CCC(CC)C)=O)CCC2(CCC(NC(=O)C(F)CC(C)C)CC2)CC1 46651,C1(C(N(CCCCNC(c2cc(COC)on2)=O)C)=O)CN(C)CCO1 46652,Cc1nn2c(c1C(=O)NCC1CCCC(NC(=O)Cn3ccnn3)C1)CCCC2 46653,N1(C(c2nnn(CC)c2C)=O)CC(CN(C)C(c2sccc2OC)=O)C2(CC2)C1 46654,C1(C(=O)NCCC(C)NC(C2(F)CC2)=O)CC(C)N(C)C1 46655,N1(C(c2cnc(C(C)(C)C)[nH]2)=O)CC(CNC(=O)CCn2ccnc2)C(O)C1 46656,c1(C(=O)NCC(C(=O)NC2(C)CCC2)OC)cccc(F)c1C 46657,c1(OC)ncc(C(N2CC(CCNC(C3CCC(C)O3)=O)C2)=O)cc1C 46658,c1(CC(C)C)occc1C(=O)NCC(C(C)C)CCN(C)C.C(=O)(COCCO)N 46659,C1(CNC(c2ccc3nn[nH]c3c2)=O)CN(C(c2cc(Cl)no2)=O)CCC1(F)F 46660,N1(C(c2cnc(C(C)OC)s2)=O)CC2C(NC(=O)Cc3cscn3)C2C1 46661,c1(OC)cc(C(=O)NC2CCN(C(=O)C3=C(C)CCC3)C2(C)C)c(F)c(Cl)c1 46662,CC1(C)CN(C(=O)CCC2CC2(Cl)Cl)CC(CNC(=O)C=Cc2cscn2)O1 46663,C1(N(C)C(c2nocc2Cl)=O)CCN(C(=O)CN2CCOCC2)CC1 46664,N#Cc1ccc(C(O)C(=O)OCC2CCC2c2ccccc2)cc1 46665,O=S(=O)(c1ccc(Br)cc1NC1COc2ccc(F)cc21)NC1CCCC1CF 46666,N1(CC2CN(C(C3(C)CCCCC3(C)C)=O)CC(C)O2)CCCC(C2CC2)CC1 46667,c1(C(=O)NCCN(C(=O)COC2CCC2)CCC)snnc1CC.C1CC1 46668,c1(C(=O)NCCN(CCOC)C(c2cccc(N)n2)=O)ccc2nc(S)[nH]c2c1 46669,c1(C(=O)NCCCN(C(C2CCC(C(N)=O)O2)=O)CC)cc(OC)cnn1 46670,N1(C(C(CO)N(C)C)=O)CCOC2CN(C(C3C4CC5C(C4=O)C35)=O)CC12 46671,CC1=C(CNC(=O)NCc2csc(-c3ccccc3F)n2)S(=O)(=O)CCO1 46672,N1(C(Cc2nc(C)sc2C)=O)CCCC(NC(C23CC(C2)C(C)O3)=O)CC1 46673,N1(C(C2(CC(C)C)CCC2)=O)CC2CCC(NC(C34CC(C3)C4)=O)C2C1 46674,C(=O)(C(C(C)C)OCC)NC.C1(=O)CC=CCOC(=O)CN1CC=C 46675,N#CC1(C(=O)NC2CCCCCN(C(c3cccnc3)=O)C2)CC12CCOCC2 46676,c1(Nc2n(CCC)cnc2-c2ccc(F)cc2)c(OC)ncc(Br)c1C 46677,N1(C(CCc2c(C)ncs2)=O)CC=C(CCNC(=O)CCCC2CC2)CC1.C=O 46678,C(=O)(CC1COc2cc(O)ccc21)NC(CC(C)(C)C)CO 46679,C(=O)(C1=CCCN(C(=O)Cc2cccc(Cl)n2)C1)NCC(C)(C)CO 46680,c1(OC(C(=O)NC2C(NC(C3(F)CN(C(C)=O)C3)=O)C2)C)ccc(Cl)cc1Cl 46681,CC1CCC(C(=O)NCc2nc(CNC(=O)C=Cc3ncc[nH]3)cs2)C1 46682,C1(NC2(c3n(CC=C)nnn3)CCN(C(C)C)CC2)CN2CCCC2CO1 46683,C=CCC(C)(CC)C(=O)NCC1CCC1C(=O)Nc1ccc(C)cc1CO 46684,C1(CNC(C2(CSC)CCC2)=O)CN(C(c2sccc2F)=O)CC12CC2 46685,C12(CNC(Cc3cc(C)[nH]n3)=O)CC1CN(C(C1(NC(C)C)CC1)=O)C2 46686,CCC(O)C(C)C(=O)N1CCCCC1CCNC(C1CCCCN1CC(F)F)=O 46687,N1(C(C)(C)CNC(=O)CCc2nc(C(=O)OC(C)(C)C)n[nH]2)CCC(F)(C#N)C1 46688,CCCCC(CNC(C1CCC(CN2CCOCC2)O1)=O)NC(=O)CC1CCC1 46689,CC1CCc2c(C(=O)NCC(C)NC(C3CCC(C)(O)CC3)=O)csc2C1 46690,Cc1cc(C(=O)N(C(CNC(c2cccc(O)n2)=O)C2CC2)C)n2nccc2n1 46691,c1(C(N2C3CC(NC(C=CC)=O)CC2CC3)=O)ccc(=O)n2c1CCC2 46692,Cc1cc(C(=O)NCC23CC(NC(=O)C(C)C4=CCCC4)(C2)C3)n2nccc2n1 46693,C(=O)(C(F)(F)C(C)O)NCC1CC(F)(CNC(c2ccc(C)cc2)=O)C1 46694,CC1CCCC(CCNC(=O)NC2(CCn3cc(Br)cn3)CCC2)O1 46695,CC(C)C(O)CC(=O)N(CCC(N1CCCC(C)(CO)C1)=O)C(C)C 46696,C1(N(C(=O)CCC2CCCCO2)C)CCCN(C(=O)COCc2nc[nH]n2)CC1 46697,CC1CC(NC(=O)CCS(N)(=O)=O)CCN1C(C1CC2(C1)CC2(F)F)=O 46698,C(=O)(C(C)CCCc1cn(-c2ccncc2)nn1)NC(CCC=C(C)C)(C)N(C)C 46699,c1(CC)cc(C(=O)NCC=CCNC(=O)C(F)(F)c2ccnn2C)oc1CC 46700,Cn1ncc(CNCCN2CCN(C(c3ccoc3)=O)CC2)c1C1CC1 46701,Cc1cc(=NC(C)Cc2cn[nH]c2)[nH]c(NC2C=CCCCC2)n1 46702,N1(C(C2C(C)(C)CCCC2)=O)CC2COCCC2(NC(=O)Cc2cc[nH]n2)C1 46703,C1(NC(CC2(C)CCN2C(=O)CCCc2cnn[nH]2)=O)CCCCC12CC2 46704,c1(C(N2CC3C(CNC(c4cn(C(C)C)nc4)=O)C3C2)=O)cccc2cnsc12 46705,c1(C(N(C2(C(=O)NC3(CO)CCCC3(C)C)CC2)C)=O)cc2ccccc2[nH]1 46706,c1(C(=O)NCC(CNC(CCC#CC)=O)(C)O)cc2ccccc2nc1C(F)F 46707,C1(C(C)CNC(=O)CCCc2cnn[nH]2)CCN(C(C2CCOC(=O)N2)=O)CC1 46708,C1(Cc2onc(CN3C(=O)COCC3)n2)CCC2(CCNC2)CC1 46709,c1(C(C(=O)NCC=C)N(CC(=O)NCc2cccnc2)C)cn(C)cn1 46710,CCC(CC(F)(F)F)NC(C1CNC(=O)CN1C(=O)C(C)c1cc[nH]n1)=O 46711,CC1OCCC1CC(=O)NOCC(=O)NCC1(CCCO)CC1 46712,C1(C2CCN(C(c3cc(N)cc(O)c3)=O)C2)(NC(CC2ON=C(CC)C2)=O)CC1 46713,C=CCCC(F)(F)C(=O)NC1CN(C(=O)Cn2cnnc2O)CC2(CC2)C1 46714,C1(NC(c2cc(SCC)ncc2)=O)CC2CN(C(=O)C=CCO)CC12 46715,CC1=NOC(=O)C1CC(=O)NC1CCC(NC(=O)CSc2nncn2C2CC2)C1 46716,O(P(=O)(OCC)C1(C)CCCN1C(=O)Nc1nc2cc(Cl)ccc2n1C)CC 46717,CCC(CN(C)C)CC(=O)N(C)CC1(O)CCN(C(c2cncn2C(C)C)=O)C1 46718,N1(C(CC2(CC=C)CCCC2)=O)CCC2CCN(C(C3C=CCC3)=O)C2C1 46719,c1(NC(C2CSCCN2Cc2scc(Br)c2Br)=O)ccc(O)cc1Br 46720,c1(C(N2C(C)CC(CNC(=O)CSc3nncn3C)C2)=O)ccc2c(c1)CCN2 46721,C1(NC(c2c(C)n[nH]c2)=O)COCCN(Cc2ccc(Br)cn2)C1 46722,c1(C(N(C)CC2CCN(C(c3cn(C(F)F)cn3)=O)C2)=O)ccc2c(c1)COC2 46723,N1(C(C(C)=CC)=O)CCCC(C)(NC(=O)Cn2nnc(-c3ccco3)n2)C1 46724,c1(OC)ccc(C(N2CCOCC2CN(C)C(C2CC(F)C2)=O)=O)cc1OC 46725,N1(C(C2(C#C)CCCC2)=O)CC2CCOCC2(NC(=O)CC(C)(C)CC)C1 46726,c1(N2CCC(CNC(C3CC4CC3C3CC43)=O)C2)ncnc(Cl)c1F 46727,c1(CC(=O)N(CC(O)CN(C)C(C2CC2(C)C)=O)C)cc(Br)nn1C 46728,C1(NC(C2(C(C)C)COC2)=O)CC(CNC(=O)C(C)CC2CC2)CC1O 46729,N1(C(CC(=C)Br)=O)CC(NC(=O)C(C)CC2CCC2)C(C(F)(F)F)C1 46730,C1(C(C)C)CN(C(=O)CCS(C)=O)CCCN1C(=O)CCC1CCN(C)CC1 46731,N1(C(COCCCOC)=O)CCOCC(C(=O)Nc2cc(Cl)ccc2C)C1 46732,C1(C(=O)NC2CC3(OCCC(N)C3)C2)CCC2(CCCCC2)CC1 46733,CC1CCCC1C(=O)NCC(C)(C)CN(C)C(c1cnn(C2CC2)c1)=O 46734,c1(C(=O)NCC#CCNC(CN(CCC#C)C)=O)csc(O)n1 46735,Cc1ccc2cc(Cl)cc(C(=O)NCCn3cc(-c4csc(C)n4)nn3)c2n1 46736,c1(NC(C2(C)CCCN(c3nnc(C)o3)C2)=O)cc([N+](=O)[O-])c(OCC#N)cc1F 46737,C12(C(=O)NC3CC(CNC(C4(OC)CCCCC4)=O)C3)CCC(C)(CO1)C2 46738,C1(C(=O)NC(C(N2CCC(c3ncco3)C2)=O)c2cccs2)CC=CC(O)C1 46739,c1(CCOC)ccc(NC(c2ccc(C3CC3)cc2)C(=O)NCCC2CC2)cc1 46740,N1(C(C(C=C)(C)C)=O)CCC2(CCCN2C(C2CCC3(CCOC3)O2)=O)CC1 46741,c1(C(=O)NCc2ncc(C)s2)ccc(-n2cc(-c3ccnn3C3CC3)nn2)cc1 46742,C(=O)(CC(C)C(C)(C)NC(=O)Cc1ccccc1O)N1CC(CC)N(C)CC1 46743,c1(C(=O)NC2C(NC(C3N(C)CCCC3)=O)CCCC2)cccc(=S)n1O 46744,c1(CC)cc(-c2nc(C(F)F)nn2CCS(C)(=O)=O)cn(C)c1=O 46745,c1(C2C(C)C2)ncc(C(=O)N(C)CCOCCCNC(=O)C(C)(C)F)s1 46746,C1(NC(c2cccc(SC)c2)=O)CC2(NC(c3c(Cl)n[nH]c3C)=O)COC1C2 46747,C(C(=O)N1CCC(NC(C2CC2F)=O)C1)(C(C)(C)C)NC(=O)OC 46748,N(C1CCCc2c[nH]nc21)C(C(C1CCC1)NC(c1cn[nH]c1)=O)=O 46749,C(CS(=O)(CCC(=O)OC(C)(C)C)=NC(=O)c1ccn(Cc2ccccc2)c1)OC 46750,C12(C(=O)NC3(CC=C)CCN(C(C4(C)C(C)(C)C4(C)C)=O)C3)CCCC1C2(F)F 46751,C(=O)(CCCCCc1cccs1)NC(C)CN(C(=O)C(O)C1CCCC1)C 46752,C(C(=O)NCC1CCC(C(=O)NCc2ncc(CO)[nH]2)CC1)(C(C)C)SC 46753,O=C(CC(F)(F)F)NCC1CCCCC1NC(c1ccc(OC(F)(F)F)cc1)=O 46754,N1(C(C(CC)(C)CO)=O)CCC2(CC1)COCC(CNC(C1(C)CCC1)=O)O2 46755,c1(C(N2CCCC(CNC(C3CCS3(=O)=O)=O)C2)=O)ccc(F)c2occc12 46756,C(=O)(C1Cc2ccc(Cl)cc21)N1CCC(C(C)(C)NC(C(C)SC(C)C)=O)CC1 46757,C(=O)(C(F)(F)C(C)O)NCCCC1CCN(C(c2cc(C)c(C)[nH]2)=O)CC1 46758,c1(C(=O)NCC(CC=C)NC(C2CS(=O)(=O)C2)=O)coc2c1NC(=O)CCC2 46759,C1(CNC(C(C)Cc2ccco2)=O)CC2CC2N1C(=O)C#CC(=O)N(C)C 46760,C1(CNC(CCCOC)=O)CC(C)(C)CN1C(c1ccc(C(=O)N(C)C)nc1)=O 46761,c1(C(=O)NC(C(C)C)CCN(C)C(c2cc(O)ncn2)=O)ccc2c(c1)C=CCC2 46762,C1(C)(C(=O)NCC(n2cc(-c3cc(CC)on3)nn2)C)COCCO1 46763,c1(C(N2CC(CC(C)NC(C(CC)c3ccccc3)=O)C2)=O)[nH]c(C)nc1C 46764,N1(C(C(COCC)(C)C)=O)CCC2(CC2NC(c2coc(C)c2)=O)C1 46765,C(=O)(C(C)CCCOC)NC1C(CCC)CN(C(c2cnn(C3CC3)c2C)=O)C1 46766,C(CC(C)(C)C)N(C(C1(C(C)NC(C2CC23CCC3)=O)CC1)=O)C 46767,c1(C2C(NC(=O)COC3CCN(C(=O)C=CCO)C3)CC2)cccc(F)c1 46768,CC1CC(N(C)C(C2CN(C(=O)C(C3CCOCC3)C)CC2F)=O)CCO1 46769,c1(C(N2C(C)CC(NC(C3CC3(C)C)=O)CC2)=O)cc(F)c(O)c(F)c1 46770,c1(C(=O)NCc2c[nH]nc2C2CCN(C(=O)C=C3CC3)C2)ccc2n[nH]cc2c1 46771,C1(NC(CCOCCN(C)C(C2CC(C)(C)CO2)=O)=O)CCN2CCCCC12 46772,C#CCCCC(c1nnnn1C1CC1)N(c1ccc(F)cc1)C(N1CCC(C)C1)=O 46773,c1(C(=O)NC2CCN(C(c3cnc(-c4ccoc4)s3)=O)CC2)cnn2c1OCC2 46774,c1(C(N2CCc3nc[nH]c3C2)C(=O)NC(C)C)cc(F)c(Br)cc1F 46775,C1(CC)CCC(C)CN1C(C1CCN(C(=O)C=CC(=O)OCC)C1C)=O 46776,CCC(CC(=O)NC(CNC(=O)COc1cc(C)on1)C1CCC1)C(C)C 46777,c1(CN(C(CN(C(C(=O)NC)c2cscn2)C)=O)C)ccc(Br)cc1Cl 46778,c1(C(=O)NC2CCN(C(C(CC)SC)=O)CC2(C)C)cc2c(C)cccn2n1 46779,C1(NC(c2cc(C)ns2)=O)CN(C(=O)CCSc2ccccc2)CC1C 46780,C1(N(C(=O)CC2COC(=O)C2)C)CCN(C(c2cnc[nH]2)=O)CC1 46781,c1(C(=O)NCCNC(C(C2CCOC2)OC)=O)cn2cccnc2n1 46782,N1(C(CC=C=C)=O)CC2(CCOCC2)CC1CNC(c1cnc2sc(C)cn12)=O 46783,c12ccccc1S2.C(CCCCC(=O)NOC(C)CC)NC(C(C)OCC=C)=O 46784,C1(C)(NC(CC2(C)N(C(c3ccc(C(C)C)o3)=O)CC2)=O)CCCC1C 46785,C1(NC(C(CC)COC)=O)CN(C(c2cnc(OC)nc2)=O)CC1S(C)(=O)=O 46786,c1(CCC(=O)N(C2CCCN(C(C3CCOC3)=O)C2)C)cn2ccccc2n1 46787,C1(NC(c2c(NCC)ccnc2)=O)CC(OC)CN1N1CCC(C(=O)NC)C1.C(C)=O 46788,C1(N(C(Cn2c(C)cnc2)=O)C)CN(C(=O)CCOc2ccccc2O)CC1O 46789,N1(C(C=C(C)C(C)(C)C)=O)CCC(N(CCO)C(C2CC(C)C2)=O)CC1 46790,Cc1cc(C(=O)NC2CCCCC2NC(C2CC(C(C)(C)C)C2)=O)nnc1C 46791,CCCCC(CC)C(=O)NCCOCCCN(C)C(C12CC(C(F)F)(CO1)C2)=O 46792,C1(NC(c2cc(C)c(Br)o2)=O)CN(C(=O)CNS(N)(=O)=O)CC1C1CC1 46793,N1(C(c2n(CC#C)ccc2)=O)CCN(C(C2CCCS(=O)(=O)C2)=O)C(C(C)C)C1 46794,Cc1nc(C(=O)NC2CCC2NC(c2csc(Cl)c2)=O)c(C)s1 46795,C#CC1(C)COCCN1C(=O)CCn1cc(-c2cnn3c2NCC3)nn1 46796,N1(C(c2n(C)nc([N+](=O)[O-])c2)=O)CCCC2(CCCCC2NC(=O)CO)C1 46797,Cc1cc(C(=O)N(C)CC2CCCCN2C(C23CCC2C3)=O)c(C)n1C(C)C 46798,C1(CC(N2CC=CC(NC(c3c(C)cco3)=O)C2)=O)CCCC(F)(F)C1 46799,CC1=CC(C)CN(C(c2ccc(C(=O)NCC(C)C)cc2)C(=O)NC2CC2)C1 46800,C1(C(N2C(C)CC(CNC(CCC(C)N(C)C)=O)C2)=O)CC2(CCO1)CC2 46801,C1(CNC(c2n(CC)cnn2)=O)CCC2(CCN(C(=O)C(F)C(C)C)CC2)CO1 46802,CC1CN(C(=O)Cc2cc(Br)ccc2C(F)(F)F)CCS1(=N)=O 46803,C1(O)(CNC(c2cc(OC(CC)C)ncc2)=O)CCCN(C(=O)CNC=O)C1.OCC 46804,C1(N(C)C)CCC(n2cc(CN(CC3CC3)CC3CC(O)C3(C)C)nn2)CC1 46805,c1(C(=O)NC(CNC(C(C)OC2CCOC2)=O)C2CCC2)ccn(C2CC2)n1 46806,C1(N(C(C(C2CC2)OC)=O)C)CCC(NC(c2nnsc2C(F)F)=O)CC1 46807,C1(C(N)=O)CC(C(=O)NCC(C)(C)CNC(=O)CCSc2ccccn2)=NO1 46808,c1(OCC(=O)NC(C2CCCCN2C(=O)C(C)O)C)cccc(-n2cnnn2)c1 46809,CC1(CC(=O)NC2CCC(NC(C3CCCC3(C)C)=O)C2)Oc2ccccc2O1 46810,C12(C(N3CC(O)(C(C)NC(=O)C(F)CC4CCC4)C3)=O)CC3CC1C2C3 46811,N1(C(c2n(CC)ccc2)=O)CCOC2CN(C(=O)C(c3ccccc3F)C)CC12 46812,CCC(C)C(C(=O)N(C)Cc1nccn1CC)NC(C1CCCSC1C)=O 46813,C(CCC(C)(C)NC(=O)C=CBr)NC(C=CCCC(C)C)=O 46814,c1(C(=O)OC)cnc(CNCCC2(C)CC2(F)Cl)[nH]1 46815,c1(C(=O)NC(CN(C(=O)C(C2CCOCC2)O)CC)C)cc(C(C)C)n(C)n1 46816,c1(C(N2C(C)(CC)CC(NC(=O)CCCCCF)C2)=O)nc2c(s1)COCC2 46817,CN1CCc2cc(C(N3CCC(N(C(=O)C=CS(C)=O)CCO)C3)=O)sc2C1 46818,CC(C)C#CC(=O)NC1CC(CNC(C2CC(O)C(F)C2)=O)C1 46819,C1(C)(C(=O)NCC(N(C(C(C)n2cccc2)=O)C)C2CC2)CCCS1(=O)=O 46820,C12(CCNC(=O)Cc3ccccc3F)CCC(C1)N(C(c1ns[nH]c1=O)=O)C2 46821,C1(CC(C)NC(C2(CC#C)CCC2)=O)CCN(C(=O)CNC(C)=O)CC1 46822,C12(C(N3CC(SC)C(NC(=O)CC4CCCN(C)C4)C3)=O)CCC(CC1)CC2 46823,C1(C(=O)NCC2CC(NC(C(COC)O)=O)C2)Cc2cc(C)ccc2S1(=O)=O 46824,c1(C(=O)NC(C)CCF)ccc(CNC(C2CC2F)=O)nc1 46825,C1(NC(CCSCCC)=O)CC(C)N(C(=O)C(=O)NCC(F)F)C1 46826,C12(NC(CCCC#C)=O)CCN(C(c3cnoc3-c3cnn(C)c3)=O)CCC1C2 46827,C1(CC(=O)NC2C(CNC(c3c(C)ocn3)=O)CC2)CCC2(CC1)CC2 46828,CCCC(CNC(=O)C(CC)OC)C(=O)NC1CCN(CCC)C1 46829,c1(C(=O)NC(CC)CN(C(=O)C=Cc2scnc2C)C)ccc(CO)cc1OC 46830,C(CC(Cc1ccco1)N(CCCN(C)Cc1ncn(C)n1)C)OC 46831,C1(NC(C(=O)N(C)C)=O)CC2CCC1N(C(c1ccccc1Cl)=O)C2 46832,c1(CC)ocnc1C(=O)N(CC(C)CNC(=O)Cn1cnnc1O)CC 46833,N1(C(C2N(CC)C(=O)CC2)=O)CCCC(NC(c2cnc(C)n2C)=O)C1C 46834,C1(C)(NC(CC2(O)CCN(C(C3C(CC(C)(C)C)C3)=O)C2)=O)CCCCC1(C)C 46835,S(=O)(=O)(c1sc(O)nc1C1CC1)NC(C)C(N1CCOCC1C)=O 46836,C=C(Cl)CC(C(=O)NCc1cnc(F)c(C)c1)NC(=O)C(C)C(F)(F)F 46837,c1(N(CC(CCC)C)C)cc(NC(COC)CC(C)C)nc(C)n1 46838,NC(=O)C(N)CCC(=O)NCC1CN(C(c2ccc(C3CC3)nc2)=O)CCO1 46839,CC1CCN(C(=O)COC2CCOC2)CC1CNC(=O)CCC(C)(C)F 46840,c1(C(=O)NC(C2CN(C(c3cnn(C4CCCCC4)c3)=O)C2)C)ccsc1C#N 46841,Cc1c(C(N2CC(CNC(=O)C(C)Cn3ccnc3)C(O)C2)=O)ccn1C1CC1 46842,CC1CC(C)CN(C(=O)NC(c2ccc(C(F)(F)F)cc2Br)C)C1 46843,CCC(C(=O)OC)C(=O)N1CCCCC1CCNC(=O)CCc1c(C)n[nH]c1C 46844,c1(CC(=O)NC(C2(O)CN(C(c3c(C#C)c[nH]n3)=O)C2)C)ccc(Br)cc1C 46845,Cc1csc2ncc(C(=O)NC3CN(C(=O)CSC(F)(F)F)CC3O)n12 46846,Cn1nc(I)cc1NC(=O)NCC1(C)CC(F)(F)C1 46847,c1(CCC)nc(C)c(C(N2CC(CNC(C3(C#N)CCC3)=O)CC2C)=O)o1 46848,C1(OC)CC(C)N(C(=O)C(=O)NC(c2nn[nH]n2)C2CC2)C(C)C1 46849,c1(C(N(C2CCC(NC(C3C(C(=O)OC)C3)=O)CC2)C)=O)cc(Cl)c(N)cc1F 46850,C#CCC(C)(C(=O)NC(C)C(=O)OCC)NC(=O)CN1C(=O)CNC1=O 46851,N1(C(c2n(C)c(S)nn2)=O)CCCN(CC(O)Cc2ccc(O)cc2)CC1 46852,C1(C(=O)NCC(C)(CO)NC(=O)CN2CC3CC3C2)CCC(=O)NC1 46853,N1(C(COC(C)C)=O)CCCC2CN(C(=O)CN3CCN(C)CC3)CCC12 46854,N1(C(C(CC)(C)C)=O)CCC2CN(C(c3c(OC)ccnc3F)=O)CCC2C1 46855,C(CC(C)C)(C(=O)N1CC(NC(C23CCCC(C2)OC3)=O)C(C)C1)OC 46856,n1(CC)nc(C(=O)NCCC2CCN(C(=O)CCC(C)SC)CC2)cc1O 46857,N1(C(C2(F)C(C)OCC2)=O)CC2CC1CCC2NC(c1nncs1)=O 46858,c1(C(C)C)nn(C)c(NC(C2(CC(c3cc(C(C)(C)C)[nH]n3)=O)CC2)=O)c1Cl 46859,Cc1nc2ccnn2cc1C(N1CC(NC(=O)C=CCF)C(C)C1)=O 46860,c1(C(=O)NC23CC(NC(c4cscc4C4CC4)=O)(C2)C3)cc(Cl)cnc1O 46861,c1(C(=O)NCC2(F)CC(CNC(c3sc(CC)c(C)c3)=O)C2)cc(N)cc(F)c1 46862,c1(N2CCCC(C(C)NC(c3cncc(Cl)c3)=O)C2)ncc2c(n1)CCCCC2 46863,N1(C(C2(CCCC)CCCC2)=O)CCC(NC(C2CCCCC2O)=O)CC(O)C1 46864,C1(NC(=O)CCCn2ccccc2=O)CN(C(=O)Cn2nccn2)CCC1CO 46865,c1(C(=O)NC2CN(C(CSc3ccc(OC)cc3)=O)C2)nc2cccnc2s1 46866,C(=O)(C(O)CCCNC(=O)CC1CCOC1(C)C)NC1CC(COC)C1 46867,S(=O)(=O)(c1cccc(Cl)c1Cl)N1CC2(CC(NC(c3c(OC)nn(C)c3)=O)C2)C1 46868,Cc1c(C(=O)N(CC(C)NC(=O)CCC=CBr)C)ccn1C 46869,N1(C(C=CCNC(C(c2ccn(C)n2)C)=O)=O)CCOC(C2CCC2)C1 46870,c1(CC)ncc(C(=O)NCCOC2CCN(C(C3CC3C(C)(F)F)=O)C2)c(O)n1 46871,c1(C(=O)NC2CCN(C(C(F)=CC)=O)CC2(C)C)cc2c(nc1O)CCCC2O 46872,Cc1nnc(N(C2COC2)C(C2(C)CCCC2(F)F)=O)nc1C 46873,c1(NC(c2n(CC)nnn2)c2ccccc2)cc(CO)ccc1OCC 46874,N1(C(CC2(CC=C)CCCC2)=O)C2CCC1C(CNC(c1cc(C)ns1)=O)C2 46875,c1(CC(=O)N(CCOCCOC)C)cc(C(=O)NCC2(CCOC)CC2)on1 46876,c1(C(N2CC(NC(C(C)(C)C3CCCCO3)=O)C(O)C2)=O)cccc(Cl)c1Cl 46877,CCCC(C(=O)NCC(CO)NC(c1c[nH]nc1CC)=O)OC 46878,CCCCC(O)C(C)C(=O)N(CC(=O)NCC1CC2C=CC1O2)C 46879,c1(C(=O)NC(C)C(CO)NC(=O)C(O)C2CC2)cnc(CC2CCCC2)nc1O 46880,N1(C(CCCCCSC)=O)CCCC(C2CCN(C(C3(CO)CC3(F)F)=O)C2)C1 46881,c1(C(=O)NC2(C(NOCC(C)(C)O)=O)CC2(C)C)cnn2c1CCC2 46882,C=CCCC(=O)NCCC(C)N(C)C(c1occc1Cl)=O 46883,c1(OCC)ccc(C2CCN(C(=O)C(N3CCOC(CN(C)C)C3)=O)C2)cc1 46884,C(=O)(C(F)CCCCC(CC)CC)N1C(C(=O)OCC)CC2(CCCCC2)C1 46885,c1(CNC(c2cccc(N)c2F)=O)nc2c(s1)CCN(C(=O)CNC(N)=O)C2 46886,C1(C(N(CC(CC)NC(CC(C=C)(C)C)=O)CC)=O)CCC2(CC1)CNC(=O)C2 46887,c1(C(=O)NC2CCN(CCNC(CCC)=O)CC2)c[nH]c2c(Cl)cccc12 46888,C1(C2CCC2)(CNC(C2C(=C)CC2)=O)CCN(C(c2cnc(O)c(C)c2)=O)CC1 46889,C1(C2CC2)(CNC(c2cc(OC)n(C)n2)=O)CCN(C(C2CN(C(N)=O)C2)=O)C1 46890,C#CCC(C)(C(=O)NC(C(F)(F)F)C1CC1)NC(C1COCOC1)=O 46891,c1(C(=O)NCC(CCNC(c2cc(OC)c(C)cc2)=O)O)cc2n(c1)CCCC2 46892,CC(CC(=O)NCCN(CCO)CCO)(C(=O)O)N.C(=O)(COCCOC)CCO 46893,CCCC(CCCNC(c1c(C)nn(CC)c1C)=O)NC(=O)Cc1nonc1C 46894,N(C(=NCC(C)Oc1ccccc1)NC1C(C)(C)C1(C)C)C(C)C1CC1 46895,c1(N2CC3OCC(COC)C3C2)nc(=NC)[nH]c(=NCCCC(=O)NC(C)C)[nH]1 46896,C(=O)(CCC(=O)c1ccc[nH]1)N(CCN(C(c1ccnnc1O)=O)CC)CC 46897,C1(NC(c2ncn(CC)c2)=O)COC2(C1)CN(C(c1c(C)cnn1C(C)C)=O)C2 46898,C12(CNC(C(F)(F)C3(OC)CCC3)=O)CCC(NC(=O)CC3CC34CC4)(CO1)C2.S 46899,N1(C(C(C(C)C)SCC)=O)CCN(C(=O)CCCc2ccc(F)cc2)C(CO)C1 46900,c1(SC)cc(C(N2CC(N(C(=O)Cc3cc(C#N)cs3)C)C2)=O)ccc1[N+](=O)[O-] 46901,C=CC(C)(CC)C(=O)NC1CCOC(C(=O)NOCC(F)(F)F)C1 46902,c1(N(C)C)cccc(CNC(c2ccn(C3CCNCC3)n2)=O)c1 46903,c1(C(C)=O)cc(C(=O)NCC2CN(C(=O)C3CC3)CCCO2)c(C)nc1C 46904,N1(C(Cc2c(C)non2)=O)CC(C)(C)CC1CNC(C1CCC1(C)C)=O 46905,CCCCCCCCC(=O)NC(C)(C)CC=CC(=O)N(CC(C)CO)C 46906,C1(NC(CS(=O)(=O)NC)=O)CCCC12CN(C(C1CCCCN1C(C)=O)=O)C2 46907,C(=O)(C1=NNC(=O)CC1)N1C(C)CCC(NC(c2cc(CCC)ncc2)=O)C1 46908,C(=O)(C1=CCC(C)(C)CC1)NCC1CCC(CNC(c2ncn(CC)n2)=O)CC1 46909,c1(NC(C2N(C(c3cc(CC)[nH]n3)=O)CC(O)C2)=O)ncc(Br)nc1C#N 46910,C=C(C)C(CC(=O)NCCCNC(=O)C(c1cc(F)cc(F)c1)O)OCC 46911,C(CCCO)CN(C(=O)C(C1CC1)N(C(=O)C=CC1CC1)C)C(C)C 46912,c1(CNC(COCC(=O)NC)=O)ccc(C(=O)NCC2(C)CC=CCC2)cn1 46913,C#Cc1ccc(Br)c(C(=O)NCC2CN(C(c3cc(C)oc3C)=O)C3CC23)c1 46914,c1(OC(=O)NCC(=O)NCC(C)N(C)C)cc(C(F)(F)F)ccc1O 46915,C1(NC(c2c(COC)cccc2)C(=O)NC)CCCCC1(C)NCC1CCC=CO1 46916,C(=O)(C(C(=O)NC(C(=O)N(CC(C)(C)O)C)C1(C)CC1)OC)OC 46917,C(C(O)(C(F)(F)F)c1nccn1C)NC(C1(CNC(CC(=O)OCC)=O)CC1)=O 46918,C(=O)(C(F)C(CC)CC)NC(C(N1CC2(CC(=C)C2)C1)=O)C1CCCC1 46919,C(=O)(C1OC(=O)c2ccccc21)NCCCNC(CSC(=N)N)=O 46920,N1(C(c2cn(CC)nc2C)=O)CCC(C)(C(=O)NC(C)CC2CCC2)CC1 46921,N1(C(c2cc(C3CCCC3)[nH]n2)=O)CC2CCC(C1)N2C(C1C2CCC1CC2)=O 46922,c1(C(C(=O)N(CCCN(C(Cc2c(C)cc(C)s2)=O)C)C)O)ccc(Cl)c(Cl)c1 46923,C1(=CCNC(C(C)CO)=O)CCN(C(=O)CN(C)Cc2ccccc2)CC1 46924,C1(NC(CC2CN(C(C(=O)NCC)=O)CC2C)=O)CCN(C)CC1C 46925,CCC(CC)(CC)C(=O)NCCN(C(=O)Cc1cnc(C)[nH]1)Cc1ccccc1 46926,N1(C(C2CN(C)C2)=O)CCn2c(-c3ccc(Cl)cc3)nnc2C1 46927,CC1CN(C(=O)C(C)n2cnnn2)CCCN1C(c1cn(C)[nH]c1=N)=O 46928,C(C1CCCn2ccc(C(=O)O)c21)NC(C(c1ccn(C)n1)C)=O 46929,c1(C(C)=O)cc(C(=O)NC2CCC(CNC(=O)Cn3cc(Cl)cn3)C2)ccc1C 46930,CCCC(C(O)C(=O)NC1CCN(C)C1=O)NC(=O)C(C)C(F)F 46931,N1(C(CNS(NC)(=O)=O)=O)CCN(C(c2n[nH]cc2C(=O)OC)=O)CC(CO)C1 46932,c1(C(N2C(CN(CCC#C)C)CCCC2)=O)cc(C)c(Cl)c(C)c1 46933,c1(OCC)cccc(CS(=O)CC(=O)OCc2ccc(CC)cc2)c1 46934,c1(C(=O)NCC2CC(NC(CCNC(C)=O)=O)C2(C)C)ccc2c(c1)COCC2 46935,c1(C(=O)NC(CSC)(C)C(=O)N2CCC2(C)CCO)nc(C)ccc1C 46936,CCC(C)C(C)C(=O)NCCN1CCN(C(c2ccnc(OC(F)F)c2)=O)CC1 46937,N1(C(C(c2ccco2)NC(CCC=C(C)C)=O)=O)CC2CC2C2CC12 46938,c1(C(=O)NC(C2CN(C(C3C(OCC)C3)=O)C2)C)nccn2ccnc12 46939,C1(CNC(CCN(CC=C)C(C)=O)=O)CCCN(C(=O)CC2(C#N)CCC2)C1 46940,N1(CC(C)C)CCCC(C(=O)N(CC(C)(C)CNC(C2CCNC(=O)C2)=O)C)C1 46941,C(CN=[N+]=[N-])(C(=O)N1CCC(CCC)C1)NC(C(C=C)OC)=O 46942,C(CCO)(C(F)F)N(C(=O)CN(C(=O)C(O)CC1CCCC1)CC1(C)CCC1)C 46943,C1(NC(C(C)SCc2ccccc2)=O)CCCC(NC(c2ccnnc2O)=O)C1 46944,c1(C(N(C)CC2CCCN2C(C2CCCC2(C)C)=O)=O)cc2c(s1)CCC2 46945,c1(C(=O)NCC(CN(C(C(=O)NCCNC(C)=O)=O)C)C)ccnc(S)n1 46946,C1(C(N2CCSCC2)=O)Cc2nccnc2CN1C(=O)C1=NOCC1 46947,C(=O)(C(C)(C)CC(C)(C)C)NCC(C)NC(=O)Cc1csc(N2CCNC2=O)n1 46948,N1(C(C(C)OC2CCCC2)=O)CCCCC1C(=O)NC1CC2(CC2)C1.C1C(=O)N1 46949,C(=O)(C(CC(C)C)ONC(=O)CCC1CCOC1)N(CC(=O)NC)CC=C 46950,C(=O)(CCCCCn1cnnn1)NC1CCCN(C(c2ccc(OC)cc2)=O)C1 46951,c1(C(N(CCOC2CN(C(=O)C(O)C(C)C)C2)CC)=O)cc(P(C)(C)=O)ccn1 46952,c1(C(=O)NCC(C)CN(C)C(C2(N(C)C)CCC2)=O)occc1C1CC1 46953,N1(C(C#CC(=O)O)=O)CCCC12CN(C(c1ccc(O)c(I)c1)=O)C2 46954,CC1CCN(C(=O)COC2CCC2)C1C(=O)NCc1ccc(F)cc1 46955,c1(C(N2CC(NC(=O)C(C)(C)CO)CC(C)(C)C2)=O)cc(Br)c2nccn2c1 46956,C(=O)(CCCC(=O)N1CC2(CCNC(=O)CN(C)CCO)CCC1C2)NCC 46957,c1(SC(C)C(=O)NC(=O)NCC(=O)OCC2OCCC2(C)C)ccc(F)c(F)c1 46958,c1(C(=O)NC2C(C)N(C(c3cccc(Cl)n3)=O)CC2)c(F)ccc(F)c1N 46959,C1(CNC(c2c(C)csc2Cl)=O)C(C2CC2)CCN1C(=O)CC(C)C(F)(F)F 46960,c1(C(=O)NC(C)(C)CNC(=O)C(C2CCCCC2)F)ccc(OCC(N)=O)cc1 46961,c1(C(=O)NCC(C)(CC)NC(C(CC)=CC)=O)cccc2c1ccn2C(C)C 46962,C1(C2CCN(C(c3ns[nH]c3=O)=O)C2)CCCCN1C(c1cscn1)=O 46963,CN(C1CN(C(=O)CCCC2CCCC2)CCc2ccccc21)C(=O)C=CCO 46964,C(=O)(C(C)(C)CC(C)(C)C)NCCC1(CNC(c2nccc(C)n2)=O)CC1 46965,CCC(N=c1cc(NCCOCC2CCCCO2)nc(C(F)(F)F)[nH]1)C(C)C 46966,c1(N2CCN(C(C)CO)CC2)nc(N(C)CC2CCCO2)c2cnn(C)c2n1 46967,C(=O)(C(F)n1ccnc1)N(C(C)C(=O)NCCN(C)C(C)=O)CC 46968,C1(CNC(C(=O)NC(C)C)=O)COCC2(CCN(C(=O)CCCC3CC3)C2)O1 46969,N1(C(C2(CCN=[N+]=[N-])CC2)=O)CC(=O)NCC1C(N1CCNC(=O)C1)=O 46970,c1(C(=O)NC(CC(C)NC(c2c(NC)cccc2)=O)C)c(F)cc(C)cc1Cl 46971,C(C)(C(C)C(=O)NCC1(C2CCC2)CC1)NC(C(C=C)C)=O 46972,c1(C(=O)NCC#CC)c[nH]nc1CCNC(C1CCN1C(C)(C)C)=O 46973,N1(CC)CC(NC(=O)Cn2cc(CNC(c3nc(C)c(C)s3)=O)nn2)C(C)C1 46974,C1(NC(C)=O)CCCCN(C(C2CC3(C2)CC2(CC2)C3)=O)CC1 46975,c1(NC(C2CC2Cl)=O)cccc(Oc2cccc(F)c2)c1 46976,Cc1cn2c(n1)C(C)N(C(=O)CC1CC3(C1)CN(C(=O)OC(C)(C)C)C3)CC2 46977,c1(C(=O)NCCN(CCC)C(C)C)cnn(CCNC(=O)CCN2CCCC2)c1 46978,N1(CC)CCCN(Cc2nc(Br)nn2CC)CCC1 46979,N1(C(CCCOCCOCC)=O)CCC(C)N(C(=O)C(C)SC2CC2)CC1 46980,C1(C(N(C(C)CNC(C23CC(C2)C3)=O)C)=O)CCCC(C)CC1 46981,c1(C(N2CCC(C)(CNC(CC3CC(OC)C3)=O)C2)=O)ncc(Br)cc1F 46982,n1(CC(=O)N(C(C)C(=O)NC(c2ccsc2)C)CCC)cc(C#N)cn1 46983,c1(OC)cc(F)cc(C(=O)NCC(O)CNC(C2(C)CC(C)=NO2)=O)c1N 46984,c1(C(=O)NC2C(NC(CCc3c(OC)cccc3)=O)CC2)ccc(Cl)c(C)c1O 46985,N1(C(c2cc(OC)n(C)n2)=O)CC(NC(C2(CC#N)COC2)=O)CC12CCOC2 46986,CC(C(=O)N1CC(NC(=O)CNC(=O)Nc2ccccn2)C1)C(C)(C)C 46987,c1(N2CC(C(=C)C)OCC2)cccc(S(=O)(=O)NCC2CC23CCCCC3)n1 46988,C(CCCC(CO)NC(c1occ(C)c1C)=O)NC(c1c(CC)cccc1)=O 46989,N1(CC(=O)NCC(OC)NC(=O)C(C)OC2CCCC2)CCOCC1C1CCC1 46990,Cn1nc2c(cc1=O)CN(C(CC(C)(C)C)C(=O)NCCC#N)CC2 46991,c1(CNC(CCn2cc(C3CCN(C)C3)nn2)=O)ccc2c(n1)OCCO2 46992,C#Cc1ccnc(C(=O)NCC(O)CNC(=O)COCC2CCCCO2)c1 46993,c1(CC(=O)NC(C)(C)CCCNC(=O)C=CC2CCC2)c(F)cccc1C#N 46994,CC1CN(C(=O)CCCNC(c2cncs2)=O)CCN1Cc1ccccc1 46995,C1(CNC(N(c2ccc([N+](=O)[O-])cc2)CCC)=O)CC(C)(C)CCC1O 46996,C1(CC(=O)NCc2c(C(=O)OC)scc2)CCN(C(=O)C(c2cccnc2)O)C1 46997,CC1CCCC1C(=O)NCCOC1CCN(C(=O)C(c2ccc(Cl)s2)=O)C1 46998,c1(C(N2CC(CC)C(NC(=O)C#CC3CCOC3)C2)=O)cc(OC)c(C)c(OC)c1 46999,C1(NC(C2C(C(=O)OC)C2)=O)CCC(CC(=O)NC2CC(=O)N(C(C)C)C2)CC1 47000,C(=O)(C1Cc2c(Cl)cccc21)N1CC(S(N)(=O)=O)C(NC(=O)CC(F)(F)F)C1 47001,c1(CC)c[nH]nc1C(=O)N(CC(C)O)CCNC(c1cnn(CC2CCCC2)c1)=O 47002,C(C)(C)(CC(=O)NCC(C)(CNC(c1cc(C)n(C)c1)=O)OC)OC 47003,C1(NC(CC#N)=O)CCN(C(c2cnc3n2CCS3)=O)CC12CCC2 47004,c1(C(N2CC3CN(C(CN(C)CC)=O)CC3C2)=O)cc2c(F)ccc(F)c2[nH]1 47005,N#Cc1c(F)ccc(-c2cn3cc(C(N4CCOCC(O)C4)=O)ccc3n2)c1F 47006,CC1(NC(C2CC2(C)C)=O)CCN(C(c2cc(C3CCC3)on2)=O)C1 47007,c1(-c2cnc(OC)c(CN3CCC4CCCC34)c2)cc2cc[nH]c2cn1 47008,N1(C(C(=O)NCCC2(C)CC2)CC2CCC3CC23)CC2CCCCC12C 47009,C1(NC(c2cc(CC)on2)=O)CC(NC(C2(NC(C)C)CC2)=O)C12CCC2 47010,N1(C(c2cccc(C)n2)=O)CCC2C(NC(c3sccc3CN(C)C)=O)C2CC1 47011,C1(Nc2nccc(C)c2[N+](=O)[O-])CC(NC(c2cscc2Cl)=O)C12CCOCC2 47012,N1(C(Cn2c(C(C)C)nnn2)=O)CCC(C2(NC(C3CC(Cl)(Cl)C3)=O)CC2)CC1 47013,c1(C(N2CC(CC=C)(NC(C3CCNC3=O)=O)C2)=O)cc(OC)cc(Br)n1 47014,CC(C)CCC(C(=O)NC1CC(CCF)C1)NC(C1CC2(CCCO2)C1)=O 47015,C1(CC(=O)NC(COCC)C(=O)NCCC(=O)N(C)C2CC2)CC=CCN1C 47016,c1(C(=O)NCC2CC(C)N(C(c3cccc(CO)c3)=O)C2)ccc(Cl)c(C#N)c1 47017,c1(COC)cscc1C(=O)NCCCOCCNC(=O)CCCc1ccccc1 47018,c1(N2CCC(NC(C(CC)C)=O)C(F)C2)nc(C)nc(C)c1F 47019,c1(NC(C=CCOC)=O)c(F)cc(F)cc1Br 47020,C1(C(N2C(CNC(CC(CC)C3CC3)=O)CCC2)=O)(OC)CCCC(C)(C)C1 47021,CCC(COC)C(=O)NCCCC(=O)NC(C(N)=O)C(C)O 47022,Cn1c(C(=O)NCC2COCC2NC(=O)Cn2ccc(C(F)(F)F)n2)nnc1S 47023,N1(C(C2(c3n(C)ccn3)CC2)=O)CC(C)(C)c2cc(F)ccc21 47024,C(=O)(CC1=CCCC1)N1CCC(N(C(=O)COCCC=C)CC#C)C1 47025,c1(OC)ccc(C(C)C)cc1CN1CCOCC(NC(C2C3COCC23)=O)C1 47026,c1(C(C(=O)NCC2CC(NC(=O)CCC3CCCC3)C2)=O)cc(F)c(F)cc1F 47027,C(=O)(CN=c1cc[nH]cc1)N1C(C)C(NC(c2ccc(=O)oc2)=O)CCC1 47028,c1(C(=O)NCCOCCCNC(c2n(C)ccn2)=O)cc2c(cc1O)CCCC2 47029,C1(OCC)CN(C(N2CCCCC2C(=O)OC(C)(C)C)=O)CC1C(=O)OC 47030,c1(C(=O)NC2CC(CNC(C(COCC)(C)C)=O)C2)ccnc(O)c1Br 47031,CCCCCCCC(O)CC(=O)N1CCNC(C(=O)NC2(CC#N)CCCC2)C1 47032,CCC(CC)CC(=O)NC1(CNC(=O)C(O)CC)CCC1 47033,c1(C(C(=O)NCC2CC2)N(CC(C)Cn2cccn2)CC)cccc2c1OCO2 47034,C12(CNC(c3c(CSC)cccn3)=O)CCC(CC1)N2C(C1C=CCC1)=O 47035,c1(OC)ccc(F)cc1C(=O)NCCC(C(C)C)N(C)C 47036,C1(C)(CC)CC(NC(=O)CC2(OC)CCOCC2)CN1C(=O)CC1CN(C)C1 47037,CC(CC(=O)NCC1(C)CCCN1C(=O)Cc1cncn1C)CC(F)(F)F 47038,N1(C(C2(C#C)CN(C(=O)CC(C)(C)OC)C2)=O)CCC2C(CCN2C)C1 47039,CCC(CC(C)C)C(=O)N1CC(C(=O)Nn2ccnn2)C(C)(C)C1 47040,C1(NC(CCCC)=O)CC2CCC(C1F)N2C(c1ccc2c(c1)CCN2)=O 47041,C(=O)(C1=CC2(CCNC2)C1)N1CCC(C(=O)N(c2ccccc2)CC2CC2)CC1 47042,C12(CNC(C(C)CN(C)C)=O)CC(CCO1)N(C(=O)C(CO)C(F)(F)F)C2 47043,c1(CC)ccc(CNC(N2CC(N(C)C)C2)=O)cc1F 47044,N1(C(Cc2cn(C)nc2)=O)CCC(O)(C(=O)NCCN2C(=O)CSC2=S)C1 47045,c1(C(N2C(C(C)NC(C3(C)CC(C)C3)=O)CCC2)=O)cn2ccccc2n1 47046,N1(C(CN(C(=O)C(=Cc2c[nH]cn2)F)C)=O)CCN(C(c2n[nH]cc2Cl)=O)CC1 47047,c1(OC)cc(C(N2CCC(C)(NC(=O)CC3CCC3(C)C)C2)=O)ccc1F 47048,OC1CC(NC(Cc2csc(Br)c2)C(=O)O)(Oc2ccccc2)C1 47049,C=CC1(c2cn(CCCCO)nn2)COCCN1C(C1(CC(C)C)CCCC1)=O 47050,C1(NC(C(C)Cc2ccccn2)=O)CN(C(c2ccc(F)c(I)c2)=O)CC12CC2 47051,c12sc(cc1C)N(CCCN)NCC(C)CN(C)C2=O.CC 47052,C1(NC(c2ccc(Cl)nn2)C)CCCN(c2ccccc2)C1 47053,C1(NC(C2CC2(F)F)=O)CCC2CN(C(C3(CF)CC3)=O)CCC2C1 47054,c1(OC)ccc(CC(N2CC(CNC(C3(C)CC3)=O)C(F)(F)C2)=O)cc1Cl 47055,C(CNC(C1CN(C)C(=O)N1)=O)(CC(=O)NC1(CO)CC(C)C1)OC 47056,N1(C(C2CCN(CC)C2)=O)CCC(N(C)C(c2ccn3nccc3n2)=O)C2(CC2)C1 47057,[N-]=[N+]=NCCCCCC(=O)NC1CCC(NC(=O)NCCOC2CCCOC2)CC1 47058,CC1(C)CCC(C(=O)NCCCC2CN(C(c3cccnc3O)=O)CCO2)CC1 47059,CCC(C(=O)N1CCC(NC(c2cc([N+](=O)[O-])ccc2O)=O)C1)C(C)(C)CC 47060,C1(O)(CNC(C2(C#C)CC2)=O)CCCN(C(=O)C(C)NC(c2ccoc2)=O)CC1 47061,C(CC1c2ccccc2CCN1C(=O)C(O)C(C)C)NC(C(Br)=C(C)C)=O 47062,C(=O)(CCCC(=O)NC(C)CCSC(C)C)NC1C(c2nc(C)[nH]n2)C1(C)C 47063,CCC(C)(CCC(C)C)C(=O)NC1COCC1NC(c1cncc2nc[nH]c12)=O 47064,CC(O)CCCCCC(=O)OCC1CCCCN(c2ccc(Br)cc2)C1=O 47065,C=C(C)CCCC(=O)N(C1CCN(C(=O)C(c2ccccc2)F)CC1)CC 47066,CC(C)(C(=O)N1CCC(Nc2ccccc2C(F)(F)F)CC1)S(C)(=N)=O 47067,c1cnn2c1CCCC2.Oc1cccc(-c2cccc(NC3CC3)n2)c1F 47068,CC1=C(C(=O)N2CCN(C(c3cscn3)=O)C(CO)C2)CCS1(=O)=O 47069,S(=O)(=O)(c1cn(C)c(C)n1)NCC(N1CC2(C(NC(C=NOC)=O)CC2)C1)=O 47070,Cc1c(C(=O)NC(C)(C)C(C)NC(=O)C(C)CC(F)F)nn(C)c1N 47071,N1(C(C(C=C)(C)O)=O)CCC2(CC1)CC(NC(c1c(C)cc(C)nc1C)=O)C2 47072,C(CCCCC(=O)N1CCCC1C(C)(C)O)N(C(C(C)CC1CCC1)=O)C 47073,CC1COC2(C1)CN(C(C1CCCN1C(C1CC(CF)C1)=O)=O)C2 47074,N1(C(C2(NC(c3ccnc(C)c3N)=O)CCCCC2)=O)CC(C)C12CCOCC2 47075,c1(CC(=O)NCC2(C)CCN(C(C3(C#N)CCCOC3)=O)C2)cc(F)ccc1F 47076,CC1(C(=O)NC2CC(C)(NC(=O)C3=CCCOC3)C2)CCC2CC2C1 47077,C1(NC(CNC(c2cccc3ccccc23)COC)=O)CNc2ccccc2O1 47078,c1(OC)cc(C)sc1C(=O)NC(C1CN(C(=O)CCCC2CCCC(=O)N2)C1)C 47079,C(=O)(CCCCCNC(=O)CC1CC(F)CN1C(c1cc(O)nc(Cl)c1)=O)OC 47080,c1(OC)c(C(=O)NCC(C)NC(c2cnc(Cl)s2)=O)csc1Cl 47081,c1(SC)c(C(=O)NC2COCC2CNC(C2Cc3cscc3C2)=O)cccc1F 47082,C(=O)(C(C#N)C(C)(C)C)N1CCC(C(=O)NC(CSCC)CO)(OC)C1 47083,C1(C(=O)NC2CC2)(CNC(C(C)NC(=O)CCOC2CC2)=O)CC=CC1 47084,C(c1ccc(F)cc1F)=CC(=O)NCC1(OC)CCN(C(C2COC(=O)N2)=O)C1 47085,C(=O)(CC(O)c1ccccc1)N(CCCNC(=O)COC1CCC1)C(C)C 47086,C1(NC(c2ccc(OC)nc2)=O)CCC(C)N(C(=O)CCOC)C1 47087,S(=O)(=O)(c1ccc2nc(C)oc2c1)N(C1C(CC)CCCCC1)C1CC2CNC1C2 47088,C(=O)(C(O)C(F)(F)F)N1CCC(C)(CCNC(c2ccc(C#C)o2)=O)C1 47089,C(CN=c1[nH]c(=NCc2cnc(O)[nH]2)c2sccc2[nH]1)C1C(C)C1 47090,C(C(=O)N1CCCc2nccn21)C1CC1.CC1(C)CC1CC(=O)N 47091,c1(-n2cc(CN(C(CNC(C3C(C)(CC)C3)=O)C)C)nn2)cccc(C)c1Br 47092,C(=O)(CC(CCCC(C)C)NC(c1cc(Cl)cc(Cl)c1OC)C(=O)OC)OCC 47093,C1(C(=O)O)CC=CCN1C(C)=O.C(=O)(C(C)N=[N+]=[N-])NCC(N1CC(OC)C1)=O 47094,C1(NC(c2n(CC)ncc2)=O)CC12CC(NC(=O)C(O)C(C)C)C2 47095,Cc1csc(=NCC(=O)N2CC3C(CNC(=O)CSC4CCCCO4)C3C2)[nH]1 47096,C1(NC(c2ccc(CC)[nH]2)=O)CCN(C(c2cc(C(C)(C)C)oc2C)=O)CC1F 47097,c1(N(c2cc(C3CC3)no2)C)ccc(COC)cc1.C1(CC(=O)O)CCCCCC1 47098,N1(C(CC(=O)OC)=O)CC2CC1C2NC(c1nscc1Br)=O 47099,C1(C(N(C(C)C(N)=O)CCOC)=O)C2CCC1(c1cccnc1)C2 47100,N1(C(Cc2ccn(CC)n2)=O)CC2(CCC(CNC(=O)CCn3cccn3)O2)C1 47101,CS(=O)(=O)c1cccc(CN2CC(C(=O)Nc3ccc(F)cc3F)CC(F)C2)n1 47102,C#Cc1cnc(NCC(CNC(c2ccccc2C)=O)Cl)nc1 47103,c1(OCc2onc(-c3ccc(OC)cc3)n2)ccc(C(C)=O)c(F)c1Br 47104,C(C1=CCN(C(c2ccnc(C(N)=O)c2)=O)CC1)NC(C(CC)NC(N)=O)=O 47105,C(C(C)C(F)C(=O)Nc1cccc(Cl)c1)NC(c1c(OC)nn(C)c1)=O 47106,Cc1ccnc(C(=O)NCC(C2CCCC2)NC(c2conc2C(C)C)=O)c1N 47107,C(CCC(O)C(=O)NC(C)C(O)C(F)F)NC(COCC)=O 47108,C1(C(=O)NCCC(CCNC(c2ccc(C(C)=O)o2)=O)C)CC2(CCCO2)C1 47109,N1(C(COCCN=[N+]=[N-])=O)CCC2(CC1)CC2NC(C1CN2CCC1CC2)=O 47110,Cc1cc(C(N2CC(CCO)(NC(=O)C(C)SC(F)(F)F)C2)=O)cnc1C 47111,C(C(C)CC(C)C)NC(C(CC1CCOCC1)NC(CCC)=O)=O 47112,C1(C(=O)NC2C=CCC2)(NC(C2CCCSC2)=O)CCOCC1 47113,c1(C(=O)NCC2CCC(NC(C3N(CCC)CCC3)=O)C2)c(C)ccc(F)c1N 47114,C1(CC(=O)N(c2ccccc2)C2(C(C3CC3)C3CC3)CC2)CCN(CCCF)C1 47115,CCCCCCCCC(C)CC(=O)NC1CCC1(C)C 47116,n1(C(C)CC(=O)NC2CCOCC2NC(=O)C2=CSCS2)cnc2ccccc12 47117,C(=O)(C(C)P(C)(C)=O)N1CCC(N(C(CC(C)OC)=O)Cc2ccccc2)CC1 47118,c1(C(=O)NCC2(O)CC(CNC(C=C(CC)C)=O)C2)cc(C)c(CO)cn1 47119,C1(CC(N2CCC(N(C(c3cn(CC)nc3C)=O)CC)C2)=O)CC2C=CC1CC2 47120,N(C)(S(=O)(=O)N(C)C)CC(N1C(CN(C(c2ncn(C(C)C)n2)=O)C)CCC1)=O 47121,Cc1cccc(-c2nnc(C(N3CCC3CNC(=O)CC3CCCCO3)C)o2)c1 47122,c1(N(CCNC(CCC(C)(C)F)=O)CC#N)ncc(Br)cc1C#N 47123,CC(C)CCCC(=O)NCC(CC(=O)N1C(CO)CC1C)C1CCC1 47124,C(=O)(CC(O)CC1CCNCC1)NC(C(c1ccccc1)OCCC(C)C)=O 47125,Cc1cc(C(N2CC=CC2CNC(=O)C(c2cccc(Cl)c2)C)=O)ccn1 47126,N1(CC2CCOC(C(C)C)C2)CCCN(C(=O)C(=O)NCC(NOCC)=O)CC1 47127,CCC1=NOC(C(=O)NC2CC(NC(C3(CC(=O)NC)CCCC3)=O)C2)C1 47128,c1(C(=O)C(N2CC3(CCCO3)C2C2CC2)=O)c[nH]c2ccc(F)cc12 47129,N1(C(c2c(C)nc[nH]2)=O)CCC(C)N(C(c2ncnc(C)c2C)=O)CC1 47130,Cc1ncc(C(N2CC(C(=O)NC3(C(F)F)CCC3)C3(CC3)C2)=O)cc1C#N 47131,C1(CNC(c2c(C)nc(O)[nH]2)=O)CC2CCCCC2N1C(C1CCSC1)=O 47132,C1(C(=O)NC2CCCCN(C(c3ccc(Cl)cc3O)=O)C2)CC2CCCCCC12 47133,C(c1ccnn1C)=CC(=O)NCCN(C(c1cc(C2CCCCC2)n[nH]1)=O)CC 47134,CC1CCN(C(C2(N3CCCC3)CC2)=O)CC1CSCC(=O)NS(=O)(=O)C1CC1 47135,C(C1=NOC2CN(C(=O)C(C)(C)C3CCC3)CC12)NC(c1cc(C)nnc1O)=O 47136,c1(C(N2C(C)CC(NC(C3(C)CC(=C)C3)=O)C2)=O)cn2cccc(F)c2n1 47137,N1(CC(=O)NC2CCC(CO)O2)CCCC2(CC2)S1(=O)=O 47138,C1(C)(CNC(c2occ(C)c2)=O)CCN(C(c2ccc(OCCF)cc2)=O)C1 47139,C#CC1(C(=O)NCC(COC)NC(=O)C(CCSC)OC)CCCC1 47140,C1(C(=O)NCC2C3CN(C(Cn4nnc(C)n4)=O)CC32)CCN2CCOCC12 47141,c1(C(NNC(c2c(C)scn2)=O)=O)cc(Cl)cnc1F 47142,C(=O)C(O)C(F)(F)F.O=C(NOCC1(F)CCC1)C(F)C1CCOC1 47143,CC1CC(C#N)(C(=O)NC2CC(NC(C3(Cl)CC3(F)F)=O)C2)C1 47144,N1(C(C(=O)N(C)C)=O)CC(O)C(C2CC2)C1 47145,CCC(C(=O)NCC(C)(C)Cn1cc(-c2cccc(F)c2C)nn1)C(C)O 47146,c1(OCCCOC)ccc(C(=O)N(CC(C)NC(c2ncccc2O)=O)CC)cn1 47147,N1(C(c2cn(CC=C)nc2)=O)CCC(NC(=O)C(F)C(C)(C)O)CC1C 47148,N1(C(c2nncc(OC)c2)=O)CCC(N(C)C(C2SCCS2)=O)C(C)C1 47149,C1(C(N2CC(CCOC)N(C(=O)CC(C)(C)OC)CC2)=O)CCCC2(CCC2)O1 47150,N1(C(C(C)(C)NC(=O)OC)=O)CCC(NC(=O)C(C)(C)C)C(O)C1 47151,C1(CC(=O)NC2CC(CNC(CCCNC(C)=O)=O)C2)COCC(C)(C)O1 47152,N1(C(c2ccc(F)c(C)c2O)=O)CC2(C1)CN(C(=O)CCCF)CC2CO 47153,C(CN=c1[nH]c(=NC)[nH]c(=NCC=C2CCOCC2)[nH]1)c1nc(OCC)sc1 47154,N1(C(CC2(NC(C)=O)CC2)=O)CCOC(C(C)NC(c2cc(Cl)cnn2)=O)C1 47155,c1(OC)cccc(=NC(=O)CN2CCN(c3cc(Br)c(C)cc3F)CC2)[nH]1 47156,c1(OC)ccc(OC)c(CC(C)C(=O)OCC(C)(O)COCc2ccccc2)c1 47157,N1(C(C2CCN(C)CC2)=O)CC2(CNC(=O)COCC3CCCO3)CC1CO2 47158,n1(C(CC)C)ncc2cc(C(=O)NCC3CCN3C(c3ccncc3)=O)cnc12 47159,CC1CCN(C(c2cc(Cl)cs2)=O)C1C(=O)N(C1CC=CC1)C 47160,CCCCCCCC(=O)N1CCCC1CNC(c1c(Br)c(C)nn1C)=O 47161,C1(C(N(CC(O)CNC(C2CC23CCCCC3)=O)C)=O)CCC(=C(F)F)CC1 47162,C1(CC=C)(NC(C2CC2(F)F)=O)CC2CCC(C1)N2C(=O)Cc1c(C)noc1Cl 47163,C1(NC(CSCC)=O)CCC2(CC1)CCN(C(c1n[nH]c3cccnc13)=O)C2 47164,C(C(O)C(F)(F)F)N(C(C(C)N(C(=O)CC1(NC(=O)COC)CC1)CC)=O)C 47165,c1(CCC(=O)NC2CC(C)N(C(=O)CC#N)C2)cc(F)ccc1Br 47166,N1(C(C2CCN(C)C2)=O)CC=CC(C(N2CCN(CC(N)=O)CC2)=O)C1 47167,C1(C(N(CC#C)CC#C)=O)CC2CC2N1C(C1CC=C(C)CC1)=O 47168,N1(C(CC2(CNC(C3CCN(C)CC3)=O)CC2)=O)CCCC(F)CC1 47169,C(=O)(C1=NOC(CNC(=O)C=C2CCOCC2)C1)N1C(CC(C)C)CCCC1 47170,N1(C(CCC(=C)C)=O)CCC(C2CC2)(CNC(=O)CC2C(C)(C)C2(C)C)C1 47171,N1(C(c2cnc(C)nc2)=O)CC2CC(C)N(C(C3CCCOC3)=O)C2C1 47172,c1(C(=O)NCCCN(C(C2(CC)CC(C)(C)C2)=O)C)ccc(C(F)F)c(F)c1 47173,N1(C(c2ccn(CC)n2)=O)CCC2(CCN(Cc3c(C)cccc3C)CC2)C1 47174,c1(CCC)cc(C(=O)N(CC(C)CNC(=O)CC(CC)C2CCC2)C)ccn1 47175,Cn1ncc(C(=O)NC2CCCCC2C(=O)NOCc2ncccn2)c1Cl 47176,c1(C(C)C)nnc(SCCCCN2CCOCC2)n1-c1ccc(F)cc1 47177,C1(C(=O)NCc2cc(OC)c(Br)cc2)CC(c2ccccc2F)=NO1 47178,c1(C(=O)NCC2(O)CC(C(=O)NCC(C3CC3)OC)C2)cc(C)oc1C 47179,c1(SC)nsc(N2CC(OCCNC(=O)C(C3(O)CCCC3)F)C2)n1 47180,N1(C(C(CC)O)=O)CC(C(=O)N(C2CCCCC2O)C)C(F)C1 47181,c1(C(=O)OC)coc(C=CC(=O)NCC2CC(NC(C3CCCCC3F)=O)C2)c1 47182,C1(CN(C(=O)CC2(CO)CCC2)CC)CCCN1C(=O)CSc1n[nH]c(O)n1 47183,C1(NC(CS(CCC)(=O)=O)=O)CCC2CCN(C(c3ccc(O)cc3Cl)=O)C1C2 47184,c1(OC)ccc(C(=O)NC2CN(C(=O)CC)C2)c(F)c1Cl.C1(OC)CCOCC1 47185,C1(n2cc(CC(C)(C)CO)nn2)CCC(NC(c2cc(F)n[nH]2)=O)CC1 47186,c1(C(N(CCCCN(C)C(c2csc(-c3cn[nH]c3)n2)=O)C)=O)cncc(F)c1 47187,C1(C(=O)NCC(C)(C2CC2)NC(c2c(C)nncc2)=O)CCCC1C1CC1 47188,CCN=c1[nH]cc(C(=O)N(CCCNC(C2CC2[N+](=O)[O-])=O)C)s1 47189,C1(N(C(CCOc2cccc(C)c2)=O)C)CN(C(c2csc(=N)[nH]2)=O)CC12CC2 47190,CC(C)(C#N)CC(=O)NC1CC(NC(C2CCC=CCC2)=O)C(O)C1 47191,c1(OC(C)C(=O)NC23CC2CN(C(C2(C#N)CC2)=O)C3)cccc(C(C)(C)C)c1 47192,C1(N(C2CC2)Cc2cnc(C)n2-c2ccccc2)CC(C)CC(C)C1 47193,c1(OCC)ccc(-c2cccc(C3(C(=O)N(CCO)C4CC4)CC3)c2)c(F)c1F 47194,C1(CC)(CC)CC(NC(C2CCCOCC2)=O)CN1C(c1ccc(OC)cn1)=O 47195,N1(C(C(C)NC(C2CCC2)=O)=O)CCCC(O)(CNC(=O)Cn2nccn2)C1 47196,c1(OC)ccnc(O)c1C(N1CC(NC(=O)Cc2cnsc2)C(C)C1)=O 47197,Cc1cc(C(N2CCN(C(C3CCCO3)=O)CC2)C(=O)NC2COC2)cc(F)c1 47198,C1(S(C)(=O)=O)(CNC(=NCCSC)NCc2c(Br)cnn2C)CCC1 47199,N(C1CC(C)(C)c2ccccc21)Cc1c(Br)cc(OC)c(OC)c1O 47200,c1(C(=O)NCCCN(C(=O)CNS(=O)(=O)N(C)C)CC)cc(S(C)(=O)=O)cs1 47201,C(=O)(C(C(C)(C)O)NC(c1ncncc1N)=O)N1CC(C)SCC1 47202,Cc1nn(C)c(Br)c1C(=O)NCC(c1ccccc1)NC(C1CC2CC2C1)=O 47203,C1(C)(CNC(C(=C(C)C2CC2)F)=O)CN(C(c2cc(=O)cc[nH]2)=O)C(C)(C)C1 47204,n1(CCCNC(C2CC3(CC3)C2)=O)cc(C2C3COCC23)nn1 47205,c1(C(c2nnnn2CC2CCOC2)NCc2cc(C)no2)cc(C)oc1C.C1CC1 47206,c1(C(CO)NC(c2cn(CC(=O)OC)nn2)=O)cncc(F)c1 47207,CCCC(C(=O)N1CC(=O)CC1C(=O)N(C)CCc1cnccn1)OC 47208,c1(C(N2CCC(O)(CNC(c3cnn(C(F)F)c3)=O)C2)=O)noc2ncccc12 47209,c1(C(=O)NC(C2CCOC2)CC)cn(CCNC(=O)C(C)SC)nn1 47210,c1(OCC)ccc(C(=O)NC(c2ccccc2)(C)CNC(C2CCCO2)=O)cn1 47211,c1(CNC(CC2C3CN(C(C(n4ccc(C)n4)C)=O)CC32)=O)ccc(F)cc1F 47212,CN1CCC(O)(CC(N2CCC(NC(=O)C(F)(F)C3(O)CCC3)C(O)C2)=O)CC1 47213,Cc1ccc(CC(N2CCC(C)(C(=O)N(C)Cc3nncn3C)C2)=O)cc1 47214,C12(CNC(=O)Cn3ncc(Br)n3)CC1CN(C(=O)CCOc1ccccc1)C2 47215,C1(N(CCCC)C(c2cc(OC)cs2)=O)CCN(C(c2n[nH]cc2Cl)=O)CC1 47216,C#CC1(CNC(C2CN(C(c3nonc3N)=O)CCO2)=O)CCCC1 47217,Cc1ccc(C(F)F)cc1OCC(N1CCSCC1NC(=O)OCCO)=O 47218,N1(C(C(C)Oc2cccnc2)=O)CCC(F)(F)C(Nc2ncc3c(n2)CCC3)C1 47219,C=C(C)CC(C(=O)NC1CCCCC1N=[N+]=[N-])NC(=O)C(C1CCOCC1)F 47220,c1(OC)noc(C2CC2)c1C(=O)NCC1(NC(C2(C#N)CC2C)=O)CC1 47221,CN1C(=O)Cc2c(-c3nc(CCCCN(C)C)nn3CC(F)(F)F)cccc21 47222,N1(C(C(C)CC2CCCCC2)=O)CCC(CF)(NC(=O)CCSCC(N)=O)C1 47223,C1(O)(CCNC(Cc2n(C)cnc2)=O)CCN(C(c2cnn(CCF)c2)=O)CC1 47224,C12(C(N(C(C3CCCCC3)C)C)=O)CC(CO1)N(C(c1ccc(Cl)cn1)=O)C2 47225,N1(CC(=O)NCc2ccnnc2NCC(F)F)CCc2ccccc21 47226,N1(CC(=O)N(CCNC(=O)CCc2ncc[nH]2)CC)CCc2sccc2C1 47227,C=C(C)c1cccc(NC(C2CC(=O)CN2C(=O)C(C(C)(C)C)OC)=O)c1 47228,c1(OC)ncc(C)c(C(=O)NC2CC(C)N(C(c3cccc[n+]3[O-])=O)C2)c1Cl 47229,c1(-c2ccc(CNS(CC=C)(=O)=O)cn2)ccc(OC(C)C)c(F)c1F 47230,Cc1c(C(=O)NCC(C)CNC(=O)C2=CCCC2C)c(O)nc2ccccc12 47231,CC1(NC(c2coc(Br)c2)=O)CCN(C(c2ccc(C3(C)CCO3)cc2)=O)C1 47232,N1(C(c2c(C)ncs2)=O)CC(C)(CNC(=O)CC2CCCC(=O)N2)CC1(C)C 47233,c1(C(=O)NC2CC(CNC(C3(CC)CC3)=O)C2)cc(Br)co1 47234,C12(C(N3C(C)CC(NC(C(C)=C4CCC4)=O)C3)=O)CCC(F)(CC1)CC2 47235,CC(C)CC(C)(CNC(=O)Cc1cccc(O)c1)NC(c1ccn(C2CC2)n1)=O 47236,N1(C(C(C2CCCO2)NC(C2CCS(=O)CC2)=O)=O)C2CCCC1COC2 47237,CC(C)(C)CC(=O)N1CCC(C(=O)NOCC2(C)CC2)CC1 47238,C=C=CCC(=O)NCC1COCC1NC(=O)CCc1cc(OC)no1 47239,c1(N(CC(C)NC(Cc2nc(C)sc2C)=O)C)nc(Cl)ncc1Cl 47240,Cc1cc(-n2ccnc2)ccc1C(=O)N(CCNC(=O)C(F)C(F)(F)F)C(C)C 47241,C1(NC(c2ccn(-c3ccc(Cl)c(F)c3)n2)=O)CCCCCC1c1ccccc1 47242,c1(C(N(CC(CNC(c2c(CC)cno2)=O)C)C)=O)ccccc1C1CC1(F)F 47243,Cc1cc(=NCC2(CCCO)CCCC2)[nH]c(NC(c2cccnc2)C)n1 47244,CN1CCC(n2cc(C3(C)CN(C(=O)C(F)C4CCOC4)C3)nn2)C1=O 47245,CC(CNC(=O)Nc1nccnc1Oc1cccnc1)(CO)CO 47246,C1(CC(=O)N(C2CCN(C(c3ncsc3C)=O)C2)CC)CCCC2CC12 47247,N1(C(C2=NNC(=O)C2)=O)CCC2(CC1)CN(C(c1cncc(F)c1)=O)CCC2O 47248,c1(OC)ccc(F)c2[nH]c(C(=O)NCC(C)(CO)NC(=O)C(O)CN(C)C)cc12 47249,c1(C(N(C(CNC(C2(CCC)CCC2)=O)C2CC2)C)=O)cn(C2CCCC2)nn1 47250,c1(N(CC(=C)C)C)cccc(S(=O)(=O)NC2CCCC(c3ccc(F)cc3)C2)n1 47251,C1(C)(CNC(c2c(CC)con2)=O)CN(C(=O)CC(C(F)(F)F)OC)C(C)(C)C1 47252,C1(NC(c2cc(C(C)C)[nH]n2)=O)CCN(C(c2cn(C)ccc2=O)=O)C1(C)C 47253,C1(C(=O)NCc2nc(C)c(C)s2)CC2(CCN1C(=O)CC1CCC(=O)C1)CC2 47254,c1(CC)cc(C(=O)NC(C2CCN(C(=O)COC(C)C)C2)(C)C)c(C)o1 47255,C1(C)(CNC(C(C)NC(C)(C)C)=O)CCN(C(=O)CC23CCCC2C3)CC1 47256,N1(C(=O)Cc2nc[nH]n2)CCOC2(CCN(C(C3CC4CCC3O4)=O)C2)C1 47257,CC(C)C(CN(C)C)N=c1nc(N2CC3CCC3C2)c2c([nH]1)CCS2 47258,Cc1nc(Cl)[nH]c(=NC2CC(NC(=O)CC3(CO)CC3)CC23CCOCC3)c1Cl 47259,Cn1nc(C(N2CCC(C)(NC(C3COC(C)(C)C3)=O)CC2)=O)c(Cl)c1Cl 47260,CC(CC(C(=O)N1Cc2cncnc2C(C)(C)C1)Nc1ccccc1)CC(C)(C)C 47261,C1(C(=O)NCCC(=C)CNC(c2csc(C)n2)=O)CC(=O)N(C2CCCCC2)C1 47262,C1(OC)CN(C(C2CC(C#N)C2)=O)CC1NC(C1(c2ccccc2F)CCC1)=O 47263,c1(CN2C(C)CN(C(c3cccc(C#N)c3)=O)CC2)csc2ccc(Br)cc12 47264,Cc1cnc(NC(C2CSCCN2Cc2c(C)cccc2Br)=O)c(Cl)c1 47265,c1(C(=O)OCC)cc2n(n1)CC(C)N(C(c1cc3occc3[nH]1)=O)C2 47266,C(C(CC1CCCC1)C(=O)N=c1ccn(C2CC2)[nH]1)NC(c1c(C)cnn1C)=O 47267,C(=O)(CC(C(F)F)NC(c1n[nH]c(O)n1)=O)NCCC(CC)(C)C 47268,Cc1cc(NC(=O)NCC2CCCC(C)C2)n(CCOc2ccccc2)n1 47269,C1(C)(C(N2CCC(=CCNC(COCCCCC)=O)CC2)=O)CCC(=O)NC1 47270,CCC(C(C)O)NC(c1ccoc1CNC(=O)COCC(C)C)=O 47271,C1(NC(c2sc(CC)c(C)c2)=O)CN(C(=O)C(F)(F)C(C)O)CC1C1CC1 47272,Cc1c(CNC(=O)NCC2(F)CCCCC2)cccc1F 47273,CS(=O)c1cccc(NC(c2noc(-c3ccccc3)n2)c2nnnn2CCl)c1 47274,C=CC1(C2(C(=O)NCCCCN(C(=O)CSc3cccs3)C)CCC2)CCC1 47275,C(c1ccc(F)cc1)=C(C)C(=O)N(C)CCN(c1cc(Cl)nc(CS(C)(=O)=O)n1)C 47276,CC1CC(NC(c2cncc(O)c2Cl)=O)CCN1C(c1ccc(F)cc1Cl)=O 47277,Cc1[nH]c(C#N)cc1C(N1CC(CC(N2CC3(CCC3)C2)=O)C(C)C1)=O 47278,N1(C(c2c(C)ncnc2)=O)CCC(F)(C(=O)N(CCCC(O)CO)C)CC1 47279,c1(OC(C(N2CCC(C)CC2)C)=O)ccc2ccccc2c1 47280,c1(NC(C2ON=C(C)C2)=O)ccc(NC(=O)CN2C(=O)CCCC2=O)cc1C 47281,C#CCCCCCCC(=O)N1CCN(C(=O)CCCSC)C2CC12 47282,N1(C(C2(C=C)CCN(C(=O)CCOC(C)C)C2)=O)CCC2(CC=CCO2)C1 47283,C(CC(O)C(=O)NCCCCC(C)NC(c1ccc(NC=O)cc1)=O)SC 47284,N1(C(c2c(C)nc(C(C)C)cc2)=O)CCC2(NC(=O)CN(C)CCO)CCCC12 47285,Cc1nn(C)c(C)c1S(=O)(=O)NCCC(=O)NCC(C)(C)NC(C1CC1C#N)=O 47286,c1(OC)ccc(NC(=O)C(C)OCCN(C)C)cc1.C12(COC1)N(C1CC1)C2 47287,c1(C(=O)NCCCC(C)NC(CC2C(OC)COCC2)=O)nc2cnccc2s1 47288,c1(C(N(C(c2ccccc2)CNC(C2CNC(=O)C2)=O)C)=O)cc2cccnn2n1 47289,C1(SCCNC2CC(c3ccccc3F)(C(=O)OC)C2)CC2CCC1C2 47290,C1(C2(C(=O)OCC)CCC2)CCCN1C(C1COCCO1)=O 47291,CC(C(=O)OC1C2CCOC2C12CCCC2)N1C(=O)COc2ccccc21 47292,Cn1cnc2c1CCCC2C(=O)NCC1(F)CN(C(=O)CCC2CCOC2)C1 47293,C1(C)(NC(C2(C#C)CCC2)=O)CCN(C(=O)CNC(=O)CNC(C)=O)C1 47294,Cc1cc(CC(N2CC(O)CC2CC(N2CCC(C)(N(C)CCO)C2)=O)=O)nn1C 47295,C=Cc1cnn(C)c1C(N1CCC1CNC(c1cnccc1N1CCCC1)=O)=O 47296,c1(C(=O)NCC2CCCN(C(C(C3CCC3)OC)=O)CC2)nc2ccccn2n1 47297,C1(C(N(CCC)CC)=O)CCCN(C2CCCCC2OC)CC1 47298,N1(C(C(CCSC)(C)C)=O)CC2CC(C1)CN(C(C1CC3CC(=O)C1C3)=O)C2 47299,C1(NC(=O)C=CC2CCOC2)CC2(C1)CC2C(=O)NC1CCOC1 47300,C(CC(O)CC(=O)NC1CCC(N(C(=O)C(C)n2cncn2)C)CC1)SC 47301,N1(C(Cc2c(C)n[nH]c2)=O)CCC(O)(C(C)NC(c2ccc([N+](=O)[O-])o2)=O)CC1 47302,c1(Cn2cc(CSC)nn2)cccc(C(=O)NC(C2CCOCC2)C)c1 47303,N1(CCn2c(C)cc(C)n2)CCCC(NC(=O)CCN2CCCCC2=O)CC1 47304,C1(CC(=O)N(C2(C#C)CC2)C)CC(O)CN1C(=O)CN1CCCC1 47305,c1(C(C)=O)cc(C(=O)NCC23CC(NC(c4cnccc4Cl)=O)(CO2)C3)n(C)c1 47306,N1(C(c2n(C)c(S)nc2)=O)CC2CN(C(c3coc(C(F)(F)F)n3)=O)CC2(C)C1 47307,C1(C(N(CCCNC(=O)CSCc2ccncc2)C)=O)CCC(=O)N2CCCC12 47308,C1(C(N2CC(CC)NC(=O)C2)=O)C2CCCC2CN1C(c1cn(C)nn1)=O 47309,C1(NC(=O)C=CCNC(=O)CC2CC=CCC2)CCC(C2CC2)O1 47310,CCC(N)CCC(=O)N1CCC12CN(Cc1ccccc1)C2 47311,C1(NC(CNC(=O)CC(F)(F)F)=O)CCN(C(=O)CSc2n[nH]c(O)n2)CC1O 47312,c1(CC(=O)NCC(CCOC)NC(=O)Cc2c(Cl)cnn2C)ccc(F)cn1 47313,C(=O)(C(F)C(F)(F)C(F)(F)F)N1CCC2CCC(NC(C3CC(C)(C)C3)=O)C1C2 47314,C1(C(N(C)Cc2cccnc2)=O)CN(C(C23C=CC(CC2)C3)=O)CC1(C)C 47315,c1(OCC)ncc(C(=O)NCCC2(NC(=O)C(C)(F)F)CCCC2)s1 47316,N1(C(CNC(C(=O)NC(c2ccc(I)cc2)CC)=O)(C)C)CCC(C)CC1 47317,C1(CN(C(=O)C(F)OC(F)(F)F)CC)CCCCN1C(=O)CCn1ccnc1C 47318,CC12CC(C1)C(C(=O)NC13CC(CNC(c4cncc(CO)c4)=O)(C1)C3)CO2 47319,N1(CCNC(C(C)(C)C2CCC2)=O)CCN(C(=O)C(C)(C)C2(C)CC2(F)F)CC1 47320,C1(NC(N2CC(NC(c3c(C)ocn3)=O)C2)=O)CN(Cc2ccccc2)CCN1C 47321,c1(NC(C(N2CC(OC)C(NC(=O)CO)C2)=O)C)ccccc1[N+](=O)[O-].C(C)(C)S 47322,CCCCC(O)C(C)C(=O)N1CC2CCC(C1)N2C(c1cnn(CC)c1)=O 47323,O=C(N1CC(O)C(O)CO1)C1CC2CC1CN(C(C13C=CC(CC1)C3)=O)C2 47324,c1(NC(COC2(C)CN(C(c3cc(CCC)[nH]n3)=O)C2)=O)cncnc1O 47325,c1(C(c2nnnn2C2(C)CC2)NCCC(=O)NCC)cc(C)ccc1Cl 47326,C=CCCC(C(=O)NOCCF)NC(C1CC=CCO1)=O 47327,C(=O)(CC(C)(C)C(F)(F)F)NCC1N(C(C(C(=O)OC)OC)=O)CC2(CC2)C1 47328,S(=O)(=O)(C(Cl)(Cl)Cl)C1C(C(N(CCC#C)CCC#N)=O)C1 47329,N1(C(Cc2c(C)nn(C)c2)=O)CCC(C)C(CC(N2CCC(SCO)CC2)=O)C1 47330,N1(C(COCC=C)=O)CC2CC(C(=O)NCCOCCC3CC3)C(C2)C1 47331,CCCCC(C)CCC(=O)NCC12CCC(CC1)N2C(=O)C(C)(C)C(=O)OC 47332,C12(C(=O)NCCc3c(CNC(=O)C=C4CCC4)nco3)CC(CF)(CO1)C2 47333,N1(C(c2cc(CC)ncn2)=O)CC(C(=O)NCc2cncn2CC)CC(C)C1 47334,C1(OC)CCCN(C(c2cc(CNC(C3CC3C3CCC3)=O)[nH]n2)=O)C1C 47335,C(CNC(=O)CCCc1cnn[nH]1)(CC(=O)N1CCC(N(C)C)C1)OC 47336,C1(NC(c2c(SC)cccc2)=O)CC2CN(C(=O)CCc3cn(C)nn3)CC12 47337,Cc1sc(C)c(S(=O)(=O)NC(=O)CCCc2ncco2)c1C 47338,N1(C(=O)CCCc2ncco2)CCC(CO)(CNC(=O)C(F)OC(F)(F)F)C1 47339,Cc1cc(-c2nc(CC(F)(F)F)nn2CCCn2ccnc2)nc2ccccc12 47340,N1(CC)C(=O)CCC1CC(=O)NC1(C)CCN(C(=O)CCc2nccn2C)C1 47341,C(=O)(C1CCc2c[nH]nc21)NC(C(N1C(C)C(=O)NCCC1)=O)c1ccoc1 47342,C(=O)(C(C(C)(C)C)NC(N)=O)N(CC(F)(F)F)CCN(C)CP(C)(C)=O 47343,c1(-c2scc(C(=O)NC(c3ccc(Cl)cc3)CF)n2)ccc2c(c1)OCO2 47344,C(C)(C(O)C(=O)NCC1CCC(CNC(c2ccncc2C2CC2)=O)CC1)OC 47345,N1(C(c2c(C)nsc2)=O)CC(C2CCCN(C(=O)C(C)(F)F)C2)C1 47346,CCCCC(O)C(=O)NC(C)CC(C)NC(c1cc(C(C)(C)C)n(C)c1C)=O 47347,C12(CC(O)C13CCC3)C(=O)N1CCN(c3cccc(c3C)C2)CC1.CCOOC.O=CN.CCI 47348,c1(C(=O)NCC2(CNC(c3sc(C)c(O)n3)=O)CCC2)c(O)cccc1Cl 47349,c1(NCC(N(C)C(c2ccncc2F)=O)C2CC2)ncc2scc(Br)c2n1 47350,N1(CCNC(C)CCN)CC2C3C=CC(CC3)C2C1 47351,N1(C(CC=CCC)=O)CCCOC(CCNC(C2(C)CN(C(C)C)C2)=O)C1 47352,C1(C(N(C2CC(C(=O)NCC(C)OC)C2)CC)=O)CCCC(=O)N1C 47353,N1(C(C2(CO)CCN(C(CCC3CC(OC)C3)=O)CC2)=O)CC2COCC(C2)C1 47354,O(C1CCCC(=O)c2ccccc21)CC(N)CC1CCCC1 47355,c1(CC#N)ccnc(NCC2CCCCN2C(=O)CSc2ccc(F)cc2)n1 47356,S(=O)(=O)(c1ccc([N+](=O)[O-])cc1Cl)NCCNC(CCCNC(=O)OC(C)(C)C)=O 47357,C(CCCCCC(=O)N(CCCCCO)C)n1cc(CC)nn1 47358,C1(CC=C)(NC(=O)C(O)C2CC2)CCCN(C(=O)CCCN(C)C)C1 47359,C1(C(N2CC(CC=C)(NC(=O)Cc3[nH]cnc3C)C2)=O)COC(C)(C)CO1 47360,C1(C(N(CCCC)CC)=O)CSCCN1C(C1(Cl)CCCCC1)=O 47361,Cc1cc(C2CC2)cnc1C(=O)N(C)CCNC(=O)CCc1ccccc1O 47362,N1(C(c2c(N(C)C)ccnc2)=O)CCC2(NC(c3ncccc3F)=O)CC2C1 47363,N1(C(Cn2ncc(CC)c2)=O)CC(O)CCC1C(=O)NCc1ccc(F)c(F)c1 47364,c1(C(N2C(CNC(CCN(C(CCC)C)C)=O)CCC2)=O)ccc2nonc2c1 47365,CC(C)(O)C#CC(=O)NCCCNC(C1(C(=O)NC)CC1)=O.C12=CC=C(C=C1)C2 47366,CC(C)C(O)CNC(C1CCC1CNC(c1cc(CO)[nH]n1)=O)=O 47367,CC1(C)COC(C(=O)NC2CCN(C(=O)CCC=CBr)C2)CO1 47368,N1(C(c2nc(OC)c(F)cn2)=O)C2CCC1CN(C(=O)Cc1cnc(C)[nH]1)CC2 47369,C1(NC(C(CSC)C)=O)COC2(CNC(c3ccc(F)cc3N)=O)CC1C2 47370,N1(C(=O)CC2C=CCC2)CCCC2C1CCCCN2C(=O)COc1cccnc1 47371,N1(C(CCOC)=O)CC(C)(C)CCC1CNC(c1ccc(C(N)=O)c(Cl)c1)=O 47372,C1(CC(N2CCC(NC(c3cc(C(=O)OC)sn3)=O)C2)=O)CCS(=O)(=O)C1 47373,C1(NC(CCc2cn(C)nc2)=O)CN(C(=O)CSc2nncn2C(C)(C)C)CC1O 47374,C1(C(=O)NC2CC(C(N)=O)C2)CCN(C(=O)CC2CCCC2N(C)C)O1 47375,c1(CC(C(=O)OCC(N2CCC(C(F)(F)F)C2)=O)O)cccc(Br)c1 47376,N1(C(CCCC)=O)CCC2(NC(=O)C(N3CCOCC3)C)CCCCCC12 47377,C(=O)(C(CC(F)F)N(C)C(c1ccc(C#N)cn1)=O)NCC(C1CCCC1)C 47378,N1(C(Cc2cc(OCC)no2)=O)CCC2(C(=O)Nn3ccc(C)cc3=O)CC2C1 47379,C#CC1(O)CC(C(N2CCC(N(C(=O)CC(C)(O)C3CC3)CC)CC2)=O)C1 47380,C1(CC)(NC(c2cc[nH]n2)=O)CCN(C(C2CCC(=O)N(CCOC)C2)=O)CC1 47381,C(=O)(CCC(C)C#N)N1CCN(c2nnc(-c3c(C)nc(Cl)s3)n2CCC#N)CC1 47382,Cc1conc1C1CN(C(C2(NC(C3C4CCCC34)=O)CCCC2)=O)C1 47383,C#CCCCC(C)C(=O)NC1CN(C(C2(n3cccn3)CC2)=O)CC1C(F)(F)F 47384,C1(C)(CNC(C=C(COC)C)=O)CCN(C(C2CC(C)C(C(=O)OC)O2)=O)CC1 47385,C(CCCCC(=O)NC1(C)CC(N(C)C)C1)N(C)C(C1CCC2CC12)=O 47386,C1(C(N2CCCC(c3n(C(C)N)cnc3)C2)=O)Cc2c(C)cccc2O1 47387,C12(CNC(c3c(C)nc(Br)s3)=O)CCC1CCN2C(=O)CC1=CCCC1 47388,c1(NCC(N2CCC(NC(C3CCCSC3)=O)C(O)C2)=O)ccccc1[N+](=O)[O-] 47389,c1(CC)ncoc1C(=O)N(CCCC(=O)NCC(c1ccccc1)F)C 47390,c1(C(=O)Nc2sc(C(C)=O)c(C)n2)cc(O)ccc1Br 47391,C1(CC(C)=O)(C(=O)OC)CCN(C(CCCC)C(=O)NCCC#C)CC1 47392,C(=O)(CS(=O)(=O)C(C)(C)C)N(CC)CC1CCN(C(C2CC2CF)=O)C1 47393,C1(CCNC(c2sccc2C2CC2)=O)CCN(C(C2(CF)CC2)=O)C1 47394,C1(NC(C=CSC)=O)CN(C(c2ncc(Cl)cc2F)=O)CC(C)(C)C1 47395,N1(C(C2(C)CC2)=O)CCN(C(CNC(=O)COC2CCOC2)C(F)(F)F)CC1 47396,C(=O)(CCCC(F)(F)F)N1CC(C(=O)NCCCOCC2CCC2)CC(C)C1 47397,C(CCC(C)C)(C(=O)NCC1CC(C)C1)NC(C1CC=C(C)CC1)=O 47398,C1(C(=O)NCC2(C(C)C)CCCC2)CC2CN(C(=O)C(C)n3ccnn3)CC2C1 47399,C1(NC(CCC(=O)N(CC)CC)=O)CCN(C(c2nn(C)cc2Cl)=O)C12CCC2 47400,c1(CNC(N2CCC(=CCc3nn[nH]n3)CC2)=O)n[nH]c2c1CCOC2 47401,c1(OC)cc(C=CC(=O)NCC2CC2NC(C2(n3cnnn3)CCCCC2)=O)sn1 47402,C1(CNC(CN(C(C)C)C(C2CC3CCC(C2)O3)=O)=O)CC12CCCCC2 47403,N(C1CCc2cccnc21)C(CCOCCNC(C1CN2CCC1C2)=O)=O 47404,C1(C(N(C(C)CC(=O)NCc2ccco2)C)=O)CC2CCC2C1 47405,c1(C(N2C(C)CN(C(=O)CC#N)CC2)=O)cccc2c1CC(=O)N2C 47406,C1(C(N2CC(C)(NC(c3ccc(Cl)s3)=O)C2)=O)CCc2nn[nH]c2C1 47407,C(=O)(C(C)CC(C)C)N(CCCC(=O)N(CCC)CC)C 47408,c1(C(=O)NC(CCOC)CNC(=O)C(F)n2cccn2)ncc(Br)cc1N 47409,c1(C(N(CC(C)CNC(=O)COCC2CCOC2)C)=O)cnn(C)c1F 47410,C=CC(C)(O)C(=O)NCC(CNC(c1sccc1Cl)=O)OC 47411,C(=O)(C(F)(F)C(F)(F)C(F)(F)C(F)F)N1CCCC(NC(C(C=C)O)=O)C1 47412,N1(C(c2ncc(C)c(C)c2)=O)CCC2(CC(NC(=O)C(C)(C)C(F)F)CO2)C1 47413,c1(C(=O)NCC(CC=C)NC(c2ccc(CC)o2)=O)cc(C(C)=O)ccc1O 47414,C(CCC(C)CC(=O)NC1CCCN(C(c2ccns2)=O)CC1)=C(C)C 47415,c1(CC(C)C(=O)N2CCC(N(C(=O)Cn3ccnn3)C)C2)cccc(Cl)c1 47416,CC1CN(C(c2ncccc2C(N)=O)=O)CC1NC(=O)CCCc1cnn[nH]1 47417,N1(C(C2(NC(CNC(CC)=O)=O)CC(O)C2)=O)CC2(CCC(=O)O2)C1 47418,C#CCCCC(C)C(=O)N1CCC(C)(CNC(c2c(F)ccc(OC)c2F)=O)C1 47419,c1(C(C)C)ccc(C(=O)NCC(C)NC(=O)CCC2CCC(O)CC2)cn1 47420,c1(CN(C)C)ccc(C(=O)NCC2CCCCN2C(C2CC3CCC2O3)=O)cc1 47421,c1(OC)ccc(C(N2CC(OCCNC(=O)C(N)=O)C2)=O)c2ccoc12 47422,N1(C(CSCCCC)=O)CC(CNC(=O)CN2CCN(C3CC3)C2=O)CCC1C 47423,C12(NC(CCc3nnc(C)n3C)=O)CCN(C(=O)CC3(C)CC3)CC1C2 47424,Cc1c(C(=O)NC23COC(CNC(=O)Cc4csc(S)n4)(C2)C3)cnn1C 47425,C(=O)(Nn1cccn1)c1cc(CNC(c2ccccc2O)=O)no1 47426,C(=O)(C(C#N)C(C)(C)C)NCC1(F)CCC(NC(COCCOC)=O)C1 47427,c1(NC(C2N(C(c3ccc(Cl)cc3)=O)CCC(=C)C2)=O)cnc2c(c1)CCC2 47428,Cc1ccc2c(C(N3CCC(CNC(=O)CC(O)C(C)(C)C)C3)=O)c[nH]c2c1 47429,c1(CN2CCC(c3cccc(C)c3)C2)c(Br)cncc1Br.C12CCC(C1)NC2=O 47430,N1(C(CSCC=C)=O)CCCCC12CC(NC(c1ncsc1C(C)C)=O)C2 47431,N1(C(CC2(OC)CCC2)=O)CCC(CF)(NC(c2ccc(C(F)F)o2)=O)C1 47432,C1(C(N)=O)CC(C(=O)NCCCNC(=O)CSCC2CC2)=NO1 47433,N1(c2n(C)c(C3(O)CC(c4ccccc4)C3)nn2)CCC2(CCCCO2)C1 47434,N1(C(CCC=C=C)=O)CC(NC(=O)CC(C)COC)C(N=[N+]=[N-])C1 47435,C1(C(=O)NC2(C)CC(NC(C3CCC(C)CC3)=O)C2)CCn2c(O)nnc2C1 47436,Cn1nccc1CCC(=O)NC1CCCC1NC(c1coc(Cl)n1)=O 47437,Cc1cc(=O)cc(CNC(C2CN(C(c3sccc3C#N)=O)CCO2)=O)[nH]1 47438,C1(NC(C(CC)C#N)=O)CC(O)(C2CCN(C(=O)CCc3csc(C)n3)CC2)C1 47439,N1(C(c2cc(COC)on2)C(=O)NCC(F)F)CC2CC2(CO)C1 47440,n1(CC(=O)Nc2c(F)cc(I)cc2F)ccc(=NC(=O)c2cc[nH]c2)nc1O 47441,c1(C(=O)NC(C)C(C)NC(c2cc(C(F)(F)F)cc(N)c2)=O)cn2c(n1)CCC2 47442,C1(C(N2CC3(C(=O)OCC)CC2(C(=O)OC)C3)=O)CCCC2CCCCC12 47443,N1(C(C(CC#C)(C)C)=O)C2CCC1C1CC1(NC(C1CCC(=O)N1CCC)=O)C2 47444,c1(C(C(=O)NC23CN(C(C(C)O)=O)C(C2)C3)=O)cc(F)ccc1F 47445,c1(SC)nc(Br)c(N(C2CC2)Cc2ccc(-c3ccncc3)o2)n2ccnc12 47446,C1(C(=O)NC(Cc2ccco2)CO)(NC(Cc2c(C)ccs2)=O)CCCCC1 47447,C1(NC(CC2N(C)CCCC2)=O)CCC12CN(C(=O)C1=NNC(=O)C1)C2 47448,N1(C(CC(=O)OCC)=O)CC2(CCCC2)C1C(=O)NC(c1nccn1C)C 47449,C1(C(C)NC(c2cn(CCC)nc2)=O)CCCCN1C(=O)Cn1nnc(C)n1 47450,S(=O)(=O)(c1cc(C)cnc1NCCO)NC(C(CC)C)C 47451,C(=O)(CN=c1cc[nH]cc1)NCC(C(=O)NCC(CCC)C)C 47452,C1(NC(C2C(=C)CC2)=O)CN(C(c2cc(Br)cn2C(C)C)=O)CC1F 47453,C(C)(C)(CC(=O)NCCC(N1CCC(O)(C(C)C)C1)=O)OC 47454,C1(C(=O)NC(C)CN2CCN(C(c3ccon3)=O)CC2)CC12CCCCC2 47455,c1(CC)cc(NC(C2CCCCC2NC(=O)CCc2ccncc2)=O)cnc1C 47456,C1(C(=O)NCCN2CCNC2=O)(CC)CCN(C(C2CCNC2=O)=O)C1 47457,c1(C(=O)NC(CNC(c2cnc(SC)n2C)=O)C)cnn2ccnc(N)c12 47458,N1(C(c2ccc(OC(C)C)nc2)=O)CC2=C(C1)CN(C(c1cc[nH]c1)=O)C2 47459,C1(C(=O)OCc2cnc(C#N)s2)CC2(CCC(F)(F)CC2)CO1 47460,C(=O)(C#CC1CCCOC1)N1CC2CCC(NC(c3cc(C)nnc3O)=O)C2C1 47461,c1(C(=O)NC2(C3CN(C(C(C)(C)CC4CC4)=O)C3)CC2)c[nH]c2ccc(F)cc12 47462,C1(NC(C2CCCOC2)=O)CC2(C1)CC(C(=O)NCC(O)C(F)F)C2 47463,CC1(F)CN(C(=O)Cc2ccon2)CCN(C(=O)CCS(C)(=O)=O)C1 47464,C(=O)(C1CCCn2ccnc21)NCCC1N(C(c2ncn(CC)n2)=O)CCSC1 47465,c1(C(N(C)CC2(O)CN(C(C(C)COc3ccccc3)=O)C2)=O)ccc(O)nn1 47466,Cc1ccc(N)c(C(N2CC(C)(C)CC2CNC(c2cn(C(F)F)cn2)=O)=O)c1 47467,N1(C(CCc2ccc(C)cc2)=O)CC2CC(O)C1C2NC(C1CCC1)=O 47468,c1(Cc2onc(C(=O)NCC)n2)cccc(Br)c1O 47469,C1(CNC(C=CC=CC)=O)CN(C)CCN1C(C1CCCN1CC(C)C)=O 47470,N1(C(C2(c3ccccc3F)CC2)=O)CCc2c(C(=O)O)cccc2C1 47471,c1(C(N(C2CN(C(=O)C(O)c3ccco3)C2)C)=O)ccc(S(N)(=O)=O)s1 47472,c1(C(=O)NC2(CC)CN(C(c3ccccc3OCCN(C)C)=O)C2)cnn(C)c1N 47473,CCC(F)(C(=O)OC)C(=O)N1CCOC(CN(C(=O)Cc2cnoc2)C)C1 47474,CC(N=[N+]=[N-])C(=O)NC(CC1CCC1)C(N1CCCCC1CF)=O 47475,C1(NC(c2ccc(C(F)F)o2)=O)CCCC12CCN(C(=O)CCc1ncc[nH]1)C2 47476,c1(C(=O)OC)cn(C)nc1C(=O)NCC1CC1CNC(C1CCCCC1C)=O 47477,N1(C(c2c(C)ccnn2)=O)CC(NC(c2ncccc2F)=O)CC12CCOC2 47478,C1(NC(CCC(N)=O)=O)CCN(C(C2CN(C3COC3)C2)=O)C(C2CC2)C1 47479,c1(C(=O)NC(CN(C(CC(CC)C(C)C)=O)C)C)c(O)cnc2cc(F)ccc12 47480,CC(C)(O)C(F)(F)C(=O)NC1CC(NC(c2sc3cnccc3c2Cl)=O)C1 47481,N1(C(C(C)CSC(F)(F)F)=O)CCC(CCN(C)C)(NC(=O)CNC=O)C1 47482,c1(C(=O)NC)ccc(COCCSCC(=O)N(CCC)C(C2CC2)C)o1 47483,N1(C(CC2(OC)CCC2)=O)C(C(=O)NCC(C)OC(F)F)CCC1C1CCCC1 47484,C(=O)(CC(=O)NCc1n[nH]cc1CC(N1CCCC1CC(C)O)=O)OC 47485,C(=O)(C(C(F)(F)F)C(F)(F)F)NCCC1N(C(c2ncn(CC)n2)=O)CCOC1 47486,Cc1cc([N+](=O)[O-])ccc1C(=O)NC1CCC1NC(=O)C(=O)NC(C)C 47487,Cc1ccc(C(=O)NC2CCC2CNC(C2COCCO2)=O)cc1Cl 47488,C1(C)(C(N(CCCC(N2CCC3CCC23)=O)C)=O)CC(=O)N(C)C1 47489,C1(C(N(CC(C)NC(C=CC)=O)C)=O)CCCN1CC(C)C 47490,N1(CCc2ccc(OC)cc2)CCCCS(=O)(=O)C1CO 47491,C1(c2ccc(C)o2)CCCCCN1C(=O)Cc1ccccc1C(=O)O 47492,C1(NC(c2cccc(SCCC)c2)=O)CN(C(c2ccc(C)cn2)=O)C(C)(C)C1 47493,CC1CCCC=C1C(=O)N1CCCN(C(C2CNC(=O)CC2(C)C)=O)CCC1 47494,C(C)(C(C)(C)NC(c1cccn1C1CCCC1)=O)NC(C(C)n1cncn1)=O 47495,c1(CCCC(=O)NC2C(NC(C(CCC)NC(N)=O)=O)C2)cc(O)ccc1C 47496,CCC(C(=O)N1CCC(NC(=O)CCNC(C)=O)C1Cc1ccccc1)C(C)C 47497,N1(C(c2cnc(CC)s2)=O)CCC2(NC(c3ccc(C)n3C)=O)CC2C1 47498,C(C(C)(C(=O)NCCC1CCSC1)NC(c1ccc(F)cn1)=O)SC 47499,C1(N(C(CCOCC#C)=O)C)CN(C(=O)CCCCC)CCC1O 47500,CC(C)CCN=C(NCC1=CCOCC1)NCC(c1c[nH]c2ccccc12)(C)C 47501,c1(C(=O)NCC2CN(C(C3C(C)C3C)=O)C2)n[nH]c(C2CC2)c1Cl 47502,C(CCN(C)C(C12CCCC1C2(F)F)=O)(C(C)(C)C)NC(C=CC=CCC)=O 47503,c1(C(=O)NCC2OCCC(NC(=O)CCF)C2)ccc2c(c1)C(=O)CCCC2 47504,c1(NC(CS)=O)c[nH]nc1C.C1(C(=O)OC)CC1(Cl)C(=O)O 47505,C1(C(=O)NC(C#C)CC2CC2)CCCCCC1NC(C1(C)CNC(=O)N1)=O 47506,C(=O)(CCCCCCCC(=O)NCCNCc1ccc2cn(C)nc2c1)OC 47507,C(CN=c1[nH]c(=NC2CC2)[nH]c2ccsc12)N1C(CSC)CCC1 47508,C1(NC(CCc2ccc(C)cc2)=O)CC12CCN(C(C1CC1C(N)=O)=O)C2 47509,C(C1=NOC2CN(C(c3cc(NC)ccc3Cl)=O)CC12)NC(CCCC(=C)C)=O 47510,C(=O)(CC(C)(O)C1CC1)N1C(C(C)NC(=O)Cc2cscn2)CC1 47511,Cc1[nH]c(C(=O)NCc2ncccn2)c(C)c1C(=O)NCc1cncn1C 47512,N1(C(c2cc(C)[nH]c2C)=O)CCCC(C)(NC(c2cnoc2C)=O)C1 47513,c1(C(=O)NCC(C)(C(C)C)NC(C=CCC)=O)c(Br)ccc(C)c1F 47514,N1(C(CCc2c(OC)cccc2)=O)CCCCC(NC(C23CC(C)(CO2)C3)=O)C1 47515,c1(CC)cccc(C(N2CC(C)C(O)C2)C(=O)NC2CCOCC2)n1 47516,n1(CC(COC)C)cc(C2(C3CC3)CC2)nn1.C12(CC1)CC2 47517,C1(C(=O)NCC2(CCNC(=O)CC3CCCC3)CC2)CC12CCCCCC2 47518,c1(OCC2CC2)cncc(NC2CCC(c3nn[nH]n3)C2)n1.CN1C(=O)N1 47519,C(=O)(C(C)(F)C(=O)NCCC(C)NC(c1cc(C)n(C(C)C)c1C)=O)OC 47520,Cc1ncnc(C)c1C(=O)NCC(F)CNC(=O)C(c1cccc(F)c1)(C)O 47521,C(=O)(CC1=CCOCC1)N(C)CC1CCN(C(=O)CC2CCCSC2)C1 47522,CCC(C)C(O)CC(=O)NCc1ccc(C(=O)NCC2CCC3(CC3)C2)cn1 47523,Cc1ccn2c(C(N3CC4CC3C4NC(=O)CC(O)CN(C)C)=O)cnc2c1 47524,n1(CC)cc(Cl)c(C(N2CCC(O)(CN(C)C(C3(C)CSC3)=O)C2)=O)n1 47525,c1(C(=O)NCC2(NC(=O)CC3CCC(O)C3)CCOCC2)cnc2[nH]nnc2c1 47526,c1(C(=O)NCC=CCNC(C(CC)(C)C#N)=O)nc2ccc(Br)cn2c1F 47527,C1(C(C)C)(C(=O)Nc2cnsc2)CCN(C(c2ccncc2O)=O)C1 47528,C12(OC)CCCCC(C(=O)NCCCCN(C(=O)C(C(C)C)C(C)C)C)(C1)C2 47529,c1(C(N2C(C(=O)Nc3cnccc3I)CC(C)C2)=O)ccc(Cl)c(C(F)(F)F)c1 47530,CCCC(C(=O)N1CC2CC1C2CNC(c1cc(C)n(C)n1)=O)OC 47531,C1(C(=O)NCCCCNC(C(CC=CC)CC)=O)OCCOC12CCC2 47532,N1(c2cc(C)nc(N3CCC(C4CCCO4)C3)n2)CCC2(CCOC2)CC1 47533,C1(CNC(C2(NC(c3nc(C)sc3C)=O)CSC2)=O)CCCN(C)C1=O 47534,c1(C(N(C2CN(C(=O)COCCCF)CC2F)C)=O)cccc(Cl)c1F 47535,c1(OC)cncc(C(N2CC(CNC(=O)CC3(C#N)CC3)CC2C)=O)n1 47536,C1(N(C(CC=CC=C)=O)CCOC)CCN(C(C2CCCCN2C(C)=O)=O)CC1 47537,c1(C(=O)NC(CC2CN(C(C3CN(CC)C(=O)N3)=O)C2)C)ccc(=N)[nH]c1Cl 47538,C1(NC(C=CC(N)=O)=O)CCCC2CN(C(=O)Cc3nc4c([nH]3)CCCC4)CC12 47539,N1(C(CCCC#C)=O)CCC2(NC(c3n[nH]cc3COC)=O)CCCCCC12 47540,c1(C(N(CC(CC)NC(c2cccn2Cc2ccncc2)=O)C)=O)cc(C)sn1 47541,c1(C(N(C)CCOCCNC(C2CCCN2S(C)(=O)=O)=O)=O)cc(Cl)n(C)n1 47542,c1(CC)ncc(NC(=O)NC2CCN(CC3CCOCC3)CC2)c(C)n1 47543,CC1CCC(C2CC2)CN1C1CCCC1.C(S(=O)(=O)N)N(C(=O)CN)CCO 47544,c1(C(N2CC(CNC(CC(C)(C)C)=O)OCC2)=O)cc(Cl)ncc1O 47545,C1(CC)CN(C(c2cncc(C)n2)=O)CCC1NC(=O)CC1CCOCC1 47546,Cc1cnc(CCNC(C2C3CN(C(=O)CCCc4cnn[nH]4)CC23)=O)cn1 47547,c1(C(=O)NC(CN(C(=O)C(C)CC2CC2)CC)C)c[nH]cc1-c1cnn(C)c1 47548,N1(C(C2C(C)=CCS2)=O)CCC(NC(C2CS(=O)(=O)C2)=O)C(C)(C)C1 47549,CC1(C)CC(NC(=O)CC2(C3CC3)CC2)CN1C(=O)CC1CN2CCC1CC2 47550,C1(C2CCN(C(=O)CC3CCNC3=O)C2)(NC(c2nnc(O)nc2O)=O)CC1 47551,N1(C(C2C(CNC(C(C(C)C)N(C)C)=O)CCC2)=O)CC(N(C)C)C2(CC2)C1 47552,C(C)(CC(=O)NCC(C)N(C)C(C1CCOCC1)=O)=C(C)C 47553,C12(CCNC(=O)NCc3cn(CCC)nc3)CCC(CC1)CC2 47554,CON1CCC(NC(C2(NC(=O)CC3CC4CC4C3)CC(F)C2)=O)CC1 47555,C(=O)(C(C)(C)C(=O)NC(C)C(C)NC(=O)CSc1ccccn1)OCC 47556,c1(CCNC(N2CC(C)S(=O)CC2)=O)nc2ccccc2s1 47557,N1(S(c2cc(CC)oc2C)(=O)=O)CCc2sccc2C1C(=O)OC 47558,C1(C(=O)NC(c2cccnc2O)C)CCCC(NC(=O)C(C2CCOCC2)F)C1 47559,C1(CC(=O)N(C(C)CN(C(=O)CN2CCCC2=O)C)C)CC=CCN1C 47560,N1(C(C(C)Oc2cccc(Cl)c2)=O)CC2CCN(C(C3CC=CC3)=O)CCC2C1 47561,c1(SCCCC)cccc(C(=O)NCCCNC(=O)CC2CC3(CC3)CO2)c1 47562,c1(CNc2c(C(=O)NCC(F)(F)F)scc2)ccc(Br)cc1Cl 47563,N1(C(C(=O)NC(c2cccc(OC)c2)CF)=O)CC2CC(C)C2C1 47564,c1(C(=O)NCC2CCCN(C(CCC=C)=O)CC2)nnc2n1CCCCC2 47565,C1(OC)(CNC(=O)Cc2ccc(F)cc2F)CCN(C(=O)CSC(=N)N)CC1 47566,CC(CN(C)C)CCC(=O)N(C)CCN(C(=O)C(c1ccc(F)cc1F)(C)C)C 47567,C(=O)(CC(C(C)(C)C)NC(c1c[nH]c(=S)cn1)=O)NC(CCC)C(F)(F)F 47568,N1(C(C(CC)(C)C#N)=O)CCC=C(C(=O)NOCC2CC(OC(C)(C)C)C2)C1 47569,CC#CCC(C(=O)N(C1CCN(C)C1)C)NC(=O)CCC(C)(C)OC 47570,n1(CC)ccc(C(N2CC(NC(=O)Cn3ccnn3)CC2C)=O)cc1=O 47571,N1(C(C2OCCN(C)C2)=O)CCN(C(c2cnn(C)c2Cl)=O)CC(CO)C1 47572,N1(C(COCC(C)C)=O)CC2CC1CCC2NC(=O)CSCc1cscn1 47573,CN1CC=C(CCNC(=O)C(C)(CO)NC(=O)Cc2ccccc2O)CC1 47574,c1(NC(CN(C(CC(CCC)N)=O)C)=O)ccc2c(c1)OCCO2 47575,C1(C)(CC(=O)NCC2CN(C(CNC(C)=O)=O)C2)CCCO1 47576,C1(O)(C(=O)NC(CNC(c2n(C)nc(C)c2Cl)=O)C)CCCC(C)(C)CC1 47577,N1(C(CN(CCC)C(c2cc(COC)on2)=O)=O)CCCC2(CC2)C1 47578,CC1=NN(C)C(=O)C1CC(=O)NC1CC(NC(C2CC(F)(F)C2(C)C)=O)C(O)C1 47579,C1(CNC(Cc2c(C)ncs2)=O)CCCN(C(C2CCC(C(C)C)CC2)=O)C1 47580,c1(C(N2CC(C)(C(N(C3C(C)CC3)C)=O)C2)=O)ccc(N)cn1 47581,c1(C2(C(=O)NCC3CCN(Cc4nc(Br)cs4)CC3)CCCC2)ccc(Cl)cc1 47582,C1(C(N(C(CC2CC2)CO)C)=O)(CNC(=O)Cc2cc[nH]c2)CC=CC1 47583,C1(C(=O)NCC(CCNC(C(C)NC=O)=O)O)CCCC(F)(F)C1 47584,C1(C)(CNC(C(C)(N(C(c2scc(OC)c2)=O)C)C2CC2)=O)NC(=O)NC1=O 47585,c1(C(=O)NC2CCN(CCCCc3ccccc3)C2)ccc2cc(Br)ccc2c1 47586,CC1(CNC(c2cccc(O)n2)=O)CCCN1C(=O)CCc1cnc[nH]1 47587,S(=O)(=O)(c1cccnc1NCC1(CC#N)CC1)NCC(CCOC)(C)C 47588,C1(C(N2C(CN(C(=O)Cc3nncn3C)CC)CCC2)=O)CC2C=CCC(C1)C2 47589,c12cccc(c1)C2O.n1(CC(=O)NC(C(C)C)c2nc[nH]n2)cc(CO)nn1 47590,c1(CC)ccc(C(=O)NC2CCC(CCNC(=O)Cn3cnc(=N)[nH]3)C2)nc1 47591,C(=O)(C1CC(=O)Nc2ncccc21)NCCN(C)C(c1cnc(CC(C)(C)C)o1)=O 47592,C(=O)(C(C)(C)CCCNC(=O)Cc1cn(C)cn1)N1C(C)CCC(C)C1 47593,C(=O)(C1CCc2c[nH]nc21)NC1CC2CC(NC(CCNC(=O)NC)=O)C2C1 47594,C1(CNC(c2nccc(C)c2)=O)CN(C(=O)C(F)=C2CCC2)CC(C)(C)C1 47595,c1(OC)cncc(C(N2CC(N3CCN(C(C4CC4CF)=O)CC3)C2)=O)c1 47596,N1(C(C)=O)CCCC1C(=O)NCCOCCN(C(=O)C(C)(C)OC)C 47597,C1(NC(C(=O)N(C2CC(C)OCC2)C)=O)CN(C(=O)C(F)(F)F)CCC1O 47598,C1(NC(c2cc[nH]c2)=O)CC12CC(NC(c1cncc(C(F)(F)F)c1)=O)C2 47599,c1(NC2C3N(C(CCCOCC)=O)CC(CC3)C2)ncnc2c1ncn2CC 47600,c1(C(=O)NCC(C)(C2CCC2)NC(CN(CCOC)C)=O)cccc(C(F)F)c1 47601,N1(C(c2c(O)ccc(C)c2)=O)CC2(NC(C3CCCCS3)=O)CCC1CC2 47602,C(=O)(CC(O)CN(C)C)NCC(C)(C1CC1)NC(c1cc(C)[nH]n1)=O 47603,N1(C(c2cc(C)no2)=O)CC2CCCC(NC(=O)C(C)CC3CCC3)(C2)C1 47604,C1(CC(=O)N(CC#C)CC)CCCN(C(c2ccc(SC)o2)=O)C1 47605,C(=O)(CS(=O)(=O)C1CC1)NCC(C1CCN(C(COCC=C)=O)CC1)O 47606,O=C1OCCC1Cc1cn(CCC(N2CC(O)(CN3CCCC3CO)C2)=O)nn1 47607,CC1(C(=O)NC2(CN)COC2)CCCN1C(C1CCOCC1)=O 47608,N1(C(C(CCC)F)=O)CCN(C(=O)CC2COC(=O)C2)CC1CCC 47609,C1(CNC(C(CC2CCC2)OC)=O)CN(C)CCN1C(=O)CC1CC1 47610,C(c1cccc(Cl)c1Cl)=CC(=O)NCCCCCCNC(=O)CC1CCOC1 47611,CONC(=O)C(=O)NCC(C1CCC1)NC(=O)Cc1nnc(S)n1C 47612,C1(C(N(C(CNC(C2CSCN2C(N)=O)=O)C2CC2)C)=O)(CF)CCOCC1 47613,N(C(=NCCCN1CCOCC1)NCC(=O)NOC)CCN(C(=O)OC)C 47614,c1(C(=O)NC(CC)CCC(=O)NCC(N2CCOCC2)=O)ccc2c[nH]nc2c1 47615,C(C(=O)SC(CNC(=O)CN(C)C(=O)OC(C)(C)C)C1CC1)=CCC.C1CC1 47616,CCC(CC(=O)NCC(C)(O)C1CCCC1)N(C(=O)C(C)OCCOC)C 47617,C(=O)(C(COC(C)C)NC(C)=O)N(C1CCN(CC2CCSC2)C1)CC 47618,c1(OC)cc(C(N2CCC(NC(=O)Cn3ccc(C)n3)C(F)C2)=O)c(F)cn1 47619,C(C1CCN(C(=O)CC2CC(F)(F)C2)CC1)=CC(=O)NCCC1C(C)CCCC1 47620,c1(C(=O)NC(C)CCNC(=O)CSC(F)(F)F)cnn(CC(F)(F)F)c1 47621,c1(C(C)NC(CC2CCN(Cc3ccn(CCC)c3)C2)=O)c(C)nn(C)c1C 47622,c1(N(CC(F)F)CCc2nc(C[Si](CC)(C)C)on2)cnc(O)cc1O 47623,n1(CCCC)nc(C(=O)N(C)CC2(CO)CC2)ccc1=O.C1(=O)C(OC)N1 47624,c1(CCC)c(C(N2CC(c3ccccc3C(F)(F)F)C2)=O)cnn1CCO 47625,C1(C(=O)NC(CCCC)COC)CC2(CCC2)CN1C(C1(N2CCCC2)CC1)=O 47626,N1(C(c2c(C)snn2)=O)CCCC(CNC(C2CN(C3CCOC3)C2)=O)C1 47627,C1(C(=O)NCC2(CN(C(CC3CC(OCC)C3)=O)C)CC2)CC2CCC1NC2=O 47628,C1(F)(C(=O)NC2CCC(C(N(C(c3ccccn3)C)C)=O)C2)CCOCC1 47629,Cc1nccnc1C(=O)NCCC(C)(C)NC(C1CC(F)(CF)C1)=O 47630,c1(CC(N2CCC(NC(CC=CC=C)=O)C2)=O)cccc(OC)c1Cl 47631,c1(C(N(CCCNC(c2csc(Cl)n2)=O)CC)=O)ccc(CO)cc1 47632,C12(NC(c3cc(-c4cccs4)[nH]n3)=O)CCCC(CN(C(=O)C(F)F)C1)C2 47633,N1(C(c2c(OC)cncn2)=O)CCC(F)(F)C(CNC(c2cc(Cl)c[nH]2)=O)C1 47634,S(=O)(=O)(c1ccc(F)cc1)N1C(CCNC(N2CCOCC(F)C2)=O)CCCC1 47635,c1(OC)cc(F)c(C(=O)Nc2cccc(NC(C34CC(C3)C4)=O)c2)cc1F 47636,C#Cc1cccc(C(=O)NCC2(OC)CN(C(C3CCC(C)CC3)=O)C2)c1 47637,N1(C(CCc2cccc(OC)c2)=O)CCC2CN(C(C3CCCS3)=O)CC12 47638,c1(C(=O)Nc2c(C(=O)OC)c(NC(C)=O)c(C)s2)c(=O)ccc2ccccc2n1 47639,C1(CC(c2nnnn2CC2CCOC2)(C)NC(C2CCCCC2)C)CC(F)(F)C1 47640,c1(SCC(=O)NCCNC(c2c(C)ccnc2)=O)ccc2ccccc2c1 47641,CC1(C)CC(CC(N2CC(O)CC2CNC(C2CC=CCC2)=O)=O)CC(C)(C)O1 47642,c1(CC)ccsc1C(=O)N(CC(C)C(=O)N(CC(CC)OC)C)C 47643,C1(CNC(CC(=C=C)C)=O)CN(C(=O)Cn2c(C)c(C)sc2=O)C(C)(C)C1 47644,CC1(C)CC(CNC(=O)CCN2CCCCC2)N(C(c2ccnc(C#N)c2)=O)C1 47645,Cc1[nH]nc(C(N2CCCCC2CN(C)C(c2cc(C#N)on2)=O)=O)c1F 47646,N1(C(c2c(CC)n(C)cc2)=O)CC2CN(C(C34CC(F)C3C4)=O)CC2C1 47647,C#CC1N(C(=O)C(=O)Nc2cccc(OCc3ccncc3)c2)CC12CCC2 47648,c1(C(C(=O)NC(C)CN(C(=O)CCc2cnn[nH]2)C)O)ccccc1C(F)(F)F 47649,C1(NC(c2nc(C)sc2)=O)CC(C(NC[Si](C)(C)C)=O)C1(C)C 47650,Cc1cc(CC(=O)NC2CCN(C(c3csc(Br)n3)=O)CC2)nn1C 47651,N1(S(c2c(OCCCCC)c(Cl)ccc2)(=O)=O)CCn2ncc(S(C)(=O)=O)c2C1 47652,N1(c2cc(C)nc(N(C)Cc3nnc(C)s3)n2)CCc2nc(Br)sc2C1 47653,N1(C(CCC(=O)N(C)C)=O)CCC2CN(C(C3CCn4nnnc4C3)=O)CC2C1 47654,c1(C(=O)NC2C(CC(=O)NCCC(C)O)CCC2)ccc(N)cn1 47655,c1(CN=C(NC(CF)CF)NC2CCSC2)ccc(F)c(Cl)c1 47656,C1(C2CCCCO2)(C(=O)NC2CC(NC(c3ccn(CC)c3C)=O)C2)CCCO1 47657,CCC(C)C(C(=O)NCC1(OC)CN(C(c2ccc(SC)nc2)=O)C1)OC 47658,C=CC(O)(C(=O)NC1CCN(C(=O)C(=O)NCCOC)CC1O)C(F)(F)F 47659,c1(NC(C2N(Cc3cc(C)cc(C)c3)CC(C)C2)=O)cc2oc(C)nc2cc1Cl 47660,C(=O)(C(O)CC[S+](C)C)NC1C(NC(c2ncc(C)c(C)c2)=O)CCCC1 47661,CC1CC(S(C)(=O)=O)CN1C(=O)Nc1ccc(-c2ncco2)cc1 47662,C1(C2CCC2)(C(=O)NCC(C)(C)OCCNC(C2CCC(F)(F)C2)=O)CCC1 47663,C=CCCCCCCC(=O)N1CC(CN(C(=O)CC2CCOCC2)C)C2(CC2)C1 47664,c1(C(N2CC(CC(C)NC(=O)CC34CCCC3C4)C2)=O)cc2cccnc2o1 47665,C1(NC(C2(CC)CCCC2O)=O)CC=C(C(=O)NC2CC3C(C2)C3(F)F)C1 47666,CC1CCc2ncc(C(N3CCCC34CCN(C(c3ccncc3)=O)C4)=O)n2C1 47667,C1(NC(c2ccnc(C)n2)=O)COC2(CCN(C(c3cnsn3)=O)C2)C1 47668,Cn1cc(Cl)cc1C(=O)NCc1ccoc1C(=O)NC1CCCC(F)C1 47669,N1(C(CC=C)=O)CCC2CN(Cc3ccc(Br)cc3O)CC12 47670,CCC(CC)(CCNC(=O)C(C(C)(C)C)SC)NC(=O)COC(F)F 47671,N1(C(C(N2CCCC(C)C2)=O)=O)CCCC2(NC(C3(C4CCC4)CC3)=O)CC2C1 47672,c1(NC)ncccc1C(=O)NCCC(O)CNC(=O)CCC1CC(C)C1 47673,c1(C(=O)NC2CC(NC(C=CCOC)=O)C2)cc2c(nc1O)CCCC2O 47674,C1(NC(C(CSC)C)=O)CCC2(CCN(C(c3ccoc3Cl)=O)C2)C1 47675,CN1CCC(N(C(c2csc(C(F)(F)F)c2)C(=O)NC2CC2)C)C1 47676,c1(C(=O)NC(C)(C)CCNC(=O)C2=C(Cl)CCCC2)c(N)c(F)cc(F)c1F 47677,c1(OC)ccc(C(=O)NCC2CCCN(C(=O)COCc3nc[nH]n3)CC2)c(Cl)n1 47678,CCCCCC(O)C(=O)N1CC2=C(C1)CN(C(c1ncc(Br)cc1N)=O)C2 47679,c1(C(=O)NC(C(C)Nc2ncc(C)c(O)n2)C)ccc2nnc(O)n2c1 47680,C#Cc1nccnc1NC(C1CC1NC(c1cnc(CC)cn1)=O)=O 47681,C(=O)(C(O)C(F)(F)F)N1C(C(N2CCC(CC(C)(C)C)C2)=O)C=CC1 47682,CC(C)CC(CNC(=O)C(C)(C1CC1)N(C(=O)CN1CCOCC1=O)C)N(C)C 47683,CC1CN2CCN1C(C(=O)NC(C)(C)CNC(=O)CCCN1CCCC1)C2 47684,c1(OC(C)C)ccc2c(c1)CCN(C(=O)C(=O)NCC1CC(O)C1(C)C)C2 47685,CCC(C)(O)C(=O)N1CCN(C2CCCC2NC(=O)C=CC2CCCCC2)CC1 47686,CC1(C)CC(NC(c2ccc([N+](=O)[O-])s2)=O)CN(C(=O)Cc2cc[nH]n2)C1 47687,C(=O)(C#CC1CC1)NC1CCN(C(CCN(C)CCO)=O)C1 47688,N1(C(C2N(C)CCCC2)=O)CCN(C(=O)CSc2ccncc2)C(CF)C1 47689,C(C(C)N=c1[nH]c(=N)[nH]c(=NCCc2c(F)cccc2Br)[nH]1)(C1CC1)OC 47690,c1(C(N2CC(C)C(CNC(C3CC34CCCC4)=O)C2)=O)ccc(F)c2c1OCC2 47691,CC1(C(=O)NCC(C2CCCC2)NC(c2cc(Br)no2)=O)CC(F)C1 47692,N1(C(C(COC)C)=O)CCC2(CCCN2C(c2cncc(OC(F)F)c2)=O)CC1 47693,C1(NC(c2c(CC)scn2)=O)CC(CNC(c2cn(C)nc2OC)=O)C1(C)C 47694,C1(C(=O)NCC=CCNC(c2cc(C)on2)=O)CCn2nccc2C1 47695,Cn1ccc2cc(C(=O)NCC3CC(CNC(=O)Cc4cnc[nH]4)CO3)cnc12 47696,C1(NC(c2nc(CC)sc2)=O)CN(C(=O)Cc2cc[nH]c(=N)c2)CC2(CC2)C1 47697,N1(C(C2(C#C)CCN(C(=O)CCC3CCCOC3)C2)=O)CC2(CC(CO)CO2)C1 47698,c1(C(=O)NCC(C)CNC(C23CCCN2CCC3)=O)ccc2c(c1)NC(=O)CC2 47699,c1(OC)ccc(C(N2CCCC2CN(C(=O)CC2CCCC2C)C)=O)cc1 47700,C1(NC(C(CCC)CNC(=O)C(C(C)(C)C)OC)=O)CC(C2CCCC2)C1 47701,C1(C)(C(N2CC(C(C)(C)O)(CNC(CCSCC)=O)C2)=O)CC2CC2C1 47702,C12(C(=O)NC3CC(CC(=O)NCC4CCCCC4O)C3)CCCC1C2(F)F 47703,CC1(C(=O)NC2C=CC(CC(=O)NCCc3ccncn3)C2)CCCOC1 47704,c1(OC)cc(CNc2cc(C(C)C)n(CC3CC3)n2)c2ccccc2n1 47705,C1(CNC(c2ccc(C3OCCO3)cc2)=O)CCN(c2ccccc2)S1(=O)=O 47706,C1(c2n(CC=C)nnn2)(NC(CC(N)=O)C2CC2)CNC(=O)C(C)(C)C1 47707,c1(C(N2C(C)CC(NC(c3nn[nH]c3Cl)=O)C2)=O)nccc2ncccc12 47708,c1(C(=O)NC2CC(NC(CN(C3CCC3)C)=O)C2)c(F)cccc1F 47709,c1(C(=O)OCC)cnc(NC)cc1C(=O)NCCSCc1ccc(F)cc1 47710,C1(CNC(C2CCC(CC)O2)=O)CCCN(C(=O)Cc2cncnc2O)CC1 47711,c1(C(=O)NC(CC)CNC(=O)CC2CCCOC2)cccc(N)c1C 47712,C1(F)(CNC(C2(C(C)C)CCC2)=O)CCN(C(C2CC(F)(CO)C2)=O)C1 47713,N1(C(C2(C)CC(C#N)C2)=O)CC23CCCC2(C1)CN(C(=O)CN1CC2CC2C1)C3 47714,C1(C#N)(C(N2CCCC(N(C(=O)C(O)C(F)F)C)CC2)=O)CC2CCC1CC2 47715,C12(CC(=O)NCC3CCC(C)S(=O)(=O)C3)CC3CC(C1)CC(Br)(C3)C2 47716,C(=O)(C(C#N)C(C)C)N1CCC(C(=O)NCc2c(C)scn2)C1 47717,C1(C#N)(C(=O)NC2CC(CNC(C(C)C(F)F)=O)C2)CC2CC2C1 47718,N1(C(C2(CSC)CC2)=O)CCC(CN(C)C(c2cc(C(C)=O)[nH]n2)=O)CC1 47719,CC1CC(C)C(C(=O)NC2CCC(CNC(c3n[nH]c(O)n3)=O)C2)O1 47720,N1(C(c2c(C#C)c[nH]n2)=O)CC(=O)NCC1C(=O)NC1CCCC12CC2 47721,S(=O)(=O)(c1c[nH]c2ccncc12)NCCN1CCCCC(C)C1 47722,N1(C(CCOCCCNC(C2CCCC(C)CC2)=O)=O)CC2(CCN(C)CC2)C1 47723,CN1CCC2CCC(C1)N2C(=O)C(c1cnn(C)c1)NC(=O)CC1CCCC1 47724,C(c1cc2ccccc2o1)=CC(=O)Nc1cc(-n2cccc2)ccc1F 47725,C(=O)(C(C)(C)S(C)(=O)=O)N(C1CCCN(C(=O)C(C)(C)COC)C1)CC 47726,C1(NC(C2(C)CC2(F)F)=O)CCC(NC(C2(F)CCC2)=O)CC1 47727,Cn1ccc2cccc(C(=O)NCC(O)CCNC(C3(C)CCCO3)=O)c12 47728,CCC(CC(=O)N1CC(F)CC1CO)NC(=O)C=Cc1cn(C)cn1 47729,CC1CCCN(C(=O)CC2CCCC2)C1CCNC(c1csc(C(C)(F)F)n1)=O 47730,c1(OC)ccc(-c2onc(C(=O)NC3CC(CNC(=O)CSC)C3)c2C)cc1 47731,c1(C(N2CC3C(CNC(c4c(C)n(C(C)C)nn4)=O)C3C2)=O)ccc(F)c(Cl)c1 47732,C(CC(C)CN=C(NC(C)C)N1CCC(NCC(F)(F)F)C1)OCC 47733,C(=O)(CC(C(F)(F)F)NC(c1sccc1F)=O)NCC1C(C(C)C)C1 47734,c1(C(C)C)oncc1C(=O)NCC1CCN(c2ccccc2)C1 47735,c1(C(=O)NC2(C(=O)NC(C=C)C3CC3)CC2C)cc(CO)[nH]n1 47736,CN1C(C)(C)C(NC(c2nnnn2Cc2ccccc2)(C)C2CC2)CS1(=O)=O 47737,N1(C(c2cc(C)n(C)n2)=O)CC2CCC1C(CNC(=O)C(C)(C)C(F)(F)F)C2 47738,C1(NC(c2cc(C3CC3)nc(Cl)c2)=O)CC1C1CCCN(C(C23CC2C3)=O)C1 47739,C1(C(N2CCC(CC(=O)N(CC(C)C)C(C)C)C2)=O)CC(=O)NC1=O 47740,C(=O)(CC(C)CN(C)C)N(CCOCCNC(c1c(C(C)C)cc[nH]1)=O)C 47741,c1(OC)ccc(CCNC(=O)C(=O)N(C2CC2)CC2(C)CCCC2)cc1C 47742,c1(C(=O)NCC2(F)CCN(C(C3CCCOC3)=O)CC2)cnc2ccnn2c1O 47743,C1(CNC(CCN(C)CC)=O)CC(CNC(=O)C(C)(C)SCc2cccs2)CO1 47744,N1(C(c2cn(C)nc2-c2ccnn2C)=O)CCCc2cc(OC(F)F)ccc21 47745,N1(C(c2c(C)n(C(C)C)cc2)=O)CC(N(C)C(c2cccc(N)c2)=O)C(C)(C)C1 47746,C(=O)(CCCCCF)N(C(C)C(=O)NC(C)(C)CCCO)CC 47747,C12(C(N3CCCC(NC(C(c4cccc(OC)c4)O)=O)C3)=O)CC(N=[N+]=[N-])C1C2 47748,C=CC(CC)CC(=O)NCCC1(C(=O)NCC2CCC(C(N)=O)O2)CCC1 47749,C(=O)(CS(=O)(=O)C1CC1)N(CCCCNC(C(C)=CC1CC1)=O)C 47750,C(CN=c1nc2cccc(Br)c2c[nH]1)C1CCN(C(c2c(C)noc2)=O)C1 47751,N1(C(C2(C=C)CCCC2)=O)CC(CO)C2(C1)CN(C(c1cnc(O)c(F)c1)=O)C2 47752,C1(NC(=O)C=C(Cl)Cl)CCCCCC1NC(C1CC2CCC(C1)C2)=O 47753,CCCCCC(=O)NCCCC(C)NC(c1ccnc(N2CCCCC2)n1)=O 47754,c1(NC(C2N(C(C(C)O)=O)CC2)=O)nc(Cl)ccc1F 47755,CC(C)C(CCN(C)C(c1csc(CO)n1)=O)NC(C1(O)CC1(C)C)=O 47756,CC(C)(C)CC(O)CC(=O)NC(CCF)C(=O)NCc1ccc(C(N)=O)o1 47757,C1(C(NNC(C=Cc2c(C)cccc2)=O)=O)C2CCCCCCC12 47758,C(=O)(C(C)CCCOC)NCCN(C(=O)CCC(C)CC)CCCCCC 47759,C1(c2nnnn2Cc2ccco2)(NC2CC=CCC2)CCC2(CCO2)CC1 47760,N1(C(CC2CC(CC)C2)=O)CCOC2CN(C(=O)COC(C)=O)CC12 47761,CC1COCC(C(=O)NCC(=O)NCC(N2CC(O)(c3cc[nH]n3)C2)=O)O1 47762,C(=O)(C1=CC2(CCOC2)C1)N(CC(C)C)CC(N1CC(CO)C(O)C1)=O 47763,c1(C(=O)NCC(CC=C)NC(=O)Cc2ccc(F)c(F)c2)onc2c1CCCC2 47764,CCC(C)CC(C)C(=O)NC1(CNC(=O)C(C)(C)Oc2cccc(Cl)c2)CC1 47765,C(CC(=O)N1CC(CC23CC(C2)C3)C1)(C(C)(C)C)N(c1ccnc(O)c1)C(C)=O 47766,c1(C(=O)NC2C3N(C(C(CCCC)O)=O)C(CC3)C2)cc2c(C)cccn2c1 47767,N1(C(CNC(CC)=O)=O)CCC(O)(CCNC(c2c[nH]nc2C)=O)CC1 47768,Cc1cc(OCC2CCCC2)ccc1NC(=O)NC1CCC2COC1O2 47769,c1(C(=O)NCC(F)CNC(c2cc[nH]c2)=O)cccn2cc(C(F)(F)F)nc12 47770,CC1CN(c2nnnn2CCC2CCCCC2)CCCO1 47771,Cc1cccc(C2CC2C(=O)Nc2cn[nH]c2)c1.N12CCC1CNCC2=O 47772,C(=O)(CCCCC(=O)NCC1CCCN(C2CCNC2=O)C1)NC 47773,N1(C(c2cnc(C)nc2C)=O)CC(NC(C2(Cl)CC2)=O)C(N=[N+]=[N-])C1 47774,c1(C(=O)NCC2(C)C(C)CN(C(c3cc(C#N)c[nH]3)=O)C2)cc2ncccn2n1 47775,c1(CC(=O)NC2CC3(CN(C(C(C=C)O)=O)C3)OC2)c[nH]c2ccc(Br)cc12 47776,N1(C(C(N2C(C3C(C)(O)CCCC3)CCC2)=O)=O)CCCc2ncc(F)cc21 47777,C=CCC(C)(C)CCNCc1ccc(-c2cc(Cl)ccc2Cl)o1 47778,C12(NC(C3(CC#C)CCN(C(c4c[nH]nc4C)=O)C3)=O)CC1COC2(C)C 47779,C1(NC(=O)CC(F)(F)F)CC2CC(NC(C3CCCC(F)(F)C3)=O)C1C2 47780,C12(NC(CNC(C)=O)=O)CCCN(C(=O)C(Cc3cccnc3)C3CCCC3)C1C2 47781,C1(Cc2oncn2)CNCC(C)(C)O1.c1(-n2c(C)ncn2)ccc(F)cc1F 47782,C1(CCCC)(C(N2CCC(C(C)NC(=O)CC)C2)=O)CCCC1.C1(C)C(=O)N1 47783,CC(c1cccnc1)=CC(=O)NCC1(CO)CCCO1 47784,C(=O)(C1=Cc2ccccc2C1)N1CC(C)(C)C(C(=O)N(CCCF)CCO)CC1 47785,C(=O)(CC1=CCCCC1)NC1(C)CCCN(C(c2cncc3nc[nH]c23)=O)C1 47786,C1(C(=O)NC(C(C)NC(=O)Cc2nnn(C(C)(C)C)n2)CO)CC12CCCCC2 47787,CC1(C(=O)NCc2ncccc2O)CCCN(C(C2CCOC2C2CC2)=O)C1 47788,C(=O)(C1=NOC(C)(C)C1)NCCCCCCN(C(C(CC#C)C1CC1)=O)C 47789,C(CC1=CCN(C(c2cc(C(C)(C)C)on2)=O)CC1)NC(c1n(C)c(Cl)cn1)=O 47790,C1(CC(n2cc(CCC3CC3)nn2)C)CCCCN1C(=O)Cn1nccn1 47791,c1(-c2cn(-c3cccc(C(CCCCOCC)=O)c3)nn2)ccc(S(C)=O)cc1 47792,c1(CC(N2C(CN(C)C(C3CC3(Cl)Cl)=O)CC(F)C2)=O)ccc2c(c1)COCC2 47793,C1(OC)CC2(CCN(C(=O)CCC3CC(NC(=O)Cn4nc(C)nc4C)C3)C2)C1 47794,c1(C(N(CC)CC2CCCCN2C(C2CC(F)(F)CS2)=O)=O)ccn2cncc2c1 47795,c1(C(=O)NCc2ccc(C(=O)NC(C)Cc3cccs3)o2)cccc(F)c1O 47796,CCCCC(CC)C(=O)N1CCCN(C(c2ccc(Cl)nc2O)=O)CCC1 47797,N1(C(CCC#CC)=O)CCC(NC(c2nn(C)c(Cl)c2C(F)(F)F)=O)C(C)C1 47798,O=C1CC(C2CC2)(C(=O)NC23CCC(NC(=O)C(O)C(F)(F)F)(CC2)C3)C1 47799,C1(C(=O)NCCOCC(=O)NCCCn2cccc2)(CO)CCCO1 47800,c1(C(N2CCn3ncc(I)c3C2)=O)cc(C(F)(F)F)nc2ccccc12 47801,C(=O)(C(F)(F)C(C)(C)O)NCC1(C(C)C)CC1.C1(C)C(=O)N1CCF 47802,C1(NC(CCCSC)=O)CCCC1(C)CNC(=O)CCc1cccc(C)c1 47803,n1(CC)cc(CC(=O)NCCCCCNC(c2cnn(C)c2N)=O)c(C)n1 47804,c1(CC)cccc(F)c1C(=O)NC(C)CNC(=O)C(C)Cc1cccc(Cl)c1 47805,N1(S(CC)(=O)=O)CCCC1C(=O)NCC(C)(CO)NC(C1CC(=C2CCC2)C1)=O 47806,c1(N2CCC(CCC)C2)nccc(=NCCC2CC(n3cc(Br)cn3)C2)[nH]1 47807,N1(C(C(C)C2CCCC2)=O)CC2CCN(C(=O)Cc3ccc(F)cc3Br)CC2C1 47808,C1(C(=O)NCC(CN(C(=O)CC2CCOC2=O)C)O)CCCC(C)(C)C1 47809,C1(C(=O)OC)C(C)OCCN1C(CCc1cccc(Cl)c1)C(=O)NCCC1CC1 47810,c1(NC(=O)NCC2N(C(c3c(COC)noc3)=O)CCC2)ccc(OCC)cc1Cl 47811,Cc1nc(C(=O)NCCn2cc(C(=O)NCC3(Cl)CC3(F)F)cn2)sc1C 47812,N#Cc1cc(C(=O)NCC2(NC(c3cn(C4CC4)nn3)=O)CCOC2)on1 47813,n1(CC#C)cccc(C(N2CCCC(CS(C)(=O)=O)C2)C(=O)NC(C)(C)C)c1=O 47814,Cc1nn(C)cc1-c1cn(CCCCC(=O)O)nn1.C(=O)(C(C(C)C)NS(N)(=O)=O)NCC 47815,C1(NC(COC)=O)CC(C(N2CCN(C(c3ocnc3C)=O)CC2)=O)C12CCC2 47816,C(=O)(CCC1=CCCCC1)NCC1(C)C(C)CN(C(c2ncn(CC)c2)=O)C1 47817,c1(C(C)(F)F)cccc(C(=O)NCC(CO)NC(c2cccn2C2CC2)=O)c1 47818,N1(C(c2ccc(C)[nH]2)=O)CCCCC(CCC(N2C3CCC2COC3)=O)C1 47819,C1(N(C(C2CC(C)N2C(=O)COC)=O)CC)CCCN(C(=O)C=CCOC)C1 47820,Cc1cc(Nc2cc(NC(C)CN3CCCCC3)ncn2)cc(C)c1 47821,c1(NC(C2CCCN(C(C3CC(=O)NCC3)=O)C2)=O)ccc(F)c(CO)c1 47822,C1(CCNC(c2ccccc2Cl)=O)CN(C(=O)C(F)(F)C2(O)CCC2)CCO1 47823,C1(NC(C(C)OCC=C)=O)(CF)CCN(C(c2ccccc2C(C)=O)=O)C1 47824,Cc1ccc(C(=O)NC2CC(N(C(=O)CCc3cscn3)C)C2)c(F)c1C 47825,C(CCN(C)C(C12CC(C1)C(C(F)(F)F)O2)=O)(C(C)C)NC(CC1CC(=C)C1)=O 47826,N1(c2nc(C)cc(C)n2)CCC2(CC1)CN(C(=O)CC1CC1C)C2 47827,N1(C(=O)CC2CCCC2)CCC(C2CCN(C(C3CC3C3CC3)=O)C2)CC1 47828,C1(C(N(C2CCCN(C(Cn3ncc(C)c3)=O)C2)C)=O)CCc2nc(C)nn2C1 47829,CC(CN=c1[nH]c(=NCC2CC(F)(F)C(=O)N2)[nH]c2c1CCC2)c1ncc[nH]1 47830,C1(NC(CNS(CC)(=O)=O)=O)CN(C(=O)C(n2nc(C)cc2C)C)CC1C(F)F 47831,C(=O)(CCC(=O)C(C)(C)C)NC1CCC(CCC(=O)NCC(N(C)C)C2CC2)C1 47832,Cc1ccccc1OCCC(=O)NC1CN(C(=O)C2=NOCC2)CC1C(F)(F)F 47833,C(=O)(C(CC(C)C)C(N)=O)NC1CCN(c2nnc(C(CC)(C)C)o2)CC1O 47834,c1(NC(C(=O)N(CCNC(C2CC(C#N)C2)=O)CC2CC2)=O)cc2c(s1)CCC2 47835,C=CCCC(CC(C)C)C(=O)NC1CN(C(=O)CCc2ncccc2C)CC1O 47836,CCCC(CCCO)C(=O)N1CCN(C(C2CCCN(C(C)=O)C2)=O)C(C)C1 47837,CN(S(N)(=O)=O)NC(C1CC(n2cc(CNCc3cncnc3)nn2)C1)=O 47838,CCCCCCC(C(=O)NC1(C)CCN(C(=O)C(C)(C)C2CC2)C1)NC(C)=O 47839,c1(C(N2CC3C(CNC(C=C(C)C(=O)O)=O)(C3)C2)=O)ccnc(Cl)c1C 47840,Cc1nc(F)ccc1-c1cccc(OCC(C)O)c1 47841,C1(SCC)CCCC(CNC(=O)CN(C)C(C)=O)C1.C12(CCCC1)C(=O)N2 47842,N1(C(C(C)(C)C2CCOCC2)=O)CC2CCCC(NC(c3cnsc3)=O)C2C1 47843,c1(C(=O)NCC23C(CN(C(c4cn(CC=C)nn4)=O)C2)C3)cccn2cnnc12 47844,CCC(C)C(C)C(=O)N1CC(O)(CNC(c2csc3nnsc23)=O)C1 47845,C(CC(C(=O)NOC(CO)C(C)C)NC(C1CC(C(C)C)C1)=O)=CC 47846,CCC(C(=O)NCC(CNC(=O)C=CCO)OC)Sc1nc(=N)[nH][nH]1 47847,N1(CC(C)(C)OCC2CCCCC2)CC(=O)N(Cc2ccc(C3CC3)o2)C1=O 47848,c1(CC)cc(N2CC(C3CC3)CC2C)n2ncc(Br)c2n1 47849,c1(CN(C(=O)C(CO)N(C(C)(C)C)C(c2ccn(CO)c2)=O)C)cccc(Cl)c1 47850,C1(C(=O)NCc2c(C)noc2)C2CCN(C(=O)CCC(C)CN(C)C)CC12 47851,C1(NC(N)=O)CC2CCC1C(NC(C(CC)N(C)CC)=O)C2.C12CC(C1)NC2=O 47852,C(C)(C(C)(C)NC(c1ccn(C(C)(C)C)c1)=O)NC(C1C(C)C1C)=O 47853,CC1CCN(CCC(=O)NCC2C(C)CCN2C(c2cc(C#N)on2)=O)CC1 47854,c1(OCC)cc(OC)ccc1NCCCC(C)C1CN(C(=O)OC(C)(C)C)C1 47855,CC(C)C(C)CC(=O)NCC1(C(C)(C)O)CN(C(=O)CC2OCCO2)C1 47856,C(c1ccc([N+](=O)[O-])s1)=CC(=O)N(C)CC1CCCCN1C(=O)C1=COCCC1 47857,Cc1oc(C(C)(C)C)cc1C(=O)NCC1CC1NC(c1cnoc1C(C)C)=O 47858,c1(C(=O)NCCCCCNC(Cc2cc(C)sc2)=O)coc2ccccc12 47859,N1(C(c2nn(C)c(C(N)=O)c2)=O)CCN(C(=O)Cc2ccsn2)C2CC12 47860,CCC(CC(=O)NC(CNC(=O)C(c1ccc(Cl)s1)C)CC)C(C)C 47861,N1(C(c2ccc(F)s2)C(=O)NC2CC2)CCCCC2(CCC2)C1 47862,C1(C(C)(C)C)CN(C(=O)C=CC2CCCO2)CCN1C(=O)C(Cl)=CCl 47863,CC(CNC(C1CCSCC1)=O)C(F)C(=O)N1CCC1(C)CCO 47864,c1(C(N2CCC(N(C(C3C(COC)C3)=O)C)C2)=O)cc(C2CC2)oc1C1CC1 47865,N1(C(C(C)(C)N2CCC2)=O)CCC(C2CCCN(C(C3CC3C(F)F)=O)C2)CC1 47866,c1(OC)cc(-c2cnc3cc(C(N4CCOCC4)=O)[nH]c3c2)cc([N+](=O)[O-])c1 47867,C1(CNCc2cccc(OCCCC)c2)CCCC1C1CC1 47868,C1(N(C(c2cc(CCC)[nH]n2)=O)C)CCCCC1N(C(=O)C=CC(C)C)C 47869,N1(C(C(CC(C)C)F)=O)CCC2CCC(C1)N2C(c1cccc(SCC#N)c1)=O 47870,N1(C(C=CCNC(C2C(C(=C)C)OCC2)=O)=O)CCc2ccc(F)cc21 47871,C(CC1c2ccccc2CCN1C(c1ccon1)=O)NC(=O)C(C1CC1)C1CC1 47872,CC1CN(C(c2cscc2C(F)F)=O)CC(CCNC(=O)C2=CCSC2)O1 47873,c1(C(N(CC(C)(C)CNC(=O)C(O)Cc2cnc[nH]2)C)=O)cc(C(F)F)ncn1 47874,C1(C(=O)NCC(NOC)=O)CN(C(=O)CNc2cccc(Cl)c2)CC12CCC2 47875,C1(CC)C(C(=O)N(CC(C)COC)C)CCN1C(=O)CC1CCCNC1=O 47876,c1(C(N2CCC(N(C)C(C3CNC(=O)N3)=O)C2)=O)ccccc1-c1cc[nH]n1 47877,C1(CN(C2CCC2)C(c2cocn2)=O)CCC(C(F)F)CC1 47878,Cc1ncc(C=CC(=O)NCC2CCCN2C(=O)C=CC(c2cnn(C)c2)=O)s1 47879,c1(C(=O)NCC2(C(=O)NCCCCO)CC2)ccc(N2CCOCC2)nc1 47880,C1(CNC(C=CC(C)(C)SC)=O)CCCN(C(C2(C)C=CCCC2)=O)C1 47881,CC(C)C(O)C(C)(C)C(=O)NCC1CCC(NC(=O)CSc2nnnn2C)CC1 47882,Cc1cc(C(=O)NCC2CCN(C(=O)C(C)n3cncn3)C2)cc(Br)c1C 47883,c1(NCCCC)ncnc(NCC(N2CCC(C(C)(C)CO)CC2)C(C)C)c1C 47884,C1(NC(c2ccc(OCCF)cc2)=O)CC2(C1)CN(C(C1CC1(F)F)=O)C2 47885,N1(C(C(C(C)C)C)=O)CCC(CNC(=O)CN2CCCS2(=O)=O)C12CC2 47886,C1(CNC(C2C3CNCC23)=O)CCN(C(=O)CCC2CCCC2)CC1 47887,c1(C(=O)OC(C)(C)C)cc(Cl)cc(Cl)c1Cl.C1(C(C)(C)C)C(=O)N1 47888,O=C1CNC(=O)N1CC(=O)NC12CC1CN(C(c1ccoc1C1CC1)=O)C2 47889,N1(C(CCC(=O)NC2C(=C)CC2)=O)CC2C(NC(=O)CCCSC3CC3)C2C1 47890,C1(NC(c2c(COC)cco2)=O)(CO)CCN(C(c2ccsc2SC)=O)C1 47891,c1(CCC(=O)NCC(C)N(C(c2nc(OCC)oc2)=O)C)c(C)noc1Cl 47892,c1(C(=O)NC2(CN=c3[nH]nc(C)s3)CCCCC2C)cnc2nncn2c1C 47893,N1(C(CSc2ccc(OC)cc2)=O)CCCC(C)C1CNC(c1ccncc1)=O 47894,CN1CCN(C(C2CCC(C(F)F)CC2)=O)CC1CNCc1ncc(F)cn1 47895,Cc1nccn1CCCC(=O)N1CCC1CC1(c2cn(C(C)C)nn2)CCCC1 47896,c1(C(=O)OCC)cnc(SC)nc1N1CC2CC1CN2Cc1ccc(I)o1 47897,Cc1ncc(NC(=O)C(C)(C)C2CCN(C(=O)C=CC3CCOC3)C2)c(C)c1C 47898,Cc1nc(NC2CN(C(c3c[nH]c4c(Cl)cccc34)=O)CC2C)c2sccc2n1 47899,c12cnc(C)c(c1)OC1CCN(C1)C2=O.C(=O)(COCC=C)NCC 47900,C1(NC(CN(C(C)C)C)=O)CCN(C(=O)C(C)(C)C2(C)CC2(F)F)C1 47901,N1(C(CCCC)=O)CC(NC(C2(F)CC2C)=O)CC2(CC2)C1 47902,N1(C(C(CC#C)O)=O)CC(NC(c2cc(Cl)ccc2NS(C)(=O)=O)=O)CC(F)C1 47903,c1(CCC(N2C(C(C)NC(C(C)=C3CCCC3)=O)CCC2)=O)ccc(N)c(F)c1 47904,CC(C)CC(CNC(C1CC1C1CCCC1)=O)C(=O)Nc1cc(O)cc(F)c1 47905,c1(OC)ccc(S(=O)(=O)N(c2cc(C3CC3)nn2C)C2CC3CCC2C3)cc1Cl 47906,c1(C(=O)NC2C(NC(=O)CSc3nc[nH]n3)C2)cc(F)cc(F)c1 47907,c1(N(CC(C)CNC(C2(CN(C)C)CC2)=O)C)cnc(C#N)cn1 47908,N1(CC(=O)NCC(CCOC)NC(C2CC23CC(O)C3)=O)CCCCCC1 47909,C1(NC(COCC(C)C)=O)CCN(C(C2CN(C3COC3)C2)=O)C(C)C1 47910,C(=O)(C(CC1CCC2CC12)N(CC(C)C(C)C)C1CC1)NC(CC)C 47911,C(=O)(CCCC(=O)N(CC(F)CC1CCCC1)CCN(C)C)OC(C)(C)C.O 47912,Cc1cc2ccc(C(N3CCN(C(c4ccsc4Cl)=O)CC(CO)C3)=O)cn2c1 47913,C=CC(C)CC(=O)N1CC2(NC(=O)CSc3ccccc3)CC1C2 47914,c1(CC)onc(C(N2CCC(NC(=O)CCc3cnn[nH]3)C2CC)=O)c1C 47915,c1(C(N(CCNC(C2C(C)C2C)=O)C2CC2)=O)cnc2ccc(F)cc2c1 47916,CC(C)CS(=O)(=O)CCC(=O)N1CC(CC(C)NC(=O)CCn2ccnn2)C1 47917,c1(C(=O)NC2(C)CN(C(C3(F)C(C)OCC3)=O)C2)cnc(O)c2cncn12 47918,N1(C(c2cn(C(C)C)nc2)=O)CCN(C(c2ccnc(C3CC3)c2)=O)C(CO)C1 47919,C1(NC(NCC(COc2ccc(CC)cc2)O)=NC)CCCCC1(C)C 47920,C1(NC(CN(C(=O)Cn2c(C)ccc2C)CC#C)=O)CCn2ncnc2C1 47921,c1(OCCNC(c2n(CCC)nnn2)c2cc(C3CC3)no2)cc(F)cc(F)c1 47922,N1(C(c2ccc(CC)[nH]2)=O)CC(C)(C)CC1C(=O)NCC1CCCN(C)C1 47923,c1(C(=O)NC2CC(NC(c3ncc[nH]c3=O)=O)C2)c(F)c(F)cc(F)c1F 47924,C(C(C)(C)CC(=O)N1CCC12CCC2)NC(C(C)=CC=C)=O 47925,c1(C(N2CCC(N(C(C3CN(C)C(=O)C3)=O)C)C2)=O)ccnc(Cl)c1O 47926,CCC(C)C(O)CNC(=O)COC(=O)CC1CCCS1(=O)=O 47927,N1(C(CCc2ccc(C)nc2)=O)CCN(C(=O)CC2CCCC2)C2CC12 47928,c1(C(=O)NC(CNC(c2n[nH]c(CC)c2Cl)=O)(C)CO)cc(F)cc(Cl)c1O 47929,CON(C)C(=O)CN=c1[nH]c(=NCc2cccc(C(N)=O)c2)[nH]c2c1SCC2 47930,C1(CC(=O)NCC2N(C(C(C)CC3CCCC3)=O)CCC2)COCCOC1 47931,c1(CC)c(C(=O)N(C)CC2(NC(=O)CCC#N)CC2)cnc2ncnn12 47932,c1(C(=O)NC2CCC(C)(CNC(C3(CCOC)CC3)=O)C2)nn(C)c(C)c1Cl 47933,C1(CNC(c2c(CC)ocn2)=O)C(C2CC2)CCN1C(c1cnn(C2CC2)c1)=O 47934,C=CCCC(F)(F)C(=O)N1CC(NC(=O)CC(C)(C)C(F)F)C2CC2C1 47935,N1(C(Cc2n(C)ncc2)=O)CCC(C(=O)N(CCCO)CCCO)CC1(C)C 47936,C1(CCC)CN(C(=O)Cc2occc2C)CC1NC(=O)C(C)CNC(C)=O 47937,C(CNC(C1CCNC1=O)=O)(CC(=O)N1CC(F)(CF)C1)OC 47938,N1(C(C2CC(SC)C2)=O)CCC(C(C)(C)NC(C2CC(C)C2)=O)C1 47939,c1(NC(C2OCCN(C(C(C=C)O)=O)C2)C)ncc(C)c(C)n1 47940,C1(CNC(CCCCC)=O)CCC(C)CN1C(c1ccc(Cn2cccn2)o1)=O 47941,C1(NC(CCC#CC)=O)CCCCN(C(=O)CCCNC(C)=O)C1 47942,C1(CNC(c2conc2C(F)F)=O)CN(C(c2n[nH]cc2Cl)=O)CC1O 47943,C(=O)(CC(C)(C)N(C)C)NCC(CC=C)NC(=O)Cn1cc(Br)c(C)n1 47944,Cc1cc(C(C)C)ccc1C(=O)NC(C1CCN(C(=O)CC2CCOC2)CC1)C 47945,C1(CC)C(NC(c2ccc(COC)o2)=O)CCCN1C(C1CCOC1CC)=O 47946,c1(C(=O)NC(CN(C(c2cc3cnccc3[nH]2)=O)CC)C)cnn2cccnc12 47947,N1(CC)CCOC(C(N2CCCC(CNC(c3ncoc3C(C)(C)C)=O)C2)=O)C1 47948,Cc1cc2ncc(C(=O)NCCC3CC(NC(C4(C)CC4(Cl)Cl)=O)C3)c(C)n2n1 47949,CC1(C(=O)NOCc2cccc(F)c2)CCN(C(c2nccnc2N)=O)CC1 47950,C(=O)(C1=CCC(C)(C)CC1)NC(CC#C)C(=O)NC1(C)CCC(C)(C)C1 47951,C=C(Cl)CC(C(=O)NC1CC(C)(O)C1)NC(c1cc(Cl)cn1C)=O 47952,N1(C(c2ncn(C)n2)=O)CC2CCCC(C1)N2C(=O)CC=C(Cl)Cl 47953,CCC(C)C(C(=O)NCc1cnn(C)c1O)N(C(=O)C#CC(C)(C)C)C 47954,Cc1ccc2c(C(=O)NC(C3CCN(C(C4CC4C)=O)C3)(C)C)c[nH]c2c1 47955,C1(NC(C2N(CC)C(=O)CC2)=O)CCC12CN(C(c1cnc(S)[nH]1)=O)C2 47956,N1(c2sc(C#N)c(Cl)n2)CCc2sc(C(=O)NCCCOC(=N)O)cc2C1 47957,CC(C)CCCCC(=O)NCC=CC(=O)NC(C1CCOCC1)C 47958,N1(C(c2c(C)cccc2F)=O)CC(NC(=O)C=CC2CCCO2)CC2(CCC2)C1 47959,c1(C(N2CCN(CC(C)NC(C(CC)C(C)C)=O)CC2)=O)cc2oc(C)cc2[nH]1 47960,C1(C(=O)NC(C=C)C2CC2)CCC(C)(C)N(C(=O)CCC(C)CN(C)C)C1 47961,CCC(C(=O)N1CC(N2CCCC2)C1)NC(=O)COC1CCCC1 47962,N1(C(=O)CNC(c2cccs2)=O)CCC2(NC(=O)Nc3cccc(Cl)c3)CC2C1 47963,c1(N(CC(CC)C)C)nnc(-c2nc(C)c[nH]2)n1CCC(=O)N(C)C 47964,N1(C(C(=O)N(CC(=C)C)C)C)CCOC(C(=O)OC)C1 47965,c1(C(C)O)ccc(C(=O)NCCC2CN(C(=O)COCP(C)(C)=O)CCO2)cc1 47966,N1(C(c2ccc(C)cc2)=O)CC(C)CCC1CNC(=O)Cc1cc[nH]c1 47967,C1(C(=O)NC2C(NC(COc3cc(C)on3)=O)C2)CCc2c(nnn2C)C1 47968,C(C(N=c1ccnc(NCCCn2cccn2)[nH]1)C1CCCO1)SC 47969,C1(NC(C(C2CCC2)SC)=O)CC(C)(NC(=O)CCC=CC(C)C)C1 47970,CCC(CN=c1ccc(Br)c(S(=O)(=O)N2CCC2c2cc(C)cc(C)c2)[nH]1)OC 47971,C(=O)(C(O)C1=CCCCC1)N(CCN(C(c1c(C)nc(CCC)s1)=O)C)C 47972,c1(C(C)C)ncc(C(N2CCN(C(=O)C=CC(C)(C)C)CC2)=O)cn1 47973,CCCC(CCCNC(=O)COc1ccsc1)NC(=O)C=Cc1c(C)coc1C 47974,N1(C(CC2C=C(C)CS2)=O)CCC(NC(C2CCCCS2)=O)C1c1ccccc1 47975,CC(C)CC(O)CC(=O)NC(c1nocc1C(N1CCC(N2CCC2)C1)=O)C 47976,CC1CCC(c2nnnn2C2COC2)(NCc2cscn2)C1 47977,c1(C(=O)NC2CCN(C(C=C(C)C(C)(C)C)=O)C2C)cc2cccc(C)n2n1 47978,c1(CC(N2C3(CNC(=O)CCC4OCCO4)CCC3CC2)=O)cc(F)c(F)cc1F 47979,n1(CC(=O)NC2C(C)N(C(=O)C=CC3CC3)CC2)sc(=O)c2ccccc12 47980,c1(-n2c(C)nnn2)cc(C(=O)NCCCNC(=O)CSC2CC2)ccc1Cl 47981,N1(C(C2CC(C#N)(OC)C2)=O)CC(C(=O)N(CCC(F)(F)F)C)OC(C)C1 47982,C1(CC(C)C)CCN(C(C2CCN(C(=O)CCc3cn(C)cn3)C2)=O)C1 47983,C1(NC(C2(CCC=C)CN(C(c3cc[nH]c3)=O)C2)=O)CCn2cncc2C1 47984,c1(C(N(C2CCN(C(c3c(COC)cc[nH]3)=O)C2)C)=O)cncnc1O 47985,C1(NC(C(CSC)O)=O)COC2(C1)CN(C(c1cnc(OCC3CC3)cn1)=O)C2 47986,c1(C(=O)NC2CCN(C(c3c(C)nc(C)o3)=O)CC2O)c(C)nc2sc(C)nn12 47987,N1(C(C2(C)CN(C(=O)C(F)C3CCCC3)C2)=O)CCCC2C(=O)NCC12 47988,c1(C(N2CC=CC(NC(=O)CCc3cnccn3)C2)=O)cc2c(s1)CCOC2 47989,C1(CCC(=O)OC)(NCN2CCC2(C)C2CCCCC2)CCNCC1 47990,C(=O)(C(F)C(C)CNC(c1ccc(O)cc1)=O)N(CC(C1CC1)OC)C 47991,C12(CNC(CCOC)=O)CCC1CCN2C(=O)C(=Cc1ccco1)C 47992,C(=O)(CC(O)C(C)(C)C)N1CCC(NC(Cn2c(C)ccn2)=O)C1C 47993,N1(C(C2N(CC)CCC2)=O)CCC(C)(CNC(c2sncc2C)=O)C1 47994,C1(CCOC)(NC(=O)CCC2CC2)CCN(CC=C(Cl)Cl)CC1 47995,c1(OC)ccc(CN2CCC2C(N2CCOC(C3(O)CC3)C2)=O)cc1 47996,c1(C(=O)NC2CCC(CNC(CC(C)c3cccnc3)=O)C2)c(SC)cnn1C 47997,C1(C(=O)NC2CC(NC(=O)COc3cccc(Cl)n3)C2)CCN(CCO)C(=O)C1 47998,C(CC(O)CC(=O)N(C)CCN(C(=O)C(C)(F)CC)C)SC 47999,[N-]=[N+]=Nc1ccnc(NC(=O)CNC23CCC2CCN3NC(=O)CCCCO)c1 48000,c1(CN2C(C(N3CCC(CCCO)CC3)=O)CC(F)C2)cnc2ncccn12 48001,Cc1nc2ccc(C(=O)NC3CC(CNC(=O)CC4CCCC4)C3)cn2n1 48002,C(C)(CNC(c1ccn(C)c1)=O)(CC(C)C)NC(Cc1nc(C(C)OC)sc1)=O 48003,N1(C(C2CC(=C)CN2C(=O)Cc2cc(Br)ccc2Br)=O)CCC(O)C(C)(CO)C1 48004,c1(CC)nc(C)oc1C(N1CC2C(N(C(=O)C(CC)SC)C)C2C1)=O 48005,Cc1cc2c(C(N3CCC(CNC(=O)CSC(F)F)CC3)=O)cccc2[nH]1 48006,C1(C)(C(=O)NC2CCN(CCC)C2)CCCN(c2cc[nH]c(=N)c2)C1 48007,c1(N2CC(CNC(C(CC)N(C)C)=O)OCC2)cc(C)c([N+](=O)[O-])cn1 48008,n1(CCOCC)c(N2CCOC(C)C2)nnc1C1(OC)CC1 48009,Cc1nc(C(=O)NCC(C)(C)CN(C)C(C2CCSC(C)C2)=O)cn1C 48010,CC1(F)CN(C(c2cccc([N+](=O)[O-])c2)=O)CCN(C(c2cccc(=O)o2)=O)C1 48011,C1(CC=O)C(=O)N(C)C(C)(C(=O)NCCOC(F)F)C1CC 48012,Cc1ncc(N)cc1C(=O)NC1COCC1NC(=O)Cc1cc(C2CC2)nn1C 48013,Cc1cccc(Br)c1S(=O)(=O)NCCCc1ccc([N+](=O)[O-])cc1 48014,CN1C(C(=O)NC2CC(C)(NC(=O)CC(C)(C)C#N)C2)CCS1(=O)=O 48015,c1(OCC#C)ccc(Oc2ccc(CN3CC=C(Br)CC3)cc2)cc1 48016,Cc1nsc(C)c1C(=O)NCC1CC(NC(C2CC2c2ccn(C)n2)=O)CC1O 48017,C(CC(=O)NCCS(C)(=N)=O)(C(F)F)NC(Cc1cc(C)n(C)n1)=O 48018,C1(O)(CCNC(C2(CC=C)CCOC2)=O)CCN(C(=O)Cn2ncc(Cl)c2C)C1 48019,c1(CC2CC(F)(F)C2)nc(-c2ccccn2)nn1-c1ccnc(F)c1 48020,C(=O)(C(F)(F)CC(C)C)NC1(COC)CCN(C(=O)Cn2cc(Cl)cn2)C1 48021,C1(CN(C)C(C2CCN(c3ncccn3)C2)=O)CCCOC1 48022,C(CS(=O)(=O)CC(=O)NCCCC1CCCCN1C(C1CC(F)C(=O)N1)=O)OC 48023,N1(C(C2C(CC)C2)=O)CC(CNC(c2cccc(CC)c2N)=O)CC12CCC2 48024,c1(CN(C)C)cnc(O)cc1C(F)(F)F.C12CC(C1)NC2=O 48025,C(C(C)(C(=O)NCC(C)O)OC)OC.C1(CCOCC(=O)NCCS)CCCO1 48026,N1(C(C2(C)C(C)OCC2)=O)CC(C2(NC(c3cnnn3C)=O)CC2)C1 48027,C1(C(N2CC3(CC(NC(CNC(CCC)=O)=O)C3)C2)=O)CC(C(C)=NO)C1(C)C 48028,CCC1=NOC(C(=O)N(CC(C)NC(c2cccc(C(C)(F)F)n2)=O)CC)C1 48029,N1(C(C(C2CCOCC2)C)=O)CCC(C)(C(=O)Nc2cccc(CO)c2)C1 48030,Cc1nc(CN2CCC(C(C)NC(c3cn(C)nn3)=O)CC2)c(C)s1 48031,C1(OCC)CN2CC1C2=O.c1(NC(=O)CC2(OC)CC2)cnccc1C 48032,c1(CC(C)C)c[nH]c(C(=O)N(C)CCN(C(=O)CC2C=CCC2)C)c1 48033,c1(C(N(C(C)CCNC(C2(F)CCCC2)=O)C)=O)cc(C2CC2)nc(O)c1 48034,O=C(C(O)C1=CCCCC1)NCC1CCN1C(=O)Cc1ccc(C(F)F)cc1 48035,CCCC(O)CC(=O)NCC(C1CCCC1)NC(=O)C(c1cccc(F)c1)C 48036,Cc1ncncc1C(N1CC(NC(C2OCCC2C)=O)C(C)C1)=O 48037,C(N=c1[nH]c(N2CC(C(F)F)C3(CCC3)C2)nc2c1COC2)c1c(C)cncc1 48038,c1(C(=O)NC(CC=C)CNC(=O)CCC=C=C)c(C)[nH]c2ccc(OC)cc12 48039,c1(CCC)c(C(N2CCC(NC(=O)C(C)C(=O)OC)C2)=O)cnn1C 48040,c1(C(C)NC(C(C)n2ccnc2)=O)ccc(N2CCCC2)cc1 48041,CC1CCCN(C(=O)C=CC(C)(C)NC(C23CC2CNC3=O)=O)C1CO 48042,N1(c2cc(Nc3cc(C(=O)OC)cc(F)c3)ncn2)CCCC(C)(C#N)C1 48043,C(CCCCC(=O)NC(CC)C(C)(C)O)NC(C1N(C(C)=O)CCC1)=O 48044,N1(C(CN(CCC)C)=O)CC(C)C(NC(c2nccc3occc23)=O)C(C)C1 48045,N1(C(C(CC)C2CCOCC2)=O)CCN(C(=O)CCCCCSC)CC2(CC2)C1 48046,N1(C(C2(C)COC2)=O)CCc2c(C(=O)Nc3cc(Br)cc(Cl)c3O)n[nH]c2C1 48047,Cc1cc(F)sc1C(=O)NCc1cccc(CN(C)C(c2nnn(C)c2N)=O)c1 48048,C1(CC(N2CC(CCNC(=O)CCn3cccc3)OCC2)=O)CCCCCCC1 48049,N#Cc1cn(CC(=O)NC2CN(C(C3NC(=O)C4CC34)=O)C2)c(=O)nc1O 48050,c1(C(=O)NC(CN(C(C)C)C)C)ccccc1NC(=O)C(C)NC(N)=O 48051,C1(CC)(Nc2nn(C)c(C)c2Cl)CCN(C(c2ncc(I)cn2)=O)CC1 48052,C1(NC(CC(c2ccc(F)cc2)C)=O)CCCN(C(C2COC2)=O)CC1 48053,c1(C(N2CCC(C(=O)OC)(OC)C2)=O)ccc(Cl)nc1Cl 48054,C(=O)(CCCCCN(C)C)NC1CC(F)(CNC(c2ccnc(CC(C)C)n2)=O)C1 48055,Fc1cccc2c1OCC2NCc1ncc[nH]1 48056,c1(C(N(CCC(C)NC(C(C(C)C)O)=O)C)=O)ccc(F)c(C#N)c1 48057,c1(OCC)ncc(C(N2CC(C(C)NC(c3cscc3C(N)=O)=O)C2)=O)s1 48058,Cc1ccc(C(=O)NC(c2ccccc2)CNC(=O)CCOCC(C)C)nc1O 48059,c1(C(=O)NCC(N(C(CC=C=C)=O)C)C2CC2)cccc2c1OCCN2 48060,C1(CNC(C2CC(CC)OCC2)=O)CC2CCC1N2C(C1CNC(=O)N1)=O 48061,N1(C(C(=O)NCCSC)CC2C=CCC2)CCOC2CCN(C)CC12 48062,c1(COC)ncsc1C(N1CCCC1CNC(=O)C(C1CC(F)(F)C1)OCC)=O 48063,C1(NC(c2ccnn2C2CCC2)=O)CCN(C(=O)CN2CCCC2)C(C2CC2)C1 48064,CC1CC(C(=O)NC2CCCCC2NC(=O)CN(C2CCC2)C)CN1C 48065,C(=O)(C(O)C(F)(F)F)NCCC(CNC(c1n(CC)ncc1)=O)O 48066,N1(C(C2C3CC(NC(C(C(C)(F)F)(C)C)=O)C(C3)C2)=O)CCCC12CCOCC2 48067,c1(CCC(=O)NC(CN(C(C2(C)CC2(F)F)=O)CC)C)ccc(C(=O)N(C)C)cc1 48068,c1(CCC)ccc(C(c2nnnn2C2CC2)NCC2CCCOCC2)cc1 48069,C1(C(=O)NCCCC(C)NC(C(C2CCCCC2)OC)=O)CN2CCCN1CC2 48070,C12(N(c3ccccc3)C(=O)CCN(C)C)C(OC)CC1NC2=O.C(C)(C)(C)OC 48071,c1(C(=O)NC(C(CO)NC(C(CSC)C)=O)C)ccc(Br)c(SC)c1 48072,C1(C(=O)NCCCCN(C(C(C)C#N)=O)C)CCn2cncc2C1 48073,N(C(=NCCN1CCCCC1)NC1CCCC1)CC(c1ccccc1F)O 48074,c1(C(C)N(C)C(C2(C(C)(C)C)CCNC2)=O)ccc(F)cc1 48075,Cc1ncc2cc(C(N3CC4CC(NC(=O)CCc5csnn5)C3C4)=O)ccn12 48076,C1(C2CC2)(CNC(C(N2CCC(C)CC2)=O)=O)CCN(C(C2(Cl)CC2)=O)C1 48077,C1(CNC(C2C(CCC)CCC2)=O)CN(C(=O)C=Cc2cnc(C)s2)CCCO1 48078,c1(CC(=O)NCC(CC)(C)NC(=O)CCC=CC(C)C)ccc(OC)cc1C 48079,N1(C(CCC(=O)NC)=O)CCOC2CN(C(c3cnc4cccc(C)n34)=O)CC12 48080,c1(C(=O)NCC2OCC(CNC(CCC)=O)C2)cc2cccc(Br)c2cn1 48081,N1(C(c2cc(C)[nH]n2)=O)CC2C3CCC(C2C1)N(c1nc(Cl)ncc1C(N)=O)C3 48082,c1(NC(=O)Cc2cncnc2)ccc2c(c1)CN(C(C1CC(=O)N1)=O)C2 48083,C1(C)(C(=O)NC2CC(CNC(C3(OC)CCC(C)C3)=O)C2)C(C)(C)C1(C)C 48084,Cc1cccc(CC(=O)N(C2CCC(NC(=O)Cc3nccn3C)C2)C)c1 48085,C(=O)(C(F)CC(C)(C)NC(c1cc(C)n(C)c1C)=O)NC(C(=O)OCC)C1CC1 48086,C(=O)(C(CC(C)C)C(C)C)NC1CC2(C(C(N(CCOCC)C)=O)C2)C1 48087,C1(CC(=O)NC(CNC(C(c2cnn(C)c2)C)=O)(C)C2CC2)CNC(=O)C1 48088,c1(C(=O)NC2CCC(n3cc(COC)nn3)CC2)c(F)ccc(SC)c1F 48089,N1(C(CCC(=C)C)=O)CCC(NC(=O)CN2CCC(C(N)=O)CC2)CC1C1CC1 48090,c1(C2C3CN(C(C4(COC)CCC4)=O)CC32)cccc(OC2COCC2CO)c1 48091,C1(CCC#C)CCCN1C(=O)C(Cc1cc[nH]n1)NC(C1CC(N(C)C)C1)=O 48092,Cc1nc(S)nc(C)c1CCC(=O)NCCN(C(C1CCN(C)C1=O)=O)CC1CC1 48093,C1(C2CCOCC2)(NC(N(CCC(F)(F)F)CC)=O)CC1 48094,c1(NCc2cnc(CC)s2)ccc2c(c1)CN(C(c1cnc(C)c(C)c1)=O)C2 48095,N1(C(=O)OC(C)(C)C)CC2CC(NCc3ccn(C4CCCCC4)n3)C(C2)C1 48096,N1(C(C)=O)CS(=O)(=O)CC1C(=O)NCC1CN(C(=O)Cc2cn3ccsc3n2)C1 48097,c1(NC(CN(C)C)C(=O)NCC2(N(C)C)COC2)ccncc1[N+](=O)[O-] 48098,N1(C(CCOC)=O)CCC2CCN(C(C3CN4CCN3CC4)=O)CC12 48099,c1(CC)nn(C)c(C(=O)NCC2CN(C(c3ccc(SC)o3)=O)CCC2C)c1Cl 48100,C1(C(=O)NCC(CNC(C(C=C)(C)C)=O)C)CC(C2CCOCC2)=NO1 48101,c1(C(=O)OC)cc(=NCC2CCC(NC(c3cc(C(C)(C)C)on3)=O)C2)[nH]cn1 48102,C1(CNC(C2CCCC2O)=O)CC2CCCCC2N1C(c1ncc(F)cn1)=O 48103,c1(NC(c2n(C(CC)(C)C)nnn2)C2CC2(C)C)ccc(F)c(SC)c1 48104,C(CCCCCCC(=O)N(CCNC(c1cnccc1Cl)=O)CC1CC1)SC 48105,CCC(CC)C(=O)NCC1CN(C(c2coc(CN3CCCCC3)n2)=O)CCO1 48106,C#CC1(C(N(C)C[Si](C)(C)C)=O)CCN(C(=O)CCn2cncn2)C1 48107,N1(C(C2(CC)CCCCO2)=O)CC(NC(=O)CCCC2CCCC2)CC(F)C1 48108,N1(C(C2CC3CC3C2)=O)CC=C(CC(=O)N2CCC3CC23)CC1 48109,c1(C(C=CC)O)nnc(N2CCN(C(c3cccs3)=O)CC2)n1CC(C)C 48110,c1(C(=O)NCC2N(C(C(=O)NC(CC)C)C)CCC2)ccn2ccnc2c1 48111,C1(C(C(=O)N(CCCC)C2CC2)C)CCCN(C(=O)C(OC)OC)C1 48112,c1(C(N2C(C(=O)NC(CCC=C)C(=O)OC)CC3CC32)=O)ccc2c(c1)OCCO2 48113,c1(C(N2CC(NC(C(C3CCC3)OC)=O)C(F)C2)=O)cc(N)ccc1SC 48114,C1(OC)(CO)CCN(C(C2CCOC2(C)C)C(=O)NCc2ccc(C)o2)CC1 48115,c1(C(N2CC(NC(C3C(C)C3C)=O)C3(C2)CC3)=O)cc2cc(F)ccc2[nH]c1=O 48116,c1(C(C2(C)CC2)NC(c2ccccc2)=O)cc(F)c(C(=O)O)c(F)c1 48117,CCCCC(O)C(C)C(=O)NCCC1CCCCN1C(c1cccn1C1CC1)=O 48118,Cc1cc(CC(=O)NC(C)C(C)(C)NC(=O)Cc2csc(Cl)c2)n[nH]1 48119,N1(C(c2cccc(CC)n2)=O)CCC2C(CCCN2C(=O)Cc2cn[nH]c2)C1 48120,N1(C(c2ccn(CCNC(CCN(CCC)C)=O)c2)=O)CCC12CCC(C)CC2 48121,C1(F)(CNC(c2n(CCC)ncc2)=O)CCN(C(C2CC3CC3CC2C)=O)CC1 48122,c1(CC)nc(=N)[nH]c(=NCCCCN(C2CC(c3ccccc3)(OC)C2)C)[nH]1 48123,N1(C(C(C)n2ccnn2)=O)CC2(CCC(CNC(=O)CCF)O2)C1 48124,C(=O)(C1CCCc2nnn(C)c21)N(CCCNC(=O)CCCN(C)C)CC 48125,C1(C(=O)NCc2ccccc2)CCC(NC2C(CCNC(C(CC)C)=O)C2)CC1 48126,C(=O)(C1=NOC(C)C1C)NC1C(OC)CN(C(=O)CCCC2CCCCC2)C1 48127,c1(C(=O)NCC2C(NC(=O)C=CC3CCCCCC3)C2)ccc2nnn(O)c2c1 48128,C1(C(=O)NCC(C)(C)NC(C2(F)C3CCCCC23)=O)CC2(C1)CC21CCC1 48129,CC(CN(C(=O)C(Cn1cccn1)NC(=O)COc1ccccc1)C)C(F)(F)F 48130,C1(C(N(C(C)CN(C)C(c2cnncc2O)=O)C)=O)CN(C)CCN(C)C1 48131,CC1=C(C(=O)NC2(CC(=O)NCC3OC(=O)NC3(C)C)CC2)CCCO1 48132,Cc1nc(Cl)nc(N2CCCC(C(C)NC(=O)C=Cc3ccncc3)C2)c1F 48133,CCS(=O)(=O)CC(=O)N1CCOC(C(=O)NCC2(C)CC=CCC2)C1 48134,C1(CC(=O)NCCC2CCN(C(=O)CN3CCCC3)C2)CCC2(CC1)OCCO2 48135,Cn1cncc1C=CC(=O)NCCN(C(C1CC1c1cccnc1)=O)C1CC1 48136,C(=O)(C1CCS(=O)(=O)c2ccccc21)NCC(CNC(Cc1ccc(C)s1)=O)C 48137,Cc1nccc(C(=O)NC2CCCCC2NC(c2cc(C(F)F)ccn2)=O)n1 48138,N1(C(C(=O)NCC2(C)CN(CC)C2=O)=O)C(=O)CCC(N(C)CCO)C1=O 48139,c1(C(=O)NC2C(NC(C(C)(C)n3ccnn3)=O)C2)cc(F)c(Cl)cc1Cl 48140,N1(C(CC(C)c2cccnc2)=O)CC2CC2(CNC(=O)CN(C)C(N)=O)C1 48141,CCCCC(CC)CC(=O)NCC1CCC2CN(C(c3ncc[nH]3)=O)CCC2C1 48142,C1(O)(C(C)NC(=O)C=CCOC2CCCC2)CN(C(=O)CCC2CC2(Cl)Cl)C1 48143,CC(C)C(O)C(=O)NC(C)CCNC(=O)CCC1CCCC1 48144,C(C)(CCC(=O)N(CCCNC(=O)Cn1nc(C)cc1C)C1CC1)SC 48145,C(C(CC(C)C)C(=O)N1CCN(C(c2ccns2)=O)CC1C(F)F)OC 48146,C1(O)(CNC(c2nc(CNC(CS(=O)(=O)NC)=O)oc2)=O)CC2CCC1O2 48147,C12(NC(=O)CSCc3ccncc3)CCCN(c3ccn4ccnc4n3)CC1C2 48148,Cc1cccc(CN(C2CCN(C(c3cc(C(N)=O)ccc3F)=O)C2)C)c1C 48149,n1(CC(=O)NC2C(SC)CN(C(C3(CO)CCCC3)=O)C2)nc(C)c(Cl)c1C 48150,CC1CC(C(N2CCCCC2c2nncs2)C(=O)NC2CCOCC2)CC(C)C1 48151,Cc1nc(O)c(C(=O)NCC23CC2CN(C(C2(CO)CC2)=O)C3)c(C)c1[N+](=O)[O-] 48152,N1(C(CNS(NC)(=O)=O)=O)CCCC2CCN(C(c3nocc3C)=O)CC12 48153,c1(C(N2CC(C)(NC(C(C)c3ccsn3)=O)C2)=O)ccc(C(F)F)nc1 48154,c1(C(=O)Nc2scc(COC)n2)cc(Br)cnc1C(F)(F)F 48155,C1(NC(=NCCC=C)NCC2(C3CCC3)CC2)CCOC2(CCOCC2)C1 48156,N1(C(CCC(=C)C)=O)CC(CNC(=O)CC(Br)(Cl)Cl)CC12CCOCC2 48157,Oc1nc2ccccc2cc1NCCN1CCCC1 48158,N1(C(C(N2CC(C)CC(C)C2)=O)=O)CCn2c(cnc2C(N2CCOCC2)=O)C1 48159,N1(CCC)C(=O)CCC1C(=O)NC(CNC(=O)C=C1CCSCC1)C1CCC1 48160,CCC1(C(=O)NCC(O)CN(C(=O)Cc2cscn2)C)CCCc2ccccc21 48161,Cc1nn(CC(=O)NCC2CCC3(CN(C(=O)C(C)CF)C3)O2)c2ncccc12 48162,C1(C(=O)NC2C(CNC(c3cnoc3-c3ccoc3)=O)CC2)CC2(C1)CC2(F)F 48163,c1(C(=O)NCC(CNC(C(C(C)(C)C)SC)=O)F)cc(Cl)c2n[nH]cc2c1 48164,Cc1cc(Cl)cc(C(N2CCOC(CN(C)C(c3ccc(F)s3)=O)C2)=O)c1N 48165,CC1CCC1C(=O)NC(C(=O)NC1CC(CCC(N)=O)C1)C1CCCC1 48166,c1(C(=O)NCC23C(CN(C(C(C(C)C)NC(C)=O)=O)C2)C3)ccc(Br)c(C)n1 48167,CCCCCC(C)(C)C(=O)NC(CC(=O)NC1CCn2ccnc2C1)CC(C)C 48168,c1(CC)cc(Br)cc(C(=O)NCC2CCN(C(=O)CCC(F)F)C2)c1N 48169,c1(C(C(=O)NC(CC)CC2CC2)C)ccc(F)cc1Br 48170,Cc1ccc(CC(=O)NC(C2CN(C(C3CC3(C)C)=O)C2)C)cc1Cl 48171,C1(C(=O)OC)CCCC1NC(=O)NCCNC(c1scnc1C)=O 48172,Cc1cccnc1C(=O)N(CC(O)CN(C)C(c1cc(CC(C)C)nn1C)=O)C 48173,CC1(C(=O)Nc2cc(O)ncn2)CCN(C(c2ccccc2C2CC2)=O)CC1 48174,C1(C(N2CCC(CO)CC2)=O)CC2CC2N1Cc1cccc(-c2ccccn2)c1 48175,c1(C(=O)NC(C)CN(C)C(c2ccns2)=O)cc(S(=O)(=O)N(C)C)oc1C 48176,C1(CNC(CSC(C)C)=O)CC(F)(CNC(C2(CF)CCC2)=O)C1 48177,N1(C(C(C)(C)C)=O)CCCC(F)(CNC(c2cccc(C3CC3)c2Cl)=O)C1 48178,c1(CC(=O)NCCCNC(=O)CC2CCC2C2CC2)c(Cl)cccc1Cl 48179,c1(C(=O)NC(C2CCCN(C(C3=C(C)OCC3)=O)C2)C)cc2c([nH]1)CCOC2 48180,N1(C(c2nc(COC)oc2)=O)CCC2CCN(C(=O)C(=O)NC3CC3)C2C1 48181,C(=O)(CS(=O)(=O)CC1CCCO1)NC(CCCNC(CC1CC(OC)C1)=O)(C)C 48182,C1(C=C)(C(N(CCN2CCCC2)CC)=O)CCN(CCSc2ccsc2)CC1 48183,c1(CN(C(C2CC(=O)C2)=O)C2CC2)c(F)cccc1F 48184,N1(C(=O)CN2CC3CC3C2)CC2CCCN(C(C3CCC(F)C3)=O)C2C1 48185,CN1CC(C(=O)NCC2CC2CNC(C2(C(F)F)CC(F)(F)C2)=O)NC1=O 48186,C(C(=O)NNc1ccc(S(=O)(=O)N(C)C)cc1)(C(C)(C)C)n1cc(COCC)nn1 48187,C12(C(N(C3CC(C)OCC3)C)=O)CCC(CC1)N(C(c1cncc(O)c1)=O)C2 48188,N1(C(C2C(C)CCC2)=O)CC2CCC1CC2NC(c1cnn(C)n1)=O 48189,c1(C(=O)NCC2CCCN(C(C3(O)COC3)=O)C2)cc2ccnc(Cl)c2s1 48190,Cc1nc2cc(C(=O)NCCN(CC(C)O)C(C3CC(=C4CCC4)C3)=O)[nH]c2s1 48191,c1(C(=O)NCCCCN(C(c2cc(C(C)=O)on2)=O)C)cc(C)c(Cl)cn1 48192,c1(N(CCNC(C2(F)CCCC2)=O)CC)ncc(C#N)cc1F 48193,N1(C(C(C)N(C(=O)C2=CCCC2)C)=O)CCCCC1C(C)(C)O 48194,c1(CS(=O)(=O)NC2CC(C(=O)NCc3ccncc3)C2)ccccc1 48195,CCC(CNC(C1(N)CCC(C)C1)=O)(CC)c1ccccn1 48196,N1(C(C2N(CC#C)CCC2)=O)CCC(NC(C2C(C)OC(C)C2C)=O)C(F)C1 48197,CP(C)(=O)c1ccc(C(N2CCC(CNC(=O)C3=CCCCC3)C2)=O)cc1 48198,c1(C(=O)NCC2(N(C)C(C3CSC3)=O)CC2)cnc(C2CC2)s1 48199,c1(C(N2CC(CN(C(c3c(OC)cnc(Cl)c3)=O)C)C2)=O)ccc(F)c(C#N)c1 48200,C1(CNC(=NC)NCC2CC(SC)C2)CCCCC(F)(F)C1 48201,c1(OC)ccccc1C(=O)NCCC1CC(NC(c2ccc(C#N)o2)=O)C1 48202,N1(C(C2(C(=O)C3CC3)CC2)=O)CCCC2(NC(=O)CCc3cccc(F)c3)CC2C1 48203,c1(C(=O)NC2CN(C(c3coc(Cl)n3)=O)CC23CC3)ccc2cccnn12 48204,c1(C(=O)NC2CCCN(C(CC(CCC)O)=O)C2)cnc2c(C)c(Cl)ccc2c1 48205,CC(CCNC(=O)CNS(N)(=O)=O)CCNC(=O)C(C)(C)C1CCOCC1 48206,C1(C(N(C2CC2C)C)=O)CC12CCN(C(=O)Cc1cccc(Br)c1)CC2 48207,CC(CC(F)(F)F)C(=O)N1CC(CCNC(c2cc(=O)cc(Cl)[nH]2)=O)C1 48208,C1(NC(C(C)OCCC=C)=O)CN(C(C2(C#N)CCCC(=O)C2)=O)CC(C)(C)C1 48209,C1(C(N2CCCCCC2CNC(=O)C(c2cccnc2)O)=O)CCCCC1(F)F 48210,c1(C(N(CC(C)O)CCNC(c2c(C)n(C)nc2)=O)=O)cccn2c(C)cnc12 48211,CC1(NC(=O)Cc2csc(C(F)(F)F)n2)CN(C(=O)CC2CC3(CC3)C2)C1 48212,N1(C(C2C(CC(C)C)C2)=O)CC2CN(C(=O)Cn3ccccc3=O)CCC12 48213,C1(CNC(C(CC)(CC)CO)=O)CCN(C(C2CC2C(=O)OC)=O)CCC1(F)F 48214,CCCCCCC(C)C(=O)N1CCN(c2ccc(-c3cc(Cl)cc(CC)n3)s2)CC1 48215,Cc1nc[nH]c(=NCC(C2CC2)N(C)C(c2c(C)n[nH]c2C)=O)c1C#N 48216,c1(CC(N2CC(NC(CC(C)(C)O)=O)C(C)(C)CC2)=O)ccc2cccnc2c1 48217,C12(CNC(CN(C3CCSC3)C)=O)CCCC1N(C(=O)CC1OCCO1)CCC2 48218,N1(C(C(COC)COC)=O)CCN(C)C(C(=O)NCCCNC(N)=O)C1 48219,CCCC(C)(C)C(=O)N(C(C)C(=O)NCC1(C)CC2(CC2)C1)C1CC1 48220,N1(C(C(C#C)(C)C)=O)CC(NC(c2ccccc2C2CCOC2)=O)C(N=[N+]=[N-])C1 48221,CCCC(C)CCNC(=O)C(C1CCN(C(c2ccccc2O)=O)CC1)C 48222,C1(N(C)C)CCCC(C(=O)OC(C)(C)C)C1.N12CCC(C1)N(C)C(=O)CC2 48223,N1(C(C(CNC(C(C=C=C)C)=O)C)=O)CCN(C)C(C)C1 48224,c1(C(=O)NC2CC(C)N(C(=O)CC3CC=CCC3)C2)cnc2cccnc2c1 48225,Cc1cc(NC(C2CCCCCC2)C)ncc1C(F)(F)F 48226,C(=O)(CC(C1CC1)C1CC1)N.C1(CN2CCC3CC3C2=O)CCCCO1.CO 48227,C1(C(N(CC=C)C)=O)CCC(C2CC2)N1C(c1cc(Cl)cs1)=O 48228,N1(C(c2cn(CC)nn2)C(=O)NCC2CCCO2)CC2(CO)CC2(C(F)(F)F)C1 48229,C1(C(N2CCC(C)(N3CCCC3)C2)C(=O)NCCCSC)CC12CCCCC2 48230,N1(C(C(CC)(C)C)=O)CCC(C2CC2)C1CNC(=O)C(c1ccccc1)N(C)C 48231,N1(C(c2c(C)nc(CCCC)s2)=O)CC(C2CN(C(C34CCC3CC4)=O)C2)C1 48232,c1(-c2c(C(N3CCOC4CC34)=O)n[nH]c2)cccnc1-c1ccccc1 48233,C(=O)(C(C)CC(C)(C)C)N1CC(F)CC(NC(c2ccc(OC)cc2C)=O)C1 48234,C#CCC(CC(=O)NC(CC)C(C)(C)C)NC(C1CS(=O)C1)=O 48235,c1(CNC(C=C2CCC(C)CC2)=O)nc2c(s1)CCN(C(=O)Cc1cocn1)C2 48236,C(CC1CCC1)(C(=O)NC(C)(C)C)N(CCCF)C 48237,N1(CC(=O)N=c2cco[nH]2)CC2CCN(Cc3nc[nH]c3C(F)(F)F)CCC2C1 48238,C12(C(=O)NCC(CNC(c3ccn4ncnc4c3)=O)O)CCC(O)(CC1)CC2 48239,C1(CCNC(c2ccc(Cl)s2)=O)CCCN(C(=O)CC(O)c2ccccc2)C1 48240,C1(CNC(C(C2CC2)OC)=O)C(C)CCCN1C(=O)C(=Cc1ccc(C)cc1)C 48241,C1(NC(c2c(C)ccs2)=O)CC2CC(NC(=O)C(O)C(C)C)CC2C1 48242,C1(NC(c2n(C)c(Cl)nc2)=O)CC2CCC(C1)N2C(=O)Cc1cccc(Cl)c1 48243,C1(C(=O)NCC2(F)CN(C(C(c3ccccc3)=O)=O)C2)CCC2C(CC1)C2(F)F 48244,N1(C(c2cc(C)ncn2)=O)CCC(C2CCN(C(c3ccccc3C)=O)C2)C1 48245,C(=O)(CCCC(C)(C)C#N)NCC(C1CCOC1)NC(c1snc(C)c1N)=O 48246,C1(C(=O)NOC(C)C(=O)OC)N(C(=O)OC(C)(C)C)CC12CCCC2 48247,Cc1n[nH]c(C)c1SCC(N1CCCC(CN(C(=O)C(C)CC2CCC2)C)C1)=O 48248,C1(CNC(c2c(C)nn(C)c2)=O)CC(C(=O)NC2CCC(C)(C)C2)=NO1 48249,CCC(C)(COC)C(=O)NCC(C1CC1)N(C(=O)Cn1cccc(C)c1=O)C 48250,c1(CC(=O)NC2CCC(NC(Cc3c(Cl)cn(C)n3)=O)C2)cc(F)ccc1Cl 48251,S(=O)(=O)(c1cc(Br)cc2c1OCC2)N.Cc1ccc(CC(=O)N2C3(CC3)C2)cc1 48252,Cc1ccccc1CC(C)C(=O)NCC1(O)CCN(C(=O)C#CC(=O)N(C)C)C1 48253,CC(C(=O)N1CCCN1C(=O)Oc1ccccc1C(F)(F)F)C1CCCNC1 48254,C(=O)(C1CCCc2c[nH]nc21)N1CC(CNC(CC(C=C)C)=O)C1 48255,C12(CNC(C3C(OC)CCC3)=O)CCC1CN(C(=O)Cc1cccc(F)c1F)C2 48256,c1(N(C)Cc2ncc(CC)s2)nc(=NC)nc(N(C)CC2CC2(C)C)[nH]1 48257,C12(C(=O)NCCCOC(=N)O)CC(CN1C(=O)CC1CCOC1)C2 48258,O=C(C#CC1CCOCC1)NCC1CN(C(c2ccc(C(F)F)o2)=O)CC1(F)F 48259,c1(CC)cc(F)c(C(=O)NC2(C)CN(C(=O)C(CC)n3cncn3)C2)cc1F 48260,C1(CC)CN(C(=O)Cc2cc(C)n(C)n2)CCC1CNC(=O)C(CC)(CO)OC 48261,c1(NCC(c2n(C)ncc2)O)ccc(S(=O)(=O)N2CCC2CO)c(Br)c1 48262,CC(CS(C)(=O)=O)C(=O)NCCN(C(=O)C=Cc1cnccn1)CC1CC1 48263,S(=O)(=O)(c1cc(-c2ccccc2)no1)C1(N(C)C2CC2)CCC1 48264,C#Cc1cccc(C(=O)NCC(C)(CC)NC(C2CCCCN2C)=O)c1C 48265,c1(C(=O)NC(C(C)NC(c2c(C)nns2)=O)(C)C)cc(C2CCCCC2)n(C)n1 48266,C(=O)(C(C)(C)C(C)NC(c1ncccc1C)=O)NC(CCC)c1ccco1 48267,S(=O)(=O)(c1ccccc1C(=O)OC)Nc1c(C(=O)OCC)n(C)c(SC)n1 48268,CC(C)CC(O)C(=O)NCC(CNC(c1cncc(N(C)C)c1)=O)CO 48269,CC(C)CC(C)(O)CNC(C1CC(CCNC(c2cccc(=O)n2C)=O)C1)=O 48270,c1(C(N2CC(OC)C(NC(c3ccc([N+](=O)[O-])s3)=O)C2)=O)ncn2c1CCC2 48271,CCCC(CNC(c1ccc(F)cc1F)=O)C(=O)N1CCCOC(CC)C1 48272,C1(CNC(CSCC#C)=O)C(C2CC2)CCN1C(c1cnc(-c2ccsc2)s1)=O 48273,C1(C(N(CCNC(CCOCC)=O)C(C)C)=O)CCC(N2CCOCC2)CC1 48274,C=CCCCCCCCC(=O)N1CC2(CCCC(CNC(C3(O)CCC3)=O)O2)C1 48275,Cc1cc(Br)cnc1C(=O)NCC1CN(C(c2ccc(Cl)o2)=O)CC1C 48276,C(=O)(C1CCc2c(Cl)cccc21)NC1CN(C(CC)=O)CC1C 48277,c1(NC(C)=O)nc(C(=O)NCC(C2CC2)N(C)C(C2CC23CC3)=O)cs1 48278,c1(C(=O)NC(CNC(c2cc(CC)c(CC)o2)=O)C(C)C)c(F)ccc(C)c1F 48279,N1(C(C2(CC(C)C)CCC2)=O)CC(NC(=O)Cc2coc(C(F)F)n2)C(C)C1 48280,C1(C)(C(=O)NCC(C)N(C)C(c2cnn(-c3ccccn3)c2)=O)CC=CCO1 48281,N1(C(C(CCC)OC)=O)CC2CC(NC(=O)CC3(O)CCOCC3)CC1C2 48282,c1(C(N(C2CCN(C(c3ccc(CC)s3)=O)C2)CC)=O)c(OC)nsc1OC 48283,C1(OC(CCCOCC(C)C)=O)CCCC(C(C)(C)C)CC1 48284,C(C(=O)NCCC1CN(C(c2cnccc2Br)=O)C1)(C(C)(C)C)NC(C)=O 48285,N1(C(C(C)(CO)OC)=O)CC(C(N2CC(N3CCNC3=O)C2)=O)C2(CCC2)C1 48286,C(CO)(C(C)NC(=O)C(n1nnnc1C(C)(C)C)C)NC(C1CC(=C)C1)=O 48287,C(C(C)C(C)C(=O)NCCOCCN(C)C(c1cc(C)nn1C)=O)OC 48288,C1(COCC)CN(C(C2CCN2C(C2CCCO2)=O)=O)CCO1 48289,C1(Cl)(C(=O)NCCN(C(c2nocc2C2CC2)=O)CC)CC12CCC2 48290,N1(C(c2cccc(CC)c2N)=O)CC2CCCC(C1)N2C(C1(C)CCCO1)=O 48291,C1(C(=O)NCCCOCC(C)C)CN(C(=O)C(C)S(C)(=O)=O)CC1(C)C 48292,C=CCC(CC=C)C(=O)NCC1CN(C(=O)CC2CCC(=O)NC2=O)CCN1C 48293,c1(C(=O)OCCC(CCC)C)ccc(C(C)(C)C)c(F)c1 48294,c1(CN(CC)Cc2ncc(C(=O)N(C)C)s2)ccc(Cl)cc1OC 48295,c1(NC(CC)CC(F)(F)F)ncccc1S(=O)(=O)NCC1CN(c2ncccn2)C1 48296,Cc1nccc2c(=O)c(-c3noc(C4CCC5(C=C5)OC4)n3)c[nH]c12 48297,c1(C(=O)NCC(C)NC(=O)CCCN(C)C)cccc2cncn12 48298,c12nc(C)c(o1)C(=O)NC2.C(CCCCC1CC1)NC(CN(C(C)=O)C)=O 48299,C(N=c1[nH]c(=NC(CN(C)C)C2CC2)c2c(ncn2C)[nH]1)c1cccc(C)c1N 48300,C1(C(=O)NC2CCN(CCC)C2)CN(C(c2cncs2)=O)CCO1 48301,Cc1cn2c(n1)CCC(CNC(=O)N(C(c1ccccc1)C(N)=O)C)C2 48302,C(=O)(C(C)(C)CC(=O)OCC)N1CCC(N(C(C(CC(=C)C)C)=O)CCC)C1 48303,C(=O)(CCS(N)(=O)=O)NCC(C(C)(C)C)NC(CN(C(=O)OC)C)=O 48304,c1(C(N(CCCCCNC(CCC(=O)OC)=O)C)=O)c(F)ccc2cnn(C)c12 48305,C=C1CCC(CNC(=O)Nc2ccsc2)CC1 48306,Cc1csc2c(C(N3CC4CC(NC(=O)Cn5cnnn5)CC3C4)=O)ncnc12 48307,C(=O)(C(O)CCC(F)(F)F)N1C(C(C)C)C(NC(C2CCSC2)=O)CC1 48308,C1(C(=O)NC2CCC(NC(C3C(C(=O)OC)C=C3)=O)CC2)CCc2nncn2C1 48309,c1(C(N2CCC(N(C(=O)CC(C)F)CC)CC2)=O)ccc(-n2cnnn2)c(C)c1 48310,C1(CNC(C2C(C)CCCC2)=O)N(C(c2cnn(C3CC3)c2)=O)CCCC1(C)C 48311,c1(C(=O)NC2C(NC(C(C)n3ccnn3)=O)CCC2)cccc(Cl)c1Cl 48312,C1(C(=O)NC(C(=O)NCCCN=[N+]=[N-])C2(C)CC2)CCCC(=O)C1 48313,N1(CC(COCC(C)C)O)CCC(N(C)C(c2cnon2)=O)CC1 48314,c1(CC(=O)NCC2N(C(C(C)C3CCC3)=O)CC(F)C2)cccc2nsnc12 48315,C(C1CCCC1)=CC(=O)N(C1(CC(=O)NCC(CO)C2CCC2)CC1)C 48316,N1(C(C(C)NC(CC)(C)C)=O)CC(C)C(NC(C2C3CC4C(C3)C24)=O)C(C)C1 48317,Cc1ccc(C)c(C(=O)NC2CN(C(=O)CCc3c(C)noc3C)CC2F)c1O 48318,c1(CNC(c2nccn2C)CC)c(C)cc(C)cc1C 48319,c1(N(CC=C)C)ncccc1S(=O)(=O)NC(c1ccccc1F)C.C1CO1 48320,CC1(CNC(C2CCCC3(CC3)C2)=O)CN(C(c2cn3ccnc3s2)=O)CCO1 48321,C1(C(=O)NC(CNC(c2c(C)n(C)nc2)=O)C(C)C(C)C)C2CCC3C(C2)CC13 48322,c1(C(Cc2ccccc2)NC(C(=O)N(CC(C)OC)C)=O)ccc(Br)cc1 48323,C12(CO)COC(CCN1Cc1n[nH]c3cccnc13)C2 48324,c1(C(=O)NC(C(C)NC(C2ON=C(C)C2)=O)CO)cnn(CCN(C)C)c1C 48325,N1(C(CC(CCC)O)=O)CC2CCC(C1)C2NC(c1cc(C)cc(F)c1)=O 48326,c1(NC(c2c(C)nns2)=O)cnc(F)cc1C(=O)Nc1cccc(CCO)c1 48327,C1(NC(c2ccsc2C(F)F)=O)CN(C(C2CCCC(O)C2)=O)CCC1CO 48328,Cc1ccc(F)cc1C(N1CCCC1CC(=O)NCC1CCC(F)(F)C1)=O 48329,N1(C(c2cc(CC)sn2)=O)CCCC(C(=O)NCC2CCN2C(C)(C)C)C1C 48330,C(=O)(CS(=O)(=O)CC1CCCO1)NC(CNC(c1c(C)nc[nH]1)=O)(C)C(C)C 48331,C1(CC)CN(C(=O)C(C)(C)c2cnsc2)CCC1NC(c1cc(O)cc(F)c1)=O 48332,CCC(C)(CNC(=O)C1=NOC(CNC(c2cc(C(N)=O)co2)=O)C1)C(N)=O 48333,S(=O)(=O)(c1cccs1)NC(C)C(=O)NCC(CO)NC(=O)Cn1cccnc1=O 48334,C1(C(N2C(C=C)CCC2)=O)CCN(C(C2CC(=O)OC2(C)C)=O)C12CCC2 48335,c1(C(=O)NCCC2N(C(C3(OC(C)=O)CC3)=O)CCC2)cnc2onc(C)c2c1 48336,c1(C(=O)NCC2COCCN2C(=O)CC23CCCC2C3)nccc(Br)c1O 48337,C(=O)(C(C)CS(C)(=O)=O)N1C(CCOC)CN(C(=O)CCc2cnoc2)CC1 48338,c1(C(c2c(C(N(C(CCC)=O)c3nccs3)=O)ccs2)=O)ccc(F)c(C)c1 48339,N(C1CCCc2c[nH]nc21)C(C(C(C)C)n1cc(-c2cccc(NC)c2)nn1)=O 48340,C1(CNC(C2CCCC(C)C2)=O)CC2(CC2)CN1C(C1CCCSS1)=O 48341,c1(C(N2C(CC)CN(C(C3CC=CCO3)=O)CC2)=O)ccc(C)c(S(N)(=O)=O)c1 48342,N1(C(=O)OCC)CCCC(NC(c2ccncc2)=O)C1.C12CC(C1)C(=O)N2 48343,CS(=O)(=O)c1nc(Cl)cc(=NC2CCCCC2NC(C2CCCOCC2)=O)[nH]1 48344,CC(C)(C)C(CO)C(=O)NCC(F)CNC(=O)CCc1cccc(C(F)(F)F)c1 48345,C(=O)(C(F)C(F)(F)F)NCC1CC(NC(CC2C(C)CCO2)=O)C1 48346,c1(C(N(C)CCNC(=O)CCc2ccc(CO)cc2)=O)sccc1S(C)(=O)=O 48347,C1(NC(c2cnco2)=O)CC(O)(C2CCN(C(c3ccccc3)=O)CC2)C1 48348,CCCC(CC)CC(=O)N1CC2CCN(C(=O)CCn3nc(C)nc3C)C2C1 48349,c1(NC2C3CN(C(=O)C(c4ccccc4F)C4CC4)CC32)ccn2nccc2n1 48350,N1(Cc2scc(C)n2)CCC2(CC1)CN(C(C1(C)CCOC(C)C1)=O)CC(C)O2 48351,C1(C(N2CCCC(C)C2)=O)CCN(C(=O)CCCC2CCC2)C12CCC2 48352,N1(C(CC(CC)O)=O)CCCC(C2CC2NC(c2cn(C)nc2C)=O)C1 48353,N1(C(C2CCCCC(=O)N2)=O)CCCC12CCN(C(C1(F)CC=CCC1)=O)CC2 48354,C1(C(=O)NC2(C)CCCN(C(c3cc(O)ncn3)=O)C2)CCc2nnc(O)n2C1 48355,C(CC(O)C(=O)NC(C1CCN(C(=O)COC2CCN(C)CC2)C1)(C)C)SC 48356,C(=O)(C(O)C(C)(C)C)N1CCN(C(CNC(C(C2CCC2)OCC)=O)C)CC1 48357,c1(NC(Cc2cccc(-c3ccc(OC)c(OC)c3)n2)=O)c(Cl)nc(C)nc1Cl 48358,C1(C(=O)NCC(C)(F)CNC(=O)CC2CCSC2)CCOC1(C)C 48359,CC(C)(C)CC(O)CC(=O)N1CCCN(C(c2noc3c2CCCCC3)=O)CC1 48360,C1(C(N2CC(C(=O)NCC)C2)=O)CN(C)CCN1C(=O)CCC1CC1(F)F 48361,c1(C(=O)O)cc(NC2C(CNC(C(CC)(F)F)=O)CC2)cc(C)c1 48362,C(=O)(CCC(C)NC(C1CN(C(=O)C(C)c2cc[nH]n2)CC1C)=O)OC 48363,C(=O)(C(CC1COCCO1)C(F)(F)F)N(C1CN(C(c2ccn(C)n2)=O)C1)C 48364,c1(OCC)cc([N+](=O)[O-])ccc1NC(C1CC1NCc1ccc(OC)nc1)=O 48365,N1(C(C)C)CCOC(C(=O)N(C2CC2)Cc2cnoc2-c2ccccc2)C1 48366,C1(NC(C(F)=CC)=O)CCN(C(c2cccc(N)c2OC(C)C)=O)CC1O 48367,CN1CC=C(CC(=O)N2CCC3CCN(C(=O)CN4CCCNC4=O)C3C2)CC1 48368,c1(OC)nc(N2CCN(C(c3cc(Cl)ccc3C)=O)CC2C(F)(F)F)ncc1Br 48369,C1(CNC(c2ncc(C)cc2C)=O)CC2CCCC2N1C(C1C2(CC2)C12CC2)=O 48370,N1(C(C(CSC)OC)=O)CCC(C2CCN(C(c3cnc(C(C)C)s3)=O)CC2)C1 48371,N1(C(CCN(C(=O)CC2CCCC23CC3)CC#C)=O)CCCCC(COCCC)C1 48372,C(=O)(CC(O)CNC(c1conc1C)=O)N(C)Cc1cnc(C)s1 48373,C(CC(N)=O)(c1cn(CCCCF)nn1)N(C)C(C1(CN(C)C)CC1)=O 48374,N1(C(C(CCOC)C)=O)CCC(C(N2CCC(C)(CN(C)C)C2)=O)C12CCC2 48375,C1(COC)(NC(c2cc(C(=O)OC)no2)=O)CN(C(=O)C(O)CSC)C1 48376,NC1(C2CCN(C3(C(=O)NC4CCCCC4)CC3)CC2)CC1 48377,C(=O)(CCS(=O)(=O)NC)N1CC(C)(NC(C2N(CC)CC2)=O)C1 48378,C1(C(C(=O)NC)N(c2cn(C)cn2)C)CCCCC1N1CCCC1=O 48379,c1(C(=O)NCC2CC(F)(CNC(Cn3c(C)ccn3)=O)C2)ccnc(CO)c1 48380,C1(C(=O)NCCNC(c2c(C)nsc2NCC2CC2)=O)Cc2cc(F)cc(F)c2O1 48381,C(CC(C)C)(CS(C)(=O)=O)NC(c1cn(CCC)nc1C)c1nnnn1C1CC1 48382,C1(NC(c2c[nH]nc2-c2ccccc2)=O)CCCCN(C(=O)C(F)(F)CF)C1 48383,Cc1ccc2c(N(CCCO)C)nc(=NCCn3cnc4c3CCCC4)[nH]c2c1 48384,C12(C(=O)NC(CC)CNC(=O)COc3cccc(Cl)c3)CCC(COC)(CC1)C2 48385,c1(C(N(C2CC2)Cc2cn(-c3c(C(=O)OC)scc3)nn2)=O)cc(=O)n(C)cn1 48386,c1(C(=O)OC)c(C(=O)NC2(CNC(=O)CSC)CCCC2)n[nH]c1C 48387,C1(OC)CC(CNC(=O)C=CC2CC2)N(C(=O)Cc2cc[nH]n2)C1 48388,N1(C(c2ccn(COC)n2)=O)CCCC12CCCN(C(=O)C(C)CC(C)(F)F)C2 48389,C12(C(=O)NC(c3cnc(C)s3)C)C(NC(=O)Cn3cnnn3)C3CC1C2C3 48390,c1(C(=O)NCC2(O)CCCN(C(COC(CC)(C)C)=O)C2)ccc(C#N)c(O)c1 48391,C=CC(C)(C)C(=O)NC(CSCC)C(=O)NCCN1CCCC(C)C1 48392,Cc1nc2ccccc2cc1C(N1CCC1NC(c1ccc(N)c(C)c1C)=O)=O 48393,CN1CCCC(CNC(=O)C(O)CNC(c2ccccc2F)=O)C1 48394,c1(SC)ccc(NC(c2cc(C(=O)OC(C)(C)C)n(CC)n2)=O)cc1 48395,C1(C)(CNC(CCCN(C)C)=O)CN(C(c2ccc(F)c(Cl)c2)=O)C(C)(C)C1 48396,Cc1cc(CC(=O)NC(C)(C(=O)N2CC(OC(=N)O)C2)C2CCC2)nn1C 48397,n1(CC(=O)N(CCOC)CCNC(=O)C(C2CCC(=O)N2)C)nc(C)c(Cl)c1C 48398,C1(C(N(CC(C2CCC2)OC)C)=O)CCCCC1(C)NC(c1cnc[nH]c1=N)=O 48399,N1(C(C(C(C)C)SC)=O)CC2(C1)CN(C(=O)C(c1ccc(Cl)cc1F)(C)C)C2 48400,C12(CNC(c3ccc(Cl)[nH]3)=O)CC(CO1)N(C(c1cc(CF)on1)=O)C2 48401,C=C(CNC(=O)CCCn1cc(CCC(C)=O)nn1)c1ccncc1 48402,N1(C(CC2C(C)CCCC2)=O)CCC=C(C(=O)NCCN(C)C2CC2)C1 48403,Cc1ccc(F)c(O)c1C(N1CC(CNC(=O)CCc2ccon2)C(C)C1)=O 48404,C1(NC(CC2CC(CC)C2)=O)CCCCC(c2ccccc2)C1 48405,c1(C(=O)NC2C(OCCCC(=O)OC(C)(C)C)CCCC2)ccc(F)c(Br)n1 48406,C1(CC(=O)N(CC(C(=O)NCC(C(=O)NC)O)C)C)NC(=O)NC1=O 48407,CC1=C(C(=O)N(C2CCCCC2N(C)C(C2CCOC2)=O)C)CCS1(=O)=O 48408,C12(C(N3CC=C(CNC(c4c(CC)cccn4)=O)CC3)=O)CCCN1CC(O)C2 48409,CCC(C)C(=O)C(=O)N1CCC(C)(C(=O)NCC2CCCC2)C1 48410,c1(C(=O)NC2C(C)(C)CN(C(C3(F)CCOCC3)=O)C2)c(F)ccc2occc12 48411,C(C(C)(CC(C)C)NC(=O)C(C)N(C)C)NC(C1(CC)CC1)=O 48412,Cc1c(C(=O)NC2CC2NC(c2ccc(C(C)C)o2)=O)cnn1C1CC1 48413,N1(Cc2cn(C)c(-c3ccccc3)c2)CCC(O)C(C(F)(F)F)(C(=O)O)C1 48414,c1(C(N2CCC(OC)(CNC(C3(C)CCSCC3)=O)C2)=O)ccc(=O)n(C)c1 48415,C=C(CNC(C1C(O)CCN1C(c1cccc2occc12)=O)=O)C1CCOCC1 48416,C12(NC(=O)COC3CC3)CCC(C(=O)NCC(O)C3CCC3)(CC1)C2 48417,N1(C(c2cnn(CC(F)F)c2)=O)CCC12CN(C(C13CCCCC1C3)=O)C2 48418,N1(C(c2n(C)ccn2)=O)CCC(C2CCN(C(c3cnco3)=O)CC2)C1 48419,N1(C(C2CC(C)(c3ccccc3)C2)=O)CCCCC12CC2 48420,C1(C(=O)NC2CCN(C3CC3)C2)CCC2(CC2)N1C(c1nc(CO)n[nH]1)=O 48421,N1(C(c2cc(C)cc(C)c2)=O)CCC2(CC1)CC2NC(C12CCN(CC1)C2)=O 48422,c1(N2CCC(C(=O)OC(C)(C)C)CC2)nccc(NCCN2CCCC(O)C2)n1 48423,c1(OCCOC)cccc(CNC(N2CCCCC2C2(CO)CC2)=O)c1 48424,c1(CC(C)NC(C2CC2NC(=O)C(C)(C)CF)=O)c[nH]c2cc(F)ccc12 48425,CN=c1nc(C(N2CC(NC(=O)C(C)(C)C(F)(F)F)CC(O)C2)=O)cc(C)[nH]1 48426,N1(C(C2CC(=C)C2)=O)CCC2OCCN(C(=O)CCc3ccc(SC)cc3)C2C1 48427,N1(C(CC=CC)=O)CCCC2(CCC2NC(C2CCCCO2)=O)C1 48428,n1(CCC(=O)NCCC(C)NC(c2c(C(=O)OC)scc2)=O)c(C)csc1=O 48429,c1(C(N2CC(C)C(CCNC(c3cccc(F)c3)=O)C2)=O)cncc([N+](=O)[O-])c1 48430,C1(NC(c2cc(SC)oc2)=O)CC(NC(=O)C2=CCCOC2)C12CCOCC2 48431,N1(C(Cc2c(C)occ2)=O)CC2C(NC(C3(c4ccc(F)cn4)CC3)=O)C2C1 48432,C1(C(=O)NCCC(C)OC)CCN(C(c2ccoc2)=O)C12CC2 48433,C1(CN(C(c2n(CCCC)nnn2)c2csc(C)c2)C)(OC)CCOCC1 48434,C(=O)(C(Cc1ccoc1)NC(=O)C(F)=CC1CC1)N(CC(C)OC)C 48435,c1(C(=O)NCCN(CCCN(C)C)C(=O)Cc2cn(C)cn2)ccc(F)cc1F 48436,C1(CNC(CC=C)=O)CC2CCC(C1)N2C(=O)CS(=O)(=O)NC1CCC(C)CC1 48437,CC1(CNC(=O)Cn2ccc([N+](=O)[O-])n2)CN(C(c2cccnn2)=O)CCO1 48438,C1(CNC(CCc2cccc(OC)c2)=O)CN(C(=O)Cc2cc[nH]c2)CCCO1 48439,c1(C(=O)NCC(CC2CN(C(CCCCC)=O)C2)(C)C)ccc2oncc2c1 48440,c1(C(=O)NC2C(NC(C3(COC)CCCCO3)=O)CC2)cc(C)ccc1C 48441,N1(C(c2nnn(CC)c2C)=O)CCC(NC(C2(Cl)CC2(C)C)=O)CC(O)C1 48442,C1(NC(c2c(C)n[nH]c2C)=O)CN(C(=O)C(=O)NOC(C)(C)C)C2(CCC2)C1 48443,N1(C(CCC2(NC(C3(C)CCC(=O)N3)=O)CCC2)=O)CC2CCC2(C)C1 48444,C1(C(N2C(C)C(NC(C3C4COCC34)=O)CCC2)=O)CCC(C2CC2)CC1 48445,S(=O)(=O)(c1ccc(N2CCC(CO)CC2)c(C#N)c1)N1CCC(C)C(CO)C1 48446,CC1CSCCN(C(=O)CC2CCCC(NC(=O)C(c3ccnn3C)O)C2)C1 48447,C1(NC(Cn2cc(CNC(C3CC(C)OC3)=O)nn2)=O)CC(C)(C)C12CCC2 48448,C1(C(N2CC(CNC(Cc3cn(C)nc3)=O)OCC2)=O)CC2C=CC1C21CC1 48449,c1(OC)cc(C(=O)NC2C3CN(C(=O)C=CSC)CC23)cc2nc(O)[nH]c12 48450,c1(C(C(=O)NCCC2CC(NC(C(C)=C(CC)C)=O)C2)C)ccncc1C 48451,c1(C(N(CC(CC)NC(=O)CC#N)C)=O)cc(C)c(F)cc1Br 48452,Nc1ccc(C(=O)NC2CCCN(C(c3cncc(F)c3Cl)=O)CC2)nc1Cl 48453,C=Cc1cnn(C)c1C(N1CCN(C(C2(C)CC2(Cl)Cl)=O)C(C)C1)=O 48454,N1(C(C(COCC)C)=O)CCN(C(c2cccc(C3CCC3)c2)=O)C2COCC12 48455,N1(C(C2CC(C(=O)O)CN(C(=O)OC(C)(C)C)C2)=O)CCC(NC(C)C)C(O)C1 48456,CC1CN(C(c2ncn3c2CCC3)=O)CCCN1C(c1cccc(N)c1O)=O 48457,N1(C(C2OCCN(C(C)C)C2)=O)CCN(C(=O)Cc2sc(O)nc2O)CCC1C 48458,C(=O)(C1=C(Cl)CCCC1)N1C(C)CC1C(=O)NC1(CO)CCCCC1 48459,CCCC(C)CC(=O)N1CCCCC(NC(c2cc(C)c(C(=O)OC)o2)=O)C1 48460,N1(C(c2ccc(CN(C)C)cc2)=O)CCC=C(CNC(=O)CC2CCC3CC23)C1 48461,c1(N2CCCC(CNC(C(Br)=C(C)C)=O)C2)nc(C(C)C)cc(C(C)C)n1 48462,c1(C(=O)NCc2nc(CNC(CCc3nc(=N)[nH][nH]3)=O)sc2)cccnc1S 48463,N1(C(C2N(C(Cn3nc(C)oc3=O)=O)CCC2(C)C)=O)CCC2(CCCCO2)C1 48464,Cn1nnc2c(C(N3CCC4C(NC(C5CCC(F)CC5)=O)C34)=O)ccnc12 48465,c1(COC)c(C)cccc1Br.N12CC=CC(C1)NC(=O)C1C(CC)(C1)C2=O 48466,N1(C(C(OCC)OCC)=O)CCC(F)(C(=O)NCC(C)(C)CN2CCCC2)CC1 48467,Cn1nc(Br)cc1NC(C1CCCN1C(=O)COc1ccccc1)=O 48468,C(N=c1[nH]c2ncc(Cl)cc2o1)c1c(C)c(C(F)(F)F)n[nH]1 48469,c1(C(=O)NCCC(C)NC(C2C3CCCCCC23)=O)c(F)ccc(F)c1Cl 48470,Cc1ccc(CC(=O)NCC(C2CCCCC2)NC(C2CCCCC2O)=O)cc1 48471,C1(C)(CNC(C(COC)O)=O)CCCN1C(=O)C(=CC1CCCC1)C 48472,c1(C(=O)NCCCN(CCOCCOC)C)cc(C)nc2c1nc(C)n2C 48473,c1(C(=O)NC2CC(NC(C(Cn3ccc(C)n3)C)=O)C2)nccc(F)c1Cl 48474,C1(CC=C)(NC(=O)CS(=O)CC)CCS(=O)(=O)CC1 48475,C1(C(N2C(CCCNC(CCC=C)=O)CCC2)=O)CCOC(C)(C)C1 48476,Cc1cc(C(N2CC(NC(c3cc4occc4n3C)=O)C(F)C2)=O)cc(N)c1O 48477,C1(COC)(NC(=O)C(C2CCOCC2)C)CCN(C(c2cc[nH]c(=N)c2)=O)CC1 48478,C1(NC(CCCNS(C)(=O)=O)=O)CCC2CCN(C(c3c[nH]cc(F)c3=O)=O)C12 48479,c1(C(c2nnnn2C2COC2)NCC(C2CCSCC2)(C)O)cccc(CO)c1 48480,N1(C(C2(CNC(=O)C=CC(C)(C)C)CC(=C)C2)=O)CC2CCC1CN2C(C)=O 48481,CC1(C#CC(=O)N2CCCC2(C)CNC(=O)C(C)(C)C2CC2)COC1 48482,C12(NC(N3C(CNC(=O)OCC)COCC3)=O)CCCC1OCC2 48483,C1(C(C)(C)C)CCCN(C(=O)C(CO)NC(C2CC(F)(CF)C2)=O)C1 48484,N1(C(c2cccs2)=O)CC(CNC(C2(C(F)(F)F)CCC2)=O)CC12CCOCC2 48485,c1(C(=O)NC(CN(C(=O)CN2CCC(C)C2)CC)C)sc2cc(F)ccc2c1C 48486,c1(CC(=O)NC(C(C)NC(=O)Cn2cnnn2)CO)coc2ccc(F)cc12 48487,c1(C(=O)NCC2(O)CCCN(C(c3cc(Cl)no3)=O)C2)ccc2c(c1)CCCO2 48488,N1(C(c2cccnc2Sc2ccccc2)=O)CC(NC(C2CC(O)C2)=O)C(F)C1 48489,CCCCCC(C)(C)C(=O)N1CC(C)(NC(=O)Cc2c[nH]c3cccc(F)c23)C1 48490,CC1CN(C(=O)CCC2CCCN2C(=O)OC(c2ccccc2)=O)CCS1(=O)=O 48491,c1(OC)ccccc1NC(C1(C)CN(C(c2cc(-c3ccccn3)[nH]n2)=O)C1)=O 48492,C(=O)(CCCCCC(C)C)N1C(C)CCC(NC(C2(CC)CC(C)(C)C2)=O)C1 48493,N1(C(CCN(C(CCC2C(C)(C)C2)=O)CCO)=O)CCc2nc[nH]c2C1 48494,C(c1ccc(C)c(C)c1)=CC(=O)NC1C2(CC(NC(C(CC3CC3)OC)=O)C2)C1 48495,Cc1cc(C(=O)NC2CCC(NC(C3CCC(C)CC3)=O)C2)sc1C 48496,Cc1ccc(C)c(C(=O)NCC(C2CC2)NC(c2cccc3scnc23)=O)c1C 48497,Cn1ncc2c1CCCC2N=c1[nH]c(=NCc2ccccc2Br)[nH]c2cc[nH]c12 48498,C1(CCO)CCN(C(=O)NC2(CNC(=O)OC(C)(C)C)CCCCC2)CC1(C)C 48499,c1(N2CCN(CC)CC2)nc2cccnc2c(=NCC2CCCC(F)(F)CC2)[nH]1 48500,c1(C(=O)Nc2cccc(NC(CC3C(CC)C3)=O)c2)c(Br)c(C)nn1C 48501,N1(C(C(C)OCC#C)=O)CCC2CN(C(C3C=CCS3)=O)C2C1 48502,C1(F)(C(N2CCC(NC(Cc3c(C)con3)=O)CC2)=O)CS(=O)(=O)CC12CCC2 48503,c1(C(N2C(CCNC(c3csc(Cl)c3)=O)CC(OC)C2)=O)cnc2nccn2c1 48504,Cc1cc(F)sc1C(=O)NC1CCC(CCNC(c2ccc(C3CC3)o2)=O)C1 48505,C1(NC(=O)CSC2CC2)CN(C(=O)C(O)CC2CCOCC2)Cc2ccnn2C1 48506,N1(C(CCC)=O)CCCC1C(=O)N(CCCN(C)C(C1CCC1OC)=O)C 48507,c1(C(c2n(CCOCC)nnn2)N)cnc2c(c1)CCC2.C(CCO)CC1CCC1 48508,c1(C(=O)OCC)ccc(CCNC(=O)C(=O)NC(C)C(C)(C)C#N)cc1 48509,N1(CC(N2CC(NC(=O)OC(C)(C)C)OCCC2)=O)CCCC2(CC2)S1(=O)=O 48510,CCCCCCC(=O)N(CCNC(c1sccc1C1CC1)=O)CC 48511,C1(C(N2CCCC2CCCO)=O)C2CN(CCO)CC12.c12cnn(c1)CCN2 48512,Cc1cc(C(N2CCCC(NC(C3C=CCC3)=O)C2C)=O)c(O)c(C)n1 48513,c1(OC)cccc(C)c1C(N1CC2CC1(CNC(C1CC3(CCC3)C1)=O)C2)=O 48514,N1(C(COCCC)=O)CCCC2(CCCN2C(=O)COCC2CC2)C1 48515,C1(NC(C(CC)N(C)C)=O)CCN(C(=O)Cc2cncn2C)C12CCC2 48516,n1(CCC2(c3nnnn3C(C)CC)CC(OCCC)C2)ccccc1=O 48517,C(C)(C(C(=O)N1C(CO)CC1CO)C(C)C)NC(C1ON=C(CC)C1)=O 48518,C1(CC(=O)NCc2cc(C(N)=O)no2)(NC(C2(CC)CC2)=O)CCCCC1 48519,c1(C(N(CCC)CCNC(C2CC=CC2)=O)=O)ccnc(-n2cccc2)c1 48520,c1(NC(c2c(NC(C(CCC)C)=O)ccs2)=O)ccc(Cl)cc1Br 48521,c1(C(=O)NC2CC(CNC(C(n3ncc(C)c3)C)=O)C2)ccc2cccnc2c1 48522,CC1CN(C(c2nnn(C)c2C(F)F)=O)CCC1NC(c1cc(Cl)cnn1)=O 48523,C#CC1(O)CCN(C(C2CCCC(NC(=O)CNC(=O)NC)C2)=O)C1 48524,C1(CCC=C)CCCN(C(C23CC2CCN3C(=O)C(=O)NOC)=O)C1 48525,CC1CN(C(=O)CC2CCCCCC2)CCC1N(C)C(c1cc(CF)on1)=O 48526,CC(C(C(=O)N1CC(C(=O)NC(C)(C)C)C1)N(C)C)OC(c1ccc[nH]1)=O.N(C)(C)C 48527,C=CCC(CC)C(=O)N1CC2(CC(CC(N3CCC(c4ccon4)C3)=O)C2)C1 48528,c1(NC(C2CC(C)CN2C(=O)Cc2ccc(Cl)s2)=O)ncnc2c1c(Br)cn2C 48529,C12(C(N(CC(=O)NC(c3cnccn3)C)CC3CC3)=O)CCCC1C2(F)F 48530,c1(CC(N2C(C(=O)NCc3cccc(C)n3)CCCC2)=O)cccc([N+](=O)[O-])c1 48531,CC1CCCC(NC(=O)C(C)CN(C)C(c2cnn(C3CC3)c2)=O)C1 48532,c1(NCC(NC(CCCOCC)=O)NC23CC(C2)C3)ccc(OCC2CC2)cc1 48533,c1(C(=O)OC)cn(C)[nH]c1=NC(=O)C(c1ccccc1)OC(c1ccccc1)=O 48534,c1(C(N2CC(NC(CN(C3CC3)CC)=O)C(C)C2)=O)c(C(F)F)nn(C)c1C 48535,N1(C(COC)=O)CC(CNC(c2c(F)ccc(Br)c2Cl)=O)C2(CCC2)C1 48536,c1(C(N(CCNC(C2C(CC)C2)=O)CC)=O)cnc(C(F)(F)F)c(F)c1 48537,C(=O)(C1=CCN(C(C2CCNC(=O)C2)=O)CC1)NCC(C)(C1CC1)OC 48538,C(CCCCC(=O)NCC1C(C)CCN1C(=O)CC1(C)CC1(Cl)Cl)OCC 48539,C(=O)(CCCCC(F)F)NCCCC(CCC)NC(=O)C(F)(F)C(O)C1CC1 48540,C1(CNC(C(CC)N(C)C)=O)(CNC(C23CC(C(F)F)(C2)C3)=O)CC(F)(F)C1 48541,CCC(CCOC)C(=O)N1CC(CN(C(=O)C(C)(C)n2cnnn2)C)C2(CC2)C1 48542,N1(c2cc(C(=O)OC)nc(Cl)n2)CC2(C1)SCCC2NC(=O)Cc1n[nH]c(C)n1 48543,c1(NC(=O)NC)ccc(NC(C2(NC3(C)CCC3)CC2)=O)c(OC)c1 48544,C1(C)(CC)COCCC1NC(=O)NN1CC(CS(=O)(=O)C(F)F)C1 48545,N1(C(C(COC)OC)=O)CC2CCC(NC(=O)CCS(C)(=O)=O)C2C1 48546,c1(C(=O)OC)cccc2c1CCN(c1cccc(Cl)c1S(=O)(=O)OC)C2 48547,c1(CNC(C(C)NC(=O)OC)=O)ccc2nccn2c1.C12CN(C1)CC(=O)NC2 48548,Cc1cc(=NC(C)CCCC(F)(F)F)[nH]c(=NCC2CC23CCC(O)CC3)[nH]1 48549,C1(C(N(CC)CC2CCCO2)=O)C2CC3C(C2NC(C2CCSCC2)=O)C13 48550,c1(C(=O)NC(C(C)NC(COC(C)=O)=O)C)cnc2snc(C)c2c1 48551,c1(CC(=O)NC2C(C)CN(C(=O)CCCCN(C)C)C2)ncn2c1CCC2 48552,CCC(C)(C(=O)N1CCC(N(C(=O)C(O)Cc2cnc[nH]2)CCO)C1)OC 48553,C1(NC(c2c(CC)cccn2)=O)CC(OC)CN(C(=O)C(C)(C)CO)C1 48554,O=C(CCCC(F)F)NCC1CCN1C(c1ccc(CO)nc1)=O 48555,C1(=CCNC(c2ccc(SC(F)(F)F)cc2)=O)CCN(C(=O)C(O)CF)CC1 48556,C1(C(=O)NCCC(CNC(C(C)C#N)=O)(C)C)CC(F)(F)CCC1(C)C 48557,N1(CCc2ccccc2)CCN(Cc2nnnn2CC2CC2)CC1.c1ccccc1 48558,C1(C(=O)NC(c2ccccn2)(C)C)CCCCC1NC(C1CNC(=O)C1)=O 48559,c1(CC)ccnc2nc(=NC(=O)c3n[nH]cc3COC(C3COC3)=O)[nH]n12.C(C)(C)C 48560,N1(C(CCC(C)C)=O)CCC2(CC1)CC(C)N(C(=O)CN1CCOCC1)C2 48561,C(=O)(C(C)CC(C)CC(C)C)NCC1(C)C(C)CN(C(C(C(CC)(C)C)O)=O)C1 48562,CCC(CC(=O)N(C1CC(NC(=O)Cc2cc[nH]n2)C(O)C1)CC)C(C)C 48563,CC(C(=O)OC(C)(C)C)C(=O)N1CC=CC1CNC(=O)C=Cc1nccs1 48564,C1(C(=O)NC2(CC=C)CN(C(=O)C(C)C)C2)C2CC2C2CC12 48565,Cc1noc(C)c1CC(C)C(=O)NCC1CCN(C(=O)CCc2cccnc2)C1 48566,C(C1CSc2ccccc21)NC(=O)CCOC1CCCCC1.c12cn(nn1)C2 48567,c1(C(c2n(CCCSC)nnn2)NCCN(S(C)(=O)=O)C)cc(F)cc(C#N)c1 48568,C(C)(CN=c1ccnc(N2CCOC(CSc3ccccc3)C2)[nH]1)SC 48569,C=CCC(CNC(c1cc(Cl)no1)=O)C(=O)NCc1cc(C)cc(O)c1 48570,c1(CN2CCCC(NC(CCC(C)C)=O)CC2)cc(Cl)c(O)cc1F 48571,Cc1cc(F)ccc1C(=O)N(CC(C)C(=O)N(C)Cc1cccc(F)c1)C 48572,c1(C(N(CCC(C)NC(C2(OCC)CCOCC2)=O)C)=O)cc(F)c(Cl)cc1F 48573,Cc1cc(C(F)(F)F)sc1C(N1CC(C)C(F)C1)C(=O)NC1CCC1 48574,Cc1cc(=NCCN(C)C(C2Cc3cccc(C)c3O2)=O)[nH]c(C)n1 48575,C1(CC(=O)NCC(C)(C)CC2CN(C(c3ccncn3)=O)C2)CCC=CCC1 48576,Cc1ccc(-c2ccc(NCc3scnc3C)cc2)cc1Br 48577,C1(NC(c2ccc(C#C)nc2)=O)CN(C(C2(C)CCC2)=O)CC12CCC2 48578,N1(CCC(CC)C)CCC(O)C(C(=O)NCCc2ccc(OC(F)(F)F)cc2)C1 48579,Cc1ccc(C)n1CC(N1CCC=CC1C(=O)NOCC1CCOCC1)=O 48580,N(C(=NCC1CN(C)S(=O)(=O)c2ccccc21)N1CCCC2(CCOC2)C1)C(C)C 48581,c1(COCC)cn(C2(C(=O)N(CC(F)F)Cc3ccccc3)CC2)nn1 48582,N1(C(c2sncc2Br)C(=O)NCCCCCC)CCCC(NC(=O)OC)C1 48583,CC1CCC(C)N1CC(=O)NC1(C)CCN(C(c2c[nH]nc2C2CC2)=O)C1 48584,N1(C(CC=CC)=O)CCC(C2CCCN(C(=O)CS(=O)(=O)CC)C2)C1 48585,CC(C)CCCCCC(=O)NC1CCN(C(c2cnn(C3CC3)c2)=O)C1 48586,c1(C(=O)NCC2CCN(C(C3CNC(=O)N3)=O)CC2)csc2cc(Cl)cnc12 48587,CCC(CC)(C(=O)N1CCCC(C(=O)Nc2ccc(OC)c(Cl)c2)C1)OC 48588,N1(C(c2c(C)nncc2)=O)CCN(C(=O)CC2(n3cccn3)CC2)C(C)C1C 48589,CC#CCC(C(=O)NCC1CC12CC2(F)F)NC(c1ccc(C)cn1)=O 48590,CS(=O)(=O)CCC(=O)NC(C(=O)NOCCCF)c1cccs1 48591,c1(OC)cnc(Cl)cc1C(N1CCC(NC(=O)C(C)(Cl)Cl)C(C)C1)=O 48592,C1(C(C)(C)C)(CNC(C(C)OCC)=O)CCN(C(C2CCC(N(C)C)CC2)=O)C1 48593,C(=O)(C1=NOC2(CCC2)C1)N1CC(C)N(C(=O)CCP(C)(C)=O)CCC1 48594,c1(C(=O)NCC(C)CN(C)C(C2CC(O)CN2C)=O)n[nH]c2c1COCC2 48595,C1(NC(C2CCN(C)CC2)=O)CN(C(=O)COCC2CCCC2)CC12CC2 48596,C(=O)(C1(C)CCn2ccnc21)NC(C(C)C)CCN(C)C(C1CSCCS1)=O 48597,C(=O)(CCC(=O)NN(C)C)NC(CC#CC)C(=O)NCc1oc(C)nc1C 48598,N1(C(C2(C)CCCN(C(COCCCC(C)C)=O)C2)=O)CC(C2CCCCC2)C1 48599,CC1(C)CC(CNCCc2c(F)cccc2F)CCO1 48600,Cc1ccc(C(N2CCCC(NC(=O)C=CC(=O)OC(C)(C)C)C2CO)=O)c(Cl)c1 48601,C(CCCN=c1[nH]nc(-c2ccon2)s1)Oc1ccc(NC(C=CC)=O)c(C)c1 48602,N1(C(c2c(C)sc(-c3ccccc3)n2)=O)CC(F)(C(=O)O)C2(COC2)C1 48603,C1(N(C(C2N(C(c3c(C)csc3)=O)CC(O)C2)=O)C)CNC(=O)C12CC2 48604,CCC(CC(=O)NCC(C(C)C)NC(c1cccc(O)c1F)=O)C(F)F 48605,c1(C(N2CCCN(C(C(N)=O)=O)CC2)=O)cccc2c3c([nH]c12)CCCCC3 48606,N1(C(CCCN(C(C(C(C)C)C2CC2)=O)C)=O)CC(=O)NCC12CC2 48607,S(=O)(=O)(c1ccc(Cl)nc1)N(C(C)CNC(C1COC2(CCNCC2)C1)=O)C 48608,Cc1n[nH]cc1C(=O)NCCCOCCNC(=O)CNC(N)=O 48609,n1(CC)ncc(C(N2CC(NC(=O)C(C)c3ccsc3)C2)=O)c1C(F)(F)F 48610,CC1=C(C)CC(C)(C(=O)NC2C=CCN(C(c3ncsc3S(N)(=O)=O)=O)C2)CC1 48611,C=CCCCCC(=O)NCC1CCC(Cn2cc(C3CC3COC)nn2)CC1 48612,CC(CC1=CCCCC1)NC(=O)CCN(C(=O)C(O)CCN(C)C)CCO 48613,N1(C(c2cc(C)no2)=O)CCC(C)C(CNC(=O)CCCOC(C)(C)C)C1 48614,C1(C(N2CC(C3CN(C(CNC(C)=O)=O)C3)C2)=O)Cc2cccc(Cl)c2C(=O)O1 48615,C(=O)(CCCCC(N)=O)N1CC(C=C)(CC(=O)NCCC2=CCOCC2)C1 48616,Cc1ccc(C)n1CC(N1CC(C)CC1C(=O)NCCc1cc(O)ncn1)=O 48617,Cc1cccc(C)c1OCC(=O)NC1CCN(C(=O)CC2CCC2)C1C(C)(C)C 48618,C1(CC(=O)N(CCNC(c2sccc2C(F)F)=O)CC)SC2=NCCN2C1=O 48619,c1(CC(N2C3(CN(C(c4c(C)nns4)=O)C3)CC2)=O)n[nH]c2ccccc12 48620,c1(OC(Cn2c(N3CCC(OC(C)(C)C)C3)nnn2)=O)ccc(Cl)cc1 48621,C(CCCC(=O)NCCCc1nncn1C)NC(Cc1n(C)ccn1)=O 48622,c1(C(=O)NC2C(CNC(CC3(C#N)CC3)=O)CCC2)ccc2cnoc2c1 48623,C1(NC(=O)C2=NOCC2)CC2(CCN(C(C3CCCCC34CC4(F)F)=O)CC2)C1 48624,CC1COCCC1N(C(=O)C(C1CCCO1)NC(=O)CCC1CCC(=O)C1)C 48625,N1(C(CN(CCOC)C)=O)CCCCC(C2CN(C(C)=O)C2)C1.C(C(C)(C)OC)NC 48626,C=CCC(C(=O)NC(CC(N)=O)C(=O)Nc1cc(C)cc(O)c1)C(C)C 48627,N1(C(C2(C(C)=O)CC2)=O)CCC(C2CCN(C(c3ccc(Cl)s3)=O)CC2)C1 48628,c1(NC(C(COC(C)C)NC(C(CC)OC)=O)=O)ccc(OC(C)C)c(C)c1 48629,c1(C(=O)NC(C2CN(C(C3CCS(=O)(=O)C3)=O)C2)C)cnc(-c2ccoc2)[nH]c1=N 48630,N1(C(CC(C)(F)F)=O)CC2COCCC2(NC(c2ccnc3[nH]cnc23)=O)C1 48631,c1(C(=O)NC(C)C(C)NC(C23CC(O)C2C3)=O)ccc(Cl)cc1 48632,C1(NC(CC(CN(C)C)(C)C)=O)C2CC(O)C1N(C(C1CSCCS1)=O)C2 48633,N1(C(c2ccc(CSCC)cc2)=O)CCN(C)C(CNC(=O)C(C)CCO)C1 48634,n1(CCC(=O)N(C(C2CCCCC2)C2CCOCC2)C)ncn(C)c1=O 48635,N1(C(c2sccc2F)=O)CCC(C2CC2)(CNC(=O)C(F)(F)C(F)(F)F)C1 48636,C(=O)(C(C(F)(F)F)=Cc1ccccc1)N1C(CNC(c2c(C)csc2)=O)CCC1 48637,n1(CC(=C)C)nnnc1C(c1nc(C2CC2)cs1)NC(C1CCC1)C1CC1 48638,C1(C2CCC2)(C(=O)NCCCC2(NC(=O)CC3CCCC(=O)N3)CC2)CC1(F)F 48639,n1(CCCC)nc(C)c(C=CC(=O)N(CC(C)C(=O)OC)CCC)c1Cl 48640,Cc1cnoc1C(=O)NCC1(NC(C2CC(n3cnnc3)C2)=O)CCC1 48641,N1(C(C2CCN(CC(C)C)CC2)=O)CCC(NC(=O)CCC(C)(C)C)C(C)(C)C1 48642,C1(C(N2CC(C)SCC2)=O)CC(O)CCN1C(c1cc(O)cc(F)c1)=O 48643,N1(CC(=C)Cl)C2CCC1C(NC(=O)C(C)OCC(=O)OCc1ccccc1)C2 48644,C(CC(CNC(=O)C(O)C1CCCC1)NC(C1(COC)COC1)=O)OC 48645,N1(C(CCC=CC)=O)CCC(NC(=O)CSCC(F)F)CC(O)C1 48646,Cc1cc(C(N2CC(CC(C)NC(c3cccc(=S)n3O)=O)C2)=O)c(F)cc1F 48647,c1(OC)cccc2c(C(=O)N(CC(C)NC(=O)Cc3cncc(O)c3)C)csc12 48648,S(=O)(=O)(c1ccc2c(c1)CC(C(=O)O)C2)NC1CCC(CSC)CC1 48649,c1(C(=O)NC(C(N2CC3(CCC(=O)N3)C2)=O)C2(C)CC2)cccc2cncn12 48650,c1(C(=O)NCC(C)NC(=O)C(O)CC2CCOCC2)cc(Cl)ccc1C(F)(F)F 48651,C1(NS(CCC)(=O)=O)CC2CN(C(c3c(I)ccnc3F)=O)CC2C1 48652,CN1CC(NC(C2C3CC2N(C(=O)C(C2CCCCC2)F)C3)=O)CC1=O 48653,C1(CNC(C(C=CC)O)=O)CCN(C(=O)C=Cc2ccccc2F)CCC1(F)F 48654,C(=O)(CCCC(=O)N1CC(C)(CCC(=O)Nc2cnc(F)cc2C)C1)OCC 48655,C1(OC)CCCC(CNC(C2CC(C)N2C(c2cscc2CO)=O)=O)C1 48656,N1(C(C(C)CC2CCC2)=O)CC2CC(CNC(c3cnc(S)[nH]3)=O)C2C1 48657,c1(C(=O)OC)c(C)[nH]c(CN2CC(NC(c3cnn(C(C)C)c3)=O)C(F)C2)c1C 48658,c1(OC)cc(CNC(C23CC(CCO2)C3)C)cc(OC)c1Br 48659,C(CC(C(=O)N1CCC(NC(=O)N(C)C)C1)NC(C1CCOC1C1CC1)=O)SC 48660,c1(C(=O)NC2C(CNC(C(CC)NC(N)=O)=O)CC2)cc2nc(=O)ccn2[nH]1 48661,C1(N(C(COC)=O)C)CCCC(N(C)C(c2cn(C3CC3)cn2)=O)C1 48662,C1(C)(CNC(CCc2n(C)cnn2)=O)CCN(C(C23CCCCC2C3)=O)CC1 48663,CC1CC(NC(C2COC(=O)N2)=O)CN1C(C1CCN(C2CC2)CC1)=O 48664,N1(C(COC(C)(C)C)=O)CCC(N(C(=O)CC2C=CCCC2)CC2CC2)C1 48665,c1(NCC)ncc(C(N2CC(NC(=O)CCCC3CC3)CC(C)C2)=O)cc1Cl 48666,N1(C(C(C=C)O)=O)CCCN(C(c2nc(OC)c(C)s2)=O)CC1C(C)C 48667,C1(C#N)(C(=O)NC2CCC(NC(c3cccc(CC)c3)=O)CC2)C(C#N)C1(C)C 48668,C1(C(=O)NC(C(C)C)CNC(=O)CCCN(C)C)CCOC(=O)N1 48669,CCC(C)CCC(=O)NC(C)C(C)(C)C(=O)NCCN(CC(F)F)C 48670,C1(N(C(C(C)=C2CCC2)=O)C)CCN(C(=O)Cn2ncccc2=O)CC1C 48671,C(CCC)(C(=O)NC1COCC1CNC(C1CSCCS1)=O)=CCC 48672,N1(C(=O)CNS(=O)(=O)C2CC2)CCCC12CCN(C(C1CC3CCC1O3)=O)C2 48673,C1(C)(CNC(C(C2CC2)NC(CCc2cn(C)nc2)=O)=O)CCCCO1 48674,c1(N2CCCC(O)(C(C)C)C2)cc2nccc(Cl)c2cc1Br 48675,CC(CN(C)C)CC(=O)N1CCC(CC(=O)NC2CC(CN(C)C)C2)CC1 48676,Cc1cc(Br)ccc1CNCC(c1cc(C2CC2)nn1CC(F)F)C 48677,C1(C(=O)NCC2CCCN(C(CN3CCC(OC)C3)=O)C2)CCC2(CCCC2)C1 48678,CCC(CCCC(=O)NC1CCCC1)NC(=O)CN(C)C(C)C 48679,c1(CC)cc(C)c(C(=O)NCC(=O)NCCCN(C(=O)C2=CCCC2)C)o1 48680,N1(C(CN(C(C(C)C)=O)C)=O)CCC2(NC(c3cc(N)cc(F)c3)=O)CC2C1 48681,C(=O)(C(O)CC(C)(C)C)NC(CC)CNC(=O)C=Cc1ccc(OCC#N)cc1 48682,C1(O)(CNC(C2(CCC=C)CC2)=O)CCCN(C(c2nnc(O)nc2O)=O)C1 48683,C1(CC(=O)NC2(c3ccnc(Cl)c3)CC2)CCN(C(C2NC(=O)NC2=O)=O)CC1 48684,c1(CC(=O)Nc2cc(Cl)c(Br)cc2O)cc2ccccc2nc1O 48685,n1(C(C)C)cccc(C(=O)NCc2cn(CCNC(C3CC(F)C3)=O)nn2)c1=O 48686,c1(C(=O)NC2CCN(C(C(C=C)O)=O)CC2)ccc(Cl)c(OC)c1 48687,CCC(C)C(O)C(C)C(=O)N1CCCC(C(=O)N(C)CC2(CO)CC2)CC1 48688,c1(C(=O)NC2CCN(C(C3C(OC)CCC3)=O)C2C2CC2)ccc(C)c(C)n1 48689,N1(C(CN(C)CC)=O)CCC(COC)(NC(=O)COc2c(Cl)cccc2Cl)CC1 48690,C1(C(N(CCCN(C(=O)CC(C)(C)F)C)C)=O)CCCCC1(C)C 48691,C1(N(C)C(C2CN(S(C)(=O)=O)C2)=O)CN(C(=O)C=Cc2cscn2)CC12CC2 48692,N1(C(c2c(OC)nc(C)cc2)=O)CCCCCC(NC(c2cnc[nH]c2=N)=O)C1 48693,N1(C(c2c(OC)ccnc2)=O)CC(NC(=O)Cc2csc(C)c2)CC(F)(F)C1 48694,C(=O)(C1CC(=O)c2ccccc21)NCC(C)NC(c1c(C)cc(C)[nH]1)=O 48695,N1(C(c2cc(C)ns2)=O)C2CCCC1CC(NC(c1c(C)[nH]c(C)c1C)=O)C2 48696,c1(C(=O)NCCOCCN(C(C(COC)(C)OC)=O)C)c(C)cccc1[N+](=O)[O-] 48697,CCCC(C(=O)OC)C(=O)N1C2CCC1CN(C(c1cnc(O)n(C)c1=O)=O)C2 48698,N1(C(C2CC(=C)C2)=O)CCC2(C1)CN(C(=O)C(C1CCC1)OC)CCO2 48699,c1(C(=O)NC2C(NC(Cc3cn(C)nc3)=O)CCC2)ccc2cnnc(O)c2c1 48700,C(=O)(CCC(C)(C)C#N)N(CCNC(=O)CCC1CC1CC1CC1)CC 48701,N1(C(C2(CC)CCCN2C(C2CC2C2CC2)=O)=O)CC2(C1)CN(C)C2 48702,C1(CNC(c2ccnc(-n3ccnc3)c2)=O)CN(C(C2CCOC2=O)=O)CCO1 48703,c1(N2CCC(C(=O)NC(CC)C(N)=O)CC2)cc(OC)nc2ccccc12 48704,c1(C(N(C(C)CNC(C2CC2C(=O)OC(C)(C)C)=O)C)=O)csc(CO)n1 48705,N1(C(C(CC)C#N)=O)CC2CCC(N(C)C(C3CCC=CCC3)=O)C2C1 48706,CCC(C)(C)CCN=c1[nH]c(N2CC(CCOC)OC(C)C2)nc2cccnc12 48707,CC(C)C(=O)C(=O)NC(c1ccnn1C)C(N1CCC(OCCO)C1)=O 48708,N(C(=NCC1COC(=O)O1)N1CC2CC(C1)c1cccc(=O)n1C2)CCN=[N+]=[N-] 48709,C1(NC(Cc2cc(C)ns2)=O)CN(C(=O)C(O)CC(=O)OC(C)(C)C)CCC1F 48710,c1(CNC(C(=O)Nc2cc(OC)ncn2)=O)cc(C)cc(C)c1 48711,Cc1cc(C=CC(=O)NC2CC(NC(C3CNC(=O)O3)=O)C23CCC3)c[nH]c1=N 48712,c1(C(=O)NC2CC(C)(NC(c3cc(C)oc3C)=O)C2)nccc2ncccc12 48713,c1(CN(C(c2cnn(C)c2C)C(=O)NCC)C)ccc(C)c(F)c1F 48714,Cc1scc(C(=O)NCC2OCCC2C(=O)NCCc2ccccc2F)c1C 48715,C1(C(N2CC(OC)C2)=O)CC(C)CN1C(=O)CCC1CC1(F)F 48716,CCC(CC(=O)NC(C)CNC(=O)CC1CC2(CC2)C1)C(C)C 48717,CC(CCC(=O)NCC1CC(CNC(C2(F)CCOC2)=O)C1)c1ccccc1 48718,CC1CCCC1(C)C(=O)NC1CC(CCNC(c2csc(CO)n2)=O)C1 48719,C1(C(=O)NCC(CC)NC(C2(N(C)C)CC2)=O)CCc2cc(OC)ccc2C1 48720,C1(NC(C2CCN(C)C2=O)=O)CC2CC1N(C(=O)CSc1nc[nH]n1)C2 48721,N1(C(CC(C2CC2)NC(c2c(CC)n[nH]c2)=O)=O)CCn2ncc(C)c2C1 48722,CC(C)C(C)C(CNC(c1csc(-c2ccsc2)n1)=O)NC(C1OCCO1)=O 48723,N1(C(C=C(C)CNC(=O)C(F)n2ccnc2)=O)Cc2ccnn2CC1C 48724,O=C1CSC2(CN(C(C34CCC(CC3NC(=O)Cc3ccccc3O)C4)=O)C2)N1 48725,c1(CC(N2CC(CC)(NC(=O)CC3CCCS3(=O)=O)C2)=O)c(C)nc(C)nc1O 48726,C1(C2CC2)(NC(C(C)OC)=O)CCN(C(=O)CCCc2sccc2C)C1 48727,c1(C(=O)NCCN(C(C(CC)n2cccn2)=O)C(C)C)c[nH]cc(F)c1=O 48728,c1(NC)cc(Cl)ccc1C(=O)NC1CC(NC(C2CCCC(O)C2)=O)C12CCC2 48729,N1(CC)CC(C(=O)N2CCC(C)(NC(=O)CS(=O)(=O)CC)C2)c2ccccc21 48730,Cc1nc2c([nH]1)CC(C(N1CCC13CCC3)C(=O)NCC1CC3(CC3)CO1)CC2 48731,C=CC1CCCN(c2ncccc2CNC(c2scc(C(=O)OC)c2C)=O)C1 48732,C1(=CC(=O)N(CCC(C)(C)NC(CC2(C=C)CCC2)=O)C)CN2CCC1CC2 48733,CC1CN(C(=O)C(C2CCCCCC2)O)CC(C)N(C(c2cc(C#N)c[nH]2)=O)C1 48734,Cc1nc(NCc2cccc3c2CNC3=O)cc(=NCC2CCCC2N(C)C)[nH]1 48735,c1(OCC(=O)NC(C2CCOC2)CNC(c2c(C)nc[nH]2)=O)cc(F)cc(Cl)c1 48736,c1(C(=O)NCC2(O)CN(C(CC(CCC)CC)=O)C2)cccc2c1CC(C)(C)C2 48737,C1(NC(c2c(C)cno2)=O)CC(CNC(c2cnc(C)cc2Cl)=O)C12CCC2 48738,N1(C(c2c(Cl)nc3sccn23)C(=O)NC(C)C)CCCCC12CCN(C)C2 48739,C1(CC(=O)N(C(CNC(COCCOCC)=O)C2CC2)C)OCCOC1(C)C 48740,c1(C(=O)NC2(CCC)CC2)ccc(CNC(C2CCOC2C(C)C)=O)o1 48741,Cc1oc2cc(C(=O)NCCN(C)C(C3(O)CC3(C)C)=O)[nH]c2c1C 48742,C1(CCOC)CN(C(=O)C(F)(F)CO)CCN1C(C1Cc2nncn2C1)=O 48743,C=CCC(C)(O)C(=O)NC(C)C(=O)NCC(C)(C)C1CCCO1 48744,C(=O)(C1CCCc2nc[nH]c21)NC(CCNC(c1[nH]nc(OC)c1Cl)=O)C(C)C 48745,CC(C)CC(CCO)NC(=O)C(C)(C1CC1)N(C)C(C12CC(C#N)(C1)C2)=O 48746,c1(C(=O)NCCC(C)N(C(C(CC)n2cccn2)=O)C)cc(C)nc(N(C)C)n1 48747,N1(C(Cc2ccc(OC)cn2)=O)CCN(Cc2ccnn2C)CC1CO 48748,N1(C(CCC=C(C)C)=O)CCC(NC(C2CCCC(O)C2)=O)CC1 48749,c1(CNC2CC(C(=O)NCc3cnc(Cl)nc3Cl)C2)c(F)cc(Br)cc1F 48750,N1(C(CC)=O)Cc2ccccc2C1C(=O)Nc1nc2ccccc2nc1OC 48751,C1(NC(C(CC=C)OC)=O)CC2(C1)CC(C(=O)NCC1C(C)C1C)C2 48752,C1(CN(C)C)CC(O)CN1C(c1n[nH]cc1CNC(c1ncncc1N)=O)=O 48753,CC(F)(F)CC(=O)NCC1CCN(C(=O)CN2CCCCC2=O)C1 48754,C1(NC(CSCC)=O)CCCCC1CC(=O)NOCC(O)C(C)(C)C 48755,C(CN=C(NCc1ccco1)NC(c1ccccc1Cl)C)N(CC)CC 48756,C(CCC(C)(C)C(=O)NCc1cc(Cl)ccn1)NC(C(C(=O)OCC)CC)=O 48757,C(=O)(CCCC(=O)NCc1csc(CNC(c2cnc(OC)s2)=O)n1)OCC 48758,N1(C(Cc2cn(C)nn2)=O)CCCC2(CCC(NC(=O)C(=O)N=S(C)(C)=O)C2)C1 48759,CC1CC2(CCN(C(=O)CS(N)(=O)=O)CC2)CN1C(C1CNC(=O)O1)=O 48760,CC(CC(=O)N(C(c1cncs1)=O)Cc1ccno1)NC(=O)OC(C)(C)C 48761,Cc1n[nH]c(C)c1SCC(=O)NC1(CNC(=O)C(C)c2cncs2)CCCCC1 48762,CC1(NC(c2nnnn2Cc2cccs2)c2cnc[nH]2)CC2(C1)CC2(F)F 48763,C#CCC(CC#C)C(=O)NCC1(C)CN(C(C2(C)CCC2)=O)CC1C 48764,N1(C(c2n(CCC)ncc2)=O)CC2CC1CN2C(c1c(Cl)sc(C)c1C)=O 48765,N1(C(CSCC#C)=O)CCC=CC1C(N1CC(C(C)C)C1C(C)C)=O 48766,Cc1cc(C)cc(C(=O)NCC(CO)NC(c2cnc(Cl)[nH]2)=O)c1C 48767,C1(c2ccccc2)(NC(CCc2cnn(C)n2)=O)CCN(C(=O)C=CC2CC2)C1 48768,N1(C(C2(C)COC2)=O)CCCC(CCCCNC(C23CCCC2(C(N)=O)C3)=O)C1 48769,N1(C(C(C)=C(C)C)=O)CC2CCC(CNC(=O)C=Cc3cccc(C#N)c3)C2C1 48770,Nc1cc(C(=O)NC2CC(CNC(c3ccc(F)s3)=O)C23CCC3)cnc1N 48771,C(=O)(CS(=O)(=O)C1CCCC1)NCC1(C)CCCN1C(C1CCCC12CC2)=O 48772,C=CCCCCC(=O)NC1CC(O)CN(C(=O)C(c2ccccc2)OC)C1 48773,Cc1nc(C)c2c(C)c(C(=O)NCC(C)NC(=O)C(C)C(C)O)sc2n1 48774,C(c1ccc(Cl)cc1)=CC(=O)NCCO.N12CCC(CC1)C2=O.C1(C)(CC)CC1 48775,c1(C(=O)NCC2(NC(c3ncc(N)cc3Cl)=O)CCC2)cnc2[nH]nc(O)c2c1 48776,c1(CN2CC3(CC(C(N4CC(C(N)=O)OCC4)=O)C3)C2)c(Br)cc(F)c(F)c1F 48777,N1(C(C(C)=C(C)C)=O)CCC2(CCN(C(=O)C(=O)Cc3ccccc3)C2)C1 48778,C#CCCCCC(=O)NCc1cc(C(=O)NCC2(C3CC3)CCCO2)n(C)n1 48779,c1(C(=O)NC2C(C(C)C)CN(C(=O)C3=CCCS3)CC2)n[nH]c2ccccc12 48780,C1(CCC(=O)NCc2c(C(C)C)c[nH]n2)CCCCN(C(=O)C2=C(Cl)CC2)C1 48781,C=C(Cl)CC(C(=O)N1CCN(C2CC2)CC1)NC(c1ccncc1NC)=O 48782,c1(CNC(C2CCCSC2)=O)nc2c(s1)CCN(C(C1CCCN1C1CC1)=O)C2 48783,c1(CN2CC(C(=O)NCC3(C(F)(F)F)CC3)SCC2)nccc2occc12 48784,C1(C(=O)NCCC)CCN(C(c2ccc(C)s2)C(=O)NCCCF)CC1 48785,CC(C)S(=O)(=O)C(C)C(=O)N1CCC(n2cc(-c3cncc(CO)c3)nn2)CC1 48786,CCC(C)C(O)C(C)C(=O)N1CC=CC(NC(c2cnc(C)c(C)c2)=O)C1 48787,C1(CC)CCc2sc(C(N3CCN(C(=O)Cc4csnc4C)C(C)C3)=O)cc2C1 48788,C1(C(=O)NC(C)CCNC(c2conc2C(C)(C)C)=O)CCN(S(N)(=O)=O)CC1 48789,C1(NC(C2(F)C(C)C2)=O)CCCCC1NC(c1c(Br)cnn1C)=O 48790,C12(NC(CCS(C)=O)=O)CCCC1N(C(c1cnn3c1CCCC3)=O)CC2 48791,c1(CNC(CCOC(C)C)=O)ncccc1C(=O)NC1CCC1 48792,CCCCC(F)C(=O)N(C1CCCN(C(=O)C(C)(C)OCC)C1)C 48793,N1(C(C(CCC)(C)C)=O)CC2(C(=O)NCc3nc(C)no3)CCC1CC2 48794,c1(NC2CCCN(C(CC(CCC)CC)=O)C2)nccc(C)c1[N+](=O)[O-] 48795,C1(C(=O)NCCOCCC#C)(CC)CCCN1C(=O)C=CCC 48796,CC1CCC(CNC(c2csc(=N)[nH]2)=O)CN1C(=O)CC1(O)CCCCCC1 48797,C(CCCCC(=O)NCC1(NC(c2csc(C)c2N)=O)CCC1)OCC 48798,CCC(CNC(=O)C(C1CCOCC1)O)(CC)NC(c1cnn(C)c1SC)=O 48799,C(=O)(CC(F)(F)CC(=O)N1CC(NC(c2ccc(C)cc2)=O)C(C)C1)OC 48800,c1(C2C(C)C2)ccc(C=CC(=O)NC2(CCNC(C3(C)CC3C)=O)CCCC2)o1 48801,C1(C(=O)NCCC(C)NC(C2(CCCC)CC2)=O)CCCCN1c1ncccn1 48802,C(C)(CCC(=O)N1CC2C(NC(C3CC(=O)N(C4CCCCC4)C3)=O)C2C1)SC 48803,CCC(CC(=O)NC(CN(C)C(c1cccc(C(C)C)n1)=O)CC)OC 48804,C(=O)(C1CCCn2nccc21)NC(CN(C(=O)CSc1ccc(F)cc1F)C)(C)C 48805,N(C1CCc2cccc3cccc1c23)C(N=c1[nH]nc(OCC)s1)=O 48806,c1(OC)c(C)cc(C(=O)NCCC(C)NC(C2(C(C)(C)C)CCC2)=O)cc1Cl 48807,C1(O)(C(C)NC(c2n(CC)ccc2)=O)CCN(c2ncncc2C#N)CC1 48808,c1(C(N(C2CCN(C(c3cc[n+]([O-])cc3)=O)CC2)C)=O)ncc(N)cc1Cl 48809,CCCC(C#N)C(=O)N1CCN(C(=O)Cc2ccncc2Cl)C(CCOC)C1 48810,c1(C(=O)NCC2N(C(CN(C)C(c3ccccn3)=O)=O)CC2)cnn(C2CC2)c1 48811,N1(C(c2ccc(CC)[nH]2)=O)CCOCC1CNC(=O)C(c1ccc(OC)cc1)O 48812,N1(C(CC(=O)NCC)=O)CCC2(CCC(CNC(=O)Cc3cnc[nH]3)O2)CC1 48813,C1(NC(C(C)CO)=O)CN(C(=O)C(C)(C)c2ccn(C)n2)CC2CCCC12 48814,c1(C(=O)NCCC(CNC(CCn2c(C)ncc2)=O)O)cncc2nc(O)[nH]c12 48815,c1(OCC)cc(C(N2CC(C3N(C(C4(OCC)CCCC4)=O)CC3)C2)=O)nn1C 48816,C1(CNC(C23CCC(OC)C2C3)=O)CCN(C(=O)C=CCN(C)C)CCC1(F)F 48817,CCCCCCC(=O)NCC(C(=O)NCC1(C)C=CCCC1)C(C)C 48818,N1(C(C=CCC(C)(C)NC(C2OCC(C)(C)C2)=O)=O)CCC(C2(C)CC2)CC1 48819,C1(CC(=O)N(C(C)C2CC2)CC)CN(C(=O)CCCC2CCCO2)CCO1 48820,c1(C(=O)NC2(CF)CCN(CC(=O)NC(=O)NCC)C2)noc2c1CCCCC2 48821,c1(Cn2cc(CN(C(c3scc(OC)c3)=O)C)nn2)ccc(F)cc1F 48822,C1(O)(CCNC(C2COCCC2(F)F)=O)CCCN(C(=O)CCc2cnoc2)C1 48823,C1(NC(Cc2ccc(C)nc2)=O)CCN(C(=O)CC2OCCCO2)CC1(C)C 48824,c1(CNC)cccc(NC(=O)C(N2CC(CN)C(C)C2)=O)c1 48825,N1(C(c2c[nH]cc(C)c2=O)=O)CC(NC(=O)Cc2nc[nH]n2)C2(CCCC2)C1 48826,C(=O)(C(F)(F)C(C)(C)O)NCC1C(C(=O)NC2CCN(CC)C2)C1 48827,CC(C)C(C(=O)NOCCCN(C)C)C(C)NC(=O)CP(C)(C)=O 48828,C(=O)(C(F)(F)CO)N1CC(OCC)(NC(C2N(CC)CC2)=O)C1 48829,C=CC(C)(CCOC)C(=O)NC1CCC1NC(c1ncoc1COC(C)=O)=O 48830,C1(Nc2cc(NCc3c(OC)cc(C)cc3)ncn2)CC2CCCCCC12 48831,N1(C(C(C)NC(C)=O)=O)CC(NC(=O)C(C)Cc2c(C)n[nH]c2C)C(C)(C)C1 48832,c1(CCC)cc(C(N2CC(C(C)(C)O)(CNC(C3(F)CC3C)=O)C2)=O)no1 48833,c1(C(=O)NC(CNC(C(CCC)OCC)=O)C)c(F)ccc(F)c1Cl 48834,C#CCCC(O)C(=O)N1CCCN(C(C2CCC(F)(F)C2)=O)CC1 48835,Cc1cc(C(N2CCC(C(=O)O)(C(C)C)C2)=O)nc(O)c1 48836,C1(CNC(=O)CCN2CCCCC2)COCCN1C(=O)COC(F)(F)F 48837,C#CCCCCCCC(=O)N1CC(N(C(=O)CNC(c2ncccn2)=O)C)C1 48838,C1(CC=C)(C(=O)NC(C(=O)NCCSCCOC)C2CC2)CCOC1 48839,CC(C)CCC(=O)N1C(CNC(c2ccc(N3CCCC3=O)cc2)=O)CC2CC12 48840,N1(C(C2C(NC(=O)Nc3ccc(F)cc3)CCC2)=O)CCC(CF)CC1 48841,C1(C(=O)NCCN(CCC)C(c2cc(N)ccn2)=O)(CC)CC(C)(C)C1 48842,c1(C(=O)NCC2(O)CN(C(CCN(CC)CC)=O)C2)cc(N)c(F)cn1 48843,C#Cc1ccc(C(=O)NC2CC(C)(NC(c3cccc(C(C)C)n3)=O)C2)cc1F 48844,N(C(=NCCCN1CCOC1=O)NCCOc1ccc(Cl)cn1)CC(C)C 48845,C=C=CCCC(=O)N(C)CC1CN(C(c2nnn(C)c2C)=O)C1 48846,c1(C(=O)NC(C2CCCN(C(c3csc(C4CC4)n3)=O)C2)C)c(O)cccc1Cl 48847,N1(C(c2c(OC)ccs2)=O)CCC(NC(c2cc(Cl)nnc2Cl)=O)C(C(C)C)C1 48848,CCCCCC(O)CC(=O)NCCC1CC(NC(c2nc[nH]c3ncnc2-3)=O)C1 48849,C1(CNC(CN(C2CCC2)C)=O)CCC2(CCC2)CN1C(=O)C(O)C(C)(C)C 48850,Cc1cccc2c1C(NC(C1(C(=O)O)CCSC1)=O)CC2 48851,c1(-c2nc(C)[nH]n2)ccc(C(N2CC(NC(c3cc(Cl)ns3)=O)C(O)C2)=O)cc1 48852,n1(C(C)C)ncc2cc(C(N3CC4CC3CN(C(C3CCSC3)=O)C4)=O)cnc12 48853,C1(CN(C(=O)CS(=O)(=O)N2CCC(C)CC2)CC)CCCCN1C(=O)CC1CC1 48854,c1(OC)cc(C(=O)NCC(CC(C)C)NC(=O)C=CC2CCOC2)n(C)n1 48855,N1(C(CC(C)OC)=O)CCCC(NC(C2CCC(CC(=O)OC)CC2)=O)CC1 48856,N1(C(CC2(C#N)CC2)=O)CCc2c(CNC(=O)CC3=CCOCC3)cccc2C1 48857,c1(C(=O)OC)cn2c(n1)CCCN2C(=O)Cc1nc(Cl)n(C)c1C 48858,CC(C)CCCCC(=O)N1CCCC1C1(O)CN(C(=O)C(=O)NC(C)C)C1 48859,C1(NC(COC2(C)CN(C(C3(C#N)C(C)(C)C3)=O)C2)=O)CCC2(CCCC2)C1 48860,C#CCC(C)(CC)C(=O)NCC1(O)CCN(C(=O)COCCCC)C1 48861,Cc1cc(NC(=O)C(=O)NC(C2COCCO2)C)ccc1NS(=O)(=O)C1CC1 48862,C(CC)(CCCCC)NC(C1(C(C)NC(C2C(=C)C2)=O)CC1)=O 48863,c1(OC(C)C(=O)NCCC(C)N(C(=O)CNc2cccnc2)C)ccccc1Cl 48864,C(=O)(C1CCc2nccn21)NCC1CC(OC)CN1C(c1cc2occc2[nH]1)=O 48865,N1(C(=O)CCc2ccon2)CCC(NC(C2(CC3CCC3)CC2)=O)CC(O)C1 48866,C(CCCC(=O)NOCCO)N(C)C(c1ccc(F)c(O)c1)=O 48867,C(=O)(CCC(F)(F)F)N1CCN(CC2(NC(=O)COC3CCOC3)CC2)CC1 48868,C1(NC(c2c(OC)cnc(Cl)c2)=O)CC2CCC(C1)N2C(C1(C#N)CCC1)=O 48869,N1(C(c2cnc(SC)s2)=O)CC2(CCN(C(c3ccncc3O)=O)CC2)CC1C 48870,O=S(=O)(c1cnccc1N1CC2C3CCC(C3)C2C1)NC(CF)CF 48871,C1(NC(CC2(C)CCOCC2)=O)CC(C(=O)NCc2nnc(O)o2)=CC1O 48872,Cc1ccc2occ(C(=O)NCC3CN(C(C4C(C)C4C)=O)CC(C)(C)O3)c2c1 48873,N1(C(c2cc(C)c(F)c(C)c2)=O)CCN(C(=O)C(O)C(F)F)C2CCCC12 48874,c1(N2CCN(C(C(=O)NCC3C(C)(C)C3(F)F)=O)CC2)ccc(C#N)cc1Cl 48875,C1(C(=O)NCCN(C(=O)CC2CCCOC2)CC)CCC(Oc2ccncc2)C1 48876,C(C)(CC(=O)N(C1CCN(C(=O)Cc2csc(NC=O)n2)C1)CCO)OC 48877,Cc1snnc1C(=O)NC(CC1CCOCC1)C(=O)NCCC(C)N(C)C 48878,C(=O)(CN1C(=O)CCc2ccccc21)NC(C)CCN(C)C(c1ccnnc1)=O 48879,CC1CCCn2ncc(C(=O)NCC3CC(NC(c4ncc(C(F)F)s4)=O)C3)c21 48880,N1(C(CCCOCC=C)=O)CCC(C)(CCNC(=O)COc2ccon2)C1 48881,C#Cc1ccc(C(=O)NC(c2ccccn2)C(=O)O)c(CC)c1 48882,CCCCCCCCCC(O)C(=O)N1CC(F)(CNC(C2C3CNC(=O)C23)=O)C1 48883,c1(CNC(=N)NC2CCN(c3ccc(F)cc3)C2=O)ccc(Cl)cc1Cl 48884,CCCC(CCCNC(=O)CCNC(C1CCCO1)=O)NC(=O)CSC1CC1 48885,C1(C(=O)OC)CCC(C)N(C(=O)Nc2cnc(C(F)(F)F)cn2)C1 48886,c1(CC)cccc(NC(C2(C)CCCN2C(=O)C(c2ccc(C)o2)C)=O)c1F 48887,N1(Cc2cn(CCC=C)nn2)CCCCC(C(=O)N(C)C)C1 48888,C12(NC(c3cnco3)=O)CCN(C(c3ncoc3-c3ccco3)=O)CC1C2 48889,C1(C)(C(=O)NC(C)Cc2ccco2)CC12CCN(c1cc(C#N)ccn1)CC2 48890,N1(C(c2scc(COC)c2)=O)CC2CCN(C(=O)CCCCCF)CC2C1 48891,N12CCCC(C1)CC=CC2=O.c1(CC(=O)NCC2C(C(=O)O)CC2)ccccc1 48892,Cc1ncccc1CCC(=O)N(CC(O)CN(C)C(C1C=CCS1)=O)C 48893,N1(C(COCc2n(C)c(S)nn2)=O)CCC2(CC1)CC2(C)C(=O)NC1CC1 48894,C12(C(=O)NC(C(C)(C)NC(Cc3c(C)n(C)nc3)=O)C)CC(CO)(C1)OC2C 48895,C(=O)(CCCCCC(C)O)NCCC1(NC(c2c(CCC)cccc2)=O)CC1 48896,C(=O)(C(C)(C)CCC#N)NCC(C)(CC(C)C)NC(CC1ON=C(C)C1)=O 48897,c1(CC)cccc(NC(=O)C(Cn2cncn2)NC(c2nonc2N)=O)c1C 48898,C(c1cc2ccccc2o1)=CC(N1C(C(=O)Nc2cc(SC)n[nH]2)CC1)=O 48899,O=C(C(=O)C(F)(F)F)NC1CN(C(c2cn(Cc3cccnc3)nn2)=O)C1 48900,N1(C(c2c(CC)con2)=O)CC2(CC(NC(C3CC(C)(O)C3)=O)c3nccn32)C1 48901,CC(C)(C)C(Cc1ccc(Cl)cc1)NC(c1csc(I)c1)=O 48902,C1(NC(COC2CC(NC(C(CC)N(C)C)=O)C2)=O)CCCOCC1 48903,N1(C(C2(C3(C)CC3)CC2)=O)CC(C(=O)NC2(C)CCSC2)C2(CCC2)C1 48904,N1(C(C(COC)(C)C)=O)CC2(C)CC1(C(=O)NC(C)CCC1CCCO1)C2 48905,C(=O)(C1(C)CCOc2ccccc21)NC(CNC(CC(CC(C)C)C)=O)C 48906,C1(C(N2CC(CCNC(=O)CSc3ccccc3Cl)C2)=O)CCCC2CCCN12 48907,C(=O)(C(CCCC)NC(C1CCCS1)=O)N1C(C=C)CCC1 48908,Cc1nc(C(=O)NC2CCN(C(c3cnn(C)c3Cl)=O)CC2C)c(C)n1C1CC1 48909,C#Cc1cccc(C(N2CCC(CN(C)C)C2)C(=O)NC2CCOCC2)c1 48910,C#CCCCCCCC(=O)N1CC2CN(C(c3c[nH]nc3C(F)(F)F)=O)CCC12 48911,N1(C(C2C3COCC23)=O)CCC(CNC(CC2CCN(CCC)C2)=O)CC1 48912,C12(C(=O)NC3CC(N(C(CC4C(C(=O)OC)CC4)=O)C)C3)CCC(OC)(CC1)C2 48913,NC(=O)N=Nc1ccc(C(=O)NCC2CC(NC(C3CCCN3C=O)=O)C2)cc1 48914,n1(C(CC)C)ncc(CNC(=NCC2CC2CN2CCCC2)NC2CC2)c1C 48915,Cn1nc(-c2nc(C3CC34CC4)nn2C2CCCSC2)c2c1CCCC2 48916,N1(C(CC(CNC(=O)CC=C(Cl)Cl)OC)=O)CC(C)(C2CCC2)C1 48917,N1(C(Cc2cccc(C)c2)=O)CC(NC(c2cncn(C)c2=O)=O)CC1(C)C 48918,c1(OC)ccc(F)cc1CNCC1CCCN1C(c1cccc(Br)c1OC)=O 48919,CC1CN(C(C2(C)CCCN2C)=O)CCC1C(N1CCCC(O)(C(N)=O)C1)=O 48920,n1(CC=C)cccc1C(=O)NCC(C)NC(=O)Cc1ccoc1C 48921,Cc1noc2nc(C3CC3)cc(C(N3CCCC(F)(F)C3)=O)c12 48922,C1(NC(C2CN(C)C(=O)C2)=O)CC2CCCC(C1)N2C(c1cccn1C)=O 48923,C1(C(=O)NCC=CCNC(C(C)=CC)=O)CCCCCS1(=O)=O 48924,c1(OC)cc(F)c(C(N2CCC(NC(C3(C)CC3(C)C)=O)CC2)=O)cc1N 48925,c1(C(N(CC(O)CN(C(=O)C(F)CC2CC2)C)C)=O)cccn2ccnc12 48926,C(c1ccccc1)=C(C(=O)NC(C)CN(C)C(c1cccnc1)=O)C#N 48927,n1(CCC)ncc(C(N2CCC(C(=O)OC)C2)C(=O)NC)c1C 48928,CC(C)(CCCF)NC(C1(C2CCCN2C(=O)CC=C(Cl)Cl)CC1)=O 48929,C1(C(N2CC(OCCCCC)C2)=O)CCN(C(c2cc(C)c(C)cn2)=O)CCO1 48930,c1(C(N2CCC(O)(CNC(CN3C(C)CC3)=O)C2)=O)cc2scnc2[nH]1 48931,Cc1ccc(C(C)OC(c2scnc2C2CC2)=O)s1 48932,N(C(=NCCOC1CCCCC1)NCc1ccco1)C1CC(OCCOC)C1 48933,C1(C(C)(C)C)(CNC(CC=C)=O)CCN(C(=O)Cc2ccnc(OC)c2)C1 48934,CC1CCCC1(C(=O)NCC1CCCC1CF)NC(=O)C=Cc1cocn1 48935,C(=O)(CCCCC(C(F)(F)F)NC12CC(C)(C1)OC2NC(=O)OC(C)(C)C)OC 48936,N1(C(CC(C(=C)C)O)=O)CCCN(C(c2ccccc2Br)=O)CC1CO 48937,C#Cc1ccccc1CC(N1CC(CNC(=O)CC(=C)Br)CC1C)=O 48938,c1(C(N(CCCNC(c2ncccc2C2CC2)=O)CC)C)ccc2n[nH]cc2c1 48939,NC(CCSC(F)(F)F)C(=O)NC12CC(c3ccccc3)(C1)C2 48940,Cn1cc(C(=O)NC2(CNC(C3CCCC(C(F)(F)F)C3)=O)CC2)c(O)n1 48941,C1(C(=O)NCC(N2CCCCC2)=O)CC2CNCC1O2 48942,C(C(C)(C)CC(=O)N(CCCNC(C1CCCN1S(C)(=O)=O)=O)CCO)OC 48943,c1(C(N2C(CNC(CC=CCC)=O)CCCCC2)=O)ncc(Cl)c(N)c1Cl 48944,c1(NC(C23C(CN(C(c4cc(OC)c(I)cc4)=O)C2)C3)=O)ccc(F)cc1C#N 48945,n1(CC)c(C(=O)N(C2CCCCC2)CCNC(=O)CCOC2COC2)cnc1O 48946,C1(CNC(C(N2CC(C)C2)C)=O)N(C(c2cnn3c2SCC3)=O)CCCC1(C)C 48947,C(=O)(C(C(C)C)C(C)C)NC1(CCNC(c2c(C)cc[nH]2)=O)CCC1 48948,N1(CCNC(C2(F)C(C)C2)=O)CCN(C(c2cscn2)=O)CC1 48949,C(C#CCN=c1[nH]ccc(=NC2CC3COCC(C3)C2)[nH]1)OC 48950,Cc1cc(Br)cc2c1CN(C(=O)Nc1cnc3c(c1)CCOC3)CC2 48951,CC1ON=C(C(=O)NCC2CN(C(=O)C(N)=O)CCCO2)C1C 48952,CCC(C)C(C(=O)NC(C)CN1CCN(C(=O)CC2CC(C)C2)CC1)NC(N)=O 48953,N1(C(c2c(OC)nc(C)cn2)=O)CC2CCC(C1)N(C(c1oc(C)nc1C)=O)C2 48954,C1(C(N2CCN(CC=C)CC2)=O)CCCCCC1NC(c1ncoc1C(C)C)=O 48955,C12(NC(c3cnco3)=O)CCCC1N(C(c1cc(-c3ccccc3)co1)=O)CC2 48956,C12(NC(CCS(C)=O)=O)CCOCC1CN(C(C1(c3ncccc3F)CC1)=O)C2 48957,C=CCC(C(=O)NC(C1(O)CN(C(c2cccc3ncsc23)=O)C1)C)C(C)C 48958,N1(CC(=O)NC2C3CN(C(c4[nH]n(C)c(=O)n4)=O)C2C3)CCC(=O)NC1=O 48959,c1(C(N2CC(NC(c3c(CC)onc3)=O)C3(C2)CC3)=O)ccc2n[nH]cc2c1F 48960,C1(C(N(OC)C)=O)CC(C)CN(C(=O)C#CC(C)(C)C)C1 48961,C1(C(N2C(CNC(=O)Cc3cccnc3)COCC2)=O)CCc2ccccc2O1 48962,CC1CN(C(=O)C(F)=CC2CC2)CCC1N=c1cc(C(N)=O)nc(Cl)[nH]1 48963,CS(=O)(=O)c1csc(C(=O)NC2CCC(CCNC(=O)C(F)=C3CCCC3)C2)c1 48964,c1(C(=O)NC2(c3ccccc3)CCN(C(C(C=C)O)=O)C2)cc(C)nnc1O 48965,C1(C(=O)NCC(CC)NC(=O)CCc2cn(C)nn2)CCCC1c1ccccc1 48966,C12CCCCN(C1)CC2=O.c1(CC(=O)NC(=O)C(F)(F)F)ncccc1F 48967,C(=O)(C(C)(C)C#N)NC1C(C(N(C(C(C)C)CO)C)=O)CCC1 48968,c1(C(N(C2CCCC(NC(=O)C(C)(C)C)C2)C)=O)cc(C2CC2)cc(Cl)c1 48969,N1(Cc2c(C)nccc2)CC2(CCC(C(=O)Nc3oncc3C#N)O2)C1 48970,Cc1nn(CC(F)F)c(C)c1C(N1CC2C(N(C(=O)CC3C=CCC3)C)C2C1)=O 48971,C(CCCCC(=O)N(C(C)CNC(C1CC(OC)C1)=O)C)=CC 48972,C(C(C)(CO)NC(=O)Cc1cccnc1)NC1(CCNC(=O)OC(C)(C)C)CC1 48973,CC(C)CC(O)C(C)C(=O)N1CCC(C)(C(=O)NCC2CCCCC2(C)C)CC1 48974,CC1CCCC=C1C(=O)NC1CCN(C(=O)CC(F)(F)C(F)F)CC1(C)C 48975,c1(OC)cc(C(=O)NCC(O)CNC(C23CC(CO)(C2)OC3C)=O)cc(OC)n1 48976,c1(C(N2CCC(N(C(=O)CCN(C)CCO)CC)C2)=O)ccc(F)cc1C(F)F 48977,N1(C(C2N(C(c3c(C)c[nH]c3)=O)CC2)=O)CCC2(CCCO2)C1 48978,C=CC1CCN(C(C2CCN2C(=O)CSCC)=O)CC1 48979,C(CCC(C)C)(C(=O)N(C)CCc1ncccn1)NC(C1C(CCC)CCC1)=O 48980,CCS(=O)(=O)C=CC(=O)N1CCC(C)(C)C(CNC(c2cccn2C2CC2)=O)C1 48981,C1(OCC)CC(CNC(=O)CN(C)C(c2cc[nH]n2)=O)C1 48982,C(c1cn(C)cn1)=CC(=O)NC(C(=O)NC(c1onc(C)n1)CO)CO 48983,C(=O)(CC1=NN(C)C(=O)C1)NCC1ON=C(C(=O)N(C2C(C)C2)C)C1 48984,N1(C(c2c(CC)cns2)=O)CC(O)CCC1C(=O)NCCn1ncnn1 48985,C(=O)(NNC(=O)C1CCCS1)NC(Cc1cc(C)[nH]n1)C 48986,N1(C(C(CC)(C)O)=O)CCCCC2(C1)CN(C(c1nn(C)cc1C)=O)C2 48987,c1(C(N2CC(O)(C(C)NC(C(CCCC)O)=O)C2)=O)cc(=O)c2ccccc2o1 48988,C1(C2CCCN(C(C3(CO)CC3)=O)C2)(NC(=O)C=CI)CC1 48989,Cc1cc(=NCC2CC(C)CC(C)C2)[nH]c(=NCCS(=O)(=O)C(F)F)[nH]1 48990,N1(C(CC2(OCC)CC2)=O)CCOCC(CC(N2CCC(C)(C)C2)=O)C1 48991,C1(C(=O)NCC(CN(C)C(c2c[nH]cc2C(C)(C)C)=O)O)C2CCCC12 48992,CCCCCC(O)C(=O)N1C(C)C2CC1C2NC(C1(C(F)(F)F)CCCCC1)=O 48993,c1(C(N(C2CCCN(C(=O)C=C3CC3)CC2)C)=O)ccc(N)c(Br)n1 48994,CCC(C)(C)CC(=O)N1CCOC(C)(CNC(=O)CC(C)OC)C1 48995,c1(C(=O)NCC2(NC(c3ccc4c(c3)NCC4)=O)CC2)cnc2[nH]ccc2n1 48996,N1(C(C=C(C)C)=O)CCOCC(CNC(C2CC(=O)N(C)C2)=O)C1 48997,c1(OC)ncc(Br)cc1CN(C1CCN(C(C2CCN(C)C2)=O)C1)C 48998,C=CCC(CC(C)C)C(=O)N1CC(NC(c2cc([N+](=O)[O-])n[nH]2)=O)CC(C)(C)C1 48999,C1(C2CCOCC2)(C(=O)NCC2N(C(CCCN(C(C)C)C)=O)CC(O)C2)CC1 49000,N1(C(C=C(C)C2CC2)=O)CC(O)CC1(C)C(=O)N(C)CC1(C)CC1 49001,Cc1sc(O)nc1C(=O)NCCC1CCCN(C(C2(N3CCCC3)CC2)=O)C1 49002,CC(C)CC(C)CC(=O)NC1(C)CCN(C(C2(C#N)CC2)=O)C1 49003,c1(C(=O)NCC(CNC(C(CN(C)C)N(C)C)=O)(C)C)cnc2ncccc2c1 49004,C1(C(=O)NCc2cnc(C)s2)CNC(=O)CN1C(c1n[nH]c2c1CCC2)=O 49005,c1(C(=O)NCCCN(C(C)C)C(C2CCCCC2(F)F)=O)cccc2occc12 49006,C(C(C)(O)CC(=O)NC(CNC(c1cc(C(N)=O)ccc1C)=O)CC(C)C)OC 49007,N1(C(Cc2ncc(C)s2)=O)CCOC(CNC(C2CN(C3CCCCC3)C2)=O)C1 49008,CC#CCCCC(=O)NC1CCC1CNC(c1ncn(CC)n1)=O 49009,CCC(CC(=O)NC(C)CC(C)NC(c1c(C)cncc1C)=O)C(C)(C)C 49010,C(=O)(CC(C)C)NC(C(=O)N(CCOC)CCOC)c1cccs1 49011,C1(NC(C(CO)N(C)C)=O)C=CCN(C(c2ccnn2-c2cccnc2)=O)C1 49012,N1(C(=O)OC)CCCC1C(=O)N(C1CC(NC(c2cn(C(C)C)cn2)=O)C1)C 49013,c1(CN2CC(CNC(C3(CC)CCNC3=O)=O)OCC2)c(F)cccc1Cl 49014,Cc1ccc(C)c(C(=O)NC2CC3CC2N(C(C2(O)CC2(C)C)=O)C3)n1 49015,C(=O)(C#CC1CCCCC1)NCC1N(C(c2cc(C)n(C(C)C)n2)=O)CCC1 49016,C1(CNC(=O)CCCC2CCC2)CC2(CCC2)CN1C(=O)Cc1ccncc1Cl 49017,N1(C(CNC(CCC)=O)=O)CC(F)CC1CNC(c1c(C)ncn1C)=O 49018,c1(C(N2CCC(C)(CCNC(CCOC(C)=O)=O)C2)=O)cnc2ccncc2c1 49019,n1(CCC(=O)NC2CC(NC(CN3CCC(C)(C)C3)=O)C2)cc(S(N)(=O)=O)cn1 49020,C(=O)(NNc1cc(F)cc(F)c1)N(CCN)CCc1ccccc1 49021,c1(CNC(c2csc(CO)n2)=O)cccc(NC(C2CCC(O)C2)=O)c1 49022,N1(C(C2N(C(CNC(=O)NC)=O)C(C(C)C)CC2)=O)CCOCC1C(C)C 49023,CS(=O)(=O)c1cscc1C(=O)NCC(CO)NC(C1(F)CC=CCC1)=O 49024,c1(-c2cnc(=NC)[nH]c2)cnn2cc(C(N3CCCC(C)(O)C3)=O)cnc12 49025,c1(C(C)=O)cc(S(=O)(=O)N2Cc3cccc(C)c3C2)cc2c1CCC2 49026,CC(C)CC(C)(O)C(=O)N1CCCC(CNC(=O)C#CC2CCC2)C1 49027,Cn1ncc(CC(=O)NC2CCC(NC(c3ccon3)=O)C2)n1 49028,c1(N(C2CCC(NCC(=O)O)CC2)C)ccc2c(c1)C(NC(N)=O)CCC2 49029,CCC(C#N)C(=O)NC1CC(CNC(=O)C(c2ncccc2F)(F)F)C1 49030,C(=O)(C(CNC=O)c1ccccc1)NCC#CCNC(C(C)N(C)C)=O 49031,CC1(C(N2CCCC(O)C2)=O)CCCN(Cc2ccccc2-c2cccs2)C1 49032,c1(C(=O)NC(CN(C(c2c(CC)non2)=O)CC)CC)coc2ccccc12 49033,c1(C(C(=O)NCCOCC)N(c2ncc(Cl)s2)C)ccc(C#N)cc1 49034,c1(C(N2CCCC(N(C(C(C)=C3CC3)=O)C)C2)=O)ccc2cc(C)cn2c1 49035,n1(CCC(=O)NC2CN(C(c3c(C)ncnc3)=O)C2)cc([N+](=O)[O-])nc1C 49036,c1(C(N2C(C(=O)NC3CCN(C(C)C)C3=O)C=CCC2)=O)ncc2ccccn12 49037,C1(C2CN(C(C3CCN(C4CC4)C3)=O)C2)(NC(c2cc(OCC)no2)=O)CC1 49038,N1(C(C(CC)SC)=O)CC(CNC(=O)CSC(F)F)C(F)(F)C1 49039,C(CO)(C(C)NC(=O)C(F)(F)c1nccn1C)NC(C(C)N(CC)CC)=O 49040,c1(NC2CCC(SCC)C2)ccc(S(=O)(=O)NCc2nnc(C)o2)cc1C#N 49041,C#CCC(C)(C(=O)Nc1nccnc1CC)NC(=O)C(=O)NC(C)C 49042,C1(C(N(CCN(C(C(CC)(C)O)=O)CC)C2CC2)=O)CCc2ncnc(C)c2C1 49043,C(=O)(C(F)(F)C(O)C1CC1)N(C)CC1N(C(C(C)OCC)=O)CCC1 49044,C(=O)(C(C)(C)C(C)O)NC1(COC)CCN(C(c2ccc(NC)cn2)=O)C1 49045,c1(OC)ccc2cc(C=CC(=O)NC3CCN(C(=O)C(C)C)C(C)C3)ccc2c1 49046,C#Cc1ccc(CNC(C2(NC(=O)CC3CCSC3)CC2)=O)cc1 49047,C#Cc1ccc(C(=O)NC(C(N2CC3CC3(COC)C2)=O)C2CCOC2)c(C)c1 49048,CCCCCS(=O)(=O)CC(=O)N1CCCC2(NC(c3ccc[nH]3)=O)CC2C1 49049,O=C(CCC(CF)CF)NC1COCC1CNC(c1cncc([N+](=O)[O-])c1)=O 49050,CCCCC(C(=O)NC1CCC(CCC(=O)N(CCC(=O)OC)CC)C1)C(C)C 49051,C(=O)(CS(=O)(=O)C(C)C)N(C)CC1CCN(C(c2c(CCC)nco2)=O)CC1 49052,N1(C(c2cnn(CC)c2C)=O)CCN(C(=O)Cc2ncc(C(C)=O)s2)C(C)C1C 49053,C(N(C)N1CC2(C=Cc3ccccc3O2)C1)C1(SCC)CC1 49054,c1(OC)ncc(N(CCCN(C(=O)COc2ccc(Cl)cc2)C)C)nc1C 49055,c1(C(=O)NCCCCC(CO)NC(C2(COC)CC2)=O)cccc2c1OCC2C 49056,C1(NC(=O)C(F)OC(F)(F)F)(CO)CCCN(C(C2(Cl)CC2)=O)C1 49057,c1(C(=O)NC(C(=O)NC2(C(C)C)CC2)Cn2cncn2)c[nH]nc1[N+](=O)[O-] 49058,c1(OC)nc(N2CC3(CCN(C(c4cncc(C)n4)=O)C3)C2)ncc1C#N 49059,NCC(CNCC(=O)NCCOCc1ccccc1)C(F)(F)F 49060,N1(C(C2=NOC(C)C2)=O)CC2CCOC2(CNC(=O)CCC(=O)c2ccc[nH]2)C1 49061,Cc1nc(CC(=O)NCC(CO)NC(=O)CCC2CCC(=O)N2)co1 49062,N1(C(=O)C=CCc2ccon2)CCC2(NC(=O)C=C3CCCC3)CCCC12 49063,c1(OC)ccc(C(N2CCC(NC(c3ccnc(Br)c3)=O)C(O)C2)=O)cc1O 49064,C(=O)(CC(O)COC)N(C1CCN(C(c2ccc(-c3ccccn3)s2)=O)C1)CC 49065,C1(CC(=O)NCC(C)N(C(c2cccc(C3CCC3)c2)=O)CC)CC(C)(C)CO1 49066,c1(C(=O)NCC2(F)CN(C(C3C(C=C)C3)=O)C2)nnn(C2CCOC2)c1C 49067,C(c1ccc([N+](=O)[O-])s1)=CC(=O)NC1CC(O)(CNC(CS(N)(=O)=O)=O)C1 49068,C(C(=O)NNC(=O)c1ccc(I)c(Br)c1)c1cccc(C)c1 49069,CC1CCCCC1(CNC(c1ccc(=N)[nH]c1)=O)NC(C1CCCN1C1CC1)=O 49070,N1(C(C=CSC)=O)CC(N(C)C)C(CNC(c2nnn(C(C)(C)C)n2)=O)C1 49071,c1(OC)ccccc1C(=O)NCC1(F)CC(NC(c2conc2C2CCC2)=O)C1 49072,C1(NC(CCOC(CC(C)C)C)=O)CN(C(=O)CNS(C)(=O)=O)CC1C(F)(F)F 49073,N1(C(c2c(C)ncn2C)=O)C2CCC1CN(C(=O)Cc1ccncc1Cl)C2 49074,CC1CC(CNC(C2(C)CCSCC2)=O)CN(C(=O)CCc2cn(C)nn2)C1 49075,C1(CNC(C=CCC)=O)CCCC2CN(C(c3ccc(CSC)cc3)=O)CC12 49076,N1(C(C2CC(CF)C2)=O)CC2CCCC2(C(N2CCCC(O)(CO)C2)=O)C1 49077,N1(C(CCCSC)=O)CCN(C(C2(C3CCC3)CC2(F)F)=O)C2(CCC2)C1 49078,c1(CC)cc2c(CC(=O)NCCOCCN(C(=O)C=C(Cl)Cl)C)csc2s1 49079,c1(NCC2CCCN(CCC(=O)OC)C2)cc(OC)ccc1[N+](=O)[O-] 49080,C1(NC(c2c(OC)cccc2)=O)CCCN(C(=O)C(=O)CC(C)C)C1C 49081,C1(CNC(c2cccc(O)c2F)=O)CC2CN(C(C3CC4CCC3O4)=O)CC12 49082,c1(C(N2C(COC)(CNC(c3nnsc3C)=O)CCC2)=O)csc(=NC2CC2)[nH]1 49083,C(=O)(C1CCSc2ccccc21)NC(CC=C)CNC(=O)CCCC(=O)OCC 49084,C(=O)(CCC(C)(C)C)N1CCC(C)(CC(N2CC(C)C(CO)C2)=O)C1 49085,C(=O)C#CC1CCOC1.c1(C(N2C(C)(C)CCC2)=O)ncsc1S(N)(=O)=O 49086,c1(C(=O)OC)ncc[nH]c1=NCC1(NC(c2cnc(C(C)O)s2)=O)COC1 49087,C1(CNC(C2(CC)CC2)=O)(C)CCCCC1.C1(N)CCSC1.C1(=O)C=CC(=O)N1 49088,N1(C(C2C(NC(=O)CC3CC4(CC4)C3)C=CCC2)=O)CCc2ccsc2C1 49089,c1(C(=O)NCCN(CCOC)C(C2C(C)(C)C2(F)F)=O)cc(F)ncc1OC 49090,c1(C(=O)NCC2CCC(C(N3CC(C)(O)C3)=O)O2)occ2c1CCC2 49091,c1(NC(C(c2ccco2)NC(COC(CC)CC)=O)=O)ccc(F)cc1O 49092,N1(C(CC(C)Oc2ccccc2)=O)CCCC(C(=O)Nc2cnc(Cl)nc2)C1 49093,C1(C)(C(=O)NCc2cn(C(C)C)nc2)CCCN1C(=O)C=CC=CCO 49094,Cc1[nH]c(C#N)cc1C(=O)NC1(C)CC(NC(C23CCCC2C3)=O)C1 49095,c1(NC)cnc(C(=O)NC2CCCC2NC(=O)CC#N)cn1 49096,CC(C)(C)C(O)C(=O)N1CCCCCC1CNC(c1cnc2sccn12)=O 49097,CCCC(O)C(=O)N1CCC(C)(NC(=O)Cc2nc(C)sc2C)C1 49098,c1(-c2cn(C(CN(C(Cc3nc(C(C)C)sc3)=O)C3CC3)C)nn2)cnccc1Cl 49099,c1(CCC)cc(C(=O)N(C)CCNC(c2ccn(C)c2C)=O)n(C)n1 49100,CCC(CC)(CC)C(=O)N1Cc2occ(C(=O)NCC3CC(F)(F)CO3)c2C1 49101,CC1(C)C(NC(C2(CO)CCOCC2)=O)CC1CNC(=O)Cc1cncnc1 49102,C1(NC(CCn2c(C)ncc2)=O)CC2CC(C1)N(C(=O)C(=O)NC(C)C)C2 49103,N1(C(CCc2cc(C)on2)=O)C(C(=O)NC2CC2C(C)(C)C)CC2CC12 49104,C(=O)(C1=CCCN(C(c2cc(F)ncc2Br)=O)C1)N(CCCN1CCCC1)C 49105,C1(CNC(C(C2CC2)OCC)=O)N(C(=O)C=C2CCCC2)CCCC1(C)C 49106,C12(C(=O)NCCC(=O)NCC(C)C)CCCN(C(=O)OC(C)(C)C)C1COC2 49107,C(=O)(C(O)CC(C)(C)C)NC(C(C)NC(=O)CSc1nccn1C)C 49108,C12(CNC(c3ccc(OC(C)C)cc3)=O)CCC1CN(C(=O)C(F)=CCCF)C2 49109,CCC(C)C(O)C(C)C(=O)N1CCN(CC(=O)NCc2ccc([N+](=O)[O-])o2)CC1 49110,C#Cc1cnn(CC(N2CCC(NC(=O)CC3CCCOCC3)C2C(C)C)=O)c1 49111,C(CC(C)N(C)CCOCCCCC)OCCOC 49112,C=C(C)C(CC(=O)N1CCCCC1C1(NC(c2csnc2CC)=O)CC1)OCC 49113,C(=O)(C(CN=[N+]=[N-])NC(C12CCCC1C2(F)F)=O)N(C1CC2(CCC2)C1)C 49114,Cc1cncc(C(=O)NC2CC2CNC(=O)C=CC(=O)NC2CC2)c1Cl 49115,O=C(CC1CC(CO)CN1C(c1ccc([N+](=O)[O-])cc1)=O)N=c1cc(C2CC2)[nH][nH]1 49116,C(=O)(C(C)C(C)S(C)(=O)=O)N(CCCNC(c1ccc(NC(=O)OC)cc1)=O)C 49117,C(=O)(C1CCc2ccccc21)NCCN(C1CCCCC1)C(c1c(C)con1)=O 49118,C1(N(C(=O)CC2(C)CCC2)CC)CCCN(C(C2(C)CCCOC2)=O)C1 49119,C1(C(=O)NCc2c(C(=O)NC3(C(C)(F)F)CCC3)c[nH]n2)CCNC(=O)C1 49120,c1(NC(c2cccc(OCCC)c2)C)cc(C)c(NC)cn1 49121,N1(C(=O)CCOC2CCC2)CC2(CC2)CC1CNC(C1(CC2CC2)CCC1)=O 49122,Cc1cccnc1C=CC(=O)NCC(C)CN(C(=O)CN1CCC(F)CC1)C 49123,CS(=O)c1ccc(C(N2CCC(C)(C)C2CNC(=O)C=C(Cl)Cl)=O)cc1 49124,C1(O)(CCNC(C=C(C)C)=O)CCCN(C(=O)C=Cc2cnc(C(C)(C)C)s2)C1 49125,C(=O)(C1COc2ccc(Cl)cc21)NC1C=CCN(C(COC2(C)CCC2)=O)C1 49126,CC(C)(CC(=O)N1CCCC1C1CCN(C(c2snnc2C2CC2)=O)C1)C(F)F 49127,c1(OC)ccc(C2(C(=O)NC3CN(C(C4CC(OC)C4)=O)C3)CCC2)cc1 49128,C(C1CN(C(=O)CNC(C)=O)Cc2ccccc21)NC(C1C(OCC)C1)=O 49129,c1(CCC(=O)NC(C2CCCN2C(c2cnc[nH]c2=N)=O)(C)C)ccc(Cl)nc1 49130,C1(C(N2CC3(CN(C(=O)CCC4CC4(F)F)C3)C2)=O)CC(c2ccncc2)=NO1 49131,NS(=O)(=O)CCCC(=O)NCC1CCCCN(C(C2CCCCO2)=O)C1 49132,N1(C(C(CC)F)=O)CCOC(CN(C)C(c2csc(-c3ccsc3)n2)=O)C1 49133,C(=O)(CCCC(=O)NCCNC(=O)NC)N1CCN(C(CN(CCC)C)=O)CC1 49134,C(=O)(C(C)(C)C(=O)N1CC2(NC(c3nnc(O)cc3O)=O)CCC1C2)OC 49135,C(F)(F)(C(=O)NOC)c1scc(Cc2ccccc2Cl)n1.C1(COC)(OC)CCCOC1 49136,CN1CC=C(CC(=O)NC2CC(C3CCN(C(=O)CC4(O)CCCC4)C3)C2)CC1 49137,C(N=c1[nH]cnc2c(Br)nn(C)c12)C1CC(NC(C(C)Cc2cnc[nH]2)=O)C1 49138,C1(NC(c2cncs2)=O)CCCOC12CCN(C(c1cc(Cl)nnc1Cl)=O)CC2 49139,n1(CC(=O)NC2CCC(CNC(CC3CC(CC)C3)=O)CC2)ccc(O)nc1=O 49140,N1(C(=O)COCC(F)(F)F)CCN(C(C2(c3cccs3)CC2)=O)CC1CC1CC1 49141,C1(CNC(C(CC)CO)=O)CN(C(=O)CCc2cnc[nH]2)CC(C)(C)C1 49142,c1(NC(=O)C(=O)NC2CCN(c3nncs3)C2)ccc2c(c1)C(=O)NCCO2 49143,Cc1c(C(=O)N(C)CCN(C(=O)CC2OCCCC2(C)C)C)cccc1CO 49144,C1(NC(C(C)=CC2CC2)=O)CC(C2CCN(C(c3cc(N)ccc3C)=O)C2)C1 49145,O=S1(=O)CCN(S(=O)(=O)c2cnccc2OCC(F)(F)F)CC12CCCC2 49146,c1(C(N(C2CCN(C(C(CC#C)O)=O)C2)C)=O)cc(S(=O)(=O)NC)c[nH]1 49147,CC(C)C(C(=O)NCc1cnn(C(C)C)c1)c1ccnc(N(C)C)c1 49148,Cc1nccnc1N1CCN(c2nnc(C3CCOC3)n2CC2CC2)CC1 49149,C1(C(CC)CC)C(=O)OCCN1CC(CCCC)CC.C(CCF)CC 49150,C1(NC(CCc2ccc(C(C)(C)C)cc2)=O)CC(O)CN(C(=O)C2=CCCC2)C1 49151,CC(C)(C)C(CCc1ccc(F)cc1)C(=O)N1CCNC2(CC2)C1 49152,C(=O)(C(C#N)CCC)N1C(C(=O)NC2(CC#C)CCCCC2)CC(F)C1 49153,C1(NC(C2(C)CC2(Cl)Cl)=O)CCCN(Cc2cn(Cc3csc(Br)n3)nn2)C1 49154,N1(C(C(C=C)(C)CC)=O)CCC(NC(=O)C2=CS(=O)(=O)CCC2)C(F)(F)CC1 49155,c1(-c2cn(CCN(C(=O)C(c3cccnc3F)(C)C)C)nn2)cnccc1Cl 49156,c1(C(=O)NCCCC(C)NC(C2N(C(C)=O)CSC2)=O)cc2ncccc2o1 49157,c1(C(=O)NC2CN(C(c3cc(CC)c(CC)o3)=O)C(C)C2)c(N)ccc(F)c1F 49158,N1(C(C=CCC)=O)CC2CC(NC(c3cn(C)nc3-c3cccnc3)=O)C1C2 49159,C(C)(c1cccnc1)=CC(=O)NC(CCOC)CNC(C1(C)CC=CCO1)=O 49160,C(c1ccccc1Cl)=C(C(N1CC(CNC(CN(C2CC2)CC)=O)OCC1)=O)C 49161,CCN=c1cc(C(N2CCCC(NC(=O)C3=C(C)CC3)C2)=O)cc[nH]1 49162,C1(C(=O)NC(c2ncnn2C)C)CCN(C(=O)CN2CCSCC2)C(C)(C)C1 49163,Cn1ncc(Cl)c1CC(=O)NCC(CNC(=O)CCCC1CCCO1)CO 49164,C1(CN(C(C)C)CC2CCCN2C(c2ccn(C)c2)=O)CCCC(C)O1 49165,N1(C(CCCCC(N=[N+]=[N-])=O)=O)CCC2(CCC2)C(CNC(C2C=CCC2)=O)C1 49166,N1(C(C(C(C)(C)C)(C)C)=O)CCC(NC(c2ccc(N)cc2O)=O)C(F)(F)CC1 49167,c1(C(=O)NCCC(C)(C)NC(c2cc(OC)no2)=O)ncccc1SC 49168,N1(C(CCSC)=O)CCN(C(=O)COC2CCOC2)CC1c1nccn1C 49169,C1(C(=O)NC(C(=O)N(C(C2CCCC2)C)C)C2CC2)CN(C)CCN1C 49170,c1(CCC(N2CCC(c3cn(C(C=C)C)nn3)C2)=O)cc(OC)c(Cl)cc1OC 49171,N1(C(C2(C)C=CCC2)=O)CC2=C(C1)CN(C(c1ccc(OCC(F)(F)F)o1)=O)C2 49172,N1(C(CCc2ncn(C)c2)=O)CC(F)CC1CC(=O)NC1(n2cccn2)CC1 49173,c1(C(N2CCC(N(C(=O)CSc3nncs3)C)C2)=O)ncc(C(F)F)cc1F 49174,c1(C(=O)NCC(CCCC)NC(=O)CC(=O)N(C)C)cc(F)c(F)cc1Cl 49175,c1(C(N2CCN(C)C(CNC(=O)C3=CCOC3)C2)=O)cc2ccccc2s1 49176,c1(OC)ccc(CN(C(CCO)C(F)F)C)c2ccccc12 49177,c1(C(=O)NCC(CN(C(C(C)(C)OC)=O)C)C)cccc2nn(C)nc12 49178,N1(C(C2(C(=O)OC)CC2)=O)CCC2(CC1)CCN2C(c1c(C)ccnc1Cl)=O 49179,n1(CC(=O)NCC(CNC(CC(C)c2ccco2)=O)O)cnc([N+](=O)[O-])c1 49180,c1(CC)ccc(NC(C2(CNC(=O)C(C)CC3CCCC3)CCOC2)=O)cc1 49181,c1(C)ccc(N(CCCNC(=O)C(C(C)(C)C)c2cc[nH]n2)C)cc1Cl.CC=O 49182,Cc1nc2cccc(C(=O)NCC34CCCC3CCN4C(c3cnsn3)=O)c2[nH]1 49183,N1(C(C2CC(CC)C2)=O)CCCC(O)(CN(C(=O)CCC(C)C)C)C1 49184,C1(NC(CC2CC(CC)OCC2)=O)CN(C(=O)C(C)(C)CSC)CC2(CCC2)C1 49185,c1(OCCC)cc(F)ccc1Cn1cc(CCCc2ccccc2)nn1 49186,[N-]=[N+]=NC1COCC1NC(C1CN(C(=O)CN2CC3CC3C2)CC12CC2)=O 49187,N1(Cc2[nH]c3ccc(C)cc3c2)C(=O)C2C(C)CCCN2C1=O 49188,C1(C(=O)NCc2cnc(C)s2)CN(C(=O)CC2CCOC2)CC1(F)F 49189,c1(C(N2C3C(NC(C4CCN(CCC)CC4)=O)C(C3)C2)=O)c(C)ncnc1O 49190,c1(C(=O)NCC2CCCN(C(c3c(OC)csc3)=O)C2)ccc([N+](=O)[O-])c(F)c1 49191,c1(NC(C2CCN2C(=O)C(c2ccccc2)=O)=O)c(Cl)ccnc1Cl 49192,N1(C(=O)Cc2c(F)cccc2Cl)CC2CCC(C1)N(C(c1ccns1)=O)C2 49193,C1(NC(c2cccc(C)n2)=O)CC2CCC1CN2C(c1ccnn1C1CC1)=O 49194,Cc1cc(Cl)c(C(=O)NCc2ccc(CNC(=O)CC3CC3(C)C)cc2)s1 49195,CCCC(C#N)C(=O)NC(c1cnn(C)c1)C(=O)NCC(C)CCC 49196,N1(C(C(OC)OC)=O)CC2(CCCCN2C(C2CCCC23CC3)=O)C1 49197,C1(F)(CNC(c2cc(C)c(O)nc2)=O)COCCN(C(=O)CS(C)(=O)=O)C1 49198,c1(C(N2C(CNC(=O)C3=CCCC3)CC(C(F)(F)F)C2)=O)ccc2ccnn2c1 49199,CC1CCC(C)(C(=O)NC2CC3(C2)CN(C(c2ncncc2F)=O)C3)C1(C)C 49200,Cc1cc(F)cnc1C(=O)NC1(CO)CCN(C(c2sccc2OC(F)F)=O)C1 49201,C(=O)(C(C(C)(C)O)NC(C1CCCN(C)C1)=O)NCCC1C(C)C1 49202,C(=O)(CCCC(F)(F)F)N1C(CCC)CN(C(=O)COC2CCCC2)CC1 49203,CCCC(CC(=O)N(C)CC1(N(C)C)CCC1)NC(c1cc(Cl)c[nH]1)=O 49204,N1(C(CCCCC(=O)OC)=O)CCC2(CCC(NC(=O)CCCSC)CC2)C1 49205,c1(C(N(CCC(=O)N(CCOC)C)C2CCC2)=O)ccnc(C)n1 49206,N1(C(C(C)(C)CF)=O)CC2(CCN(C(=O)CCCC3CCCC3)C2)C1 49207,N1(C(CCCCOC)=O)CCOC(C)(CNC(=O)C(F)(F)C(O)C2CC2)C1 49208,C1(NC(=O)Cc2cccs2)CN(C(c2coc(C(F)F)n2)=O)C2(CCCCC2)C1 49209,c1(C(C)NC(=O)NCc2sc(C(=O)OC)c(C)n2)ccc(C#N)cc1F 49210,c1(C(=O)NCC(Cn2cc(-c3cccc(OC)n3)nn2)(C)C)cc(N)c(F)cn1 49211,C12(C(=O)NC(C)C(C)(C)C#N)CCC(CN(C(=O)CC(C)C(F)(F)F)C1)C2 49212,C1(C(=O)Nc2ccc(COC)nc2)CCN(C(=O)C(C)C2CCOCC2)O1 49213,N1(C(c2c(NC)n(C)nc2)=O)C(CC(=O)N(C)CC2(N(C)C)CC2)C2CCCC12 49214,N1(C(C=CC(C)NC(=O)C(F)CC2CCOC2)=O)CCCCCC1 49215,CCC(C)(C)CCNC(=O)CC(CNC(C1CCCS1)=O)C1CCC1 49216,C(=O)(C1CCc2nccn21)N1CCN(N2C(C)CCCC2)CC1C1CCCC1.C=O 49217,c1(OCN2C(COC)CN(C(=O)OC(C)(C)C)CC2)c(Cl)ccc(F)c1Cl 49218,CC1CC(C)OC1C(=O)NC(C)CCNC(c1ccsc1-n1cnnn1)=O 49219,C(CC(C(=O)NCCC1CC(C)(C)C1)NC(=O)OC(C)(C)C)=CC.C1(=O)CN1.SCC 49220,c1(C2(C(C)NC(C3CCN(C(COCCC=C)=O)C3)=O)CC2)cccc(F)c1C 49221,C1(CC(=O)NCC2N(C(c3c(C)nn(C)c3Cl)=O)CCC2)CCC2(CCC2)CO1 49222,C(C(C)(C)CC(=O)NC(C1CCCC1)CO)NC(C1(CC)CCCC1O)=O 49223,c1(CN(C2CCNCCC2C)C(c2c(C)cccn2)=O)ccc(F)c(Cl)c1 49224,C(=O)(C1CCCc2nn(C)cc21)N(c1cn(CC(C)C)nc1)C1CCCC1 49225,C(CC(C)(C)C(=O)N1C2CCC(C2)C1CNC(=O)Cn1[nH]cnc1=N)SC 49226,c1(C(=O)NCC2N(C(CC(CCSC)O)=O)CC2)[nH]nc2ncnc(O)c12 49227,C1(c2nc(CCCCC)nn2-c2ccc(OC)c(Cl)c2)CCC2CC1C2(C)C 49228,CN1C(=O)c2ccccc2C1CNC(N1CCC(C2CC(=O)NC(=O)C2)CC1)=O 49229,C1(S(=O)(=O)N2CCOC(CNC(=O)CC(C)C)C2)(CC)CC1 49230,N1(C(C2CC=C(C)CC2)=O)CC2(C(N3Cc4c[nH]nc4C3)=O)CCC1CC2 49231,C(=O)(CCCCCN(C)C)N1CC=C(C)CC1.C12(CCCCC1)C(=O)N2 49232,c1(C(N2CCN(CC(C)(C)NC(=O)Cn3ccnn3)CC2)=O)nnc(O)cc1O 49233,C(C(=O)N1CC(CO)(NC(=O)CCCCN2CCOCC2)C1)(C(C)C)SC 49234,C1(NC(C2C(CC)C2)=O)CCC(NC(=O)CCOc2ccc(Cl)cc2)CC1 49235,N1(C(C2C(=C)CC2)=O)CCCC(C2CN(C(c3nc[nH]c3C(C)(C)C)=O)C2)C1 49236,C1(NC(C2N(C(=O)OC)CCC2)=O)CCCCC1NC(C1(C)CCSCC1)=O 49237,c1(CCC)ccc(C(N2CCC(CF)(NC(=O)NC3CC3)C2)=O)cc1.C(C)(C)(C)O 49238,C(=O)(C1=CC(O)CCC1)NC1CCN(C(C2CC(C)(C(=O)OC)C2)=O)CC1 49239,Cc1csc2c(NCC3CCN(C(c4cc(Cl)cc(Cl)c4O)=O)C3)ncnc12 49240,c1(OC)cccc(C(=O)NCC2(O)CCN(C(c3ncccc3N)=O)C2)c1 49241,C1(NC(c2cn(CC)nc2C2CC2)=O)CCN(C(=O)Cc2cccs2)CC1C 49242,N1(CC(=O)NC2CCN(C(C34CCOCC3C4)=O)CC2O)Cc2ccccc2C1 49243,c1(CN2C3C(C(N4CCC(C(N)=O)CC4)=O)C(C3)C2)c(F)cc(Br)cc1F 49244,c1(C(CNC(=O)CC2CCCCC2)O)cccc(-c2cccnc2)c1 49245,N1(C(CC2CC(C)C2)=O)CCC2CN(C(=O)CSc3ccc(F)cc3)CCC12 49246,N1(C(c2c(C)ccn2C)=O)CC(CCNC(c2oc(CO)cc2C)=O)OC(C)C1 49247,c1(C(=O)NC2CCCC(N(C(Cc3cnc(C)o3)=O)C)C2)cc2c[nH]cnc-2n1 49248,Cc1c(C(N2CCC(C(=O)NCC3CC3c3ccco3)(C(C)C)C2)=O)nnn1C 49249,Cc1cc(C(=O)NC(C)CCNC(=O)C2=CCCC2)cc(Cl)c1 49250,c1(CN)ccc(CNC2CC2NC(=O)Nc2cccc(F)c2)cc1 49251,C(=O)(C(C)(C)C1=CCSCC1)NC1C(NC(CC(COC)(C)O)=O)CCC1 49252,C(=O)(C(C)(C)S(=O)(=O)C1CC1)N1CC2C(NC(C(C)CC(F)F)=O)CC(CC2)C1 49253,c1(C(=O)NCc2cccc(F)c2)ccc(F)c(S(=O)(=O)N2CCC2)c1 49254,N1(C(C=C(CC)CC)=O)CC2CC(NC(c3ccnnc3S)=O)CC2C1 49255,C1(C(=O)NC2(CC=C)CN(C(C3(CF)CC3)=O)C2)CCCCC1C1CC1 49256,Cc1nn(C)c(=O)c(C(=O)NCCCCN(C(=O)Cc2cscn2)C)c1C 49257,CC1CC(CNC(=O)COC2CCC2)CCN1C(c1ncoc1-c1ccco1)=O 49258,C(=O)(C(F)CCC(C)C)NC(CC)CC(=O)NCCCC(C)O 49259,C1(CC)CN(C(=O)C(O)C(C)(C)C)CCC1NC(c1cc(N)ccc1C)=O 49260,N1(C(C(C)=C(CC)C)=O)CCC2(CCN(C(=O)C(C)(C)C(F)F)C2)C1 49261,C1(NC(c2c(C)scn2)=O)CCCC(N(C)C(C2CCC(C)CC2)=O)C1 49262,C1(C(=O)NC2CC3C=CC2C3)CCCN(C(=O)CN2CC(=O)NC2=O)CC1 49263,c1(CNC(c2cnc(C)n2C)=O)ccc(CNC(c2c(C)ncn2O)=O)c(F)c1 49264,c1(C(=O)NC2(C)CCN(C(C3CC(C4CC4)=NO3)=O)C2)csc(=NC2CC2)[nH]1 49265,Cc1cnc2cccc(C(=O)NC(C)C(C)NC(=O)COC(C)C)n12 49266,CC(C)(C)CCC(N)CNCc1cnccc1Cl 49267,C(=O)(CCCS(C)(=O)=O)NCC1(F)CC(NC(C(c2c(C)cccc2)C)=O)C1 49268,c1nc(N2CCOCC2)[nH]c(=NC(CCc2cccnc2)C2CCC2)n1 49269,N1(C(CCCO)C(F)(F)F)CCc2cc(Nc3ncccn3)ccc21 49270,CC1=C(C(=O)N2CCC(NC(=O)CC3CCCC3)C(CO)CC2)CCS1(=O)=O 49271,C1(C#N)(C(=O)OCc2cc(C)c(Cl)cc2)CCCCCCC1 49272,c1(C(=O)NCCOC2CCN(C(CCSC)=O)C2)nn(C)cc1Br 49273,Cc1cn(C)cc1C(=O)NCC(C(=O)N(CCC(=O)NC1CC1)C)N(C)C 49274,N1(C(Cn2c(C)nc(C)n2)=O)CCC2CCN(C(C3CCNC3=O)=O)CC2C1 49275,C1(NC(C2CCN(C3COC3)CC2)=O)CCN(C(c2ccncc2Cl)=O)C12CC2 49276,C(=O)(C1=NN(C(C)C)C(=O)CC1)N1C2(C#C)CC(C1)C2 49277,CC(CC(F)(F)F)C(=O)NC(C)CN(C)C(c1c(O)cc(O)cc1O)=O 49278,N1(C(C2CN(C(C)=O)C2)=O)CC2(NC(c3cncs3)=O)CC1C2 49279,c1(OC)ccc(CC(=O)NCC2C(C)CCCN2C(c2cocc2C)=O)cc1Cl 49280,CCC(C(=O)NCC1(C(N2CC(C3CC3)(COC)C2)=O)CCCO1)C(C)C 49281,C(C(=O)NOCCN(C)C)(N(C(C(C)n1cncn1)=O)C)C1CC1 49282,c1(CN(C(=O)NC(c2ccc(C(C)C)cc2)C)CC)onc(C)c1CO 49283,C(=O)(CC(C)(C)C(F)F)NC1C(NC(C(C)S(N)(=O)=O)=O)CCC1 49284,CN1CCN(C(c2cc3ccsc3s2)=O)C(CNC(c2ccc(O)c(O)c2)=O)C1 49285,Cc1nc(Cl)[nH]c(=NCC2CCCC(NC(=O)Cn3ccc(O)nc3=O)C2)c1Cl 49286,N1(CC(=O)N(C)CC2(NC(C3CCC(CC)O3)=O)CC2)CCC(=O)NC1=O 49287,C#CCCCCCCC(=O)NC1CC(F)CN(C(=O)C(c2ccc(C)o2)C)C1 49288,N1(C(C(C)NC(COC)=O)=O)CC2CCC(C1)C2NC(=O)CC1CC=CCC1 49289,c1(C(=O)NCC2(C)CCN(C(CCNC(COC)=O)=O)C2)c(C)nn(C)c1OC 49290,c1(-c2cc(C(=O)Nc3cc(C(=O)OCC)cc(Cl)c3)n[nH]2)c(F)cc(O)cc1F 49291,Cc1cc(C)c(C(=O)NCCCCN(C(=O)COCCOCCO)C)s1 49292,c1(NC(C(C)(N(C)C(c2ccnnc2)=O)C2CC2)=O)ccc(O)c(=O)cc1 49293,c1(C(=O)NC2CN(C(C(C=CC)O)=O)CC2O)cnc2c(c1)COCC2 49294,C(CC(=O)N1CCC(C(=O)OC)C1C)(C(F)F)NC(c1cnc(CC)s1)=O 49295,C1(O)(CNC(c2cc(CNC(=O)Cc3ccc[nH]3)on2)=O)CCCCC1 49296,c1(CC)cc(C(=O)N(CC(C)(C)C(=O)NC(CO)C(=O)OC)C)nn1C 49297,C(C)(CCC(=O)NCC1(F)CCC(NC(=O)CSc2cccc(F)c2)C1)OCC 49298,C(=O)(CC(C)P(C)(C)=O)N(CC(C)(C)NC(C=C(C)c1ccsc1)=O)C 49299,C1(CO)CN(CCCOC)CCN1CC1CC1 49300,C(=O)(C(C)C(F)(F)F)NCCN(C(=O)C(C)COC)CCC 49301,c1(C(CC=CCONC(C2CCC(C(C)(C)C)CC2)=O)=O)ccc2nn[nH]c2c1O 49302,C1(CCC)CN(C(=O)Cc2cncnc2O)CCN1C(c1cnc(O)c(Cl)c1)=O 49303,C(=O)(CC(=O)N(CCNC(=O)C(C)(C)C1CC1)CCOC)OCC 49304,C1(C(=O)NC23C(CN(C(c4cc(C)[nH]n4)=O)C2)C3)CCc2ccc(F)cc2C1 49305,c1(C(=O)NC(CC)CNC(c2csnn2)=O)cc(N)c(N)cc1F 49306,N1(C(CCN(CCCCC)C)=O)CCN(C(C2CC2OC)=O)CC1C1CCC1 49307,c1(OC)ccc(CC(N2CCC(CNC(C34CCC(CO3)C4)=O)C2)=O)nc1 49308,c1(C(C)C)cc(=NCC(C)(C)NC(c2ccc(Cl)nc2)=O)[nH]cn1 49309,C1(CCOC)CN(C(=O)CC2CCCC2)CCN1C(C1CCCC(=O)N1C)=O 49310,C12(NC(c3ncn(CC)c3)=O)CCCC(NC(c3ccsc3C)=O)(C1)C2 49311,c1(C(=O)NCC2(NC(COCC)=O)CC3CCC2C3)ccc2snnc2c1 49312,C12(C(N(C)Cc3ncco3)=O)CCC(CC1)N(C(=O)C=CC1CCOC1)C2 49313,C(=O)(CCC(=O)N1CC(N2CC(C(C)OC)CC2=O)C1)NCC.n12cc(nn1)C2 49314,S(=O)(=O)(CC(=O)NC1CCN(CC(=O)NCC2CCCC2)CC1)NC(C)(C)C 49315,C1(C(=O)OC)CC(n2cc(C3CC=CCC3)nn2)CN1C(C1CCCCC1O)=O 49316,c1(OC)cccc(C=CC(=O)NC(C)CC(C)NC(c2ccc(C)nc2C)=O)c1 49317,c1(C(=O)NC2CC(CC(=O)NC(C=C)(C)C)C2)cn(C)nc1SC 49318,c1(C(=O)NCCCCNC(C2C(C(N(CC#C)C)=O)C2)=O)cccc(CO)c1 49319,c1(CC)nc(C(=O)NCC2COCC2NC(=O)Cn2cc(Cl)cn2)co1 49320,C1(NC(c2ccc(F)o2)=O)CCC12CCN(C(c1ccc(F)c(F)c1F)=O)CC2 49321,c1(NC(C2(NC(CC3CCC(C#N)C3)=O)CC2)=O)cccc([N+](=O)[O-])c1 49322,c1(C(=O)NCC2(OC)CN(C(=O)C(C)(CO)OC)C2)nc2ccccc2cc1Cl 49323,C12(C3(O)CN(C3)C1=O)CC2.C1(O)(CC(=O)N(C)CC2(C(=O)OC)CC2)CCC1 49324,C1(C(N)=O)CCCN1C(=O)CC1(CNC(c2ccn(C3CC3)n2)=O)CC1 49325,c1(C(N(CC=C)C(C2(c3sccc3C)CC2)=O)=O)nnn(CC2C(SC)CC2)c1C 49326,C1(N(C(=O)COCC2CCOC2)CC#C)CCN(C(C2CC23CCC3)=O)CC1 49327,C1(C(=O)NCCn2ncc(CC)c2)C=CCCN1C(c1cn(CC)nn1)=O 49328,N12CC3C(CC1c1nc(no1)NC2=O)C3.n1(CCC)ccc(CC)c1 49329,c1(C(=O)NCC2(C)CN(C(C(C)O)=O)C2)cc(C(C)(C)C)ccn1 49330,C(N=c1[nH]ccn2cnnc12)c1cc(OC)c(Br)cc1 49331,C1(N(C(c2nc(C(C)OC)oc2)=O)C)CCN(C(=O)COC2CCOC2)CC1 49332,C=Cc1cnn(C)c1C(N1CC2CC1CC2NC(=O)C(=O)C(C)(C)C)=O 49333,CC1CC(C2CC2)CN1Cc1ccc(C(=O)NN(C)C)[nH]1.c12ccc(o1)CNC2=O 49334,Cc1ccc2c(c1C)OCCC2NCc1cc(F)ccc1C#N 49335,C1(C(=O)NCCC2C(C)C2)CN(C(=O)CC2CCOC2=O)CC12CC2 49336,n1(CC)cc(-c2ccccc2)nc1N(C)Cc1cc(C)nn1Cc1ccccc1 49337,c1(CNC(C2(SC)CC2)=O)ccc(C(N2CCC(C(C)O)C2)=O)cn1 49338,C1(C(=O)OCCOC)CC(F)(F)CCN1C(=O)OC(C)(C)C 49339,C#CCC(C(=O)N(CC(C)N(C(=O)Cc1csc(Cl)n1)C)C)C1CC1 49340,N1(C(c2cc(C)oc2)=O)CCC2(NC(c3cc(CC(C)C)c[nH]3)=O)CCCC12 49341,c1(C(C)(C)C)nocc1C(=O)NCC(C)(O)CNC(c1cnc(C2CCC2)s1)=O 49342,c1(CCC(=O)N(C2CCN(C(C3C(=C)C3)=O)CC2)CC)cnc2n1CCCCC2 49343,C1(C(N(C)Cc2ccoc2)=O)CC(NC(c2nc[nH]n2)=O)CCO1 49344,N1(C(C2(F)C(C)C2)=O)CCC2(CCC2CNC(c2ccco2)=O)CC1 49345,CC(C)CC(=O)NCC1CCN(C(C2CNC(=O)N2)=O)C1 49346,CC(C)CCCOCC(=O)N(CCCN(C)C)CCNC(C1CC1CC(C)C)=O 49347,C1(OC)CCC12CC(C(N1CCN(C(=O)CN3CCS(=O)CC3)C(CO)C1)=O)C2 49348,c1(C(=O)NCC2CC3(CC(NC(CCSCCC)=O)C3)C2)cnc2n1CCCC2 49349,CC(C)(C(=O)N1CC(n2cc(CNC(=O)C(C)(O)CC3CC3)nn2)C1)C1CCC1 49350,c1(CC(=O)NCC2CCN(C(C3CNC(=O)N3)=O)C23CC3)ccc(Cl)c(Cl)c1 49351,Cn1nc(CC(=O)NC(C)(CNC(C2CC23CCC3)=O)CO)cc1C(F)(F)F 49352,c1(OC(C)CNC(=O)NCc2nc(-c3ccccn3)no2)ccccc1Br 49353,N1(C(C2C(C#N)C2)=O)CC2CCC2(CNC(C2CC2c2ccc(Cl)cc2)=O)C1 49354,c1(C(C(=O)NCCN(C(C)C)C(c2ccco2)=O)C)c(Cl)cccc1Cl 49355,C1(C)(C(=O)NCc2cn(CC(C)NC(c3ccc(CO)s3)=O)nn2)CCOC1C 49356,c1(CC(=O)NCCCCCNC(=O)CC2(O)CC2)ccc2n[nH]cc2c1 49357,c1(C(c2nnnn2CC2CC2)NC(C(C)(C)OC)C)cnc(Cl)n1C.C1CC1 49358,n1(C(C)C)nncc1C(=O)N(CC(C)NC(=O)CN1CCCC1)C 49359,N1(C(C=C(C)C)=O)CC(C)(C)OCC1CNC(c1cccc(O)c1)=O 49360,C1(CNC(C#CC2(CC)CC2)=O)CCC(C)(C)CN1C(c1csc2nnsc12)=O 49361,C=CCC(C(=O)NC1CCSC12CN(C(c1ccc(Cl)o1)=O)C2)C(C)C 49362,N1(C(C2CN(OC)C(=O)C2)=O)CCc2sccc2C1CNC(c1ccon1)=O 49363,C1(c2c(CC)cccc2)CCCN(C23CC(C)(C2)C3)CC1 49364,C1(NC(c2c(C)con2)=O)CCN(C(c2ccc(C3CC3)cn2)=O)CC12CCC2 49365,C(=O)(C(C)(C)CCCF)N(CCCCCNC(C(C(C)C)OCC)=O)C 49366,CC12CCC(C(=O)NCC(O)CNC(=O)C(C)(C)n3cc(Br)cn3)(CC1)CO2 49367,C1(NC(Cc2[nH]c(=N)sc2)=O)C2CN(C(C3(C4CCCO4)CCC3)=O)CC12 49368,N1(C(c2ccn(CCOC)n2)=O)CCC2CN(C(C3CC4(CC4)CO3)=O)C2C1 49369,C1(C(N2C(C(C)C)CNC(=O)C2)=O)CCN(C(=O)C(C)c2ccco2)CC1(C)C 49370,c1(C(=O)NC2CC(CNC(c3ccc(-n4cccn4)nc3)=O)C2)c(Cl)csc1Cl 49371,c1(CC)ccccc1C(N1CCOC(CCCNC(C2CCCN2C=O)=O)C1)=O 49372,N1(C(CCC(C)=O)=O)CCCC1C1CCCN1C(=O)CCC1CCC(C)(C)CC1 49373,C1(CC(=O)NC(CCNC(C(C)O)=O)C)CC(F)(F)C1 49374,C1(CNC(CC(C)(C)C)=O)CC2(CCN(C(c3ccc(N)c(Cl)c3)=O)C2)CO1 49375,N1(C(CC(=O)OC(C)(C)C)=O)CCC(NC(C2CC2(F)F)=O)C12CCCC2 49376,CCCC(C)CC(=O)NC1(C(=O)NC2CCCNC2=O)CCOCC1 49377,C(=O)(C(O)C(C)(C)C)NCC1(OCC)CN(C(=O)C2=CCCCC2)C1 49378,c1(C(=O)NCC2CN(C(C3N(S(CCC)(=O)=O)CCC3)=O)C2)nccc(C)n1 49379,C(=O)(C1=CS(=O)CCC1)NCCCN(C(C)C)C(C1CCCN1N=O)=O 49380,N1(C(C)=O)CCc2cc(NC(c3ccccc3C(N)=O)=O)ccc21 49381,c1(C(N2C3CCC(CNC(C(C)(C)SC)=O)(C3)C2)=O)ccc2c(c1)COC2 49382,c1(NC(=O)CC2CCN(C(=O)Cc3ccc(F)cc3Br)C2)ccc2c(n1)CCC2 49383,N1(C(C(c2cnn(C)c2)C)=O)CCC12CN(C(c1cc(O)cc(Cl)c1)=O)C2 49384,c1(OC)ccccc1S(=O)(=O)NC(=O)C(c1sc(Br)cc1C)N1C(C)CC1(C)C 49385,CP(C)(=O)c1ccc(C(=O)NCC2(F)COCCN(C(=O)CC3CCC3)C2)cc1 49386,C1(NC(CNC(C=NOC)=O)=O)CCC=CCC1 49387,CCCS(=O)(=O)CC(=O)NC(C)CC(C)NC(=O)COc1ccc(Cl)cn1 49388,N1(C(CNC(=O)NC)=O)CCCN(C(c2cc(C(=O)C(C)C)c[nH]2)=O)CC1 49389,C=C(C)c1ccccc1NC(c1cc(CNC(C2C3CC(=O)CC23)=O)no1)=O 49390,N1(C(c2c(CC)cns2)=O)CCOCC(C(N2CC=CC2C(=O)NC)=O)C1 49391,CN1CCCC(CCC(=O)NCC2CCN(C(C3CCC3)=O)CC2)C1 49392,c1(OCC2N(CC(=O)N(CC)CC3CC3)CCC2)cccc(C)c1.C1(=O)CN1 49393,C#Cc1ccc(C(=O)NCC2COC(CNC(c3ccc(C#N)o3)=O)C2)cc1C 49394,C(C(C)CC(=O)N(C1CC1)C1CC1)NC(CC=CCC)=O 49395,c1(C(=O)NC(CN(C)C)C(=O)NC2CCC(C)(C)C2)ccc([N+](=O)[O-])o1 49396,N1(C(c2cc(CC)nn2C)=O)CC(C(=O)NC(CO)C(N)=O)C(C2CC2)C1 49397,C1(C)(NC(N(C2CCC2)CC2CCN(CC(C)C)C2)=O)C(C)(C)C1(C)C 49398,Cc1cc(C(N2CC3C(NC(=O)CC4CCC(C)(C)C4)C3C2)=O)n(C)n1 49399,CCC(C(F)(F)F)NC(C1CCCCN1C(=O)COCC(F)(F)F)=O 49400,CC(C)C(C(=O)N1CCC(NC(C2CC3(CC3)C2)=O)C1)n1cncn1 49401,c1(-n2c(-c3ccc(C(CC)C)cc3)nc(C(C)C3CC3)n2)ccc(F)c(Cl)c1F 49402,c1(C(N2CC3C(CNCc4ccc(C(=O)O)cc4)(C3)C2)=O)ccc2scnc2c1 49403,c1(OC)ccc(C(=O)N(C)CC2CCCN2C(c2coc(O)n2)=O)c(O)c1F 49404,CCC(C)(C)C(C)CC(=O)NCCC(C)NC(c1ccc(OCCOC)nc1)=O 49405,C1(CNC(COC(C)=O)=O)C2CN(C(c3cnn(-c4cccc(Cl)c4)c3)=O)CC12 49406,C1(C(=O)NCc2nc(-c3ccc(C)cc3)oc2)CN(C)CC(C)O1 49407,N#Cc1ccc(C(N2CC(CO)(NC(=O)C=Cc3cscn3)C2)=O)s1 49408,C1(NC(C23CC(C#N)(C2)C3)=O)CC(C(=O)NC2CNC(=O)C2(C)C)=CC1O 49409,c1(C(=O)NC(C)CCCNC(=O)C(C)C)ccccc1C1CC1.C1(=O)CC(=O)N1 49410,C1(NC(=O)CCCC2CCOCC2)CCCC(NC(=O)COc2ccccc2)C1 49411,c1(C(=O)NC2(n3cccn3)CC2)cc(O)nc2c1CN(C(C1(F)CC1)=O)CC2 49412,C1(NC(C=NOC)=O)CCC(O)CN(C(=O)CC(C(F)F)n2cccn2)C1 49413,C(=O)(CC(C)CCC)N1CCC(C(C(=O)NC2CCN(C(CC)=O)C2)(C)C)C1 49414,CCC(CC(=O)NC(CC1CCC1)CO)N(C(C1CC12CC2)=O)C1CC1 49415,C1(CC=C)(NC(=O)CC2CC3C=CC2CC3)CCCN(C(=O)Cc2nc[nH]n2)C1 49416,CCCCC(C(=O)NO)NC(=O)NC1CCOCC1F 49417,C1(C(=O)Nc2c(F)cccc2Cl)CCC2CCCCN2C1 49418,c1(OC)cccc(C(=O)N(CCCNC(=O)CCc2ccc(F)cc2)C)c1OC 49419,c1(COC)nc(NCC2CC(=O)N(C)C2=O)cc(=NCc2cccs2)[nH]1 49420,c1(N(CCOC)C)ccnc(C(N2CCC2CNC(C2(SC)CCC2)=O)=O)c1 49421,S(=O)(=O)(c1ccc(F)c(C(=O)O)c1)CN1CC2CN(S(CC)(=O)=O)CC21 49422,c1(C(=O)NC(Cc2ncn(C)n2)C(=O)O)ccc(CO)cc1 49423,c1(C(N(C2CCN(C(=O)CSc3nncn3CC)C2)CC)=O)ccn(C2CC2)n1 49424,N1(C(c2cc(-c3cccs3)on2)=O)CC2(CCN(C(C3(C(F)(F)F)CC3)=O)C2)C1 49425,C1(C(=O)NCC2CC(NC(c3ccn(C)n3)=O)C(O)C2)Cc2c(F)cccc2O1 49426,C1(C(c2nnnn2C2COC2)NC(=O)CCCN(C)C(C)C)(OC)CCCC1 49427,N1(C(COCCC)=O)CC2(CC1CNC(=O)Cc1cc(C)[nH]n1)CC2(F)F 49428,c1(C(N(C2C3CCCC23)C)=O)cc(CNC(=O)CC2CC(=O)C2)[nH]n1 49429,C1(C2CCN(C(=O)C=CC3CCC3)CC2)(NC(c2cc(OC)no2)=O)CC1 49430,C(=O)(CCCCCC)N(CC(=O)NCC12COC(COC)(C1)C2)CC#C 49431,c1(C(=O)NC(CC)CNC(=O)C(C)c2cncs2)ccc(F)cc1OC 49432,C(=O)(CCC(=O)c1cc(Cl)sc1Cl)NCC(C)N(C)C(c1cnccn1)=O 49433,CC(C)CC(N=C1NS(=O)(=O)c2ccccc21)c1nc(-c2cccnc2Br)no1 49434,O=C(CC(C(F)F)NC(C1(F)CC1)=O)NCC1(F)CCOCC1 49435,CN1CCC2C(CCN2C(=O)CCC2(NC(=O)COc3ccccc3)CC2)C1 49436,C1(C(=O)NC2(C(=O)NCCOC3CCCC3)CCN(C)C2)CCCC1C1CC1 49437,C(=O)(N1CCC(C(=O)NCC(F)CO)O1)c1nc(=N)[nH]cc1 49438,C1(NC(c2c(C)cno2)=O)CN(C(C2CC2c2ccccc2F)=O)CCC1C 49439,C1(C2CCC2)(COC2C(C(=O)NC3CC(OC)CN3C(C3(CC)CC3)=O)C2)CCC1 49440,C(=O)(N=c1[nH][nH]c2cccnc12)C1CCC(NC(c2ccccc2O)=O)C1 49441,C(=O)(CCC(F)(F)F)NCC(CCNC(c1cc(C(C)C)on1)=O)O 49442,C(=O)(C1CCSc2ccccc21)NCC(CNC(=O)C(C)C)OC 49443,N#Cc1c(C(=O)NCC2(O)CCN(C(=O)C(=O)NCC(F)(F)F)C2)cccc1F 49444,c1(C(N2C(CC(=O)NCC(C)S(N)(=O)=O)CC(F)C2)=O)cn(C)ccc1=O 49445,N1(C(c2c(CC)[nH]cc2)=O)CCC(C)(CNC(C2CCC(CC)O2)=O)C1 49446,Cc1cc(F)c(C(=O)NCC2CCN(C(=O)CP(C)(C)=O)C2)c(Br)c1 49447,c1(OC)ccc(CCC(=O)N(C)CC2CCCN(C(C3(CF)CC3)=O)C2)cn1 49448,C(=O)(CCS(N)(=O)=O)NCC(C)(C)OCC(=O)N(C)Cc1nccn1C 49449,C(=O)(CCCCC(C)(C)C)NCC(C)(CC)NC(CCC(=C)Br)=O 49450,CCCCC(CNC(c1cc(Cl)cnc1O)=O)CCC 49451,C1(C(N2CC(C)C(CCNC(=O)CCCCCF)C2)=O)CCc2c[nH]nc2C1 49452,c1(CC)nnc(C)cc1C(=O)NC(C)(CNC(c1cc(C(F)F)[nH]n1)=O)CO 49453,Cc1cc(O)ncc1C(=O)NC1C2CC1N(C(=O)CN1CCC(=O)CC1)C2 49454,Cc1nc2sccn2c1C(=O)NC1CN(C(c2cc[nH]c2)=O)CC1C 49455,C1(C(=O)NC(C)C(=O)NO)CCC(C)(C)N(C(=O)CC2CCCCCC2)C1 49456,C(=O)(CCC(=O)Nc1nccs1)NCC(C)N(C)C(c1cccc(O)c1)=O 49457,N1(C(C(C)CO)=O)CCN(C(=O)CCC2OCCO2)C(CF)C1 49458,c1(C(=O)NC2(C)CC(C(=O)Nc3cnc(OC)nc3)C2)nccc(C)c1F 49459,c1(OCC(=O)NCC2N(C(CSCC(C)C)=O)CCC2C)cc(Cl)cc(Cl)c1 49460,Cn1cc(C(F)=CC(=O)NC2CC(NC(c3conc3C3CCCC3)=O)C2)cn1 49461,C(=O)(C(CC(C)C)C(C)C)NCC1OCCN(C(CC2(COC)CCC2)=O)C1 49462,c1(OC)ccc(OC)c(CN2CC3C(C2)N3C(C2CC3CCC2O3)=O)c1.C(C)(=O)O 49463,c1(C(=O)NCCC2N(C(Cn3ncc(C)c3)=O)CCC2)cncc2cnccc12 49464,C12(NC(=O)Nc3ccc(OCCO)nc3)CCC(O)(CC1)C2 49465,CCCCCC(F)C(=O)N1CCC(C(=O)NCC23CCC(CO2)C3)(CC)C1 49466,C1(CC)CC(NC(=O)CC(C)(C)NC(C2CC(CF)C2)=O)CCO1 49467,C1(CNC(c2c(OC)cncc2)=O)CN(C(=O)CC2CCCSC2)CC(C)(C)C1 49468,C#CC1CCCN(C(=NCCOCC2CC2)NCC(CC(C)(C)C)C(C)(C)C)C1 49469,C1(CCC)CN(C(c2cc(C)no2)=O)CC1C(N1CCOCC1CC(C)C)=O 49470,C=CC(C)(CC)C(=O)NC1CCCC1NC(c1c(C)coc1-c1ccccc1)=O 49471,N1(C(C(C(=O)OCC)F)=O)CCN(C)C(C(=O)NCC2=CCCC2)C1 49472,c1(OC)ccc(CC(=O)N(C)CC2CN(C(=O)Cc3ccsc3)CCO2)c(F)c1 49473,c1(C(C(=O)NCC2CCCO2)N(CCCC)CC)nc(C2CC2)cs1 49474,C(=O)(NNc1ccc(S(=O)(=O)C(F)F)cc1)c1c(OC)c(Br)c(F)c(F)c1 49475,N1(C(C2OC3CCC2C3)=O)CC2=C(C1)CN(C(C1(n3cnnn3)CC1)=O)C2 49476,C1(C)(C(=O)NC2(CC(=O)OC)CCC2)CCCN(C(c2cccnc2Br)=O)C1 49477,N1(C(c2ccc(NC(N)=O)cc2)=O)CCC2CCN(C(=O)CC3CC34CC4)CC12 49478,c1(C(N(C2CCCN(C(C3(CC#C)CCC3)=O)C2)CC)=O)nccc2ccccc12 49479,C(C)(CCCCNC(=O)C(C)c1cccs1)NC(C1N=C(C)SC1)=O 49480,C1(C(=O)NCCOC(C)(C)C)CC2(CCN(C(c3ccnc(Cl)c3)=O)CC2)CO1 49481,c1(C(=O)NC(CCOC)CNC(C2(C)CC=CC2)=O)ccc2cnn(C)c2c1 49482,CC1(C(N2CC(NC(C3CCOC3)=O)C(O)C2)=O)CC2CCC1C2 49483,CON(C(=O)c1cc2cn[nH]c2cn1)C1CCCC1 49484,c1(C(=O)OCC)cc(C(=O)NC23CC(NC(=O)CN(C)C4CC4)(C2)C3)ccc1Cl 49485,Cn1ccc2cccc(C(N3CC4CC4(CNc4ncc(C(F)F)cn4)C3)=O)c12 49486,N1(C(c2cnc(SC)s2)=O)CCN(C(C2CCCC2c2cnn(C)c2)=O)CC1 49487,C1(C(=O)NC(C2CCCC2)CNC(C2(CC=C)CC2)=O)CS(=O)(=O)CC(=O)N1 49488,n1(CC)nc(C(=O)NC2CC(C(N3CC(CO)CC3CO)=O)C2(C)C)cc1O 49489,C(=O)(C(C(C)CC)NC(=O)C(C(CC)CC)OC(=O)OC(C)(C)C)NCCOC 49490,C1(CNC(c2cc(CCC)ncc2)=O)CCN(C(=O)C(C2CC2)OC)CC1O 49491,c1(C(=O)OCCCN(C)C)nc(=NCc2cccc(Cl)n2)[nH]c2c1COC2 49492,Cc1ccnc(C(=O)NCC(O)CCNC(C2CCCCCN2C)=O)c1F 49493,Nc1ncccc1C(N1CC2C(CNC(c3cc(=O)cc[nH]3)=O)C2C1)=O 49494,C(=O)(C(O)CC(C)(C)C)N1CCCC(N(C(COCc2ncc(C)o2)=O)C)C1 49495,c1(NC(C2C(C)(COC)C2)=O)cccc(NC(c2coc(Cl)c2)=O)c1 49496,C1(NC(CC(C(=C)C)OCC)=O)COC2(C1)CN(Cc1sccc1Cl)C2 49497,N1(C(C(CC=C)C)=O)C2CCC1CC(C(=O)NC1(C(=O)OC)CC1)C2 49498,c1(COC)cc[nH]c1C(=O)NCC1COCC1NC(=O)CCC1CCOC1 49499,C1(C(=O)Nc2ccc(C#C)cc2)CN(C(=O)CC2CCCCCC2)CCC1(C)C 49500,C1(C(N2CCC(NC(C3(C(F)(F)F)CCCCC3)=O)CC2)=O)CC12CC(F)(F)C2 49501,CN=c1nc(N(C)Cc2ccccc2C)[nH]c(N2CCOCC(CO)C2)n1 49502,N1(C(c2c(CC)ocn2)=O)CCCC(NC(=O)C(C)(O)C2CCC2)CCC1 49503,CCC(CC)CC(=O)N1CCCC1CCC(=O)NCc1ccc(C)cc1F 49504,C1(CNC(c2ccco2)=O)COCC2(CCN(C(=O)CC3CC4(CC4)C3)CC2)O1 49505,c1(CC)cc([N+](=O)[O-])ccc1C(N1CCC(C2CCCCN2C(=O)CO)CC1)=O 49506,Cc1cnc(Cl)c(C(=O)N(C)Cc2cccc(CNC(c3sncc3C)=O)c2)c1 49507,N1(C(C2N(C)CCOC2)=O)CC2CCN(C(c3ccc(Cl)c(Cl)c3)=O)C(C2)C1 49508,N1(Cc2onc(-c3ccc(C)c(C)c3)n2)CCC2(N=N2)C(F)(F)C1 49509,C(=O)(CS(=O)(=O)C1CC1)NC1CCCC(NC(=O)COc2cccnc2)CC1 49510,N1(C(CN(S(C)(=O)=O)C)=O)CCC2C(NC(c3sc(F)cc3Cl)=O)CC12 49511,C(=O)(C(C)(F)C(=O)NC(C)C(=O)N(CCC(F)CN=[N+]=[N-])C)OC 49512,c1(SC)cn(C)nc1C(N1CCCC(C(C)NC(C2(O)CCOCC2)=O)C1)=O 49513,N1(C(CNC(CC)=O)=O)CC2CN(C(c3ccc(-c4nnc(C)o4)cc3)=O)CCC12 49514,N1(C(=O)NCc2cc(C)no2)CCC(C2CC2)(C(=O)N(C)C)C1 49515,c1(C(=O)NC2CCN(C(CCCCOC)=O)C2(C)C)cc(F)c(F)c(F)c1F 49516,C(=O)(CCCCCN=[N+]=[N-])N(C1CN(C(=O)CC2CC(C(F)F)C2)C1)C 49517,Cc1ccc2cc(C(=O)NC3CCCC34CCN(C(C3(CO)CC3)=O)C4)[nH]c2c1 49518,C1(NC(CCOCCC)=O)CC(C)(NC(=O)CC2CCCN2CC)C1 49519,CC(C)(C(=O)NCC(=O)NCC1(CNc2ncccn2)CC1)N1CCCC1 49520,N1(C(COCCOC)=O)CC=CC1CNC(=O)CN1CCC(C)C1 49521,Cc1ccn2ncc(C(=O)NCC3CCN3C(C34CC(CN3C3CC3)C4)=O)c2n1 49522,c1(C(=O)NCC2C(NC(C3C(C(=O)OC)C=C3)=O)C2)n[nH]c2nccc(Cl)c12 49523,CC1CN(C(C2(F)CCOC2C)=O)CC1NC(C1CCCN1N=O)=O 49524,N1(C(C(COC)NC(C(COC)OC(F)F)=O)=O)CCN(C)C(=O)C1C 49525,c1(CS(N2C(C(=O)O)CC(=C)C2)(=O)=O)c(SC)cccc1Br 49526,C(CS(=O)(CCO)=NC(=O)c1ccc(-n2ccnc2)cc1)NC(=O)OC(C)(C)C 49527,CC1CN(C(=O)CC(C(F)(F)F)NC(C2(C)CC(=O)N(C)C2)=O)C12CCOCC2 49528,C12(C(=O)OC)CC(C(=O)NCC3CCC(NC(=O)CCc4ccncn4)C3)(C1)C2 49529,c1(C(=O)NCC2CCCCN2C(=O)C=Cc2ccncc2)cnc2c[nH]nc2c1 49530,C1(n2cc(C#CCNC(=O)CC(O)C(F)F)nn2)CCOC2(CCOCC2)C1 49531,c1(CNC(CC(=O)NC)C)ccccc1Cl 49532,N1(C(C(c2c(C)n[nH]c2C)C)=O)CCN(C(=O)COC=CCl)C(C2CCCC2)C1 49533,c1(CC(N2CC(C)N(C)CC2)=O)c[nH]c2ccc(-c3cncc(N(C)C)c3)cc12 49534,c1(C(=O)NC2C3(CC(NC(Cc4cnc(C)[nH]4)=O)C3)C2)ccc(N)c([N+](=O)[O-])c1 49535,c1(C(C)(C)C(=O)OC(C)(C)Cc2ccccc2)cccc([N+](=O)[O-])c1 49536,C#Cc1ccc(F)c(C(N2CC3CCC2(CNC(=O)Cc2ccsc2)CC3)=O)c1 49537,C1(NCC2CCN(C(C)C)C2)CCCCN1C(c1ccn(CCF)n1)=O 49538,O=C(C#CC1CCCO1)NCC(c1ccc(F)cc1)NC(c1cc(Cl)no1)=O 49539,C1(N(C(C(CC)C)=O)C)CCCCN(C(C2CC=CC2)=O)C1 49540,C12(OC)CC(C(=O)NCC(C)(C)NC(c3cccc(F)c3)=O)C(C1)C2 49541,c1(N2CCCC(C(N3CCN(CC#C)CC3)=O)C2)n[nH]c2c1CCC(F)(F)C2 49542,c1(C(=O)NCc2nc(C(N3CCCC3c3ncc[nH]3)=O)co2)c(O)cccc1Cl 49543,c1(-c2nc(C(C)OC)nn2CC2CCOC2)cc(=O)c2ccccc2o1 49544,c1(OCC)ccc(CN2CCCC(C)(NC(c3nccn3C)=O)C2)cc1OC 49545,C1(NC(C(CCC)OCC)=O)CCN(C(c2cc(C)n(C(C)C)c2)=O)CC1F 49546,N(C1CCOc2ccccc21)(CC#C)C(C12CC1CN(C(=O)C(C)(C)O)C2)=O 49547,CC1Cn2nc(C(N3CC(N(C)C(c4ccoc4Cl)=O)C3)=O)cc2C(=O)N1 49548,c1(CC(C)C(=O)NCC#CCNC(C2CC3(CCCO3)C2)=O)ccc(C#N)cc1 49549,C1(C(N2CC(CNC(C=C(C)C)=O)OCC2)=O)CCN(C)S1(=O)=O 49550,c1(NC(C(C)C)C(C)NC(=O)Cc2cnccc2Cl)ncnc2c1cnn2C 49551,Cc1cc(Cl)c(Br)cc1C(N1CCCC1C(=O)Nc1nc(C#N)cs1)=O 49552,C=CC1(C(N2CCC(C(F)(F)F)C2)=O)CCN(C(C2CCC2C)=O)C1 49553,N1(C(COCCCC)=O)CC2CCC1C(CNC(=O)CCCc1cnn[nH]1)C2 49554,N1(C(c2ncn(CC)n2)=O)CC(CNC(=O)C=Cc2ccsc2)C2(CCC2)C1 49555,c1(C(N2CC3OCC(NC(=O)C(F)(F)F)C3C2)=O)cccc2ncsc12 49556,C1(COC)(NC(=O)C(C2CCC(=O)N2)C)CCN(C(=O)C2=CCCCC2)CC1 49557,n1(C(C(=O)NCC(=CC(=O)NC(CCOC)C)C)C)ccnc1C 49558,c1(OC)ccc(CCC(=O)NCC2CCC2NC(C2CC3C=CC2O3)=O)c(F)c1 49559,N1(C(c2c(OC)ccc(C)c2)=O)CCC2C(CCN2C(c2cnncc2C)=O)C1 49560,c1(CC)nc(C)c(C(=O)NCC(C2CCCN2C(C2CCCOC2C)=O)(C)C)s1 49561,N1(C(C2(C)CCCCC2)=O)CC(CO)C2(CCN(C(C3COCCO3)=O)CC2)C1 49562,C1(CNC(C2(C)CCNC2=O)=O)CN(C(c2c[nH]nc2Cl)=O)C2(CCC2)C1 49563,c1(CC)ccc(O)c(C(=O)N(C(C)CCNC(C2CCC2(C)C)=O)C)c1 49564,C1(CC)C(NC(=O)CCC=C(C)C)CCN1C(=O)CCC(C)Oc1cccc(F)c1 49565,N1(C(c2ccc(C(C)=O)cc2)=O)CCN(C(=O)C(C)C(C)O)CC1CC(F)F 49566,C1(N(C(C2C=CC(NC(c3c(CC)non3)=O)C2)=O)C)CCC(O)CC1 49567,Cn1cc(C=CC(=O)NC(Cc2ccoc2)C(=O)NCC2(Cl)CCC2)nn1 49568,N1(C(c2cc(C)c(O)nc2)=O)CCC=C(C(=O)N2CCCCC2C#N)C1 49569,C12(CNC(c3cccc(CNC)n3)=O)CC=CC(C1)OC2.C1(C=O)C(C)(C)C1(C)C 49570,c1(N(C)C)ccc(C(N2CC3C(NC(=O)CN4CC(C)(C)C4)C3C2)=O)cn1 49571,CC1=C(C(=O)N2CCC(CC(N3CC(Nc4ccccn4)C3)=O)C2)CCO1 49572,CCCC(CCO)NC(=O)CN(C(=O)C(C)C#N)CC 49573,C(c1cccc(Cl)c1)=CC(=O)NC(C1CCN(C(c2cc(C)c(C)[nH]2)=O)C1)C 49574,N1(C(C(C)C#N)=O)C2CCC1CC(NC(c1ccncc1Br)=O)C2 49575,S(=O)(=O)(c1ccc(C(N2CCC(C(C)NC(c3cc[nH]c3)=O)C2)=O)o1)NC 49576,c1(OC)c(C(=O)NC(C)C(C)NC(c2cc(-c3ccco3)c[nH]2)=O)csc1Cl 49577,C1(C)(C(=O)NCC2CCN(CCC)C2)CCCN(C(c2cc(Br)nc(Br)c2)=O)C1 49578,C1(CCOC)(NC(=O)CC2(CO)CC2)CCN(C(C2CC2C(C)O)=O)CC1 49579,N1(C(C(COC)N(C)C)=O)CC(CNC(=O)CCn2ccc(C)n2)C2(CC2)C1 49580,c1(CC(N2CCC(CNC(c3ccnn3CCF)=O)C2)=O)cccc(C(F)(F)F)n1 49581,CC(C)C(O)CCNC(C1CC=CCN1C(C1CC2C=CC1O2)=O)=O 49582,C(C(CNC(=O)CC1CCC(=O)N1C)C(F)(F)F)NC(c1c(SC)nn(C)c1)=O 49583,Fc1cccc2c1CN(c1nccc(=NCCN3CCCS3(=O)=O)[nH]1)C2 49584,n1(CCOCC)cc(C(=O)N(C)CCNC(C2CCC(C(N)=O)C2)=O)cn1 49585,c1(OCC(N2CCC(N(C)Cc3cccnc3O)C2)=O)cc(F)cc(Cl)c1 49586,CCC(C)C(=O)N(C)CC1(O)CN(C(C2C=C(C)CS2)=O)C1 49587,c1(C(N2CC(NC(C(CCC)O)=O)C(OC)C2)=O)cnc2c(c1)CNC2=O 49588,Cc1ccc(C(=O)O)c2c1N(CC(=O)NCCC1CCC1)CCC2 49589,c1(N(CC=C)C)[nH]c(=NC2CC3(CCCC3)C2)nc2c1ncn2C 49590,CC(C)CCCC(C)NC(=O)CN1CCN(C(C2C=CC=CC=C2)=O)CC1 49591,N1(C(c2c(C)csn2)=O)CCN(C(c2ccc(F)cc2O)=O)C2CCCC2(C)C1 49592,N1(C(C2(COC)C=CCC2)=O)CCCC(NC(c2nnsc2SC)=O)C1 49593,CC1=C(C(=O)NC(CNC(c2cc(C(F)(F)F)n[nH]2)=O)CC(F)(F)F)CCCO1 49594,N1(C(Cn2c(C)ncc2)=O)C2CCC(C2)C1CNC(C1COC2(CCC2)C1)=O 49595,N1(C(c2ccc(C(C)=O)cc2)=O)CC(C2CCCN(C(=O)C(C)(C)C(C)O)C2)C1 49596,N1(C(c2n(CC#C)cnn2)=O)CCC2C(C(=O)NCCOCC(N)=O)C2C1 49597,Cn1ccc(C(N2CC(C)(NC(=O)CC3(O)CCOC3)C2)=O)c1C1CCC1 49598,C1(NC(C2CC2(F)Cl)=O)CCN(C(=O)C(C2CCCC2)C2CCCC2)CC1 49599,N1(C(C2CC(CC)C2)=O)CC2CC2(NC(=O)CNC(c2cccc(NC)c2)=O)C1 49600,C1(CC(=O)O)CCC(C)(C)CO1.CC1CN(C(=O)OC(C)(C)C)C1CN(C)CC 49601,c1(C(N2CC(NC(C3(OC)CCOC3)=O)C2)=O)cc2c(C)c(Cl)ccc2[nH]1 49602,N1(C(CCC2CC(OC)C2)=O)CCCN(C(c2cc(C#N)ccc2Cl)=O)CC1C 49603,Cc1cc(N2CCCCC2)cc(NCc2ncc(F)cc2O)c1 49604,C1(CNC(c2cn(C(C)C)nn2)=O)(CO)CCCN(C(C2CCCC(F)C2)=O)C1 49605,c1(N(C2CCCO2)C(N(C2CN(C(=O)OC(C)(C)C)C2)C)=O)ccc(F)c(F)c1F 49606,c1(C(=O)NC2CC(CNC(Cc3c(C)nsc3)=O)C2)coc2c1CCCC2 49607,C1(C(=O)NC(C)CNC(=O)Cc2nc[nH]n2)CCCCN1S(N)(=O)=O 49608,CC1CCN(C(=O)C(N2CCC(C)(c3ccccc3)C2)=O)CC1C 49609,CC1=NOC(C)(C(=O)NCCC(=O)NCCS(C)(=N)=O)C1 49610,C1(CC(N2C(CNC(CSC)=O)COCC2)=O)CN2CCN1CC2 49611,Cc1ccc(N2CC(NC(C3(N4CCCC4)CCCC3)=O)CC2=O)cc1 49612,c1(N(CCCOC)C)nc(N2CCCC(OC3CC3)C2)nc2scnc12 49613,CC1CC(=O)NC1C(=O)NCC1CC(NC(c2cnn(C(C)(C)C)c2)=O)C1 49614,CC1CC(NC(c2cc(CF)on2)=O)CN(C(c2c[nH]nc2C2CCC2)=O)C1 49615,C12(NC(c3c(C)cc(C)s3)=O)CCOC(CNC(C3CCC(=O)NC3)=O)(C1)C2 49616,CCCC(C)(O)CC(=O)NCC1CC(F)CN1C(=O)Cc1nccs1 49617,Cc1oc(C(=O)NCCC2(O)CN(C(c3ccc(C(C)C)cn3)=O)C2)cc1CO 49618,C#Cc1ccc(CC(N2CCOC(C)(CNC(c3cnnc(O)c3)=O)C2)=O)cc1 49619,c1(C(=O)NCC(C2CC2)NC(c2n(C)nc(C(F)(F)F)c2)=O)c(F)cc(Cl)cc1F 49620,c1(C(N2CCCC(O)(CNC(CCCOC)=O)C2)=O)cc(OC)cc([N+](=O)[O-])c1 49621,CC1CC(C)(C)CN1Cc1nc(-c2cn(-c3ccccc3F)nc2C2CC2)no1 49622,Cc1c(Br)sc(CNCC(C)(C)CN)c1Br 49623,c1(C(=O)NCC2(OC)CCN(C(c3ccon3)=O)C2)ccc(F)c(SC(C)C)c1 49624,N1(C(C2(NC(c3n(C=C)ncc3)=O)CCN(C)C2)=O)CCC2(CCC2)C(O)C1 49625,N1(C(C(C)SC(C)C)=O)CCC2C(C1)CN2C(=O)CCCc1ccc(Cl)c(Cl)c1 49626,c1(N2CCCC(NC(C)=O)C2)ncnc(NCC2CCCC2(C)C)c1C 49627,C1(C(=O)NC(C2CCCN2C(C2CC2(C)C)=O)C)CCN(C(=O)OC(C)(C)C)CC1 49628,C1(N(C)C(C2CC23CCC3)=O)CC2CC1N(C(c1ccc(N)cc1F)=O)C2 49629,C1(NC(c2ccccc2)=O)N(C(=O)CC(O)c2ccccc2)CC12CCCC2 49630,N1(C(c2c(SC)ccs2)=O)CCOC2(CCN(C(C3CCOCC3)=O)CC2)C1 49631,C1(NC(=O)Cc2cccc(F)c2Cl)CC12CCC(NC(c1cnsn1)=O)CC2 49632,Cc1cnc(C(N2CCC(C)(C(N3CC(N4CCCC4=O)C3)=O)CC2)=O)c(F)c1 49633,Cc1oc([N+](=O)[O-])cc1C(=O)N(CCCNC(=O)C=CC1CCCN1C)C(C)C 49634,CN(CCCC(=O)NCC1(C)CCCN(C(C2CCN2S(C)(=O)=O)=O)C1)N=O 49635,c1(C(=O)NC2C(NC(=O)Cc3ncncc3Cl)CCOC2)cnc2nccn2c1 49636,C1(COC)(CNC(C2CCCCC2O)=O)CCCN1C(=O)CC1(C)OCCO1 49637,c1(C(=O)NC23CC(NC(CC4CC(C(=O)OC)C4)=O)(C2)C3)ncc(C)cn1 49638,C#CCC(C)(C)C(=O)NCCC1CCC(NC(c2n[nH]cc2OCC)=O)C1 49639,N1(Cc2ccc(OC(C)(C)C)cc2)CC2CC(C1)N2C(c1cc(F)c[nH]1)=O 49640,c1(C(N2CCC(CNC(C(CCC)CC)=O)C23CC3)=O)ccc2c(c1)NC(=O)C2 49641,O=C(CCCCCCCO)NC1CC(CC(=O)NCc2nnco2)C1 49642,c1(C(=O)NC(C)CCNC(C2(F)CCCC2)=O)cc(Cl)cc(Br)c1N 49643,N1(C(c2ccn(CC)n2)C(=O)NC2CCCCC2)CC2CCC(O)CC2C1 49644,C1(NC(C2CCC(C)C2)=O)CN(C(C2C3CCCC23)=O)CCC12CCC2 49645,n1(CC(N2CC(CC(C)NC(C(C=C=C)C)=O)C2)=O)ccc2ccccc2c1=O 49646,C(=O)(CC(C)(C)Cn1cc(CN2CC(=O)CCC2=O)nn1)N(CC)CC 49647,c1(CCC)onc(C)c1C(=O)NC1CN(C(=O)CCc2ccc(OC)cc2)C1 49648,C1(NC(C=CCOCCOC)=O)COCCN(C(c2cnc(S)n2C)=O)C1 49649,C=C(C)C(CC(=O)NC1CN(c2cc(O)nc(SC)n2)CCC1C)OCC 49650,C12(C(N3CC(O)(C(C)NC(c4ccc(Br)c(O)n4)=O)C3)=O)CC(C)(C1)OC2C 49651,c1(CC)cccc(C(=O)N(C(C)CN(C)C(C2(Br)CC2)=O)C)n1 49652,C(CCCC(C)(C)C(=O)NNC(=O)C(C)CC=C)OCC#C.N1CCCC1 49653,N1(Cc2cnc(C)nc2)CC2CCC(C1)C2CC(N1CCC(C#N)C1)=O 49654,CC1CC(C)CN(C(C2CC(N(C(=O)CN3CCCCC3C)C)C2)=O)C1 49655,C(=O)(C(O)CC(F)F)NC(CC)CNC(=O)Cc1cc(-c2ccccc2Cl)on1 49656,c1(C(=O)NC2C(NC(CC(C)(C)C)=O)CCC2)cc2ccccc2cc1N 49657,c1(C(=O)NCCN(C)C(C2C3CC3C3CC23)=O)cccc(OCC(F)F)n1 49658,N1(C(CCCCOCC)=O)CCN(C(c2cn(CCO)nc2C)=O)C(C2CC2)C1 49659,C=CCCCC(=O)N1CCC(n2cc(CNC(C34CC(F)(C3)C4)=O)nn2)C1 49660,C1(NC(C(C)(C)SC)=O)CCCC(CNC(c2ccc(O)cn2)=O)C1 49661,c1(OC)cnc(F)c(C(=O)NCC(C2CCCCC2)NC(=O)C(F)(F)CF)c1 49662,Cc1ccc2c(C(N3CC(CC(C)NC(C4(S(N)(=O)=O)CC4)=O)C3)=O)csc2c1 49663,C1(CC(=O)NC(c2nocc2C(=O)NCC(F)(F)C(F)F)C)CCCC(C)C1 49664,c1(C(=O)NCC2C(NC(C(C)OC)=O)C2)ccc(C(N)=O)nc1 49665,CC(CC(=O)NC1CC2CCC(C1)N2C(c1csc(C(=O)O)c1)=O)C(C)(C)C 49666,c1(C(=O)NCC2(CNC(c3c(CC)ocn3)=O)CCC2)ccc(F)c(C(F)F)c1 49667,n1(CC(N2CC3C(NC(c4c(C)cns4)=O)(C3)C2)=O)nc2n(c1=O)CCCCC2 49668,C(CC(C)C(=O)N(C1CCC(CNC(c2cc(Cl)cs2)=O)CC1)C)=CC 49669,C1(C(=O)NC2C=CCN(C(C3N(CCC)CCCC3)=O)C2)CCc2nncn2C1 49670,C1(C(N(C)Cc2ccc(CC)o2)=O)CCCN(C(=O)COC(C)=O)C1CC 49671,CCC(C)(CNC(C1CC2CC2C1)=O)C(=O)NCCCn1cnnc1C 49672,c1(C(=O)NCc2ccn(CC)n2)cccc(CNC(C2CCCN2C)=O)n1 49673,CC12CCC(C(=O)NCCC3CN(C(C4CCCCCC4)=O)C3)(CC1)CO2 49674,c12ccc(F)cc1NC2=O.N1(C(c2c(C)n[nH]c2)=O)CC2C(C1)N2S(C)(=O)=O 49675,c1(-c2cn(S(CCC)(=O)=O)nn2)cc(F)ccc1Br.C1CCN(C(=O)C(C)(C)C)C1 49676,C1(CC(=O)N(C(c2ccccn2)C)C)CCCN(C(C2CCCO2)=O)CC1 49677,N1(Cc2cc(C)nn2C)CCn2nc(C(C)C)cc2C1.C1(N2C(=O)N2)CCC1 49678,C1(NC(C(C=C)OC)=O)CC2CCC1(C(=O)Nc1cnc(O)c(C)c1)C2 49679,c1(CC)c(C(=O)NC2CCCC2CNC(=O)Cc2csc(C)c2)csc1C 49680,N1(C(C(C)SCCCC)=O)C2CCC1C(C)C(NC(c1nc(C)oc1C)=O)C2 49681,c1(OC(C(=O)N(CCC)CCNC(=O)C(C)n2cnnn2)C)ccc(C)cc1 49682,c1(C(N2CC(F)(CNC(c3cc(C(F)F)no3)=O)C2)=O)nccc(F)c1Cl 49683,N1(C(=O)NCc2c(OCCOC)cccc2)CCCC(CO)CC1 49684,C(=O)(C(CN(C)C)NC(=O)Cn1ccnn1)N(C(C(C)SC)C)C 49685,N1(C(CN(C(c2cnc(O)cc2C)=O)CC)=O)CCSC(C)C1C 49686,c1(CC(=O)NC(C)CC2CN(C(C3CC(C)(O)C3)=O)C2)cc(F)ccc1Br 49687,Cn1cccc1C=CC(=O)NCC1(F)CC(NC(=O)C=Cc2cnccn2)C1 49688,OC1(C2CCCN(Cc3cn(C4CC5CC45)nn3)C2)COC1 49689,C1(C(=O)NCCOCCNC(c2nn(CC)nc2C)=O)C2CS(=O)(=O)CC12 49690,N1(C(C(c2ccc(F)cc2)=O)=O)CC(NC(C2CC3C=CC2CC3)=O)CC(O)C1 49691,C1(C(N(C)CC2(NC(C(C)Oc3cccc(C)c3)=O)CC2)=O)CC2(CCCC2)C1 49692,C(CCCCCNC(=O)CCc1cccnc1Br)N(C(C1C(=C)CC1)=O)C 49693,C(=O)(CCCN(C)N=O)N1CC(CCCNC(CCC2CC(OC)C2)=O)OCC1 49694,c1(CC)cnccc1C(=O)N(C1CC(C(=O)NC2(C)CC2)C1(C)C)C 49695,N1(CC)CCC2(CC(NC(=O)COCNC(=O)NC)C2)C1.C12CC(C1)CN2 49696,C=CC(CCC)CC(=O)NC(C(=O)NC1CCCCCCC1)C(C)(C)C 49697,N12CCCC(C1)C2=O.n1(CC)cc(NC(c2c(OC3CCCC3)c[nH]n2)=O)cn1 49698,c1(OC)cc(C(=O)NCC2(F)CC(NC(=O)C(F)OC)C2)c(OC)cc1C(F)F 49699,c1(CN2CCN(C=O)CC2)cc(Cl)c(Cl)c(Cl)c1.c1(N)ccc(ON)cc1 49700,N1(C(Cc2cc(C)on2)=O)CC23CCCC2(C1)CN(C(=O)CN(C)C)C3 49701,N1(C(c2nc(C(N)=O)sc2)=O)CC2(COC(CNC(c3coc(Cl)n3)=O)C2)C1 49702,NCCCC(O)C(=O)NC(Cc1ccccc1O)C(=O)O 49703,C(=O)(CC(F)(F)C(C)(F)F)N1C(C)CCC(CNC(=O)CCc2nncs2)C1 49704,N1(C(c2c(CC)noc2)=O)Cc2n[nH]cc2C1C(=O)N1CC(N2CCC2)C1 49705,c1(N2CCCCC(CO)C2)nc2c(c(=NCC3CC3(F)F)[nH]1)CSC2 49706,C(=O)(C1=NOC2COCC12)N1C(C(=O)NC(CC#C)CO)(CC=C)CCC1 49707,Cc1nc(C2CCC2)sc1CC(=O)N(CCCNC(C1CC1CF)=O)C1CC1 49708,N1(C(CCC(CC)=O)=O)CC2(CCCC2NC(=O)C=CC2CCCN2C)C1 49709,c1(C(=O)NC2CC(C(C(N3C(C(C)O)CC3)=O)F)C2)cc(C(N)=O)co1 49710,CC(CCCNC(=O)C(O)Cc1ccccn1)NC(=O)C=CC=C(Cl)Cl 49711,C1(NC(C2(C)C=CCC2)=O)COCCN(C(=O)Cc2ccsc2)C1 49712,N1(C(C=CCC)=O)CC(F)(n2cc(COCC(=O)O)nn2)C1 49713,n1(CCC)cc(C(=O)NCCCC2CCCN2C(C2CCS2(=O)=O)=O)nn1 49714,N12CCC(CC13CCC3)C2=O.N1(C(c2nc(C3CC3)no2)C)CCC(C)C1 49715,C1(C(=O)NCC2CN(C(Cc3cc(C)on3)=O)C(C)C2)CCC2(CCOCC2)O1 49716,c1(CC(=O)NC(CC)CNC(C2(C3CCCO3)CCC2)=O)c(OC)cccc1Cl 49717,c1(OC)ccc(C2CCN(CCn3cccn3)C2)c2ccccc12 49718,C=Cc1ccc(C(N2CCN(C(C3C(F)(F)C34CC4)=O)C(CCC)C2)=O)cc1 49719,CC1OCCCC1C(N1CCC(CCC(=O)NCCCN2CCOCC2)CC1)=O 49720,C1(C2CC2)(C(N(CC(C(C)C)C)C)=O)CN(C(C2CCCSC2C)=O)C1 49721,c1(CC)ccnc(C(N2CCCC2CNC(=O)CCC2CC=C(C)CC2)=O)c1F 49722,n1(CC)ncc(C(=O)NC(C2CCN(C(=O)CNC(=O)COC)C2)C)c1C1CC1 49723,C1(NC(C(C)Oc2ccccn2)=O)(CNC(C2(C(N)=O)CC2)=O)CCOCC1 49724,c1(CCC)cc(=NCCCOCCNC(c2nc(O)n[nH]2)=O)[nH]cn1 49725,N1(C(COC2CC(NC(C3CCC(=O)N3)=O)C2)=O)CCN(CCCO)CC1 49726,n1(CCC)nnnc1C(c1ccc(CCC)s1)NCCc1ccoc1 49727,c1(C(=O)NC(C)CN(C(=O)Cc2ccc(F)cc2)C)c(F)ccc(Cl)c1F 49728,CC1CN(C(=O)C=C2CCN(C)C2)CCCN1C(=O)CN1CC(=O)N(C)C1=O 49729,c1(OCC(=O)NCC(C)N(C)C(c2ccc(CC#N)cc2)=O)ccc(Cl)cn1 49730,c1(CC(N2C(CNC(=O)C=Cc3ccccc3)CCCC2)=O)cc(F)ccc1O 49731,Cc1cccc2c(C(=O)NCC3CC3NC(=O)CSc3cccc(Cl)c3)n[nH]c12 49732,N1(C(CN2C(C)CCC2C)=O)CCC2(CCCN(C(=O)CCCCF)C2)C1 49733,c1(C(N2CC(NC(=O)COc3ccc(Br)cc3)C2)=O)ccc2nncn2c1 49734,N#Cc1cc(C(=O)NCC2(NC(c3ccc(Cl)o3)=O)CCC2)cc(O)c1 49735,C12(C(N3C4C(NC(c5cc6c(s5)CCC6)=O)C(C4)C3)=O)CCC(O)(CC1)CC2 49736,C1(CNC(c2ccc(OC)cc2F)=O)C2CCCC1N(C(c1coc(Br)n1)=O)C2 49737,N1(C(c2c(C)nccn2)=O)CCC(NC(=O)COC2(C)CCC2)C12CC2 49738,CC1(C)COCCC1C(N1CCC(CCNC(=O)C=CC2CC2)C1)=O 49739,CN1CC2(CCN(C3CC4(C3)CN(C(C3CCS(=O)(=O)C3(C)C)=O)C4)CC2)C1 49740,C1(CCOC)CN(C(C2(Cl)CC2(C)C)=O)CCN1C(c1ccn(C)c1)=O 49741,N1(C(C2C(NC(C(C)n3ccnc3)=O)C3CCC2C3)=O)CCc2nc[nH]c2C1 49742,Cc1cccc(CC(=O)NC2CC2CNC(C2CC2CN(C)C)=O)c1 49743,c1(N(CC(C)C#N)Cc2ccc(C)cc2)ccc2ncc(I)n2c1 49744,c1(C(C)(F)F)csc(C(=O)NC2(CO)CN(C(c3csc(Cl)c3)=O)C2)n1 49745,N(C(=NCc1cnn(C)n1)NCC(F)F)C(C)CCc1ccccc1 49746,c1(C(=O)NC2C(NC(CCOC)=O)CCC2)cc2c(cc1Br)OCO2 49747,c1(C(=O)NC(CCNC(C2(SC)CC(O)C2)=O)C)ccc(C)c(CO)c1 49748,N1(C(c2cc(C3CC3)nc(O)c2)=O)CC2CC1CN2C(C1C=CCCC1)=O 49749,CC1CC=C(C(=O)NCC23CCC(CC2)N(C(C2CC4CC2CC4O)=O)C3)CC1 49750,C(=O)(C1=C(c2ccccc2F)CCC1)ONC(CN1C(c2cc(C)sc2)CCC1)=O 49751,CC1CCC(CCNC(=O)C(Cc2ccoc2)NC(C2CCC(O)C2)=O)CC1 49752,C(C)(CCC(=O)N(CCCN(C(=O)Cc1cnc(C)o1)C)C)SC 49753,c1(CSC)ccc(SCCCCC(=O)N(C(=O)NC(C)(C)C)C(C)C)cc1C 49754,C(C(C(C)C)NC(c1ccccn1)=O)(C1CCCCC1)NC(CCCC)=O 49755,CN1CC(F)CC1C(N1CCC(C(F)C(=O)NCC2CNC(=O)C2)C1)=O 49756,Cc1cnc(NC(=O)C(C2CCCCC2)NC(c2cn(C)nn2)C2CC2)c(C)c1 49757,N1(Cc2cccc(C)c2O)CCc2nn(C)c(C(=O)Nc3cccc(Cl)n3)c2C1 49758,CCC(CNC(C1(F)CCCC1)=O)N=c1[nH]nc(CO)s1 49759,N1(C(C2CCC(C)O2)=O)CCCC2C1CCN2C(c1cccc2c1CC(=O)N2)=O 49760,c1(CC)sc(C(=O)NCC2(C)CCN(C(=O)C(c3cccnc3)C)C2)cc1C 49761,CC1CC2(CC(C(=O)NC3CCN(C(C4CCS(=O)(=O)CC4)=O)CC3F)C2)C1 49762,c1(CC(N2CC(C(C)(C)O)C2)=O)cc(F)cc(F)c1.c12ccc(cc1)C(=O)NC2 49763,C1(C(=O)NCCOCCC#C)C2CC3C(C2NC(=O)C(C)(C)Cl)C13 49764,C1(C)(CC)CC(C(=O)NCCCNC(=O)CC#N)CCO1 49765,c1(C(N(C(CNC(CCc2ncc(C)[nH]2)=O)C2CC2)C)=O)ncccc1C(F)F 49766,Cc1nnn(C)c1C(N1CCC(C)(CNC(c2ccccn2)=O)C1)=O 49767,c1(C(=O)NC2CCN(C(C(C)=CC)=O)C2CC)cnn2cccc(Cl)c12 49768,C1(C(N(CCC(C)F)CCN(CC)CC)=O)CCC2(CCOC2)O1 49769,C#CC1CN(C(=O)CN(C)C(C)C)CCN1C(=O)CC1(C2CC2)CC1 49770,N1(c2c(C#N)cc(Br)cn2)CCCC(C2(NC(C3CCCC(O)C3)=O)CC2)C1 49771,CC1(CNC(C2CC(O)C2)=O)CCN(C(c2cc(C(F)F)on2)=O)C1 49772,CC(O)C(C(=O)N1CCN(C2CCC2)CC1)NC(=O)CC1CC2C=CC1C2 49773,CC(C)(C)C(CNC(C1CC1Cl)=O)C(=O)NCC1(c2ccon2)CC1 49774,C1(NC(c2cc(C)[nH]c2)=O)CC2C1CCN2C(c1cnn(CC(C)(C)O)c1C)=O 49775,c1(C(=O)NCC(C)NC(C(CC)(O)c2ccccc2)=O)ccc2c(c1)CNC2=O 49776,Cc1cc(C)c(C(N2CC(O)(CCNC(=O)C(C)OCCN(C)C)C2)=O)c(O)c1 49777,N1(C(C2C(=C)CC2)=O)CCN(C(c2cc(C(C)C)on2)=O)C(c2ccccc2)C1 49778,C1(CCOC)(NC(=O)CSc2nncs2)CCN(C(c2ccc(CO)cn2)=O)C1 49779,CC1CC(CNC(c2cc(C(F)(F)F)on2)=O)CN1C(=O)C(F)C1CCOC1 49780,N1(C(Cc2c(C)nn(C)c2C)=O)CC(C)OC2(CCN(CC3CCOC3)CC2)C1 49781,Cc1ccc(C(=O)NCC2(O)CC(NC(C3CCN(C)C3=O)=O)C2)cn1 49782,C1(NC(=O)COC2CC2)CC2CN(C(c3cc(Br)c(F)cc3F)=O)CC2C1 49783,C1(CNC(=O)C(F)C(F)(F)F)CC2CCC(C1)N2C(c1ccc2c[nH]nc2n1)=O 49784,S(=O)(=O)(c1ccc(=NCCNC2CC2)[nH]c1)N(C)CCOCCCN1CCOCC1 49785,C1(CC(=O)NC2(CCOC)CCCC2)CCCCN1C(=O)C=C(C)C(C)C 49786,N1(C(C2C(CC)CCO2)=O)CCCC(C(=O)NCC(=O)OC(C)C)CC1 49787,C1(n2cc(-c3c(C)nccn3)nn2)CC2CCC1(NC(=O)Cn1cc(Cl)cn1)C2 49788,N1(C(c2c(OCC)ccc(Cl)c2)=O)CCC=C(C(=O)N2CCC(O)(CO)C2)C1 49789,N1(C(C23CC(n4cc(CCSC)nn4)C2C3)=O)CCN(CCN(C)C)CC1 49790,C1(NC(C#CC2(C)CC2)=O)CN(C(C2(c3ccsc3)CC2)=O)C2(CCC2)C1 49791,C#CCC(C(=O)NC)NC(c1cc(CNC(c2nccnc2C)=O)[nH]n1)=O 49792,C1(O)(CNC(CCOCCN(C)C(c2cocn2)=O)=O)CCOC1 49793,c1(-n2cc(CN(C(=O)C(O)C(F)(F)F)C(C)C)nn2)cccc(S(C)(=O)=O)c1 49794,C1(C2CC2)(NC(c2c(C)nc[nH]2)=O)CCN(C(=O)CC2OCCOC2(C)C)C1 49795,c1(OC)cccc(CN2CCC(CNC(c3c(C4CC4)noc3C)=O)CC2)c1 49796,CC1(C)CC(F)(F)CCC1C(N1CCOC(CCNC(=O)C2=CCC2)C1)=O 49797,n1(CC)cc(C(=O)NCCCC2CN(C(=O)C(C)c3cc[nH]n3)CCO2)c(C)n1 49798,c1(OC)ccc(F)c(C(=O)NC2CCCCC2NC(c2cccnc2)=O)c1F 49799,C1(C(=O)Nc2cn(CC(=O)OC)nc2)CCC(NC(=O)CNC=O)CC1 49800,Cc1cc(C(N2CCCC(CNC(=O)CC3OCCCC3(C)C)C2)=O)ccc1N 49801,C1(CNC(c2c(C)cn(C)n2)=O)C2CCC(C2)N1C(C1(CCF)CC1)=O 49802,C1(NC(C2(COC)C=CCN2C(=O)CCc2ccc[nH]2)=O)CCCCCC1(C)C 49803,c1(C(N(CC(C)NC(C2CCC3(CCC3)O2)=O)C)=O)csc(S(C)(=O)=O)c1 49804,CC1(C(=O)NCCNC(=O)CCc2nc(O)n[nH]2)CCc2ccccc21 49805,C1(C2CCN(C)CC2)(C(=O)NCCC(C)NC(c2cccc(C3CC3)c2)=O)CC1 49806,c1(C(N2CCCC(C3N(C(CCCC#C)=O)CCCC3)C2)=O)c(C)nn(C)c1Cl 49807,N1(c2n(C(C)OCC=C)c(COCCO)nn2)CCOC(CC)(CC)C1 49808,C1(n2cc(CNC(C)=O)nn2)CCN(C(c2ocnc2C)=O)CC1 49809,c1(SC)nc(=NC2CCCN(C(c3ccccc3C(C)(F)F)=O)C2)s[nH]1 49810,C1(CNC(C2CCC(C)CC2)=O)C(C)CCCN1C(=O)CC1CCN(C)C1=O 49811,c1(C(=O)NCC(CC)NC(COC(CC)C)=O)cnn(C2CCCC2)c1 49812,N1(C(C2(C)N(Cc3c(C)scc3)CC2)=O)C2CCCC1COC2 49813,C=CC1(CC)COCCN1C(c1ncc(Br)cc1Cl)C(=O)NC(C)(C)C 49814,c1(C(=O)Nc2c(C(N(CC(C)C)CCC)=O)n[nH]c2)cc2ccccc2o1 49815,Cc1ccc(CC(N2CC3(CNC(C4CN(C)C4)=O)CCC2C3)=O)cc1F 49816,Cc1cc(C=CC(=O)NC(C(=O)NC2COCC2CO)C2CCCO2)on1 49817,N1(C(C(COC(C)C)(C)C)=O)CCCC(NC(c2cnc(O)c(F)c2)=O)C(F)C1 49818,c1(C(=O)NC(C)CCCCNC(=O)C2CC2)coc2c1COC2 49819,C1(NC(c2ccc(Cn3cccn3)o2)=O)CCCCC1CNC(C1(CF)CC1)=O 49820,N1(C(C2CC(NC)C2)=O)CCC2(CC1)OC(=O)NC2C 49821,N1(c2ncccn2)CCC2CN(c3ncc(C4CC4)cn3)CC2C1 49822,C1(NC(C2CCC(N(C)C)CC2)=O)CCN(C(=O)Cc2ccnn2C)CC1O 49823,N1(C(C2C(=C)C2)=O)CCN(C(c2ncc([N+](=O)[O-])n2C)=O)C2(CCC2)C1 49824,C1(N(C)C)(CNC(=O)NCc2ncoc2-c2ccccc2)CCSC1 49825,c1(C(=O)NC2C(NC(c3cc(C)nn3C)=O)CC2)c(C)nc(O)nc1C 49826,C1(NC(C2CC(C)(C)C2)=O)(CO)CCCN(CC(c2cc(C#N)on2)=O)C1 49827,c1(C(CCOC)NC(=O)C(C)O)cc(C(F)(F)F)ccc1C(F)(F)F.C(C)(=O)N 49828,c1(OC)cc(C=CC(=O)NC23CCCC2CN(C(c2cscn2)=O)C3)ccc1F 49829,c1(C(=O)NC(C)CCN(C)C(c2ccco2)=O)nccc(Cl)c1Cl 49830,c1(OC)ncc(Br)c(C)c1NC(=O)N(C)Cc1cc(F)ccc1C(F)(F)F 49831,C(=O)(C(C)CC(N)=O)NCc1cc(N2CCN(C(CN(C)CC)=O)CC2)ncc1 49832,C1(C(N2C(C)(C)CC(NC(c3cc(Cl)ccn3)=O)C2)=O)CN2CCCCC2CO1 49833,c1(NS(CC)(=O)=O)ccc(C(=O)NC(CNC(C2(C)CCNC2=O)=O)CO)cn1 49834,c1(C(=O)NC(CNC(c2cc(CSCC)on2)=O)C2CCC2)cc(Cl)ccc1O 49835,c1(CC(=O)NC2C(CNC(C3CC(OC)C3)=O)CCCC2)ccc(O)c(C)c1 49836,C1(CNC(C(CC)(C)OC)=O)C2CCC(C2)N1C(=O)CCc1ccc(Cl)cc1 49837,c1(CCC)ccc(C(=O)NCC(C2CCC2)NC(=O)C(N2CCNC2=O)C)[nH]1 49838,N1(C(C(CCCC)C)=O)CC2=C(C1)CN(C(C1CCCCC1CC)=O)C2 49839,Cc1cc(Cl)c(C(=O)NC(C2CN(C(c3cnc(S)nc3)=O)CCO2)C)cc1N 49840,N1(C(c2ccc(CC)o2)=O)CCC(NC(c2sc(C)c(C)c2C)=O)CC1C1CC1 49841,N1(C(CCC=CC(C)C)=O)CCN(CCNC(C2(C)CC=CCC2)=O)CC1 49842,C1(NC(c2c(C)ncc(C)c2)=O)CCCC12CCN(C(c1cn[nH]c1)=O)C2 49843,c1(C(N(C(CCNC(c2c(C)nn(CC)c2Cl)=O)C)C)=O)cccc2c1CCN2 49844,c1(C(C)NC(=O)CN(C(=O)CCC2CC2(F)F)C)nncn1C 49845,C(=O)(C(F)(F)CC)NCC(CCOC)NC(C1N(C(CCC)=O)CSC1)=O 49846,C1(C(=O)NCC(C(C)C)NC(=O)CCn2cccn2)CCC2(CC2)C1 49847,c1(C(N(C)CC2(CNC(c3cccs3)=O)CC2)=O)nc(O)nc(O)c1N 49848,c1(-c2scc(C(N3C(CNC(COCC=C)=O)CC3)=O)n2)ccc(O)cc1 49849,c1(C(=O)NC2(COC)CCN(C(c3ccccc3)=O)C2)ccc(=O)n(C)n1 49850,N1(C(C)=O)CCCC1COC(C)CNC(C1(Nc2ccccc2)CCC1)=O 49851,C(CC(F)F)(C(=O)NCC(=O)NC1CCCC1)N(C(c1cncc(CC)c1)=O)C 49852,C(C(=O)N(CCCCCCNC(=O)C=C1CCC(C)C1)C)(C(C)C)OCC 49853,C1(C)(C(N(CCC)CCNC(c2ccc(Cl)o2)=O)=O)SCCCS1 49854,C1(C(N(CCCN(C(c2c(C)ccc(O)c2)=O)C)C)=O)CCCCC1P(C)(C)=O 49855,Cc1nn(C)c(Cl)c1CC(=O)NCC1CCN1C(C1(C)CC(F)(F)C1)=O 49856,c1(N2CC(C)NC(=O)C2)nc(N2C3CCC2COC3)nc2c1COC2 49857,c1(N2CCC(NC(c3c(C)cc(OC)cc3C)=O)C2)ncnc2cc(C)[nH]c12 49858,C12CN(CCN1C(c1nocc1Br)=O)C(=O)C2.c1(CC)scnc1C 49859,C#Cc1cnc(C(=O)NC(CC2CCC2)C(=O)N(CCC=C)C)c(C)c1 49860,C1(CCC)CN(C(c2cnc(Br)c(OC)c2)=O)CCN1C(=O)CCSC 49861,C(=O)(CC(CC1CC1)NC(C1(CC)CCOC1)=O)NCC(CC)O 49862,N1(C(C2(C)CC2)=O)CC2(C1)CN(C(c1csc(Cl)c1Cl)=O)CC2CO 49863,c1(C(=O)NC2C(C)CN(C(C3CC(Cl)(Cl)C3)=O)CC2)cc(C#N)c(F)cc1F 49864,C1(OC)CN(C(c2c(Cl)cccc2Br)=O)CCC1NC(=O)CC1CCCCO1 49865,C1(C(N(CC(=O)OC)C2CC2)=O)CCC(n2cc(CCCNC(C)=O)nn2)C1 49866,N1(C(Cc2c(F)ccc(C)c2)=O)CC2CCN(C(c3cn(C)nn3)=O)CC12 49867,N1(CC(N2CC(O)(CNC(C3(c4cccnc4)CCCC3)=O)C2)=O)CSCC1=O 49868,N1(C(COC2(C)CN(C(=O)CCc3cccnc3)C2)=O)CC2(CC(CO)CO2)C1 49869,N1(CC2N(CC)CCC2)CCCC(C(=O)N(C)Cc2nncn2C)CC1 49870,C(C(C(=O)NCc1ccc(CNC(=O)C(C)O)s1)N(C)C)OC(C)C 49871,C1(C(=O)NCC2C3CN(C(=O)CCN4CCOC4=O)CC23)CCc2cnnn2C1 49872,c1(C(=O)NCCC(F)(F)F)cnc2ncc(-c3cccc(C(=O)C(F)(F)F)c3)cn12 49873,CC1CC2(CC(C(=O)NC(CC(C)C)C(=O)Nc3cncnc3O)C2)C1 49874,Cc1cccc(NC(=O)NC2(CO)CN(C(=O)Nc3ncccc3F)C2)c1C 49875,c1(C(N(C(CNC(C(C)OC)=O)C)C)=O)ccc(F)c2c1OCC2 49876,CC(C)C(O)C(C)(C)C(=O)NC1CCN(C(=O)C2=CCCC2)CCC1CO 49877,Cc1ccc(F)c(CNC2CC(n3cc(-c4nn(C)cc4[N+](=O)[O-])nn3)C2)c1Br 49878,c1(OC)ccc(C(C)C(=O)NCC(O)CNC(c2cnc(N)c(N)c2)=O)c(C)c1 49879,C(N=c1ccnc(NC(=O)C(C)(C)C)[nH]1)c1c(N(C)CCOCC#N)cccc1 49880,C1(NC(c2coc(Cl)n2)=O)C2CC3CN(C(=O)C4=CCCSC4)C1C3C2 49881,C(=O)(CCCCCC(C)(C)C)N(CCCNC(CCc1ccc(C)s1)=O)C1CC1 49882,c1(OC)ncc(F)cc1C(=O)NC1(CNC(c2ccc(-n3cccc3)nc2)=O)CC1 49883,N1(C(c2c(N)cc(F)cc2)=O)CCCC(C2(NC(C3CCCCO3)=O)CC2)C1 49884,C(CC(C(C)C)NC(C1CCC(=O)C1)=O)NC(C(=O)NCC)=O 49885,c1(C(N(C(CC)C(=O)N2CC(NC(C)=O)C2)C)=O)cccc2cc[nH]c12 49886,C(=O)(C1=CCCCCC1)NCC1(OC)CCN(C(CSCCCC)=O)C1 49887,C(=O)(CC(CC=C)NC(c1ccnc(O)c1F)=O)NC(C#C)CC1CCC1 49888,C(=O)(C(F)(F)C(O)C1CC1)N1CCC(CN(C)C(C2COC(C)(C)CO2)=O)CC1 49889,c1(OC)cccc(NC(=O)COCCNC(c2csc(C(F)F)c2)=O)c1C 49890,c1(CC(=O)NC(CC)CN(C(C2CC2F)=O)CC)ccc2scc(C)c2c1 49891,c1(C(=O)NC2C(C)CN(C(C34C(=O)C5CC3C4C5)=O)CC2)cc2ccccn2c1 49892,c1(C(=O)NCC(COC)NC(=O)C(OC)OC)cccnc1-n1ccnc1 49893,C1(NC(CCOCCC)=O)CC(C2CCN(C(c3cc(O)nc(C)n3)=O)C2)C1 49894,c1(C(=O)OC)[nH]c(=NCC23CCC(C)(CC2)CO3)sc1Cl 49895,C(C(F)(F)C(F)(F)F)n1ncc(CN2CCC(N(C(CCC#C)=O)C3CC3)C2)c1 49896,c1(C(=O)NCCCCCCNC(=O)CC2CC(=O)NC2=O)cnc2[nH]cncc1-2 49897,c1(NCC(CCCC)NC(C2(C)CCCCN2)=O)cnc(C#N)c(C#N)n1 49898,CCCC(CC)C(=O)NCC(C)CN(C)C(c1cc(F)ccc1NC(C)=O)=O 49899,C1(CNC(C2(C)C=CCCC2)=O)CCN(C(=O)CCCS(N)(=O)=O)CC1C1CC1 49900,c1(OC)ccc(C(=O)NC(C)(CNC(=O)C(C)CO)CC(C)C)cc1C 49901,N1(CC)CCCC1CC(=O)NCC#CCNC(=O)CCOCC1CC1 49902,C1(OC)(OC)C(C(=O)NCC2(C)CCCN2C(C)=O)CC1(F)F 49903,c1(SCC)ccccc1NC(=O)CC1CCCC1.c12ccc(cn1)s2 49904,Cc1cncc(C(=O)N(C2CCCN(CC=Cc3ccccc3)C2)C)c1Cl 49905,S(=O)(=O)(c1c(Cl)ccc2c1OCCO2)Nc1ncnc2sc(C)c(C)c21 49906,c1(C(=O)OC2CC(C)C(F)N(C(=O)OC(C)(C)C)C2)ccc(N)cc1S(N)(=O)=O 49907,Cc1nc2c(C#N)cnn2c(C)c1CCC(=O)N=c1ccn(C)[nH]1 49908,C1(NC(C2CCN(CC)C2)=O)CCC12CN(C(=O)Cn1cc(C(F)(F)F)nn1)C2 49909,C1(C(=O)NCC(CC)NC(c2sc(C3CC3)nc2C)=O)CC(=O)N(CC2CC2)C1 49910,C(CC(C)C)(C(=O)NCCNC(c1cscn1)=O)NC(CNC(=O)OC)=O 49911,CCCC(CCC)CC(=O)NC1(C)CN(C(c2cc[nH]c2C2CCC2)=O)C1 49912,c1(C(=O)NC(CC=C)CNC(=O)Cc2ccsc2C)cc2c(O)ncnc2cn1 49913,c1(C(C)C)nc(-c2ccc(C(F)F)cn2)n(CC2CCOC2)n1 49914,C1(Nc2c(C(=O)OC)c(Cl)ncn2)CC1C1CCCN(C(=O)C2=NOCC2)C1 49915,c1(N2Cc3c(nc(COC)s3)CC2)nc(=NC(C)CC(N)=O)[nH]c2c1CCCCC2 49916,CC1(C)CCCC(O)(C(=O)NC2CCCCN(C(=O)CC3CC=CCC3)C2)C1 49917,CCCCC(O)C(=O)NC(CNC(C1CCCSC1)=O)C(C)C 49918,Cc1cc(C(=O)NC2CC2CNC(c2cc(Cl)c(Cl)s2)=O)c2nccn2c1 49919,C1(NC(C(C(C)O)N(C)C)=O)CCN(C(=O)CC2CC(C(C)(C)C)C2)CC1O 49920,c1(OC)cc(Cl)ccc1CC(=O)N(C(C)CN(C)C(C1CC2CCC1CC2)=O)C 49921,CC1(C(N2CCC(COC3CCN(C(c4cscn4)=O)C3)CC2)=O)CCCCC1 49922,c1(NC(C2CCCN2C(c2ccc(F)cc2)=O)=O)c(F)ccc(CO)c1F 49923,c1(-c2onc(Cc3c(OC)cc(C#N)cc3)n2)cc(Cl)cc(Br)c1F 49924,C(=O)(C1=CCc2ccccc21)NCC1C(NC(=O)CC2CC3(CC3)CO2)COC1 49925,CCC(C)(C(=O)NC(C)C(CO)NC(C1CC(F)(F)CS1)=O)C(N)=O 49926,c1(C(=O)NCCn2cc(C(=O)NCC(=O)NCC(C)C)nn2)ncccc1F 49927,C(=O)(C(O)CC(C)C)N1C(C=CC(N2CC(O)(CC=C)C2)=O)CCC1 49928,C1(C(N2CCC(NC(=O)N(C)C)C2)C(=O)Nc2nc(C)sc2)CC12CCOC2 49929,c1(OC)ccc2c(C(C)NC(=O)NC(C)COCC(C)C)c[nH]c2c1 49930,C(CC(=O)NOCC1CC2C=CC1C2)C1CCN(C(c2[nH]cc(C(N)=O)c2)=O)C1 49931,N1(C(c2ccc(C#C)o2)=O)CC2(CCCC2)C1C(=O)NCC1CCc2nccn21 49932,C1(CNC(=O)C=Cc2ncc[nH]2)CC(O)CN1C(=O)CC1CCC(O)CC1 49933,N1(C(c2n[nH]c(CC)c2Cl)=O)CCC2(CCC2CNC(=O)C(C)C(C)C)CC1 49934,c1(C(=O)NC2CC(CCNC(C3C(C)C3)=O)C2)sccc1S(=O)(=O)N(C)C 49935,c1(C2(C(N3C(CC(=O)OC)CCC3)=O)CCC2)ccc(C2=COCC2)cc1 49936,c1(OCC)cccc(C(=O)NC2C3CC2N(C(=O)CC(C)C2CCCO2)C3)c1 49937,c1(C(=O)NC(C2(O)CCN(C(C(=O)NCC)=O)C2)C)ccc2ncn(C)c2n1 49938,N(C(=NCC1CCCSCC1)NC1CCN(CC(F)(F)F)C1)C(CC)CC 49939,CON=C(C(=O)N1CCCC(CO)(NC(=O)C(C)C2CC2)C1)c1ccco1 49940,C(=O)(CCS(C)=O)N1CC(N(C(=O)CCC2CC2(C)C)C)C1 49941,CCCC(CCCNC(C1(C)CCNC(=O)C1)=O)NC(C1CN(C(C)=O)C1)=O 49942,N1(C(CC2CC(SC)C2)=O)CC(NC(C2(C)CCCOC2)=O)CC(C)C1 49943,N1(C(C=C(C)Cl)=O)CC2CC(NC(C3(CCN(C)C)CCCC3)=O)CC2C1 49944,Cc1cccc(Br)c1C(C(N1CCC(CO)CC1)=O)NC(c1cnn(C)c(=O)c1)=O 49945,c1(C(=O)NC(C)CCCCNC(c2cnc(C#N)s2)=O)cccc2nccnc12 49946,C(=O)(C(C)C(C)S(C)(=O)=O)N(CCNC(C(F)=CC)=O)CCC 49947,CC(C)C(C(=O)N1CCC(C)(C)CC1C(N1CCCC1CF)=O)C(C)C 49948,c1(CN(C)C)ccc(C(=O)NCC2CC(F)CN2C(=O)CSc2cccs2)cn1 49949,c1(C(=O)NCC2N(C(C3CC(=C)C3)=O)CCOC2)c[nH]c2cc(OC)ccc12 49950,C1(N(C(C(CC)n2cccn2)=O)CCF)CCCN(C(=O)C=CC(C)(C)SC)C1 49951,CC1(C(=O)NCC2CC3CCC2N3C(C2(CO)CCC2)=O)CCCNS1(=O)=O 49952,C1(NC(c2cc(Cl)cnn2)=O)CCN(C(c2ccc(Cl)cn2)=O)CC1O 49953,N1(C(c2scc(C)c2)=O)CC2CC2(NC(c2ccnc(C3CC3)n2)=O)C1 49954,C1(C)(CNC(c2c(CC)c[nH]n2)=O)COCCN(C(C2CC2CC)=O)C1 49955,C1(OC)CC(C(N2CC=CC(O)C2)=O)N(C(c2sccc2Cl)=O)C1 49956,Cc1cccnc1CC(=O)NC1CC(C)N(C(=O)CN2CCOCC2)C1 49957,N1(C(C2N(C(C(N)=O)=O)CC2)=O)CCOC2CC12 49958,C1(CC)C(NC(=O)CCOc2cccc(F)c2)CCN1C(=O)C(CO)N(C)C 49959,c1(CC)ncc(C(N2CCN(C(=O)CCn3cccn3)C(CC)C2)=O)c(O)n1 49960,C(=O)(C1=NOC(CNC(=O)CC2NC(=O)NC2=O)C1)N1CC(C(=O)NCC)C1 49961,c1(OC)nn(C)cc1C(N1CC(C(=O)NC2CCN(CCCO)C2)C(CO)C1)=O 49962,c1(C(N(CC(C)NC(C2CCCN2Cc2nnn(C)n2)=O)C)=O)ccc(Cl)cc1 49963,Cc1cc(C(=O)NC2CC(F)(F)CC2NC(=O)C2=CCOCC2)cc(Cl)c1 49964,N1(C(C(C)OCCC=C)=O)CC2CC1(CNC(C1CC(C)=NO1)=O)C2 49965,c1(C(C)C)cc(C(N2CC3(C2)CN(C(C2OC4CCC2C4)=O)C3)=O)nc2ncnn12 49966,N1(C(C(F)=CC)=O)CCC2CN(C(c3sc(C)cc3Cl)=O)CCC12 49967,CCC(C)(C(=O)NC1CC1NC(c1nc(=O)n(C)[nH]1)=O)OC 49968,N1(CCC2N(C)CCC2)CC(=O)N(CC2(n3ccnn3)CC2)C1=O 49969,c1(C(N2CC(O)(CNC(C3C(OC)C3)=O)C2)=O)ccc(Br)cc1O 49970,Fc1cccc(CN=C(NCC2CCN2C2CCOCC2)NCC(F)F)c1F 49971,c1(C(N2CCC3CCN(C(CC(C)(C)O)=O)CC32)=O)c[nH]c2ccccc2c1=O 49972,Cc1ccc(CCC(=O)N(CCCCNC(=O)CC2CCCC(C)C2)C)cc1 49973,c1(CC)nc(=NCC(C2CCCCC2)C(=O)NC2(C3CCC3)CC2)s[nH]1 49974,C1(C(N2CC(C)(NC(=O)Cc3cnn(C4CC4)c3)C2)=O)CC2(CCCC2)CO1 49975,c1(OCC=C)ccc(Cl)nc1C(=O)NC1CCC1NC(=O)C(C)c1ccco1 49976,c1(C(N2CCCC(CN(C(=O)C(O)c3ccco3)C)C2)=O)cc(F)ncc1Br 49977,N1(C(C23CCC(OCC)(CC2)C3)=O)CCSC(C)(C)C1CN(C)C 49978,C1(CN2CC(C(F)F)NCC2)CCOC12CCC2 49979,C(C1CN(C(C2CC3(CC3)C2)=O)CC1C(N1CCOC(C2(C)CC2)C1)=O)=CC 49980,N1(C(C2N(C(N)=O)CCCC2)=O)CCC(NC(C2(O)CCC2)=O)C(F)C1 49981,C(CCN(C)C(c1ccc(CC)s1)=O)(C(C)C)NC(c1cc(CCC)[nH]n1)=O 49982,N1(C(C23CC(C#N)(C2)C3)=O)CCC2(CCN(C(=O)C=Cc3cncs3)CC2)C1 49983,CCCS(=O)(=O)C(C)C(=O)NC1CN(C(c2cc(C)ncc2C)=O)C2(CCC2)C1 49984,c1(CC)ccc(C(C)CC(=O)NCC(O)CN(C(=O)Cc2cc[nH]n2)C)cc1 49985,C1(C(=O)NCC2(C)N(C(c3ncc(NC)nc3)=O)CCC2)C2CCCCCC12 49986,C12(C(=O)OC)CC(CNC(c3ccn(C)c3C)=O)(C1)OC2C.C12(CO)CN(C1)C2=O 49987,Cc1ccc(C(=O)NCC(C)(C2CC2)NC(=O)COCP(C)(C)=O)c(C)c1 49988,c1(-c2ccc(CN(C(c3c(CCC)nccc3)=O)C)cc2)cc(OC)cc(O)c1 49989,c1(NCC(C)(C)N(C)C)cc(Br)ccc1S(=O)(=O)NCC1CCOC(C(C)C)C1 49990,C1(C(=O)Nc2c(NCCC)ccc(Cl)c2)CC2(C)CCCN2S1(=O)=O 49991,C(CCCC(=O)N1CC2CC2(CNC(=O)CNC(c2ccc(Cl)cc2)=O)C1)OC 49992,c1(C(N(C2C(N(C)C(C3CC3F)=O)CCCC2)C)=O)cnc2ccnn2c1 49993,N1(C(CSCCCC)=O)CCC12CN(C(=O)CCC(C)(C)F)C2 49994,C1(NC(c2cn(C)nc2O)=O)COC2(C1)CN(C(=O)Cc1cc(F)cc(Cl)c1)C2 49995,C(CCCCC(=O)NC1CCC1O)N(C(=O)Cc1cncnc1)C 49996,N1(C(CN(c2ccncc2)C)=O)CCCCCC1CNC(c1ccccc1F)=O 49997,CC1=C(C(=O)NC2COC3(C2)CN(C(c2scnc2C2CC2)=O)C3)CCS1(=O)=O 49998,c1(NC(CN(C(=O)C(F)OC(F)(F)F)C(CC)C)=O)cc(C)cc2c1NCCC2 49999,CC1CC(NC(c2c[nH]c(C(N)=O)c2)=O)CCN1C(=O)CC1(C)CC1 50000,C(=O)(CCCCCc1cn(C(C)C)nn1)OCC1C(C)C1 50001,CC(C(=O)NN1CCCC1C(=O)NCCCN1CC=CCC1)C1CCC1 50002,Cc1nccc(C(=O)NC23CC2CN(C(=O)C#CC2CC2)C3)c1C 50003,CCCCCC(O)C(=O)N1CCCC(CCNC(C2(OC)CCSCC2)=O)C1 50004,C(C(CCOC)NC(=O)CC1CCCC1)NC(COCCC=C)=O 50005,N12CCCC1C2=O.N1(C(C2(C(=O)OC)CC2CO)=O)CCC(N2CCCCC2)C1 50006,C#Cc1ccc(C(N2CCC(NC(C3(F)CCOC3)=O)C(O)C2)=O)c(F)c1 50007,C#CC1CCC(C(=O)NC(C)CNC(C2(OC)CCCCC2)=O)CC1 50008,CC(C)C(C)(CNC(c1ccc(C(O)CF)cc1)=O)NC(=O)CSc1nc[nH]n1 50009,c1(C(C)(C)C)cccc(COc2cnc(C3CN(C(=O)OC(C)(C)C)C3)o2)c1 50010,n1(CC)nnc(C(=O)NCCC2(C)CCN(C(C3CCS(=O)(=O)N3)=O)C2)c1C 50011,C1(NC(CSc2n(C)ccn2)=O)CC2CCC1N2C(c1coc(C(C)(C)C)n1)=O 50012,n1(CC(=O)NCC2(NC(C(C)OCC3CCCO3)=O)CCOC2)ncccc1=O 50013,CON1CCC(CC(=O)NC2CCN(C(C3(OC)CCCCCC3)=O)C2C)CC1 50014,C(CC(=O)NCC1CC[Si](C)(C)C1)(CC(C)C)NC(C(C)OCC)=O 50015,Cn1cnc2ncnc(Nc3cc(-c4ccc([N+](=O)[O-])nc4)ccn3)c12 50016,C(=O)(CCCS(C)(=O)=O)N(C1(CNC(=O)CC(C)(C)C(F)F)CC2CCC1C2)C 50017,c1(C(=O)NC2CC(NC(C34C(C(=O)OC)(CCC3)C4)=O)C2)ccn2nnnc2c1 50018,c1(C(C(=O)N(C2(C(=O)OCC)CC2)C)NC(N)=O)ccccc1 50019,CC1CCC(CO)CN1C(=O)C(CCCc1ccccc1)N1CCNCC12CC2 50020,C1(C(CNC(C(C2CCCO2)OC)=O)=O)CC=CCC1 50021,c1(CC(=O)NC(C2CN(C(c3ccccn3)=O)C2)C)ccc2c(c1)COCC2 50022,Cc1ccc(C(N2CC(F)(F)CC2C(=O)NCCC(C)C)=O)c(O)c1 50023,C1(C(c2n(C(CC)(C)C)nnn2)(C)NCCc2ccncc2)CC2CCC1O2 50024,N1(CC)CCC1C(=O)NC(CNC(C1(C2CC2)CC1)=O)C1CC1.C1CC1 50025,N1(C(CC(c2ccc(C)cc2)C)=O)CC(CNC(=O)C2=CCOCC2)C(C)(C)C1 50026,CC1(C)CC(NC(C2C(C(F)F)C2(C)C)=O)CN1C(c1ccc(Cl)cc1N)=O 50027,Brc1cc(NCc2csc3c2CCNC3)c2c(c1)OCO2 50028,c1(OC)ccc(CC(N2CCNC(C(=O)Nc3c(Br)ccnc3C)C2)=O)cc1Cl 50029,N1(C(C2CC(=O)NC2)=O)CCCC(C2CCN(C(=O)CCc3ccc[nH]3)C2)C1 50030,C1(C(C)NC(=O)CC2(C)CCCC2)CN(C(=O)CC2CC3(CCC3)C2)CCO1 50031,C1(CNC(CN(C(C)=O)C)=O)CCN(C(=O)CCc2ccncn2)CC1 50032,c1(CC)cn2c(n1)CC(C(=O)NCC1C=CCN1C(=O)CNc1nccs1)CC2 50033,N(C(=NCCC1CC1(F)F)NCC1CCC(C)CO1)C(C)C 50034,N1(C(c2c(C(C)C)occ2)=O)CCCC(C2CN(C(=O)C(C)NCCC#N)C2)C1 50035,CCCC(O)CC(=O)N(CCC(C)NC(c1occc1-c1ccc(F)cc1)=O)C 50036,N1(C(C2(CC)CCCCO2)=O)CCN(C(=O)CCc2cncnc2)CC(CO)C1 50037,N1(C(CCc2cncc(C)c2)=O)CCN(C(=O)Cc2ccc(C)nc2)CC(O)C1 50038,C1(CNC(C=Cc2ccc(C)o2)=O)CN(C(c2cnn(CCF)c2)=O)CCN1C 50039,N1(Cc2cccc(OC(F)F)n2)CC2CC3CCCN3C2C1 50040,C12(NC(=O)Cc3cc[nH]n3)CCCC1CN(C(c1c(F)cncc1Cl)=O)C2 50041,Cc1cn2ccnc(C(=O)NCCCC3CCN(C(c4cc[nH]n4)=O)CC3)c2n1 50042,c1(C(=O)OCCOC)ccc(CCN(C)C)cc1.C1(C(=O)CN)CCCC1(OC)OC 50043,C1(CNC(c2ccnn2CCF)=O)CC(O)CN1C(=O)Cc1ccn(C(F)F)n1 50044,C1(C)(C(=O)OC)CC(F)(F)CN1C(=O)CC1CNCC(C)(C)O1 50045,C1(C(N2C(C)(C(=O)NC(CC)C(C)CN(C)C)CCC2)=O)CCC(F)(F)CC1 50046,c1(NC(C2(F)CN(C(C3CC(O)C3)=O)C2)=O)c(Br)cccc1[N+](=O)[O-] 50047,c1(OCOC)ccc(C(=O)NC(C)(C)CNC(C2CCCC23CC3)=O)cc1 50048,Cc1nsc(C(=O)N(CCCN(C(=O)C(C)Cn2ccnc2)C)C)c1N 50049,CC(C)(C#N)CCC(=O)N1CCSCC1C(N1CCS(=O)(=O)CC1)=O 50050,c1(CC)cnccc1C(=O)NCC1CCN(C(C2C=CCC2)=O)C1 50051,CC(C(=O)NCC1C=CCN1C(=O)C=Cc1cn(C)nn1)C(F)(F)C(F)F 50052,C(C(C)(C)SC)(c1nnnn1CCCC(=O)OCC1CC(OC)C1)NCC 50053,C1(NC(c2cccc(SCC)c2)=O)CCN(C(=O)C(C)S(N)(=O)=O)CCC1(F)F 50054,c1(CC(=O)NC(C(C)C)CNC(c2ncsc2C2CC2)=O)ccc(Br)cn1 50055,C(C(O)C(=O)NC1(CN2CC(C(=O)NCC3CCCCC3)C2)CCOC1)OC 50056,Cc1nn(CC(=O)N(CC(C)NC(c2n[nH]cc2C(F)(F)F)=O)C)cc1Cl 50057,C12(C(N(C3CCN(C(C(C(C)C)F)=O)C3)C)=O)C3CC(CC13)C2(F)F 50058,c1(CN=C(NC(c2ccc(OC)cc2)C)NC(C)C2CC2)cn(C)c(=O)nc1O 50059,CC1(C)OCC(CCN=C(NCC2CCCO2)NC2CC=CC2)CO1 50060,C(CS(=O)(=O)NC(=O)CC1CC1C1CCCC1)OC 50061,C(=O)(CCCS(N)(=O)=O)N1CC(N(C(=O)C(c2ccccc2)O)C)C(O)C1 50062,C1(C(=O)NC2CCCC(NC(c3c(C)cc(F)s3)=O)C2)CC2C(C1)C2(F)F 50063,N1(C(c2c(OC)cccn2)=O)CC2(NC(=O)Cc3ccc(F)cn3)CCC1CC2 50064,CCCC(C)(CCC)C(=O)NCCCCCN(C(=O)C=Cc1ccccc1)C 50065,N1(C(C=C(C)Cl)=O)CC2CCC1(CNC(=O)C(c1ccc(F)c(F)c1)O)CC2 50066,c1(CCC(=O)N(CCN(C(COCCC#C)=O)CC)CC)ccccc1Cl 50067,C1(CN(C(=O)CN(C)C)C)CC(F)CN1C(=O)CNC(=O)CCn1ccnc1 50068,c1(OC)noc(C)c1C(=O)NC1COCCC1NC(C1CC12CCC2)=O 50069,CCC(C(=O)NC1CCCC1NC(C1(OC)CC1)=O)SC 50070,C1(C(N(CCCNC(C2(C)CCN(C)C2=O)=O)CC)=O)COCCN1C=O 50071,C(C(CC(=O)N1CC2=C(C1)CN(C(C1C3C4CCC(C4)C13)=O)C2)C(F)(F)F)OC 50072,S(=O)(=O)(c1cccc(=NCC(O)c2ccccc2C)[nH]1)N1CC(CCC)OCC1 50073,C1(CNC(CSCCCC)=O)N(C(=O)C(C)C(=O)OC)CCCC1(C)C 50074,CC(CC(=O)NCC1CC1CNC(c1ccc2c(n1)CCCN2)=O)CC(C)(C)C 50075,CC(C)CCC(C(=O)NCC(CO)C(C)C)NC(=O)CCN(C)CCO 50076,c1(C(=O)NC(CNC(c2c(C)ccnn2)=O)C)cn2cccc(F)c2n1 50077,CCCC(CC)CC(=O)N1CC(C2CN(C(c3c(C)ccc(Cl)c3O)=O)C2)C1 50078,C(=O)(C(C)(C)Cc1ccccc1)N(CCN(c1nnc(C)s1)C)C 50079,c1(N(C(C2(CNC(=O)OC(C)(C)C)CCCC2)=O)CC)ccc(Br)cn1 50080,C(=O)(C(C)CC(F)F)N.c1(C(N2C(C(C)O)CCC2)=O)cc(OC(F)F)ccn1 50081,C(c1ccc(Br)cc1)=CC.C(C=O)(N(CC(=O)NCCCOCCOC)C)C1CC1 50082,C#CCCC(C(=O)NCC(F)(F)Cl)NC(c1cnc(O)cc1C)=O 50083,c1(OC)cccnc1C(=O)N(C1CCN(C(C2CCOC2C2CC2)=O)CC1)C 50084,c1(C(c2n(CCOC)nnn2)NC(C2(OC)CCC2)C)c(Cl)cnc(F)c1Cl 50085,C1(C(=O)NCCOCC(C)(C)O)CC2(CC2)CN1C(=O)C=CCN(C)C 50086,N1(C(CN(C(=O)CC(O)C(C)C)CCC)=O)CCC(C)(C)C1C 50087,N1(C(C2C(C3C(C)C3)C2)=O)CC2(C1)CN(C(C1CCC(=O)N(C)C1)=O)CC2CO 50088,Cc1cnncc1C(=O)NCC(C1CCC1)NC(=O)C(C)Cc1cccc(Cl)c1 50089,C1(OC)CN(C(=O)CO)CC1NC(=O)C(C(C)C)n1cnnc1 50090,C(=O)(C(C)C(C)NC(=O)CCN1CCCC1=O)N(C)CC1C(C)OCC1 50091,n1(CCC)nnnc1C(CCC)(C1CC1)NCc1cnc(CC)s1 50092,c1(C(=O)NCCN2CCN(C(CC(C(=C)C)OCC)=O)CC2)ccc2n[nH]cc2n1 50093,CCC(C)C(O)C(C)C(=O)NC1(C(N2CCCC(CC(N)=O)C2)=O)CC(F)(F)C1 50094,C1(CCNC(C2CN(C(N)=O)C2)=O)CN(C(c2nnsc2C(F)F)=O)CCO1 50095,N1(C(=O)C(c2cccc(Cl)c2)O)CCCC(NC(C2CC(C(F)F)C2)=O)CC1 50096,c1(CC(=O)NCCCN(C)C(C2(c3nc[nH]n3)CC2)=O)cnsc1 50097,CC1CC(NC(=O)C(C)(C)CC2CC2)CN(C(=O)Cc2cncn2C2CC2)C1 50098,C1(NC(C(c2cnn(C)c2)OC)=O)CC12CC(NC(=O)CCCC1CCCC1)C2 50099,CC1=C(C=O)CCCO1.C12(C(=O)NCC3(F)CNC3)CCC(CO)(CC1)CO2 50100,C=CCC(C)(C)C(=O)NCC1CN(C(c2cscc2C(N)=O)=O)CCC1C 50101,Cc1ccc2c(c1)C(C(=O)N1CCCC(NC(C3(C)CSC3)=O)CC1)OCC2 50102,C1(NC(CCOCC)=O)COC2(CCN(C(c3ncsc3NCC)=O)C2)C1 50103,C1(N(C(C(CCCC)N(C)C)=O)C)CC2CCC(C1)N2C(c1ocnc1C)=O 50104,c1(C(=O)NCC2CCC2NC(C2CCC2(F)F)=O)cncc(N2CCCC2=O)c1 50105,Cc1c(C(=O)NC(CNC(C2CCS(=O)CC2)=O)C2CCC2)c[nH]c2nccc1-2 50106,N1(C(C2CN(C)C(=O)N2)=O)CCN(C(=O)CCCC2CCOCC2)CC(O)C1 50107,N1(CC(=O)NC(C2CCCN2C(c2c(Cl)cnn2C)=O)C)CCN(C)C(=O)C1 50108,[N-]=[N+]=NCC(C(=O)NCCN1CCC(CO)C1)NC(c1nnsc1N)=O 50109,C1(NC(C2(CC#C)CC2)=O)CCC2CCN(C(=O)C(c3ccc(C)cc3)C)C12 50110,C1(NC(Cc2n(CC)cnc2)=O)CCCC(N)CC1 50111,N1(C(Cc2c(C)occ2)=O)CC(NC(=O)C(c2cccc(F)c2)C)C(C)C1 50112,c1(OC)cc(C)cc(CN2CC3C(C(=O)NC4CCCCCC4C)C3C2)c1O 50113,C(CCC(C)(F)F)N(C)C(C1CCCN(C(=O)CSCCC#N)C1)=O 50114,N1(C(C(CC)n2cncn2)=O)CC(NC(=O)CC2CCCN2CC)C2CCCC12 50115,N1(C(CC(C)(C)O)=O)CCC2(CCN(c3ccnc(C4CC4)n3)C2)C1 50116,c1(OC)ccc2[nH]c(CN3CCC(O)CC3C(=O)Nc3csc(C)n3)cc2n1 50117,c1(C(N2C(C)C(NC(=O)CCCC(F)F)CCC2)=O)cnc([N+](=O)[O-])n1C 50118,CC1CN(C(=O)CO)CC(C)N(C(c2cc(Cl)cc(Br)c2F)=O)C1 50119,C=CCC(C)C(=O)N1CCC(CCC(N2CCC(CCC)CC2)=O)C1 50120,C1(C(N2CC(OC)C(NC(=O)CC34COCC(C3)C4)C2)=O)CC2(CCCO2)C1 50121,Cc1cc2ccccc2n1CC(=O)NC1(C)CCN(C(C2(C)CC2C)=O)C1 50122,Nc1cc(C(=O)NCC2CCCN2C(c2cnccc2C(F)F)=O)cc(F)c1O 50123,S(=O)(=O)(c1cccc(=NCc2cnc(N3CCCC3)nc2)[nH]1)NC(C(CC)(C)C)C 50124,N1(C(CSC)=O)CCc2nc(CNC(C3(C)CC3(F)Cl)=O)sc2C1 50125,CC1CCN(C(=O)Nc2ccc(Cl)c(-n3nnnc3C)c2)CCN1C(=O)C(F)F 50126,c1(OCC)c(C(N2CC(C)(NC(c3c(C)cccc3Br)=O)C2)=O)cccc1F 50127,S(=O)(=O)(c1ccccc1Cl)NCC(=O)N(C1CC(NC(c2occ(C)c2)=O)C1)C 50128,c1(NC(CCC)CC)[nH]c(=NC2CSCCC2C)nc2c1ncn2CC 50129,N1(C(c2cncc(NC)c2)=O)CCC2C(NC(C34CCCC3C4)=O)CC12 50130,C1(C(=O)NC(C(=O)NCC(C(C)O)O)(C)C2CCC2)C(C#N)C1(C)C 50131,c1(NC2CCN(C3CCN(C(c4n(CC)nnn4)OC)C3=O)C2)cnn(C)c1Cl 50132,C1(C(=O)NC2CC(C)(NC(C(CC)Sc3ccccc3)=O)C2)CC(F)CN1C 50133,C1(C(=O)NC(C2CCCC2O)C)CCCC1CNC(c1cc[nH]n1)=O 50134,c1(N(C(N(C2CCC2)C)=O)Cc2ccc(F)cc2F)ncnc2[nH]cnc12 50135,c1(CC)ccsc1C(=O)NC(C1CCN(C(C2(c3cccs3)CCCC2)=O)C1)C 50136,Cc1nc2ccnn2cc1C(N1CC(O)(CNC(C2CC2(C)Br)=O)C1)=O 50137,N1(C(C(C)C2CCC2)=O)CCC(CO)(CNC(c2ccnc(Cl)c2N)=O)CC1 50138,C1(CN(CCNC(c2ccoc2-c2cnn(CC)c2)=O)CC)CC12CC2(F)F 50139,CCCC(C)C(=O)N1CCC(N(C(=O)CC=C(Cl)Cl)C)CC1 50140,N1(C(C(c2cccc(OC)c2)(F)F)=O)CCC2(CC(NC(c3ccsn3)=O)C2)C1 50141,C1(C#N)(CNC(=O)NC(Cc2nc(C)[nH]n2)C)CCCC1 50142,CC1CCCCN1C(C1CC(NC(c2cc(Cl)cs2)=O)C(O)C1)=O 50143,C1(NC(CCC(CC)NC(=O)CCCn2ccnc2)=O)CCC(=O)N(C)C1=O 50144,c1(C(N(CC(C)(C)NC(=O)C2=NOCC2)C)=O)cc(F)cc2nc(S)[nH]c12 50145,C(C(CC)CCO)NC(CCN(CC#C)C(c1cnc(Cl)s1)=O)=O 50146,N1(C(CCCC#CC)=O)CC2(C1)CN(C(c1cc(C)c(Cl)s1)=O)CC2CO 50147,Cc1cc(C(c2nnnn2C2CC2)NCC(C)(C)C(N)=O)cc(C)n1 50148,C1(c2nnnn2CCN2CCOCC2)(NCc2ncc(C)o2)CC(C)SC(C)C1 50149,C1(NC(c2ccc(C#N)o2)=O)CC(C(=O)NCC2CCCC2O)C12CCC2 50150,CCCCC(C(=O)NCC(C)N(C)C(c1nc(C(F)(F)F)cs1)=O)C(C)C 50151,N1(C(c2cc(Cl)c3n[nH]cc3c2)=O)CCC2(CCN(C(C3CC3(Cl)Cl)=O)CC2)C1 50152,C(=O)(CC1=CCN(C(=O)CC2CCCCC2C)CC1)NCC1(C#C)CCCC1 50153,CC#CCC(C(=O)NC1CCC12CCCC2)NC(c1ccc(OC)nn1)=O 50154,C(=O)(C(C)C(=O)NCCOCCCNC(C1CNC(=O)C1)=O)OC 50155,C1(N(C(C23CCC(OC)C2C3)=O)C)CN(C(C2CC3(CCOC3)C2)=O)CCC1O 50156,S1(=O)(=O)c2ccc(cc2)CNC(=S)N1.c1(COCC)cnn(Cc2ccccc2)c1 50157,N1(C(C23CC(COC)(OC2)C3)=O)CCCC(NC(C2ON=C(C)C2C)=O)CC1 50158,C1(CC=C)(NC(=O)C2=CCC2)CCN(C(c2ccc(CCC)cc2)=O)CC1 50159,c1(C(=O)OCC)nc(C(=O)NCCN(C(C2COCCO2)=O)CC2CC2)cs1 50160,C(=O)(CCCC(C)(C)NC(c1cnn(CCF)c1)=O)NCC1N(C)CC(O)C1 50161,N1(C(C(COCC)C)=O)CC2CCC(C1)N2C(c1cccc(F)c1O)=O 50162,Cc1nc(C(C)(C)C)sc1C(N1CC(NC(=O)C2=CCC2)CC1CO)=O 50163,c1(C(N(CC(C)N(C(CN(CCC)C)=O)C)C)=O)sc(Cl)c(Cl)c1C 50164,c1(CC(=O)NCCC2(NC(c3cn(C(C)C)nn3)=O)CC2)ccc(F)cc1 50165,C1(C(C)NC(=O)CCN(CC(F)(F)F)C)CCCN1C(=O)CC1(C)CCCO1 50166,N1(C(C2(C(C)(F)F)CCC2)=O)CC(NC(=O)CC2OCCC2(C)C)CC(F)C1 50167,C1(C(=O)NCc2cncnc2)(COC)CCN(C(=O)C(CO)NC(N)=O)C1 50168,CC1=C(C(=O)N2CCC(C(C)C(=O)NCc3cnsc3)C2)CCC1 50169,C1(NC(C=CC(C)C)=O)CN(C(=O)CSC(C)C)CC1C(F)(F)F 50170,C(=O)(C(C)CCCOC)NC(C(=O)Nc1cn(CCC)nc1)(C)C 50171,Cc1c(Cl)c(Cn2cc(C(N)CCC(N)=O)nn2)nc2ccccc12 50172,CCCC(C)CCCC(=O)N1CCCC1C1CCN(C(c2ccc(C)nc2)=O)C1 50173,c1(OC)c(C(N2CCC(N(C)C(c3csc(SC)n3)=O)C2)=O)cccc1F 50174,c1(OCC)cccc(C(c2nnnn2C(C)C)Nc2cc(CC)on2)c1C 50175,c1(C(=O)NCC2CC(C)N(C(c3cscc3C(F)(F)F)=O)C2)ccnc(C#N)c1 50176,C1(C(C)NC(=O)C(F)n2cccn2)CCCCN1C(c1ccc(CO)cc1)=O 50177,N1(C(C2CCC(C)(C)O2)=O)CCC2CN(C(=O)CCCC#N)CC2CC1 50178,N1(C(C2=CN=C2C(F)F)=O)CCN(C(c2cc(C3CC3)sn2)=O)C(C2CC2)C1 50179,C(=O)(C1(N2CCCC(O)(C3CC3)C2)CCc2c(OC)cccc21)OC 50180,C(CCC(C)C(C(=O)NCC1CCCCO1)N(C)Cc1ccc(Cl)cc1)=C(C)C 50181,CC(COC(c1nnn(C(F)F)c1C(F)(F)F)=O)CC(F)F 50182,c1(NC(C(C)CSC(F)(F)F)=O)cccc(-c2cn(CCCN(C)C)nn2)c1 50183,c1(CNC(C)=O)ccc(CC(N2CCC2C(=O)Nc2cc[nH]c(=N)c2)=O)cc1 50184,N(C(=NCCN1CC2CC2C1)NCc1ccco1)Cc1scc(C#N)n1 50185,O=C(C1=CCC(NC(c2n[nH]c(O)n2)=O)C1)NC(CC1CC1)C1CC1 50186,CCCC(F)(F)C(=O)NCC1CC1CNC(=O)CCn1cncn1 50187,C(=O)(C(C)(C)C(=O)NC1CC(NC(=O)C(C(C)C)n2cc(Br)cn2)C1)OC 50188,N1(CC2C(C)CCO2)CC(=O)N(Cc2cnn(CC(F)(F)F)c2)C1 50189,C12(NC(CCCOC(C)=O)=O)CCC(CC1)N(C(C)=O)C2 50190,c1(C(N(C2CCCN(C(=O)CCc3cnc[nH]3)C2)CC)=O)cc(F)cnc1O 50191,C1(CNC(C(CCOC)C)=O)(NC(C2CCC(F)(F)C2)=O)Cc2ccccc2C1 50192,c1(SCC(=O)NC2(CN(C(COCCC#C)=O)C)CC2)n[nH]c(C)n1 50193,C12(NC(c3cc(CCC)[nH]n3)=O)CCC(CC1NC(=O)C(C)n1cncn1)C2 50194,c1(SCC(=O)NCC2C(NC(C(F)OC)=O)C2)nnnn1C1CC1 50195,Cn1cc(-c2ocnc2C(N2CCC(NC(=O)CC3CCC3(F)F)C2)=O)cn1 50196,C1(NC(C2CC2C(F)(F)F)=O)CCC2CCN(C(c3coc4ccccc34)=O)C12 50197,CC(CN1CCC1)CN=c1[nH]c(=NCC2(Cl)CC23CCC3)[nH]c2c1CCCCC2 50198,c1(C(N2CCC(N(C(C(C(CC)C)OC)=O)CC)C2)=O)c(F)ccc(F)c1N 50199,C(CCCCC(=O)NCC1CCN1C(=O)CCn1cnc([N+](=O)[O-])c1)NC(N)=O 50200,CC1CN(C(c2cnc(O)cc2O)=O)CC(CCNC(c2ccn(C)c2)=O)O1 50201,c1(C(=O)NCC(CC=C)NC(C2(CCC)CCNC2=O)=O)cc2cccnn2c1 50202,CC(C(=O)N1CCC(C(C)(C)C)(CNC(=O)C(CO)NC(N)=O)C1)S(N)(=O)=O 50203,CC#CCCCC(=O)NNC(=O)Nc1ccc(N2CCCCC2=O)cc1C 50204,N1(C(C(=Cc2cn[nH]c2)C)=O)CCN(C(c2csc(C(F)(F)F)n2)=O)CCC1C 50205,N1(C(C(=CC2CCCC2)C)=O)CC2OCCN(C(=O)CCS(C)=O)C2C1 50206,CCCCC(C(=O)NC1CCCCCC1C)NC(=O)C=CCN1CCCC1 50207,C(=O)(CCC(C)S(C)(=O)=O)NCC1CC(NC(CC(C)C(F)(F)F)=O)C1 50208,Cc1cc(CC(=O)NC2CC(C)(CNC(c3c(C)cccc3F)=O)C2)cc(F)c1 50209,Cc1ncc(C(N2CCCC2(C(=O)Nc2ccc(O)nc2)C(C)C)=O)c(=N)[nH]1 50210,c1(CCC)ccccc1C(=O)NC(C1CN(C(c2cc(CC(C)C)on2)=O)C1)C 50211,C(=O)(CCCCC1CC1)N(CCCC(=O)NC1(CCOC)CCOC1)C 50212,Cc1ccc2[nH]c(C(N3CC4CCC4(NC(C4(F)CCOC4)=O)C3)=O)cc2c1C 50213,N1(C(=O)CN2CCCC2CO)CC2(NC(C3CC(n4cnnc4)C3)=O)CCC1C2 50214,c1(OC(C)C)cncc(C(=O)NC2CN(C(=O)CCOCC3CCC3)CC2O)n1 50215,C1(CN(C(Cc2cc(C)no2)=O)C)CCCN(C(c2occc2Cl)=O)C1 50216,C=Cn1nncc1C(=O)Nc1cccc(NC(=O)CC(O)c2ccccc2)c1 50217,C(C(N=[N+]=[N-])C(=O)N1CC(=O)CC1C(=O)NC1(CC(N)=O)CC1)OCC 50218,N1(C(C2=CCC(NC(c3c(NC)cncc3)=O)C2)=O)CCC(C2CC2OC)CC1 50219,N1(C(C2CCC(CSCC)C2)=O)CCN(CC(C)NC(C2CC(OC)C2)=O)CC1 50220,C1(NC(=O)CC2CCC(=O)O2)(CO)CCN(C(=O)CCCn2ccnc2)CC1 50221,C1(S(C)(=O)=O)(C(=O)NCC2C(CNC(CSC)=O)C2)CCCCC1 50222,c1(C(C(=O)OCC)NC(=O)CCC(C)C2CN(C(C)=O)C2)ccc(C)cc1 50223,C(CC1=CCN(C(C2CC23CC3)=O)CC1)NC(c1n[nH]c2c1CCCC2)=O 50224,Cc1cccc2c(CCN)cn(C)c12.c1(CC2(C)COC2)nnnn1CC(F)F 50225,N1(CC)Cc2ccc(NC(=O)NC(CNc3ccccc3)C(C)(C)C)cc2C1=O 50226,N1(C(=O)OC(C)(C)C)CCC2(CCCCN(C(C3CCC4(CCC4)C3)=O)C2)C1 50227,Cn1nc(C(N2CC3CC3(CNC(=O)CN3CCC(C(N)=O)CC3)C2)=O)cc1O 50228,C(=O)(C1c2c[nH]nc2CCC1C)N1CC2N(Cc3cc(C)on3)C(CC2)C1 50229,C1(=O)CCC(C)(C)N1CC(=O)N(C1CN(C)C1)C.C1(C)(N(C)C)CCCC1 50230,c1(CNC(CCOC2CCN(C)CC2)=O)ccc(Br)cc1F 50231,C1(NC(CCC(=C)Cl)=O)CN(C(=O)C(CC(=C)C)NC(C)=O)CC1(C)C 50232,S(=O)(=O)(c1cc(C(=O)OC)c(C)c(Cl)c1)N1CCN(CCCOCC)CC1 50233,C(=O)(CS(=O)(=O)N1CCN(CCCNC(C2(C)CC2F)=O)CC1)OCC 50234,N1(C(c2ccnc(C)n2)=O)CCC(C)CC1CNC(=O)CCOC(C)CC(C)C 50235,C1(C)(CNC(C)=O)CCN(c2nnnn2CC2COC(C)(C)O2)CC1 50236,CN1CC(C(N2CC(O)(C(F)C(=O)NCC3CC(O)C(O)C3)C2)=O)CCC1=O 50237,c1(CCC(=O)NC23CC(NC(=O)C(O)C4CC4)(C2)C3)cccc(O)n1 50238,c1(NC(C(N2C(c3c(C)noc3C)CCC2)C)=O)c(C)nn(C)c1C 50239,C(=O)(CC(O)CC(C)(C)C)N(C(CC(C)C)C(=O)NCC1(F)CCN(C)C1)C 50240,c1(SCC(=O)NC2CC(C)N(C(=O)CCSC3CC3)C2)ccc(F)c(F)c1 50241,c1(C(N2CC(OCCNC(=O)CSc3nc[nH]n3)C2)=O)cc(C(F)F)cc(F)c1 50242,N1(C(c2cc(C3CC3)[nH]n2)C(=O)NC)CCN(C2CCOCC2)CC1 50243,c1(OC)cccc(C(=O)NCCC2CN(C(c3cnc(Cl)s3)=O)CCO2)c1OC 50244,CS(=O)(=O)c1ccccc1CN1CC2C(C1C(N1CCCC1CO)=O)C2(C)C 50245,C(=O)(C1CCc2cc(Cl)ccc21)N1CC(NC(c2nc(C)n(C)c2)=O)C(F)C1 50246,c1(C(=O)NCC2CN(C(C(CC=C)NC(C)=O)=O)C2)cc2nc(OC)ccc2[nH]1 50247,C1(NC(C2N(C(C)=O)CCC2)=O)CC(NCC2CCC3(CC2)CC3)C12CCC2 50248,C1(CNC(c2ccc(Cl)o2)c2nnnn2CC2CCCO2)CCCCCC1 50249,c1(C(N2CCC(NC(c3cc(CCCO)on3)=O)C2)=O)ccc2c(n1)CCCC2 50250,c1(CNC(=O)Cn2cnc(C(F)(F)F)c2)cc[nH]c1C(=O)NC1C(OC)C1 50251,c1(CNC(Cn2c(C)ccn2)=O)cccc(NC(C2CCCCC2C)=O)c1 50252,c1(C(=O)NC2(C)CCN(C(C(C)SCC)=O)C2)cc2c(Br)c(C)ccc2[nH]1 50253,C1(N(C)C)CN(C(C2CSCCS2)=O)CC1CNC(c1csc(C(F)F)n1)=O 50254,N1(C(C(C)C)=O)CCC(C)CC1CNC(c1ccc(SCCC#N)cc1)=O 50255,C1(C(N2CCC(OC)CC2C)=O)CN(C(=O)C(C)CCOC)CCC1(C)C 50256,C1(C(N2CC3CC3(C(N3CCC(c4ncco4)C3)=O)C2)=O)CC2CC1CC2O 50257,c1(C(N(C2CCN(C(=O)NC3CCOCC3)C2)C)=O)ccc(Br)cc1OC1CC1 50258,c1(N2C3CN(C(C(C(C)C)NC(C)C)=O)C(C3)C2)ccc(Cl)cc1Cl 50259,C1(NC(C2CC(OCC)C2)=O)CCCN(C(c2cc(C)c(C)s2)=O)C1C 50260,CCCCC(C)(F)C(=O)NCC1CC(NC(=O)CC2(N(C)C)CCCC2)CCO1 50261,Cc1onc(Cl)c1C(N1CC2C(CNC(c3snc(Cl)c3Cl)=O)C2C1)=O 50262,N1(C(C)C)CC(NC(=O)CN2CCN(C(=O)Cn3ncccc3=O)CC2)CC1=O 50263,C1(NC(C=C(C)C(C)C)=O)C2CC1N(C(=O)Cn1cc(C)cn1)C2 50264,C1(CNC(CCCN(C)C(C2(C3CC3)CC(=O)C2)=O)=O)CC2CCCC2C1 50265,c1(C(N2CCCC(CCNC(C(COCC)(C)C)=O)C2)=O)cnc2scc(C)n12 50266,N(S(=O)(=O)N1CCC2(CCCC2)C1)C(C1CC(CC)OCC1)=O 50267,C1(C2CCN(C(=O)CC3=CCCC3)CC2)(NC(CC2(N(C)C)CCCC2)=O)CC1 50268,N1(C(C(C)N(C)C)=O)CCC(N(C)C(c2ncc(C(F)F)s2)=O)CC1 50269,N1(C(C(C)OC)=O)CC2(CC(NC(c3cn4cc(C)ccc4n3)=O)CO2)C1 50270,C1(C(=O)NC(C2N(C(c3n[nH]c(CC)c3Cl)=O)CCC2)(C)C)CCOC(C)(C)C1 50271,c1(COC)nc(C)c(C(=O)NCCCC2CCCN2C(=O)CN2CCC2)s1 50272,N1(C(C2N(C)C(=O)CC2)=O)CC2CCC(Nc3ncc4c(n3)CCCC4)CC2C1 50273,C1(CC(=O)Sc2ccccc2)(N(C(=O)CSC(F)(F)F)C2CC2)CCOC1 50274,C1(CNC(C(C)c2ccon2)=O)(NC(c2cc(Cl)no2)=O)CCCCC1 50275,C1(C(=O)NCC(C(C)(C)C)NC(c2c(CC)c[nH]c2)=O)CCCCC(=O)N1 50276,c1(OC)cc(CN2CC(O)CN2C)c(-c2ccc(C)c(F)c2)cc1OC 50277,CCCCC(C)(C)NC(C1(CC)CCN(C(=O)C(c2cnn(C)c2)C)C1)=O 50278,N1(C(c2c(OCC)nsc2)C(=O)NCCC2(C)CC2)CCC(C2(OC)CC2)CC1 50279,c1(OC)ccc2c(c1)C(C(=O)Nc1ccc(C(=O)NCCC(C)(C)O)cc1)CC2 50280,n1(CC)cc(C(=O)NC(C)CC(C)NC(=O)CN2CCNC(=O)C2)c(C(C)C)n1 50281,C1(OC)CCCC(C(=O)NCCCN(C2CCCC2)C(c2cn(C)c(C)n2)=O)C1 50282,C(N=c1[nH]cnc(Cl)c1F)C1C(NC(CCCn2c(C)ncc2)=O)CCCC1 50283,CCC(CC)CCC(=O)NCCC1(C)CCN(C(C2CC(OC)C(OC)C2)=O)C1 50284,C(=O)(C(F)C(=O)NC(C)(CSC)C(=O)NCC=C(C)C)OCC 50285,C(=O)(C(C)(CCC)CCC)N1CCC(=C)CC1C(=O)NCC(O)C(C)(C)C 50286,N1(C(CC#N)=O)CCC2(CC2C(=O)Nc2cc(C(F)F)no2)C1 50287,c1(C(N(C(CNC(C=COCC)=O)C)CC)=O)ccnc2ncnn12 50288,c1(OC)ncc(C(=O)N(C2CC3CC2N(C(=O)CSCC(C)C)C3)C)cc1Cl 50289,Cn1nc(Br)c2c(NCC(C)(C)NC(c3ccc(Cl)cc3F)=O)ncnc12 50290,C(=O)CCCC(C)(C)C#N.C1C(C(C)C(C)C)NC(=O)C(=CC=C(Cl)Cl)O1.CO 50291,N1(C(CCCC#C)=O)CC2CCCC1C2CNC(=O)CC=C 50292,c1(CC)ncc(CNC(=O)C(C(C)C)NC(=O)OC(C)C)c(=N)[nH]1 50293,c1(SC)ccncc1OCCNC(c1nncn1C)=O 50294,N1(C(c2cc(C#C)c(Cl)cc2)=O)CCC2(C1)CN(C(=O)CCN(C)CC)CCO2 50295,N1(C(C(C)=CC2CC2)=O)CC(C(N2CCC(CCO)C2)=O)(SC)C1 50296,Cc1cnc(NCc2csc(C)c2C)c(S(=O)(=O)NC2CC3CC(CO)CC23)c1 50297,c1(C(N(CCN(C(=O)CC(C)(C)CC)CC)CC)=O)cc([N+](=O)[O-])c(C)cc1C 50298,c1(C(=O)NC2CC(CNC(C(C(C)c3ccccc3)O)=O)C2)ccnc(F)c1O 50299,C1(C)(C(=O)NCCC(C)N2CCC2)CCCN(C(C2CCOC2(C)C)=O)C1 50300,CC(C)C(O)C(C)(C)C(=O)NC1COCC1C(N1CC(C)(CF)C1)=O 50301,c1(C(=O)OC)cccc(C(=O)NCC)c1.N1(C(C2(Cl)CC2)=O)CCOCC1CO 50302,C1(NC(CCC)=O)CC(CNC(=O)CCCOC(C)C)C1(C)C 50303,N1(C(=O)NCC(=O)OCC)C2CCC1CC(CN(C)C)C2.C12CCC(CC1)C2 50304,N1(C(C=CC(C)(C)NC(=O)Cc2cc[nH]n2)=O)CC(O)(C(N)=O)C1 50305,C1(C(=O)NC(C(C)C)CCN(C)C(C2CC2(F)F)=O)CC1C1CCCCC1 50306,C(=O)(CCCCCCN=[N+]=[N-])N1C(C)(C)CC(C)(CNC(C2CC2(C)C)=O)C1 50307,Cc1ccc(C(O)C(N2CCCC(NC(c3ccc(Cl)nc3)=O)C2)=O)cc1 50308,CC(CN(C)C)CC(=O)NCC1C2CC1N(C(=O)Cc1nc[nH]n1)C2 50309,N1(C(C(CC)(C)COC)=O)CCCCC(CNC(=O)Cc2ccc(C)cc2)CC1 50310,c1(CNC(c2c[nH]c(C(=O)NC3N(CC)CC3)c2)=O)cc(OC)c(OC)cc1OC 50311,C1(CC#C)(C(=O)NCC(O)C(F)F)CCN(C(=O)CCCC#N)C1 50312,c1(C(C(=O)NCCCOC)N(CCC(N)=O)CC2CC2)nc(C#N)cs1 50313,Cc1cc(C(=O)NC2(CC(=O)Nc3nnc(C)o3)CCC2)nc(C)c1 50314,Cc1cnc2c(NC3(c4nnnn4CCN(C)C)CCCSCC3)nccc2n1 50315,C(C)(C)(CC(F)C(=O)NC1(c2ncc(C)o2)CC1)NC(c1c(CC)nn(C)c1)=O 50316,c1(C(N2C(CN(C(c3nccc(C)c3)=O)C)COCC2)=O)cc2c(ncn2C)[nH]1 50317,c1(C(=O)NC2C3CN(C(c4ccn(C(C)(C)C)n4)=O)C2C3)n[nH]c2c1COCC2 50318,C1(NC(c2sc(C)c(O)n2)=O)CC2CC(C1)N(C(C1(C)CCCCC1)=O)C2 50319,c1(CC)nc(C(=O)NCC2C(NC(=O)Cc3cnns3)CC2O)co1 50320,c1(-n2cc(CN3CCCC(NC(c4ccno4)=O)C3)nn2)ccc2c(c1)CCO2 50321,C(=O)(C(C)(F)F)N(CC(C)N(C)C(c1ccc(CN(C)C)o1)=O)C 50322,CC1CN(C(C2CC2c2cn[nH]c2)=O)CCCN1C(c1csc(C(F)(F)F)c1)=O 50323,CC(CCCNC(c1nc(Cl)cs1)=O)NC(=O)C(C)(C)c1cscn1 50324,C1(COC)(NC(=O)C(C)n2cccc2)CN(C(=O)C(C2CCCCC2)F)C1 50325,C(C)(CSc1ccn(C)c1C)(C(C)C)NC(=O)NC1N(C(CCCC)=O)CSC1 50326,c1(OC)ccc(N)c(C(=O)N(C)CC2COCCN2C(=O)C(C)CF)c1 50327,C1(C(N2CCN(CC(=O)Nc3csc(CO)n3)CC2)=O)CC12CCCCC2 50328,CC1N(C(C2N(C(c3ccc[n+]([O-])c3)=O)CCC2(C)C)=O)CCOC1(C)C 50329,c1(C(N2CCC(N(C(C(CC(C)C)C)=O)CCO)C2)=O)nn2cccnc2c1Cl 50330,Cc1cnc(CCNC(C2CCCN2C(=O)C(C)(F)F)=O)o1 50331,c1(C(N2CCCCC3CCC23)C(=O)NCCOC)ccc(F)c2ncccc12 50332,C1(CC)CNC(=O)CN1C(=O)CC1CN(C(=O)Cc2cccc(C)c2)CC1C 50333,CC1(C)CN(C(C2CCC(=O)NC2)=O)CC1CNC(=O)Cc1ccc(O)cc1 50334,Cc1ccc(Cl)cc1C(N1CC(NC(=O)C=Cc2cn(C)cn2)CCC1C)=O 50335,C(=O)(C1SCCc2sccc21)NCCNC(C(c1c(C)nn(C)c1)C)=O 50336,CN1CCC(CC(=O)NCC(C2CCN(C(=O)C(C#N)=CC3CC3)CC2)F)C1=O 50337,C1(C)(CNC(CCN2CCC(C)CC2)=O)COCCN(C(C2CNC(=O)C2)=O)C1 50338,C(=O)(CCC(=O)NC(CNC(C1CCCN1C)=O)C1CC1)NCCCOC 50339,C(=O)(C1=COc2ccccc2O1)NCCN(C)CCNC(C12CCCCC1C2)=O 50340,c1(C2CC2)ncccn1.C(C(=O)N1CC(C(F)(F)F)C1)(C1CCCC1)NC(=O)C1CC1 50341,CC1CN(CCCN2CCCC2=O)CCN1C(c1cccnc1)=O 50342,N1(Cc2n(CC)cnc2)CC(C(N2CCC(C(=O)OC)C2)=O)C2(CC2)C1 50343,C#CC1(C(=O)NC2CC3CCCCN3C2)CCN(C(=O)CC2OCCCO2)CC1 50344,c1(CC(=O)NCCN(C(C(CC)(C)F)=O)CC(C)O)c(C)nn(C)c1C 50345,C1(CC(=O)NC2CC(NC(Cc3cn(CC)nc3)=O)C2)CCC(=O)NC1=O 50346,Cc1cc(I)c(C(N2C3CCC2CC(NC(=O)C(C)(C)CN(C)C)C3)=O)cc1C 50347,C(=O)(C(C)(C)C(=O)N1CCOCC(C(N2CCN(C)C(CO)C2)=O)C1)N(C)C 50348,N1(C(COC(C)C)=O)CCN(C(=O)Cc2cncnc2)C(CS(C)(=O)=O)C1 50349,CCCC(CNC(c1cc(CO)c(C)o1)=O)C(=O)NCC1CC1Cl 50350,C(CCCC(=O)NC1CCC(NC(C2(C)CSC2)=O)C1)SC 50351,C(=O)(CC(C(F)(F)F)OCC)N1CCC(CC=C)(NC(=O)COCCCOC)C1 50352,N1(C(CC(C)CNC(=O)CCc2ccc[nH]2)=O)CC2(CNC(=O)N2)C1 50353,C1(NC(c2nc(C(C)OC)sc2)=O)CN(C(=O)Cc2ccccc2F)CC1(C)C 50354,CC1Cc2cc(OCc3ccc(C(C)C(F)(F)F)cc3)ccc2O1 50355,CN1C(=O)CSC1=CC(=O)NCC1CC2CCC1N2C(=O)CN1CCCCC1=O 50356,Cc1ncc(C=CC(N2CCC3CN(C(c4cc(C)nn4C)=O)CC23)=O)c(O)n1 50357,N1(C(C(=O)NC)=O)C2CCC1CC(N(C)C(C1CC(C(F)(F)F)(OC)C1)=O)C2 50358,Cc1ccc(C)c(C(=O)NC2CN(C(C3CC3C3CC3)=O)CCC2(F)F)c1O 50359,c1(CC(=O)NCC(C)N(C(=O)Cc2nccn2C)CC)ncc(F)cn1 50360,C1(C(=O)NC2(CNC(C3(F)CCS(=O)(=O)C3)=O)CC2)CC(c2ccccn2)=NO1 50361,C1(CC(=O)OCC)CCN(C(c2cccc(Br)c2Cl)C(=O)NCCSC)C1(C)C 50362,c1(C(N2CC(NC(C(C(COC)C)C)=O)(CO)C2)=O)ccc2c(c1)SCC(=O)N2 50363,N1(C(C(C=CC)O)=O)CCN(C(=O)CCn2cc(C)cn2)C2CC12 50364,CC1CC(C(=O)NCC2(CNC(=O)C(O)CF)CCC2)CN1C(=O)OC(C)(C)C 50365,N1(C(=O)COc2cccc(Cl)c2Cl)CCC2(CC(NC(C3(CO)CC3)=O)CO2)C1 50366,c1(OC)ccc2c(CC(=O)NCC3CCN(C(C4(C)CCC4)=O)C3)coc2c1C 50367,c1(CC)ccc2c(c1)OCC2C(=O)N1CCC(C)C(F)(F)CC1 50368,C(=O)(CCC[N+](=O)[O-])NC(CC)CNC(=O)C(C)Oc1cccc(F)c1 50369,c1(C(=O)NC(CNC(CNS(CC)(=O)=O)=O)(C)C2CCC2)cccc(F)c1Cl 50370,CC1(C(F)(F)F)CS(=O)(=O)CCN1C(=S)NCC1(O)CCCCC1 50371,CS(=O)(=O)C1CCCN(C(c2cc(Cl)ncc2C(F)F)=O)C1.C12CCCN1C(=O)C2 50372,C(CC(C)C)(C(=O)N(C1CC(C(N)=O)C12CCC2)Cc1ccon1)OC 50373,CC(C)CC(C)(O)C(=O)N1CCN(CCCNC(=O)CCNC(C2CCC2)=O)CC1 50374,c1(C(=O)NC(CCNC(c2cc(C)n(C)n2)=O)C)c[nH]c2cccc([N+](=O)[O-])c12 50375,CCC(CC(=O)N1CCN(C(=O)C(=Cc2cccnc2)C)C2(CC2)C1)C(F)F 50376,c1(C(=O)NCC2C(NC(C3(OC)CC3)=O)CCCC2)c(OC)cc(OC)cc1N 50377,c1(C(=O)NCC2CCS(=O)(=O)C2)cc(-c2cccnc2C2CC2)cc2c[nH]nc12 50378,C(=O)(CC1OCCc2ccsc21)NCC1C(C)CCCN1C(=O)Cc1cccs1 50379,CC1CCN(CC(=O)Nc2ccnc(C(=O)NCc3cccnc3O)c2)CC1 50380,N1(C(C(COC)N(C)C)=O)CCOC(CCNC(=O)CSc2cccc(Cl)c2)C1 50381,Cc1cc(CCC(=O)NCC2CC(NC(=O)Cn3nccn3)C(O)C2)nn1C 50382,c1(C(=O)NC2(CNC(C(Br)=C(C)C)=O)CC2)cn(C2CCC2O)nn1 50383,C12(NC(C=C(C)C3CCCCC3)=O)CCCCCC1N(C(C1CCC1)=O)CC2 50384,c1(C(=O)NC(C)CCNC(=O)CSc2nnc(S)s2)cc2cccnc2[nH]1 50385,Cc1nc(O)sc1C(=O)NC1CCOCC1C(=O)NCCC1CC(F)(F)C1 50386,Cn1c(COC(C2OCC2(C)C)=O)ccc1Cl 50387,c1(C(=O)NC2CN(C(C3(C=C)CCC3)=O)CC2C)ccc(NC(=O)OC)cc1Cl 50388,c1(CC)ncc(C(N2CCC(CF)(NC(=O)CC3C=NN(C)C3=O)C2)=O)c(C)n1 50389,C1(CNC(C(CC#C)C2CC2)=O)CN(C(=O)CNC(C)=O)CC12CCC2 50390,CCC(C(=O)NC(C)(C)C=CC(=O)NC(C)CCC1CC1)n1ccnc1 50391,c1(-n2c(C3C(CC)C3)nc(C3CC3(C)C)n2)ccc(C)cc1OC 50392,CCC(C)CC(=O)C(=O)NC(c1cn(C)nn1)C(=O)NCc1cc(Cl)ccn1 50393,C1(CC(N2CC(C)(C(=O)NCC3(F)CCOCC3)C2)=O)(OC)CCOCC1 50394,C1(NC(C2CC(=C)C2)=O)CC(CNC(c2ccc(NC3CC3)nc2)=O)C1(C)C 50395,c1(C(=O)NC(CNC(CN(C(C)C)C)=O)C(C)C)cn2c(n1)SCC2 50396,S(=O)(=O)(c1nc(N2CCC(C(C)(C)CO)CC2)ccc1Br)NC(CC)CO 50397,c1(C(=O)NCC2(C)CCN(C(C3CCCCO3)=O)C2)ccc2cnsc2c1 50398,N1(C(C)=O)CSCC1C(=O)NCC(O)CNC(C1(NC(N)=O)CCCC1)=O 50399,C1(CC(=O)N(CCO)Cc2cc(CCOCc3cccs3)on2)CCCCO1 50400,c1(CNC(C(N2C(=O)CCC2=O)CC)=O)ccccc1CNC(C1SCCS1)=O 50401,c1(C(=O)Nc2c(C(N(C)Cc3ccc(CC)cc3)=O)c[nH]n2)cc2occc2[nH]1 50402,c1(N(C)C)ccccc1N(C(=O)C(=O)NCC(=O)Cc1ccccc1)C 50403,C(=O)(C(C)C(O)CCCC)NC1(CC(=O)N(CCCCCC=C)C)CCCCC1 50404,Cc1ccc2nn[nH]c2c1NC(=O)N=c1cc(C2CCCO2)[nH][nH]1 50405,CCCCCCC(CC)C(=O)N(CC(CC)NC(c1nnn2c1CCC2)=O)CC 50406,C1(C(=O)NC2CC(C(CC)CC)OCC2)CC2(CCOCC2)CCO1 50407,N1(C(=O)Cc2ccccc2F)CCC(CCCNC(C23CCC2C3)=O)CC1 50408,N1(C(CC(C)F)=O)CCN(C(c2csc(CO)n2)=O)CC1c1ccc(F)cc1 50409,N1(C(C(C)(CO)NC(CCCCC=C)=O)=O)CC(C)OC2(CCC2)C1 50410,C1(C(=O)NCC2N(C)CCC2)CCCC(NC(C2(CO)CCCC2)=O)CC1 50411,N1(C(=O)OC(C)(C)C)CC(NC(C2CCCCC2C#N)=O)CC(C)C1 50412,C1(C(N2C(C(N(CCn3c(C)ncc3)C)=O)C(C)C2)=O)CCCC(C)(C)C1 50413,C12(C(=O)NCCC(CNC(c3cc(C)nc(O)n3)=O)(C)C)OCCCC1C2(F)F 50414,C1(N)CCCCN1S(=O)(=O)N(C)C.Cc1ccccc1Nc1nc(C)cs1 50415,c1(C(N2CCC(NC(c3c(C(C)C)[nH]cc3)=O)C(C)C2)=O)cccc2cnnn12 50416,c1(C(N2CCC(NC(C3C(=C)CC3)=O)(CO)C2)=O)cc2c(Br)cccn2n1 50417,N1(C(=O)C2=CS(=O)CCC2)CCOCC2(COCCN2c2nc(Cl)ncc2F)C1 50418,CCS(=O)(=O)CC(=O)N1CCCCC1C1CCN(C(C2CC2F)=O)C1 50419,c1(NC(c2c(CC)sc(=N)[nH]2)=O)cc2c(cc1Br)CCC(=O)N2 50420,N1(C(C2C(C(C)C)C2)=O)CCC(O)(CN(C)C(c2ccc(CC3CC3)cc2)=O)C1 50421,CC1CN(C(=O)CC2C(C)(C)C2(C)C)CC1NC(c1ccc(CO)cn1)=O 50422,c1(CC)cnccc1C(N1CCOC(C(=O)NCC2COC(=O)N2)C1)=O 50423,N1(CC(CC(C)C)c2ccccc2)CCNCC(O)C1 50424,c1(C(=O)NCC(CN(C(C2CCC(C)C2)=O)CC)(C)C)cn2c(n1)SCC2 50425,CC1(C)CCCCC1(C)NC(c1cccc(CNC(c2cscn2)=O)n1)=O 50426,N1(C(C2OCCC(C)C2)=O)CC2CN(C)CC(C1)O2 50427,c1(C2(CNC(=O)NCCC(COC)OC)CC2)nc(C)cc(O)n1 50428,C1(C2CCN(C(C3CCCC3)=O)C2)(NC(C(C)c2ncco2)=O)CC1 50429,c1(C(=O)NCC=C2CCN(C(CC(C)C3CC3)=O)CC2)cc(Cl)cc([N+](=O)[O-])c1 50430,C1(NC(=O)CCC2CC2(F)F)CC2(C1)CC2NC(=O)CC1CCCC1 50431,c1(C(N(C2CC2)CC)=O)cc2cc(-c3cccc(S(C)=O)c3)ccn2n1 50432,N1(C(CCCCC#C)=O)CCC2(CC1)CC2CNC(c1c[nH]ccc1=O)=O 50433,C1(C(N2C(CC(=O)Nc3cncc(Cl)n3)CCC2)=O)CCCN(CC(F)(F)F)C1=O 50434,N1(CCc2cccc(C(N)=O)c2)C(=O)CN(CC2CC(F)C(=O)N2)C1=O 50435,CC1CN(C(=O)CCC(F)(F)F)CC1(C)C(N1CC(F)CC1CO)=O 50436,c12ccoc1CNC2C.c1(CNC(C2(CCC)CCC2)=O)noc(C(C)(C)C)n1 50437,N1(C(c2c(Cl)nc(OC)s2)=O)CC(C)CN(C(c2n[nH]c(=N)s2)=O)C(C)C1 50438,c1(OC)cncc(CC(=O)N(C2CCN(C(=O)C(C)(F)F)CC2)CC(C)C)c1 50439,C(=O)(C1=NOC2(CCC2)C1)NCC(CN(C)C(c1ncc(C(F)F)s1)=O)(C)C 50440,c1(CC)cccnc1C(N1CCC(C(C)NC(=O)CNC(C2CCC2)=O)CC1)=O 50441,C1(NC(C(Cc2ccsc2)NC=O)=O)CC2CCC1N2C(=O)Cc1ccn(C)n1 50442,N1(C(C(CC=C)C)=O)CCC(C2CCN(C(C3(c4ccnn4C)CC3)=O)C2)CC1 50443,c1(C(=O)NC(C)C(C)(C)NC(=O)CSCCC(C)C)cc2nc(O)[nH]c2cc1N 50444,Cc1ccncc1C(=O)N(C)CCOCCN(C(=O)Cc1cscc1F)C 50445,CCC(CC)C(F)C(=O)NCCN(C(=O)Cn1cnnn1)C 50446,Cc1ccc(Cl)c(C(N2CCC(O)C(NC(=O)C(C(C)(C)C)C3CCC3)C2)=O)c1 50447,N1(C(CCCC2CCCC(=O)N2)=O)CC2CC(N=c3cnc(F)c[nH]3)C2C1 50448,c1(C(=O)NC2C(C)CN(C(=O)C=CC(C)(C)C)C2)nn(C)cc1S(C)(=O)=O 50449,N#CC1(CC(=O)NC2CCOC(CNC(=O)C=CC3CC3)C2)CCCCC1 50450,c1(Cc2nnn(CC(F)(F)F)n2)nc(O)c2cnn(C)c2n1.CN1CCN1C 50451,c1(C(=O)NC(CN(C(=O)CN2C(=O)CNC2=O)CC)C)ccc2cc[nH]c2n1 50452,C1(C(=O)NCC(C)NC(=O)CCCC(N)=O)CC12CCC1(CC2)OCCO1 50453,c1(C(N(C2C3CN(C(c4cnc(C5CC5)[nH]4)=O)CC23)C)=O)ccc(O)nc1Cl 50454,C1(C(C)(C)NC(C2CN(C(C)C)C2)=O)CCN(C(=O)Cc2nncn2C)CC1 50455,c1(C(N2C(CCCC)C(=O)NCC2)C(=O)NC(C)C)ccc2c(c1)cc(C)n2C 50456,C(C1CN(C(=O)CC2CCN(C)C2=O)CC1C(=O)NCC1(CCCO)CC1)=CC 50457,c1(NC(C2N(C(C3(COC)CC3)=O)C(C)CC2)=O)nnc2ccc(Cl)nn12 50458,O=C(NN1CC(C(N2CCCC(F)C2)=O)C1)C1CC=CCC1C(=O)O 50459,CCC(C)C(CC(=O)N1CC(O)C1)NC(C1CCCS1)=O 50460,c1(C(C(=O)NC2CCCN(C(Cn3c(C)cc(C)n3)=O)C2)O)cc(F)cc(F)c1 50461,C(=O)(CCCC(=O)N1CC2(CNC(=O)CC3(C)CC(F)(F)C3)CC1CO2)N(C)C 50462,c1(NC(C2(C)CCCN2Cc2ccc(O)cc2O)=O)ncnc2sc(Br)cc12 50463,c1(C(N(CC(CNC(CSCC(C)C)=O)C)C)=O)cc([N+](=O)[O-])c[nH]1 50464,c1(C(=O)NC2CN(C(c3c(C)nns3)=O)C(C)CC2)cccc2nc(Cl)cn12 50465,c1(NC(C2CCCN(C(=O)CSc3cccc[n+]3[O-])C2)C)ncc(C#N)cc1Cl 50466,N1(C(COCC#C)=O)CC2CC2(C(=O)NC(COCC2CC2)CC)C1 50467,Cc1cnc(C(=O)NCC2CN(C(C34CC(F)(CO3)C4)=O)C2)cc1Br 50468,C1(C(N2CC(C)(c3cn(CC4CC5CCC4C5)nn3)C2)=O)CCC(C2CC2)C1 50469,C1(O)(C(C(=O)N(C(=O)CSC2(c3cc[nH]n3)CC2)CCS)F)CCCC1 50470,C1(NC(C(C=C)(C)C)=O)CCCC2CN(C(c3cnc(SC)nc3O)=O)CC12 50471,C1(C(=O)NCC(CNC(c2c(C)noc2)=O)(C)C)CCCCC1F 50472,N1(C(COC)=O)CCC(CCCCCNC(c2ccnc(C(C)(F)F)c2)=O)CC1 50473,C1(CC#C)(C(=O)NCC2CCN(C(=O)C(c3ccccc3)C)C2)CCCC1 50474,n1(CC(=O)NC2(C3N(C(CC(C)F)=O)CCC3)CC2)cc2ncccc2n1 50475,N1(C(Cc2cccc(C)c2)=O)CCCC2(NC(c3cnc(Cl)[nH]3)=O)CC2C1 50476,C#CC(CC(C)C)NC(=O)C(C)CN(C(=O)C(C)(C)CC)C 50477,CN1CCCC12CN(C(C1(C(=O)O)CCN(C(=O)OC(C)(C)C)CC1)=O)C2 50478,c1(OC)ccc(C(N2CCN(C(C3CN(C)CCO3)=O)CC2C)=O)c(OC)c1C 50479,C(CC(C(C)C)NC(c1cccc(-n2cncn2)n1)=O)NC(C(C=CC)O)=O 50480,C(CN=c1nc(C(=O)OC)nc[nH]1)C1CCC(NC(CC2(OCC)CC2)=O)C1 50481,C(CCC1CCC1)(C(=O)N(C1(CO)CC1)C)NC(COC(CC)CC)=O 50482,c1(CC)cccc(CN2CCC(C(N)=O)(Cc3ccccc3)C2)c1F 50483,c1(C(N2CC3CC3(C(=O)NCc3ccccn3)C2)=O)c(F)ccc(F)c1Cl 50484,N1(C(Cn2ccc(C)n2)=O)CC2(CC2)CC1C(=O)NCC1CCCO1 50485,c1(C(=O)NC(CC2CN(C(C3CC(CCC)C3)=O)C2)C)cc(C)nn1C 50486,C12(NC(CSS(C)(=O)=O)=O)CCOC(CNC(C3CC3C(N)=O)=O)(C1)C2 50487,c1(C(=O)NCC2(O)CN(C(C(C)NC(=O)NC)=O)C2)ccc2cc[nH]c2c1 50488,Cc1cccc(C(=O)NC2CCCCC2CC(=O)NC(c2cccnc2)C)c1N 50489,C1(C(=O)NCCc2ncccc2F)COCCN(C(c2n[nH]c3c2COC3)=O)C1 50490,c1(CNC(=O)NC2(C)C(C)OCC2)ccc(S(N)(=O)=O)cc1 50491,c1(C(N2CC3C(C(=O)Nc4ncc(SC)s4)(C3)C2)=O)cc(O)c(O)c(Cl)c1 50492,c1(C(=O)NC(C2CN(C(=O)C=CCN(C)C)C2)C)ccnn1C1CC1 50493,C1(CC)CCCCC1C(N1CC2C(CNC(=O)CCc3ccncc3)C2C1)=O 50494,n1(CC)cc(C(=O)N(C2CCN(C(=O)C(O)COCc3ccccc3)C2)C)nn1 50495,N1(C(C2(CCCC)CC2)=O)CC(NC(=O)CNS(=O)(=O)C2CC2)CC(O)C1 50496,N1(C(C(C)CO)=O)CCCCC(N(C)C(c2cnnc(-c3ccccc3)c2)=O)C1 50497,N1(C(c2c(C)cn(C)n2)=O)C2CCCC1CC(NC(c1cn(C)[nH]c1=N)=O)C2 50498,N1(C(c2cc(C)nnc2)=O)CC(=O)NCC1C(=O)N(CC(=O)N(C)C)C 50499,C1(C(=O)NCCCCC2CN(C(C3CCC(C(=O)OC)C3)=O)C2)CC12CCOC2 50500,N(C(=NCCc1ccccn1)N1CCCC(O)CC1)CC(C(=O)OC)C 50501,C(C(C)C(C)C(=O)N1CC(C(C)NC(c2ccc(F)cc2F)=O)C1)OC 50502,CCC(C)CCC(=O)NCC12CC1CN(C(=O)C=CSCc1ccco1)C2 50503,N1(C(c2c(C(C)(C)C)ncnc2)=O)CC2(C1)CN(C(=O)CC1CCC(C#N)C1)C2 50504,N1(C(C2C(NC(c3c(C)n[nH]c3)=O)CCC2)=O)CCN2CCOCC2C1 50505,C1(C(N2CCC(C)(NC(C3N(C)CCCC3)=O)C2)=O)CN2CCN1CC2 50506,N1(C(CCC)=O)CCN(C(C2CC=CCO2)=O)CCC1C 50507,C1(CNC(CC2ON=C(C)C2)=O)(CNC(c2cncc(Cl)c2)=O)CC12CCC2 50508,c1(C(N2CC(COC)(NC(=O)CN(C(=O)C(C)C)C)C2)=O)ccc2c(n1)CCOC2 50509,C1(NC(C(C)Cn2cccn2)=O)CC(F)CN(C(c2cn(CC3CC3)nn2)=O)C1 50510,Cc1c[nH]cc1C(N1CCC(NC(c2ccsc2-n2cnnn2)=O)C1)=O 50511,Cc1cnn2ccc(C(=O)NCC3C4CN(C(=O)C(O)CC(N)=O)CC34)nc12 50512,N1(C(C2CCC(=C)CC2)=O)CCOC2CN(C(c3cc(COCC)no3)=O)CC12 50513,C(N(O)C(=O)C(O)Cc1cc(F)c(F)c(F)c1)c1cc(=N)[nH]cc1 50514,C=C(C)CCC(C(=O)NCCCC1CC1)N(CC(F)(F)CCC(=O)OCC)C 50515,N1(C(CN(C)CC)=O)CC2CCC1C(C(=O)Nc1cc(Cl)ccc1O)C2 50516,n1(CC(N2C(C(CNC(C)=O)Cc3ccccc3)CCC2)=O)cc(F)ccc1=O 50517,c1(C(=O)NCC(=O)Nc2ccc(C(C)=O)cc2)c(N)cc(F)cc1Cl 50518,C=C(Cl)C(C)(C)C(=O)N1CC(CCNC(=O)CCn2cc[nH]c(=O)c2=O)C(C)C1 50519,c1(C(N2CCCCC(NC(C(COC)OC)=O)CC2)=O)nc2n(c1Cl)CCCC2 50520,O=C1CC2(C1)CC1(CC(NC(C3CCC(c4ccccc4)C3)=O)C1)C2 50521,N1(C(C=CCOC)=O)CC2CCCC1C2CNC(=O)CSCC(F)F 50522,Cc1occc1CC(=O)NC1CC1CNC(c1nocc1-c1ccccc1)=O 50523,C1(CC)CCCN(C(c2cc(CNC(=O)CCc3ccn(C)n3)nn2C)=O)CC1 50524,c1(C(=O)NC(C2CCCCC2)C(N2CC(O)C(O)C2)=O)ccn2nccc2c1 50525,C(=O)(C(C)(CO)NC(=O)CC1CCN(C(=O)CCC2CCC2)C1)OC 50526,N1(C(c2ccc(CN(C)C)nc2)=O)CC2CC(C1)C2NC(c1ccccc1F)=O 50527,N1(C(CC2(COC)CCCCO2)=O)CCC2(CCC(NC(=O)C3CC3)C2)CC1 50528,N1(C(Cc2ccc(C#C)cc2)=O)CC2CCC(C1)N2C(C1CC1C(=O)OC)=O 50529,c1(C(c2n(C(C(=O)OC)C)nnn2)NCCP(C)(C)=O)ccc(Br)c(F)c1F 50530,N1(C(c2c(OC)c(C)cs2)=O)CCOCC(NC(C2CCS2(=O)=O)=O)C1 50531,c1(C(=O)NCC2(NC(C3CN(C)C3)=O)CCCCC2)cc2c(cc1N)CCC2 50532,C1(C(=O)NC(COC)CO)N(C(=O)CCOC2CC2)CCCC1(C)C 50533,c1(CCC(N2C(CNC(C3CCCCC3)=O)CC(O)C2)=O)cc(Cl)ccc1Cl 50534,Cc1ccc(CCC(N2CC(C)(NC(c3cscc3F)=O)C2)=O)cc1 50535,N1(C(C(C(C)O)(F)F)=O)CCC2(CC1)CCN(C(C1(C(=O)OCCO)CC1)=O)CC2 50536,C1(CNC(C2(C)CC3CC3C2)=O)CCN(C(=O)CC2CC2C2CC2)CC1(F)F 50537,c1(N(C)C)ccc([N+](=O)[O-])c(C(=O)NC2CN(C(C3CCC3(F)F)=O)CC2O)c1 50538,C1(C(=O)NCC(C#C)OC)(COC)C=CCN1C(=O)CCOCCN(C)C 50539,CC1(C)CC(CNc2cc(N3CCOC(c4ccc(F)cc4)C3)ncn2)CO1 50540,c1(CCNC(C(=O)Nc2cn(C(C)(C)C)nc2)=O)ccc(Br)cc1Cl 50541,C1(CNC(c2c(CC)noc2C)=O)CCN(C(c2c[nH]c(C)c2)=O)CCC1(F)F 50542,N1(C(CC(C)F)=O)CCCC(CNC(C2(F)CCCCC2)=O)CC1 50543,CC(CF)CC(=O)NC(CNC(=O)C(c1ccc(Cl)cc1)(F)F)CO 50544,c1(C(=O)NCC(C)NC(c2c(F)ncc(OC)c2)=O)ccc(F)c(C)c1N 50545,C1(COCC)CCCN(C(CC2CCC3CC23)C(=O)NC2CC2)C1 50546,CCC(C)(C(=O)NC1CN(C(c2ccccc2C)=O)C(CC)(CC)C1)OC 50547,c1(NC(CC)=O)cccc(C(N2CC(NC(c3csc(Cl)c3)=O)C3CC23)=O)c1 50548,c1(-n2cc(CN(C(=O)Cc3cccnc3)O)nn2)ccnc(Cl)c1F 50549,C(=O)(C(CC(C)C)NC(C)=O)N(C1C2CN(C(C3(CO)CCCO3)=O)CC12)CC 50550,c1(C(N2C(CCNC(c3ccc(CC)cc3)=O)CC2)=O)cc2cc(Cl)ccc2s1 50551,c1(C(=O)NC2(CN(C(C3CC(C)NC(=O)C3)=O)C)CC2)ccc(Cl)c(F)c1N 50552,c1(CC)ccc(C=CC(=O)NC2CN(C(=O)CCN3CCCC3)CC2SC)o1 50553,CC(CS(C)(=O)=O)C(=O)NCCC1CCN(C(c2cc3c(ccn3C)[nH]2)=O)C1 50554,C1(OC)CC(N(CC(=O)OCCOc2ccc(C)cn2)C)C12CCOCC2 50555,c1(CCC(N2CC(NC(CSCCCC)=O)C2)=O)cc2ccccc2o1 50556,C1(C(=O)NCC(CCC)C)(C(C)C)CCN(C(=O)C(CO)NC(N)=O)C1 50557,Cc1cc(C)n(CC(N2CC(N(C(=O)Cc3c(C)noc3Cl)C)C2)=O)c(=O)n1 50558,c1(C(=O)NCC2CC(F)(CNC(c3cncs3)=O)C2)cc2cccnn2n1 50559,C1(C(=O)NCC(=O)OCCCC)CCCN(C(=O)C2=NNC(=O)C2)CC1 50560,c1(OC)ccc2c(CNC(c3cnn(C(F)(F)F)c3C)=O)c[nH]c2c1 50561,c1(C(=O)NCC2(F)CCN(C(CNC(CC)=O)=O)C2)cccc(F)c1Br 50562,C1(C(N(C)CC2(C)CC2)=O)CC(C)(NC(=O)Cn2cc(CO)nn2)C1 50563,c1(C(N2CCN(C(CNS(NC)(=O)=O)=O)C(C3CC3)C2)=O)ccc(O)c(C)c1C 50564,c1(CC(=O)NCC(CNC(c2nc(CCC)sc2)=O)O)ccc(CO)c(C)c1 50565,C1(NC(c2cnc(C3CC3)[nH]2)=O)CC2CC1N(C(c1csc(Cl)c1Cl)=O)C2 50566,c1(C(N2CC=CC(C(=O)O)C2)=O)cnc2[nH]ccc2n1 50567,N1(C(C2C(C)C2(F)F)=O)CCC(C)N(C(c2cc(C3CCOCC3)on2)=O)CC1 50568,N1(C(c2ccc(C(=O)OC)[nH]2)=O)C2CCCC1CN(C(C1(F)CCOC1)=O)CC2 50569,Cc1cccc(C)c1CS(=O)(=O)NC(C1CCC(F)(F)C1)C 50570,C1(C(=O)NC(C2CC=CCC2)C(=O)NCCC2(O)CCCC2)(SC)CC(=O)C1 50571,C12CN(CC13CC3)C2=O.Cc1ocnc1CC(=O)NC1CC(=C2CC2)C1 50572,Cc1nc(-c2c[nH]c(C(=O)N(C)CC3CCN(C(C4CC4[N+](=O)[O-])=O)C3)c2)cs1 50573,N1(C(C(CN(C)C)(C)C)=O)CCC2(CCN(C(=O)CC3CCCCC34CC4)C2)C1 50574,C1(CC(=O)N(CC(=O)NCCOC(CC)CC)C2CC2)CC2C=CC1C2 50575,n1(CC(=O)NCC(c2ccn(C)c2)C)cc(NC(C(C)C)c2nc[nH]n2)cn1 50576,CC1CCC(C2CCCC2)CN1Cc1cn(CCC2CCCNC2)nn1 50577,c1(OC)ccc(Cl)cc1C(N1CCC(NC(=O)CC2(C(F)(F)F)CC2)C(O)C1)=O 50578,N1(C(CC2(C=C)CCC2)=O)CC2CC2(CNC(=O)CC2CCC(=O)N2C)C1 50579,c1(C(N(C2CCN(C(=O)C=Cc3cn[nH]c3)CC2)C)=O)cc(O)cc(C#N)c1 50580,COn1cnc(C)c1C(=O)NCc1ncncc1C(=O)NCCC(C)CO 50581,C(=O)(CC(C)CC(C)C)NCCCCN(C(c1cccc(NC(=O)OC)c1)=O)C 50582,C(=O)(C1CCc2c[nH]nc21)N1C(C(N(CC#C)CCO)=O)C2(C1)CCCC2 50583,N1(C(C(CC)(C)C)=O)CC2CCC2(NC(=O)COc2cccc(F)c2)C1 50584,C(=O)(C1CCCc2scnc21)NC1CN(C(COCCOCC#C)=O)C1 50585,Cn1nc(C(=O)NC2CCN(c3nc(C4CC4)ns3)CC2O)c2c1CCCC2 50586,C1(CNC(C2CCC(=C)CC2)=O)C(C)CCCN1C(=O)Cn1cc(C)cn1 50587,C1(CNC(CCC2N(C)CCCC2)=O)CCN(C(c2ccc[nH]2)=O)CC1O 50588,CC1(NC(=O)C(O)C(C)(C)C)CCN(C(=O)Cn2cnnc2)CC1 50589,C(=O)(C(C(C)O)NC(=O)CC1CCCN(C)C1)N(C1CC(C)C1)C 50590,C1(C(N(CCCNC(=O)COC2CCOC2)C2CC2)=O)CC=CCC1 50591,Cc1noc2nc(C(=O)NC3CCCN(C(=O)CC4CNC(=O)C4)C3)ccc12 50592,CC(c1ccccc1)=CC(=O)NC1CC1CNC(=O)C(C)n1ccnn1 50593,C1(NC(=O)CSC2CC2)CC2CN(C(c3cccc(-n4cccc4)c3)=O)CC12 50594,C1(COC)CN(C(C2(C)CCCCO2)=O)CCN1C(=O)CN1CCC(O)CC1 50595,N1(C(CC2OCC(C)(C)C2)=O)CC(C(N2CC(N3CC(F)C3)C2)=O)C(F)(F)C1 50596,c1(C(=O)NC2CCCN(c3ccc(C#N)cc3)C2)cc(Cl)sc1S(N)(=O)=O 50597,c1(CNC(C2(C)CCN(Cc3ncn(C)c3)CC2)=O)ccc(C#N)c(F)c1 50598,c1(N(CCOC)C)nnc(CN(S(C)(=O)=O)C)n1CC(C)C 50599,c1(N2CCN(C)C(CNC(c3cn4c(n3)CCC4)=O)C2)ncnc2[nH]ccc12 50600,c1(C(C(=O)NCCC(C)F)NC(C(C2CCC2)OCC)=O)ccccc1 50601,C1(C)(C(=O)OC)CNCCN1Cc1ccncc1 50602,c1(NC(C(c2ccc(Cl)o2)N(C2CCC2)C)=O)ccc(Oc2ccccc2)cc1 50603,CN(CCOCc1ccccc1)N1CC(CO)OC2(CCC2)C1 50604,n1(CC(=O)NCC2CC(O)CN2C(=O)Cc2ccc(Cl)s2)nc(Cl)ccc1=O 50605,C1(C(=O)NCCOCCOCCNC(C2(C)CC2)=O)CCCCC12CCC2 50606,N1(C(C(CCC#C)NC(c2cnc(S)nc2)=O)=O)CC(O)C2(CCCC2)C1 50607,c1(CC)cc(C(N2CCCC2CCC(C)C)C(=O)NCCC#N)ccc1Cl 50608,Cc1nc2cccc(C(=O)NCC(O)CNC(=O)Cc3cncc(O)c3)c2[nH]1 50609,C12(CNC(c3ccn(CC(F)F)n3)=O)CC1CN(C(C1CC=CC1)=O)C2 50610,CCC(O)C(C)(C)C(=O)NCC1CC2CCC1N2C(C1C2CCCC1CCC2)=O 50611,c1(OC(C(=O)NCCC(C)N(C(c2n(CC)ncc2)=O)C)C)cccc(CO)c1 50612,c1(C(=O)NCC2CC(C)N(C(c3ccoc3Cl)=O)CC2)ccc2c(n1)CCC2 50613,CCN(NC(=O)C(O)CCn1cc(CO)nn1)C(=O)OC(C)(C)C 50614,C1(C(N2CC(c3onc(C)n3)C2)=O)CCOCC1NC(C12CC(C#N)(C1)C2)=O 50615,N1(CCCC(=O)N(C)C)CC2C(Cc3ccccc3)CS(=O)(=O)C2C1 50616,CCCC(CC)CC(=O)N1CCCCC(NC(c2cc(C3(Cl)CC3)n(C)n2)=O)C1 50617,C1(NC(C(C)CC(N)=O)=O)CC12CCN(C(C1(O)CCCCCC1)=O)CC2 50618,C1(COC)CN(C(C2(CC(F)(F)F)CC2)=O)CCN1C(=O)CCS(C)=O 50619,N1(C(N(c2ccccc2)CC(C)(C)C)=O)CCN(S(=O)(=O)N2CCOCC2)CC1 50620,CC(C)(C)S(=O)(=O)CC(=O)NCC1CCN1C(C1(C)CCC(=O)N1)=O 50621,C1(C(=O)NCC2(CC)CCOC2)CCCCCCN1C(=O)C(C)CC(=O)OC 50622,CCCC(CCNC(=O)CCC1(C)CN(C(C2CCC(O)CN2C)=O)C1)CCC 50623,C12(C(N3CCC(N(C(C4CCCS4)=O)CC4CC4)C3)=O)C3CCC(CC13)C2(F)F 50624,c1(OCC(N2CC(NC(=O)C=Cc3ccccc3)C(O)C2)=O)ccc(F)c(Cl)c1 50625,C(c1ccccc1)=CCN(C(C1N(C(C)=O)CCC1)=O)C.C12CN(C1)C2=O 50626,C1(CNC(Cc2ccc(C)s2)=O)CCC2(CN(C(c3ccccc3O)=O)C2)O1 50627,CCC(CC(=O)N(CCOC)Cc1ccc(F)c(-c2nn[nH]n2)n1)C(F)F 50628,N1(C(C2C(C=C)C2)=O)CC(O)(CNC(=O)CC2COCC2O)C1 50629,Nc1cnc(C(=O)NC2CCC2NC(=O)C=Cc2ccccc2Br)c(Cl)c1 50630,C=CC(C)(O)C(=O)NCC1C(CNC(=O)CC(CC)OC)C1(F)F 50631,CC#CCC(C(=O)NCCC(O)CCC)NC(=O)C(C)OC1CCCC1 50632,c1(NC(C(C2CCN(C(c3nc(CC)sc3)=O)C2)C)=O)ccc(C)cc1CO 50633,N1(C(CCCOCC=C)=O)CCN(C(CNC(c2cc(C)cs2)=O)C(F)F)CC1 50634,C(=O)(CC(CC)C(C)(C)C)NC(C(=O)Nc1cnc(CCC)nc1)CC=CC 50635,c1(C(N2CC(C)(NC(CC(CCC)C)=O)C2)=O)cc2c(nc1O)CCC(CC)C2 50636,n1(C(CC)C)cc(-c2nc(COc3ccccc3)no2)c2ccccc12 50637,Cc1c(C(C)NC(c2ccc(O)nc2)C)cccc1Cl 50638,N1(CC(=CC(=O)NC(CNC(C(C)SCCOC)=O)CO)C)CCOCC1 50639,C(=O)(C(F)C(F)(F)F)NC(C)CCNC(C1(CNC(N)=O)CC=CC1)=O 50640,C=CCCCCCC(=O)N1CC2CC(NC(c3cc(C)oc3CC)=O)CC2C1 50641,C=CCCCCC(=O)NC(C1CCN(C(=O)C=C(Cl)Cl)C1)C 50642,c1(C(=O)NC2(CC=C)CN(C(=O)CS(=O)CC)C2)cnc(F)c(C)c1 50643,C1(C(CNC(C2(C)CCCC2)=O)O)CCN(C(c2ccc(O)nc2)=O)CC1 50644,C(CNC(c1cccc(CCCCO)c1)=O)(CC(F)(F)F)NC(C(C)OCC)=O 50645,S(=O)(=O)(c1ccc(-c2ccc(C(C)NC)cc2)s1)N(CC=C)C(C)C 50646,c1(C(=O)NCC2CCCN(C(c3c(CC)n(C)nc3)=O)C2)c(C)cc(O)cc1C 50647,C1(OC)CC(N(C(=O)CCOC2CN(C(=O)CCc3cccnc3)C2)C)C1(C)C 50648,c1(CNC(N2CCC(CC(=O)N(C)C)C2)=O)ccnc(Cl)c1 50649,C=C(C)CCCC(=O)N1CCC(C)C(CC(N2CC=CC2(C)CO)=O)C1 50650,c1(C(N2CC(C)C(NC(=O)CCCCC3CC3)C2)=O)ncc(CO)cc1Cl 50651,c1(N2CCC(OC)CC2)nc2c(c(=NC3CCCSC3)[nH]1)CC(C)CC2 50652,C(=O)(CCCCCNC(N)=O)NC1(F)CN(C(CN2CC(C)(OC)C2)=O)C1 50653,C1(CCC)CCN(C(=NCCc2ccncn2)NCCNC(=O)OC)C1 50654,N1(C(CC)=O)CC(=O)N2CCOCC2(CNC(=O)CC2CCCCC2(F)F)C1 50655,c1(CC)cccc(C(=O)NC(C(=O)NC2CN(C)NC2=O)C2CCCC2)c1 50656,C1(CCOC)(NC(c2c[nH]nc2C(C)C)=O)CCN(C(c2nnc(C)s2)=O)C1 50657,c1(CC(=O)NCC(C2CCOC2)NC(CC(C)(C)C)=O)csc2ccccc12 50658,C1(C)(C(N(C2CCCCCC2)C)=O)CC12CCN(CCc1ncccn1)CC2 50659,c1(C(=O)NCCC(CNC(C2(CSC)CC2)=O)O)ccc(-c2cnc[nH]2)cc1 50660,N1(C(CNC(CCC)=O)=O)CCN(C(=O)C(C)OCC(C)C)C(CC(C)(C)C)C1 50661,CCCCCC(F)C(=O)N1CCCC1(C(=O)NCC(C)C(=O)OC)CC 50662,Oc1nc(COC(c2cc3c(O)ncnc3cn2)=O)nc2ccccc12 50663,c1(OC)cc2c(cc1OC)C(NC(c1occ3c1CCC3)=O)CCCC2 50664,c1(OC)c(Cl)cc(C(N2CCC(NC(=O)CCC3CCC(=O)N3)C2)=O)cc1Cl 50665,N1(C(c2c(CCC)occ2)=O)CC2(CC(NC(=O)CN3CCCC3CO)C2)C1 50666,c1(N2CCC(CC)C2)nc(=NCc2nc(C(F)(F)F)n[nH]2)[nH]c2c1CCCC2 50667,c1(CC(C)N(CCCCN(C(C(CN(CC)CC)F)=O)C)C)c(F)cccc1F 50668,CC(C)CC(C)(C)C(=O)NC1COCC1NC(c1ccccc1OC1CC1)=O 50669,c1(C(N2CC3(C(NC(c4c(C)onc4)=O)CC3)C2)=O)cnc2cc(O)ccc2c1 50670,C1(C(=O)NC(C)CNC(=O)CCF)(CC)CCNC1=O 50671,c1(CCC)cc(C(=O)N(CCC(C)NC(=O)C(=C2CCCCC2)F)C)ccn1 50672,Cc1cccc(CCNC(=O)CCC2(C)CN(C(C3CC(C(C)C)C3)=O)C2)n1 50673,C(C(CO)C(C)(C)C)c1onc(-c2ncc(C)o2)n1 50674,C1(C(N2CC3C(NC(Cc4cc(C)c(Cl)cc4)=O)(C3)C2)=O)CCCC(F)(F)CC1 50675,C1(C)(C(N2CC(CC)(NC(c3ccc(C(F)(F)F)cn3)=O)C2)=O)COCC1(F)F 50676,S(=O)(=O)(c1nc(N2CCCC(OCC)C2)ccc1Br)NCC(c1ccccn1)(C)C 50677,C1(C(=O)NC2(CN(C)C(c3csc(CO)n3)=O)CC2)CC2CC(=O)C1O2 50678,N1(C(C(CC)O)=O)CCC(F)(C(=O)NC2(C3CCCCO3)CC2)CC1 50679,C12(CO)CCCC(CC1)C2.Cc1cncc(-n2cc(C3CCN(C=O)C3)nn2)n1 50680,C(=O)(C(F)CC(CC)CC)NCc1cc(C(N(CC#C)OC)=O)no1 50681,O=C1CCC(C(=O)NC(Cn2cccn2)C(=O)NCCCCN2CCCC2)O1 50682,c1(OC)c(F)ccc(F)c1C(=O)NC1CCN(C(c2cc(C)ccn2)=O)CC1F 50683,C1(C(N2CCN(CC(C)NC(C3(C)CC4CC4C3)=O)CC2)=O)Cc2cscc2C1 50684,N#CC1CN(Cc2ccc(O)c(O)c2)CC1NC(=O)Cc1cccc(C(N)=O)c1 50685,N1(C(c2ncn(C)n2)C(=O)NCC2(CC3CC3)CC2)CCC(O)C(F)C1 50686,Cc1ccccc1C(C)CC(=O)NC1CCN(C(=O)CCCF)C1 50687,N1(C(C2C(C(C)NC(c3ccc(COC)o3)=O)C2)=O)CC(CO)C1(C)C 50688,C1(NC(C2(CCC)CC2)=O)CC2CC(C1)N(C(=O)C(C)(C)C(F)F)C2 50689,c1(CC)c(NC(CNC(c2cnc(C)[nH]2)=O)C(C)C)ncnc1Cl 50690,CCC(C)(C(=O)N(CC(C)C(=O)Nc1cnn(C(C)(C)C)c1)C)OC 50691,CC(C)CC(C(=O)NCC1COCCN(C(=O)C(O)Cc2cnc[nH]2)C1)N(C)C 50692,Cc1cn(C)cc1C(=O)N(CC(C)NC(c1cc[nH]c1C)=O)C 50693,c1(C(=O)NCC2(C(=O)NC(C#C)CC3CCCC3)CCC2)cn(C(C)C)cn1 50694,CCC(C)(C(=O)N1CC(NC(=O)C(F)(F)c2cnn(C)c2)C(SC)C1)OC 50695,C1(NC(c2c(CC)scc2)=O)CC(NC(=O)C(C)C)C12CCOCC2 50696,N1(C(CCCOC)=O)CC(N=[N+]=[N-])CC1C(N1CCC(CF)C1)=O 50697,c1(OCC)nc(Cl)ccc1C(c1nnnn1-c1ccc(Cl)cc1F)NCCOC 50698,c1(C(=O)NC2CCC2NC(c2n[nH]cc2Br)=O)cccc(F)c1 50699,N1(C(COc2ccc(OC)cc2)=O)CC(NC(=O)C(F)C2CCC2)CC(O)C1 50700,CC(C)CC(F)C(=O)NCC1(C)CCCN(C(c2c(Br)cnn2C)=O)C1 50701,N1(C(C2N(Cc3c(OC)ncc(F)c3)C3C(C2)C3)=O)CCCC2(CCO2)C1 50702,CC(CC(=O)NCC(C)NC(c1cnc(C(F)(F)F)s1)=O)C1CC1 50703,CCC(C)(COC)C(=O)NCC(C)N(C(=O)CC1CCC=CCC1)C 50704,N1(c2n(CCC#C)c(-c3ccccc3Cl)nn2)CCc2cc(Cl)c(Cl)cc2C1C 50705,N1(C(c2cncc(N=[N+]=[N-])c2)=O)C2CCCC1CN(C(c1coc(CO)c1)=O)C2 50706,CCCCC(CNC(c1cccc(OC)c1)=O)NC(=O)CC1(OCCF)CCC1 50707,CC1CCN(C(C2(C)SCCCS2)=O)C1c1cn(-c2ccc(Cl)nc2)nn1 50708,CC1CN(C(c2ccnc(Br)c2F)C(=O)NC2CCC(F)(F)CC2)CC(=O)N1 50709,N1(C(Cc2cc(C)ns2)=O)CC2CC(NC(C3CC4CCC3CC4)=O)CC1C2 50710,N1(C(C(C=C)(C)O)=O)CC2CCCC(NC(=O)Cc3ccn(C)n3)C2C1 50711,N1(C(C(C)CO)=O)CCN(C(=O)CN2CCn3nccc32)CC1CCO 50712,N1(CC(=O)NCCC2(C)CC2)CCN(C(=O)Cc2cnoc2)CC1 50713,C(C)(CNC(C1(F)CC1)=O)(CC(C)C)NC(CCOc1c(C)cccc1)=O 50714,C1(NC(CCCC#CC)=O)CCC(C)(C)CC1CNC(c1cnc(N)c(N)c1)=O 50715,C(C(=O)NC)(C(C)CCc1ccccc1)N(CCOCCO)CC 50716,C1(O)(Cc2scc(C)n2)CCN(C(=O)CCn2cccnc2=O)CC1 50717,C1(C(=O)NC(C)Cc2cccnc2)CC2CCC1N2C(C1(C#N)CCCC1)=O 50718,N1(C(C(C)OC(C)=O)=O)CCC(NC(C2CC(O)CN2C(N)=O)=O)C(C)C1 50719,S(=O)(=O)(c1ccc(N)c(NC(C2CCCC(COC)O2)=O)c1)NCC 50720,C1(CC(C)NC(C(COC)O)=O)CCN(C(c2cncc(F)c2)=O)CC1 50721,C=Cc1ccc(C(N2CCC(C)C(NC(=O)CCC(C)(C)F)C2)=O)cc1 50722,c1(C(N(CC(C)NC(c2ccoc2Br)=O)C)=O)c[nH]cc(Cl)c1=O 50723,N1(C(C(CC)OC)=O)CC2(CNC(c3cc(OC)cc(F)c3)=O)CCC1CC2 50724,C1(CC)CN(C(=O)C=CC=C(Cl)Cl)CCC1CNC(c1cc(Cl)ccc1O)=O 50725,C1(C(=O)NCCNC(CC(C)F)=O)CC(c2cccc(Br)c2)=NO1 50726,c1(C(N(C(CCNC(C2N(C(C)=O)CCOC2)=O)C)C)=O)nccc2n[nH]cc12 50727,c1(CC)cnc(O)c(C(=O)NCC(CO)NC(=O)C(c2ccnn2C)C)c1 50728,n1(CCC)nnnc1C(c1cnc(C(=O)OCC)s1)NCCC(C)OC(C)(C)C 50729,Cc1c(C(C)NC2(C)CC2(C)C)cnn1-c1ccc(F)cc1 50730,c1(CC(=O)NC(C2CCCC2)CNC(CNC2CCC2)=O)cc(C)oc1C.CO 50731,C1(C(C)C)N(C(C2CSCN2)=O)CC12CCCOC2 50732,CC1(C)CN(C(=O)Cc2ccc(C#N)cc2)CC1NC(C1(CC2CC2)CC1)=O 50733,N1(C(Cc2nn(C)c(Cl)c2)=O)CCC2C1CCCN2C(=O)C(S(C)(=O)=O)C1CC1 50734,C1(F)(C(=O)NCC2CC(C#N)C2)CCN(C(=O)Cn2cncn2)C1 50735,CC1COc2c(C(N3CC(CCO)(NC(c4ccc(O)cc4)=O)C3)=O)cnn2C1 50736,C1(C)(NC(C(C)Cc2cnn(C)c2)=O)CCN(C(C2CCCOC2)=O)CC1 50737,Cc1sc(Cl)nc1C(=O)NCC1COCCN1C(=O)CCn1nc(C)nc1C 50738,N1(C(CN(C(C)C)C)=O)CCC2(NC(c3cc(F)ccc3Cl)=O)CC2C1 50739,C1(NC(CCc2ncc(C)[nH]2)=O)CN(C(c2cc3c[nH]nc3s2)=O)CCC1C 50740,C(C(C)C(F)C(=O)NCc1cccnc1O)NC(C1(CC#C)CC1)=O 50741,c1(C(=O)Nc2ccc(Cl)c(OC(F)F)c2)noc2c1COc1ccccc1-2 50742,N1(C(C(C)C)C)CCC(C)(C)C1.C1(=O)CCCn2cc(nn2)C(C)(C)N1 50743,N1(Cc2c(C)noc2)CCC2(NC(c3ccnn3CC3CCC3)=O)CCCC12 50744,C1(C)(OC)CCN(C(C2C=CC(NC(c3cccc(Br)c3F)=O)C2)=O)CC1 50745,N1(C(C=C(C)C(C)C)=O)CCCC12CCCN(C(=O)CC1(O)COC(C)(C)C1)C2 50746,c1(OC)ccc(C(=O)N(CCCCN(C(=O)C(F)OC(F)(F)F)C)C)nc1N 50747,c1(C(=O)NC2CN(C(c3cn(CC=C)nc3)=O)CC(C)C2)cc(C)c(=O)n(C)c1 50748,N1(CCC=CCC)CCC(C2CCN(C(C3(C)CCS(=O)(=O)CC3)=O)CC2)C1 50749,N1(C(Cc2cccc(C)c2C)=O)CC2CCN(C(c3cn[nH]c3)=O)C2C1 50750,c1(C(=O)NCCC(C)N(C)C(c2ccnn2CC2CC2)=O)cc(C(F)F)ccn1 50751,c1(OC)cscc1C(=O)NCC1CCC1C(N1CCCC1C(C)(C)C)=O 50752,c1(OCC)ccc(C(=O)NC(C)CCCNC(=O)C=CC2CCCN2C)cc1C 50753,C(=O)(CCC(CC)CCC)N1CC(NC(CC(=O)NCC)=O)C1 50754,C1(NC(c2cc(C)ncc2)=O)COCCN(C(=O)CNC(=O)NC2CC2)C1 50755,c1(CC(=O)N(C2CC(NC(=O)C=CCO)C2)C)ccc2c(c1)OCO2 50756,C(=O)(C1CCCc2n[nH]cc21)N1CC(CCCNC(CC=CCC)=O)OCC1 50757,CC(C)(CCC(=O)NC1CCN(C(c2ccc(Cl)cc2)=O)C12CCC2)[N+](=O)[O-] 50758,C(=O)(C1=C(Cl)CCCC1)N(CC(=O)N(C1CCCC(C)(C)C1)C)C(C)C 50759,c1(C(C)(F)F)cc(C(N2CCC(NC(=O)C=CSCc3ccco3)C2)=O)ccn1 50760,CC(C)(CC(=O)N1CCC(NC(c2conc2C2CCC2)=O)C1)c1cccs1 50761,C1(O)(CC=C)CCN(C(=O)NCC2CCC2NC(=O)OC(C)(C)C)CC1 50762,c1(CCC)cc(C(N2CC=CC2CNC(C2(OCC)CCCOC2)=O)=O)ccc1C 50763,Cc1c([N+](=O)[O-])c(C(=O)NCC(C)(CO)NC(=O)CCC(C)(C)C)nn1C 50764,Cc1cc(C(=O)NC2CCCC(CNC(C3COC(=O)O3)=O)C2)n(C2CCC2)n1 50765,CC(O)CCCC(=O)NC(C1CCN(Cc2nc(-c3ccsc3)no2)CC1)C 50766,N1(C(c2n(CC)ccc2)=O)CCOCC(F)(CNC(C2C3CC4C(C3)C24)=O)C1 50767,CC(C)CCCCC(=O)NCC1CN(C(C2OCCC2C(F)(F)F)=O)CC1C 50768,N1(C(C(CC)=CC)=O)CCC(C(C)C(=O)N(C2CCC(F)(F)C2)C)CC1 50769,N1(C(C(CC)O)=O)CCC12CCCN(C(C1(Br)CC1)=O)C2 50770,C=C(C)c1cccc(NC(C2CCN(C(c3cscn3)=O)C23CCC3)=O)c1 50771,C(=O)(CCCCC(N)=O)NCC1(C)C(C)CN(C(CCOCC#C)=O)C1 50772,C1(CC)CCCCN1C(=O)C(CCN(C)C)NC(=O)C(CN(C)C)CC 50773,N1(C(C(C2CCCC2)OC)=O)CCN(C(c2cnc[nH]2)=O)C(C2CC2)C1 50774,c1(C(=O)NCCN(C(c2cnn(CCF)c2)=O)CC)cc2cccc(C)c2nn1 50775,C(C(C)C(C)C(=O)N(C)CC1(O)CCN(C(c2cn(C)cn2)=O)CC1)OC 50776,C(=O)(C1=CCC(F)(F)CC1)NC1CC2CN(C(c3ccc(C=C)cc3)=O)C1C2 50777,C1(CNC(CSCC#C)=O)CC2(CCC2)CN1C(C1CCC(C(C)C)NC1=O)=O 50778,C(=O)(CCCC(C)(C)C)N1CCC(C)CC1CNC(=O)CCc1cccnc1Cl 50779,C1(CC)CN(C(C23CC(F)(C2)C3)=O)CCC1NC(c1ccccc1O)=O 50780,N1(C(C2(CSCC)CC2)=O)CC(CNC(=O)OC(C)(C)C)C2(CCCC2)C1 50781,CC(C)C(O)C(C)C(=O)NCC1CN(C(c2ccn(CCO)c(=O)c2)=O)C1 50782,CC1CN(C(C2(CCF)CC2)=O)CCC1CNC(c1cc(N(C)C)ccn1)=O 50783,n1(CC)nccc1-c1cn(CCCOCCNC(c2cnc(Cl)[nH]2)=O)nn1 50784,C(=O)(CS(=O)(=O)C1CC1)NC1C2(CN(C(c3c(C)cc(O)nc3)=O)C2)CC1 50785,c1(C(N2CCN(C(c3occ(OC)c(=O)c3)=O)C(C)C2)=O)c(C)ccc(F)c1N 50786,C1(C(C)C)(C(=O)N(C)CC2(O)CCCCC2)CCN(C(C2CCCOC2)=O)C1 50787,C=C1CCN(C(C2CCS2(=O)=O)=O)C(C(=O)NC(CCC)C(=O)N(C)C)C1 50788,N1(C(=O)Cn2cc(C3CCCOC3)nn2)CCCC2(C1)C(O)CC2O 50789,N1(C(c2c(CC)ncc(Br)c2)=O)CC2CCC(C1)N(C(=O)C(C)C)C2 50790,Cc1cc(F)c(N)cc1C(N1CCCN(C(c2cscc2C(F)F)=O)CC1C)=O 50791,N1(C(CNC(C)=O)=O)C(CC(N2CCC2C2CCCCC2)=O)C2CCCC12 50792,C1(C(=O)NC2CCN(C(=O)OC)CC2)CCC(C)(C)CC1 50793,N1(C(CCC=CC(C)C)=O)CC(CNC(C2CCC(CO)CC2)=O)C(C)C1 50794,CC(C(=O)NC1C2CN(C(=O)CCc3cccc(C(F)(F)F)c3)CC12)C(C)(F)F 50795,c1(C(=O)NCC2CC(NC(=O)C(=Cc3cccnc3)F)C2)ccc2nsnc2c1 50796,CCC(C)C(O)CC(=O)NC1C2CC(NC(C3CCOCC3)=O)CC12 50797,C1(CC)CN(C(=O)CN2CCC(O)CC2)CCN1C(=O)CNS(N)(=O)=O 50798,c1(C(=O)NC(CCNC(C(CC=C)C)=O)C)cnc2c(c1)N(C)CCO2 50799,c1(OC)ncccc1C(N1CCCC(CC(=O)NC(C)(C)CN2CCCC2)C1)=O 50800,CCC(CC)C(=O)NCC1CC(F)(Cn2cc(C3CC3C(=O)O)nn2)C1 50801,C(CC(=O)N1CCn2ccnc21)(C(F)(F)F)NC(C=CC(CC)C)=O 50802,N1(C(c2cc(C)n(C)c2C)=O)CC2COCCC2(NC(=O)COCC(C)(C)C)C1 50803,c1(C(=O)NCCNC(c2cccc(OC)c2F)=O)cc2ccncc2[nH]1 50804,CCCCC(O)CC(=O)N1CC(C(=O)NC23CCC(CO)(CC2)C3)C(C)C1 50805,CCCC(CCCNC(c1cnc(OC)cn1)=O)NC(c1cnc(C)o1)=O 50806,Cc1ccc(C(N2CC(C(N3CCCC3C(F)(F)F)=O)C2)=O)c(O)c1 50807,C1(C(=O)NC(CC=C)CNC(=O)CSS(C)(=O)=O)CC(=O)N(CC)C1 50808,C1(NC(C(CC)N(CC)CC)=O)CCN(C(c2cc(C)cs2)=O)C(C)C1 50809,c1(C(=O)NC2CN(C(c3ccc(C)c(CO)c3)=O)C2)cc(N)c2ncccc2c1 50810,CC1CCC(CO)CN1C(c1cc(CNC(c2ccoc2)=O)cs1)=O 50811,C(=O)(C(O)CCCNC(c1ccccc1Cl)=O)NCCNS(N)(=O)=O 50812,CC1(C)CCCC(C(=O)NC(CNC(=O)CCc2ncco2)C2CC2)C1 50813,c1(C(=O)NCCC(=C)CNC(C2(OC)CS(=O)(=O)C2)=O)ccc(-n2cccn2)nc1 50814,C(c1cnccn1)=CC(=O)NCCCC1CN(C(=O)Cn2cnnc2)CCO1 50815,C1(C(=O)NCC(c2ccccn2)C)CCC2(CC2)N1C(=O)C(C)CC(F)F 50816,CCCC(CCC)C(=O)NCC1CC2(CC2)CN1C(c1[nH]nc(OC)c1Cl)=O 50817,Cc1c(C(=O)NC2(C#N)CCN(C(c3ccon3)=O)C2)cncc1Br 50818,Cc1c(C(N2CCC(NC(=O)C=CC3CC3)C23CC3)=O)sc(Cl)c1Cl 50819,C1(C(=O)NCC(C(C)C)(C)F)CCCC(NC(C2CCCSC2C)=O)CC1 50820,N1(C(CCc2cc(C)on2)=O)CC(N(C(=O)Cc2nn(C)cc2Cl)C)C(F)C1 50821,C(=O)(C(CCF)NC(=O)CC#N)N(CC(O)CO)C 50822,N1(C(CCCCCOCC)=O)CC(C(=O)OC)C2(C1)CN(c1ccncn1)C2 50823,N1(C(CCCSC)=O)CC(NC(=O)C(C)(C)c2cccnc2)CC1C 50824,C1(C(N2CCC(C)(CC(=O)NC3C(C(=O)NC)CCC3)C2)=O)CCCCCN1C 50825,C(=O)(C(O)C1=CCCCC1)N(CC(=O)NC(c1csnn1)C)C(C)C 50826,Cc1cc(Cl)nc(Cl)c1NC(C1CC(O)CN1C(c1cc(F)c(F)cc1O)=O)=O 50827,C1(C(N2CC(N(C(c3ccc(C)cc3)=O)CCO)C2)=O)CC2CCC(C1)C2(F)F 50828,Cc1cc(C)c(C(N2CC=C(CNC(=O)CC3CCOC3(C)C)CC2)=O)cc1N 50829,N1(C(C2(C)C=CCC2)=O)CCN(C(c2onc3ccccc23)=O)CC(O)C1 50830,C(=O)(CC1CCCc2ccccc21)N(CCNC(C(CC#C)C)=O)C1CC1 50831,c1(C(N2CCC(NC(CC(CC)C3CC3)=O)C2C)=O)cc2n(n1)CCNS2(=O)=O 50832,CC(C)CC(CN(C)C)N=c1nc2c(ncn2C)c(NCCc2c[nH]c(=N)s2)[nH]1 50833,c1(C(=O)NCC(C(=O)NC(CCC)C)N2CCOCC2)ncccc1C 50834,c1(SCC)nc(C(=O)NC2CC(C)N(C(=O)CCSC3CCCC3)C2)cc(=N)[nH]1 50835,CS(=O)(=O)CCC(=O)NCCCC1CCCN1C(=O)CCc1cncc(F)c1 50836,N1(C(C(C)N(CC)CC)=O)CC(NC(C2CN(C(=O)N(C)C)C2)=O)C2(CCC2)C1 50837,c1(C(C)O)ccc(C(=O)N(C2CCC(NC(=O)CC3CCCCO3)CC2)C)cc1 50838,C1(C(N2C(CNC(c3cn(-c4ncccn4)cn3)=O)CC2)=O)CCc2nncn2C1 50839,C1(NC(C2(OCC)CCOCC2)=O)CC2CN(C(C3CCCCC3C)=O)CC2C1 50840,Cc1c(CN(C(=O)CCCCNC(c2ccncc2)=O)C)cnn1C 50841,C#CCCC(=O)N(CCC(=O)NC1CCOC1=O)CCCO 50842,Cc1ccc(NC(C2CCCC2CNC(c2ccc(CO)s2)=O)=O)c(C)n1 50843,C1(CC)(CNC(C2CC(O)(CNC(=O)C(C)C3CCC3)C2)=O)CCCC1 50844,C12(C(=O)N(CCC3(NC(c4cc(CCC)on4)=O)CCC3)CC)CCCN1CCC2 50845,C(CCC(C)C(=O)NCCCCC(=O)NC1CCN(C)C1=O)OC 50846,Cc1c(Cl)sc(Cl)c1C(=O)N(CCCN(C)C(c1cccc(=O)o1)=O)C 50847,Cc1cc(C(=O)N(CC(=O)NCC2CC(O)C23CCC3)C2CCC2)cnc1O 50848,N1(C(C(C)(C)CCl)=O)CCOC2(CCN(C(=O)C(O)O)C2)C1 50849,Cc1cc(C(F)(F)F)nn1CC(=O)NCCC1CCN(C(c2cncs2)=O)C1 50850,N1(C(C(C)NC(=O)C2CC2)=O)CC(C)(C)CC1CNC(=O)CC1(C)CC1(F)Cl 50851,C1(CC)C(C(N2CCC2(C)CCO)=O)CCN1C(=O)Cc1ccc(C)o1 50852,C1(CNC(C2(CC=C)CCCC2)=O)CN(C(=O)Cc2ccnc(O)c2)CCN1C 50853,C1(C2CCCO2)(C(=O)NCC2CC(C)N(C(c3ccncc3F)=O)C2)CCCO1 50854,C1(NCc2c(C)ncs2)CCN(C(=O)CC2(O)CCCC2)CC1C 50855,C(=O)(CC(=O)NCCC1(C(=O)NCCC(O)CO)CCCC1)N(C)C 50856,C(=O)(CC(O)C(=O)N1CC2CC2(CNC(c2coc(Cl)c2)=O)C1)OC(C)(C)C 50857,Cc1cnc(C(=O)NC2CC(F)CN(C(=O)C3=CCCCC3)C2)cc1C 50858,N1(C(CCC(C)(C)NC(=O)C=Cc2ccccn2)=O)Cc2ccccc2C1 50859,C1(CCNC(CN(C)CCO)=O)CC(F)(F)CN1C(c1cccnn1)=O 50860,c1(C(=O)NCCCN(C)C)ccc2c(c1)CN(C(=O)C(=O)NCC(F)F)C2 50861,C1(NC(C(C)=C2CC2)=O)CN(C(c2nn(C)nc2C(F)(F)F)=O)CCC1C(F)(F)F 50862,C(=O)(CCCCCC(C)O)NC1C=CCN(C(C(CC(C)C)O)=O)C1 50863,C1(C(=O)NCCCCNC(c2cn(C)nc2O)=O)CS(=O)(=O)CC1C(F)(F)F 50864,C1(C#N)(C(N2CCCC(NC(c3nc(OCC)sn3)=O)C2)=O)CCCOC1 50865,CN1CC(C(N2CCC(F)(C(=O)NCCC(F)=C(F)F)C2)=O)CC1=O 50866,C1(NC(c2nc(C)n(C)c2)=O)CCCC(C(=O)N(CC(Cl)Cl)C)CC1 50867,CC1CN(C(c2ccc([N+](=O)[O-])[nH]2)=O)CCC1NC(=O)CC12CCC(CC1)CC2 50868,c1(CC(=O)NC2CCC2CNC(c2ccncc2)=O)ccc(F)cc1C(F)(F)F 50869,c1(C(N2CC3C(NC(C(CC=C)OC)=O)C3C2)=O)coc2ccc(OCC)cc12 50870,CCC(CC)CC(F)C(=O)NCc1cc(C(=O)N(CC(O)C(F)(F)F)C)cs1 50871,c1(C(=O)NCCc2ccc(C(=O)O)s2)cnc(O)c2ccsc12 50872,C12CCC(CC1)NC2=O.C(=O)(C(C)=O)N(C1CCCC1)CC 50873,N1(C(C(C)=C2CCCC2)=O)CCN(C(c2cc([N+](=O)[O-])c[nH]2)=O)C(C)C1C 50874,C1(NC(CC(C2CC2)NC(C)=O)=O)CCCC(CNC(=O)C=C(C)C(C)(C)C)C1 50875,C(CC(C)C(=O)N(CCNC(c1cnc(O)o1)=O)C1CC1)=CCC 50876,C1(CCC)CN(C(=O)C(CC(C)C)NC(N)=O)CCN1C(=O)C=CC=C(Cl)Cl 50877,CC(CCNC(=O)C(C)Cc1ccco1)CCNC(=O)CCc1cn[nH]c1 50878,N1(C(C2CCCC(C)C2)C(=O)NCC=C)CCC2(CC1)CCN(C)C2=O 50879,C1(NC(=O)NC(C(C)C)c2cccs2)CCCCCN1C(c1ccccc1)=O 50880,C(C)(CN=c1ccn2ncc(S(=O)(=O)NCc3ccccc3Br)c2[nH]1)OCC 50881,c1(OC)cnc(C(N2CCCC(NC(=O)CC3CN(C)C3)CC2)=O)c(OC)n1 50882,C1(NC(COCCC)=O)CC2(N(C)C(C3CCN3CC)=O)COC1C2 50883,C(C)(CO)(C(=O)NCCC(C)F)NC(C(C)OCCC#C)=O 50884,C#Cc1cc(C(=O)NC2CC(CNC(c3ccccc3C#N)=O)C2)cc(F)c1 50885,CCC1=NOC(C(=O)NC(CNC(=O)Cc2ccn(C)n2)CO)C1 50886,c1(C(N2CC(CCCCNC(C3(O)CC4CCC3C4)=O)C2)=O)cc2sccc2s1 50887,C1(OC)CC(NC(c2cc(C)nn2C)=O)C12CCN(C(c1scnc1C)=O)CC2 50888,c1(CC)cc(CNC(c2ncc(C)s2)C)cc(Cl)n1 50889,CC1(NC(=O)CC2CC(F)C2)CCC(NC(c2ncoc2C(C)(C)C)=O)CC1 50890,CC1CC(CNC(=O)CCCc2cnn[nH]2)CCN1C(=O)CC1CCCO1 50891,c1(C(=O)NCC2CCN(C(=O)C=Cc3cnc[nH]3)C2)coc2c1CSC2 50892,c1(C(=O)NCC2CC2NC(C2CCC2)=O)ccc2nc(O)nc(O)c2c1 50893,N1(C(C(COC)OC)=O)CCC(CCC(C)(C)NC(c2cnc(S)[nH]2)=O)CC1 50894,C1(C(=O)NC(c2cccc(NS(C)(=O)=O)c2)C)CCS(=O)(=O)C(C)(C)C1 50895,N1(C(CCOC)=O)CCCCC(N(C(=O)CC(C(C)C)c2ccccc2)C)C1 50896,Cc1cc(C(=O)NCC(C)N(C(=O)CCc2cccc(O)n2)C)c2n[nH]cc2c1 50897,Cc1c(O)ccc(CNC2CC(C(=O)Nc3conc3C)C2)c1O 50898,O=C(CC(C(F)(F)F)NC(=O)NCc1ccccc1)NC1(C2CCC2)CC1 50899,N1(C(CC(C=C)(C)C)=O)CCN(C(=O)CCCN(C)C)C(C)C1C 50900,C(=O)(C(C(C)CC)NC(c1ccc(SC)o1)=O)NCCSCCC=C 50901,c1(CC)c(C(=O)NC(CNC(=O)COCC2CCCO2)CC2CC2)cccc1F 50902,CN1CCC(C(=O)NCc2nc(CNC(=O)C3=CCCC3)cs2)S1(=O)=O 50903,Cc1cnc(NCC2CCCCC2NC(C2(O)CCOCC2)=O)nc1O 50904,C1(Cc2ccc(C(C)(C)Cc3ccccc3)s2)CC2(C(=O)O)COC1C2 50905,N1(C(COCc2cccc(C)c2)=O)CCC(NC(=O)CCOC2COC2)C(O)C1 50906,N1(C(c2n[nH]c(C)c2Cl)=O)CCC(O)(CN(C)C(C2CCC(C(N)=O)C2)=O)CC1 50907,CC(C)C(C)C(CNC(=O)C=Cc1ccoc1)NC(=O)CCCCCN(C)C 50908,c1(C(=O)NC(CNC(C(CCCC)CC)=O)CO)cccc([N+](=O)[O-])c1OC 50909,CC(C)C(C(=O)NC1CCN(c2ccnc(Cl)n2)CC1)c1ccc(-c2nn[nH]n2)cc1 50910,C1(CNC(CCc2cc(C)on2)=O)CC2CN(C(=O)C3=CCCO3)CC12 50911,C1(C(N2C(CNC(CC3CC(=C)C3)=O)CC(C(F)(F)F)C2)=O)CCCCC(=O)N1 50912,C12(NC(C3C(CCOC)C3)=O)CC(COC)(CN1C(=O)COc1cnn(C)c1)C2 50913,C1(C2CCOCC2)(C(=O)NC2C(NC(C(C(C)C)NC(COC)=O)=O)CCC2)CC1 50914,C(=O)(C(O)CC(C)(C)C)NC1CCC(CNC(c2cc(C)[nH]c2)=O)C1 50915,C=C1CCN(C(c2nonc2N)=O)C(C(=O)Nc2cnc(F)nc2)C1 50916,C(=O)(CC1=CCCC1)OC(C(C(=O)OCC)=O)C 50917,c1(C(N2CCC(N(C(c3cscc3OC)=O)CC)C2)=O)oc(C)nc1C 50918,C(c1cc[nH]c1)=CC(=O)N(CC(C)NC(c1cn(CC2CCCOC2)nn1)=O)C 50919,c1(OCC)cccc(NC(c2sccc2CNC(=O)COCCC(C)C)=O)c1 50920,N1(C(C(C)=C2CCC2)=O)CCC(NC(c2cc(C(F)F)ccn2)=O)CC1C 50921,C(C(=O)N1CCCN1)NC(C1CC2CCC1C2)=O 50922,CC1CCN(C(c2cccc(F)c2O)=O)CCN1C(c1cc2c[nH]nc2s1)=O 50923,N1(C(c2ccc(CC)o2)=O)CCC(O)(C2CCN(C(c3cnns3)=O)CC2)C1 50924,N1(C(CC2CN(C(CC3(C)CC3)=O)CC23CC3)=O)CC2CCC(O)C(O)C12 50925,C(C(C)(CC(C)C)NC(c1csnn1)=O)NC(c1c(C)cc(C(F)(F)F)s1)=O 50926,C1(CNC(C2(C)CCCC2)=O)CCN(C(=O)Cc2ccc(O)c(Cl)c2)CC1(F)F 50927,C1(CNC(c2ccc(CC)cn2)=O)CCC2(CCC2)C1NC(=O)C=C1CCC1 50928,CC(C)CC(CNC=O)CC(=O)NC1CCCN(C(=O)C=CCN2CCCC2)C1 50929,N1(C(CCCc2c(C)nc[nH]2)=O)CC(C)C(NC(=O)C=CBr)C(C)C1 50930,c1(C(=O)NC2(C3N(C(COC)=O)CCC3)CC2)ccc(OCC(C)(C)C)cc1F 50931,C(=O)(C1COc2ccc(Cl)cc21)N1CCC(CN(C)C(C2CC3CC3C2)=O)C1 50932,c1(C(N2C(C)(CNC(c3cnc(SC)[nH]3)=O)CCC2)=O)cccc(N)c1O 50933,C(=O)(C(F)(CNC(=O)C(C#N)C(C)(C)C)C(C)C)N(CC(C1CC1)OC)C 50934,CC(C)C(F)C(=O)NCCC1CCC(NC(=O)CC2CC=CC2)C1 50935,N1(C(C(CC=C)C)=O)CCC(C2CCN(C(=O)C(C)(C)CC(C)=O)C2)CC1 50936,C1(NC(=O)CSc2nc[nH]n2)CCCC(NC(c2c[nH]cc2Br)=O)C1 50937,C1(NC(C=C(COC)C)=O)CN(C(c2cc(CC(C)C)c[nH]2)=O)CC1N=[N+]=[N-] 50938,c1(C(=O)NCC(C(C)C)NC(C2COCCO2)=O)sc(N2CCOCC2)nc1Cl 50939,c1(OCC(N2CCC(N(C(=O)CC34CC(C3)C4)CC)C2)=O)cc(Cl)ccc1Cl 50940,C=Cc1ccc(C(=O)NC(C2(O)CCN(C(=O)CSc3nncs3)C2)C)cc1 50941,c1(C(=O)NC23CCN(C(=O)C(N4CCOCC4)O)CC2C3)ccc(Cl)cc1Cl 50942,N1(C(=O)Nc2ccc(-c3ccco3)cc2)CC2(CCN(S(=O)(=O)c3ccc(Br)s3)C2)C1.C1CCCCC1 50943,c1(OC)cc(CN2CCNCC2)ccc1I.c12ccc(nc1)[nH]2 50944,c1(CC)nn(C)c(Cl)c1C(=O)NCC1(O)CC(CNC(=O)C2=C(Cl)CC2)C1 50945,CCC(C)C(C)C(=O)NCC12CC(NC(=O)Cc3ccc(C(=O)OC)cc3)(C1)C2 50946,c1(C(N2CC(O)(C(C)NC(CNC(=O)OCC)=O)C2)=O)cnc2c(c1)CCOC2 50947,Cc1ccc(-c2cn(C3CCN(C(=O)CC(=O)N(C)C)CC3)nn2)cc1N 50948,NS(=O)(=O)c1ccc(C(=O)NC(CNC(C2CCCO2)=O)CO)o1 50949,C1(C(N(C)C)=O)(NCCN(C(=O)CCCF)C(c2cccc(F)c2)=O)CCCCC1 50950,c1(C(N2CCN(C(=O)Cc3nc[nH]n3)C(CO)C2)=O)nc(Br)c2n1CCCC2 50951,C1(C(=O)NCCC(=O)NCC)CC2(CCN1C(c1cn(C)nn1)=O)CC2 50952,C1(CNC(N(CCNC(=O)OC(C)(C)C)CC)=O)CCCC1 50953,c1(C(N2C(C)(C)CC(NC(=O)C(O)C3CC3)C2)=O)cc(N)cc([N+](=O)[O-])c1 50954,c1(C(=O)NC(CCNC(C2CC(C)(CC)C2)=O)C)cc(C#N)c(F)cc1F 50955,N1(C(COC(C)=O)=O)CCOCCC1C(=O)N(C)CC1CCN(C)CC1 50956,CCCC(C(=O)OC)C(=O)NC1COCCC1NC(c1ccc2n[nH]cc2n1)=O 50957,c1(C(N2CCCC(NC(CCOCCOC)=O)C2C)=O)cc2c(s1)CCC(C)C2 50958,CCCCC(O)CC(=O)NC(CC(F)F)C(=O)N1CCOC2CC12 50959,N1(C(c2c(CC)csc2)=O)C(C(=O)NCCOC(C)=O)CCC12CC2 50960,C1(C(=O)OCC)CN(C(C)=O)CC1(F)F.C12(CC=CCC1)NC2 50961,c1(OCCCC)ccc(Cl)cc1NC(N1CCC(C)C1(C)C)=O 50962,CC1CN(C(C(=O)NCC2CC2)C(C)CC2CCCCC2)CC(C)(C)C1 50963,c1(OC)ccccc1N(C)C(c1n[nH]cc1CNC(=O)C(N1CCNC1=O)C)=O 50964,C1(NC(CCc2cc(C)no2)=O)(CO)CCCN(C(C2CC23CC(C)(C)C3)=O)C1 50965,N#CC1(C(=O)NCCc2ccc(Br)cn2)CC12CCCC2 50966,N1(NC(C(C)C)CNC(=O)OC(C)(C)C)CCN(CCCC(C)(C)C)CC1 50967,c1(N(CC(CCC(=O)NCc2cc(C)c(C)[nH]2)C)C)ncc(Cl)cc1Cl 50968,N1(C(c2ncn(CC)c2)=O)CCN(C(=O)C(F)(F)C(F)F)CC1CO 50969,N1(C(c2n(C)cnc2)=O)CCCC2(CCC(NC(c3coc(Cl)n3)=O)C2)C1 50970,C=C(C)CC(C(=O)NC(COC)CSC)NC(=O)CN1CCOCC1=O 50971,N1(C(=O)Nc2cccc(N3CCNC3=O)c2)CCN2C3CCC(C3)C2C1 50972,C1(CC)CN(C(C2(NC(=O)C(CC3CCC3)OC)CCOCC2)=O)CCO1 50973,C(CC(=O)N1CCCC1CN(C)C)(C(F)F)NC(C1N(C)CC(F)C1)=O 50974,CCCS(=O)(=O)CC(=O)NC1CN(C(c2ccc(O)nc2)=O)CC1CO 50975,C1(C)(NC(C2(NC(CC=CCC)=O)CC(O)C2)=O)CCC(C)C1 50976,c1(C(=O)NCC(F)CNC(C2CC(F)C(=O)N2)=O)cc2cccc(O)c2[nH]1 50977,c1(N2CC3C(NC(c4ccc(S)cc4)=O)C3C2)ncnn2cccc12 50978,N1(C(c2sc3ncn(C)c3c2)=O)CCC2CCN(C(c3cccc(O)n3)=O)C2C1 50979,C=C1CC(CN(C(C(=O)OC)C2CN(C(=O)NC(C)(C)CC)C2)C)C1 50980,CCCS(=N)(=O)c1cccc(SCc2cccc(C#N)c2F)c1 50981,C=CC(CC)CC(=O)N(C1CCCC1)CCCNC(C12CCN(CC1)CC2)=O 50982,C=C(C)CCCC(=O)N1CC=CC(NC(C2(Cc3cccc(F)c3)CC2)=O)C1 50983,C1(C(N2C(C)CCC(NC(CN(CCOC)C)=O)C2)=O)CC2(C1)CC1(CCC1)C2 50984,CC1(C)CN(C(=O)C2=CCOC2)CC(C)(C)C1NC(C1CC2(CCC2)CO1)=O 50985,c1(C(=O)NCC(C)N(C(COCCCCC)=O)C)[nH]c(C)cc1C 50986,N1(C(C(C#C)(C)C)=O)CCN(C(=O)CC2CCN(C)C2)C(CCC)C1 50987,C(C(COC)C(=O)N1CC(C)(CCC(=O)NC2CC(OC)C2(C)C)C1)OC 50988,C(C(=O)NCCCCC(C)C)(C(C)C)NC(CCCNC(C)=O)=O 50989,Cc1cc(C(=O)NCC(C)NC(=O)C(c2cscn2)N(C)C)c(N)c(C)c1 50990,CC1CC(NC(=O)CC(C)(O)C2CC2)CN1c1nnc(-c2ccccc2)s1 50991,c1(CC)ccc(C(=O)N(CC(C)NC(=O)Cc2ccsn2)CC)cc1 50992,C1(O)(CC(=O)NC2C(C(=O)NCC(C(=O)OC)O)CCC2)CCCCC1 50993,CC1(C)C(NC(C2(Br)CC2C(=O)O)=O)C(C)(C)C1O 50994,C=CC(CC(=O)N(c1ccccn1)CCNC(=O)COCC)c1ccccc1 50995,Cc1ccnn1C(C)C(=O)NC1CCCCC1.C12CC(C1)CNC2=O 50996,c1cn2c(n1)C(NCC1CCNC3(CC3)C1)CCC2 50997,N1(C(c2cn(C3CCC3)nn2)=O)CCN(C(=O)CN2CCCS2(=O)=O)C2CCC12 50998,C(CC)(C(=O)NC(C1CN(C(=O)CC2CC2C)C1)C)=CC 50999,N1(C(c2c(C)noc2N)=O)CCN(C(C2CCC(=O)N(C(C)C)C2)=O)C(C)C1 51000,c1(OC)cccc2c1CCCC2NC(=O)C(=O)NCC(c1ccc(F)cc1)(F)F 51001,c1(NC2CC(NC(C3C(OCC)C3C)=O)C2)ncc(C(N)=O)cc1Cl 51002,c1(C(=O)NCC(CC(C)C)NC(CC2CC(CC)C2)=O)c(F)cncc1Br 51003,c1(C(=O)NCC2CCN(C(C(CC=CC)C)=O)C(C)C2)cn2ccccc2n1 51004,c1(CCCNC(c2ccccc2)CC)ccccc1Br 51005,C1(C(C)C)CN(C(C2CNC(=O)C2)=O)CCN1C(=O)CCc1cnc[nH]1 51006,c1(CCCC(=O)NCC2CC(OC)CN2C(=O)C(F)F)c(F)cccc1F 51007,N1(C(COCCC)=O)CCN(C(=O)CCc2cc(C)n(C)n2)CC2(CC2)C1 51008,CCCCCCC(CC)(c1nnnn1CCOC)NCc1ccc([N+](=O)[O-])o1 51009,N1(C(COCC)=O)CCC(N(C(c2ncoc2C)=O)Cc2cccnc2)CC1 51010,C(Nn1cncn1)c1nc(-c2ccccc2)no1.n12ccnc1C(=O)C2C 51011,c1(C(N2C(C(=O)Nc3ncncc3Cl)CC(F)C2)=O)c(F)cccc1F 51012,C1(C(=O)NCC2(C)CCN(C(c3cnco3)=O)C2)(CC)CNC(=O)C1 51013,c1(C(=O)NC2CN(C(c3nc(C)nn3C)=O)CC2C)cnn2ccn(C)c12 51014,Cc1cccc(C(C)(C)C(=O)NCCN(C(=O)C(F)CC2CCC2)C(C)C)c1 51015,C#CC(N(C)N(C)Cc1ccc(-c2ccc(F)cc2)cc1)c1ccccc1 51016,Cn1cc(S(N)(=O)=O)c(C(=O)NC2CC(C)(NC(=O)CC3CCC(=O)N3)C2)n1 51017,CC(C)(C)C(CO)C(=O)N1CC2CC1C2NC(=O)CCCOC1CCOCC1 51018,CCCC(C)(CC)C(=O)NCC(C1CCC1)NC(c1cnc(OCC)c(Cl)c1)=O 51019,N1(Cc2nnc(CCC)s2)C2CCC1CN(C(c1ccnn1C1CCC1)=O)CC2 51020,Cc1c(C(=O)N(C)CCOCCCNC(C2(O)CC(F)(F)C2)=O)cccc1F 51021,N1(C(C(C2CCCC2)OC)=O)CC(=O)NCC1C(=O)NCCC(F)=C(F)F 51022,N1(C(CC(=C)C)=O)CCN(C(=O)COc2ccccc2C#N)CC1C1CC1 51023,C1(C(=O)NC2(CC=C)CCN(c3ncccc3C(C)=O)C2)CCOC2(CCC2)C1 51024,c1(OC(C)C)ccc2c(c1)CCN(c1nccc(=NCC3CCOCC3C)[nH]1)C2 51025,C=CCC(C)(O)C(=O)NC1CCC1C(=O)N(C1CC(C)(C)C1)C 51026,CCCC(CCC)C(=O)N(CC(C)C(=O)NC1CCCC(OC)C1)C 51027,c1(C(N(CC(CC)NC(c2c(OCC)cccn2)=O)C)=O)c(OC)cccc1C 51028,c1(CC)oc(C(=O)NC2CC(CNC(C3CC34CCC4)=O)C2)cc1C 51029,C(C)(C)(CCC(=O)NCCC(=O)OC(C)C)NC(C1(OC)CCC(C)C1)=O 51030,C1(CC)CC(C(=O)N(C2CCC2C)C)CCN1C(c1nn(C)cc1Cl)=O 51031,N1(C(C2=NOC(C)C2)=O)CCC(C2(NC(=O)C=Cc3nccs3)CC2)C1 51032,C1(OC)CN(C)CC1NC(=O)C(C1CCCC1)NC(C1CC1(C)C(F)F)=O 51033,C(=O)(CCCC(C)=O)NCC(CC=C)NC(=O)C=Cc1ccco1 51034,CC1(C)CCCC(C(=O)NCC2(O)CN(C(C3C4CCCCC34)=O)C2)C1 51035,C1(C(N2CC(N(C)CCO)C2)=O)(COC)C=CCN1C(C1C2CCCOC12)=O 51036,C(=O)(C(CC)C(C)C)N1CC(C=C)(CC(=O)NC(CO)CC=CC)C1 51037,N1(C(C(COC(C)=O)C)=O)CCC(C(=O)NCCNC(=O)C(C)C)CC1(C)C 51038,c1(C(=O)Nc2nc(CC(C)C)[nH]n2)c2c(cc([N+](=O)[O-])c1[N+](=O)[O-])OCCO2 51039,N1(C(C=CC(C)(C)SC)=O)CCN(C(C2CC2c2cccs2)=O)C(CCOC)C1 51040,CCCC(C(=O)N(CCCN(C(=O)CCc1cc(C)sc1C)C)C)NC(N)=O 51041,Cc1nn(C)c2[nH]c(=NCCC3CC3NC(C3CC34CC4)=O)c(C#N)cc12 51042,CC1COCCC1NC(=O)C(=O)N(CCCC1CC2CCC1C2)C 51043,CN1CCC(CCNC(=O)CC2C=CC(NC(c3cncn3C)=O)C2)C1 51044,Cc1cc(CC(N2CC(NC(=O)C=Cc3cc[nH]c3)C(C(F)F)C2)=O)ccn1 51045,C12(C(=O)NCC3C(C)(C)N(C(C4CCCOCC4)=O)CC3)CCC(N=[N+]=[N-])C1C2 51046,Cn1nnc2cc(C(N3CCC(CCNC(C4CCCC(F)(F)C4)=O)C3)=O)sc12 51047,C1(NC(c2c(COC)noc2)=O)C2CCN(C(C3CC4(CC4)C3)=O)CC12 51048,c1(CC)ccc(C(=O)N(CCNC(C2(C(F)(F)F)CCC(F)C2)=O)C2CC2)cn1 51049,C1(C(N(CCCNC(C(n2ccc(C)n2)(C)C)=O)C2CC2)=O)C(Cl)(Cl)C12CC2 51050,N1(C(C=COCC)=O)CC(NC(=O)CCC2CCCCN2C)CC(C)(C)C1 51051,C(=O)(CCCCCCC(=O)OC)NC1CN(C(CC=CC)=O)CC(F)C1 51052,Cc1ncc(C(=O)N(C)CC2(NC(=O)C3=COCCC3)CC2)c(Br)c1Cl 51053,Cc1cccc2c1OC(C(=O)NC1CN(C(c3ccon3)=O)CC1C)C2 51054,C1(C(N(CCNC(c2ccc(OC(C)C)nc2)=O)CC)=O)CCC(F)(F)C1O 51055,C(CN=C(NCC(C)C)NCC1CCN(S(C)(=O)=O)CC1)c1ccc(OC)cc1 51056,C1(NC(Cc2c(C)ccc(F)c2)=O)CCCC12CN(C(C1NC(=O)C3CC13)=O)C2 51057,CC(CC(=O)N1CCN(C(=O)C=C2CCOCC2)CC1)C(C)(C)C 51058,c1(C(=O)NCC2(OC)CN(C(c3nocc3C)=O)C2)n[nH]c(C(C)C)c1Br 51059,NS(=O)(=O)c1n[nH]cc1C(N1CC2CCC1C2NC(=O)Cn1cnccc1=O)=O 51060,CCCC(CCC)C(=O)NCc1occc1C(=O)NC1CCOC1C1CC1 51061,c1(C(=O)NC2CN(C(c3ccc(C(C)C)o3)=O)C3C2C3)cc(F)cc(F)c1 51062,c1(OC)ccncc1C(=O)NC1CCN(C(C2CC2C)=O)C1C 51063,c1(C(=O)NC(CNC(C2C(C)CC2)=O)(C)C)ccc(C(F)F)cc1Cl 51064,C(CN=c1ccc(Br)c(S(=O)(=O)NCc2c(F)cc(Br)cc2F)[nH]1)C1(C)CC1 51065,Cc1ccc(SCC(=O)NCC2CC(O)(CNC(=O)C(C)NC(N)=O)C2)c(Cl)c1 51066,CC1CN(C(C2C(F)(F)C23CCC3)=O)CCC1CNC(=O)CC1OCCC1(C)C 51067,C1(OC)CCC(C(=O)NC(C)CNC(c2sccc2C(C)(C)C)=O)CC1 51068,C(C)(C)(C(=O)NCCCC1(NC(=O)CC2CC(F)C2)CC1)OCC 51069,C1(C(=O)NC2CCCN(C(Cc3n(C)nc(C4CC4)c3)=O)C2)C2CC3C(C2=O)C13 51070,CC1OCCC1(O)CNC(C1(NC(C2CNC(=O)N2)=O)CCCCC1)=O 51071,N1(C(CN2CCC(C)C2)=O)CC2CCC1CN2C(=O)C(C1CCCCC1)O 51072,CCCCCC(=O)NC1CN(C(c2cnn(C(C)C)c2C)=O)C2CC12 51073,CC1CN(C(c2ccn(CCN(C)C)n2)=O)CC(C)N(C(=O)C(C)C2CC2)C1 51074,c1(C(C(=O)NCC=C)N(C2CCN(CC)C2)CC)cnn(C)c1Br 51075,C(=O)(C1CCc2c[nH]nc21)N1CCC(C(C)NC(c2cnsc2)=O)CC1 51076,C1(C(N2CCC(C#CC)C2)=O)N(C(=O)Cc2ccc[nH]2)CCCC1(C)C 51077,C#CCC(CC#C)C(=O)OCC1CCCC1c1ccccc1 51078,CC(C(=O)N1CC(NC(C2CNC(=O)N2)=O)C(C)C1)C(C)c1ccccc1 51079,c1(C(CC)C)ccc(C(c2nnnn2C)NCCc2csc(C)n2)cc1 51080,C(C(=O)NCCC(C)(C)NC(=O)Cc1c(Cl)cnn1C)(C(C)C)n1ccc(C)c1 51081,C1(C2CCN(C(C3(C)CC3C(F)(F)F)=O)CC2)(C(=O)OC)CC(F)(F)C1 51082,N1(C(C2(CNC(C3C=CCC3)=O)CC2)=O)CCN(c2ccccc2)C(=O)C1 51083,c1(C(N2CC(CNC(c3ccc(SC)cc3)=O)C3C2C3)=O)cncc(Cl)c1C 51084,Cc1ccc2c(=NC(C)C3CSC3)[nH]c(=NCc3c(F)ccc(F)c3F)[nH]c2c1 51085,CC1CN(C(c2cccc(C(N)=O)c2)=O)CCCN1C(c1ccns1)=O 51086,N1(C(CC(C)C(F)F)=O)CCC2CCCC12C(=O)NC(C1CCC1)C1CC1 51087,CCC(CO)(C(=O)NCC1(CNC(=O)COC2CC=CC2)CC1)OC 51088,c1(-c2nc(C(N3CC4(CCC4O)C3)=O)sc2)ccc(O)cc1Cl 51089,C12(C(=O)NC3CC(CNC(c4ncc(OC)cc4F)=O)C3)CCCCC1OCC2 51090,C#CC1CC2CCC1N(C(C1CCN(C(=O)CCC3CCCN3C)C13CC3)=O)C2 51091,Cc1ccc(CC(=O)N(CC(O)COCc2ccccc2)C)o1 51092,N1(C(c2c(C)nc(-c3cccc(F)c3O)s2)=O)CCCC2(CNC(=O)O2)C1 51093,c1(C(N(CC)CC2CCCN2C(C2OCCC2C(C)C)=O)=O)cccc(=S)n1O 51094,CC(C)(C(=O)NCCN(C1CCCC1)C(C1OCCOC1C(F)(F)F)=O)C(N)=O 51095,N1(C(CCC=C)=O)CCN(C(=O)C(c2ccccc2F)C)CC1CCO 51096,CCC(C)(COC)C(=O)N1CC(C2CC2C(N2CCOC(C(C)C)C2)=O)C1 51097,N1(C(CCP(C)(C)=O)=O)CC(CNC(=O)Cc2cccc(C#N)c2)CC12CCC2 51098,c1(OC)ccc(Cl)cc1CC(=O)N(C1CC(NC(=O)CC2(O)CCCC2)C1)C 51099,c1(C(N2CC(CC(=O)NC3CC4C=CC3C4)OCC2)=O)cc2n(n1)CCC2 51100,C1(CCC)CN(C(c2oc(C)cc2C)=O)CC1NC(c1ccsc1C)=O 51101,N1(C(CCC)=O)CCN(C(c2cc(C)nn2C)=O)C(CCO)C1 51102,C1(C(=O)NCC(CNC(=O)CN2CCS(=O)(=O)CC2)O)CC2C=CC1C21CC1 51103,c1(C(N2CCC(CNC(C(CC)O)=O)C2)=O)cc2ccccc2c(=O)n1C 51104,CC1CCN(C(C2CNC(=O)O2)=O)CCN1C(c1ccnn1CCF)=O 51105,N1(C(c2ccc(C(CC)=O)cc2)=O)CCN(C(c2coc(C)n2)=O)CC1C1CC1 51106,Cc1ccc(C(=O)NCCSCC(=O)NCC(C)(C)O)c(F)c1 51107,c1(OC)cc(C)sc1C(N1CC(OC)C(NC(=O)C=C2CCN(C)CC2)C1)=O 51108,N1(C(c2c(C)snn2)=O)CCCC(C(C)C(=O)Nc2ccc(Cl)cc2)C1 51109,C1(C#N)(C(N(CC(C(=O)NC(CCOC)CO)C)C)=O)CCCOC1 51110,N1(C(CNC(C(C)(C)C)=O)=O)CCC2CCCC12CNC(c1ccc(C(N)=O)s1)=O 51111,CCC(C)(C)CC(=O)N1CC(N(C(=O)C(C)OC)C)C(O)C1 51112,C1(CNC(C=CC=CCC)=O)CN(C(=O)C(=O)NC(C)C)CCC1C 51113,N1(C(CN(C2CC2)CC)=O)CCCN(C(=O)Cc2sc(S)nc2C)CC1C 51114,N1(C(C2CC(OC)CN2C(C2CCCCCC2)=O)=O)CC(C)N(C)C(C)C1 51115,N1(C(CNS(CCCC)(=O)=O)=O)CCc2nc[nH]c2C12CCN(C(=O)C(N)=O)C2 51116,c1(C(=O)NCCC(C)NC(CC=CC)=O)cnc2ccccn2c1=O 51117,Cc1ccc(C)c2c(C)c(C(=O)NCC3(NC(C4CSCC(=O)N4)=O)CC3)oc12 51118,c1(C(C(=O)NCCCCCN(C(=O)CCOC2CC2)C)F)ccc(F)cc1 51119,C1(CC(=O)NC(C(C)NC(c2ccsn2)=O)(C)C)CCC(=O)NC1=O 51120,c1(NC2CC(C)N(C(c3cc([N+](=O)[O-])c[nH]3)=O)CC2)ncc2c(c1C#N)CCC2 51121,C1(C)(C(=O)NC)C=CCN1C(C1CS(=O)(=O)C1)=O 51122,c1(C(N2CC(CNC(C(C)c3ccsc3)=O)C2)=O)ccc(-c2ccco2)o1 51123,N1(C(C2(COC)CC2)=O)CCC(N=c2ccc(C#N)n[nH]2)(CO)CC1 51124,Cc1cc(O)ncc1C(=O)N(CCCN(C(=O)CC1CCC(=O)N1)C)C 51125,N1(C(=O)CCCCn2cc(CO)nn2)CC2(COC(COc3c(F)cccc3F)C2)C1 51126,Cc1ccc(C(N2CCC(C)(C(N3CC(c4ncc[nH]4)C3)=O)CC2)=O)nc1C 51127,N1(CC)Cc2ccccc2OC(C)C1.C1(=O)N2CCC(CO2)CO1 51128,C1(CC=C)CCCN(C(=O)CCC2(C)CCN(C(C3(n4cccn4)CC3)=O)C2)C1 51129,Cc1ccc(C(=O)N(C)CCN(C(=O)C(C)N(C)C)C)cc1I 51130,c1(C(C)C)cc(C(=O)NC2CCN(C(c3ccc([N+](=O)[O-])[nH]3)=O)C2)cc(Br)c1 51131,C1(NC(=O)C=CBr)CN(C(=O)COc2ccsn2)CC(F)(F)C1 51132,CC(C)(CCNC(=O)C(O)C1CC1)NC(C1C(c2ccccc2)C1(F)F)=O 51133,C1(C2(O)CCC2)(C(=O)NC(C)C(CO)NC(C2CC3CC2CC3O)=O)CC1 51134,c1(CC)cnc(C(=O)NCC2(NC(C3CCC34CCC4)=O)CCCC2)cn1 51135,N1(C(=O)C(c2cccnc2)O)CC2CC(C(N3CCCC4CC34)=O)(C2)C1 51136,c1(C(N2C3C(NC(C(C(CC)CC)C)=O)C(C3)C2)=O)nc(N)cc2ccccc12 51137,N1(C(C(CC)(F)F)=O)CCC(C)C(NC(c2ccc(C(OC)OC)o2)=O)C1 51138,C1(NCC2CCCN(C(Cc3c(C)cccc3)C)C2)CCC2CC2CC1 51139,C1(CC=C)(NC(c2cc(Br)oc2C)c2nnnn2CCC)CCOCC1 51140,C1(NC(C(CC#C)O)=O)C2CCN(C(c3cnc(C4CC4)o3)=O)CC12 51141,c1(NC(C2C(C)C2c2ccccc2)=O)ccc(CCC(=O)O)cn1 51142,CC1(C)CN(C(=O)Cn2nnc(C3CC3)n2)CC1NC(C12CC(CO)(C1)C2)=O 51143,c1(C(=O)NC(CC=C)CNC(c2cnc(C)n2C(F)F)=O)cnc(CO)nc1C 51144,CCC(C)C(C(=O)NCC1COCCN1C)NC(C1CCC1(F)F)=O 51145,CCCC(O)CC(=O)NCCCN(C(=O)C(N1CCCC(O)C1)C)CC1CCCC1 51146,c1(-c2ccc(C(=O)NC(CNC(C3CCSC3)=O)CO)s2)cccc(F)c1 51147,C1(C(=O)NCC(CN(C(COCC(C)C)=O)C)C)CCC(N(C)C)CC1 51148,C1(C(N(CC(F)F)C)=O)CCCC1CNC(=O)Cc1ccn(C)n1 51149,C1(CNC(=O)CNCc2cnn(C)c2C(=O)NC2CCC2)CC2C=CC1CC2 51150,C1(CC(=O)NC2CC(N(C(CSCC(C)C)=O)C)C2)CN(C)CC1O 51151,O=C1NC(COc2ccccc2)C(=O)N1C1CC(=O)N(c2ccccc2)C1 51152,C1(C(N2C(C(C(=O)NCCn3ccc(C4CC4)n3)O)CC2)=O)CC2CCC1C2 51153,CC(=O)N=c1nc(C2CCN(C(C3CCN(C(=O)C(C)C)CC3)=O)CC2)[nH]n1C 51154,N1(C(c2ccc(OC)cc2C)=O)CCN(C(=O)C=CC=C(Cl)Cl)C(C)C1C 51155,C(C)(CCC(=O)NCCCCCO)NC(C1ON=C(C)C1)=O 51156,N1(C(C2CC2F)=O)CCC2(CCN(S(=O)(=O)c3ccc(O)cc3)CC2)C1 51157,c1(NC(=O)NC(C2CCOCC2)C)ccc(C#N)c(Cl)c1 51158,Cc1cccnc1C(=O)NC1CC1CNC(c1c[nH]nc1C1CCC1)=O 51159,C1(C(N(CC(C)NC(=O)C(C)(C)N(C)C)CC)=O)CCC(O)CN1C 51160,Cc1ccc(C(C)C(=O)NCc2nc(CNC(=O)CC3C=CCC3)cs2)cc1 51161,C1(C(C)NC(c2ccc(C)o2)=O)CN(C(=O)CC23COCC(C2)C3)CCO1 51162,c1(OCC)cc(NC(C2CCCC(CNCC3(C)CNC3)C2)=O)ncn1 51163,C1(C(=O)NCC2OCCN(CC)C2)CN(C(=O)C(CO)C(F)(F)F)CCC1(C)C 51164,C1(NC(CC=C)=O)CCC(C)N(C(c2cc(C)nn2CC)=O)C1 51165,N1(C(C(CC)(C)O)=O)Cc2nccn2CC(NC(C2SC3C=CC2CC3)=O)C1 51166,C1(NC(c2ccc(-c3ccccc3)cn2)=O)CCc2ncccc2C1 51167,Cc1nccn2c(C(N3CCNC(=O)C3(C)C(C)C)=O)cnc12 51168,c1(C(=O)NC(CNC(C(CC=C)C)=O)CO)cccc2[nH]c(C)cc12 51169,c1(N(C)Cc2ccc(C)o2)ccc(Br)c(S(=O)(=O)NC2CN(C)C3(CCC3)C2)n1 51170,c1(CC(N2CCC(N(C(c3cc(Cl)cs3)=O)CC)C2)=O)ccc(F)c(F)c1 51171,N1(C(C2CCN(CC)CC2)=O)CCCC(O)(Cc2nc(C3CC3)no2)C1 51172,N1(C(C(C=CC)O)=O)CCOC(CCCNC(C2(SC)CCC2)=O)C1 51173,C1(CC)COC(C)(C)CN1C(=O)C1=CCN(C(=O)CCC2CCCCO2)C1 51174,C1(CNC(COCCC)=O)CCCCC1NC(=O)Cc1ccc(Cl)s1 51175,C(=O)(C1=NOC2(CCC2)C1)N1CC(C)C(C(=O)NC2(c3nn[nH]n3)CC2)CC1 51176,N1(C(C(CC)F)=O)CC(C2CCCCN(C(C3CCc4n[nH]c(C)c4C3)=O)C2)C1 51177,c1(CC)cc(C(N2CC(Cc3ccoc3)C2)=O)nn1C.C1(=O)CC2(CC2)N1C 51178,C12CCN(C1(C)C)C2=O.C1(C(C)C)CCN(C(=O)Cc2nc(C3CC3)n[nH]2)CC1 51179,c1(C2C(NC(C3C(C(=O)O)NCC3)=O)C2)ccc(Cl)cc1 51180,c1(C(C)C)cnc(C(=O)N(C)CCOCCNC(=O)C(O)C(C)C)nc1 51181,C1(NC(C(COC)C)=O)CCS(=O)(=O)C12CN(c1nc(C(C)C)ncc1Br)C2 51182,c1(C(=O)NC2(COC)CCCN(C(=O)CC(C)(F)F)C2)ccc(C)c([N+](=O)[O-])c1 51183,C(=O)(C1=CCOCC1)N1CC(CCNC(=O)C(Cc2ccccc2)C2CC2)C1 51184,c1(C(=O)NC2(CO)CN(Cc3ncsc3Br)C2)cccc(C(F)(F)F)n1 51185,C1(NC(c2c(C)ccc(Cl)c2)=O)COC2(C1)CN(C(c1ccnc(Cl)c1N)=O)C2 51186,Cc1cccc(C(C)C)c1-n1nc(Cn2cncn2)nc1CCCC(C)(C)C 51187,C1(N(C(=O)CNC(C)=O)CCOC)CCN(C(c2n[nH]c(C(C)(C)C)n2)=O)C1 51188,c1(C(N2CC(C)C(NC(=O)Cc3cnn(C)c3)CC2)=O)ccn2nccc2n1 51189,C(C)(C)(CC(F)C(=O)NCC1CCOC(C)(C)C1)NC(C(C(=O)OC)OC)=O 51190,CN1CCN(C(=O)CN2CCCC2=O)CC1C(=O)NOCc1ccncc1 51191,C1(C(N2CC(O)(CNC(c3cnc(C4CCOC4)s3)=O)C2)=O)CC2(C1)CC2(F)F 51192,CCCC(C)(O)C(=O)NCC1CCC1NC(c1ccc(N)c(CC(C)C)c1)=O 51193,CC1CC(NC(=O)CC2CCN(C(C3CC(F)CN3)=O)C2)C(=O)O1 51194,N1(C(C(=O)NCC2CC(SCC)C2)=O)CCC(COC)C(F)(F)C1 51195,CN1CCC(C)(C(=O)NCCOC2CCN(C(=O)CSCCC(F)(F)F)CC2)CC1 51196,C=CC(CC)CC(=O)NCC1CCN(C(c2cc(C(F)(F)F)ccc2O)=O)C1 51197,c1(OC)c(C(=O)NCCCCCNC(c2c(Cl)cnn2C)=O)ccnc1Cl 51198,Cc1ccnc(O)c1C(=O)N(CCNC(C12CCCCC1C2)=O)C1CC1 51199,Cc1c(C(N2CC(F)(C(=O)NC3(C)CCCC3(F)F)C2)=O)cccc1O 51200,C=CC(C)(O)C(=O)N1CCCC(CN(C)C(c2sc(C)nc2C(F)(F)F)=O)C1 51201,[N-]=[N+]=NCCC(=O)NC1CCC(C(=O)NC2C3CCCCC23)C1 51202,C(CCCCC(=O)NCC1(O)CCN(C(=O)CCn2ccnc2)C1)NC(N)=O 51203,C1(C(=O)NC(C2CN(C(c3ncoc3-c3ccon3)=O)C2)C)C(C)(C)C1(C)C 51204,c1(OC)ccccc1C(CNC(C1CCC2CC12)=O)NC(C12CC(CO1)C2)=O 51205,C=CC1(CC(N2CCC(C)C2CO)=O)CN(C(c2nn(C)cc2C)=O)C1 51206,C(=O)(CC(C)CNC(=O)COC(C)=O)NC1(CC=C)CCOC1 51207,CCCS(=O)(=O)CC(=O)NCC(C)(O)CNC(C1CC2(CCC2)CO1)=O 51208,N1(C(c2c(C)nc(N)cn2)=O)CCC2(CCC(NC(=O)C#CC3CCOC3)C2)C1 51209,c1(CC)ccc(CC(=O)NCC2CC2NC(c2cc(=O)n(C)cn2)=O)cc1F 51210,C1(C(N2CC(CNC(c3ccc[nH]3)=O)C(F)(F)CC2)=O)CC2CCCCCCC12 51211,c1(C(N2CC(CNC(C(C=C)O)=O)OCC2)=O)ccc(C)c(S(=O)(=O)CCO)c1 51212,Cc1ccc2c(C(=O)N(C)CCN(C(=O)CC3CC(=O)C3)C)coc2c1 51213,N1(C(C(CC=C)CC)=O)CC2COCCC2(NC(c2cnc(Cl)s2)=O)C1 51214,c1(CNC(CC2OCCN(C(C3CC(C)(F)C3)=O)C2)=O)ccc(F)c(O)c1 51215,N1(C(CC(=O)OC)=O)CCC(C2(NC(c3cc(C)ccn3)=O)CC2)CC1 51216,C(C(CC)CO)NC(C1(C(C)NC(COCCC=C)=O)CC1)=O 51217,c1(C(N2C(CC(C(=O)NCCN3CCC(OC)C3)C)CCC2)=O)sc(C)nc1C 51218,CCCCC(O)CC(=O)NCC12CCCN1C2=O.c1(SCC)ccc(F)c(O)c1 51219,c1(CCC(=O)NCC(O)CNC(C2(F)CCCC2)=O)ccc2c(c1)OCO2 51220,C1(C)(C(=O)NCC(CNC(C2(CC#C)CCCC2)=O)O)Cc2ccccc2N1 51221,C1(NC(c2ccc(C(C)(C)C)cc2)C=C)CCCC2C1C2[N+](=O)[O-] 51222,CC1CN(CC2CCCC2N2CCOCC2)CCN1S(=O)(=O)Cc1ccccc1 51223,c1(OC)c(F)cc(Br)c(C(=O)NNC(=O)Cn2nc(C)cc2C)c1F 51224,c1(C(=O)NC2CC2NC(c2cnns2)=O)cc([N+](=O)[O-])c2nsnc2c1 51225,c1(OC)nccc(C(N2CC(OC)CC2)=O)n1.C(CN(C)C)(CO)NC=O 51226,Cc1nn(C)cc1C(=O)NCCCC1CCCN1CC(O)COCc1cccs1 51227,c1(C(=O)NC2CCC(NC(C(N3CCCCCC3)C)=O)C2)cncc(N)n1 51228,c1(N(C2CCCOC2)C)cc(Br)ccc1S(=O)(=O)NC1(C2CC2)CC1 51229,Cc1cccc(CN2CCC(C)(CN)C2)c1Br 51230,N1(C(C=NOC)=O)CCCCC1CN(C(=O)CCc1nccs1)C 51231,C(C(CC(=O)NC(CC1CC1)CO)NC(=O)C(C)c1cc[nH]n1)OC 51232,C1(CNC(CCNS(CC)(=O)=O)=O)COC(CNC(c2ccc(C)o2)=O)C1 51233,c1(C(N(CCCCNC(C(C(CC)C)O)=O)C)=O)cc2ncn(C)c2cn1 51234,CCC(CN(C)C)C(=O)NC1CN(C(=O)C(c2cccnc2)O)CC1CC1CC1 51235,C(=O)(C(F)C(C)(C)O)NCc1ccc(CNC(C2CCC(C)(C)C2)=O)cc1 51236,C1(C(NOC(C=C)C)=O)N(C(c2csnn2)=O)CCCC1(C)C 51237,N1(C(=O)CCc2ccccc2)CCC(C2CCCN(C(c3ccco3)=O)C2)C1 51238,Cc1sc(-c2ccccc2)nc1C(N1CC(Oc2ccccc2)C2(CC2)C1)=O 51239,c1(C(=O)NC2CC(CNC(C3(C)N(C)CC(O)C3)=O)C2)ccc2nc(=N)[nH]n2c1 51240,C1(NC(c2n(C)ncn2)=O)CC2CN(C(=O)Cc3c(Cl)cnn3C)CC12 51241,C#CC1CN(C(C2CCN(C)C2)=O)CCN1C(c1cc(F)n(C)n1)=O 51242,C1(C(N(C)CC2C(NC(C3CC(C(C)C)C3)=O)CCC2)=O)CCc2nc[nH]c2C1 51243,CCCCCCCCCCC(=O)N1CCCC(N(C(=O)C2=CSCS2)CCO)C1 51244,N1(C(c2ncn(CC)c2)=O)CCC(NC(=O)C(C)Cc2ccc(F)cc2)C(F)C1 51245,Cn1cc(C(=O)NC(C)(C)C(=O)NC(C)CC2(O)CCC2)nn1 51246,N1(C(CCOCC#C)=O)CC(CNC(c2c(NC(C)=O)c[nH]c2C)=O)CC1C 51247,c1(C(=O)NC(CC(=O)N2C(C)(C(=O)OC)CC2)COC)coc2c1COC2 51248,c1(C(=O)NC23CC(NC(C45CC(CCO4)C5)=O)(C2)C3)ccc(F)cc1C(F)(F)F 51249,N1(C(C(C)N(C)Cc2ccccc2)=O)CCC(O)C(C(N2CCCC23CC3)=O)C1 51250,C1(O)(CCNC(c2c(C)coc2)=O)CCN(C(c2cc(Br)c[nH]2)=O)C1 51251,N1(C(c2ccc(OC)cc2)=O)CC(C)C(C)(CNC(=O)CCCCSC)C1 51252,CCCC(O)C(=O)NCC1(CNC(=O)C(C)SC)CCCCC1 51253,CCC(C)(CCC(C)C)C(=O)N1CCOC(C(N2CCC(F)(F)C2)=O)C1 51254,c1(C(=O)NC2C(C#N)CN(C(c3ccno3)=O)C2)ccc2ccccc2n1 51255,CCC(CC(=O)NC(C(=O)NC(C)COC)c1cccs1)C(F)F 51256,C1(CNC(CN(CCC#C)C)=O)CN(C(=O)CC2CN3CCC2CC3)CC1(C)C 51257,N1(C(C(C)C2CCC2)=O)CCCC(C2CN(C(c3cccc(C4CC4)n3)=O)C2)C1 51258,N1(C(c2cccc(CNc3ccc(C)cc3)c2)=O)CCNc2cc(C)ccc2C1 51259,c1(C(N2CCC(NC(c3n(C)ccn3)=O)C(F)C2)=O)cncc2[nH]ccc12 51260,C1(CC(=O)OC)CCN(C(=O)C(C2CCN(CCC3CCCCC3)CC2)C)CC1 51261,C1(C(C)(C)C)CC(C(=O)N2CC(CNC(=O)CCc3cn[nH]c3)C(C)C2)=NO1 51262,c1(C(=O)NCC2(C(C)(C)C)CCN(C(c3c(C)ncs3)=O)C2)ccc(N)cc1Cl 51263,c1(C(N2CC=CC(NC(=O)C3=CCC3)C2)=O)ccc2c(=O)ccoc2c1 51264,Cc1ccc(C(N2CCC(CNC(=O)COC3(C)CCCC3)C2(C)C)=O)c(C)n1 51265,c1(C2C(C(N(C(C3CCOCC3)C)C)=O)C2)ccc2nsnc2c1 51266,c1(OC)cc(C(O)CN(C)Cc2ccc(Cl)cc2)ccc1O.N12CCC(CC1)C2 51267,N1(C(C2(NC(Cc3scc(C)c3)=O)CCCC2)=O)CCCN(C)C(=O)C1 51268,c1(CC)noc2ncc(C(N3CCN(C(C4CCC=CCC4)=O)C(C)C3)=O)cc12 51269,c1(C(=O)NC2CCN(C(C3OCCN(C)C3)=O)C2)ccc2c(n1)OCC(=O)N2 51270,S(=O)(=O)(C1CN(C(=O)NCC2CCOC2(C)C)CC1)NC 51271,C(=O)(C(C#N)C(C)C)N1CCC(C(C(=O)NC(c2nccn2C)CC)F)C1 51272,C(=O)(CCCCCNC(=O)C(C)C)OCC.C12CC1C(=O)NC(=O)CNC(=O)N2 51273,c1(NC(CC=C(C=C)COC)=O)cc(NC)ccc1C 51274,N1(C(c2c(CC)nco2)=O)CCOC(CCNC(=O)C(C)CF)C1 51275,c1(OC)cccc(C(=O)NC(C2CCN(Cc3cnc(C)s3)CC2)C)c1O 51276,C1(C(N2C(C(CNC(C(CSC)O)=O)(C)C)CCC2)=O)CN2CCN1CC2C 51277,Cc1nc(Nc2ccc(F)cc2F)ncc1-c1nc(C(F)F)nn1CCN(C)C 51278,C=CC(CCC)CC(=O)N1CCOC(C)C1C(N1CCC(OCC)C1)=O 51279,S(=O)(=O)(c1ccc(OC2CCOCC2)cc1C)N(C)Cc1c(CCC)cccc1 51280,N1(C(c2n(CC)nc(Br)n2)C(=O)NCC(F)F)CCC(C)(C)CC(C)(C)C1 51281,N1(C(C(CC)C)=O)CCc2nc(O)cc(C(=O)NC3CN(C(C)=O)C3)c2C1 51282,c1(OCC)cc(N)c(F)cc1C(=O)NC(Cc1ccnc(Br)c1)C(=O)O 51283,Cc1ccc(Cl)cc1C(N1CCC(n2cc(C3(NC(N)=O)CC3)nn2)CC1)=O 51284,C1(CC(=O)NCC=CCl)CCCCN1C(c1ccc(Cl)o1)=O 51285,C1(NC(CCc2c(C)cccn2)=O)CCN(C(C2(C)CCCC2)=O)CC1(C)C 51286,C(N=c1[nH]c(=N)[nH]c(=NC2CCN(CCF)C2)[nH]1)C1CC(CC)C1 51287,CC1C(NC(=O)Cc2cccs2)C(C)CCN1C(c1cnc2n1CCC2)=O 51288,C1(C(=O)OC)CC(CN)CN(C(=O)C(CC)(CC)OC)C1 51289,C=CC(C)(C)CC(=O)NCC1C2CN(C(=O)C=CC(c3cnn(C)c3)=O)CC12 51290,C1(F)(CNC(C2C(CC(C)C)C2)=O)CCN(C(C2CCN(c3ccccc3)C2)=O)C1 51291,N1(C(C(c2cn(C(C)C)nn2)C2CCCO2)=O)CCN(CC(F)(F)F)C(C)C1 51292,C1(O)(CN(C)C(c2ocnc2-c2ccccc2)=O)CCN(C(=O)CCC(N)=O)C1 51293,c1(NCC)cncc(C(=O)N(C)CCOCCNC(=O)CCc2cn(C)nn2)c1 51294,c1(OC)ccc2cc(C(=O)NC3CC(N(C(=O)CC(C)C(F)F)C)C3)[nH]c2n1 51295,c1(NCC2(COC)CC2)nc(N2CCC3(CC(=O)NC3=O)C2)nc2scnc12 51296,N1(C(C(COC)Cl)=O)CC2(C(N3CCNC(C)(C)C3)=O)CC1CO2 51297,c1(C(=O)NCC(C)CNC(=O)CC2CC3(CC3)C2)sccc1C#N 51298,C1(F)(CNC(COC(CC)C)=O)CCN(C(c2cc(F)ncc2OCC)=O)CC1 51299,C=Cn1nncc1C(=O)NC1CCC(NC(C2(CCC)CCC2)=O)C1 51300,c1(OC)cc(C)c(C(=O)NC2CN(C(=O)CCc3cnc(O)[nH]3)CC2O)c(C)c1 51301,n1(CC)nc(C)cc1C(N1CC(F)CC1C(N1CCC(O)(CC)C1)=O)=O 51302,C1(CN(C(=O)CCc2nccs2)C)CCCN(C(c2cnsn2)=O)C1 51303,N1(C(C(C(C)NC(c2cc([N+](=O)[O-])c[nH]2)=O)(C)C)=O)CC(O)C2(CCCC2)C1 51304,c1(C(N2C(C3CCN(C(C=CC(C)(C)SC)=O)C3)CCC2)=O)cc(C)c(C)o1 51305,CCC(C)(C)C(C(=O)NC1(CO)CCC(C)C1)OC.c12nc(co1)C(=O)NC2 51306,N1(C(c2ccc(CCC)cc2)C(=O)Nc2ccccc2)Cc2ncsc2C1 51307,Cc1sc(C(=O)NC2CC(O)CN(C(c3cccc(O)n3)=O)C2)cc1S(N)(=O)=O 51308,C1(OC)CN(C)C(C)(C(=O)NCC(CO)NC(c2ccsc2SC)=O)C1 51309,N1(C(C(C)(F)F)=O)CCN(C(=O)CN2CC=CC2)CC(O)C1 51310,N1(C(c2cc(SC)oc2)=O)CCN(C(=O)CNS(=O)(=O)N(C)C)C(CC2CC2)C1 51311,C1(C(=O)OC)CC2CC2N1C(=O)C(N1CC2CC2C1)C 51312,CCC(C)(C)C(=O)C(=O)N(CCO)CCOCCCONC(COOCCO)=O 51313,c1(-c2ccc(C(=O)NCCN(C(=O)CCCc3ncco3)C)[nH]2)ccccc1F 51314,c1(C(N(CC(C)NC(=O)C(C)(O)c2ccccc2)CC)=O)ccc(C)nc1OC 51315,Cc1ccc(C)c(CN(C(c2cccc(Br)c2)C(=O)O)C)c1 51316,c1(C(=O)OC)cc(C#N)cnc1NC(=O)NCC(O)COc1cccc(Cl)c1 51317,c1(C(=O)NC2(C)CN(C(C3CC(C#N)C3)=O)C2)nnn2c1CSCC2 51318,c1(C(N2CC(COC)(NC(c3cccc(OC)c3)=O)C2)=O)ccc(OC)c(C)n1 51319,Cn1ncc2c(N3CCC4(CC4)C3)nc(=NCCCOCc3ccccc3)[nH]c12 51320,C1(NC(=O)C(F)CC2CC2)CN(C(c2cccc(Br)c2)=O)CC2(CCC2)C1 51321,c1(C(=O)NC2CN(C(CC(CCC)O)=O)CC(C)C2)cc2ccc(F)cc2[nH]1 51322,C1(COC)(CNC(=O)C2=CCSC2)CCCN1C(c1ccc(C#N)s1)=O 51323,C[Si](C)(C)CC(C(=O)O)Oc1ccc(NC(=O)C(Cl)=CCl)cc1 51324,CCCC(CCC)CC(=O)NCC1CCC(C)(C)CN1C(c1sncc1CC)=O 51325,CN1CCC(NC(C2C3CN(C(=O)NC)CC23)=O)CC1=O.C(c1ccccc1F)=CC=C 51326,c1(CC(=O)N(CCCNC(C(OCCC#C)OCC)=O)CCO)cnccn1 51327,c1(C(N2CCCC(CCNC(CCCCCC)=O)CC2)=O)cc2cccnc2o1 51328,CCCCCC(O)CC(=O)N1CCCC(C2CCCCN2C(c2cnns2)=O)C1 51329,CC(C)CC(O)C(=O)ONC(=O)CC1CCCCC1.CC(CO)C(C)C 51330,C1(NC(CN(S(C)(=O)=O)C)=O)CC(N=c2[nH]c3ccc(N)cc3s2)C12CCC2 51331,c1(CNC(C2(C)CN(C)C(=O)C2)=O)ccc2c(c1)CN(C(=O)CS(C)(=O)=O)C2 51332,c1(C(=O)NC(CC)CN(C(c2cc(F)n(C)n2)=O)CC)c(OC)ccnc1F 51333,C1(C(N2C(C)CC(O)C2)=O)N(C(c2cnccc2C#N)=O)CCCC1(C)C 51334,c1(C(=O)NC2C(CNC(c3c(COC)nn(C)c3)=O)C2)cc2occc2n1C 51335,N1(C(N2C3(C)CC(C(F)F)(C2)C3)=O)CCCN2CCCC12 51336,CC(C)CC(CNC(C1(C#N)CCOC1)=O)NC(=O)C(C)(C)CC1CCOCC1 51337,CCC(C)(CCNC(=O)Cc1ccn(CC)n1)NC(C1CC1C(C)C)=O 51338,C1(OC)CCC(C(N2CCC3CC23C(N2CCC2C2CCC2)=O)=O)CC1 51339,C1(C(N2CC(OC)C(NC(C3CC3C3(C)COC3)=O)C2)=O)CCC(O)CN1C 51340,c1(C(=O)NCC2C(CNC(C3(C(C)C)CC3)=O)C2)cnc2[nH]ncc2c1 51341,N1(C(=O)C(F)C2CCOC2)CCCC(N=c2[nH]ncs2)(CO)C1 51342,c1(NC2(c3n(CC(=C)C)nnn3)CC3CC3C2)ccc2[nH]c(C)cc(=O)c2c1 51343,CC(C1OCCc2ccccc21)N(C)C.C1CS(=O)(=O)c2cccc(c2)NC(=O)N1 51344,c1(N2CC(C(C)NC(=O)CSC3CC3)OCC2)cc2nncn2cn1 51345,C#CCC(O)C(=O)N1CCOC(CNC(C2C3CCCCC23)=O)C1 51346,N1(C(c2cncc(C#C)c2)=O)CCC2(CC1)CN(CCc1ccnn1C)CCO2 51347,c1(CCNC(=O)NC(CSC)(C)CO)cc(C)ccc1Cl 51348,C=C1COc2c(C(=O)NC3CC(CO)N(C(C4(N(C)C)CCC4)=O)C3)cnn2C1 51349,Cc1nc(Cl)ccc1S(=O)(=O)N1CCC(F)(C(=O)NCC(F)F)C1 51350,c1(OCCCOC)ncccc1CNC(c1nnc(C2CCNCC2)s1)=O 51351,N1(C(CC(C)C)=O)CCSCC1CCNC(c1cnoc1C1CCC1)=O 51352,Cc1ccccc1C=CC(=O)NC1C2CC3C(C2)C13 51353,c1(NCC(N2C(C)(CNC(C)=O)CC(F)(F)C2)=O)ccc(S(N)(=O)=O)cc1 51354,C1(NC(N2C(C)CC2)=O)CC12CCN(C(=O)C(C)CC#N)CC2 51355,CN1C(=O)CCC1CC(=O)NCC=CCNC(c1ocnc1C1CC1)=O 51356,N1(C(c2cccc(OCC)c2)=O)CCN(C(=O)CSC)C(c2ccnn2C)C1 51357,c1(C(N2CCCC(N(C(=O)C3=CCCO3)C)CC2)=O)ccc2cncn2c1 51358,C=CCC(F)(F)CNC(=O)CN(C)C(C1CCN1C(C)(C)C)=O 51359,C1(C(N(C(C)CC(=O)N(C)CCC2CCCO2)C)=O)C2CN(C)CC12 51360,c1(NC(C)=O)ccc(Cl)c(C(N2CCOCC2CNC(=O)CNS(N)(=O)=O)=O)c1 51361,c1(-c2ccc(CN3CC(C(=O)OC)C(C)CC3)s2)cccc(F)c1C#N 51362,C=C(C)CC(=O)NCC(C(C)C)NC(C1CCCN1Cc1ccccc1)=O 51363,C(=O)(CC(C)CC(=O)N1CCC(C)(C)C1C(=O)NCCCc1cc(C)no1)OC 51364,c1(CC=C(C)C)ccccc1C(=O)NC(C)CN(C(=O)Cc1c(C)noc1C)C 51365,C1(NC(C=Cc2c(C)ccs2)=O)CN(C(=O)C(=C2CCCCC2)F)CC12CCC2 51366,C1(C)(NC(C(C2CCN(C(CCC)=O)C2)(C)C)=O)CCSCC1 51367,c1(C(N2CCC(NC(C3(C)CCC(=O)N3)=O)C(O)C2)=O)cc2ccc(F)cc2s1 51368,c1(C(=O)NCC2CC(NC(=O)CC3CC(F)(F)C3)C2)nccc(Br)c1O 51369,CC(F)(C(=O)N1CCC(CCNC(c2ccccc2F)C)CC1)C(F)(F)F 51370,CCCC(C(=O)NCC)NC(=O)C(c1cn(C)nn1)NC(=O)CC1CCN(C)C1 51371,C1(C(=O)NC2CN(C(c3ccc(C#C)o3)=O)C2)CS(=O)(=O)CC1C(F)(F)F 51372,c1(C(N(C2CCCN(C(C(C)NC(C)=O)=O)C2)CCO)=O)ccc(F)c(C)c1N 51373,c1(Cc2cn(C)nc2-c2ccnn2C)ccc(F)c(F)c1.c12noc(n1)C2 51374,CC1CN(C(C2CCN2CC(F)(F)F)=O)CC1(C)CNC(=O)CCOCC(F)F 51375,Cc1cnc2c(C(=O)NC3CN(C(=O)CO)CC34CC4)cccn12 51376,C1(C(N(C(C)COC)CC)=O)(CNC(=O)C(N)=O)CCCCC1 51377,c1(C(=O)NC2(C)CCN(C(C3CCC3)=O)C2)nc(Cl)ccc1N 51378,N1(C(C2(CC)CC2)=O)CCCC(C(N2CCC2CC2CC2)=O)CC1 51379,N1(C(CCc2cc(C)sc2C)C)CCN(C(C)C)CC1C 51380,c1(CCC)cccc(C(N2CCC(C)(CNC(=O)CCS(C)=O)C2)=O)c1 51381,N1(C(C2CN(C(C)=O)C2)=O)CC(C(=O)NCC(C)(F)C(C)C)C(F)(F)C1 51382,c1(C2C(C(=O)NCC3CC(NC(=O)C(F)=CCCF)C3)C2)ccc(F)cc1F 51383,C(c1ccccn1)=C(C)C(=O)NC(C)C(C)NC(=O)CN(CC(C)(C)C)C 51384,CC(c1cccs1)=CC=CC(=O)NC(C)C.C12(C)CCCN1C(=O)C2 51385,N1(C(C(Cc2cn[nH]c2)NC(COCC(=C)C)=O)=O)CCC2CC12C 51386,C#CCC(CC(=O)NCC#CC1CC1)NC(=O)CSCC=C 51387,C(C)(c1ccco1)=CC(=O)N(CCC)CCNC(=O)Cc1ccn(CC)n1 51388,C1(NC(c2n(CCC)nnn2)c2conc2CSC)CC2(C1)NC(=O)NC2=O 51389,c1(C(N2CC3C(CNC(COCC(=C)C)=O)(C3)C2)=O)c(C)cc(C)cc1O 51390,C1(F)(C(N2CCC(OCC=C)C2)=O)CCCN(C(c2c[nH]c(C)c2)=O)C1 51391,c1(C(=O)NCCN(CC(C)O)C(=O)Cn2ncnn2)cc(F)cc(S(N)(=O)=O)c1 51392,c1(C(=O)NC2CN(C(c3cc(CC)[nH]n3)=O)C(C)C2)ccc(=O)n2c1COCC2 51393,C1(C(=O)NC(C23CCC(CC2)C3)CNC(COC(CC)C)=O)CCOC(=O)CC1 51394,c1(OCCN(C)C)ccc(C(N2CC(NC(=O)Cc3ccsn3)C(O)C2)=O)cc1N 51395,c1(C(=O)NC2CN(C(C3(F)CC=CCC3)=O)C2)cc(O)nc(O)n1 51396,C1(NC(C2C(C)(CC)C2)=O)CC2CCC(C1)N2C(C1(N(C)C)CC1)=O 51397,c1(C(=O)NCC(CC=C)NC(C2CCCC(O)C2)=O)cccc2c1CCCN2 51398,C1(C(=O)NC2CC(NC(C(C)OCC=C)=O)C2)CCC2(CC1)CC2(F)F 51399,Cc1cc(C(=O)NCCC(O)CNC(=O)CC(C)C)n(C2CC2)n1 51400,CCCC(C)(O)C(=O)NCCN(C(c1nc(C)nn1C)=O)Cc1ccc(Cl)nc1 51401,C1(NC(=O)NC(c2ccc(OC)nc2)C)(CO)CCCCC1C 51402,N1(C(C2C(C)CCO2)=O)CC=CC(C(=O)N(C)CC2CC2)C1 51403,CC1CN(C)CC(C(=O)NCC23CC(NC(C4CC=CC4)=O)(CCO2)C3)O1 51404,C(c1cccc(Br)c1)=CC(=O)NC(CC)CNC(=O)Cc1ncn(C)c1C 51405,C(CC(C)C)(C(=O)Nc1cncnc1C(C)C)ONC(C(C)NC(C)=O)=O 51406,c1(CNC(c2cccc(C)n2)CC)nn(C)c(Cl)c1I 51407,C(=O)(C(O)CC[S+](C)C)NCc1cn(CC(C)NC(c2cc[nH]n2)=O)nn1 51408,n1(CCC(=O)N(CCCCCCCN)C)nc2ccccn2c1=O 51409,Cc1nnccc1C(=O)NCC(C1CCOC1)NC(=O)CN1CCOCC1 51410,c1(OC)c(C)cc(C(N2CCCC2CNC(=O)C=C2CCC(C)C2)=O)cc1C 51411,Cc1c(C(=O)NCCc2n[nH]cc2C(=O)NC2COCC2C)nnn1C 51412,C1(NC(c2c(OC)nccc2)=O)CC(F)CN(C(C2CCC(=O)NC2)=O)C1 51413,C1(NC(C2CCC(=C)CC2)=O)CCN(C(=O)Cn2cc(C(F)(F)F)nn2)C(C)C1 51414,C1(C(=O)NCC(C)(C)CC2CN(C(c3cncnc3)=O)C2)C(C)(C)C1(F)F 51415,C1(F)(C(=O)NC2C(C(C)C)CCCC2)CCN(C(c2ccccc2)=O)CC1 51416,C1(CNC(=O)CSC(F)F)CN(C(C23CC4CC2C3C4O)=O)CCC1(F)F 51417,N1(C(c2cnc(CC)s2)=O)CC2(CC(CC(=O)N(C(C)C)CC3CCC3)C2)C1 51418,c1(C(N2C(CNC(C=C(C)CCc3ccccc3)=O)CC2)=O)ccc(F)cc1O 51419,N1(C(C(C)N2CCC2)=O)CC2(C1)CN(C(C1(C#N)CCOCC1)=O)C2 51420,CC1(c2cn(CC3CCC(C(N)=O)O3)nn2)CCCN1C(=O)COC1CCOC1 51421,N1(C(C2(COCC)CC2)=O)CC2C(CC(=O)NC3(C(N)=O)CCCC3)C2C1 51422,C1(NC(C2N(C(C3C(OC)CCCC3)=O)CCN(C)C2)=O)CCCC(C2CC2)C1 51423,c1(C(N(C(C(=O)NCCC#N)C2CC2)C)C2CC2)ccc(F)c(F)c1 51424,C(CCCC(=O)N(C)CC1CCCN1C(=O)CNc1ccccc1)OCCC=C 51425,c1(C(N(C2CCN(C(CN(CCOC)C)=O)CC2C)C)=O)cc2cccnc2o1 51426,CC1C(NC(c2cnn[nH]2)=O)C(C)CCN1C(C1CCCCCC1)=O 51427,Cc1nnc2n1CCCC2C(=O)c1noc(-c2cc(F)ccc2F)n1 51428,N1(C(CC2C(C)(C)C2)=O)CCC(C=CC(=O)NCC=C(Cl)Cl)CC1 51429,C1(NC(CCN2CCC(C)CC2)=O)CCCN(C(C2CCCS2)=O)CCC1 51430,C1(C(=O)NC(C(=O)OC)C2CC2)CCCCN(C(=O)C(C)N2CCCC2)C1 51431,CC(C)(CC(F)(F)F)C(=O)NCC1(F)CC(CNC(C2CN3CCN2CC3)=O)C1 51432,C1(O)(CN(C)C(c2ccnn2CC#N)=O)CCN(C(=O)COC2CCOC2)C1 51433,C1(C)(C(=O)NCCNC(C2N3C(C)CN(CC3)C2)=O)Cc2ccccc2NC1=O 51434,CC1CN(C(c2cscc2Cl)=O)CC1NC(c1cccc(OC(F)(F)F)n1)=O 51435,c1(OC(C)C)c(F)cc(-c2ccccc2C(N2CC3CCC2C(O)C3)=O)cc1F 51436,C1(NC(CSCC(C)C)=O)CCN(C(=O)Cc2cnccc2Cl)CC1 51437,N1(C2CC(C(=O)OC)C2)CCCN(C(=O)NC2CCCN(C(=O)C(C)C)C2)CC1 51438,C(=O)(C(C)CC(C)C(C)=O)NC1C2OCC(NC(c3c(CC)n(C)nc3)=O)(C2)C1 51439,c1(CC)cncc(CNC(C2CC2CNC(C2CCCC(O)C2)=O)=O)c1 51440,C1(CNC(c2c(C)coc2)=O)CN(C(=O)C(O)C2CCCC2)CC1(F)F 51441,C(CO)(CCCCNC(c1ccnn1C(F)F)=O)NC(c1c(C(C)C)ncs1)=O 51442,N1(C(CN(C(C(C)C)=O)C)=O)CCCC(C)(NC(=O)C(O)C(F)F)C1 51443,c1(CCNC(C(c2cnn(C)c2)NC(C(C)=CC2CC2)=O)=O)nnc(C)n1C 51444,C1(NC(c2c(C)nccn2)=O)CC=C(C(=O)NCC(F)(F)F)C1 51445,N1(C(CCC#CC)=O)CCC2(CC(NC(=O)Cc3nc([N+](=O)[O-])n[nH]3)CO2)C1 51446,c1(C(=O)NC(C2CCN(C(c3c(C(C)C)csc3)=O)C2)C)n[nH]cc1[N+](=O)[O-] 51447,Cc1cc(Cl)cc(C(=O)NCC(C)(C)CN(C)C(c2cc(Cl)ccn2)=O)c1N 51448,C(=O)(CP(=O)(C(C)C)C(C)C)NC(CN(C(c1cc(COC)[nH]n1)=O)CC)C 51449,c1(OC)cccn2ncc(C(=O)N(CCO)Cc3cc(F)ccc3Br)c12 51450,c1(Cn2c(N(C(C)=O)CCO)nnn2)cc(CC2(C)CSC(C)=N2)cc(C)c1 51451,C(=O)(C(C)S(N)(=O)=O)NCC1(O)CC(C(=O)NCCc2cc(C)no2)C1 51452,N1(C(C2(C)CCCN(S(=O)(=O)CCBr)C2)=O)C2CCCC1COC2 51453,CCCCCC(CC)C(=O)NC1CN(C(c2cc(C)cnc2N)=O)CC1C1CC1 51454,C1(C(N)=O)(COC)CCCN(C(c2ccc(OCC(F)F)nc2)=O)C1 51455,C1(C(=O)NCCC2CCN(C(C=Cc3nc(C)sc3)=O)C2)Cc2ccccc2O1 51456,c1(C(N(CC(=O)NC2CCC2NC(C2CC23CC3)=O)C)=O)ccccc1Cl 51457,c1(-n2cc(CN(C)C(c3cc(O)cs3)=O)nn2)cccc(Br)c1 51458,CN1CCC(NCC(=O)NC2CC2NC(=O)C(N2CCC(O)CC2)C)CC1 51459,CC(C)(CC(F)(F)F)C(=O)NCC1C=CCN1C(=O)CC(C(F)F)n1cccn1 51460,c1(NS(C)(=O)=O)ccc(F)c(F)c1.c12cncc(c1)C(=O)N(N(C)CCO)C2 51461,N1(C(C=C(C)c2ccco2)=O)CCCC1C1CCCN1C(=O)Cc1nonc1C 51462,c1(OC(C)(C)C)cc(NCC2CC(N3CCCC3)C2)[nH]n1 51463,c1(C(=O)NC2CC(CCNC(c3cc(C)sc3C)=O)C2)cnc2n1CCCC2C 51464,C1(C(=O)NCC(F)F)CC12CCN(C(=O)C=Cc1cscn1)C2 51465,Cc1cc(=NCCCN2CCC(C)CC2)[nH]c(N2CCC(c3nncs3)CC2)n1 51466,N1(C(C(CC(=C)Cl)NC(=O)Cc2ccn(C)n2)=O)CC(=O)NC(C)(C)C1 51467,c1(C2C(C(=O)NCC(CNC(c3cc(OC)ns3)=O)(C)C)C2)cccc(C#N)c1 51468,C1(C(N2CC(OC)C(C(=O)NC3C(C)(C)C3(C)C)C2)=O)CCCCNC1=O 51469,c1(N(C)Cc2cccc(OC)c2OC)nccc(=NC2CCCC2S(C)(=O)=O)[nH]1 51470,C1(C(C)N(C(=O)CCN(C)C(C2CCO2)=O)C)CCOCC1 51471,N1(C(CCCSC)=O)CCC2(C1)c1[nH]cnc1CCN2C(=O)CCc1nccs1 51472,N1(C(COCC)=O)C(C(N2CSCC2C(N)=O)=O)CCC12CC2 51473,C1(C(N(C(C#C)C)C)=O)C2CCC(C2)C1NC(C1CCC1C#N)=O 51474,C=CCC(C(=O)NC1C=CCC(C(=O)NC(c2ccc(C)nc2)C)C1)C(C)C 51475,Cc1occc(=O)c1NC(C1(CNC(c2cnnc(O)c2)=O)CC1)=O.N1CCC1CO 51476,N1(C(C(C)n2ccnc2)=O)CCC2(CC(C(=O)Nc3cncc(Br)n3)=NO2)C1 51477,c1(C(C(=O)NC2CCN(C(c3cnc(CC)[nH]3)=O)C2)C)c(C)n[nH]c1C 51478,N1(C(C2CN(OC)C(=O)C2)=O)C(C)CC2CN(C(=O)CCC(C)CN(C)C)CC12 51479,C1(F)(CNC(C(C2CCN(C(=O)C=CC(=O)N(C)C)C2)C)=O)CCN(C)C1 51480,C12(C(=O)NC(CCCC)CNC(=O)C(F)n3ccnc3)C3CC(CC13)C2(F)F 51481,N1(C(c2c(OC)cncn2)C(=O)NCCCSC)CC(N(C)C)C(C2CC2)C1 51482,c1(CN(CCF)CC)cn(CCNC(C)C(=O)Nc2ccc(C(=O)O)o2)nn1 51483,C1(C(=O)NC(CC=C)CNC(c2cnc(C)[nH]2)=O)CCC(n2ccnn2)CC1 51484,c1(C(=O)NCCC(CC)(C)NC(=O)C(n2nccc2C)C)ncnc(C)c1C 51485,C(CC(C)(C)NC(=O)CNC=O)NC(CN(c1ccccc1)C)=O 51486,C1(NC(C)=O)CCCCN(C(c2cc(C)n(CC3CC3)c2C)=O)C1 51487,N1(C(c2c(C)nn(C)c2)=O)CCc2c(C(N3CCCCC(O)C3)=O)csc2C1 51488,CCCCCC(O)CC(=O)N1CC2CCCC2C1C(=O)NCC1(C)COCCO1 51489,c1(C(=O)NC2C(C)N(C(=O)CCc3ccc(Cl)nc3)CC2)ccc2c(c1)COC2 51490,c1(OC)cncc(C(N2CCOC(CNC(C3CC(=O)N(O)C3)=O)C2)=O)n1 51491,Cc1ccc([N+](=O)[O-])cc1C(=O)NC(C)C(C)NC(=O)C(CO)C(C)(C)C 51492,C(CNC(=O)C(C1CCCCCC1)C)(CC(C)C)NC(CC1(C=C)CCC1)=O 51493,C1(C(=O)NCC(COC)O)CCCN(Cc2ccc(CN(C)C)cc2)C1 51494,C12(C(N(CCN(C(=O)CCc3ccnn3C)CC)CC)=O)CC(CO1)C2(C)C 51495,c1(C(C)N(C(c2cnc(N(C)C)nc2)C(=O)NCCN(C)C)C)ncc(Cl)n1C 51496,c1(CCCCC)nc(C(=O)NCC(CC)NC(=O)CCc2nc(=N)[nH][nH]2)cs1 51497,c1(C(=O)NCC(CCNC(CC(CC)SC)=O)O)ncn2c1CCCC2 51498,CC1CCC(C(=O)NCCn2ccc(C(=O)NCC(F)(F)C(N)=O)c2)CC1 51499,c1(C(=O)NCCN(C(Cc2c(C)ccs2)=O)C)ccc2[nH]ccc(=O)c2c1 51500,C1(C(=O)NC(CNC(C2(COC)CCCO2)=O)C2CCC2)CC2CCC(C1)C2 51501,C1(C)(CC)NC(=O)N(CC2(C)CN(Cc3scnc3C(=O)OC(C)(C)C)C2)C1=O 51502,c1(C(C(N2CCC(CNC(CNC(=O)OCC)=O)CC2)=O)O)c(C)cccc1C 51503,Nc1cccc(C(=O)NCCCNC(=O)Cn2cc(I)nn2)c1 51504,c1(OC)noc(C)c1C(=O)NC1CCC(CC(=O)NC2CC2c2cncs2)CC1 51505,c12ccccc1CN(CC)CCO2.c1(NC(C)=O)ncc(OC(F)(F)F)cn1 51506,Nc1ccc(F)c(C(N2CCC(NC(=O)Cn3cc([N+](=O)[O-])cn3)C(F)C2)=O)c1 51507,C(CC(C)C)(C(C(=O)NCC(F)F)N1CCSCC(C)C1)OC 51508,c1(CC(CO)NC(C2COCCN2C(=O)C(O)C2CC2)=O)ccc([N+](=O)[O-])cc1 51509,c1(OC)cc(C)c(C(N2CCC(CNC(=O)C3=CCOCC3)C(C)C2)=O)c(C)c1 51510,n1(CC(=O)NC(CNC(c2ccc(C)s2)=O)C2CCC2)nc(C)c([N+](=O)[O-])c1C 51511,c1(C(=O)NCC(F)CNC(C2(C(F)F)CC2)=O)cccc2ccnn12 51512,c1(C(=O)NCC2C(C)CN(C(C3CC(O)C3)=O)CC2)nc(Cl)c(=O)[nH]c1N 51513,C1(NC(C(CSC)OC)=O)CC(=O)N(C2CN(C(=O)CC3(C)CC(F)(F)C3)C2)C1 51514,c1(C(=O)NC(CNC(c2cnc(OCC)nc2)=O)CC(C)C)ccc(F)cc1C 51515,c1(C(N2CCCC(NC(c3cncc(F)c3Cl)=O)C2)=O)nc2cc(O)ccc2[nH]1 51516,N1(C(CCCCC#C)=O)CCS(=O)(=O)C(CCNC(=O)C(O)P(C)(C)=O)C1 51517,N1(C(C2C(OCC)CC2)=O)CCC(N(C(=O)CSc2cccc(C)c2)C)C(C)C1 51518,C1(O)(C(=O)NC2CCC(CNC(C(N3CCOCC3)C)=O)C2)CCCC(C)(C)C1 51519,c1(C(=O)OC)ccnc(C(N2CCNCC2C)=O)c1F 51520,S(=O)(=O)(c1cc(Br)c(Br)s1)N1CC2N(Cc3cncc([N+](=O)[O-])c3)C(C2)C1 51521,C(=O)(C(CC1CC1)NC(c1cocn1)=O)N(CCOC)C(C)C1CC1 51522,C1(NC(c2cc(N)c(Cl)nc2)=O)CCCC12CCN(C(c1ccnnc1O)=O)C2 51523,c1(C(N(CC(O)CNC(C2(n3cccn3)CCC2)=O)C)=O)csc(Cl)c1 51524,C(C(=O)N=c1cc(C(N)=O)n(C)[nH]1)C1N(C(C(C=C)O)=O)CC(O)C1 51525,C(C(CNC(c1ccc(SC)cc1)=O)C(F)(F)F)NC(CCCC#C)=O 51526,c1(C(N(C)CC2N(C(CC(C=C)C)=O)CCCC2)=O)cc(C)cc2cccnc12 51527,C1(NC(C2C(C)(C)C2)=O)C=CCCC1C(N1CCC2C(C(N)=O)C2C1)=O 51528,c1(OCC(=O)N(C(CN(C(c2c(C)c[nH]n2)=O)C)C)C)ccccc1C(C)(C)C 51529,c1(C(N2CCC(C(N(CC#C)CC3CCCO3)=O)(CO)C2)=O)cccc(=O)n1C 51530,C(Cc1ccccc1)(CCCO)NC(c1ncn(CC)n1)=O 51531,c1(SC)ncc(C(=O)NCC(O)CNC(C2CCCN2C(=O)NC(C)C)=O)s1 51532,c1(C(C(N2CCN(C(C3(OC)CCOC3)=O)CC2)=O)C)ccc(F)c(F)c1 51533,N1(C(C(c2ccc(C)cc2)CC)=O)CC2(CCC(CNC(=O)CC(C)F)O2)C1 51534,N1(C(C2(SC)CCC2)=O)CCN2CCN(C(=O)C#CC3CCOCC3)CC2C1 51535,N1(C(c2c(COC)cccn2)=O)CCC(NC(=O)C(F)CC(C)(C)C)C(C)(C)C1 51536,c1(N2CCC(N(C)C(C34CCOC3CCOC4)=O)C2)nc2c(cc1C#N)CCOC2 51537,CCS(=O)(=O)CCN(CC(=O)NCc1cccc(Oc2ccccc2)c1)C 51538,C1(CNC(c2[nH]cc(CC)c2)=O)CN(C(=O)CC(F)(F)F)CC1C(F)(F)F 51539,C(=O)(C(C)CC(C)(C)C)N1CC(OC)C(CNC(=O)COC(F)(F)F)C1 51540,N1(C(=O)CC2CC=CC2)CC2CCN(C(C3CCOC3C3CC3)=O)C2C1 51541,N1(C(c2c(CNC(C(CCCC)=O)=O)occ2)=O)CC(C)OC2(CCC2)C1 51542,C#Cc1ccc(C(N2CCC(CCNC(c3cnc(C)s3)=O)CC2C)=O)c(F)c1 51543,CCC(C(=O)N1CC=CC1CNC(c1ncccn1)=O)NC(N)=O 51544,c1(C(=O)NC2C(NC(C(CC)n3cccn3)=O)C2)cc(OC)c(Cl)cc1OC 51545,c1(C(N2CC(CCNC(Cc3n(C)ccc3)=O)OCC2)=O)cnc2[nH]ccc2n1 51546,Cc1c(C(=O)NC2CN(C(=O)CC3CCCOC3)CC2O)oc2c(Cl)cccc12 51547,C1(NC(C2(CCC)CCC2)=O)CCCC(NC(=O)C(c2ccc(O)cc2)(C)C)C1 51548,N1(C(C(C)OCC)=O)CCC(F)(CNC(c2ccc(N)cc2Br)=O)CC1 51549,c1(NC(=O)CSCC=O)nc[nH]n1.c1(CC(=O)NCC(C2CC2)S)ccno1 51550,Cc1c(C(N2CCCN(C(c3ccsc3)=O)CC2)=O)cc(F)cc1Br 51551,c1(COC)nc(NCCCCS(C)(=O)=O)cc(=NC2CCCC(O)C2)[nH]1 51552,C1(C(=O)NC(c2ncc[nH]2)(C)C)CN(C(=O)CN2CCC(=O)CC2)CC1(F)F 51553,N1(C(C2N(CC#C)CCC2)=O)CCCC2(CC(NC(C3CC(F)(CO)C3)=O)C2)C1 51554,N1(C(C(CO)NC(c2ccc(F)cn2)=O)=O)CC2CC1CO2 51555,C(CN=c1[nH]c(=NC2C=C(c3ccccc3)C2)[nH]c2cccnc12)NC(=O)OC 51556,c1(CCC)c(C(=O)NCC(CC)NC(=O)CC2CC=CCN2C)cnn1C 51557,C1(N(C(CCC#C)=O)C2CCCC2)CC2CC1N(C(=O)CC(CC)C1CCC1)C2 51558,c1(C(=O)NCC2(COC)CN(C(c3cccnc3N)=O)C2)ccc2ccnn2c1 51559,C1(C2(O)CN(C(c3n[nH]cc3Br)=O)C2)(CNC(=O)C(F)=CCCF)CC1 51560,C(=O)(CCCC(F)F)N1CCC(NC(C(C(C)C)C)=O)CC1 51561,C1(OC)CCCC(C(N2CCCC2CCCNC(=O)Cc2c(Cl)cnn2C)=O)C1 51562,N1(C(CCOCCOCC)=O)CC(C)N(C(C2CCC(C)(C)OC2)=O)CC1C 51563,C=CC(C)CC(=O)NCC=CCNC(c1coc(C(F)F)c1)=O 51564,c1(CC)ccccc1C(=O)NC1CCOC(C(=O)NOCCCN(C)C)C1 51565,c1(N2CCC(N3C(=O)CC(OC)C3)CC2)ccnc(C2CC2)c1O 51566,C(N=c1[nH]c(=N)[nH]c(=NCc2ccccn2)[nH]1)C1(N(C)C)CCCC1 51567,C1(C(C)=O)CC1(Cl)C(=O)NC1CC1NC(=O)COc1cn[nH]c1 51568,CCC(C)CC(C)C(=O)N1CCC(F)(C(N2CC(O)C(N=[N+]=[N-])C2)=O)CC1 51569,c1(OC)ccc(-c2cc(NC(=O)NC3CCC3S(C)(=O)=O)no2)c(Cl)c1 51570,N1(C(CC2CC(OC)C2)=O)CCN(C(=O)C(CN(C)C)N(C)C)CC1CS(C)(=O)=O 51571,N1(C(CCc2ncc(C)[nH]2)=O)CCCCC(CNC(C2CCCN2C(C)C)=O)C1 51572,C1(NC(C(CC#C)NC(=O)C(C)CC2CC2)=O)CCCOC12CCC2 51573,N1(C(C(=O)NCCNC(C)=O)=O)CCN(C(=O)CC(C)P(C)(C)=O)CCC1C 51574,C(C)(CCCCN=c1nc2c(c[nH]1)CCCCC2)NC(C(C=C)(C)CCOC)=O 51575,C1(O)(C(C)C)CCN(C(C2(NC(=O)C(C)C3CC3)CCOCC2)=O)C1 51576,CC1=C(C(=O)N2CC3CC2CN3C(c2[nH]nc3cnccc23)=O)SCCO1 51577,Cc1ccc2c(=NCC3(C)CCC(=O)N3)[nH]c(=NC(C)c3cscn3)[nH]c2c1 51578,C12CCCC1C(=O)NC2.C1(OCC)CCC1CNC(=O)CCC1CCCC1 51579,N1(C(c2cnns2)=O)CCC2CN(C(C3CN4CCN3CC4)=O)C2C1 51580,C(C(C)(C)C#CC(=O)N(C(CC)CO)CC)NC(C(CC)N(C)C)=O 51581,C1(C)(CCNC(CCC=CCC=C)=O)CCN(C(C2(C=C)CCOCC2)=O)CC1 51582,C1(C(=O)NCC2(C)CC3CC3C2)CN(C(C2(C)CC=CCC2)=O)CC1(F)F 51583,N1(C(CCc2n(C)ccn2)=O)CC2(CC(CC(=O)NCC(c3cccs3)O)C2)C1 51584,c1(C(=O)NCC2N(C(CCCCCOC)=O)CCN(C)C2)ccc(F)c(C#N)c1 51585,c1(C(N(C(C)C(=O)NC(C)CC2CCCCC2)CC)=O)ccc(=NC)[nH]c1 51586,C1(C(=O)NC(CC)CSC)CC(NC(=O)Cc2ccco2)CCO1 51587,N1(C(C2CC(=C)C2)=O)CCC2(CC(NC(c3c(-c4ccccc4)coc3C)=O)C2)C1 51588,N1(CC(=O)NC2C=CCN(C(c3c(C(C)(C)C)[nH]cn3)=O)C2)CCCCS1(=O)=O 51589,N1(C(C(C)SC)=O)CCC(C2CCCN(C(c3c(Cl)nn(C)c3Cl)=O)C2)C1 51590,C1(C)(C(=O)NCC2CN(C(c3sc(CC)c(C)c3)=O)CC2C)CCC(C)CC1 51591,C12(OC)CC3CC(C1)C(NC(=O)N(C)CC1COC(C)C1)C(C3)C2 51592,C1(NC(CCCCOC)=O)CC2CCCC(C1)C2NC(c1ccco1)=O 51593,CC(C)S(=O)(=O)C(C)C(=O)NCC1(O)CCCN(C(=O)C(F)(F)C2CC2)CC1 51594,N1(C(C(C)OC)=O)CCN(CCC2CCCCN2C(c2cc(C#N)cs2)=O)CC1 51595,c1(C(N2C(C)CC(NC(CC(C)(C)SC)=O)C2)=O)cccc2[nH]cc(Cl)c12 51596,C(=O)(CC(O)CN(C)C)NC1(C(=O)NCc2ncn(C(C)C)n2)CC1(C)C 51597,CON1CC(C(=O)NCC2CCCC2C(=O)NCC2(C)CC2)CC1=O 51598,C(CCCl)(CCCl)(c1n(CCOC)nnn1)NCC1(c2ccccn2)CC1 51599,c1(N(CCNC(c2csc(C(C)C)n2)=O)CC)nc(O)c2ccc(Cl)cc2n1 51600,N1(C(c2c(SC)cnn2C)=O)CC2CC(C)N(C(c3cccc(F)c3C)=O)C2C1 51601,c1(OC)ccc(NC(C2CC(NC(=O)C3=CCCOC3)C2(C)C)=O)cc1C 51602,N1(C(CC(CC)OC)=O)CC(N(C(=O)CCOC)CC)C2(CC2)C1 51603,c1(C(=O)NC2(CNCc3c(C)ccc(F)c3)COC2)cc(C)c(C)cc1I 51604,O=C(CCCc1ccncc1)NNC(=O)C1CCC(c2cc(F)cc(F)c2)C1 51605,C1(CC(=O)NCCN(C(c2n[nH]cc2OC)=O)CC)CCCC(=O)N1 51606,Cc1cc(N2CCCC(C(C)(C)C)C2)nc(=NCCc2cnc3n2CCOC3)[nH]1 51607,C1(CC#C)(NC(=O)C=CCNC(=O)CC2CCCO2)CCC1 51608,c1(CN(C2CC2)CC)cc(-c2coc3ccccc23)c(OC)c(Cl)c1 51609,C(CC(C(C)(C)C)NC(C1CC2CC2C1)=O)N(C(c1cn(CCC=C)nn1)=O)C 51610,N#CC1(C(N2CCOC(CNC(=O)CCC(N)=O)C2)=O)CC(F)(F)C1 51611,c1(CC(=O)NC(C)CC(C)NC(C2CCCC2c2nc[nH]n2)=O)ccc(O)nc1 51612,C1(C(=O)NC(CN(C(c2c(C)nc(C)[nH]2)=O)C)(C)C)CC2COCC2C1 51613,C(CC(C)CC)(C(=O)N(CC(C)(C)CO)C)NC(CC1CC(=C)C1)=O 51614,c1(CNC(=O)NC2CCC3CC23)ccc(C2CCC2)cn1 51615,C1(NCCC(=O)NC(CC)C)CCc2cnnn2C1 51616,C1(CCCNC(C(C2CC(F)(F)C2)OC)=O)CCCN1C(=O)C=CCO 51617,c1(CC)c(Cl)nc[nH]c1=NCC1CN(C(C2CC(=O)N2)=O)CC1C 51618,N1(C(CCCOCC)=O)CCN(C(c2cc(OC)ns2)=O)CC1C1CC1 51619,N1(C(C(C=C)(C)C)=O)CCC2(CC1)CC(NC(=O)C(CC)n1nccc1C)CO2 51620,N1(C(COCCC#C)=O)CC(C)N(C(c2cc(OC)c(C)c(OC)c2)=O)CC1C 51621,c1(C(N2CCCC(NC(N(C)C)=O)C2)=O)cc(O)cc(Br)c1 51622,Cc1cccc(C(C)NC(C2(NC(=O)CC3CC=CCC3)CCSC2)=O)n1 51623,N1(C(c2ccccc2)CCNC)CCC(S(=O)(=O)N2CCCC2)C1 51624,N1(C(CCC(=O)NC)=O)CC(CO)C2(C1)CN(C(c1n[nH]cc1Cl)=O)C2 51625,c1(C(=O)NCCF)cc2n(n1)CCCN(C(c1ccc3nc(O)oc3c1)=O)C2 51626,c1(CCC(=O)NC2C(C(=O)OC)C3C2CCCC3)c[nH]c2cc(C)ccc12 51627,C12(CNC(C3CC(O)(CC#C)C3)=O)CCCC1N(C(=O)C(C)CSC)CCC2 51628,N1(C(c2cc(Br)cc(F)c2F)=O)CCOC2(C1)CN(C(C13COCC1C3)=O)C2 51629,N1(C(C2CC(=C)C2)=O)CCC(NC(c2sc(SC)cc2C)=O)C(F)C1 51630,C12(C(=O)NCC3(C(=O)NC(CCOC)CO)CCCC3)CC(C#N)(C1)C2 51631,N1(C(C(C=C)(C)O)=O)CCCC(C)(C(=O)NC2CCOC2=O)C1 51632,CCC(C(=O)NCC(C)N(C)C(C1(C#N)CC1(C)C)=O)C(C)C 51633,c1(CNc2ccnc(SC)n2)cc(O)cc(O)c1.C12CCNCC1N2 51634,c1(C(=O)NC2C(CNC(c3c(C)ncn3C)=O)C2)cc(Br)cc2c1OCC2 51635,N1(CCCC(=C)C)CCC2(CC1)CC(N=c1[nH]nc(C(F)F)s1)CCO2 51636,Cc1ccc(NC(C2CCCCN2C(=O)CC2CCCC(=O)C2)=O)c(C)c1 51637,c1(C(=O)NC(CCNC(c2c(C)snc2)=O)C)nn(-c2ccccc2)cc1Br 51638,C1(CNC(C(CC(C)C)O)=O)CN(C(c2ccccc2O)=O)CCC12CCC2 51639,c1(SC)ccc(C=CC(=O)NC(C2CCN(C(C3CCCCC3O)=O)C2)(C)C)s1 51640,C1(C(=O)NC2(C=C)CCC2)CCN(C(C2CCCN2CCC)=O)C1(C)C 51641,c1(CC)ccc(NC(C2(N(C(=O)C(C)=C(C)C)C)CC2)=O)c(F)c1 51642,Cc1ccc(Cl)c(C(=O)NCC2CC2CNC(C2(n3ccnn3)CC2)=O)c1O 51643,CC(C)CC(C)(O)C(=O)NC1CN(C(c2cc3nc[nH]c3cn2)=O)CC1C 51644,C1(OCC(C)NC(=O)NC(C)CC2(O)CCC2)CCCCC1 51645,c1(CC(=O)NC2CC(F)(CNC(c3nc(Cl)cs3)=O)C2)c(F)cncc1Cl 51646,C12(CNC(C3(C(=O)NC4CC4)CC3)=O)CCC(C1)N(C(=O)C(C)n1cccc1)C2 51647,C1(CC)(CC)CC(C(=O)NCC2(C(=O)NC3CCCC3C)CCCO2)C1 51648,c1(C(=O)NC(c2cn(C)nn2)C(=O)NCC(CC)N(C)C)cncc(C)n1 51649,Cc1cc(C(=O)NCC(CNC(=O)C(C)C(F)F)CO)c(Br)s1 51650,S(=O)(=O)(c1cccnc1N1CCn2cnnc2C1)N(CC(C)(C)N(C)C)C 51651,C(=O)(C1CCOc2ccccc21)N1CC(NC(c2nocc2C)=O)CC(OC)C1 51652,C=C1CC2CCCC(C1)N2C(C1CCCN(C(c2csc(=N)[nH]2)=O)C1)=O 51653,C(=O)(C#CC1(C)CCCO1)NCC(C)N(C(c1cc(Cl)ccc1O)=O)CC 51654,c1(-c2n(CC(=C)C)c(SC)nn2)c(Br)ccc2c1OCCO2 51655,CCCCC(O)C(=O)N1CC(CC(=O)N(CCCOC(C)C)C)C2(CC2)C1 51656,C1(C(=O)NC2(CF)CCN(C(C3CCC(C)(C)C3)=O)C2)CC2(CC(=O)N2)C1 51657,N1(C(c2ncc(CC)cn2)=O)CCC2CCCC12C(N1CC2C(C1)C2(F)F)=O 51658,c1(C(=O)NC(C2CCCCN2C(=O)CC2CSC2)C)ccc(S(=O)(=O)N(C)C)cn1 51659,C1(C2CC2)(NC(c2cc(CNC(C3CCCC3)=O)[nH]n2)=O)CCCC1 51660,C(=O)(C1CC(=O)Nc2ncn(C)c21)NC1C(C)N(C(=O)C=Cc2ccsc2)CC1 51661,Cc1nn(C)c(F)c1C(N1CCC(CNC(c2ccnc(OC(F)F)c2)=O)C1)=O 51662,CCC(CC(=O)N1CC(C)(C)CC1CNC(=O)CCNS(C)(=O)=O)CC(C)C 51663,CC(CC(=O)NCCCNc1ccccc1)N(C1CCCC1)C 51664,C(CC(C)C)(C(=O)N1C(CC(=O)Nc2ccc(O)c(C)c2)C2CCCC12)OC 51665,CCCCS(=O)(=O)N1CCCC(C(=O)N(CCC2(C)CCO2)CCO)C1 51666,C(=O)(C#CC1(CC)CC1)N(CCNC(c1ccncc1N(C)C)=O)CC 51667,CC1CN(C(=O)OC(C)(C)C)CCN1N1CCSC(C)(C)C1CO 51668,N1(C(COC)=O)CCC(CNC(C2CC(Cc3ccccc3)=NO2)=O)C1(C)C 51669,c1(C(N2CCC(NC(c3cc(C(C)C)no3)=O)C(O)C2)=O)ccc2snnc2c1 51670,N1(C(C(CCC)N(C)C)=O)CC(N(C(=O)C=Cc2cccnc2)C)C2(CC2)C1 51671,CC1(C)CC(NC(c2cnc[nH]2)=O)CN(C(=O)Cc2csc(C3CCCC3)n2)C1 51672,C12(C(N3CC(CC(C)NC(c4c(C)occ4)=O)C3)=O)COCC(C1)C2 51673,C(C(CC(C)C)C(=O)N1CCC(C)(C)C(O)C1)NC(COCCC=C)=O 51674,CCC(CCC(=O)NCCC1(CO)CC1)NC(=O)CC1(C)CCCCC1 51675,C(=O)(C(C)CC(F)F)NCCN(C(C(CSC)(C)C)=O)C1CC1 51676,C12(NC(C(C#N)C3CC3)=O)CCC(CC1)N(C(=O)CC(=O)NC1CC1)C2 51677,NS(=O)(=O)c1cc(C(=O)OCC2C3CCCCCC23)c(F)c(Br)c1 51678,c1(C(=O)NCCCOCCC(=O)NC2CCC(N(C)C)C2)cnc(NC)cn1 51679,c1(CCC)cnnc(C(c2nnnn2CC2CC2)NC(CC(F)(F)F)C2CC2)c1 51680,N1(C(CCSCCC)=O)CCN(C2CCCN(C(=O)CSCCC#N)C2)C(=O)C1 51681,c1(OC)cc(NCC(C)CNC(=O)C(=O)NCC2CC2)ncn1 51682,c1(C(=O)NC2CC(NC(C34CCC(F)(CC3)C4)=O)C2)c[nH]c2ncc(Br)cc12 51683,C(c1ncc(C)[nH]1)=CC(=O)O.C1(F)(CC)CC(N(C(C2(c3ccno3)CC2)=O)CC)C1 51684,Cc1cc(=O)c(-c2nc(CO)nn2C(C)C(C)(C)C)cn1C 51685,C1(NC(C(C)(C)OC)=O)CN(C(c2cn(C)nc2C2CC2)=O)CC1C 51686,C(C)(C)(C(=O)NCC1(CNC(=O)Cc2ccnn2C(C)C)CC1)OCC 51687,CCCCC(C(=O)N1CCN(C(=O)CSC)CC1c1ccccc1)NC(N)=O 51688,c1(C(N(CCN(C(=O)CSCC(F)F)C(C)C)C)=O)cnn2cccc(Cl)c12 51689,N1(C(C2=C(C)CC2)=O)C(CC(N2CC3CCCCC23)=O)C2CCCC12 51690,c1(ON(C)CC)nc(C)cc(C)c1NS(=O)(=O)c1sccc1C1OCCO1 51691,c1(CC(=O)NCCC2CC(NC(CCc3ccc(C)s3)=O)C2)cn(C)nc1C 51692,c1(CC)csc(Cn2cc(CNC(=O)CNC(=O)C(N3CCOC3=O)C)nn2)n1 51693,N1(c2n(CC)c(C3(Cc4ccccc4)CC3)nn2)CCN(C)C2(CCOC2)C1 51694,C=CCC(Cc1ccccc1)C(=O)NC1CCCC1NC(=O)CC(F)F 51695,c1(NC2CCC(C)(C)C2)ccc(S(=O)(=O)NCCC2(C)CC2(F)F)cn1 51696,N1(C(C(C(C)C)OCC(C)C)=O)CCN(C(=O)COc2ccncc2)C(CF)C1 51697,c1(C(N2CC3C(CNC(C4(C)CCN(C)C4)=O)(C3)C2)=O)cc(F)ccc1C1CC1 51698,S(=O)(=O)(c1ccc(F)cc1)NCCC(=O)N(C(c1cn(C(C)C)nn1)C)C 51699,C1(NC(c2cc(F)n[nH]2)=O)CC(NC(C2CC(CF)C2)=O)C12CCC2 51700,C(C(=O)N(CCCCNC(=O)C(C)Sc1ccccc1)C)(C(C)C)NC(C)=O 51701,CC1C(=O)N(CC(=O)NC2(CNC(=O)Cc3nncs3)CCC2)C(=O)C1C 51702,C#CCCCCC(=O)N(C1CCC(NC(c2ccnnc2NC2CC2)=O)CC1)C 51703,N1(CC)CC(C(=O)NC2CCCN(C(C3CN4CCN3CC4)=O)CC2)CCC1=O 51704,n1(CC(=O)NC(C)CC(C)NC(C2CCC(=O)C2)=O)ncccc1=O 51705,C(C(C)(C)C(F)F)NC(C(C1CCN(C(=O)C=Cc2ccccc2)C1)C)=O 51706,c1(C(=O)NCC(CNC(Cn2c(C)ncc2)=O)CO)cc(C(F)(F)F)cc(N)c1 51707,c1(CCC(=O)NC(C=CC(=O)OCCC)C)nc2ccccc2o1 51708,N1(C(COC(C)C)=O)CCC(NC(=O)C(C)CCc2cccc(F)c2)C12CCC2 51709,c1(OC)ncccc1C(=O)NC(C)(C)CN(C(=O)Cn1ccc(C)n1)C 51710,c1(C(=O)NCCN(C(=O)C(C)C2CCCC2)C(C)C)cc2n(n1)CCCNC2=O 51711,c1(C(=O)NC(CNC(COC2(C)CCOCC2)=O)CO)ccc2sc(O)nc2c1 51712,C1(NC(C(C)NC(c2ccco2)=O)=O)(CNC(=O)C(C)O)CC2CCC1CC2 51713,Cc1cc(C(C)C(=O)N2CC(CNC(c3nc(C(C)(F)F)cs3)=O)C2)c(C)o1 51714,C1(C(N2CCCCC(C)C2)=O)COC2(C1)CN(C(c1ccc(O)cc1F)=O)C2 51715,c1(CC)nc(C)[nH]c1C(=O)NC(CNC(=O)C(C(C)C)SC)CC(C)C 51716,CC(C)(C(=O)NCC1CCCN(C(=O)CCOCC(F)(F)C(F)F)C1)C(F)(F)F 51717,C(N=c1ncc(CCOC)c[nH]1)C1CCC(C(C)OC)CC1 51718,N1(C(C(C(CC)CC)OC)=O)CC2CCCC(NC(=O)C(C)(COC)CC)C2C1 51719,c1(C(=O)NCCC(CCNC(CC(CC)O)=O)C)coc2cc(F)cc(F)c12 51720,c1(OC)ncnc(OC)c1CN1CCCC1CC(=O)Nc1sccc1CO 51721,CN1CCN(C(c2ccc(C3CC3)o2)=O)CC1C(N1CCCC1CO)=O 51722,CCCCCC(=O)NN(CCNC(=O)C(C(C)C)Oc1ccc(Cl)cc1)C(C)=O 51723,C1(N(C(=O)COC)CC)CCCN(C(C2CC(c3cccc(Br)c3)(O)C2)=O)C1 51724,CC(CC(=O)N1CCCC1C(=O)N=c1cc[nH]cc1C(=O)O)CC(C)(C)C 51725,C1(NC(c2c(C)nn[nH]2)=O)CCC2CC1CN2C(=O)CCCCCC#N 51726,c1(C(=O)NCC(C)(C)C(=O)N2CCCC2)cccc2c3c([nH]c12)CCCCC3 51727,C1(C(N(CCOCCCN(C)C(c2ccc(CO)s2)=O)C)=O)CCCCCN1C 51728,C1(NC(c2c(C)ccs2)=O)CCCCN(C(c2cnc(C(C)(F)F)s2)=O)C1 51729,C1(NC(c2c(CC)n[nH]c2)=O)CC2(CNC(=O)CCC3CCOCC3)CC1CO2 51730,N#Cc1cc(C(=O)NC2(CNC(c3scnc3Br)=O)CCC2)co1 51731,c1(C(N2CC(NC(C3CCC4CCC3O4)=O)C2)=O)cccc(Br)c1F 51732,C(=O)(C1=CCC(F)(F)CC1)N1CC(C2(NC(c3cc(C)no3)=O)CC2)C1 51733,C#CCCC(=O)NCCn1ccc(C(=O)NCC2(SC)CC2)c1 51734,C1(CNC(C=CCOC)=O)CC(NC(=O)CN(CC(=O)NC(C)C)C)C1(C)C 51735,c1(Oc2nnc(NC(=O)NC3C(C=C)OCC3)n2C)c(OC)cccc1C 51736,c1(C(=O)NC(C)CC(C)NC(=O)CC(F)(F)F)c(O)nc(=O)n2c1CCC2 51737,C(=O)(CS(=O)c1ccc(Cl)cc1)NC1CC(N(C(=O)C(C)(F)F)C)C1 51738,C1(C(=O)NC(C)CCCCNC(C2CC3(CCOC3)C2)=O)CCS(=O)(=O)C1(C)C 51739,N1(C(C(=O)NCC=C)C(C)C)CCOC(C)(C(F)(F)F)C1 51740,C(C(F)(C(=O)NCC1CCCCO1)C(C)C)NC(c1c(C)nsc1C)=O 51741,CCC(CCC(=O)NC1CC2(C1)CC2C(=O)N(C)CCOC)OC 51742,N1(C(C=Cc2n(C)cnc2)=O)CCC2CCC(C1)N2C(=O)CC1(C)CC1 51743,C12(NC(c3ncc(C(F)F)s3)=O)CCC(C1)N(C(c1ccncc1C(F)F)=O)C2 51744,C1(CNC(CC)=O)CCC2(CCN(C(c3ccccc3COC)=O)CC2)O1 51745,CON1CC(C(=O)NCC2(O)CCN(C(=O)Cc3ccn(C)n3)C2)CC1=O 51746,C12(CNC(CCc3onc(CSC)n3)=O)CCCN(C(=O)COC(C)C)C1C2 51747,c1(C(=O)NC2C(CNC(COc3ccc(OC)cc3)=O)CC2)cnc(Cl)c(N)c1 51748,C1(NC(C)=O)CN(C(=O)CCc2cc(Cl)cc(Cl)c2)CC12CC2 51749,c1(NC(C(c2ccccc2)N(CCC(C)(C)C)C)=O)nn(C)cc1Cl 51750,c1(C(=O)NCC=CCNC(c2c(SC)cccc2)=O)ncc(C)cc1Br 51751,CCCCCC(O)C(C)C(=O)N1CCCC(CCNC(c2ccoc2Cl)=O)C1 51752,c1(C(N2CC(NC(C=CC(C)C)=O)C(O)CC2)=O)cc2c(Cl)c(Cl)ccc2[nH]1 51753,CCCC(CC)C(=O)NC(CC(=O)NCC1(C#N)CCC1)C(C)OC 51754,n1(CC(C)CO)nc(-c2ccccc2)nc1CC1CC1(C)C 51755,c1(CNCCc2c(OC)cncn2)cc(F)cc(O)c1F 51756,Cc1cnn(CCC(=O)NCC(O)CNC(c2csc(Cl)c2)=O)c1 51757,C12(C(=O)NC(C)C(C)NC(c3cncn3C)=O)CC(CCO1)C2 51758,C1(CNC(C(c2cncnc2)C)=O)COC(C)(C)CN1C(c1ccoc1C)=O 51759,c1(OC)cccc(CCC(=O)NCC(C)NC(=O)C(C)C(F)(F)F)c1F 51760,C12(SCC(N3CC(C)C(C)(CN=c4ccnc[nH]4)C3)=O)CC3CC(CC(C3)C1)C2 51761,c1(C(N(C2CCN(C(C(CC)O)=O)C2)CCO)=O)ccc2c(c1)nc(O)n2C 51762,c1(CC(N2CC3CC(CNC(C4(CC5CC5)CC4)=O)C2C3)=O)c(Cl)cccc1Cl 51763,Cc1cc(CNC(=O)CC(C)NC(c2ccccn2)=O)cc(C#N)c1 51764,c1(CC)ccnc(C(=O)NCc2ccoc2C(=O)NC2COC(C3CC3)C2)c1 51765,N1(C(C2(C)CSC2)=O)CCC2(CC1)CC2C(=O)NCCCCc1ncc[nH]1 51766,C=C=CC(C)C(=O)N1CCCC1CN(C(c1cc(C(C)(C)C)on1)=O)C1CC1 51767,c1(NC(C2N(C(c3c(OC)ccc(F)c3)=O)CC(O)C2)=O)cccc([N+](=O)[O-])c1 51768,CC(CCCNC(=O)CCc1cnoc1)NC(=O)CSc1nncs1 51769,C1(NC(C2C(CC)C2)=O)CC2CC(NC(c3cc(Cn4cccn4)on3)=O)CC12.COC 51770,c1(CCC(=O)NC23CC2CN(C(c2ccoc2Cl)=O)C3)nnc(O)nc1O 51771,Cc1ccc(O)cc1C(N1CCC(NC(=O)C=C2CCN(C)C2)C(F)C1)=O 51772,C#CC1(C(=O)NC(CN)C2CC2)CCN(C(=O)C(C)OC)C1.C1(O)CCCC1 51773,c1(C(=O)NCC(C2CCCN(C(C(C)C)=O)C2)(C)O)cc2cccn2c(O)n1 51774,N1(C(c2ccc(C)nc2)=O)CCC2C(CCCN2C(c2c[nH]cc2C2CC2)=O)C1 51775,c1(C(C)NC(=O)NC(CC2CC(F)(F)C2)CO)nc2c(o1)CCSC2 51776,c1(C(=O)OC)c(C)[nH]c2ccc(NC(=O)NCC3CS(=O)(=O)CCO3)cc12 51777,CCC(CC(=O)NCCOCCNC(C1CC2(CCC2)CO1)=O)CC(C)C 51778,N1(C(C2(C(=O)OC)CC2)=O)CC(NC(c2ccn(C(F)(F)F)n2)=O)CC(F)C1 51779,Cc1cnccc1-c1cn(CCO)nn1.C1(CC(N2CCCC2)=O)CC2CCC1O2 51780,C#Cc1cccc(OCC(=O)NC2CCOCC2NC(=O)CC(=O)N(C)C)c1 51781,c1(C(N2CC(CN(C)C(C3CCCS3)=O)C2)=O)csc2nccn12 51782,C(C1=CCN(C(c2cc(CCCO)on2)=O)CC1)NC(=O)C(F)=CCCF 51783,C1(CC=C)(C(=O)NC(CSC)CCOC)CCCN1C(c1cccs1)=O 51784,C1(NC(c2cc(C)nc(C)c2)=O)CN(C(=O)CC2CCCN(C)C2)CC(C)(C)C1 51785,C(C(C)(C(=O)N1CC2C(C)C2C1)NC(c1cccc(CC#N)c1)=O)SC 51786,c1(C(=O)NCCCCCO)nc2ccc(Br)cn2c1F 51787,C(CC(C)C)(C(=O)NC1CC2(C1)CC2NC(c1ccc(NC(C)C)nc1)=O)OC 51788,C1(CC)CN(C(C2(C)C=CCC2)=O)CCN1C(=O)COc1cc(C)on1 51789,C12(C(=O)NC(CC)C(=O)NC)CC(CN(C(c3cnccc3C#N)=O)C1)C2 51790,N1(C(C2N(C)CCN(C(C3CC3C3CC3)=O)C2)=O)CCC(C2(C)CC2)CC1 51791,C=CCCC1C(=O)N1c1cn(C)nc1Oc1ccccc1.c1(C(F)(F)F)ccccc1F 51792,Nc1ccc(O)c(C(=O)NCc2ccccc2Oc2cccc(Cl)c2)c1 51793,Cc1ncnc(N2CCC(CNC(=O)COC(F)(F)F)C2)c1Br 51794,c1(C(=O)NC(CC)(C)CNC(=O)COCP(C)(C)=O)ccc(Br)cc1 51795,N(C(=NCC(C)C)N1CCC(COC)C1)C(c1ccc(F)cc1)C#C 51796,c1(C(N2CC(OC)(CNC(=O)C3=C(Cl)CC3)C2)=O)c(C)nc2cccnn12 51797,c1(OC)cncc(C(=O)NC2CN(C(=O)C(CO)N(C)C)CC2CC(C)(C)C)n1 51798,C(=O)(CC(C)CNC(C1CCOC1C1CC1)=O)NCC(CSC)OC 51799,N1(CC(N2CC(c3n(C)cnc3)C(NC(=O)CNC=O)C2)=O)CCC(=O)NC1=O 51800,N1(C(c2ncc(NC)nc2)=O)CCN(C(=O)C=CSC)C2CS(=O)(=O)CC12 51801,C(C(C(C)C(C)C)NC(=O)Cn1ccc(C)cc1=O)NC(C)=O 51802,C1(C(=O)NC(C)CN(C)C(c2cn(C)nc2C2CCCO2)=O)CN2CCC1CC2 51803,n1(CC(N2CC(OC)C(NC(C3CCC=CCCC3)=O)C2)=O)c(C)c(C)sc1=O 51804,C1(CNC(CNC(=O)NC)=O)CCCN(C(C2CCC(C)(C)C2)=O)C1 51805,C12(CNC(c3cc(C)sn3)=O)CC3CC(CC(C3)C1NC(C1CNC(=O)C1)=O)C2 51806,CC(CN=c1[nH]nco1)(C1CC1)NC(c1cc(S(N)(=O)=O)co1)=O 51807,CCC(CC)C(=O)NCc1nnn(C)c1C(N1CCCCC1C1CC1)=O 51808,C1(C(=O)NC(C2N(C(CCC(=O)NC)=O)CCCC2)C)C2(CCC2)C12CCC2 51809,C(=O)(C(C)N(CC(C)NC(=O)C(C)C1CC1)C)N(C1CC1)CC 51810,n1(CC)nc(C)cc1C(=O)NC(C)C(C)(C)NC(C1CNC(=O)C1)=O 51811,C1(NC(Cn2c(C)ccc2C)=O)CCN(C(C2CC(=C(F)F)C2)=O)CC1C 51812,N(C1CCCn2ncnc21)C(C(C)(N(C(COC)=O)C)C1CC1)=O 51813,c1(NC(C(OC)OC)=O)cc(Cl)c(Br)cc1C.C1(=O)N(C)CCO1 51814,C(=O)(CC1=CCOCC1)NCC(CC)N(C)C(C1CC(C)(C)CCO1)=O 51815,N1(C(C(CC(C)=O)(C)C)=O)CCC2(CCCN2C(=O)CC2CCCC2C)C1 51816,N1(C(C=CC(=O)OCC)=O)CCCC2CCN(C(c3n[nH]c(C4CC4)n3)=O)CC12 51817,N1(C(=O)Cc2ccccc2)CC2CC(C1)N2C(=O)C(F)C1CCOC1 51818,C(C(C)(C)CC(=O)NC1CCOCC1NC(=O)CSCC(F)(F)F)OC 51819,C(C(C(=O)Nc1cnn(CCF)c1)C(C)(C)C)NC(c1c(C)n[nH]c1C)=O 51820,c1(NC(C)C)ncc(Br)c(C(N2CCN(C(C3CC34CC4)=O)CC2)=O)n1 51821,N1(C(C(N2C(=O)CCC2=O)C)=O)CC2CN(C(C3C(C)(C)C3(C)C)=O)CC2C1 51822,c1(CC(N2C(CCNC(C(CC)C)=O)CCCC2)=O)cc(C)cc(F)c1 51823,Cc1nc(CNC(C2C=CCCN2C(c2cc(C3CC3)[nH]n2)=O)=O)[nH]c1C 51824,CC1(C)CCC(C(=O)NCCc2ccncc2)(NC(C2CC(N(C)C)C2)=O)C1 51825,N1(C(C(C)(C)C2CCCCO2)=O)CCC12CN(C(=O)CCSc1ccccn1)C2 51826,C1(C(=O)NCCOCCCNC(c2ncsc2C2CC2)=O)CCC(C2CC2)C1 51827,C1(C(=O)NC(C(=O)O)C2(C(=O)O)CCC2)COC2CCCCC12 51828,N1(C(c2c(OCC(=O)NC)cccc2)=O)CC2CC1CN2C(C1CCOC1=O)=O 51829,c1(C(=O)NC(C)CNC(=O)CN2CCSCC2)ccc(SCc2cnc[nH]2)cc1 51830,N1(C(C2N(C(c3c(CC)cno3)=O)CC=CC2)=O)CCCC(O)(C(N)=O)C1 51831,c1(OC)c(C)csc1C(=O)NC1CN(C(c2cn[nH]c2)=O)CC1C 51832,CC1CCCc2ncc(C(=O)NC3CC34CCN(C(=O)Cc3cnoc3)CC4)n21 51833,C1(CC)(NC(c2ccn(C)c2)=O)CCCN(C(C2CCCN(CC(C)C)C2)=O)C1 51834,C12(CNC(C3(C#C)CCC3)=O)CCC(CC1)N(C(c1ccoc1)=O)C2 51835,c1(C(c2n(CCCF)nnn2)NC2(Cc3ccsc3)CC2)ccccc1OCC 51836,C1(C(N(CCN(C(c2cnn(CCF)c2)=O)CC)CC)=O)CC(NC)CCO1 51837,S(=O)(=O)(c1ccc2ccccc2c1)NC(c1cc(N)n(-c2ccccc2F)n1)=O 51838,c1(C(=O)NC(CCOC)CNC(=O)Cc2cc(C)ns2)nccc2cc[nH]c12 51839,C1(CC(=O)NCCc2ccccc2O)CN(C(c2cccnc2)=O)CC12CC2 51840,c1(C(CNC(N2CCCC2c2ncno2)=O)O)cccc(Br)c1 51841,N1(C(CC2(COC)CCCC2)=O)CC2CCN(C(=O)Cc3csc(C)n3)CC12 51842,Cc1ccc(C(N2CCC(CN)C2)=O)cc1C1C(C(=O)NC2CC2)C1(C)C 51843,N1(C(CCCCCCC)=O)CCN(C(C2CCc3nn[nH]c3C2)=O)CC2(CC2)C1 51844,CCC(CCC(=O)OC)N=C(NCCCCC(C)(F)F)NCC(C)(C)C 51845,C1(NC(c2ncn(CC)c2)=O)CCC(N(C(=O)COc2cn[nH]c2)C)CC1 51846,C1(C(=O)NCCN(C(=O)C(F)C2CCOC2)CCOC)CCC=CCCC1 51847,Cc1cccc(C(=O)NC(CNC(=O)CN2CCOCC2=O)C(C)C)c1F 51848,c1(OC)ccc(C)nc1C.N1CCOC(C2CN(C(C3(OC)CC(CF)C3)=O)C2)C1 51849,c1(C(N2C(C)CN(C(=O)CCC#N)CCC2)=O)cc(=O)c2cc(Br)ccc2o1 51850,Cc1csc(C(N2CCCCC2CCC(=O)NCC(C)(O)C(C)C)=O)c1C 51851,CC(N=c1nn[nH]n1C)C1CCCCN1C(c1c(Cl)cnn1C)=O 51852,N1(C(CC(C=C)C)=O)CC2CC(C1)C(CO)C2NC(=O)CCCCSC 51853,N1(C(C(C=C=C)C)=O)CCC(CC(=O)NCC(C2CCCC2)C)C1(C)C 51854,CCC(CC(=O)NCC1CCC(CNC(=O)C=CC2CCCN2C)CC1)SC 51855,CN1CCC(NC(N2CCOC(CO)C2)=O)C(c2ccccc2)C1 51856,N1(CC(c2nccs2)=O)CC(n2cc(C(c3ccccc3)O)nn2)C(O)C1 51857,C1(NC(C=NOC)=O)CN(C(=O)CCC2OCCO2)C2(CCOCC2)C1 51858,c1(OC)ccsc1C(=O)NCC1CCCC1C(=O)NOCc1nc[nH]n1 51859,c1(C(N2CC(CNC(C3CCC34CCC4)=O)C2)=O)cccc(C#CCO)c1 51860,c1(C(=O)NCC2C(C)CCN(C(=O)COc3ccsc3)C2)cc2ccccn2n1 51861,C1(NC(c2cc(CCC)[nH]n2)=O)CCN(C(C2OC3CCC2CC3)=O)CC(O)C1 51862,C1(CNC(C=CSC)=O)CCN(C(=O)CCc2ccccn2)CC1(F)F 51863,c1(C(=O)NC(c2ccccc2F)CNC(C2(C)CC2(F)F)=O)nccnc1O 51864,CC1CC(C(N2CCN(C(=O)CCNc3ncccn3)CC2)=O)CC(=O)N1 51865,N1(C(CC(C)(C)OC)=O)CCC2CCCC12C(N1CC2C=CC1CC2)=O 51866,C1(NC(=O)CC2CC=CCC2)CCC2(CC1)CCN(c1nc3ccccc3o1)C2 51867,c1(C(N2CCOCC(CNC(COCC=C)=O)C2)=O)ncc2ccccn12 51868,CC1(C(N2CC3(CCC3NC(=O)Cc3ccccc3F)C2)=O)CCCCCC1 51869,CC(C)C(N=c1[nH]nc(CC(F)(F)F)o1)C(C)NC(=O)CCC1CC(C)(C)CO1 51870,C1(CNC(Cc2c(C)nc(C)s2)=O)CC2(CO1)CN(C(=O)C(C)CS(C)(=O)=O)C2 51871,N1(C(C=Cc2ccc(C)s2)=O)CCCCCC1CNC(=O)CC1CC=CCN1C 51872,CCCC(O)CC(=O)N(CCNC(=O)C(F)C(C)(C)O)CCOC 51873,C=CCN=c1ccc(S(=O)(=O)N2CCCCC2c2ncc(Br)cn2)c[nH]1 51874,N1(C(c2cc(OC)ncn2)=O)CC(NC(=O)COC(F)(F)F)CC1(C)C 51875,C1(CC(=O)OCC2(C)CCCC2O)(NC(=O)OC(C)(C)C)CCCCC1 51876,CCC(CNC(c1cc(C#N)oc1C)=O)(CC)C(=O)NC12CCCCC1C2 51877,CCCCS(=O)(=O)CC(=O)NCC(CO)NC(c1csc(C)n1)=O 51878,Cc1ccc(C)n1CC(N1CCC(C)C1C(=O)N(CCC(O)CO)C)=O 51879,C(=O)(C1=CS(=O)(=O)CCC1)NC1CCC(CNC(C2(C#C)CCCC2)=O)C1 51880,N1(C(CSc2ccc(C)cc2C)=O)CC(CNC(=O)CC#N)C2(CCC2)C1 51881,C1(NC(c2nccc(C)c2)=O)CCN(C(c2cncc(C(C)(C)C)c2)=O)CC1O 51882,C(C(=O)N(C(C(=O)NCC1CCOC1C)C1CCOC1)C)(C(C)(C)C)OC 51883,N1(C(C(C)=CC=C)=O)CCC(C(=O)NCc2ncsn2)=C(F)C1 51884,c1(C(N(C(C)C(=O)N(CCC(=O)NC2CC2)C)CCC)=O)cnc(C)o1 51885,C(C(C)(C1CC1)NC(=O)CNS(C)(=O)=O)NC(COC(CC)C)=O 51886,c1(COC)csc(C(C(=O)NC(C)(C)C)N(C2(c3cc[nH]n3)CC2)C)c1 51887,Cc1cc(C)n(CCC(N2CC3CC2C3NC(c2ccc(C(F)F)cn2)=O)=O)n1 51888,c1(NC(=O)CC2CCCC2C(N2CCCC2C2CCCOC2)=O)ncccc1O 51889,C1(NC(c2c(C)ccs2)=O)CC(F)(F)CC1NC(=O)COc1ccccc1 51890,Cc1cc(CNC(=O)NCC(c2ccccc2Cl)O)ccc1-c1ccncc1 51891,C#CC1CC2CCC1N(C(=O)C=CC(C1CC1)NC(=O)CSCCOC)C2 51892,Cc1nsc(CNC(c2nnnn2CCN2CCOCC2)C2CC=CC2)n1 51893,C1(CC)(CO)CCCN(C(=O)C(=O)NCCOCCS)C1.c1(O)ccccc1 51894,C1(C(=O)NC2(CC#C)CC2)C=CCN1C(C1CC(n2cccn2)C1)=O 51895,c1(CC)nc(C)c(C(=O)NC(C)CCN(C(=O)COCC2CCCO2)C)s1 51896,C(C1COc2ccccc21)NC(NC(c1ccc(Br)cc1)C#C)=NCCF 51897,C(=O)(CC(=O)N=c1ccn(-c2ccc(Cl)cc2O)[nH]1)NC(N=c1ccn(C)[nH]1)=O 51898,c1(OC)ccc2c(c1)CC(C(=O)NC1CCCC1NC(C1(CO)CC1)=O)CO2 51899,CCCC(C)(O)C(=O)N1CC(NC(c2ccc(CC)c(F)c2)=O)C1 51900,C1(C(=O)NC2CC(CCNC(c3cc(C4CCC4)no3)=O)C2)CC2(C1)OCCO2 51901,N1(C(=O)C=Cc2ccco2)CCCC2(NC(C3CC(O)C3)=O)CC2C1 51902,c1(C(N2CC(OC)(CNC(C3CC3CF)=O)C2)=O)c(O)cc(=O)n2c1CCCC2 51903,N1(C(C(C)SCCCC)=O)CCC(C(=O)NOCCCCC2CC2)C(C)C1 51904,c1(OC)cnc(Cl)[nH]c1=NC1CC2CCC1N(C(c1cc[n+]([O-])cc1)=O)C2.C1CC1 51905,c1(C(N2CC(F)(C(=O)NCC3(CCO)CCC3)C2)=O)ncccc1Cl 51906,c1(C(=O)NC2CC3(CC(CNC(C4ON=C(C)C4)=O)C3)C2)c(Br)ccc(F)c1C 51907,C1(CNC(c2cnc(CC(C)(C)C)s2)=O)CN(C(C2CSCCS2)=O)CC1O 51908,c1(C(=O)NCC2CCC(NC(=O)C(Cl)=CCl)C2)cccc(C(F)(F)F)n1 51909,C(=O)(CCCCCC(C)C)NCC1N(C(c2c(C)ccc(Cl)c2)=O)CC(F)C1 51910,c1(NC2CCN(C(n3cc(CSC)nn3)=O)CC2)ccnc(OC(C)C)c1 51911,C1(CC(=O)N(C(C)C(=O)NCCn2cnnc2C)CC)CCC(C)CO1 51912,N1(C(C(C)Cc2cccc(O)c2)=O)CCC(F)(F)C(CNC(=O)CP(C)(C)=O)C1 51913,N1(C(C=NOC)=O)CCC(C(C)(C)NC(=O)C(C2CCOCC2)OC(C)C)CC1 51914,CCC(C(=O)N1CCN(C(c2ccnnc2O)=O)C(CO)C1)C(C)(C)CC 51915,CC1(C=CC(=O)N(C2CCCN(C(=O)CC3CC34CC4)C2)CCO)CCOCC1 51916,S(=O)(=O)(CCCCS(N)(=O)=O)N1C(C(C)(C)O)C(O)CC1 51917,n1(CC(=O)NC(C(C)NC(CCC(=O)NCCC)=O)(C)C)nc(O)ccc1=O 51918,C(=O)(C(F)(CNC(c1ccccc1C1CC1)=O)C(C)C)N(CC=C)CC 51919,C1(C(=O)NC(CC)CC(=O)OC)CCC2(CN(C(=O)C(Cl)(Cl)Cl)C2)O1 51920,c1(-n2c(COCC(C)C)nc(-c3cnccn3)n2)ccc(Cl)c(Cl)c1 51921,CCC(CC)C(C(=O)NC1(C(=O)NCC(C)CC2CC2)CSC1)OC 51922,C(N=c1[nH]cnc(NCc2ccc(Cl)c(F)c2F)c1C)c1cc(CC)no1 51923,c1(CC)nc2c(C(=O)NCC(C)(CO)NC(=O)C(C)C3CC3)ccnc2[nH]1 51924,CCC(CC)CCC(=O)NCC1CCCN(C(C2(CC)CC=CCC2)=O)C1 51925,Cc1nnc2c(C(N3CCCOC(CNC(=O)C(C)(C)C)C3)=O)cccn12 51926,C1(C(C(=O)NC(c2cccnc2)C(=O)N(C2(CC)CC2)C)C)CCOCC1 51927,c1(OC(C)C)cncc(C(=O)NCCCC(C)(C)NC(c2ccco2)=O)c1 51928,c1(OC)cc(Cl)c(Br)cc1CN=c1[nH]c(-c2ccc(O)c(C)c2)cs1 51929,c1(C(=O)NCCC2N(C(C3C(CC)C3)=O)CCC2)cc2c(nc1O)CCOC2 51930,N1(C(c2c(COC)noc2)=O)CCC2(NC(c3cnc(C)nc3O)=O)CCCC12 51931,C(c1ccnn1C)=CC(=O)NC(C(=O)NC(c1n(CC)ncc1)C)c1ccco1 51932,c1(C(N)=O)ccc(C(=O)NCC2(O)CC(C(N3CC(c4cc(O)no4)C3)=O)C2)o1 51933,CCCC(C(=O)NCC(CNC(=O)Cn1cnccc1=O)OC)c1ccccc1 51934,C1(C(=O)NCC(CSC)OC)CCC(O)CN1C(=O)Cc1nocc1C 51935,N1(C(C2N(CC)CCC2)=O)CC2CC(C(=O)NCc3cc(C)sc3C)(C2)C1 51936,C1(NC(c2cc(OC)n(C)n2)=O)CN(C(=O)C2CC2)CCC1c1ccccc1 51937,CC1CCN(C(c2ccccc2C2CC2(F)F)=O)CC1NC(C1CCCS1)=O 51938,c1(CN(c2cncc(Cl)c2)C(=O)NCC)nc2c(s1)CCCC2 51939,c1(COC)ccc(C(N2CC(NC(=O)CC3COC(=O)C3)CC2C)=O)cc1 51940,c1(C(N2CCSC2c2ccc(Cl)s2)=O)cccnc1NC(=O)Cn1cccn1 51941,CC(CC(F)F)C(=O)N(CCCCCCNC(C1(F)CCC1)=O)C 51942,C12(C(N3CCCC(CCC(=O)N(C)CCC4CCCC4)C3)=O)CCCC1C2(F)F 51943,n1(CC(=O)NC(c2ccccn2)(C)C)cc(C#N)c(O)nc1=O 51944,C(=O)(C(C)(C)C(c1ccccc1)NC(C1CC(=O)NOCC1)=O)OC 51945,Cc1c(C(=O)NCC2CC(CNC(=O)CSC(F)F)CO2)sc2ccc(F)cc12 51946,C(=O)(C(C)(C)C(=O)NCC(O)CN(C(=O)CCn1cc[nH]c(=O)c1=O)C)OC 51947,C1(CC=C)(NC(C2CC2(C)C)=O)CCN(C(=O)Cc2c[nH]ccc2=O)C1 51948,C1(F)(C(=O)NCCC2(O)CCN(C(C(C)SC)=O)C2)CC2(CCC2)C1 51949,c1(C(=O)NC2CCN(C(CN3CCP(C)(=O)CC3)=O)C2)ccc2nsnc2c1 51950,c1(C(N2CC3C(NC(C(C)S(N)(=O)=O)=O)(C3)C2)=O)cccc2cc(O)ccc12 51951,N1(C(CCCCC)=O)CCN(C(=O)C(C)OC2CCCCC2)CC1CC(F)F 51952,CC1(C)CCC=C1C(=O)NCCNC(n1ccc(=O)n(Cc2ccccc2)c1=O)=O 51953,C(=O)(CCCCCCCCCO)NCC1C(C)(C)CN(C(C2C=CCCC2)=O)C1 51954,Cc1nc(N2CCC(NC(=O)C(C3CC3)C3CC3)CC2C)cc(C#N)n1 51955,c1(C(=O)NCCC2(O)CN(C(c3cnc(OCC)s3)=O)C2)ccc(C(C)C)nc1 51956,C1(O)(CNC(C(CCOC)OC)=O)CCCN(C(=O)Cc2cnc(C)s2)CC1 51957,c1(CCC(=O)N(CCCNC(=O)CCCCC2CC2)CCO)c[nH]c2ncccc12 51958,c1(C(=O)NCC2C(NC(COCC)=O)C2)cc(OC)c(OC)cc1N 51959,N1(C(c2cc(C)cc(OCC)c2N)=O)CC2CC(C1)CN(C(C1CC13CC3)=O)C2 51960,CCCCCC(O)C(=O)N1CCCC1Cn1cc(CNC(C2(F)CC2)=O)nn1 51961,N1(C(CC(C)(F)F)=O)CCOC2(CCN(C(c3sccc3SC(F)F)=O)CC2)C1 51962,c1(CN2CCC3(C(C(=O)NCCn4cccc4)C3)C2)cn2ccccc2n1 51963,N1(C(=O)CC(F)F)CCN(C2CCC(NC(=O)C(F)C3CCOC3)CC2)CC1 51964,CCC(O)CC(=O)NCC1CCC(NC(=O)CC2CSC2)CC1 51965,CCCC(CCCNC(c1ccc(=O)n(C)c1)=O)NC(c1sc(C)cc1C)=O 51966,c1(C(=O)NCC(C)N(C(c2cc(CC)[nH]n2)=O)C)ccc2cnsc2c1 51967,N1(CC(C)NC(=O)CCc2ccc(C(F)F)cc2)CCN(C(=O)C=C2CC2)CC1 51968,c1(C(N2CC3C(CNC(C4CC=C(C)CC4)=O)(C3)C2)=O)cc2cn[nH]c2cn1 51969,C(=O)(C1CCCn2ncnc21)NC(C(C)C)CNC(=O)CCC(N)=O 51970,CC(C)(CO)C(=O)NC1(C)CCN(C(=O)COc2cccc(Br)c2)C1 51971,N1(C(C(c2ccc(Cl)cc2)C)=O)CC(NC(=O)C=CC(N)=O)Cc2ccccc21 51972,C1(C(N2CCC(CCN(C(=O)CN(C)CCO)C)CC2)=O)CCn2ncnc2C1 51973,C1(CNC(CC(n2c(CC)ncc2)C)=O)CC2CCC1N(C(=O)Cc1cc[nH]n1)C2 51974,N1(C(Cc2c(Br)cn(CC)n2)=O)CC(C2(NC(=O)C3=CCCS3)CC2)C1 51975,CC1CCOCC1C(=O)NCc1cccc(C(=O)NC2(CO)CCC2C)n1 51976,C=CC1(CNC(C2(C)CC(O)CN2C(=O)C(C)c2cccs2)=O)CCOCC1 51977,C1(C(N2CCC(NC(=O)CCCCCF)C2)=O)(COC)CCCNS1(=O)=O 51978,C1(C2(O)CCC2)(C(=O)NC2C(CNC(c3cnc(C(C)(C)C)[nH]3)=O)C2)CC1 51979,n1(CC(=O)NCc2ncc(C(=O)O)s2)cc(CCO)nn1 51980,C1(CN(C)C)CC(O)CN1C(C1C=CCN(C(=O)CCCNC(N)=O)C1)=O 51981,C1(C(N2CC(NC(C=C(C)C(F)F)=O)C3(C2)CC3)=O)CCOCC12CCCCC2 51982,N1(C(C(C)n2cncn2)=O)CCC(CNC(=O)CNS(N)(=O)=O)C(C2CC2)C1 51983,C(=O)(C1CCCc2ncnn21)N1CCN(C(c2[nH]nnc2C2CC2)=O)CC(C)C1 51984,N1(C(c2c(C)c[nH]n2)=O)CCC(O)C(C(=O)NCc2ccccn2)C1 51985,c1(OC)ncc(CNC(=O)C(C2CCC(=O)N2)C)s1 51986,Cc1cc(C(=O)NC23CCCN(C(c4ccsn4)=O)C2C3)ccc1Br 51987,c1(C(C)NC(C2C(NC(c3c(C)nc(CC)s3)=O)C2)=O)ccc2c(c1)OCO2 51988,N1(C(CCC(=O)NC)=O)CCN(C)C(CNC(C2(c3nccs3)CC2)=O)C1 51989,c1(C(=O)NC2CCCC(N(C(=O)Cc3ccoc3)C)C2)ccc2ccn(C)c2c1 51990,N1(C(CC)C(=O)O)CCc2c[nH]c(=N)nc2C1 51991,c1(C(C)C(=O)NC2CC(CNC(c3ccc(N)cn3)=O)C2)cc2ccccc2o1 51992,N1(C(c2c(N)ncc(O)c2)=O)CCCC2(CCCCC2NC(C2CC23CC3)=O)C1 51993,C1(CNC(c2n(C=C)ncc2)=O)CC2CCC1N2C(C1SCCCS1)=O 51994,C1(NC(=O)CCCN2C(=O)CNC2=O)CC2CC(C1)N(C(c1nccs1)=O)C2 51995,C(C(O)CCNC(C1(n2nccn2)CC1)=O)NC(COCCSC)=O 51996,c1(C(=O)NC(CNC(C(c2ccc(CC)cc2)C)=O)C2CC2)cc(C)cc(N)c1 51997,N1(C(C(CC)CC)=O)CCC(NC(=O)C(CC)n2ccc(C3CC3)n2)C2(CCC2)C1 51998,CC1CN(C(C2(C)CCCOC2)=O)CCC1CNC(c1ccc(F)cc1F)=O 51999,C1(CNC(C(C)NC(N)=O)=O)CN(C(=O)CC2CC(F)(F)C2)CCC1(C)C 52000,N1(C(C2CC(C#N)(OC)C2)=O)CC(NC(c2ccc(OC)s2)=O)C2(CCC2)C1 52001,C=C(C)C(O)CC(=O)NC1CN(C(c2cc(OC)ccc2F)=O)CC1C 52002,CN1CC(C(=O)NCC(c2ccc(F)cc2)Nc2cnc(F)cn2)CC1=O 52003,Cc1ncc(C(=O)NC2CC(CNC(c3ccc(F)cc3)=O)CC2O)n1C 52004,Cc1cc(Cl)ncc1CC(=O)NC1CCC(CNC(=O)CC2CCC3CC23)CC1 52005,C1(NC(CCCC)=O)C2CC3C1C3C2C(=O)NCC1CCC(C(N)=O)O1 52006,C(C(CC(C)C)c1nccn1C)CCCCC.C(=O)(C(F)(F)Cl)NCC 52007,c1(-n2c(C(CC=C)CC)nc(-c3occc3C)n2)ccc(C)c(F)c1 52008,C=C=CCCC(=O)N1CC(CNC(C2CN(C)C(=O)N2)=O)C1 52009,c1(C(=O)NCC(C)CNC(c2nnn3c2CCC3)=O)nccc2ccncc12 52010,c1(C(N2C(CCNC(C(CC#C)O)=O)CSCC2)=O)cccc(F)c1C 52011,Cc1nc(CC(=O)NCC(O)CN(C)C(c2cc(F)n(C)n2)=O)[nH]c1C 52012,CCC(F)(F)C(=O)NCC1CC(NC(c2cnc(C)nc2)=O)C1 52013,c1(C(N2CC3C(CNC(=O)C4=CC5CCC4C5)(C3)C2)=O)cc(Cl)cc([N+](=O)[O-])c1 52014,CC(C)(C)C(C#N)C(=O)N1CC=CC(C(=O)Nc2cccc(F)c2)C1 52015,C1(NC(CC2CCN(C(c3c(COC)cco3)=O)C2)=O)CCn2cnnc2C1 52016,C(=O)(C1=NOC2COCC12)NC(C(C)C)CCN(C(=O)CCC1CC(F)(F)C1)C 52017,C1(C(=O)NCC(C=C)(F)F)CC2(CCO2)C1 52018,N1(C(CC(C)O)=O)CCCCC(N(C)C(c2cc(C(F)(F)F)ccn2)=O)C1 52019,C1(CC(=O)NC(C#C)C(C)C)CC2(CC2)CN1C(c1cc(CO)n(C)n1)=O 52020,C(=O)(C(C)(C)CC(C)(C)C)NC1CN(C(C(C(CC)CC)C)=O)CC2(C1)CC2 52021,c1(C(N(C(CC)C(=O)N2CC(C)(CF)C2)C)=O)cc(=O)cc[nH]1 52022,C1(C(=O)OCC)CCN(C(=O)CN(C)CCOC(C)=O)CC1(C)C 52023,C1(C(=O)NCC2OCCN(C(C(C=C)O)=O)C2)CC2CCC1CC2 52024,Cc1nc(NCCN2CC3CCC3(CO)C2)cc(N2CCC(CCO)C2)n1 52025,CC(C)(CNC(=O)NCC1CCC12CCCO2)CS(C)(=O)=O 52026,c1(CC(=O)NC(C)C(C)(C)NC(=O)CCCN2CCCC2)ccc2c[nH]nc2c1 52027,c1(C(=O)NC(C(N2CCCC(C=C)C2)=O)C2CCOC2)coc2ccccc12 52028,C1(C(=O)NC2CCCN(C(C3CN(CC)C(=O)C3)=O)C2)CCOC(C)(CC)C1 52029,N12CCC(C)(CC1)NC2=O.Cc1cncc(N(CCO)Cc2cccnc2)c1 52030,CC1CN(C(=O)CC2CC2CNC(=O)C=Cc2cccnc2)CCS1=O 52031,c1(OCCC)ccc(C(=O)NC2(CO)CCOC2)cc1OC 52032,c1(C(N2CCCC(O)(CNC(C(=O)NCC)=O)C2)=O)cnc2cc(OC)ccn12 52033,C1(C(N(CC(C)NC(=O)CCc2ccc(N)cn2)CC)=O)CCc2nn[nH]c2C1 52034,c1(C(N2CC(NC(C(C)SCCCC)=O)C(C)C2)=O)sc2nccnc2c1NC 52035,C(=O)(C1=CCCOCC1)N1C(C)CC(C(=O)NCCCCCCF)CC1 52036,C1(NC(C2CN(CC)C(=O)N2)=O)CN(C(c2cocn2)=O)CCC1F 52037,C(=O)(C1CCc2ccccc21)N1CCC(N=[N+]=[N-])(C(=O)NCC(C#C)C(C)C)C1 52038,N1(CC)CCOCC1C(=O)NCCCCC(=O)NCCC1CCCN(C)C1 52039,C1(C(=O)NC(C)(CO)C2CCC2)CCN(C(=O)C(CO)NC(N)=O)C(C)(C)C1 52040,CC1OCCCC1C(=O)NC1CCC(NCC(O)CNC(N)=O)CC1 52041,C(c1ccccc1)=CC(N1CC(CCCCNC(CC2C(CC)C2(C)C)=O)C1)=O 52042,C(=O)(C(O)C(C)(C)C)N1CCC(O)(CN(C(CCOCCC)=O)C)C1 52043,Cn1cc2c(n1)CCCC2C(=O)NC1CC(F)CN(C(=O)CC(C2CC2)C2CC2)C1 52044,C(=O)(C1=CCCOCC1)N1CC(COC)N(C(=O)C(n2cc(C)cn2)C)CC1 52045,CC1(C)CCC=C1C(=O)N1CCCCC1CNC(c1cn2cnnc2cn1)=O 52046,C(CC(F)(F)F)N(C)C(C1(CNC(=O)CC2CCOCC2)CC1)=O 52047,Cc1cccc(C(C2CC2)NCC(N2CCC(c3cn(CC(=O)O)nn3)CC2)=O)c1 52048,c1(N2CC(C(C)NC(c3csnn3)=O)C2)c(F)cc([N+](=O)[O-])cc1F 52049,c1(C(=O)NC(CNC(C(N)=O)=O)CO)ncccc1Br 52050,c1(C(c2n(CCOC)nnn2)NCc2csc(N(C)CC)n2)cc(C)cc(F)c1 52051,C1(NC(=O)COC(F)(F)F)CN(C(c2cnn[nH]2)=O)C2CCCCC12 52052,c1(C(=O)NC2(CNC(C(CSC)C)=O)CCCCC2)[nH]cc2c1CCS2(=O)=O 52053,c1(CC(=O)NC2CN(C(C(C)=C3CCC3)=O)CC(C)C2)ccc(S(N)(=O)=O)cc1 52054,CC1CN(C(=O)CCc2ccccc2)CC1NC(=O)CC1CCCN1C(C)C 52055,C1(CNC(C2(CCC)CC2)=O)CN(C(c2csnc2Cl)=O)CC1C 52056,CC(CCN(C)C)C(=O)NCC1C2CN(C(=O)C(C)(C)N(C)C)CC12 52057,c1(C(=O)NCC(C)N(C(=O)C(C2CCCCC2)O)C)cscc1C(N)=O 52058,c1(C(=O)NC2(CNC(CC(CC)C)=O)CCCC2)cc2c(Cl)cccc2nc1C 52059,CC1CN(C(=O)C(C2CCOCC2)C)CC(C)N1C(c1ncncc1Cl)=O 52060,c1(C(=O)NCC2(C)CCC(NC(=O)CN3CCCC3=O)C2)cncc([N+](=O)[O-])c1 52061,C1(C(=O)NC2(CNC(C3(CN(C)C)CC3)=O)CCOCC2)Cc2nncn2C1 52062,C1(NC(c2cccc(-n3cccn3)c2)=O)CC(F)CN(C(c2n[nH]cc2Cl)=O)C1 52063,c1(C(N2CCC(CNC(C(C)Oc3ccc(C)cc3)=O)C2)=O)c(C)[nH]c(C)c1C 52064,CCC(C)(CNC(C1(NC(=O)CC2CCCCO2)CC1)=O)OC 52065,C=CCN=C(NCC(=O)Nc1cccs1)N1CCC(c2cccc(C)c2)C1 52066,c1(C(N2CCN(C(COCCC#C)=O)C(C3CC3)C2)=O)cc(Cl)cc2c1CCC2 52067,c1(C(=O)NC(CNC(C(C=C)(C)CC)=O)CO)ccc2c(c1)nc(C)c(=O)n2C 52068,C(C1CN(C(=O)C(O)Cc2ccccc2)CC1C(=O)NCC(F)C1CCC1)=CC 52069,C1(c2cn(CCF)nn2)(C(=O)OC)CCN(C(c2ncc(Br)s2)=O)C1 52070,c1(C(=O)NCC2(C(=O)NCCNS(CC)(=O)=O)CCCC2)nccnc1C 52071,C1(NC(C2=CC(C)(C)C2)=O)CCN(C(=O)COC2CCCOC2)CCC1(F)F 52072,CCC(C(=O)OCC)C(=O)N(CCC(=O)NCc1nc(C(N)=O)co1)OC 52073,C(C1CCN(C(c2nccn2C2CC2)=O)CC1)=CC(=O)NCc1c(C)cnn1C 52074,c1(C(=O)NCC2N(C(c3c(NC)nc(C)cc3)=O)CC=C2)nc(C)c(C)nc1C 52075,CN1CCN(C(C2CCSC2)=O)CC1CNC(C1CC(F)(CO)C1)=O 52076,N#CC1CCC(NC(=O)C(CCOC)NC(=O)CCOCC(F)F)CC1 52077,C1(NC(C(C)Cc2ccco2)=O)(CO)CCCN(C(c2cnc(Cl)cc2Cl)=O)C1 52078,c1(CCNC(=O)NCC2CCCCS2)ccc(Cl)cc1 52079,N1(C(c2nc(C(=O)NCc3ccc(Br)cc3)sc2)=O)CC2CCC1CO2 52080,c1(CNC(=O)CCOC2CC2)cnn2c1CN(C(C13CC(C1)C3)=O)CC2 52081,C(=O)(C(C)(C)CS(C)(=O)=O)N1CC(NC(=O)C(C)(C)N2CCCCC2)CC(C)C1 52082,N1(C(C=C(CC)C)=O)CCCC(C(=O)NC2(c3noc(C)n3)CC2)CC1 52083,CN1CCN(C(c2cc(C3CC3)no2)=O)C(C(=O)N(C)Cc2ncnn2C)C1 52084,N1(C(c2cc(C)n(C(F)F)n2)=O)CC2(CC(NC(=O)CCCC(C)O)CO2)C1 52085,Cc1cc(C(N2CCC(C(c3c(C)nn(C)c3Cl)CCNC(C)=O)CC2)=O)cnc1O 52086,C(C)(C(C)C(=O)NC(C)C)NC(C1(CC)CCC1)=O.C1(N)CN(CC)C1 52087,C(CC(C(C)(C)C)NC(c1ccc(F)o1)=O)N(C)C(c1cc(F)ccc1F)=O 52088,C1(CC(=O)NC2CCCOC2)(NC(=O)COC(F)F)CCCCC1 52089,C=CC1(C(N2CCCC(C)C2CO)=O)CCN(C(c2ccc(C)c(F)c2)=O)C1 52090,C1(CC=C)(NC(=O)CSCCCC)CCN(C(c2cc(Cl)c(Cl)[nH]2)=O)C1 52091,N1(C(c2[nH]cc(C#N)c2)=O)CCOC2CN(C(c3cccc(F)n3)=O)CC12 52092,O=C1COc2nc(C(=O)NCC3(F)CCN(C(C4C=CCCC4)=O)C3)ccc2N1 52093,c1(C(=O)NCCC2CCN(C(C3CC3F)=O)C2)csc2cccc(F)c12 52094,C1(C(=O)NCCCC(C)(C)NC(=O)CN2CC3CC3C2)CCc2nnc(O)n2C1 52095,CC(O)C(C(=O)NCC1(NC(c2csc(C3CC3)n2)=O)CCCCC1)N(C)C 52096,c1(C(N2CC3CN(C(C)=O)CC3C2)=O)cc2cc[nH]c(=O)c2s1 52097,N1(C(c2c(OC)c(C)sc2)=O)CCCN(C(=O)CC2CCN(OC)CC2)C(C)C1 52098,c1(OC(=O)NCc2nn[nH]n2)c(Cl)cc(NC2CCC23CC3)cc1Cl 52099,C(=O)(CC(F)(F)C(F)F)NCCNC(=O)C(N1CCC(F)(F)C1)C1CCCCC1 52100,C12CC(C)N1C2=O.n1(C2(CNC(COC(C)C)=O)CC2)cccn1 52101,C1(C(=O)NCCCCN2CCCC2)CN(C(C2COCOC2)=O)CC12CCC2 52102,C(N=c1cc[nH]cc1S(=O)(=O)NC1CN(CC2CC2)C1)C1CCC(C)O1 52103,c1(C(N(CCN(C(C2(CCC)CC2)=O)C)C)=O)nc(O)c(C)s1 52104,CCS(=O)(=O)CC(C)NC(c1cc(N(C)C)ccc1C)c1nnnn1CC(F)F 52105,c1(OCCC(=O)NC2CCC(NC(c3scnc3Cl)=O)CC2)ccc(F)cc1 52106,c1(C(=O)NCC(CO)NC(=O)Cn2cc(C3CC3)nn2)cc(C(F)F)ccc1F 52107,Cc1ccnc2c(C(=O)N(C)CCNC(=O)CC3CCCC4(CCC4)O3)cnn12 52108,c1(CC)ccc(C(=O)N(CCC(C)NC(=O)CCC2CCC(=O)NC2)C)cc1 52109,C1(NC(c2c(CC)nc(C)[nH]2)=O)CCN(C(C2CCN(C(N)=O)CC2)=O)CC1C 52110,c1(CC)cccc(C(N2CCOCC2CCNC(c2ncccc2F)=O)=O)c1N 52111,C1(C(N(CCC(C)NC(C=Cc2scc(C)n2)=O)C)=O)CCCCN1N=O 52112,C12(C(N3C(C)(CC(=O)NCC4(SC)CC4)CC3)=O)CCCC1OCC2 52113,C12(NC(c3ccon3)=O)CC(CNC(c3cnn[nH]3)=O)(C1)C2 52114,O=S(=O)(c1cccnc1N1CCOCC(O)C1)NCCCC1CC1 52115,C(=O)(C1=C(C)CCCC1(C)C)NCCC(CNC(c1cc(C)oc1)=O)O 52116,c1(C(=O)NCCN(C(COCC)=O)CC(C)O)sc2c(Br)csc2c1C 52117,c1(CN(C(CCN(C(C(n2ncc(C)c2)C)=O)C2CC2)=O)C)ccc(C)nc1 52118,CC1=NOC(C)(C(=O)NC2CC(n3cc(-c4ccncc4Br)nn3)C2)C1 52119,c1(SC)ncc(CN2CCC(N(C)C(=O)Nc3ccccn3)C2)c(Cl)n1 52120,C1(C(N(C(C(C)SC)C)C)=O)CC2(CCC2)CN1C(=O)C(Cl)Cl 52121,c1(C(=O)NCC(C)(C)OCCNC(C2C(C)CCOC2)=O)cnn2ccccc12 52122,Cc1cc(C(=O)NC2CC(NC(c3cc(Cl)ncc3Cl)=O)C2)cc(C)c1Br 52123,C1(C(=O)NC2(CCC)CCC2)CCN(C(=O)C2(C)CC(=O)N(C)C2)O1 52124,N1(C(C2CC(SC)C2)=O)CCCC2(C1)CN(C(c1cccc3nsnc13)=O)C2 52125,C1(c2n(C)cnn2)CCCN(C(=O)CN2C(=O)CC2=O)C1 52126,CC1(C)CCCC(CN=c2[nH]nco2)C1.C(=O)(C(C)(C)C(N)=O)N 52127,Cc1cccc(OC(C)C(N2CCC(NCC(=O)NC34CC(C3)C4)CC2)=O)c1 52128,c1(C(C)C)cccc(C(N2CC(NC(C3CC4CCC4C3)=O)C(C)C2)=O)n1 52129,n1(C(C)C)cnc2ccc(CN3CCC(C(=O)NC)CC3)cc12 52130,c1(NC(C2(C)CCN2C(c2cccc(CO)n2)=O)=O)ccc(I)c(Br)c1 52131,C1(NC(C2C(C=C)C2)=O)CCC(NC(c2nnn(COCC)c2N)=O)CC1 52132,Cc1sc(O)nc1C(=O)NC1CCCCC1N(C)C(c1cc(C(F)F)ncn1)=O 52133,C(=O)(C1=CCC(C)(C)CC1)NCCC(C)NC(=O)CCCOc1cccc(F)c1 52134,N1(C(=O)OC(C)(C)C)CCC2(CCC2)C(NC(C2(S(N)(=O)=O)CCCC2)=O)C1 52135,c1(CNC(C2CCC(CNC(C3CC34CCOC4)=O)O2)=O)cnccc1Cl 52136,Cc1ccnnc1C(N1CCCC1C(C)(C)C(=O)N(C)Cc1ncco1)=O 52137,C12(CCC1)CC=CC(=O)N2.C(C(=O)NCCOCCOC)=CC=CC 52138,N1(C(C2=CCCC2C)=O)CC(CO)C2(C1)CN(C(c1sccc1Cl)=O)C2 52139,C1(C(=O)NCC(C)CN(C)C(c2cccc(N)c2N)=O)CC2CCC(C1)C2 52140,c1(CCNC(CC2(C)CN(C(c3cnc(Cl)s3)=O)C2)=O)cccc(S(C)(=O)=O)c1 52141,CCC(CN=c1cccc(S(=O)(=O)NCCN(C2CC2)CC)[nH]1)N(C)C 52142,N1(C(c2cc(C)sn2)=O)CCC(C)(CC(N2CCC(F)CC2)=O)C1 52143,n1(CC)nc(C(=O)NC2CN(C(C3(Br)CC34CCC4)=O)C2)cc1C 52144,c1(OC)nc(C(=O)NC(C)(CNC(=O)CCc2nccs2)C2CCC2)sc1C 52145,c1(CNC(COCCC=C)=O)nnn(C)c1C(=O)NC(CO)C(O)CCC 52146,c1(C(=O)NCC(C)(C)NC(=O)Cc2sc(O)nc2O)ccc(O)c([N+](=O)[O-])c1 52147,C1(CC(N2CCC(NC(CCOC)=O)C2)=O)CCCC(C)C1 52148,N1(C(=O)C(Cl)=CCl)CCC2CN(C(=O)CNc3ccccc3Cl)CCC2C1 52149,c1(CC)ccc(C(=O)NCC(C)N(C(=O)COCc2ccccc2)C)o1 52150,N1(C(CCOCCC)=O)CCC(O)C(NC(C2(C)CNC(=O)C2)=O)C1 52151,N1(C(C2C(CC)C2)=O)CCC2(CC1)CC(NC(c1cnc(C(C)(C)C)s1)=O)CO2 52152,C12(C(N(CCCNC(=O)CC(F)(F)F)CC)=O)CCCC(CCC1)C2 52153,C1(C(=O)NCC(=O)OCC)(CC)CCCN(C(C2CC3CCCC3C2)=O)C1 52154,C(=O)(CCCCC(N)=O)NCc1ccc(NC(C)C)cc1.C12CCCCN1C2 52155,n1(Cc2n(C3C(C)OCC3)nc(-c3ccnc(Cl)c3)n2)cc(Br)ccc1=O 52156,C1(C(=O)NC2C(c3n(C)ncc3)CN(C(C3CCO3)=O)C2)CCC2CC1C2(C)C 52157,CC1(C)COC(CCC(=O)NCCC2(O)CN(C(c3cc(O)cs3)=O)C2)C1 52158,c1(CC)cccc(OCC(=O)NC2CCCC2NC(C2CC23CCC3)=O)c1 52159,C1(C(N(CCCCC2CCOCC2)C)=O)CCC(C)(C)N(C(C)(C)C)C1 52160,N1(C(C2(C3CCN(C(=O)C(C)OCC)CC3)CC2)=O)CCOCC1NC(N)=O 52161,N1(CC(=O)NC2CN(C(CCCCC#C)=O)CC2O)C(=O)NC(C)(CC)C1=O 52162,c1(OCC)ncccc1C(=O)NC1CCCCC1NC(C12CCCC1(CF)C2)=O 52163,N1(C(C)=O)CC(O)CC1C(N1CCSCC1CCNC(=O)CC(=O)N(C)C)=O 52164,C1(C(=O)NCC2(CC(C)C)CCC2)CCOCCN1C(=O)CCN1CCOCC1 52165,C1(C(N2CC(C)(c3cn(-c4ccccn4)nn3)C2)=O)CC12CCCC2 52166,N1(CN(CCCCC(C)C)C)CC(=O)N(CC(c2ccn(C)n2)(C)C)C1=O 52167,CCCC(O)C(=O)NC1CN(C(c2ncncc2Br)=O)CC1C 52168,N1(C(c2cn(CC)nn2)=O)CC2(NC(C3CC3c3ccc(F)cc3)=O)CCC1C2 52169,N1(C(CCCCCC)=O)CCC(CNC(c2cccc(C)c2F)=O)C(F)(F)C1 52170,Cc1cc(CCC(=O)NC2CCN(C(=O)CNC(=O)C(C)C)CC2F)ccc1O 52171,C(=O)(C(C)(C)C(=O)NCc1c(Br)nn(C)c1C)NC 52172,CCCCC(CN=c1[nH]cnc(Cl)c1Br)NC(=O)C1CCc2ccccc21 52173,C(=O)(C(C)(O)CC(C)C)NCC(CO)NC(c1ccc(OCCC)cc1C)=O 52174,CCCCCCC(=O)NC1CC2(C1)CC(CNC(C1NC(=O)C3CCC13)=O)C2 52175,C1(C(NOC(C)C)=O)CN(C(C2CC(C)(C)CN2C)=O)CCN1C 52176,C(=O)(CC(C)CC(F)(F)F)NCCC1N(C(c2nc(C)[nH]n2)=O)CCOC1 52177,c1(C(=O)NCC2CCN(C(C(C)CF)=O)C2)cnnc2ccccc12 52178,N1(C(C2CC(C#C)(O)C2)=O)CC2CC(NC(=O)C(C)OCC(C)C)CC1C2 52179,Cc1ccc(N)cc1C(N1CC2(NC(=O)C(CO)NC(N)=O)CC1C2)=O 52180,N1(C(C(C)OCC(C)C)=O)CCN(C(c2cccc(N)c2C(F)F)=O)CCC1C 52181,CCC(C)CC(C(=O)N1CC(N(CC(C)C)C)C1)NC(c1cccn1C)=O 52182,C(CC(C(=O)Nc1ccco1)N1CCCC1CN(C)C)SCCOCC(F)(F)F 52183,Cc1cccc2oc(C(=O)NC3CC(O)CN(C(c4ncc[nH]c4=O)=O)C3)cc12 52184,CC1(C(=O)NC2CCCN(C(=O)C3CC3)C2)CCCN(Cc2cccc(CO)c2)C1 52185,c1(C(=O)NCc2occ(C(N(C)CC3C(C)OCC3)=O)n2)cc2ccccn2c1 52186,c1(C(C(=O)NCc2nncs2)NC(CSC(C)C)=O)cnn(C)c1 52187,CN1CC2CC1CN2C(C1CC(NC(c2ncn3c2CCC3)=O)C1(C)C)=O 52188,c1(-c2cn(CCC=O)nn2)ccc2c[nH]nc2c1.c1(OC)cccc(C(F)(F)F)c1 52189,C(=O)(C(O)CC(=O)OC(C)(C)C)NCC(C)(C)NC(=O)CC1CCCO1 52190,C(c1cnccn1)=CC(=O)NC1CCC1NC(C1CCCCC1O)=O 52191,N1(C(C2CCC(C)(CC)O2)=O)CCN(C(=O)CCCn2cccn2)C2COCC12 52192,N1(C(COC(CC)(C)C)=O)CCNCCC12CCOCC2 52193,N1(C(C=CCN(C)C)=O)CCCCC(C2CN(C(=O)CCC(C)(C)C#N)C2)C1 52194,C1(NC(c2c(OC)cccn2)=O)CCN(C(=O)C(O)Cc2[nH]cnc2C)CC1F 52195,Cc1cc2nc(N3CCC(CNC(=O)C(C)(C)C(F)F)CC3C)cc(=O)n2o1 52196,c1(CC(=O)NCCC(=C)CNC(=O)CCCn2ccnc2)ccc(C(C)C)cc1 52197,C1(NC(CCOCC(C)C)=O)CCCC1C(=O)NOCC(C)(C)O 52198,N1(C(c2ncc[nH]2)=O)CCC(C2CCN(C(=O)C(O)C3CCC3)CC2)C1 52199,Cn1c(I)cc2c(N(C(=O)CC(F)(F)F)C3CCNC3)ncnc12 52200,N1(C(C(C)O)=O)CCC2C(C1)OCCN2C(c1nc(=O)n2[nH]cnc2n1)=O 52201,C=CC1CN(C(=O)CCN(C)CC)CC1NC(C1CCN(C2CCCCC2)C1)=O 52202,c1(C(=O)NCC(CNC(c2cn(CC)nc2C2CC2)=O)F)coc2ccccc12 52203,c1(C(=O)NCC2C(NC(C(CC=CC)C)=O)COC2)cc(OC)cc2ccoc12 52204,CC(C)(CC(=O)NC1CC(c2ncc[nH]2)C1)NC(C1CC2CC2C1)=O 52205,C1(CCNC(CCCc2c(C)ccs2)=O)COCCN1C(=O)Cn1cnc(=N)[nH]1 52206,N1(C(c2c(OC)scc2)=O)CCC(NC(=O)CNc2ncccn2)C(CO)C1 52207,C(=O)(C(CC)CC(F)(F)F)NCCCCC(CO)NC(C1(CCCC)CCC1)=O 52208,CC(C)(CNC(C1CCNC(=O)C1)=O)CC(=O)NCC1CCCOCC1 52209,N1(C(C2(CC)CCN(C(C3CCCN3C=O)=O)C2)=O)CCCCC(CO)C1 52210,C=C1CC2(C1)CC(C(=O)N(C(CNC(c1ncccc1F)=O)C1CC1)C)C2 52211,N1(C(C2C(C)(CC)C2)=O)CC2(CCN2C(=O)CCN(S(C)(=O)=O)C)C1 52212,C1(NC(C(CC=C)CNC(C2(O)CCC2)=O)=O)C2CCN(CC2)C1C 52213,N1(C(C(c2n(C)cnc2)O)=O)CC=C(C(=O)NCc2ccc(F)c(F)c2)CC1 52214,CN1CCC(C(=O)NC2CS(=O)(=O)C23CCN(C(=O)CO)CC3)c2ccccc21 52215,c1(CCNC(N2CC3CCC(N)C3C2)=O)cccc2c1OC(F)(F)O2 52216,C(=O)(CC1=NNC(=O)C1)NCCOCCCNC(C1C(C(C)C)CCC1)=O 52217,C1(N(C(=O)NCC(CC)NC(=O)OCC)CC)CCCN(c2ccc(C)cc2)C1 52218,C1(c2onc(C)n2)CCCCN1C(c1ncnn1C)C(=O)NC1(C)CC1 52219,c1(C(N(C2CN(C(C3N(CCC)CCC3)=O)C2)C)=O)cc(OC)cc2c1CCC2 52220,c1(C(=O)NC(C(C)C)CNC(c2coc(CO)c2)=O)cc(Cl)cn1C 52221,Cc1cccc(C(N2CCCC(C(C)Nc3nccnc3C#N)C2)=O)c1Cl 52222,C1(CCCNC(CCCOC(C)C)=O)CCN(C(=O)CC2CCOC2)CC1 52223,CCC(C)CC(C)N(C(=O)CN(C(=O)CNC(C)=O)CC1(OC)CC1)C 52224,c1(OC)ccc(C)c(CN2CCC3(CC3C(=O)NCC=Cc3ccccc3)C2)c1 52225,N1(C(CC=C)=O)CC2CC(C)N(C(=O)CCOc3ccc(Cl)cc3)C2C1 52226,c1(OC(C)C(=O)N(CC(C)NC(C2(CN(C)C(C)C)CC2)=O)C)cccnc1 52227,c1(C(=O)NC2C(NC(C3(CC)CCNC3=O)=O)CCCC2)cnc(Cl)cc1N 52228,C12(CNC(Cc3ncc(C)o3)=O)CC1CN(C(=O)C=Cc1cnc[nH]1)C2 52229,CCCCC(C)CCC(=O)NC(Cc1cnn(C)c1O)C(=O)NCCCN=[N+]=[N-] 52230,c1(OC)nc(C(=O)N(C2CCN(C(=O)C(C)(C)C(F)F)C2)CCO)ncc1F 52231,c1(SC)c(C(=O)NC2CC2NC(c2cnc(OC(C)C)nc2)=O)cnn1C 52232,C1(C)(NC(C(CNC(CN(C)CC)=O)C)=O)CN2CCC1CC2 52233,N1(C(C(=Cc2cn[nH]c2)C)=O)CC2CCN(C(C3CCCCO3)=O)C2C1 52234,C(=O)(NNC(=O)C1OCCc2ccccc21)NC(CC)C 52235,N(C1COc2c[nH]nc21)C(CCC(CC)NC(c1cccc(F)c1N)=O)=O 52236,CCC(C)C(O)CC(=O)NCC(C)(F)CNC(c1ccnc2cc[nH]c12)=O 52237,O=C1CCCC(C(N2C(C(=O)NC3CC3)CC3CC23)=O)C1 52238,C(CCO)(C(=O)N1CC(NC(C2CCN(C)C2=O)=O)C1)N(C)C 52239,C(CCC(C)C)(C(=O)NCC1CCCC1(C)C)NC(CN(CCOC)C)=O 52240,N1(C(C2(CC#C)CC=CCC2)=O)CCC2(CC1)CN(C(c1nccnc1C)=O)C2 52241,CC(CCC(=O)NCC1COC(C)(C)C1)NC(=O)C(F)C1CCC1 52242,c1(C(=O)OC2C(C(=O)OC)CCCC2)cccc(C(C)S(N)(=O)=O)c1 52243,Cc1ncc(C#N)c(N(C)CC2CN(C(c3c(C)cc(O)cc3O)=O)C2)n1 52244,C(CC(F)F)(C(=O)NCCS(=O)(=O)CC)NC(C(C)(C)OCCC)=O 52245,C1(CCNC(C2(CCNC(C(C)C3CC3)=O)CC2)=O)CSCN1C(=O)C(C)(C)C 52246,N1(C(C2(C(C)C)CC2)=O)C2CCC(C2)C1CNC(c1cc(C(N)=O)ccc1F)=O 52247,C(c1cncn1C)=CC(=O)NC1CC(CNC(CSCCC)=O)C1 52248,Cc1ccc(C(=O)N(CCNC(C2CC(C)CO2)=O)CCOCCO)nc1 52249,n1(CC(=O)NCC2N(C(COCC(=C)C)=O)CCC2C)cccc(C)c1=O 52250,CCC(CN(C)C)CC(=O)NC(C)(CSC)C(=O)N(C)CCN(C)CCO 52251,CC1C2CC(C2NC(=O)CSCc2cccc[n+]2[O-])N1C(C1CCCO1)=O 52252,C1(CC)CCN(C(C2CN(C(C3CCCCCCC3)=O)CC23CC3)=O)CCO1 52253,C1(C(N2CC(COC)(NC(C3CCCC3F)=O)C2)=O)CC(O)C(F)C1 52254,N1(C(c2cccc(OC)c2OC)=O)CCN(C(C2(S(N)(=O)=O)CC2)=O)CC(O)C1 52255,N1(C(c2ccc(C3CC3)s2)C(=O)Nc2ccc(OC)cc2)CCCC(C)(OC)C1 52256,C1(C(=O)NC2CCCC(N(C(=O)C=CBr)C)C2)CC2(CCC2=O)C1 52257,C(=O)(C#CC1CCCCO1)NC1CCCN(C(C)=O)C1C 52258,Cc1[nH]c(C#N)cc1C(=O)NC(C)(CNC(C1CC2CC2C1)=O)Cn1cccn1 52259,c1(CC)cnn(CC(=O)NC2(CC(=O)NCCC(=O)NCC(C)C)CCC2)c1 52260,Cc1ccc(CC(=O)NC(C)C(C)NC(c2ccnn2C2CCC2)=O)cc1 52261,CCC(CC)C(C)C(=O)N(CC(C)NC(c1cccc(C(=O)NC)c1)=O)C 52262,CC(C)(CCC(=O)N1CCC(=CCNC(=O)CC2CCC(=O)N2)CC1)[N+](=O)[O-] 52263,C1(CN2CCC(C(N)=O)C2)CCC2(CCC3(CC2)OCCO3)O1 52264,N1(CC(=O)NCCN(C(=O)C(F)(F)c2csc(Cl)c2)C2CC2)CC2CC2C1 52265,N=c1cc(C(N2CCC(F)(CNC(C3CC3c3ccc(Cl)s3)=O)C2)=O)cc[nH]1 52266,C1(CNC(c2c(CC)c[nH]c2)=O)CCCC(CNC(=O)CCC2CCCCO2)C1 52267,CC(CC(=O)c1cccc(F)c1)C(=O)Nc1ccnc(OCCO)c1 52268,c1(CC)nc(C(N2CCC(C(C)NC(C3(CO)CCOC3)=O)CC2)=O)c(N)s1 52269,c1(CNC(C(COC)NC(=O)CC2COCC2O)=O)cc(C)ccc1O 52270,N1(C(CC(C)C)=O)CCC2(CC1)CC2C(=O)Nc1cc(I)ncn1 52271,c1(NC)ccc(C(=O)NC2CC2CNC(c2sc(F)cc2C)=O)c(Cl)c1 52272,C1(NC(C2(NC(CN(C3CCCC3)C)=O)CC2(C)C)=O)CCn2ccnc2C1 52273,C1(F)(C(N2CCN(C(c3cc(Br)cnc3Br)=O)C3C2C3)=O)CCCCC1(F)F 52274,N1(C(CC(CC)NC(c2cccc(F)c2)=O)=O)CC(C)CCC1CC 52275,C1(NC(c2ccncc2F)=O)CCCC12CN(C(c1sccc1F)=O)C2 52276,CC1CCN(C(C2(O)CC2)=O)C1CNC(c1cnn(C2CC2)c1)=O 52277,N1(C(c2cnc(OC)s2)=O)CC2CC(C)N(C(C3(F)CCCCC3)=O)C2C1 52278,CC1(C(N2CCOC(CNC(=O)CSCc3ccncc3)C2)=O)CC(C#N)C1 52279,C(=O)(C(C)(C)S(C)(=O)=O)NCC1CC(NC(C(c2c(OC)ccc(F)c2)=O)=O)C1 52280,C1(C)(CCNC(C2(CC)CCCN2C(=O)C(=O)NCCOC)=O)NC(=O)NC1=O 52281,C(C(C)(C)CC(=O)NCC1(C)CCN(C(c2ccc(C3CC3)c(F)c2)=O)C1)OC 52282,c1(N2CCC(NCc3cn(C(C)(C)C)nc3)CC2)ncccc1C#N 52283,CC(C)CC(CNC(C1(P(C)(C)=O)CC1)=O)NC(C1CCCC(CF)C1)=O 52284,N1(C(c2cc(C)ns2)=O)CC2CC(C1)CN(C(c1ccc(C(O)CF)cc1)=O)C2 52285,c1(C(=O)NC2C=CC(CNC(c3cnns3)=O)C2)ccc(OCCO)cc1 52286,O=C(C(=O)N=c1nc[nH]n1-c1ccccn1)N1CCC(C(O)CO)CC1 52287,n1(CC(=O)Nc2cccc(Cc3nc[nH]n3)c2)cc(C(F)(F)F)c2ccccc12 52288,c1(C(C(C)NC(C2CCCNC2C)=O)=O)ccccc1O 52289,C1(C(=O)NC(C(=O)NC(c2nn[nH]n2)C)=O)C(C(=O)C2CC2)C1(C)C 52290,c1(C(=O)NC(CNC(C(CCCC#C)C)=O)C)cc(C)c2occc2c1 52291,CC1CC(C)N(C(c2nccc(N)c2Cl)=O)CCN1C(c1cnns1)=O 52292,n1(C(C)C)nnc2c(NCCC3(NC(=O)C(C)OCCN(C)C)CC3)ncnc12 52293,N1(C(C2ON=C(C)C2)=O)CC(NC(=O)C(C)N2CCC2)C(CO)C1 52294,C12(C(=O)NC(C(C)NC(=O)C=CC3CCCCC3)C)CC3CC(CC(C3)O1)C2 52295,O=C(C#CC1CCC1)NC1CC(C(=O)NCC(O)C2(Cl)CC2)C12CCC2 52296,C1(CNC(Cc2c(C)nc[nH]2)=O)CCCCCN1C(c1cnn(CC2CC2)c1)=O 52297,c1(CN2C3CN(C(C(n4[nH]cnc4=N)C)=O)C(C3)C2)cc(F)c(F)c(Cl)c1F 52298,N1(C(c2cc(OC)ncn2)=O)CC2(CCN(C(c3ccc(Cl)nc3Cl)=O)C2)C1 52299,C1(C(N2CCCN(C(C3CC3c3ccccc3)=O)CC2)=O)CCCC1C1CC1 52300,C1(CNCC2CCCC2C(N(C)CC2(CC(C)(C)C)CC2)=O)CC(F)(F)C1 52301,c1(CNS(=O)(=O)CCc2cc(Br)cc(Br)c2)cc(F)c(Cl)cc1Cl 52302,CC(C)C(C(=O)NCCCS(N)(=O)=O)NC(=O)Cn1cnnn1 52303,c1(C(N2C(CNC(c3coc(Cl)c3)=O)CC(F)(F)C2)=O)cn2c(n1)CCCC2 52304,C1(NC(C(N(C)O)=O)C2CC2)CCS(=O)(=O)CC1 52305,c1(OC)cc(C2CC2)ccc1C(=O)NC1CN(C(C23CC(F)(C2)C3)=O)CC12CC2 52306,N1(C(C2(C)CCC2)=O)CC2(CCC2CNC(=O)C(C)(C)C2CCCC2)C1 52307,CC(CO)C(=O)NCC(C)(F)CNC(c1n[nH]cc1C1CC1)=O 52308,C1(NC(c2c(C)nc(O)s2)=O)(CO)CCCN(C(=O)CC(C)C(C)C)C1 52309,c1(C(N(C2CCN(C(=O)CC(=O)NC3CC3)C2)CCC)=O)cnc(Cl)c(Cl)c1 52310,C(C(O)C(=O)NCC(C)(C)CNC(=O)C(C)OC1COC1)=CCCC 52311,c1(OC)ncc(-c2cnn(CCN(C)C)c2)cc1C(N1CCC(OC)CC1)=O 52312,CCC(C)(C)CCCC(=O)NCCN(C(c1cc(O)n(C)n1)=O)C(C)C 52313,N1(C(c2cn(CC3CC3)nn2)=O)CCCC(C2CCN(C(c3ccoc3)=O)C2)C1 52314,C(=O)(C1=CC2(CN(C(c3cc(C)sn3)=O)C2)OC1)NCC1(OC)CCOC1 52315,n1(CC)cnc2nc(=NCCCc3nc(C)cs3)[nH]c(NC3CN(C(C)=O)C3)c12 52316,c1(NCC(N2CCN(C(=O)CC3C=CS(=O)(=O)C3)CC2)=O)cccc(F)c1 52317,c1(C(N2C(CNC(CC(C)SC)=O)CCC(C)(C)C2)=O)cnc2sc(C)c(C)n12 52318,C(=O)(C(C)(C)CCC#N)NCCC1CCN(C(c2c(C)nc(Cl)cc2)=O)C1 52319,c1(C(=O)NC2CC(C)CN(C(C3CC4(C3)CC4F)=O)C2)cccc2cccnc12 52320,c1(C(=O)NC2C(NC(c3c(CC)n[nH]c3)=O)COCC2)n[nH]c2c1CCC2 52321,S(=O)(=O)(c1ccc(N2CCN(C(C3CCCO3)=O)CC2)nc1)N(CCCCC)C 52322,c1(C(N2CC(CNC(=O)Cn3ncnn3)OCC2)=O)cc2cc(F)ccc2cn1 52323,C=CC1CN(C(c2c(C)nn(C)c2C)C(=O)NC2CCC2)CC1O 52324,C#CCCC(O)C(=O)NC1(CO)CCCN(C(c2c[nH]nc2CC)=O)C1 52325,C1(CC)CN(C(C2CC(C)(C)O2)=O)CCN1C(C1CN(C(N)=O)C1)=O 52326,c1(C(N2CC(NC(Cc3c(C)non3)=O)C(C)C2)=O)cnc2sccc2c1 52327,N1(C(c2c(C)nn(C)c2C)=O)CCN(C(c2cccc3c2CCC3)=O)CC(O)C1 52328,C1(NC(c2c(C)cns2)=O)CN(C(C2CC(F)C(=O)N2)=O)CC2(CCC2)C1 52329,C(=O)(CCCC(=O)N1CC=CC(NC(=O)C(CC)NC(N)=O)C1)OCC 52330,c1(OC)ccnc(NCC(=O)NC2CC2CNC(c2cc(Cl)cs2)=O)n1 52331,N1(N(C)C)CCN(C(c2ccnc(NCc3nc(C(C)OC)sc3)c2)=O)CC1 52332,C1(C)(C(=O)NCC(C2(O)CCN(C(C(C)NC(C)=O)=O)C2)(C)C)CCCN(C)C1 52333,N1(C(CC(CN(C)C)O)=O)CC=C(CC(=O)N2CCCC(N(C)C)CC2)CC1 52334,N1(C(c2ccc(NC)cc2)=O)CC2CCCC2C1C(=O)NCc1ccco1 52335,c1(N(C(C)=O)C)ccc(NC(C2CCCN(Cc3ccncc3)C2)=O)cc1 52336,c1(C(=O)NCCCOCCC(=O)N(C(C)CCO)C)cnn(C)c1 52337,C1(C(=O)NCc2c(C(=O)NC(Cn3ncc(C)c3)C)scc2)CC2CCCC2C1 52338,CCC(C)C(O)C(C)C(=O)N1CCOC(CN(C(=O)CCC(C)C)C)C1 52339,C(=O)(C1Cc2c(Cl)cccc21)N1CC(CCNC(c2cc(F)c(F)cc2O)=O)C1 52340,c1(OC)ccc(C(=O)N(CCC(C)NC(c2ccc(F)s2)=O)C)cc1OC1CC1 52341,N1(C(c2cc(CNC(COCCC#C)=O)sc2)=O)CCCC2(C)CCCC12 52342,c1(C(=O)NC2CCCC(N(C(CCC#C)=O)C)C2)c(Cl)ccc([N+](=O)[O-])c1Cl 52343,c1(C(=O)NCC2N(C(C(C(C)C)O)=O)CCCC2C)ccn2ccnc2n1 52344,Cc1ccc(C(N2CCCC2CN(C(=O)CNC(c2cccs2)=O)C)=O)nn1 52345,C(=O)(CCCCCC(C)(C)C)NCC1CC(NC(C(C(C)O)C)=O)C1 52346,C1(C(=O)NCc2c(OCC(=C)C)cccc2)CC(F)CN(C(=O)CCSC)C1 52347,C1(C(N2CCC(CC)C2)=O)COCCN(C(C2CC(N=[N+]=[N-])C2)=O)C1 52348,CC1(C)CN(C(c2csnn2)=O)CC(C)(C)C1NC(c1csc(C(F)F)c1)=O 52349,C#CC1CCCC(NC(C2CCOC2CNC(=O)Cc2c(C)cnn2C)=O)C1 52350,C(=O)(CC1=CCOCC1)NCC(C1CC1)NC(=O)CC(F)F 52351,N1(C(C(CC2CCCC(O)C2)NC2CC(CC)(CC)C2)=O)CCC(O)(COC)CC1 52352,N1(C(C2(C)CCNC2=O)=O)CCC(NC(=O)CC(O)c2ccccc2)C(F)C1 52353,C=CCC(C)(C)CC(=O)NCc1cc[nH]c1C(=O)NCC1CC2CC1CC2O 52354,c1(OC)ccc(C(=O)NCC2CC2NC(c2ccnc(C)c2)=O)c(Br)n1 52355,C1(C)(C(N2CC(C)C(CC(=O)O)CC2)=O)CC2(C1)CC(F)(F)C2 52356,C(=O)(C(C)=Cn1ccnn1)NC(c1ccc(CNC(CC(=O)OCC)=O)cc1)C 52357,C(=O)(C1CCCc2ncc(C)n21)N1CCN(C(C(CCCC=C)(C)C)=O)CC1C 52358,C1(CCNC(CNC(C)=O)=O)CCN(C(c2c[nH]c(=N)nc2C)=O)CCC1(F)F 52359,C(=O)(CC(O)CC(C)(C)C)N(C)Cc1c(F)cc(C#N)cc1Cl 52360,N1(C(C(CC)C)=O)CCC2(CCCC2CNC(=O)CCOC2CCCC2)CC1 52361,C1(C(=O)NCC(O)Cc2ccccc2)C2CCC(C2)N1C(c1cccc(F)n1)=O 52362,C(=O)(CCC(O)C(C)(C)C)N1CC(CNC(c2nc(CC)oc2)=O)C(C)CC1 52363,C(=O)(C(O)CCc1ccccc1)NC1C(CNC(=O)Cc2cc[nH]c2)COC1 52364,n1(C(C)C(=O)O)cc(C2(O)CN(C(C3(c4ccccn4)CCC3)=O)C2)nn1 52365,CC1(C)CC(NC(=O)CCc2ccc(F)cc2Cl)CN(C(=O)Cc2nc[nH]n2)C1 52366,c1(C(N2CCC(NC(c3c(C)[nH][nH]c3=N)=O)C2)=O)ccc(C)c2ccccc12 52367,Cc1nc(NCC(C)(C2CC2)NC(c2ccsc2C)=O)c(C)c(O)n1 52368,N1(C(=O)NC)CC(C(=O)NCC#CCNC(=O)CC2CCCO2)C1 52369,n1(CC)ncc(C(=O)NCc2ocnc2C(=O)NC2(C)CCOC2C)c1C 52370,N1(C(CC(C)F)=O)CCN(CC(C)(C)NC(c2cc(CCO)on2)=O)CC1 52371,CCC(C)(C)C(O)C(=O)N1CC(C(=O)NCc2ccncc2C)C(C)(C)C1 52372,c1(C(=O)NC(CN(C(c2n[nH]cc2Br)=O)CC)C)ccc(C)cc1 52373,C1(NC(C=CSC)=O)C(C)CCN(C(c2cnc(C3CC3)o2)=O)C1C 52374,CC1CCCCC1(C)C(=O)NC1CCCN(C(c2csc(O)n2)=O)CC1 52375,N1(C(c2c(C)ccc(C)c2)=O)CCCCC2(CCN(CC3CCOC3)C2)C1 52376,N1(C(C(CC(=O)OC)N(C)C)=O)CC2CCC1CN2C(c1coc(N(C)C)n1)=O 52377,N1(C(c2c(CC)ncs2)=O)CCCN(C(c2ccc(O)c(O)c2)=O)CC1C 52378,C1(CNC(c2c[nH]cc2Br)=O)CC2(CCC2)CN1C(=O)C=Cc1ccc(O)cc1 52379,N1(C(C=CC=CC)=O)CCCCC2(C1)CN(C(c1ccc(OCOC)cc1)=O)C2 52380,c1(C(=O)NCc2c(C(N3CC(C#CC)C3)=O)nn(C)c2)cc2ccccn2c1 52381,C1(C)(CNC(c2ccc(C)o2)=O)CCCN(C(C2CC3(CC3)CN2C)=O)C1 52382,C1(C(N2CCC(NC(c3c(C)[nH][nH]c3=N)=O)C2C)=O)CCC2(CCC2)O1 52383,C(=O)(C(O)C(C)(C)C)NCCC1(O)CCN(C(c2cc(C)c(Cl)s2)=O)C1 52384,c1(C(=O)NCCc2nc3scc(C)n3c2)ccc2cc(I)ccc2n1 52385,Cc1cc(C(=O)NC(C(=O)NC(c2nc[nH]n2)C2CC2)C2(C)CC2)ncc1N 52386,N1(C(C2(C)CCCN2C(c2cnn3ccncc23)=O)=O)CCn2cccc2C1 52387,CCCCC(CC(=O)NCC(F)(F)C(C)C)NC(c1cc(C)ncn1)=O 52388,C=CCCCCCCCCc1nc(CCCCC)nn1C1CCC1 52389,CCCC(C(=O)NCC(F)CNC(c1ccccc1Cl)=O)NC(N)=O 52390,Cc1ncnc(C)c1CC(=O)NC1CC2CN(C(=O)C(C)n3ccnc3)CC12 52391,C=CC(CC)CC(=O)N1CCN(C(=O)C2=CCSC2)C(CCO)C1 52392,CC1(C)NC(=O)CCC1NC(=O)COc1cccc(Cl)c1 52393,CCCC(CC)CCC(=O)NCc1cc(C(=O)NC2(c3noc(C)n3)CC2)cs1 52394,CC1CN(C)CCN1C(C1CC2(CC2)CN1C(=O)Cc1nccn1C)=O 52395,n1(CC(=O)NC(C)C(C)NC(=O)Cc2cccc(F)c2)nnc2c1CCCC2 52396,O=C(C1=CCS(=O)(=O)C1)NCC1CCN1C(C1CC(Cc2ccccc2)C1)=O 52397,C12(C(N(CCCNC(C(C(C)(C)C)SC)=O)C)=O)CCC(C)(C(=O)O1)C2(C)C 52398,C(C1CCc2nccn21)NC(C1=NOC(CNC(C(CC)OC)=O)C1)=O 52399,c1(SC)ccccc1C(=O)NC1CN(C(=O)COc2ccsc2Cl)CC1F 52400,C1(C(=O)CNC(C(C)OC2CCCC2)=O)CCC(ON)CC1.CCOCCOC 52401,C1(CN(C(CC2C(C)OCC2)=O)CC(O)C2CC2)CC(CCC(C)(C)C)C1(C)C 52402,Cn1ncc2cccc(-c3nc(C(F)F)nn3CCN3CCCCC3)c12 52403,N1(C(CC(C)(C)C#N)=O)C(CNC(C2CC2(C)C)=O)CC2CCCCC12 52404,N1(CC(=O)NCC(CN(C(=O)C(C)C2CCCC2)CC)(C)C)CC(=O)N(C)C1=O 52405,c1(CNC2CC(CC(=O)Nc3cnc4cnccn34)C2)c[nH]c2nccc(Cl)c12 52406,C1(CNC(c2nccc(CC)c2)=O)CCCN(C(C2CC(F)C(=O)N2)=O)CC1 52407,c1(CC(N2CCCC(NC(C(CC)(C)C)=O)C2)=O)ccc2c(c1)CCCC2 52408,CCCCC(O)C(=O)NC(C1CCCC1)CNC(c1ncc(F)cn1)=O 52409,Cc1cnc2cc(C(=O)NCC34CC(NC(C5(C)CCCCO5)=O)(C3)C4)nn2c1 52410,CCC(CC1CCCCC1)C(=O)NC1CCOC(CNC(C2(CO)COC2)=O)C1 52411,N1(C(CCC2CCC(C)N2)=O)CCC2(CCN2C(=O)OC(C)(C)C)C1 52412,C(CCCC(=O)NCC(C)N(C(=O)Cn1nnc(-c2cccs2)n1)C)OCC 52413,N1(C(=O)NCC(C2CCCC2)(C)C)CCC(Cn2cncn2)C1 52414,c1(C(N(CCOC)CCNC(=O)CCSCC(C)C)=O)ccc(S(C)(=O)=O)cc1N 52415,N1(C(CN(CCC)C(c2ccc(C#N)cc2)=O)=O)CCS(=O)C(C)C1 52416,c1(OC)ccc(C(=O)Nc2nc(C(C)(C)C)co2)cc1.C12(CNC1)CO2 52417,C1(NC(Cc2ccc(C(=O)NC)cc2)=O)CCN(C(=O)CCNC(C)=O)C(C)C1 52418,c1(NCC(C)CN2CCCCC2)nccc(=NC2CCc3cccnc32)[nH]1 52419,C1(CC(=O)N(C2C(C)CC2)C)CN(C(=O)C(C2CCOCC2)O)CCO1 52420,N1(C(C(CC)(C)C(N)=O)=O)CCCC(C2(NC(=O)CCN3CCCC3=O)CC2)C1 52421,c1(C(C)C)ccc(C#N)c(NCC2CCCN2C(C2CCCC3CCCN23)=O)n1 52422,c1(C(N2CC(CCNC(C3C(OCC)C3)=O)OCC2)=O)cnc2c(n1)CCCC2 52423,c1(C(=O)NCC2(CNC(Cn3ccc(C)n3)=O)CC2)c(C)cc(Cl)cc1C 52424,Cc1ccccc1CCC(=O)NCCCCCNC(C1CCC(F)C1)=O 52425,c1(C(=O)NCCC(Cc2ccccc2)NC(=O)CC2CC=CC2)cccc[n+]1[O-] 52426,N1(C(c2nc(CC)sc2)=O)CC(NC(=O)C(C)CCOC)C(C)(C)C1 52427,c1(CC)ccc(C(=O)NCC(C2CCC2)NC(=O)CC(=O)OC)cc1[N+](=O)[O-] 52428,c1(C(=O)NC2CC(C)(CC)N(C(C3(OC(C)=O)CC3)=O)C2)c(C)nc2sccn12 52429,c1(C(=O)NC(CN(C(C2C(OCC)C2)=O)C)(C)C)cnc(Cl)s1 52430,c1(C(N2CC(NC(=O)Cn3ccnc3)C(O)C2)=O)ccc(Cl)c2ccccc12 52431,C(=O)(CCCC(C)NC(=O)CC(C)COC)N1CC(CC)SCC1 52432,C(=O)(C(O)CCCNC(=O)CCCC1CC1C)N(CCC(=O)NC)CC 52433,C(=O)(C(O)CC(C)C)N(C(C)C(=O)NCc1nn(C)cc1CO)CC 52434,CC1(C)CCCN(C(=O)C=Cc2cnc(O)nc2O)C1CNC(C1OCCO1)=O 52435,c1(N(CC(CC)CCCC)CCCC)cc(OC)c(OC)c(Cl)c1 52436,n1(CC)nc(C)cc1C(=O)NC(C(=O)NCC1(CC)CCC1)C1(C)CC1 52437,c1(C(N2CC3C(NC(C4CN(C)C(=O)C4)=O)C3C2)=O)cc2c([nH]1)CCCC2 52438,C12(C(=O)NCC3(NC(CNC(N)=O)=O)CCCCCC3)CCCCC1C2(F)F 52439,c1(CN2CCC(NC(=O)NCCCCC#C)CC2)c(Cl)cccc1Cl 52440,CN1CC(C)(C(N2CC(N(C(=O)CSc3nncn3C)C)C2)=O)CCC1=O 52441,C1(NC(CCC2CC(OC)C2)=O)CC2CCC1(C(N1CC(C3CCCO3)C1)=O)C2 52442,C1(CC(N2CC(CNC(c3c(C)n[nH]c3)=O)C(F)(F)C2)=O)NC(=O)CN(C)C1=O 52443,N1(C(CCCOCC=C)C(=O)NCCC)CCC(F)(F)C2(CCOC2)C1 52444,C1(CC)CN(C(=O)CC(F)(F)CC)CCN1C(=O)COc1cc(F)ccc1F 52445,C1(CC)CC(O)CCN1C(C1CCOC1CNC(c1cnnn1C)=O)=O 52446,CCC(CC)C(=O)NCc1csc(C(=O)NC(C)CS(C)=O)c1 52447,c1(C2C(NC(C(C)N(C(=O)CN3CCOC3=O)CC)=O)C2)ccccn1 52448,C1(NC(C=C(C)C)=O)CCC(C)N(C(C2C3COCC23)=O)C1 52449,C=C(C)C1OCCC1C(=O)NCCC1CC(NC(=O)CCSC(F)(F)F)C1 52450,C1(C(CNC(C2C(CC)C2)=O)(C)O)CCN(C(C2(C(N)=O)CC2)=O)CC1 52451,Cc1ccn2c(C(N3CCOC(CCNC(c4ccccn4)=O)C3)=O)cnc2c1 52452,C1(C(=O)NCC2(F)CCCN(C(CCCNC(C)=O)=O)C2)CC2CCC1C21CC1 52453,C1(CNC(C2CCS2(=O)=O)=O)CCN(C(c2csc(C(F)F)c2)=O)C1 52454,c1(C(N2CCC3(C(C(=O)OC)C3)C2)=O)cc(N)c(Br)cc1C 52455,C(=O)(C1=NOC(C)(C)C1)N(C1CCCC(NC(c2c(CC)[nH]cc2)=O)C1)C 52456,c1(CNC(c2c(C)c[nH]n2)=O)cccc(C(=O)NC(C)CN2CCCC2=O)n1 52457,C#Cc1cccc(CC(=O)NCC2(NC(c3[nH]c(C)nc3C)=O)CCOCC2)c1 52458,c1(C(=O)NCC(CC)NC(=O)C(F)(F)c2csc(Cl)c2)n[nH]c2c1CC(C)CC2 52459,S(=O)(=O)(c1cccc(C(C)=O)c1)N(C(C)CCNC(=O)C(=O)N(C)C)CC 52460,C#CCCCC(C)C(=O)NC1CC(C(=O)NCCCN2CCCC2)C1 52461,Cc1cc(C(N2CC(O)(CCNC(C34CCCCC3C4)=O)C2)=O)cc2nn[nH]c12 52462,C1(NC(=O)C(=O)NC2COC3CC2C3)CCC2(CCOCC2)C1 52463,c1(SC)nc(NC2(CNC(=O)C(C(C)C)N3CCCCC3C)CCC2)cc(O)n1 52464,C(=O)(C(C1CCCC1)SC)N(C(C)CNC(=O)CNC(C)=O)CC 52465,N1(CC(=O)NC(C(C)C)CNC(c2cc(Cl)n[nH]2)=O)CCC(=O)NC1=O 52466,C1(N(C(C2C(=C)C2)=O)CCO)CCCN(C(c2ccn(C(CC)CC)n2)=O)C1 52467,C1(OC)(CNC(C2(CF)CC2(F)F)=O)CCN(C(=O)CCn2nc(C)cc2C)C1 52468,C(=O)(CCCCCOC)N(C(C)C(=O)N(C)CC1CCCCC1)CC 52469,CC1CC(NC(=O)C(C)(F)F)CCN1C(C1(c2ncccn2)CCC1)=O 52470,c1(C(N2CCC(O)(C(=O)NC(C=C)C)C2)=O)ccc2nc(Cl)sc2c1 52471,c1(CN2CC(CNC(C(CC)C)=O)OCC2)nc2ccccc2[nH]1 52472,N1(C(C#CC(C)C)=O)CCCC(C2CC2NC(=O)CC2CCCCCC2)C1 52473,c1(C(N2C(CN(C(=O)C=CC3CC3)C)CCC2)=O)c(O)nc(=O)n2c1CCC2 52474,n1(CC(=O)OC)cnc(C)c1C(=O)NC1CC(C)(NC(c2cccnc2C)=O)C1 52475,c1(C(c2n(C(CC)C)nnn2)NCCCn2ccnn2)c(Cl)ncn1C 52476,O=S(=O)(c1[nH]cc2c1CCS2(=O)=O)Nc1ccncc1C(F)(F)F 52477,Cc1ccnc(N(C)CC2CCCN2C(=O)C(C)Oc2ccccc2)c1[N+](=O)[O-] 52478,C12(NC(C(C3CCCCCC3)C)=O)CCC(CC1)N(C(C1CCCCC1(C)C)=O)C2 52479,c1(N(CCCC(=O)OC)CC2CCCO2)ncc(-c2cccs2)cn1 52480,C1(F)(CNC(C2ON=C(C)C2)=O)CC2CCC(C1)N2C(=O)CN(CC(C)(C)C)C 52481,C(=O)(C(CCOC)NC(=O)CCc1nc(C)no1)NCCC=CC=C 52482,N1(C(C2CN(Cc3ccncc3O)CCS2)=O)CCN2CC(O)CC2C1 52483,CC1CC(C(=O)NC23CC(C(N4CCCC4)=O)(C2)C3)N(c2ccncc2)C1 52484,N1(C(C2=CCN(C(c3cnc(C)[nH]c3=N)=O)CC2)=O)CCC2CCC(O)C1C2 52485,c1(C(N(CCOCCCNC(C(C)OCCC=C)=O)C)=O)cc(Cl)c(Cl)[nH]1 52486,C(=O)(C(O)CC(F)(F)F)N1C2C(CNC(CCN(C)CC)=O)C(C2)C1 52487,C(=O)CCCCCCS(N)(=O)=O.N1(C(CC#N)=O)CCC2(CCC(=O)NC2)CC1 52488,c1(N2CC3(C(NC(C4CC5C=CC4C5)=O)CCC3)C2)c(Cl)cc([N+](=O)[O-])cc1Cl 52489,Cc1cc(C(=O)NC(C)CNC(=O)C(C)(C)OC(C)C)nc(O)c1 52490,C#CC1(C(=O)NCc2cc(C)c(C(=O)NC(C)C(C)CO)o2)CCCC1 52491,C1(C(N2CC(CO)C(O)C2)=O)(COC)C=CCN1C(c1csc(O)n1)=O 52492,C=CCCC(C(=O)N1CCC(C(F)F)CC1)NC(c1ccc(C)cc1)=O 52493,CN1CC=C(c2ccc(CNC(=O)NCC3CC3c3ccccc3)cn2)CC1 52494,C1(CNC(C2(CC)CCCO2)=O)CC(OC)CN1C(=O)CC1(CN2CCCC2)CC1 52495,c1(C(=O)NCC(O)CO)cncc(NCc2ccncc2)c1 52496,c1(CC(=O)NCC2C=CC(NC(=O)C(F)=C3CCCC3)C2)cccc(C(F)(F)F)n1 52497,C1(C(=O)NCC(C)NC(=O)C(C2CC(F)(F)C2)O)CCCN(C)C1 52498,CN1C(=O)COCC1CNC(=O)CC1CC(NC(c2csnc2Cl)=O)C1 52499,N1(C(CCC=CC(C)C)=O)CCC(C2CCN(C(c3c[nH]nc3C3CC3)=O)C2)C1 52500,C(=O)(C(F)(F)CN1CCCC1)NCCCN(C)C(C1(F)CCCCC1)=O 52501,c1(C(N2CC(NC(c3ccc(C#C)cn3)=O)C(C)C2)=O)ccc2cn(C)nc2c1 52502,N1(C(c2n(CC#C)ccc2)=O)CCCN(C(c2cccnc2)=O)C(C)C1 52503,Cc1c(C(=O)NC(C2CCN(C(c3ccc(=O)oc3)=O)C2)(C)C)c[nH]c1C(C)C 52504,C1(CC(=O)NCC2CCCCS2)CCN(C(c2nc(Cl)cs2)=O)CC1 52505,C1(OC)(OC)CC(CNC(C2CCN(C(=O)CCC3CCCOC3)C2)=O)C1 52506,c1(C(=O)NCC(C)CNC(=O)CC(c2ccc(Cl)cc2)O)ccc2c(c1)OCC2 52507,C(=O)(C(CCF)NC(=O)CCCNC(=O)C1CC1)NC(C)CCCO 52508,C(CS(=O)(=O)CCCCNC1CC(C(O)C(F)(F)F)C1)N(C)C 52509,N1(C(C2CC(CC)C2)=O)CC2(C(=O)NCC3CC(C(C)(C)C)C3)CC1CCO2 52510,C(=O)(C1=CCCCCC1)NCC(CC=C)NC(C1CC(Cl)(Cl)C1)=O 52511,C1(O)(CNC(c2cc(C)c(F)cc2)=O)CCCN(C(C2C=CCS2)=O)CC1 52512,C1(NC(C=CCCC)=O)CC2(CNC(=O)CC(C)c3cccnc3)CC1CO2 52513,n1(CC)cnc(C(=O)NC2CC(C(=O)NCCCCO)C2)n1 52514,N1(C(c2c(C)ocn2)=O)CCN(C(C2(C3CCC3)CC2(F)F)=O)C2COCC12 52515,c1(C(C)Nc2ccnc(O)n2)c[nH][nH]c1=NC(=O)c1ncccc1C(F)(F)F 52516,N1(C(C2CCN(C(C)=O)CC2)=O)CCC2(CCCN2C(=O)Cn2cc(C)cn2)C1 52517,Cc1cccc2[nH]cc(CC(N3CCC(C(C)O)C3)=O)c12.C1(=O)COCCN1 52518,c1(C(N2C(CNC(C3CCN(C)CC3)=O)COCC2)=O)cnc2c(n1)CCCC2 52519,N1(C(Cc2c(C)n[nH]c2)=O)CC(NC(=O)C(C)(C)C#N)C(c2ccc(F)cc2)C1 52520,CCCCC(=O)C(=O)NC(CN(C)C)C(=O)N(CC)Cc1ccoc1 52521,C1(n2c(NC(=O)C(C)CCC)ccc2)CCCN(SC)C1.N12CCC(C)(C1)NC2=O 52522,N1(C(c2cc(F)c(N)c(F)c2)=O)C2CCCC1CN(C(C1(S(N)(=O)=O)CC1)=O)C2 52523,C1(C(=O)NCC2(O)CCC2)CC(F)CN(Cc2ncc(Cl)cc2F)C1 52524,CCC1(CNC(C)(CCBr)c2nnnn2CC2CC2)OCCc2ccccc21 52525,N1(C(C(C2CC(F)(F)C2)OC)=O)CC(C)(C)CC1CNC(C1CC(SC)C1)=O 52526,c1(N2CCC(n3cc(CCCC(C)=O)nn3)C2)n[nH]c2c1CC(C)CC2 52527,CCC(O)C(C)C(=O)N1CCCC(CCNC(c2cc(C3CC3)n(C)n2)=O)C1 52528,c1(C(N2CCCCC(CNC(C3C(CC(C)C)C3)=O)C2)=O)cnn2c(=N)[nH]cnc12 52529,N1(C(C(CC)C(C)C)=O)CC2(C1)SCCC2NC(c1cccn2cncc12)=O 52530,C1(C(=O)NCC(c2ccccc2)C)CC(O)CN1C(=O)CC1CC(=O)NC1=O 52531,C#Cc1cc(C(=O)NCCC(O)C(=O)NC(C)CC(=O)NC(C)C)ccc1C 52532,C1(C2CCCCO2)(C(=O)NCC(C)N(C)C(c2ccc(C3CC3)o2)=O)CCCO1 52533,n1(CC(=O)NCC2(CNC(CCSC)=O)CCC2)cc2ccccc2n1 52534,N1(C(c2c(C)cc(F)s2)=O)CCC(C2(NC(=O)C(O)C3CC3)CC2)CC1 52535,C1(C(N2CCCC(N(C(CCN3CCN(C)CC3)=O)C)C2)=O)CC(C2CC2)=NO1 52536,CC1CN(Cc2ccccc2)C(C)CN1C(=O)CC1CCCNC1 52537,C1(NC(C2(CO)CCCO2)=O)CN(c2ncnc3scnc23)CCC12CCC2 52538,c1(CNC(CCCOCCOCC)=O)ccc(C(=O)N)nc1.n12cc(nn1)C2.OC 52539,c1(C(=O)NC2CCN(C(CSCCOC)=O)C23CC3)nc(C)c(C)nc1C 52540,N1(C(=O)C=CC2CCCC2)CCC2OCCN(C(C3CCCS3(=O)=O)=O)C2C1 52541,c1(C(N2CC(O)CC(NC(C3CC(CC)C3)=O)C2)=O)n[nH]c2c(C)cccc12 52542,C12CCN(C1(C)C)C2=O.C1(C(N(CC(N2CCCC2)=O)C)=O)CC(=O)NC(=O)N1 52543,c1(CCC(=O)NC(C(C)NC(C(F)=CC)=O)C)nc(C)cs1 52544,CCC(C)C(C(=O)NC1C2CC3C1C3C2C(=O)NCCCO)OC 52545,C1(CN(C(COCC=C)=O)C)C2CN(C(=O)CCCc3nc(C)no3)CC12 52546,c1(NC(=O)Cc2cc(=O)n(-c3ccccn3)[nH]2)ccc(F)cc1C(N1CCCC1)=O 52547,N1(CC)CCC(C(=O)NC23CC(C(=O)NCC(O)C(F)F)(C2)C3)C1 52548,CCC(C)C(C)C(=O)NC1CN(C(=O)C=C(C)Cl)C1 52549,C(=O)(C(CCCC(=O)OC)N1CC2CCCC(C2)C1)NCC(=C)C 52550,N1(C(CCc2ccc(C)cc2C)=O)CC(CNC(C2(C)CC2C)=O)CC(C)(C)C1 52551,N1(C(C2C(C)CC=CC2)=O)CCOCCC1C(=O)N(C1CCC(F)(F)C1)C 52552,N1(C(C(C)N(C(c2cnnn2C)=O)CC)=O)CCN2C(=O)NCC2C1 52553,N1(CC)C(=O)CCC1CC(=O)NC(C)(C)CCN(C(=O)C(F)OC)C 52554,CC(=O)C(C)(C)CC(=O)N1CC2(CC(C(=O)NCC3(C)CC(C)=NO3)CO2)C1 52555,N1(c2cc(C)nc(N3CCc4cc(Cl)sc4C3)n2)CCC2(CCCCC2)CC1 52556,C1(NC(=O)C(N2CCSC3CCC23)=O)(Cn2cnnc2)CC2(CCC2)C1 52557,CC1(CC(=O)NC(CO)C(F)(F)F)CCN(C(c2nccnc2N)=O)C1 52558,CCC(C)CC(C(=O)NCC(C)(C)C(F)(F)F)NC(=O)CN(C)CC 52559,C1(C(=O)NCCC2(OC)CN(C(c3ccnnc3O)=O)C2)CCC(C)NC1=O 52560,C1(=CCNC(C(C)(O)C2CCOCC2)=O)CCN(C(=O)C(F)OC(F)(F)F)CC1 52561,C1(OC)CC2CC(C1)N(C(=O)CC1CCCCC1NC(c1cc(C#N)oc1C)=O)C2 52562,CCC(F)(F)CC(=O)NC(CC1CC1)CC(=O)Nc1cnn(C(C)(C)C)c1 52563,C1(NC(C2N(C(CC3CN(C(C)=O)C3)=O)CC3CC32)=O)CN(C)C2(CCC2)C1 52564,c1(CC(=O)NCC(=C)CCNC(c2cc[nH]n2)=O)nc(C2CC2)nn1C 52565,c1(C(C(=O)NCC2CCOC2)N(C2CCCS2(=O)=O)C)cccc(Cl)c1Br 52566,c1(C(=O)NC2C3CN(C(C(C(C)C)N(C)C)=O)CC32)cc2cc(Cl)ccn2n1 52567,C(=O)(C1=COc2ccccc2O1)N1CCC(CNC(COCCCC)=O)(CO)C1 52568,C(=O)(CCS(=O)(=O)CC(C)C)N.C=CC(CO)NC(=O)OC 52569,C1(CN(C(=O)Cn2cnnn2)CC)CCCN(C(=O)CCOCCCOC)C1 52570,C1(NC(CCN(CCC)C)=O)CCCCCC1NC(=O)CC1CCC(F)(F)CO1 52571,c1(C(=O)NC2CCCN(C(C34CCC(C3)OC4)=O)CC2)cc2ccccn2n1 52572,C(=O)(C(F)C(C)(C)O)NCC1(C(=O)NCC=CC2CC2)CC(=C)C1 52573,c1(CNC(C(C)NC(=O)CN(C)C(N)=O)=O)ncoc1C1CC1 52574,Cc1cc(F)ccc1C(O)CNC(C)CC(c1ccc(F)cc1)O 52575,N1(C(c2n[nH]c(C)c2O)=O)CCC(CNC(=O)Cn2cc(Br)cn2)C1(C)C 52576,C(=O)(C=CSc1ccccc1)NCCN(C(c1nscc1N)=O)CC 52577,Nc1ccc(C(N2CCCCC(CNC(=O)CCNS(C)(=O)=O)C2)=O)nc1F 52578,N1(C(C2C(CC)CCN2C(C2CC3CCCC23)=O)=O)CCSC2(CCC2)C1 52579,N1(C(COCCCC)=O)CC2CCN(C(C3CCCCS3)=O)CC12 52580,N1(C(c2c(OC)nccn2)=O)CC(C2CCCCN(C(=O)COC3CCC3)C2)C1 52581,C1(CC)C(=O)NCCN1C(=O)CC(CNC(=O)CNC(C1CCC1)=O)C1CCC1 52582,N1(C(CS(=O)(=O)NC)=O)CCCC(C)(C)C1C(=O)NC1CN(C)C(C)(C)C1 52583,C1(NC(c2cn(CC(C)C)nc2)=O)COCCN(C(c2ccc(=O)n(C)n2)=O)C1 52584,c1(C(=O)NC2CCC(CNC(c3nocc3Cl)=O)C2)ccc(F)c2cnccc12 52585,c1(CC(=O)NC2(C)CN(C(C3C4CCC(=O)C34)=O)C2)ccc(F)cc1Br 52586,N1(C(CNC(=O)OCC=C)=O)CCCC1C(C)NC(C1(C(F)F)CC1)=O 52587,C1(NC(c2cnc(C)[nH]2)=O)C2CCC(C2)C1C(N1CCC(O)C(F)C1)=O 52588,C(CNC(c1ccc(-n2cncn2)cn1)=O)(C(C)(C)C)NC(C(C)OC)=O 52589,C1(C(=O)O)=NC2C(=C1)N=CN2CCN=C1NCC(CC(F)(F)F)N1 52590,C(=O)(C(C)Cn1ccnc1)N(C)CC1(NC(CCN(C(C)=O)C)=O)CC1 52591,C(c1ccc(F)c(F)c1)=CC(=O)N(CCCNC(=O)CSC(C)C)CC 52592,c1(C(=O)OC)cc(CNC(=O)N(c2ccccc2)CC(C)O)ccn1 52593,Cn1nc(Cl)c(C(=O)NC(C2CCCCC2)CNC(c2cncc(F)c2)=O)c1Cl 52594,C1(S(N)(=O)=O)(C(=O)NC2C(CNC(c3cc(C)oc3)=O)C2)CCC1 52595,C1(C(N(CCCCN(C(C(CCN(C)C)N(C)C)=O)C)C)=O)CCCC(=O)CC1 52596,C1(C(=O)NC(CCC)C)(CNC(=O)CC2(O)CCCC2)CC12CCC2 52597,C(=O)(C(C)(C)C(=O)NC(C)(C)C)N1CC(C(C(=O)NC(C2(C)CC2)CO)O)C1 52598,C1(C)(CC(=O)N(C)CC2CCCN2C(C2(C)COC2)=O)CCCCC1 52599,CC(C(=O)N1CCC(C)(C(=O)NCCOC2CCC2)CC1)S(C)(=O)=O 52600,S(=O)(=O)(c1cc(Cl)ccc1F)N1C(C(=O)Nc2ncc(OC)cc2F)COCC1 52601,CS(=O)(=O)c1ccc(C(=O)NCC(C2CC2)NC(C2(CO)CC2)=O)o1 52602,C#CCC(C)(C(=O)NCc1cnc(O)c(F)c1)NC(c1cnccc1C)=O 52603,C1(NC(c2c(C)cccc2)=O)CN(C(=O)CC2CNC(=O)C2)CC(C)(C)C1 52604,C1(NC(C=CC=CC)=O)CC2CCC1CC2NC(c1ccncc1O)=O 52605,N1(C(C2C(C)C2)=O)CCN(C(C2CC3CC2C3)=O)C(CS(C)(=O)=O)C1 52606,CCS(=O)(=O)c1ccc(CC(=O)N(C2CN(C(=O)C(C)NC(N)=O)C2)C)cc1 52607,C=CCCC(F)(F)C(=O)N1CCC(C(F)C(=O)NCC(=O)N(C)C)C1 52608,C(=O)(C(O)CCSc1cn(CC2CCCC(=O)N2)nn1)NCC1NC(=O)OC1 52609,c1(C(=O)NCC2C(C)(C)CCN(C(CCCOC)=O)C2)cnn2c(Cl)cccc12 52610,N1(C(C2CCC(C)CC2)=O)CC2(CO)CC1(C(=O)NC1CCN(C(C)(C)C)C1)C2 52611,N1(C(Cc2c(C)nsc2)=O)CC(C(N2CCCC2C(=O)N(C)C)=O)C2(CC2)C1 52612,Cc1ccc2c(C(=O)NC(C3CCCN3C(c3c[nH]c(=N)s3)=O)C)c[nH]c2c1 52613,C(C)(C(CC(=O)NC(c1noc(C)n1)(C)C)NC(c1[nH]cc(C)c1C)=O)OC 52614,C(=O)(C(C(C)C)C(C)C)N1C(CNC(C2CCCC(=O)N2)=O)CC(OC)C1 52615,CCCC(CCO)NCC1CCCN(c2cccnn2)C1 52616,N1(C(c2c(CC)scc2)=O)CCOC(CCNC(=O)CCCn2cccc2)C1 52617,C12(NC(c3cccc(O)c3)=O)CCC(C(N3CC4(CCC4)C3)=O)(CC1)CC2 52618,C(C)(C)(CCC(=O)NC1CCN(C(c2cc(F)cs2)=O)CC1C)OC 52619,Cc1cc(NCc2ccc(S(N)(=O)=O)cc2)ncc1S(=O)(=O)NC(C)CS(C)=O 52620,c1(C(N2CCC(O)(C(CNC(C(C)=C3CCC3)=O)C)C2)=O)cnc2scc(C)n12 52621,CS(=O)(=O)C(C(=O)NCC1(O)CCN(C(=O)CC2CC(C3CC3)C2)C1)C1CC1 52622,c1(C(=O)NC2C(C)N(C(c3cn4c(n3)SCC4)=O)CC2)cc(F)c(Cl)cc1Cl 52623,CC(C(C)C(=O)NC1(C2CCCCO2)CC1)NC(c1ncccn1)=O 52624,c1(CC(N2C(C)(C(=O)Nc3cncc(OCC)c3)CC2)=O)ccc(F)c(F)c1 52625,C1(CNC(CC(OCC)OCC)=O)CCCCC1NC(=O)CCCF 52626,Cc1ncc(C=CC(=O)NC2CCC(CCNC(=O)CCS(N)(=O)=O)C2)c(O)n1 52627,C(CCCC(CO)NC(C1ON=C(C)C1C)=O)NC(c1c(C)nc(CCC)o1)=O 52628,Cn1ncc2c(NCCCCCO)[nH]c(=NCC3CCc4ccccc43)nc12 52629,c1(C(=O)NC2C(NC(Cc3c(C)scc3)=O)CCOC2)ccc(N)c(Cl)n1 52630,c1(OC)cccc(N(CCCC2CCCO2)C)c1NC(c1ccccc1)=O 52631,Cc1ncc([N+](=O)[O-])cc1C(=O)NCCCCN(C)C(C1(C(C)(C)O)CC1)=O 52632,C1(C(=O)O)CC(F)(CNC(C2C=CCCN2)=O)C1 52633,CC1C(C(=O)NC(CCO)C2CCCC2)CCN1C(c1ccco1)=O 52634,N1(C(C2C(C)(C)C2CO)=O)CCCC(Cn2cc(-c3cncc(Cl)c3)nn2)CC1 52635,C1(NC(c2cc(C)[nH]n2)=O)COC2(CCN(C(C3(CO)CCOCC3)=O)C2)C1 52636,CCCS(=O)(=O)CC(=O)NCC1CC2(CO1)CN(C(c1c(C)ncn1C)=O)C2 52637,c1(-c2n(-c3cccc(C)c3)nc(C3CCOC3)n2)cn(C)cc(Br)c1=O 52638,c1(OC)ccc(N(C)C(C)=O)cc1.c12cc(n[nH]1)C(=O)COCC(=O)N2 52639,C(=O)(C1c2c[nH]nc2CN1C(c1cncn(C)c1=O)=O)N1CC(C(C)O)OCC1 52640,N1(C(CCNC(C(C)(C)C)=O)=O)CC(O)(C2(CNC(=O)CC(C)(C)O)CC2)C1 52641,c1(C(=O)NCCCC(C)NC(c2c(C)oc(C3CC3)n2)=O)ccc(O)c(F)c1 52642,c1(C(=O)NC(CC(=O)N(C)CC)C)ccc(OC)c(C#N)c1F 52643,c1(NCCN(C(c2ccn(CCC)n2)=O)C)cc(O)nc(O)n1 52644,C1(C(=O)NC(CC=C)CO)CC12CCN(Cc1cc(C(=O)O)cc(C)c1)C2 52645,N1(C(C(C2(O)CN(C(c3ccc(OC)o3)=O)C2)F)=O)CC(=O)NCC1C 52646,N1(C(c2cc(C)oc2)=O)CC(NC(=O)C(C)Cc2cnc[nH]2)C(N=[N+]=[N-])C1 52647,C(C(F)(C(=O)NC(CC)C(N)=O)C(C)C)NC(c1ccn(CCC)n1)=O 52648,c1(NCC(CNC(C2CC=CC2)=O)O)cc2nncn2cn1 52649,n1(CC(C)NC(=O)CCc2ncc[nH]2)cc(CNC(=O)C(C)(F)F)nn1 52650,c1(-c2n(-c3c(CC)cccc3)nc(C(O)CC)n2)ccc(F)c(Cl)c1F 52651,c1(C(N(C)CC2CCN(C(=O)C=CC3CCOCC3)C2)=O)cn2c(n1)CCCC2 52652,N1(C(c2c(C(C)=O)cccc2)=O)Cc2nccn2CC(NC(=O)C(C)CF)C1 52653,c1(C(N2CCCC(n3cc(C(C(C)C)O)nn3)C2)=O)ccc2ncn(C)c2c1 52654,C1(C)(CC(=O)NC(c2ccccn2)CC)CCN(C(=O)CCN2CCOC2=O)C1 52655,Cc1cc(C(=O)NCC(C2CC2)N(C(=O)CSS(C)(=O)=O)C)c(O)c(C)c1 52656,N1(Cc2cccc(N3CCC(COCCOC)C3)n2)CCNC(=O)C1 52657,c1(OC)cc(Br)c(CNC(=O)C(C2CCS(=O)(=O)CC2)F)cc1C 52658,c1(C(=O)NCCCNC(N)=O)ccc2cc(-c3ccc(F)s3)n(C)c2c1 52659,N1(C(c2c(C)nc(CO)nc2)=O)CCN(C(c2ccccc2O)=O)CC12CCC2 52660,C1(CCC(=O)NCC(CC)O)CCCCN(C(c2ccc[n+]([O-])c2)=O)C1 52661,C(=O)(CCCCC(F)F)NC(C)CCNC(C1(CF)CCOCC1)=O 52662,N1(C(C(CC)OC2CCCCC2)=O)CCCC(C)(CN=c2[nH]nc(C)o2)C1 52663,CC1CC(NC(c2ccnn2C2CCOCC2)=O)CN1C(=O)C=C1CC1 52664,N1(CC(C)NC(CC=CC)=O)CCN(C(c2cccc(C3CCC3)c2)=O)CC1 52665,C(F)(F)(C(F)(F)F)N(C(c1ccc(C(N)=O)cc1)C(=O)NC(CC)C)C 52666,c1(C(=O)NC(CNC(c2nc(OCC)sn2)=O)(C)C(C)C)ccc(N)c(C)c1F 52667,n1(CC)nc(C(=O)NC(C2CN(C(=O)Cc3ccncc3Cl)CCO2)C)cc1C 52668,Cc1[nH]nc(C(F)(F)F)c1C(=O)NC1CC(C)N(C(=O)CC(=O)NC2CC2)C1 52669,C1(C(=O)NC2C(NC(CN(C)C(c3cccs3)=O)=O)CCC2)Cc2cscc2C1 52670,C1(NC(c2ccc(F)c(Cl)c2F)=O)CCC12CCN(C(C1CCC(O)C1)=O)CC2 52671,c1(-c2n(C3CCN(CC)CC3)nc(C3CCCO3)n2)ccc([N+](=O)[O-])[nH]1 52672,CC(CN(C)C)CC(=O)NCCCCCNC(=O)CCc1nncnc1O 52673,C1(C(N(CCOC)CC)=O)CCOCCN1C(c1nc(C)ccc1F)=O 52674,N=c1cc(C(N2CCN(CC3CN(C(=O)C=CI)C3)CC2)=O)cc[nH]1 52675,C1(C)(C(=O)NCC(C)CNC(C2CC2C2CCC2)=O)SCCCS1 52676,C#CC1C(C(N2CCC2CNC(=O)CN2CCC(O)CC2)=O)C1(C)C 52677,C(=O)(CC(O)CC(C)C)N(CCOC)CCNC(=O)Cn1nc(C)nc1C 52678,N1(CC)CCN(CC(=O)NC(C)CCNC(C2CCC2C(F)(F)F)=O)CC1 52679,Cc1c(Br)csc1C(N1CCCC1Cn1cc(C2OCCO2)nn1)=O 52680,n1(CC(=O)NCC2C(NC(C=C(C)C3CC3)=O)COC2)ncn2nccc2c1=O 52681,c1(C(=O)NCCC(C)(C)NC(C2CCC(C)S2)=O)ccccc1-c1ncnn1C 52682,N(C(=NCCC1CCC2(CCC2)O1)NCc1cccc(F)c1)C1CC(C)C1 52683,C1(NC(=O)Cc2cncnc2)CC12CCC(NC(c1cc(Cl)cs1)=O)CC2 52684,c1(OC)ccn2ncc(-c3ccnc(NC(=O)C(F)(F)C(O)C4CC4)c3)c2c1 52685,CC1(c2nn[nH]n2)CCCN(C2CC2c2c(F)cccc2Cl)C1 52686,N1(C(c2sccc2I)=O)CC2CC2(C(=O)NC(CO)C2CC2)C1 52687,c1(C(C(=O)NCCCCCNC(=O)CC(C)c2ccco2)OC)ccc(Cl)cc1 52688,c1(-n2c(C)ncc2)cc(NC(c2cn(C3CC3)nc2C)=O)ccn1.c1nnco1 52689,C12(C(=O)NCCNC(C3CN(C(C(c4cnn(C)c4)C)=O)C3)=O)C=CC(CC1)C2 52690,Cc1c(Cl)sc(Cl)c1C(=O)NCCN(CC(C)O)C(=O)Cn1ccnn1 52691,CCCC(C(=O)N1CC(NC(=O)C=CC2CCC2)CC(F)C1)S(N)(=O)=O 52692,C1(NC(=O)Cn2cc(Br)cn2)CN(C(C2CC3(C2)CC3F)=O)CC12CCC2 52693,C(=O)(CC(C)(C(F)F)N(C)C)NCCN(C(C1(C)CCC(=O)N1)=O)CC 52694,CC12CCC(C(=O)NC3CC3NC(C3(O)CCC3)=O)(CC1)CO2 52695,CC1CC(C)C(CNC(C23CCC(CC2)C3)=O)CN1C(=O)C1=CCCCC1 52696,c1(CN2C(Cc3ccc(F)cc3)CCCC2)ccc(F)c(F)c1Br 52697,c1(C(=O)Nc2[nH]nc(CC)n2)cn(CC)nc1C(C)C 52698,C(CC(=O)N(C)CC1(CO)CC1)(C(C)(C)C)NC(c1cc(C)c(=N)[nH]c1)=O 52699,c1(C(=O)NCC(C)N(C(C(CC)CCOC)=O)C)cc2c(OC)ccc(C)c2[nH]1 52700,C(=O)(CCN(CCCO)C(C1CC1C(C)(C)C)=O)N(C(C#C)C)C 52701,CN1CC=C(CCNC(=O)CN(C(=O)CNC(=O)CC2CCOC2)C2CC2)CC1 52702,C1(N(C(c2ccc(SC)o2)=O)C)CCCN(C(=O)C=Cc2ccn(C)c2)CC1 52703,O=[N+]([O-])c1cc(S(=O)(=O)N2CC3CC2CN3C(=O)CN2CCCC2=O)ccc1Cl 52704,c1(C(=O)NCC(CC)(CC)NC(C2CC(C)(C)C2)=O)ccc(C)c(OCCF)c1 52705,c1(OC)cnc(C(=O)NC2CCN(C3CCCC3O)CC2)c(C)c1 52706,c1(SC)cn(C)nc1C(=O)NC1CC1CNC(c1ccc(CN(C)C)cc1)=O 52707,c1(C(N2CCCC(C(C)NC(CCOCCC)=O)C2)=O)nnc(O)cc1O 52708,c12ccccc1C(=O)N(C)C(C)CNC2=O.C(C(=O)NC)OC.C1CCC1 52709,C1(C(=O)NC(CNC(c2c(OC)noc2C)=O)C)CCCCCC1(F)F 52710,N1(C(C=Cc2ncn(C)c2)=O)CC(C2CC2C(=O)NCC2(C3CC3)CC2)C1 52711,c1(CC(=O)N(CC(CNC(C(CCC)OC)=O)C)C)ccc2ocnc2c1 52712,c1(C(N(C2CN(C(C)=O)C2)C)=O)cc2c([nH]1)CCOC2.C12(CCCCC1)C(=O)N2 52713,C(=O)(C1=CCCCC1C)NCC1CN(C(C2(C(=O)OCC)CCC2)=O)CC1O 52714,n1(CC(=C)C)c(N2CCCC2COc2ccccc2)nnc1-c1noc(C)n1 52715,C1(NC(C=COCC)=O)(CNC(C2CCCS2)=O)CCC(C)(C)CC1 52716,CC1(C)CCN(C(C2(C#N)CC2)=O)CC1NC(=O)CCCOCc1ccccc1 52717,O=C1CC(C(=O)NCC2CCN2C(c2ccccc2-n2cnnn2)=O)=NN1 52718,N1(C(COCC)=O)CC2CC(N(C)C(c3ccn(C(F)F)n3)=O)C1C2 52719,C1(C(N2C(CNC(CSc3nc(C)[nH]n3)=O)CC2)=O)CC(=O)N(c2cn[nH]c2)C1 52720,CN1CC2(C1)N=C1C=CN=C(N1)N(CC1CCCC1(C)CO)Cc1c2cccc1 52721,CC(C)C(C(=O)N1CC(NC(=O)C(c2ccc(F)cc2)O)C(O)C1)n1cccc1 52722,Cc1ccc(C(CNC(c2cnc(S)n2C2CC2)=O)NC(=O)CC(C)F)cc1 52723,CC1CC(C(=O)NCCn2ccc(C(=O)N(C)C)n2)CCS1(=O)=O 52724,C12(C(=O)NCC3C(NC(C=C(CCC)C)=O)CCC3)CC=CCN1CCC2 52725,CCCCCCCCC(CCCCCC)C(=O)NCC1CCN(C(=O)CC)C1 52726,c1(CCC(=O)NCCCN(C)C(c2ncccc2Cl)=O)ccc2cccnc2c1 52727,C(=O)CC.N(C1=CCCCC1)C(=O)NCCC(=O)OCC 52728,N1(C(C(C)n2cnnn2)=O)CCC2CN(C(C3(c4cccc(F)c4)CC3)=O)CC12 52729,c1(OCCCNc2cnc(CC(=O)OCC)nc2)ccc(S(N)(=O)=O)cc1 52730,Cc1ccc(CC(N2CCCC2CN(c2nc(Cl)ncc2Br)C)=O)cc1C 52731,N1(C(C2(OC)CC2)=O)CC(CNC(C2(C)CC(F)(F)C2)=O)OC(C)(C)C1 52732,c1(C(=O)NCCN(C(CS(CC)=O)=O)Cc2ccccc2)cc(C#N)cc(C)n1 52733,C(c1ccc(Br)s1)=CC(c1nnnn1C1CCOC1)NCC(CC)(C)C 52734,C1(CNC(=O)NC2N(C(CCC)=O)CCCC2)(CO)CC2CCC1C2 52735,CN1CCn2nc(C(=O)NCC3CCN3C(c3cccc([N+](=O)[O-])c3)=O)cc2C1 52736,Cn1cc(CC(N2CCCC2CCC(=O)NC2C=CCC2)=O)nn1 52737,CCC(C)(C(=O)NC1CCC(NC(c2ccnc(C)n2)=O)CC1)C(N)=O 52738,c1(C(N(C(CCNC(c2c(CC)nns2)=O)C)C)=O)ccc(C)n1C 52739,N1(C(C2C(CC)CCC2)=O)CCN(C(c2ccc(C)c(O)c2)=O)CC1C 52740,N(C1CCC=Cc2ccccc21)c1cc(NC(c2ccc(O)nc2)C)ncn1 52741,C1(N(C)C)CCCN(C(C2CN(C(=O)CC3CCCC4CC34)CCO2)=O)C1 52742,CC1(C)CC(CC(N2CCCC2CNC(C2(c3ccsc3)CC2)=O)=O)C1 52743,Cc1c(C(=O)NC2CN(C(C3(F)C(F)(F)C3(F)F)=O)C2)oc2ccc(Cl)cc12 52744,C(C)(C(CCc1ccccc1)NC(c1cc[nH]n1)=O)NC(Cc1cc(C)sc1)=O 52745,c1(C(N2CCC(C(NOCC)=O)C2C2CC2)=O)cnn2cccc2c1 52746,Cc1c(C(=O)NCC(F)CNC(=O)C(C)(Cl)Cl)oc2cc(Cl)ccc12 52747,C(=O)(C1=CCCCC1C)NCC(C(=O)NC1CC(CSC)C1)C 52748,N1(C(c2c(CC)nccn2)=O)CC2CCCC2(C(=O)N(C2CCOC2)CC)C1 52749,C1(NC(C=CCOC)=O)C2CC3C1C3C2C(=O)N(C(CF)CF)C 52750,c1(OC)ccc(C(=O)NCC2CCN2C(C2(CO)CC(C)(C)C2)=O)c(O)c1F 52751,C1(COC)(NC(=O)CC2(OC)CCC2)CCCN(C(=O)C(C)(C)CCOC)C1 52752,N1(C(CSCC(C)C)=O)CCOC2(CCN(C(=O)CC3CN4CCN3CC4)C2)C1 52753,c1(C(N2CCC(C(C)NC(Cc3cc(CC)no3)=O)C2)=O)c(C)noc1C 52754,S(=O)(=O)(c1ccc(NC2CCOCC2C)cc1Cl)NCC(C)(C)OC 52755,c1(OC(C)C(=O)NC2CCCN(C(=O)CCCF)C2)ccccc1Br 52756,C1(NC(c2cccc(=O)n2O)=O)CC2(CCN(C(c3ccno3)=O)CC2)C1 52757,N1(c2nc(C)c(Br)cn2)CC(C)CN(C(C2C3CCCC23)=O)CC1C 52758,N1(C(C2C(C)(C(=O)O)C2)=O)CCOCC1Cc1cn(C2CCCC2)nn1 52759,N1(C(C2CCN(C(C=CCC)=O)C(C)C2)=O)CCCN(C=O)CC1 52760,c1(C(=O)NC(CC=C)CNC(=O)C(C)OCCN(C)C)ccc(O)nc1Cl 52761,N1(C(CCCn2cc(-c3cn(CC)nc3)nn2)=O)CCCC(CC(N)=O)CC1 52762,N1(Cc2c(C)nn(C3CCOCC3)c2Cl)CC=C(c2ccnn2C)CC1 52763,c1(N2C3CN(C(C(CC)(C)CC)=O)C(CC3)C2)ccc([N+](=O)[O-])c(O)n1 52764,c1(NC)snc(C)c1C(=O)NC1CCC(N(C)C(c2ccc(O)nc2)=O)CC1 52765,N1(C(CC=CCC)=O)CC(OC)CC1(C)CNC(c1ccc(C)cc1N)=O 52766,N1(C(c2c(OCCC)cccc2)=O)CCC(NC(c2cnsc2C)=O)C(C)C1 52767,N1(C(c2c(Cl)ccc(C)c2)=O)CCC2CN(C(C3(C(C)C)COC3)=O)CCC2C1 52768,c1(CN2CCCC(NC(=O)COC(F)(F)C(F)(F)F)CC2)cc2ccccc2o1 52769,Cc1cc(C)c(C(N2CC=CC(NC(c3ccsc3C)=O)C2)=O)c(Cl)n1 52770,C(=O)(C1=CC2(CCOC2)C1)NCC(CN(C(c1cc(N)c(C)c(N)c1)=O)C)C 52771,CC(C)C(F)(F)CC(=O)N1CC(CNC(c2c[nH]c(C(N)=O)c2)=O)CC1C 52772,c1(SCC(=O)NCC(O)CNC(c2c[nH]ccc2=N)=O)ccsc1[N+](=O)[O-] 52773,N1(CC(=O)N(CCC(=O)NC(C2CCCC2)C)CC#C)CCCC1C 52774,CC(C)CCCCC(=O)N1CCN(C(c2cccc(-c3nc(O)n[nH]3)c2)=O)CC1 52775,CCCCC(O)CCC(=O)NC(C1CCN(C(=O)CN2CCC(C)CC2)CC1)C 52776,CCCC(O)CC(=O)NCCN(C(=O)C(c1ccc(CC(C)C)cc1)C)C 52777,N1(C(=O)NC)CCC(NCCCOC(C2CCC2)C)CC1 52778,CC1(NC(c2ncc(Cl)nc2Cl)=O)CCCN(C(c2cscn2)=O)C1 52779,N1(C(c2c(C)cn(C)n2)C(=O)NCC(C)C)CCC(O)C(CC(C)C)C1 52780,C1(NC(c2c(OC)cc(O)nc2)=O)CCC2(CC1)CN(C(=O)C(C)(C)Br)C2 52781,C(=O)(C(C)(C)CC(F)F)NCC(CN(C(=O)C(Cc1cccc(Cl)c1)=NO)C)O 52782,N1(C(C(C)SC(F)(F)F)=O)CCOCC(NC(C2(c3ccno3)CCC2)=O)C1 52783,c1(C(=O)NC(c2ccc(CNC(=O)C(O)CN(C)C)cc2)C)cnc(O)n(C)c1=O 52784,N1(C(C(C)C2CCOC2)=O)CCC(C2CC2)(CNC(=O)COCC2CCCC2)C1 52785,Cc1c(C(N2CC(NC(C3CCCO3)=O)C(F)C2)=O)cc(F)cc1Br 52786,c1(NC(CNC(Cc2cc(C)on2)=O)C(C)C)ncnc2sccc12 52787,C1(C(=O)NCCN(C(C2CC2F)=O)CC)(CO)CCCC1 52788,Cc1nnc2cc(NCCCCNC(=O)C(c3cccc(Cl)c3F)(C)C)ncn12 52789,C1(NC(C2CCC(=O)NC2)=O)CN(C(=O)CC23CCC(CC2)C3)C2(CCOC2)C1 52790,C1(NC(CS(C)(=O)=O)=O)CN(C(=O)C=Cc2cccc(F)c2)CCC1O 52791,C1(NC(c2nc(CCC)oc2)=O)C2CC3CN(C(=O)CC4=NNC(=O)C4)C1C3C2 52792,CC(CC(=O)N(CCCNC(=O)CCC1CC(F)(F)C1)CCO)C1CCCO1 52793,c1(C(=O)NC2C=CCN(C(c3c(OC)cccc3O)=O)C2)c[nH]c(C)c(Cl)c1=O 52794,Cc1ccc([N+](=O)[O-])c(C(=O)NC2COCCC2NC(c2ccncc2C)=O)c1 52795,C(=O)(C1=CCCCC1P(C)(C)=O)N1CC2(OCCN(C(C(C=C=C)C)=O)C2)C1 52796,c1(C(=O)NC(c2cn(Cc3ccc(Cl)nc3)nn2)CCC)cn2ccccc2n1 52797,c1(CN=C(NC(CC)C)NCC2OCC2(C)C)ccc(C#N)c(F)c1 52798,C1(C(=O)NCCCNC(=O)CC2CCCO2)(Cc2cccs2)CCCCC1 52799,C(CNC(=O)C(N1CCCC(C)C1)=O)(C(F)(F)F)OCC(=O)OC 52800,c1(C(N2CC(C(C(=O)NC(C(C)C)C3CC3)OC)C2)=O)cc(O)cc(=O)o1 52801,C1(C(N2CCCC(CNC(=O)CN3CCCNC3=O)C2)=O)COC2CCCCC12 52802,N1(C(c2c(C)nc(CSC)s2)=O)CCC(NC(=O)C(C(C)C)NC(N)=O)C(O)C1 52803,CC1(C)CCC(CNC(C23CC=CC(C2)OC3)=O)N(c2cc(Cl)ncn2)C1 52804,C1(C(=O)NC(C2(O)CN(C(C3(CC4CC4)CC3)=O)C2)C)CC12CCCCCC2 52805,Cc1ccc(F)cc1C(N1CC(C(=O)N(C(CCO)C(F)F)C)C(F)(F)C1)=O 52806,n1(CCC)ccc(C(=O)NCCCCN(CCCNC(C2C=CCS2)=O)C)n1 52807,C12(C(=O)NC3CCC(C)N(C(=O)CCC(N)=O)C3)CCC(CC1=O)C2(C)C 52808,c1(CC(=O)NCC23OCCC(NC(C(CC)C#N)=O)(C2)C3)nc2ccccc2s1 52809,N1(C(c2c(Cl)ccc(C)c2)C(=O)NC2CC(F)(F)C2)CCCC1C1CCCO1 52810,C(C(F)C(=O)NOCC(O)CO)C1CN(C(C(CC)N(C)C)=O)C1 52811,C1(NC(Cc2ccc(SCC)cc2)=O)CC2CCC(C1)N2C(=O)C(C)(Cl)Cl 52812,Cc1ccc2[nH]c(C(=O)NCC(O)CCNC(=O)CCC(C)C)cc2c1 52813,C1(NC(C(C)SC)=O)CCN(CC2CCCCO2)C(C)C1 52814,c1(C(=O)NC(CC=C)CNC(=O)Cn2cnnc2O)ccc2nc(C)cn2c1 52815,C1(N2CC(C)C(NC(c3ccc[n+]([O-])c3)=O)CC2)CCc2ccccc2NC1=O 52816,c1(C(N2CCCC(C)(NC(C3C(C)C3)=O)C2)=O)cncc2ccsc12 52817,c1(OC)ccc(-c2n[nH]cc2CNC(N2CC(CO)CC(CO)C2)=O)cc1Cl 52818,N1(C(c2ccc(O)c(O)c2)=O)CC(C(N2CC3COCC3C2)=O)CC(F)(F)C1 52819,c1(NC(c2[nH]cc(COC)c2)=O)cccc(NC(C2(C)CCCO2)=O)c1 52820,N1(C(c2ccc(I)s2)C(=O)NC(C(=O)OC)C)CCOC(C(F)(F)F)C1(C)C 52821,c1(Nc2cc3c(cc2)OC(C)C3)nccc(=NC2CCCn3nccc32)[nH]1 52822,N1(C(CC(CC)(C)C)=O)CC2OCCN(C(C3CCCN4CCCCC34)=O)C2C1 52823,C1(CC(=O)NCC2CCN(C(=O)C=Cc3cccs3)C23CC3)CC(O)C12CCC2 52824,C1(C(=O)NCCCOCCCNC(CC(C)N(C)C)=O)CC12CCC1(CC1)CC2 52825,c1(CCOC)cccc(CNC(=O)C(c2ccc(Cl)cc2)N(CC(=O)OC)C)c1 52826,C1(C(=O)OC)CC2CN(C(=O)C(N3CCCC(O)C3C(=O)OC)=O)CC12 52827,c1(OCC)ccc(NC(=O)CN2CCC(c3ccccc3F)C2)cc1 52828,C1(NC(c2cc(C)no2)=O)CCCCC1C(=O)N(C)CC1(N(C)C)CC1 52829,N1(C(c2ccc(F)c(C(F)(F)F)n2)=O)CC(CO)c2ccccc21 52830,c1(C(N2C(CNC(C(C(=O)NC)(C)C)=O)CC(O)C2)=O)cc2[nH]nc(C)c2cn1 52831,C1(C(=O)NC2(C#C)CC(F)(F)C2)C(C2CC2)CCN1C(=O)C=Cc1ccoc1 52832,N1(C(c2n(CC)cnn2)=O)CCC2(CCCC2NC(c2ccc(C)s2)=O)C1 52833,C(C(CC(C)C)NC(=O)CC(O)C1CC1)NC(c1c(NC(C)=O)cccn1)=O 52834,c1(CC(=O)NCC2CN(C(C3CCC4CC34)=O)C2)nnc(-c2ccccc2)o1 52835,C1(OC)CN(C(=O)CCC2CCC(C(N)=O)O2)CC1NC(c1cccc(Cl)c1)=O 52836,C1(CN(C)CCN(C)C(c2ccccc2Cl)=O)COc2ccccc2O1.C1CN1 52837,N1(C(C(c2n(C)cnc2)O)=O)CC2(CCC(NC(c3cnnn3C)=O)CC2)C1 52838,C(=O)(CC(C)CC(F)(F)F)NC1CCC(NC(c2nn(CC)c(C3CC3)c2)=O)C1 52839,c1(NC(CC2N(c3nccc(OC)n3)CCC2)=O)cc(Br)cnc1I 52840,c1(SCC2(C)C(C(C)O)C2)ccc(C2CC2)cc1 52841,C(=O)(CC1CCc2ccccc21)N1CC(C2CN(C(C(C)(C)C)=O)C2)C1 52842,C(=O)(CS(=O)(=O)C1CC1)N1CCC(NC(CC2C=NN(C)C2=O)=O)C1 52843,CCCC(C(=O)NCCCCCNC(=O)C=Cc1cn[nH]c1)S(N)(=O)=O 52844,C(=O)(C(C)(C)CCCC(=O)N(C)C(c1cn(-c2c(C)nn(C)c2Cl)nn1)C)OC 52845,C1(CNCC(c2ccc(Br)cc2)C)CCC2(C1)CC2(F)F 52846,C1(NC(c2[nH]cc(CC)c2)=O)CC(F)CN(C(c2cccc(F)c2)=O)C1 52847,C1(NC(CCc2cc(C)on2)=O)CN(C(=O)CN2CC(C)(C)C2)CC(C)(C)C1 52848,Cc1nc(C(=O)NCCc2csc(NC=O)n2)cc(O)n1 52849,c1(C(N2C(CNC(=O)CC3CC4CCC3CC4)CC2)=O)c(F)cc(F)cc1Cl 52850,CC(N=c1ccc(C#N)n[nH]1)C1CCCCN1C(=O)CCN1CCCC1 52851,N1(C(C(Cc2c(C)n[nH]c2C)C)=O)CCCC2(NC(c3n[nH]cc3Cl)=O)CC2C1 52852,N1(c2c(OC)cncn2)CCC2(CC1)OCCCC2NC(C1CCC(=O)N1)=O 52853,C1(CNC(CCC)=O)CN(C(C2CCCCC23CC3)=O)CC12CCC2 52854,N(C(=NCc1cc(C)ccc1O)N1CCCC(OC)C1)C(COCC)C 52855,C#Cc1cccc(C(N2CCC(C3CCN(C(=O)CN(C)C)CC3)C2)=O)c1C 52856,c1(N2C(C)CC(NC(c3c(C)cc(Cl)cc3)=O)C2)cc2nnc(C)n2cn1 52857,C(=O)(C1=CC(C)(C)C1)NC1C=CCN(C(C(c2ccc(N)cn2)C)=O)C1 52858,C(CS(=O)(=O)CC(=O)N(C)CC1CCCN(C(c2ccc(OC)cc2)=O)C1)OC 52859,Cc1cc(C(=O)NC(Cn2ccnn2)C(=O)NCC2(C)CCCC2O)nnc1C 52860,C(CC(C)(C)CBr)(c1nnnn1CCCl)NCC(C)C(F)(F)F.C1CS1 52861,C1(CC)COCC1NC(=O)C(C)(C)NC(=O)C(C)=CC(C)(C)C 52862,c1(NCC=CCNC(C(CC)C(=O)OC)=O)ccc([N+](=O)[O-])cc1C(F)F 52863,N1(C(C(C)Cc2cnc[nH]2)=O)CCC(C)(CNC(=O)CCc2nncs2)C1 52864,C1(NC(C2C(OCC)C2)=O)CC1C1CCCN(C(=O)CCc2cccnc2Cl)C1 52865,c1(OCC)nc(C(=O)NC(C)(C)C(C)NC(=O)C(C)NC(=O)C(C)(C)C)ns1 52866,C(=O)(CC(C)C(C)C(C)C)N1CC(C(C)(C)O)(CNC(C(CCCC)C)=O)C1 52867,C1(C(=O)NCC(CNC(=O)OC(C)(C)C)CO)CC2(C1)CC(N=[N+]=[N-])C2 52868,C12(CNC(c3ccc(-c4ncc[nH]4)nc3)=O)CC1CN(C(c1coc(O)n1)=O)C2 52869,C1(C(N2CC3CCCC3C2)=O)CN(Cc2cc(Br)ccc2Br)CCC1(F)F 52870,C1(NC(N(C2CCCC2C#N)CC(C)C)=O)CC2C=CC1CC2 52871,c1(OC)ccc(Br)c(C)c1C(=O)NC1CN(C(c2cc(C)c(C)cn2)=O)C1 52872,N1(C(C(n2ccc(C)n2)C)=O)CCC2(CCN(C(=O)CCCC3CC3)CC2)C(C)C1 52873,C1(C(N2CCCC(N(C)C(c3scnc3Cl)=O)C2)=O)CCc2cncn2C1 52874,c1(COC)cc(CC(=O)NCC(C)N(C)C(c2c[nH]nc2C(C)C)=O)no1 52875,C(=O)(C(C)(C)C(F)F)N1CC(OCC(=O)NCc2cc(C)c(C)s2)C1 52876,c1(NCC(=C)C)cc(N2CCCC(OCC)C2)nc(C(F)(F)F)n1 52877,N1(C(c2n(C)nnc2)=O)CC2(CC2)CC1CC(=O)NCC1(C)CC1(F)F 52878,CC1CN(C(=O)CN(C)C)CC2(CCN(CC(=O)N(C)C)C2)O1 52879,N1(C(C(C2CCN(C(C(C)=CCC)=O)C2)F)=O)C2CCC1CC1(C2)N=N1 52880,C(=O)(CCCN(C)C)N(C(C)C(=O)NCC1(CCO)CCCC1)C 52881,CC(C)C(O)CC(=O)NC12CC(NC(=O)CCC3(C)CC3(F)F)(C1)C2 52882,c1(SC)nc(=NC(CNC(=O)C(C2CCCCCC2)OC)CO)s[nH]1 52883,CC1(CNC(=O)CCCCNC(N)=O)CCCN(C(=O)C(F)OC(F)(F)F)C1 52884,c1(C(N2CCCC(N(C(=O)C#CC3CCC3)CCO)C2)=O)cn2ccccc2n1 52885,c1(-c2nccc(NCc3c(CC)c(C)ccc3)c2)c(F)cc(CO)cc1F 52886,c1(-c2cn(C3CCN(C(C(C)OCCC=C)=O)C3)nn2)cc(F)ccc1F 52887,C1(N(C(c2c(COC)ncs2)=O)C)CC2CCC(C1)N2C(c1ccc(F)s1)=O 52888,C1(CNC(CC2(CSC)CC2)=O)CN(c2ncns2)CCC12CCOC2 52889,C(=O)(N=c1cc[nH]cc1I)NC(C1(F)CC1)C 52890,N1(C(CC=CC=C)=O)CCCC2(C1)CN(C(=O)CC1CCCOC1)CCO2 52891,CC(C(=O)NC(CNC(=O)CCCn1c(O)nnc1O)C(C)(C)C)C(C)(F)F 52892,C1(NC(C2CCC(CCCC)O2)=O)CN(C(c2cc(OCC)ncn2)=O)CC1F 52893,c1(C(N2CCCC(C3N(Cc4ccc(OC)s4)CCC3)C2)=O)ccnc2[nH]nnc12 52894,c1(CNC(c2cccc(F)c2)c2onc(C)n2)nn(C)c(C(N)=O)c1Cl 52895,Cc1cc(CCNC(C2CCN(c3cccc(F)c3)CC2)=O)c(C)s1 52896,C1(C(N2CC(C)=C(C)CC2)=O)N(C(c2cn(C3CC3)cn2)=O)CC12CCCC2 52897,O=C1C2CC(O)CCN2C(=O)N1CCOC.C1(C(O)C2CC2)CCCCC1 52898,C1(CNC(Cc2cnn(C)n2)=O)CC2(CO1)CN(C(c1nc(Cl)ccc1N)=O)C2 52899,N1(Cc2c(Cl)ccc(Cl)c2)CCc2c(Cc3ccccc3)cccc21 52900,CC1=C(C(=O)N2CC(NC(c3csc(-c4cnccn4)n3)=O)C3(CC3)C2)CCC1 52901,C1(CC=C)(C(=O)NCC(C)(C2CCC2)NC(C2(CSC)CC(=O)C2)=O)CCCC1 52902,C(=O)(CC(C)CN(C)C(=O)NCc1cc(C)nn1C)OC 52903,C1(C(=O)NC(C)C(c2ccc(Cl)cc2)O)CCC(=O)C(C)C1 52904,C(CCCCCNC(C1OC2CCC1C2)=O)n1cc(-c2cc(C(=O)OC)on2)nn1 52905,c1(CC(=O)N(CCCNC(=O)CCC2CC2(F)F)CCO)ccc(Cl)nc1 52906,N#CC1CCCC1OCCNS(=O)(=O)NC1CC1 52907,CC1CN(C(C23CC2COC3(C)C)=O)CCN1C(c1ncn(C(C)(C)C)n1)=O 52908,CCCCC(C)C(=O)N1CC2(CC2)CC1CNC(=O)CCCN1C(=O)CNC1=O 52909,C1(CC)CCCCC1C(=O)NCc1ccc(CNC(C2CCCC(=O)N2)=O)cc1 52910,C1(NC(C(C)=C(CC)C)=O)CC2CC1CC2C(=O)OC(c1ccccc1Br)C=O 52911,c1(CC(C)NC(=O)NCCCCC(=O)NCC(F)(F)F)ccc(F)c(Cl)c1 52912,C1(CNC(c2c(SC)nccc2)=O)CN(C(C2CCC(C)CO2)=O)CCN1C 52913,Cc1cc(C(=O)N(C2CCN(C(=O)CSc3n[nH]c(=N)s3)CC2C)C)nnc1C 52914,C(=O)(C1CCCc2nc(C)[nH]c21)NCCN(C(=O)C(C)n1ccnc1)CC 52915,C1(NC(C2(CCN(C)C)CCCC2)=O)CCCN(C(C2CNC(=O)C2)=O)CC1 52916,C1(NC(Cn2c(C)c(Cl)cn2)=O)CN(c2cc(C3CC3)ncn2)CC2(CCC2)C1 52917,C(=O)(C(O)CC(C)C)NC(C(=O)NCc1c(C)cccc1)c1ccco1 52918,C1(CN2CCCC(C(N3CCN(C)CC3)=O)C2)CN2CCC1CC2 52919,C1(N(C(CC2(OCC)CCC2)=O)C)CCC(NC(=O)C=Cc2nc(C)cs2)CC1 52920,C(=O)(C1CNC(=O)c2ccnn21)N(CCCNC(=O)CN(C)S(=O)(=O)N(C)C)C 52921,C1(N(C(=O)COC2CCCCC2)C)CCCN(C(=O)CCC2CC2(C)C)C1 52922,N1(c2n(C)nnn2)CC2CC(NC(C3CN(C4CCOC4)C3)=O)C2C1 52923,C(=O)(CCCC(F)F)N1C(CNC(=O)CC23CC(C2)C3)CC(OC)C1 52924,c1(C(=O)NCC2N(C(c3ccc(C)nc3N)=O)CCC2C)ccc2scnc2c1 52925,C(C)(C(O)C(F)F)NC(C(CNC(c1cc(C(F)F)[nH]n1)=O)OC)=O 52926,C1(C(CNC(C2(CC)CCOC2)=O)C)CCN(C(c2cccn2COC)=O)CC1 52927,c1(C(=O)NCCOCCCNC(c2cc(O)cs2)=O)csc(-c2ccsc2)n1 52928,C12CCCN(C1)C2=O.n1(CC(COC)O)cc(C(O)C(C)(C)C)nn1 52929,c1(CCNC(c2c(CC)noc2)=O)cc(F)ccc1C 52930,c1(C(=O)NCCOC2CCN(C(CCNC(C)=O)=O)C2)c(Cl)ccc2c[nH]nc12 52931,Cc1c(C(=O)N(C)CCOCCNC(=O)CN2CCC(C)CC2)cccc1Cl 52932,N1(C(C(C)CN2CCOCC2)=O)CCC2CN(C(c3cc[nH]c3)=O)CC12 52933,c1(CC(=O)OC)ccc(C(=O)NC(C)(C)C(C)NC(C2CC23CCC3)=O)cc1 52934,CCS(=O)(=O)CC(=O)NCc1cccc(C)c1.C1C(CC(C)O)N1C 52935,c1(-c2ccc(C(=O)NCCSC)s2)ccccc1-c1cnc(F)cc1 52936,CC1CC(C(=O)N)C1(C)C.N1(CCn2cc(-c3cscn3)nn2)CCN(CCO)CC1 52937,c1(N(C(=O)COC)CCS)cc(C)ccc1C 52938,C1(C(CC)C(=O)N2CC(NC(C3(C)CC3)=O)C2)CCC(C)CC1 52939,C1(NC(=O)NCCCCCO)C2Cc3ccc(Br)cc3C12 52940,C1(C(=O)NC(C2(O)CCN(C(C3(C)CC(=O)C3)=O)C2)C)CCCOCC1 52941,N1(C(CC2CCCN(C(CC(CC)(C)C)=O)C2)=O)CCn2ccnc2C1C 52942,c1(C(c2n(CC)nnn2)NC2CCCC2CCOC)cccc(C)c1C 52943,c1(C(=O)NCC23CC(NC(=O)COc4ccsc4)(C2)C3)ccc(F)cc1F 52944,c1(Cc2nc(C3OCCN(CC(=O)NC(CC)(C)C)C3)on2)c(C)cc(Br)cc1C 52945,N1(C(CCCNC(N)=O)=O)CC2CCC(C1)N2C(C1CC1c1ccc(Cl)cc1)=O 52946,C1(c2n(C(C(=O)OC)C)nnn2)(NCCS(=O)(=O)CCO)CC2(C1)OCCO2 52947,Cc1cc(F)ccc1C(=O)NC(C1CN(C(C2(C(C)C)CC2)=O)CCO1)C 52948,CC(C)CC(C)C(=O)NCC(C)CN(C)C(c1nccc(Br)c1O)=O 52949,CC(C)C(C(=O)NC1COCC1CNC(c1cc(O)n(C)n1)=O)c1cnn(C)c1 52950,N1(C(c2c(CC)cc[nH]2)=O)CCC(CO)C(NC(C2(CCF)CCC2)=O)C1 52951,C(C(C(=O)N1CCCC1CNC(C)=O)C(C)(C)C)NC(CC(=O)OC)=O 52952,N(C(=NCCCCl)N1CCCC2(CCCOC2)C1)Cc1cccc(C#N)n1 52953,CN1CCC(C(=O)N(C2CCCN(C(=O)CC(C)(C)c3cccs3)C2)C)C1=O 52954,S(=O)(=O)(c1cccc(F)c1C)NCC1(O)CN(Cc2c(OC)c(F)ccc2)C1 52955,N1(C(c2c(C)n(C)cn2)=O)CC(C)N(C(C2CC2(C)C(C)C)=O)CC1C 52956,c1(CC(C)C)ccc(NC(=O)C(N2CCNC(CCN(C)C)C2)=O)nc1 52957,C1(NC(CC(C)N2CCCC2=O)=O)C2CC1CN(C(c1ccc(Cl)c(Cl)c1)=O)C2 52958,c1(CCC(=O)NCC(CNC(c2ccccc2)=O)CO)cnc2ccccc2c1 52959,C1(NC(=O)CC(F)F)CC2CC(C1)N(C(C1CCS(=O)(=O)C1)=O)C2 52960,N1(C(CCNC(C2(O)CCSCC2)=O)=O)CCC(O)(CO)CC1 52961,c1(C(=O)NCCC2CCCN(C(c3cc(OC)ncc3)=O)C2)cc(C#N)[nH]c1C 52962,c1(C(=O)NCCCCC(C)NC(c2c(CCC)n[nH]c2)=O)cc(C)ccc1C 52963,CN1CCN(C(C2C3CCC(=O)C23)=O)C(CNC(c2ccno2)=O)C1 52964,C1(NC(CC(C=C)CC)=O)CC2CCC(C1C)N2C(=O)CC1=CCCCC1 52965,c1(CC)ccc(C(=O)NC2CC(CCNC(=O)C(n3cc(Br)cn3)C)C2)o1 52966,c1(NCC)cnc(C(=O)Nc2c[nH]nc2-c2cccc(OC)n2)cn1 52967,c1(C(=O)NCC2CCC(N(C(C(C)OCC#C)=O)C)CC2)ccc(O)c(Cl)n1 52968,CCC(C)CC(C)N(C(=O)C(CCOCCO)NC(=O)C=CC(F)(F)F)C 52969,c1(C(C(=O)N(CCNC(C(C=C)c2ccccc2)=O)CCC)C)cccc(O)c1 52970,c1(C(=O)OCC(=O)NC(C(=O)NC)(C)C)cccnc1N1CCCC1 52971,C(CC(C)C(=O)NC(CNC(c1coc(CS(C)(=O)=O)n1)=O)CO)=CC 52972,C1(C(N2CC(CCCCNC(CNC(CC(C)(C)C)=O)=O)C2)=O)CCC(C)(C)OC1 52973,N1(C(CC(COC)C)=O)CCCC2(C1)CN(C(=O)CC(C)CN(C)C)C2 52974,C1(CNC(=O)CC2CN(C(=O)CCN3CCCC3=O)C2)CCC(C(F)(F)F)CC1 52975,c1(C(=O)NC2(C)CCN(C(C3C(C)C3C)=O)C2)cc(O)nc2ccc(F)cc12 52976,C1(CNC(C(=O)NCc2ncc[nH]2)=O)CCCN(c2nc(C(F)(F)F)ns2)C1 52977,c1(NC(CCN(CC=C)C(C2CC2C2CC2)=O)=O)ccccc1CCC 52978,C(=O)(C(C)CC1CCC1)NCC(CC)N(C(=O)CSCc1cccs1)C 52979,CCC(C)(C(=O)NCC1(C(C)NC(=O)CC2C(C)(C)C2(C)C)CC1)OC 52980,n1(C(CC)C)ccc(=NC(=O)C(O)CCCNC(=O)C=Cc2cncs2)[nH]1 52981,n1(CCC(=O)NCCCN(C(C(C)=C(C)C)=O)C2CC2)nc(C)cc1C 52982,O=C(CSC1CCC1)N=c1ccn(C(F)F)[nH]1.C1(=O)CN1CC1CCC1 52983,C1(C(=O)NC(CN(C(=O)C=NOC)CC)C)CCN(c2cnccn2)CC1 52984,N12CCC(CC1)C2=O.N1(CC2(NC(=O)CC34CCCC3C4)CC2)CC2CCC1C2 52985,c1(NC(=O)NC2CCCN(C3CCCC3)C2)ccc(F)c(Br)c1F 52986,c1(C(=O)NC(C(C)NC(CCc2c(C)noc2C)=O)C(C)C)cc(Cl)ncc1O 52987,C=CCC(CC=C)C(=O)N1CCCC(C)C1CNC(c1cnc(S)nc1)=O 52988,C(CC1CC1)(C(=O)N(C)CCC1CCCN1C)NC(CC1CC(C)C1)=O 52989,c1(OCC(N2CC(CNC(C(n3c(C)cc(C)n3)C)=O)C2)=O)ccc(Cl)c(F)c1 52990,Cc1c(Cl)ccc(C(=O)NC2CCC(N(C(=O)COCC(C)(C)C)C)C2)c1N 52991,c1(CN(C)CC2CCCN(C(c3cnc(Cl)cc3I)=O)C2)cc(Br)cc(O)c1O 52992,Cc1nc2ccc(C(=O)N(CC(C)NC(C3CC(C)(C)CN3C)=O)C)cc2s1 52993,c1(C(=O)NCCNC(CC2CC(C)(C)OCC2)=O)cc(Br)cn2ncnc12 52994,C12(NC(c3ccc(C)c(F)c3)=O)CCCC1N(c1ncc3ccnc-3[nH]1)CC2 52995,c1(C(=O)NCC2(CCNC(CC(CC)CC)=O)CC2)[nH]c2cc(C)ccc2c1C 52996,C(CCS(=O)(=O)NCC(=O)NCCOC1CCN(C(=O)C=NOC)C1)OC 52997,C#Cc1ccc(OCC(=O)NCCNC(=O)CC2CC(CC)=NO2)cc1 52998,N1(C(C2OCCN(C)C2)=O)CC2CC(C1)C2NC(=O)CCSCc1ccccn1 52999,CC(CCCO)N=c1[nH]c(N2CC(C)(C)Oc3ccccc32)nc2c1SCC2 53000,c1(C(=O)NCC(C)(C2CC2)NC(c2ccnc(C3CC3)n2)=O)cc(F)cnc1O 53001,C1(C(=O)NCCc2ccn(C)n2)CCN(C(c2cn[nH]c2)=O)C(C)(C)C1 53002,CC1(C)CC(NC(C2COCC2C(F)F)=O)CN(C(c2ccon2)=O)C1 53003,Cc1cc(C(=O)Nc2nc(Cl)cc(Cl)n2)cc2nc[nH]c12 53004,c1(OC)ccccc1C1(C(=O)NC(C)CNC(=O)OC(C)(C)C)CCC1 53005,c1(CC)cc(CC(=O)NCC2CC(NC(=O)C(C)(C)C3CC3)C2)n(C)n1 53006,c1(C(N2C(C)(C3(C(=O)OC)CC3)CC(NC(C)=O)C2)=O)ccc(OC)c(F)c1N 53007,n1(CC(=O)NCCC(CC)(CC)NC(C(CC)C)=O)ccc(=O)c2ccccc12 53008,Cc1c(C(=O)NCC(C)CNC(C2(C(C)C)CCCO2)=O)cnc2ncnn12 53009,CC(C)(O)C#CC(=O)NC1CN(C(=O)CCNC(=O)C=CCl)CC1(C)C 53010,N1(C(C=C(C)C(F)F)=O)CCCCC(CNC(=O)Cc2nc(C(C)(C)C)cs2)C1 53011,Nc1cc(F)c(C(N2CC=CC(NC(=O)C3=CCCC3)C2)=O)c(F)c1 53012,CC1(C)CN(C(c2ccn(C3CCC3)n2)=O)C(CNC(=O)CNS(N)(=O)=O)CO1 53013,c1(C(=O)NC(CC)CN(C(=O)CCC(=O)N(C)C)CC)coc2c(F)cccc12 53014,CCCCC(CC(=O)NC(COC)CCO)NC(C1(C2(O)CCC2)CC1)=O 53015,C12(C(N3CC(NC(C4(C)CCO4)=O)C3)=O)CC3CC1(CO)CC3C2 53016,c1(C(=O)NCC2C3CN(C(CCC(N)=O)=O)C2CCC3)cc2cccc(F)c2o1 53017,c1(CC)n[nH]cc1C(=O)NCCCCCN(C)C(c1cn(CC)cn1)=O 53018,c1(OC)cc(C(N2CC(C)(NC(c3ccc[n+]([O-])c3)=O)C2)=O)ccc1Cl 53019,N1(C(c2cn(CC=C)nn2)=O)CCN(C(=O)C(n2cc(C)cn2)C)CC(O)C1 53020,c1(CC(=O)NCC(CC)NC(c2cc(O)cc(N)c2C)=O)ccc([N+](=O)[O-])cc1 53021,N1(C(C(C(C)C)NC(C)=O)=O)CCCN(C(c2sc(F)cc2Cl)=O)CC1 53022,c1(CCC)cccc(C(N2CC(NC(=O)C3=NOCC3)C(O)C2)=O)c1 53023,C1(O)(CNC(c2cnc(O)c(Cl)c2)=O)CCCN(C(c2ccnn2C2CC2)=O)C1 53024,Cc1cccc(Br)c1C(C(=O)NCc1c(C)n[nH]c1C)NC(c1csnn1)=O 53025,c1(C(C2CC(C)C23CCC3)=O)cc2c(cc1Cl)OCCO2 53026,Nc1cc(Cl)cc(F)c1C(N1CC(CNC(C2CC=CC2)=O)C2(CCC2)C1)=O 53027,c1(OC)ccc(CCC(=O)Nc2c(C)cccc2Cl)c(F)c1.C12CN(C1)C2=O 53028,CC(CCO)C(=O)N1CCC(CNC(c2ccc(Cl)cc2)=O)C1 53029,C=CCC(C(=O)NCC1CCN(C(c2ccn(C3CC3)c2C)=O)CC1)C(C)(C)C 53030,N1(C(C(=O)NCC)=O)CCC(NC(c2cn(CC(N)=O)nn2)=O)C(F)C1 53031,C1(NC(C(CC)C)=O)CC1C1CCCN(C(c2cnc(C#N)s2)=O)C1 53032,CCCC(CCC)CC(=O)N1CCC(O)C1C(=O)NCC(O)C1(Cl)CC1 53033,CCCC(C)CC(=O)N1CCC1(C)CC(=O)NCCC1CC(C)(C)C1 53034,c1(NC(C(CC)CC)c2nnnn2CCCSC)cc(C#N)cnc1C 53035,c1(C(C)NC(C2CC(C)CN2C(c2ccn(C(F)F)n2)=O)=O)cccc([N+](=O)[O-])c1 53036,C1(c2ccccc2)(NC(CC2CC(C)C2)=O)CC(NC(=O)C(C)CO)C1 53037,C1(C(=O)NC(c2cnc(C)s2)C)CC(O)CN1C(C1(C)CC(=O)C1)=O 53038,C1(NC(C(C=CC)O)=O)C(C)(C)C(NC(=O)Cc2cccs2)C1(C)C 53039,C=C(C)CCCC(=O)N.c1(NC(CC)=O)cc(OC)ccc1-c1nnc(C)o1 53040,c1(C(=O)NC2C(C)CCN(C(CCN(CC)CC)=O)C2)cc(N)c(F)cc1F 53041,S(=O)(=O)(c1ccc(NCC2CC2C)cc1Br)N1CCC(CCOC)CC1 53042,c1(C(=O)NC(CNC(C2CCCC2)=O)C2CC2)cncc(F)c1Cl 53043,N1(C(C(C=CC)O)=O)CC2(C1)CN(C(c1ccc(Cl)cc1C)=O)CC2CO 53044,N1(C(=O)NC(c2cc(C3CC3)no2)C)CC(C)OC2(CCOCC2)C1 53045,C1(C)(C(N(C)CC2CN(C(C3CCCC3)=O)CCO2)=O)CCCCNC1=O 53046,c1(-n2cc(C3(C)CN(C(Cc4scc(CC)n4)=O)C3)nn2)ccc(Cl)cc1 53047,c1(C(N(C)CCN(C)C(c2cc(C(N)=O)c[nH]2)=O)=O)cc(C(F)(F)F)n(C)n1 53048,CC1=C(C)CC(C)(NC(=O)C(C)CN(C)C(c2cc3ccncc3[nH]2)=O)CC1 53049,N1(C(CCCC=C)=O)CC2(CCN(C(C3CC3c3cscn3)=O)CC2)C1C(C)C 53050,Cc1cccc(C)c1C(C(=O)O)NC(c1nc(N(C)C)sc1Cl)=O 53051,C1(C(N(CC)CC2CCCN2C(=O)CP(C)(C)=O)=O)OCC2CCCC12 53052,c1(C(=O)OC)nc(C(=O)NCC2(NC(=O)C(CO)N(C)C)CCC2)co1 53053,C(=O)(C(O)CC(C)C)N1CC(N2CCN(C(c3c(C)nns3)=O)CC2)C1 53054,C=CC(C)(C)C(=O)N(CCC)CCNC(=O)CC1CC1C1CC1 53055,c1(C(=O)OC)cc(C(=O)NCC(O)CN(C)C(c2ccn(C)n2)=O)c(C)s1 53056,C=CCC(CC)C(=O)NCC1CN(C(c2csc(CCC)n2)=O)CC12CC2 53057,c1(C(=O)NC2CN(C(CCSCC(C)C)=O)CC23CC3)cc(S(N)(=O)=O)cn1C 53058,N1(C(c2nc(CNC(C3C(=C)C3)=O)oc2C)=O)CCCC2C1CCN2C 53059,C1(CN(C(C2CN(C(C)=O)C2)=O)CC)CCCCN1C(=O)CCC1CCCC(O)C1 53060,C1(C)(CCNC(CN(C(C)=O)C)=O)CCN(C(c2sccc2Cl)=O)C1 53061,C1(C(N(CC(COC)C)C)=O)CCN(C(C2C(C)(C)C2(C)C)=O)CC1O 53062,C1(CNC(c2nc(C)[nH]c2C(F)(F)F)=O)CC2CCC1N2C(=O)CSCC(N)=O 53063,c1(SC)nn(C)cc1C(=O)NCC1(O)CN(C(=O)C=C(C2CC2)C2CC2)C1 53064,C=CC(C)(O)CC(=O)NCCOC1CCN(C(=O)CCC2CCC(=O)NC2)CC1 53065,N1(C(C)=O)CC(C)(C)OC2(C1)CN(C(c1nn(-c3ccccc3F)cc1O)=O)C2 53066,C1(NC(C(CC)n2cccn2)=O)CCCCCN(C(=O)C=Cc2cnc[nH]2)C1 53067,Cc1ccc(F)c(C(=O)NCC2CC(C)N(C(=O)CSCc3ccncc3)C2)n1 53068,c1(CC)nc(C(N2CCC(O)(Cn3cc(-c4csnn4)nn3)C2)=O)c(C)o1 53069,c1(C(=O)NC2CCC(NC(C(c3cccs3)SC)=O)C2)cnc2nccn2c1 53070,C(CN=c1nc(N(C)CC2CC2(C)C)c2cc(Cl)ccc2[nH]1)(OCC)OC 53071,c1(C(=O)NC2(CO)CCN(Cc3c(F)cccc3Cl)CC2)nc2ccccn2n1 53072,N1(CC(N2CC(CNC(=O)Cc3ccsc3Br)C2)=O)CCCNC1=O 53073,N1(C(C(C)OC)=O)CCCCC2(C1)CN(C(=O)Cc1csc(S)n1)C2 53074,CCC(CC)C(F)C(=O)N1CCC(CC(N2CCCNC(=O)C2)=O)C1(C)C 53075,c1(OC)cc(C#N)ccc1C(N1CCC(C(F)(F)F)CC1)C(=O)NC(C)(C)C 53076,C1(CC(C)NC(C2N(CC)CC2)=O)CCN(C(=O)CCC2CCC(=O)C2)CC1 53077,C1(NCC2CCCN(C(C)(C)C)C2)CC(c2ccccc2[N+](=O)[O-])=NO1 53078,C(C(=O)NNC(=O)c1coc(-c2ccc(C)cc2)n1)NCC(F)F 53079,N1(C(c2c(C)cno2)=O)CC(NC(c2c(Cl)cncc2Cl)=O)CC(O)C1 53080,C(CC1CC1)(C(=O)NC1CCC(C(=O)NC2CC2)C1)NC(CNC(C1C(C)C1)=O)=O 53081,N(C1CCc2c(Cl)ccc(F)c21)CCCN1CCN(C(C)(C)C)CC1 53082,C1(NC(C=CSC)=O)CCCC(N(C)C(c2cc(N(C)C)ccn2)=O)C1 53083,C1(CC)C(C(=O)NCC2C3CCCOC23)CCN1C(=O)Cn1[nH]cnc1=N 53084,N1(C(C=CC(=O)OCC)=O)CCC2(C1)CN(C(C1(C)CCOC1)=O)CCO2 53085,c1(CC)nc(C)cc(=NC(CCN(C)C(C2CC3(CCOCC3)C2)=O)C(C)C)[nH]1 53086,C1(C(=O)Nc2c(OC)cccc2Cl)CCC(N=c2ccn3ncc(Br)c3[nH]2)CC1 53087,C1(CCC(=O)NCC(CC)N(C)C(C2CC(=O)N(C)C2)=O)CCCCN1C 53088,NS(=O)(=O)c1ccc(C(=O)Nc2ccsc2C(N2CCCC3(CCO3)C2)=O)cc1 53089,C1(C)(C(N2CCOCC(NC(CSCCC)=O)C2)=O)CCCNS1(=O)=O 53090,C(=O)(C1CCCc2scnc21)N1CC(O)CCC(NC(c2n[nH]c(C)c2C)=O)C1 53091,N1(C(CCOC(C)=O)=O)CCCC(N(CCO)C(C)=O)C1 53092,Cc1oc(Cl)nc1C(=O)NCCCCC1CN(C(=O)C(=O)NCC(F)(F)F)C1 53093,C1(C#N)(C(=O)NCC2CN(C(c3c(C)n(C)nn3)=O)C2)CCOCC1 53094,c1(C(CNC(c2c(C(N)=O)coc2)=O)O)c(F)cc(F)cc1F 53095,C1(CC)CN(C(=O)COCC2(F)CC2)CCC1NC(=O)CCc1ncc[nH]1 53096,CC(C)C(F)(F)CC(=O)NC1CCCC1NC(c1cc(Cl)cn1C)=O 53097,c1(COC)cnc(OC)c(C(N2CC(CNC(C3(C4CC4)CC3)=O)CC2C)=O)c1 53098,c1(OC)c(C(N2CCC(C(N3CC(O)C3)=O)C2)=O)cnn1-c1ccccc1 53099,Cc1nc(CCC(=O)NCCC2CCN(C(c3c[nH]nc3C(F)F)=O)C2)cs1 53100,c1(CCNCCN(C)C)ccc(OC2CCCO2)c(ON)c1.C1(C(=O)OC)(NC)CC1 53101,C1(NC(C(NOC)=O)=O)C2CCC1CN(C(=O)COc1cccc(C)c1)C2 53102,C1(CC(N2C(CCC=C)CCC2)=O)CCCCN1C(c1cnnn1CCOC)=O 53103,CC1CN(C(=O)C(C)(C)C(F)(F)F)CC(C)C1NC(=O)C(c1ccc(F)cc1)=O 53104,N1(C(C(C)NC=O)=O)CCC(CN(C)C(c2cc(CF)on2)=O)C1 53105,c1(C(N2C(C)CC(CNC(CC3CC(=C)C3)=O)C2)=O)ccc2nccn2n1 53106,n1(CC)ncc2c(N3CC(CNC(=O)CC(C)(C4CCC4)N(C)C)C3)ncnc12 53107,C1(CC(=O)N(C2CCN(C(COCCOCC#C)=O)C2)C)CCCN(C(C)C)C1 53108,N1(C(=O)OC(C)(C)C)CCC2CCN(C(C3CC3c3ncccc3Br)=O)C2C1 53109,C1(C2CCN(C(=O)C3CC3)CC2)(NC(CC2CC(C)C2)=O)CCC1 53110,C1(C(=O)NCC(CN(C(C2(CC=C)CC=CC2)=O)C)O)CC(F)(F)C1(C)C 53111,c1(CC(=O)NCCCCn2cc(Br)cn2)ccc(C(F)(F)F)c(F)c1 53112,c1(C(N2CCC=C(C=C)C2)C(=O)NCCC(=O)OCC)ccc(F)cc1Br 53113,c1(OC)cnc(C(N2CC=CC(C(N3CCC3C(=O)N(C)C)=O)C2)=O)cn1 53114,CC1(C)C(C(N2CC(O)(CNC(=O)C(F)=C3CCCC3)C2)=O)C1(F)F 53115,C1(NC(c2scc(OC)c2)=O)COCCN(C(=O)C(F)(F)c2cnccn2)C1 53116,C(=O)(C(O)C(C)CC)NCC(CC(C)C)NC(=O)C(C)NC(N)=O 53117,N1(C(c2ccc(CC)nc2)=O)CCCC(NC(c2cn[nH]c2)=O)C1C 53118,c1(N2CCC(CC=C)C2)nc(N(C)Cc2sccc2C)c2ncn(C)c2n1 53119,N1(C(C2=CCCC2C)=O)CCC(C(=O)NCC2CC3CCCC3C2)C12CCC2 53120,c1(C(=O)NC(C)C(C)NC(C2(CCO)CC2)=O)cnc(-c2ccccc2Cl)nc1 53121,N1(C(CCc2cn(C)nc2)=O)CCCC1(C)CNC(C1CC1c1ccco1)=O 53122,C#Cc1ccc(C(=O)N(CCC(=O)NCC2CC2C(N)=O)C)c(C)c1 53123,N1(C(C23C(C(=O)OC)(CCC2)C3)=O)CCCCC(NC(C2(C)CC(C)(C)C2)=O)C1 53124,c1(OC)c(C(=O)N(CC(C)C(=O)N2CC(N(C)CCO)C2)C)cnn1C 53125,C1(NC(CC2N(C(c3n(CC)ccc3)=O)CC(O)C2)=O)CCCCC1(C)O 53126,N1(C(=O)C=Cc2ncc[nH]2)CCCC2(CNC(C34CCN(CC3)C4)=O)CCCC12 53127,C(CCC(=O)NCC1CCCCC1)(C(C)C)NC(c1nccc(C)c1N)=O 53128,Cc1ccc2c(N(C3CNCC3F)C(c3ccc(Cl)cc3CO)=O)ncnc2c1 53129,c1(C(=O)NC(C(C)C)CCNC(=O)C(C)C2CCCO2)cccc2nc(CO)[nH]c12 53130,n1(CC)cc(C(=O)NCC(C)NC(=O)CCC2NC(=O)NC2=O)c2ccccc12 53131,c1(C(=O)Nc2c(C(=O)OC)cc(Br)cn2)cn2c(n1)CN(Cc1cc[nH]c1)CC2 53132,N1(C(CSCC)=O)CCc2ccccc2C(NC(=O)CC2(COC)CC2)C1 53133,c1(CNC(=O)CC2(O)CNC2)ccc(CNC(=O)C(c2ccccc2)F)cc1F 53134,CCC(C)(C(=O)NC(CCN(C(=O)CCn1ccccc1=O)C)C(C)C)C(F)F 53135,c1(C(C)NC(c2c(C#C)c[nH]n2)=O)cc2ccccc2n1C 53136,C1(CC(=O)NCC2CN(C(C(OC)OC)=O)C(C)(C)C2)NC(=O)CN(C)C1=O 53137,C1(F)(CNC(C(CCC)=CCC)=O)CCCN(C(C2CNC(=O)CC2C)=O)CC1 53138,c1(N2CCC(CCC)C2)nc2ccccc2c(=NCC(F)(F)Br)[nH]1 53139,C1(C(=O)NCCOC2CCN(C(c3cc(CO)on3)=O)C2)CCc2nc[nH]c2C1 53140,N1(C(CCC=C)=O)CCC2CCCN(C(=O)CSCc3ccccc3)C2C1 53141,Cn1cc(C2CC(C(N3CCC(N4CCOC4=O)CC3)=O)C2)c(C2CC2)n1 53142,N1(C(CSS(C)(=O)=O)=O)CCCOC(CNC(=O)CC2CCCCO2)C1 53143,N1(C(c2c(CC)con2)=O)CC2CC1CC2NC(c1cc(C(=O)OC)co1)=O 53144,c1(C(C)N2C3(CCC3)CC2=O)cc2ccccc2o1.C1(O)(COC)CCCCC1 53145,Cn1cc(C(=O)NCC23CC2CN(C(c2cc(CC4CC4)on2)=O)C3)c(O)nc1=O 53146,N1(C(c2cc(C)nn2C)=O)CCn2c(C(N3CCN(C)CC3)=O)cnc2C1C 53147,C(=O)(C=C1SCC(=O)N1C)NC1(C)CCN(C(C(C)OC2CCCCC2)=O)C1 53148,c1(COC)ccc(C(=O)NCC2CCC2NC(=O)C(C)(C2CC2)NC(C)=O)o1 53149,c1(-c2c(CNC(c3sccc3C3CC3)=O)occ2)ccc(Cl)cc1 53150,c1(C(=O)NCC2(CNC(CCN(C(CCC)C)C)=O)CC2)csc(Cl)c1Cl 53151,c1(CC(C)C)ccc(C(C)C(=O)NCCCCNC(C2CCOC(=O)N2)=O)cc1 53152,Cc1cc(=NC(=O)Cc2csc(=NCc3ccc(I)c(O)c3)[nH]2)[nH][nH]1 53153,N1(C(C2(CC)CN(C(C3(C)CCCCC3)=O)C2)=O)CCCC(C)(COC(C)=O)CC1 53154,c1(C(N2CCC(NC(C3CCCC34CC4)=O)(CF)C2)=O)cc2ccccc2cn1 53155,c1(NC(CC=CCNC(C2CC(=O)NCC2)=O)=O)cccc2c1CCO2 53156,C1(NC(C(CNC(C(C)NC(C)=O)=O)CC2CCCC2)=O)CCCCCCC1O 53157,C1(C(=O)OC(C)(C)C)(NC(C2CCC(C3CC3)C2)=O)CC2(CCCCC2)C1 53158,CC(CCN(C)C)C(=O)N1CCC(N(C(=O)CN(CC(C)(C)C)C)C)C1 53159,C(C)(C)(CC(=O)N1CCC(c2cnco2)C1)N(C(COC(C)=O)=O)C 53160,c1(C(=O)NC(CC(C)NC(C2C(CCC)C2)=O)C)cc(S(N)(=O)=O)cc(F)c1C 53161,C1(NC(C2(C#C)CN(C(=O)C(C)C#N)C2)=O)CCOCC12CCC2 53162,C1(C(=O)NCCC(CNC(c2cnc(C(C)C)s2)=O)O)CCC(=O)N(C)C1 53163,N1(C(c2cn(CC)nc2)=O)CCC(C(=O)NCCCC2CCCCC2)C12CCC2 53164,N1(C(c2c(CC)c[nH]c2)=O)CC(C)N(C(=O)C=CC(=O)NC2CC2)CC1C 53165,c1(C(=O)OC)ccc(C(=O)NC2CN(c3ncc(F)cn3)C2)cc1C 53166,N1(c2cc(OC)ncn2)CCC2CC(CNC(c3ccc[nH]3)=O)CCC2C1 53167,O=C1CC2CC(C(=O)NCc3cc(C(N4CCCC4C4CCCC4)=O)no3)C1O2 53168,CC1CN(C(=O)CC(C)CNC(=O)C(C)(C)C(C)(C)C)Cc2c[nH]nc21 53169,CCCC(C)CC(=O)N1CCCC(N(C)C(c2ccc(CC3CC3)cc2)=O)C1 53170,Cn1cc(C#N)cc1C(N1CCCC(n2cc(C3CCCN3C)nn2)C1)=O 53171,c1(C(N2CC(COC)(CNC(=O)C(F)(F)C3CCCC3)C2)=O)ccnc(C)c1O 53172,C1(NC(C(C)n2ccnn2)=O)CCC(C)(NC(C2COCCOC2)=O)CC1 53173,C1(CC)CCN(C(=O)C(F)F)C(C(=O)NCC2(C)CCCOC2)C1 53174,N1(C(c2c(C)ocn2)=O)CCN(C(=O)CNC(c2ncn(C)n2)=O)CC1 53175,c1(CC)cc(NC2CC(NC(=O)CCC(C)C)C2(C)C)ncn1 53176,C(=O)(C(O)C(F)(F)F)N1CC(OCC)C(CNC(=O)CC)C1 53177,c1(C(N2C(CNC(=O)C(O)C3CC3)CC(O)C2)=O)cnn2c1OCCC2 53178,C1(C(=O)OCC2N(CCC(C)C)CCC2)CCN(C(C2CCCO2)=O)CC1 53179,N1(C(c2cnc(CCC)s2)=O)CCCC(N(C)C(c2ccn(C(C)C)n2)=O)CC1 53180,C12(C(N(CCNC(c3cc(C)oc3C)=O)C3CC3)=O)C3C4C1C1C2C3C41CO 53181,N1(C(C(C)C2CCCC2)=O)CC2CCC1C2NC(c1ccc(Cl)c(O)c1)=O 53182,Cc1ccc(C=CC(=O)NC2CCN(C(C3CS(=O)(=O)CCO3)=O)CC2F)nc1 53183,N1(C(=O)NC2CCC2CC(F)(F)F)CCC(OCC2CC2)C1 53184,C=CCCCCNC(=O)C(O)C1CN(C(=O)C(n2ccnc2C)C)C1 53185,Cc1c(CC(=O)NCCCNC(=O)CC2C=CCC2)cccc1[N+](=O)[O-] 53186,c1(CC)cc(C(=O)NCC(C(C)C)NC(=O)C(C2CCC2)OC)ncn1 53187,CC12CCN(C1)C2=O.C1(OCC(=O)NCC(F)(F)F)CC(=O)N1 53188,C1(OC)CC2(C1)CC(C(=O)NC1CC3CC1CC3CO)C2.C12(CC1)C(=O)N2 53189,C1(NC(C2CCN(C(c3cn(CCC)nc3)=O)C2)=O)CCN(C)CC1C#N 53190,C1(C(=O)NC(C)CC2CCOCC2)CCC(C)N1C(=O)CC1CC1C1CC1 53191,C(CCN=c1[nH]c(N2CCOC(CF)C2)nc2c1SCC2)OCC(C)C 53192,c1(CNC(C2CC(O)CN2C(c2nccnc2Br)=O)=O)ccc2cc[nH]c2c1 53193,Cc1cccc(C(=O)NCC2CCCC2NC(C2(O)CCC(C)CC2)=O)c1N 53194,N12CC(C3(CCN(C(=O)CCC)CC3)C1)C2C(=O)NCCCC.C(C)(=O)OC 53195,C1(NC(C2C(C)CCC2)=O)(CNC(C2CC(F)(F)C2)=O)CCOCC1 53196,C1(CNC(C2CN(C(=O)CO)CCO2)=O)COc2ccccc2O1 53197,C(c1cccnc1)=CC(=O)NCC(CCOC)NC(=O)CCc1cnn(C)c1 53198,C1(CC(C)NC(c2cn(C3CCOC3)nn2)=O)CCN(C(=O)CSC(F)F)CC1 53199,C1(C(=O)NCC(C)CC2CC2)CCC2CCC1N2C(=O)Cn1cnnc1O 53200,N1(C(c2c(CCC)nns2)=O)CCN(C(=O)C(C)OC2CCCCC2)CC1CF 53201,CC(CC(=O)NOC(c1ccccc1)CNC(=O)C(F)(F)CO)C1CCCC1 53202,C(=O)(CC(C(F)(F)F)OC)N1CC(F)(CNC(CC2(CC=C)CCCC2)=O)C1 53203,N1(C(C2(CC#C)CCCCO2)=O)CCC(Nc2ncnc(=N)[nH]2)C(F)(F)CC1 53204,C(=O)(C1=CC2CCCC12)N(C1CCN(C(c2c(O)cccc2O)=O)C1)CC 53205,N1(C(C(CCF)NC(C(CC=CC)C)=O)=O)CCCNC(=O)C1 53206,C1(NC(C2CC3CC2C2CC32)=O)CCC2CN(C(=O)C=Cc3cscn3)CC2C1 53207,N1(C(C(CC2CCC2)NC(Cc2cccc(C#C)c2)=O)=O)CC(F)(F)CCC1C 53208,c1(OCCC)ccc(C(C)NC(=O)OC2CC2(F)F)cc1OO.OC 53209,Cc1sc2ncnc(N3CCC4CCC(C3)N4C(=O)C(C(C)C)N(C)C)c2c1C 53210,c1(C(N2CCC(CNC(CC(C)OC)=O)CC2)=O)ccc2c(c1)CC(C)(C)C2 53211,c1(CNC(=O)CCN2CCOC2=O)ccc(-c2ccccn2)cn1 53212,Cn1cc2c(n1)CCCC2C(=O)NCC(C)(O)CNC(=O)CCC1CCCCC1 53213,N1(C(c2cnn(CC)n2)=O)CCCC(NC(c2ccnc(Cl)c2O)=O)C1C 53214,C#CC1(CC)COCCN1C(c1nc(CO)cs1)C(=O)NC1CC(F)(F)C1 53215,C1(C(N2CCSCC2C2CC2)C(=O)NC2(C)CC2)CCOC2(CCOCC2)C1 53216,N1(C(CC(CC)O)=O)CC(C)CN(C(c2cc(F)n(C)n2)=O)CC1C 53217,Cc1c[nH]c(=NCCC2CCCN(C(c3ccnc4ccnn34)=O)C2)nc1O 53218,C1(C(=O)NCC(CN(C(=O)C(C)(C)N2CCCC2)C)(C)C)CCCCC1C(N)=O 53219,c1(CN(C(C(=O)N(C)C)=O)C)ccc(CNC(C2C3CCC2CC3)=O)cc1 53220,CC1CN(C(C2CC(O)(c3cccnc3)C2)=O)CCCN1CC1CCCCC1O 53221,Cc1sc(O)nc1C(N1CCCC(NC(c2cnc(Br)s2)=O)C1)=O 53222,C(=O)(CCCCC(N)=O)NC(C(N1C(CSC)CCC1)=O)Cn1cccn1 53223,N1(C(C2CC(C)(C)C2)=O)CC2CCCC(NC(c3nc(Cl)c(Cl)s3)=O)C2C1 53224,C1(C(N(CCN(C)C(c2cccc(=O)o2)=O)C)=O)CC(C)(C)OC1(C)C 53225,C(=O)(C(C)(C)S(C)(=O)=O)NC1CN(C(c2c(OC)c(F)ccc2)=O)CC(C)C1 53226,CC(C)CCC(=O)NCCNC(C1(N(C)C)CC1)=O.C12CC1CN2 53227,C1(C#N)(C(=O)NCC(C)(C)NC(C2CCCN(CC(F)(F)F)C2)=O)CC12CCC2 53228,N1(C(=O)COc2cccc(CO)c2)CCN(C(=O)CN2CCCCC2)C2CC12 53229,C1(C(=O)NC2CC(N(C(CC(C)C)=O)C)C2)CC(C)CC(C)(C)C1 53230,N#Cc1ccc(=NCC(=O)N2CCC3(CC2)CC(NC(=O)C2=CCCS2)C3)[nH]c1 53231,C(CN=C(NCc1cc(Cl)ccc1Br)N1CCC(C2CCOC2)C1)N(CC)CC 53232,N1(C(c2c(C)cc(C(=O)OC)o2)=O)CCC2(C1)CN(C(c1ccn(C(F)F)n1)=O)C2 53233,c1(CC(N2CCCC(N(C(=O)CC(C)(C)F)C)C2)=O)noc2ccc(O)cc12 53234,Nc1c(C(N2CC(O)CC2C(=O)NCc2ccc(Cl)o2)=O)cccc1F 53235,C1(C(=O)NCC(CNC(C2(COCC)CC2CC)=O)(C)C)(OC)CS(=O)(=O)C1 53236,c1(CC)cc(N)c(C(N2CCCCC2C2CC2)=O)cc1F 53237,c1(C(=O)NCC2(O)CN(C(C(CC)C(C)O)=O)C2)cnc2c(F)cccn12 53238,CC1(C)CCCCC1CS(=O)Cc1nc(C2CCCCCCC2)no1 53239,c1(OC)ccc(CC(=O)NC2(C)CCN(C(C34CCC(OC)C3C4)=O)C2)cc1Cl 53240,C1(C(N(C2CCN(C(=O)Cn3nnc(C)n3)CC2)CCC)=O)CN(C)CCO1 53241,c1(NC(=O)NCC23OC(C)C(CC2)C3)cc2ccccc2s1 53242,c1(CC)ncc(C(=O)NCCC2COCCN2C(=O)C(O)CCN(C)C)c(O)n1 53243,Cc1nc(N2CC(NCc3ccccc3Br)C3(CC3)C2)c2c[nH]nc2n1 53244,C1(NC(C=CC=CC)=O)CS(=O)(=O)CC1NC(C1(S(C)(=O)=O)CC1)=O 53245,C1(C(N(c2cccc(O)c2)CC)=O)CCC2CCC1N2C(=O)C(O)CC(C)C 53246,C1(C(N(C2CSC2)CCC)=O)CCN(C(=O)C(CC)N(C)C)O1 53247,C(=O)(C(CC(F)F)NC(=O)CSc1cn[nH]c1)NC1CC(C(=O)OC)C1 53248,CCCCC(=O)C(=O)N1CC(C)CC1C(N1CCCC(CN(C)C)C1)=O 53249,C1(C(N(C)CC2CCCN2C(c2ccc(Cl)o2)=O)=O)CC2CC1C1CC21 53250,C1(CNC(=O)COC(F)(F)F)COCC2(CCN(C(=O)CCc3ccoc3)C2)O1 53251,CCCCCC(=O)N1CCC(F)(CNC(=O)C(C(C)C)c2cnn(C)c2)C1 53252,C(=O)(C1CCCc2cn(C)nc21)NCCC(C)NC(c1cccc(O)n1)=O 53253,C1(C2CCN(C(c3cncc(Cl)c3)=O)C2)(NC(C(Cc2c(C)nc[nH]2)O)=O)CC1 53254,C(=O)(CCC(C)S(C)(=O)=O)NC12CC(NC(C3N(CCC)CCC3)=O)(C1)C2 53255,C1(CNC(c2n(C)cnc2)=O)CCC(F)(CNC(C2(C)CCCNC2=O)=O)CC1 53256,N1(C(C(CCC)C(C)C)=O)CCC2(CC1)COC(CNC(c1cscn1)=O)C2 53257,c1(OCC)cc(CCCNC(N2CCCC23CC3)=O)cc(F)c1F 53258,CC(C)CCC(O)C(=O)NC1CCN(C(=O)C2=COCC2)CC(O)C1 53259,N1(C(c2c(C)scc2)=O)CCCC2(NC(=O)Cc3ccccc3[N+](=O)[O-])CC2C1 53260,Cc1oc(Br)cc1C(=O)NC1CC(C)(CNC(C2(C)CNC(=O)C2)=O)C1 53261,N1(C(C=COCC)=O)CCOCC1CN(C(C1(C)CC1c1ccccc1)=O)CC 53262,Cc1c(F)ccc(C(N2CCOCC2)C(=O)N(C2CC2)Cc2ccccc2)c1Cl 53263,c1(C(N(CC(CC)NC(=O)CCCF)C)=O)cc(C)nc2c(F)cccc12 53264,C1(CC(N2CCCC(C)C2CNC(=O)C=C2CCCC2)=O)Cc2ccccc2N1 53265,N1(C(C2CCN(C)CC2)=O)CC2CCC(C1)N2Cc1ccncc1C(F)(F)F 53266,C1(C(=O)NC2(CC=C)CN(C(C3(COC)CC3)=O)C2)CC2CCC1C2 53267,N12CCOCC1Cc1ccc(o1)C2C.C(=O)(CC=CC(C)(C)C)OC.C1CS1 53268,Cc1coc(C)c1C(=O)NCC(C)CN(C(=O)CSCc1csc(=N)[nH]1)C 53269,n1(C(=O)NCC2CCCN2Cc2c[nH]c3ncccc23)c(=O)oc2ccccc12 53270,CCC(O)C(C)C(=O)NCC(C)(C(C)C)NC(=O)Cc1ccc(Cl)cc1 53271,c1(CC)nccnc1CNC(=O)C(C)(CSC)NC(=O)C=CC1(C)COC1 53272,Cc1cn2c(n1)C(C)CC(C(N1CC3(CC(NC(=O)Cn4ncnn4)C3)C1)=O)C2 53273,N1(C(C(CC=C)CNC(=O)C=Cc2cncn2C)=O)CC2CCC(CC2)C1 53274,c1(C(N2CCC(C)(NC(c3n(C)c(S)nc3)=O)C2)=O)nc2c(s1)COCC2 53275,C(=O)(CCC(F)(F)CN=[N+]=[N-])NC1CC(C)(CNC(C=CCOCCOC)=O)C1 53276,CC1(C)OC(C(=O)NCC(CO)NC(c2conc2C2CCC2)=O)C(C)(C)O1 53277,C(=O)(CC1CCCc2ccccc21)NC1CC(CNC(C2(C)CC=CCC2)=O)C1 53278,C(=O)(C1=COCCC1)NCC1CCN(C(C(C(C)C)OCC(C)C)=O)C1 53279,N1(C(C(CC)=CC)=O)CC(NC(=O)CC(C)n2ccc(C)n2)C(C)C1 53280,n1(CC(N2CC(SC)C(NC(=O)C(F)CCC(C)C)C2)=O)nc2c(n1)CCCC2 53281,CN1CCCC1(C)CNC(=O)Nc1nc(-c2ccncc2)cs1 53282,C1(OC)CC(N2CCN(C3CC(OC)C(C(=O)OC)C3)CC2)C12CCOCC2.CCS 53283,C(=O)(C1=CCCN(C(c2ncccc2F)=O)C1)NC(c1ccc(O)nc1)C 53284,C1(C(=O)NC(c2ncc[nH]2)CC)CN(C(=O)C(c2ccn(C)n2)C)CC12CCC2 53285,c1(OC)cc(NC(=O)C(C)N(C(=O)CC(C)n2ccnc2)C)ccc1F 53286,c1(C(N(C)CCOCCNC(C2COCC2c2ccccc2)=O)=O)cn(C)c(O)n1 53287,N1(C(C(C(C)C)NC=O)=O)CC2CN(C(=O)C=CC3COC(C)(C)O3)CC2C1 53288,c1(N(CCC)CCNC(=O)CC2=NNC(=O)C2)cnc2cc(F)c(F)cc2n1 53289,n1(C(C(=O)N(CC(C)C)C(C)C2CC2)C)cc(C(C)N(C)C)nn1 53290,C1(OCC)CCN(c2nnc(Cc3ccccc3Cl)n2CC2CC=CCO2)CC1 53291,C#CCC(C)(C)C(=O)N1CC(C(=O)NCC(CC)C(C)(F)F)C(CCC)C1 53292,CC1=NN(C)C(=O)C1CC(=O)NCC1CC1CNC(=O)COCC1CC1 53293,C1(C(N(C(C)CNC(=O)CC2COCCO2)C)=O)CCCCN1C 53294,N1(C(C(C2CC2)OCC)=O)CCC(CN(C)C(C2C(C(F)F)C2(C)C)=O)CC1 53295,C1(NCc2ccc(C(=O)O)cc2)CC2(C1)CC(NC(=O)Nc1cccnc1)C2 53296,c1(OCC)ccc(C(N2CCN(C(=O)CSC)CC2)C(=O)NCCC(C)O)nc1 53297,C1(C(N(C(C)CNC(=O)Cn2ccnn2)C)=O)CCCC(=O)C1 53298,c1(C(=O)OC)cc(C(=O)NC2CCC2NC(=O)COC2CC=CC2)ccc1F 53299,N1(C(CC(CC)CN(C)C)=O)CCCC2(CCCN2C(=O)C2=C(Cl)CCCC2)C1 53300,c1(NC(C2CCN(C(CCN(C)CC)=O)C2C)=O)cc(C)cnc1O 53301,C1(CC)CC(C(=O)NC2CN(C(=O)Cc3ccc(C)cc3)CC2C)CCO1 53302,CC#CCCC(=O)NC(CC1CC1)C(=O)NCCN1CCCC1C 53303,c1(C(N(CCNC(c2cnc(Cl)s2)=O)CC2CC2)=O)nnc2ccccc2n1 53304,N1(C(C(N2CC(C)C2)C)=O)CCCCC1CC(=O)NCc1cnc[nH]1 53305,Cc1cc2c(C(=O)NC3CC3C3CCCN(C(c4cnn[nH]4)=O)C3)cccc2o1 53306,N1(C(CC2N(C(c3c(C)nc(C)[nH]3)=O)CCC2)=O)CC=C(c2ccccc2)CC1 53307,C(=O)(C1=C(C)OCCC1)NC1C(NC(c2nc(OC)c(F)cn2)=O)CCC1 53308,c1(C(N(C2CCCC(C(=O)NC3CCCCC3)C2)C)=O)cncc(N(C)C)c1 53309,Cc1ccnc2c(C(N3CCOCC3CN(C)C(C3CC3C)=O)=O)cccc12 53310,c1(NC(c2ccccc2C(F)(F)F)=O)ccc(O)c(=O)cc1 53311,CC1=CCC(C(=O)NCCCC2CCCCN2C(=O)C(F)=CC2CC2)CC1 53312,N1(C(C2=NOC(C)C2)=O)C2CCC1CC(NC(=O)Cc1ccc([N+](=O)[O-])cc1)C2 53313,c1(CC)ccc(Cn2nccc2NC(C2ON=C(C)C2C)=O)cc1 53314,C1(C(N(CCCOC)CCO)=O)CCC(C)(C)N(C(=O)C(CO)C(F)(F)F)C1 53315,N1(C(C(COC)N(C)C)=O)CCCCC1C(=O)Nc1cccc(C)n1 53316,Cc1cc(C(=O)NCC2CC2CC(=O)NCc2[nH]ccc(=O)c2O)ccc1F 53317,C1(NC(C(CC)N(C)C)=O)CCC12CCN(C(c1oc(SC)cc1C)=O)CC2 53318,N1(C(C2N(C(C(c3ccc(OC)cc3)C)=O)CC=C2)=O)CCCC2(COC2)C1 53319,N1(C(C(=O)NCCC)CC2CC2(Cl)Cl)CCOCC1(C)Cc1ccccc1 53320,C1(C(C)C)CN(C(=O)CN2CCC(F)CC2)CC1C(=O)N(C1CC1)C(C)C1CC1 53321,c1(C(=O)NC(C(CO)NC(C(CC#C)O)=O)C)nn(C)c2c1CS(=O)(=O)CC2 53322,C1(C(=O)Nc2nc(C)ncc2Br)(OC)CCN(C(C2CC2F)=O)CC1 53323,N1(C(C2C(C(C)=O)C2(C)C)=O)CCN(C(=O)C(CO)N(C)C)C(CO)C1 53324,C1(N(C(C(C)N(C)C)=O)C)CCN(C(=O)CCc2ccc[nH]2)C1.C1(C)CCCO1 53325,C1(NC(c2cccnc2)=O)(CO)CCN(C(=O)CNCc2ccc(C3CC3)o2)C1 53326,c1(COCC)cn(CCCC(=O)NCc2ccsc2C(=O)O)nn1 53327,C(C(CC(=O)NCCC1CCC(C)(C)O1)NC(=O)C(O)CCSC)OC 53328,N1(C(C(C)OCC2CCCCO2)=O)CC2CN(C(C3CCC4(C3)N=N4)=O)CC2C1 53329,C(=O)(CCC(C)NC(=O)C(C1CCN(C(=O)CN2CCC(OC)C2)C1)C)OC 53330,c1(CC(N2CCCC(C)(OC)CC2)=O)ccc2c(c1)CC(C)O2 53331,C(=O)(CCP(C)(C)=O)N(CCCCNC(C(c1ccccc1Cl)C)=O)C 53332,CC1CCC2(CC1)CCN2C(=O)CCCCCCn1cc(-c2ccc(Cl)cc2)nn1 53333,C(C(=O)N1CCN(C(C2CCCCN2CC(F)F)=O)CC1C)(C(C)(C)C)SC 53334,Cn1ccc(C(=O)NCC2CCCN(C(C3(C(F)F)CC3(F)F)=O)C2)cc1=O 53335,c1(C(C)(C(=O)NCC(CNC(=O)CCCC2CC2)CO)N(C)C)ccc(F)cc1 53336,N1(C(c2cc(N)c(Cl)cn2)=O)CCOC2CN(C(=O)CC3C=CCC3)CC12 53337,C(C(CCO)NC(C1=NOCC1)c1nnnn1CCCOC)OC 53338,n1(CC2CC(=O)C2)cc(C(=O)NCC2CC2NC(c2cc(C(F)F)c[nH]2)=O)cn1 53339,N1(C(CCC2(C#N)CC2)C(=O)NCCC2CC2)CCC(S(=O)(=O)C(F)F)C1 53340,C1(C(=O)NC2C(C(N3C(C(=O)OC)CCC3)=O)CCC2)CC2C=CC1C2 53341,N1(C(C2(CC(C)C)CC2)=O)CC2ON=C(CNC(c3cn(C(C)C)nn3)=O)C2C1 53342,c1(C(=O)NCC2C(NC(c3cnc4[nH]cncc3-4)=O)C2)ccc(Cl)c(F)c1F 53343,N1(C(C=CCCC)=O)CC2CC(C(N3CCC(CO)C(C)C3)=O)C(C2)C1 53344,Cc1ccccc1C=CC(=O)NC1CC2(C1)CC2NC(C1CCC(=O)N1C)=O 53345,N1(C(CC(CC)(C)C)=O)CC2CC(CNC(=O)C(C)(C)SC)CC1C2 53346,CCC(CC(=O)NC(C)CCCNC(c1nc(C(C)C)oc1C)=O)C1CC1 53347,c1(C(CC)C)ccccc1OCC(=O)NCc1ccn(C(C)CC)n1 53348,C(=O)(C(O)CC(F)(F)F)NCCCOCCC(=O)NCCCOCCN1CCCC1 53349,Cc1cc(Oc2ccccc2)c(CC(=O)NNC(=O)c2cc(C)oc2C)cc1Cl 53350,C1CCC2C(N3CCC(OCC4CCCO4)C3)C2CC1 53351,CCC(CC)N(CCOC)C(=O)NC1CC1C1CCCO1 53352,C1(C(N2CC(OCCOC)C2)=O)CCC(CNC(=O)CCCF)O1 53353,C1(CN(C(CC(CC)C2CCC2)=O)C)CCCN(C)C1c1ccnn1C 53354,N1(C(C2CNC(=O)N2)=O)CC(NC(c2ccoc2Br)=O)C2(CCC2)C1 53355,c1(C(=O)NCC(CNC(CC(C)O)=O)F)c(Br)ccc2n[nH]cc12 53356,C1(C(=O)NCC(C2CCC2)OCC)(CO)CCN(C(C2CCN(C)C2)=O)C1 53357,N1(C(C2C3CN(C(C4C(OC)CCCC4)=O)CC32)=O)CC2CC2C2CC12 53358,c1(C(=O)NCCCN(C)C(c2cnc3ccoc3c2)=O)cncc(P(C)(C)=O)c1 53359,C(C1=NOC2CCCC12)NC(=O)NCC(=O)NCC1(CS(N)(=O)=O)CC1 53360,C1(O)(CC(N2CC(CCNC(=O)C(O)c3ccco3)C2)=O)CCCOC1 53361,c1(NCC2C3CN(C(CC4CCN(C)CC4)=O)CC32)cncc(C#N)n1 53362,c1(CNC(N2CC(C)(C#N)C2)=O)ccc(N=[N+]=[N-])cc1 53363,C1(C(C(=O)NC)N(c2ccc(OC)c(Br)c2)C)CCC2COCCC2C1 53364,c1(C(N(CC(CC)NC(C2(CF)CCC2)=O)CC)=O)ncn2ccc(C)cc12 53365,CCC(C)CCC(O)CC(=O)N1CCCC1C1CCN(C(=O)CCCNC(C)=O)C1 53366,C1(CNC(C2C(C(N)=O)C2)=O)C2CC1N(C(C1CCCC1F)=O)C2 53367,c1(C(=O)NC2C(CNC(Cc3n(C)nc(CC)c3Cl)=O)C2)nc2c(s1)COCC2 53368,C1(CNC(=O)CCNC(=O)C2CC2)C2CN(C(C3CC(n4cncn4)C3)=O)CC12 53369,c12cc3sc(cc3o1)NC2=O.C1CC12CC2.N(CCNC(=O)OC1CC1)(CC)C 53370,CCC(F)(F)CC(=O)NC(C)(CNC(c1ccc(C)cc1F)=O)C1CC1 53371,c1(CC(=O)NCC2=CCN(C(CCSC)=O)CC2)ccc(S(=O)(=O)C(F)F)cc1 53372,c1(CN2CCN(CC(=O)NC(c3ccc(CC)cc3)CC)CC2)cc(Br)ccc1Cl 53373,C(=O)(CC(N)C(=O)NCCC(C1CCC(O)C1O)=O)OC 53374,N#Cc1ccc(C(=O)Nc2cccc(NC(=O)CC3CC4CC4C3)c2)cn1 53375,c1(C2CN(NC(C3C(C)(C)C3)=O)C2)ocnc1-c1cn(CCC=CCO)nn1 53376,CC1(C#CC(=O)N2CCCc3ncccc32)CN(C(C)(C)C)C1 53377,c1(C(=O)NC2CC(N(C)C(C3CCCCCC3)=O)C2)cc(F)c(F)c(Cl)c1F 53378,N1(C(C2(CC)CCOC2)=O)CCCN(Cc2nncn2C)CC1 53379,n1(CC)ccnc1C=CC(N1CCOC(CCNC(C2CCS2(=O)=O)=O)C1)=O 53380,C(=O)(C(F)C1=CCCCC1)NCC(C1CCCC1)NC(c1c(CC)n[nH]c1)=O 53381,c1(CNC(CSC)=O)cc(C(=O)NC(C)CC(N)=O)no1 53382,N1(C(C(C)SCC)=O)CCCC(C)(CNC(=O)CCc2cc(C)nc(C)c2)C1 53383,C1(OC)CN(C(=O)CS(C)(=O)=O)CC1C(N1CC(c2cc(O)n[nH]2)C1)=O 53384,C1(NC(C(C=C)C)=O)CCCCC1CC(N1CCC1C1CCC1)=O 53385,c1(CNC(=O)Cc2ccon2)nc2c(s1)CN(C(=O)C(O)(C1CC1)C1CC1)CC2 53386,CC(C)CCC(O)C(=O)NC(Cc1ccoc1)C(=O)NCC1CC(C)(O)C1 53387,c1(C(=O)NC(CNC(C2(C)CC2C(F)(F)F)=O)C2CC2)cncc2sccc12 53388,O=C(N=S(=O)(c1ccccc1)C(F)F)c1ccc(OC2CC2)cn1 53389,N1(C(c2ccc(NC)cn2)C(=O)NC2CCOCC2)CCC(C)C(C)C1 53390,c1(CN(CC(C)(C)SC)C)c[nH]c2cccc(Br)c12 53391,c1(CC(=O)NC2CC(C)(NC(C(C3CCC(=O)N3)C)=O)C2)csc(Br)c1 53392,C1(CNC(C(c2cncnc2)C)=O)CC2CCC1N2C(c1ncccc1Cl)=O 53393,C(C(C)(C)CC(=O)NCCN(C)CCF)NC(c1c(C)oc(COC)c1)=O 53394,CCCC(C)(C)CC(=O)N1CCC(NC(=O)C(C)(C)CC(F)F)C(C)C1 53395,c1(C(N2CCN(C)CC2CNC(c2ccnnc2O)=O)=O)cc2c(o1)CCCC2 53396,C1(NC(c2cc(N)sc2)=O)CC2(NC(c3cc(-c4ccco4)no3)=O)COC1C2 53397,CON=C(C(=O)N(C(CNC(=O)C(C)(C)C1CCCO1)C1CC1)C)c1ccco1 53398,N1(C(C2CCCCN(C(CC3CC(OCC)C3)=O)C2)=O)CCC2(CC1)CC(O)C2 53399,c1(C(N2CC3CCCC23)C(=O)NC(C(=O)OC)C)ccc2c(c1)ncn2C 53400,N1(C(C(C2CCN(C(CS(CC)=O)=O)CC2)C)=O)CCc2nn[nH]c2C1 53401,c1(NC)cccc(C(N2CC(F)CC2CNC(c2cnn(C(C)C)c2)=O)=O)n1 53402,N1(C(c2c(CC)nc(C)o2)=O)CC(NC(=O)C(C(C)C)C2CCC2)CC(F)C1 53403,c1(C(=O)NC(C)(C)CF)n[nH]c2c1CN(C(C1(C)CCC(=O)N1)=O)C2 53404,c1(C(=O)NC(CN(C(CCCOCCC)=O)CC)CC)cc(Cl)ccn1 53405,c1(C(C(=O)NCCCN(C(C23CCC(CC2)O3)=O)CC)=O)cc(F)cc(Cl)c1 53406,N1(C(c2c(C)n(CCO)cc2)=O)CCC(NC(c2cc(C3CC3)no2)=O)C12CC2 53407,C1(NC(C(CSC)O)=O)CCCC(C(=O)N(C2C3CCCC23)C)CC1 53408,N1(C(CC(CC)O)=O)CCC(C2CC2)C1C(=O)NCCC(=O)N(C)C 53409,c1(OC)ccc(CC(=O)NC(C)(C)CNC(c2cc(CN(C)C)on2)=O)c(C)c1 53410,c1(C(=O)NCC(CC)(C)NC(C2CC2F)=O)ccc(F)cc1OC 53411,C1(NC(C2(C(=O)OC)CC2)=O)CC(NC(=O)Cc2c(F)cncc2Cl)C12CCC2 53412,C=CC(C)C(=O)N(CCC(=O)NC(C1CCC1)C)C 53413,C1(C(=O)NCc2cn(C3CCN(C(CC)=O)CC3)nn2)CCS(=O)(=O)C1(C)C 53414,N1(C(C(C)(C)CC2CC2)=O)CCC2(CCN(C(c3csc(CO)n3)=O)C2)C1 53415,Cn1ncc(CNC(=O)CC23CCCC2C3)c1C(=O)NCCF 53416,Fc1cncc(Cc2nc(-c3ccccc3)nn2C2(c3ccccc3)CCC2)c1 53417,C(N=c1[nH]c(=NC2CCOCC2)[nH]c2c1CCC2)c1cn(C)nc1C(F)F 53418,C1(N)CN(C(=O)C=CC(c2cnn(C)c2)=O)CC12CCC2.CC1CCN1CC(=O)N 53419,C1(CNC(C2(N(C)C)CCC2)=O)CC2(CCC2)CN1C(=O)CCC1CC(F)(F)C1 53420,C1(NC(c2n(C(CC)C)ncc2)=O)(CO)CCCN(Cc2ccc(Br)s2)C1 53421,C(=O)(C(C)P(C)(C)=O)N(CCNC(c1occc1Cn1cc(Br)cn1)=O)CC 53422,C1(C)(CNC(c2c(C)nsc2)=O)CCN(C(c2cc(C3CC3)ns2)=O)C1 53423,N1(C(CCC2C(C)C2)=O)CCOCC1CCNC(c1cc(C2CCCC2)no1)=O 53424,C=CCC(C)(C)CC(=O)NC1CN(C(=O)CCc2ccc(=N)[nH]c2)CCC1CO 53425,c1(-c2ccc(C(=O)NC3C(N)CC3)s2)cc(OC(F)(F)F)cc(F)c1 53426,n1(CC)nc(C(=O)NCCN(C(c2csc(C(F)F)n2)=O)C(C)C)c(C)n1 53427,CC(C)CC(O)C(=O)NC1CCCC(C(=O)N(CC(F)(F)CO)C)C1 53428,c1(OC)ncnc(N2CCOC(C(C)NC(c3cnccn3)=O)C2)c1OC 53429,N1(C(C(C)(F)F)=O)CC2CCN(C(c3ccnc(C(C)(F)F)c3)=O)C(C2)C1 53430,C(=O)(C(C)(C)S(C)(=O)=O)NC1C(C)CCN(C(c2ccc(F)c(C(F)F)c2)=O)C1 53431,N1(C(=O)NC(C(C(C)C)C)Cc2ccccc2)c2ccc(Cl)cc2OCC1C 53432,N1(C(C2(CCC=C)CN(C(c3cccc(C)c3O)=O)C2)=O)CC2CCCC2C1 53433,C12(C(=O)NCC3(NC(c4ncccn4)=O)CCCC3)COCC1CS(=O)(=O)C2 53434,C=CC(CCC)CC(=O)N(C)CC1CN(C(c2ccccc2)=O)CCO1 53435,CC1(NC(c2cc(CC3CC3)cs2)=O)CCN(C(=O)CCC2CCOCC2)C1 53436,C=CCC(C)(CC)C(=O)N1CCC(NC(c2ccnc(C(F)(F)F)n2)=O)CC1 53437,C1(C#N)(C(N2CC(NC(c3ccc(OC)s3)=O)C(C)C2)=O)CCSCC1 53438,c1(C(N2CC(CCCNC(=O)C=CC3CC3)OCC2)=O)cccc2[nH]cc(Cl)c12 53439,C=CCC(C)(C)CC(=O)NC(CCF)C(=O)NC(CN(C)C)CC(C)C 53440,C1(C(C(=O)N(C(C)CNC(=O)Cc2cnn(C)c2)CC)O)CCOCC1 53441,c1(C(N(CC(CNC(CC(CCCC)O)=O)C)C)=O)cc2c(C)cc(C)nc2s1 53442,N1(C(C(C)(C)C)=O)CC(NC(=O)CCc2nc3ccccc3s2)C(C2CC2)C1 53443,N1(C(C(C)N=[N+]=[N-])=O)CC2COCC2(C(N2CCSC(C)C2)=O)C1 53444,C(=O)(C1OCCc2ccccc21)NC(CCCNC(c1c(COC)nn[nH]1)=O)C 53445,CC1(C#CC(=O)N2CCCC2C2CCN(C(c3ccc(C4CC4)s3)=O)CC2)CC1 53446,C#CC1(C(N2CC(SC(F)F)C2)=O)CCN(C(=O)C=CC(=O)NC2CC2)CC1 53447,N1(C(CN(C2CC2)CC)=O)CC=CC(NC(c2cccc(C(C)(C)C)n2)=O)C1 53448,CCCCCCC(CNC(c1nc(C)c(C)nc1C)c1nnnn1C)CC 53449,CN1CCN(C(=O)CCc2nccs2)C(C(=O)NC2C3CCC(F)(F)C23)C1 53450,c1(N2CCC(NC(c3c(C)ncs3)=O)C2)cc(-c2ccc(Cl)cc2)ncn1 53451,c1(C(N2C(CNC(=O)CC3CCCCCCC3)C=CC2)=O)n[nH]c2c1CC1CC21 53452,C1(CCC)CN(C(C2(Cl)CC2C(C)=O)=O)CC1C(=O)NCC(C)(CC)OC 53453,c1(C(=O)NC23CC(NC(c4ccnc(F)c4Cl)=O)(C2)C3)cc2cc[nH]c2cc1F 53454,N1(C(CC(C=C)C)=O)CC2(CC(NC(c3c(C)cc(C)nc3S)=O)CO2)C1 53455,c1(CNC(c2nnc(C)n2C)c2n(CCOC)nnn2)cccc(Br)c1 53456,C(=O)(C(CCC(C)C)NC(=O)C(=O)NCC)NC1C(CC=C)COC1 53457,C1(N(CC(=O)NC2CC2)C)CCCC12CN(C(=O)C=Cc1ccccc1F)C2 53458,Cc1cncc(CC(=O)NC2C=CCN(C(c3sccc3CC#N)=O)C2)c1 53459,C(C(C(F)(F)F)N1CCOCC1)NC(=O)CCCn1cc(Cn2cncn2)nn1 53460,N1(C(C2C3CN(C)CC32)=O)CCC(C(N2CCC(F)(F)CC2)=O)C(C)(C)C1 53461,c1(C(=O)NCCCCn2cc(CNC(N)=O)nn2)cc(Br)sc1Cl 53462,Cc1cccc(C)c1NCC(N1CCCN(C(=O)CCC2CCC(C)O2)CC1)=O 53463,NC1CN(C(C2(Cc3ccc(F)cc3)CCCN2)=O)CCc2ccccc21 53464,C1(C(=O)NC2CCN(C(CCCC)=O)C23CC3)CCn2cnnc2C1 53465,C1(NC(C(=O)NC)=O)(CNC(C2CCC(C)S2)=O)CCC(F)(F)CC1 53466,c1(C(N2C(C(=O)NCc3cnc(C)nc3)CC3CC32)=O)ccc(Cl)c(Br)c1 53467,c1(C(N(C)CCN(C)C(C2CCOC2C2CC2)=O)=O)ccccc1OC(F)F 53468,CC(C)C#CC(=O)N1CCC(O)(C(C)CNC(=O)C(C)(C)c2ccn(C)n2)C1 53469,C1(CCC(=O)NC(C(C)NC(CCCCCC)=O)CO)CCc2cnn(C)c2C1 53470,Cc1[nH]c2ccccc2c1C(N1CC(C)CN(C(=O)CCOC2CC2)C(C)C1)=O 53471,c1(CC(=O)N(C(C)CNCCF)CC)ccc[nH]1.S(=O)(=O)(CC)NC 53472,CCN=C(NCC(C1(CO)CCCC1)(C)C)N1CCN(S(=O)(=O)C(C)C)CC1 53473,C(C(F)(F)C(=O)NC1CCC(NC(=O)C(c2cccc(Cl)c2)C)C1)OC 53474,CN=c1[nH]nc(CC(=O)NCC2(O)CCN(C(C3(F)CCCC3)=O)C2)s1 53475,C1(CNC(c2cnc(C)o2)=O)CC(C)CCN1C(=O)C(Cc1ccsc1)NC=O 53476,N1(C(c2c(C)n(C3CC3)cc2)=O)CCN(C(=O)C(C)OCCN(C)C)CCC1C 53477,c1(CN2C(CNC(=O)C=CCN3CCCCC3)CSCC2)c(Cl)ccc(F)c1F 53478,C(=O)(C(C)(C)S(=O)(=O)C1CC1)N(CCN(C(c1cccc(COC)c1)=O)C)C 53479,N1(C(C(C)NS(C)(=O)=O)=O)CC2CC2(CNC(c2n[nH]cc2Br)=O)C1 53480,N1(C(CC(CC)O)=O)CC2(CCC(NCc3c(Br)ccc(Cl)c3Cl)C2)C1 53481,C1=CC(=O)Nc2c(N)ccc1c2.C1(CC=C)C(OC)CC1OC(C)(C)C 53482,n1(CC)nc(C(=O)NC(CO)C(C)NC(C2CCNC(=O)C2)=O)cc1C 53483,c1(CC)nn(C)c(C(=O)NC2CC(Nc3ncncc3I)C2)c1Cl 53484,N1(C(=O)C(O)C(F)F)CCC2(CCCN2C(C2(C3CCC3)CC2)=O)C1 53485,c1(C(=O)NC(CC)(C)CNC(=O)C=C(C)Cl)cc2c(cn1)NC(=O)CO2 53486,N1(C(COCC=C)=O)CC(C(=O)NCCc2cnn[nH]2)(SC)C1 53487,c1(C(=O)NC(CC)(C)CNC(=O)Cc2c(C)noc2C)n[nH]c2c1CCCCC2 53488,C1(O)(C(=O)NC2CN(C(C(COCC)N=[N+]=[N-])=O)CC2C)CCCC(C)CC1 53489,C1(O)(CN(C(=O)Cc2nc[nH]n2)C)CCCN(C(=O)C2=CSCCO2)C1 53490,N1(C(CS(CC)(=O)=O)=O)C(C)CC2CN(C(=O)Cn3nccc3C)CC12 53491,CC#CCC(C(=O)NCC1CC1(F)F)NC(c1c[nH]c(C)c1)=O 53492,C1(C(=O)NCC(N2CCC(NC(c3cscc3Cl)=O)C2)=O)CCC(F)CC1 53493,c1(C(=O)NC2CCN(C(=O)C3=CCCC3)C(C3CC3)C2)ccn2cccc2c1 53494,N1(C(C2C(C)OCCC2)=O)CC2CCC(CNC(c3cncn(C)c3=O)=O)(C2)C1 53495,c1(COC)c(C(=O)NC2CC2NC(C23CCCC2(C(N)=O)C3)=O)cnn1C 53496,N1(C(C(CC(C)C)F)=O)CCc2sccc2C1CNC(=O)CC(C)(C)CC(F)F 53497,N1(C(c2c(=N)[nH]cnc2)=O)CC2CCOCC2(NC(=O)C=Cc2cccnc2)C1 53498,CC(C)CS(=O)(=O)CC(=O)NC1C=CCN(C(c2cnc3n2CCC3)=O)C1 53499,C(=O)(C(CCCCC(=O)OC)N1CCCC(CCO)C1)NCCC 53500,Cc1ncc2c(n1)CCC(C(=O)NC1CN(C(=O)C#CC3(C)COC3)CC1O)C2 53501,N1(C(C2CCOC2)=O)CC2OCCN(C(c3cc(C4CCOCC4)[nH]n3)=O)C2C1 53502,C(=O)(CCOCCN(C)C)OC(C(N1CCC1)=O)C.C=CCOC(C)=O 53503,c1(CC)nocc1C(=O)NCCN(C(=O)C(C)COC)C 53504,C(=O)(CC(C)(O)CCC)N(C1C(C)CCN(C(C(C=C)c2ccccc2)=O)C1)C 53505,c1(CC(=O)N(C2CC(C(=O)NCC(CC)C)C2)C)cccnc1C 53506,N1(C(c2cnc3n2CCCCC3)C(=O)NC2CC2)CCCCC(C2CCOCC2)C1 53507,N1(C(C(C=C)O)=O)CCC(CO)C(NC(c2ccc(Br)c(C)c2)=O)C1 53508,c1(C(=O)NC2CC(F)(CNC(C(CC=C)CC)=O)C2)cc2nn[nH]c2cc1F 53509,Cc1ccc2c(c1)CCN(CCc1cc3cc(Cl)ccc3[nH]1)C2 53510,c1(N2CCC(CNC(c3cncc(OC)n3)=O)C(C)C2)nc(O)c2c[nH]nc2n1 53511,N1(CCNc2scc(-c3ccc(Br)cc3)n2)CCC2CCCC(C1)N2 53512,N1(C(c2ccc(SC)s2)=O)CC(C(=O)NC(C)(C)C)C(C)C1 53513,c1(CC)[nH]nc(Cl)c1C(=O)NC1CC2C(NC(c3ncsc3C)=O)C2C1 53514,N1(C(C)=O)CCCCC1C(=O)NC1(C)CC(NC(C2CCNC2=O)=O)C1 53515,Cc1cc(NC(=O)C(C)OCc2ccccc2C#N)cc(C)c1Br 53516,C(=O)(CCCC(=O)N(C)CC1COCCN1C(c1cncc(Cl)c1)=O)N(C)C 53517,c1(C(=O)NC(CNC(C=C(CCC)C)=O)CO)ccc(CCC)c(Cl)c1 53518,c1(OCC(=O)NC2CC(CCNC(CCCC=C)=O)C2)cccc2cccnc12 53519,C#Cc1cnn(CC(=O)NC(CC2CCC2)C(=O)NC2CC(N3CCCC3)C2)c1 53520,c1(NC(C(c2ccccc2)NC(=O)OCC)=O)ncc(C(=O)O)s1 53521,Cc1ccc(-c2cc(C(=O)N(C3CN(C(=O)CN4CCC4C)C3)C)n[nH]2)s1 53522,CCCC(C#N)C(=O)N1CC(C)(C)CC1C(=O)NCCc1n[nH]c(CC)n1 53523,c1(OC)cc(NC(C2C3CC2N(Cc2cc(Cl)ccc2I)C3)=O)ccc1C 53524,c1(C(N2CCCC(C)C2CNC(=O)C(C)C2CCCO2)=O)cncc2[nH]ccc12 53525,c1(C(=O)NCC2CCCN2C(=O)CSc2nc[nH]n2)cccc(-c2nccs2)c1 53526,c1(C(N(CC)CC2CCCN2C(=O)CC(C)(C)O)=O)cc(Cl)cc(Cl)c1 53527,N1(C(CCCN(C(C)=O)C)=O)CCC(C)(C)C1C(=O)N(C1CC(O)C1)C 53528,C1(N(C(=O)CC2CSC2)CC)CCN(C(=O)C(C2CCOCC2)F)CC1 53529,C(CC(CC)C(=O)NC1CC(C)(NC(=O)C(CC)C(=O)OCC)C1)=CC 53530,c1(NC(CN(C(=O)CN2C(C)CCC2C)CCC)=O)ccc(F)c(O)c1 53531,Cc1ccc(NC(=O)C(Cc2cn[nH]c2)NC(=O)CC2(C)CC2)cc1O 53532,Cc1cc(C(=O)NCCN(C(=O)C(O)CC(N)=O)C2CC2)cc(S(N)(=O)=O)c1C 53533,C(=O)(C(C(C)C)NC(=O)C(C1CCCCC1)C)NCC#CCC 53534,N1(CC(=O)NCCCN(CCCCNC(=O)CCC2CC2(C)C)C)CC(=O)N1 53535,Cc1nc(=O)c2c(C)c(C(=O)OCCC(C)NC(=O)OC(C)(C)C)sc2[nH]1 53536,C1(CCOC)(C(=O)Nc2cncnc2C)CCN(C(=O)C(C(C)C)SC)C1 53537,C(=O)(CS(=O)c1ccc(Cl)cc1)NCC(C1CC1)NC(=O)Cc1cnsc1 53538,Cc1oc(C#N)cc1C(N1CC(F)(C(N2CCCC(c3nc[nH]n3)C2)=O)C1)=O 53539,c1(-n2c(C)cnn2)ccc(C(=O)NCC2CCCC2NC(=O)CC(C)C)cc1 53540,C1(=O)N=C2NON=C2C12CC2.C(=O)(CCC(=O)NCC1CCCC(=O)N1)OC 53541,C(N=c1[nH]c(=NCc2cccc(Br)c2Cl)[nH]c2cc[nH]c12)C1(C(C)(C)C)CC1 53542,CC12CN(C(=O)Cc3ccns3)C(C(=O)NCC(C3CCCC3)O)(C1)C2 53543,c1(C(=O)NC2C(NC(CCC)=O)CC2)cn(C)nc1C(C)(C)C 53544,CC1(CNC(C2(F)CCCC2)=O)CCCN1C(C1CCCCO1)=O 53545,CS(=O)(=O)c1cc(CC(=O)N=S2(=O)CCCC2)ccc1F 53546,N1(C(CC=CCC)=O)CCN(c2ncncc2C)CC1C 53547,C1(C(=O)NCc2nncs2)(NC(C2C(C)C2)=O)CC1(C)C 53548,C(=O)(C1CCCc2c1ncn2C)NC1(C)CCN(C(c2n(CC)ncc2Cl)=O)C1 53549,C(=O)(CC(C)C(C)C)N(CC(=O)NC(c1c(C)noc1C)C)CC(C)C 53550,C(=O)(CC(F)(F)C(F)F)N(CC(CC)NC(c1cc(Br)n[nH]1)=O)CC 53551,C1(NC(C2(O)CCCC2)=O)CCC(CCNC(=O)C(C2CCOCC2)O)C1 53552,N1(C(Cn2c(C)c(Br)cn2)=O)CCCC2(NC(c3nccnc3N)=O)CC2C1 53553,c1(C(=O)NC2CN(C(C(C)(C)c3ccc(Cl)s3)=O)CC2F)ncc(F)cc1F 53554,C1(NC(Cc2c(C)con2)=O)CCCCC1NC(=O)C(C)(C)c1ccn(C)n1 53555,N1(C(CSCCC(C)C)=O)CCCCC1C1(NC(=O)C2=CCSC2)CC1 53556,N1(C(CCCC)=O)CCC2(CC1)CN(C(c1n[nH]c3c1CC1CC31)=O)CC(C)O2 53557,c1(C(=O)NC2C(NC(C3C(C(C)C)CCO3)=O)C2)ccccc1[N+](=O)[O-] 53558,c1(C(N(C2CCCC(NC(c3ccc(C)s3)=O)C2)C)=O)cc(C)c(C#N)cn1 53559,c1(C(C(=O)NCC(C)CC2CC2)NC(=O)CN(C)C(N)=O)cccnc1 53560,C(=O)(C#CC1CCCCC1)NCCC1N(C(c2c(CC)cco2)=O)CCCC1C 53561,N1(C(C(C)Cc2ccco2)=O)CC(C(N2CCS(=O)CC2)=O)CC(F)(F)C1 53562,N1(C(c2n[nH]c(CC)c2Cl)=O)CC2(CCCC(CNC(c3oncc3C)=O)O2)C1 53563,C1(CNC(C=Cc2cc(OC)ns2)=O)CC2CC(C1)N(C(=O)CC(C)C)C2 53564,C1(CCC)CN(C(=O)C(C)(C)COC(C)C)CCN1C(C1CCCS1)=O 53565,N1(C(CC(C=C)C)=O)CC2(C1)CN(C(c1nnn(CC)c1C(F)F)=O)CC2CC 53566,CC(C)CC(C)(CNC(=O)CN(C)C(=O)C1CC1)NC(c1cnc(O)c(Cl)c1)=O 53567,c1(C(=O)NC(C(=O)OC)Cc2cn(C)nn2)cnn2c(Br)cccc12 53568,C(=O)(C(C)C(O)CCCC)NCCCCCC(=O)N1CC(CC(C#C)C)C1 53569,N1(C(c2cc(Cl)cc(Br)c2F)=O)CCCC2(CCCO2)C1 53570,Cc1cc(C(=O)N(C)CC=CC(N2CCCCC2CCO)=O)cc(O)c1 53571,C1(NC(C2C(=O)NCCCC2)=O)CCN(C(C2(Cl)CCCCC2)=O)CCC1CO 53572,c1(CC(=O)NC(C)CC2CCN(c3ccnc(C#N)n3)CC2)cc(Cl)ccc1Cl 53573,Cn1cncc(C(=O)NCC2(O)CC2C(=O)NC2COC3(CCC3)C2)c1=O 53574,N1(C(CC(C=C)C)=O)CC2CN(C(=O)CC(=O)OCCC(C)C)CCC12 53575,Cc1cc(C(=O)NCC2CC3CC3N2C(c2ccc[nH]2)=O)c(C)cc1Br 53576,CCCS(=O)(=O)C(C)C(=O)N(C1CN(C(c2cc3cccn3cn2)=O)CC1O)C 53577,c1(OC)ccc2c(c1C(=O)NCCN(C(=O)C1=CCCSC1)C1CC1)CCC2 53578,c1(C(=O)NCC2C(C)CN(C(c3coc(C(N)=O)c3)=O)C2)cc(F)cc(Cl)c1N 53579,N1(c2c(Br)cnc(OC)n2)CCCC2(CCCCC2NC(=O)CC(C)(C)O)C1 53580,c1(C(=O)NCCN(C(=O)CCn2ccnn2)C)ccc2cc(F)c(F)cc2n1 53581,C1(C(=O)NCC2N(C(c3c(OCC)ccs3)=O)CCC2)CCCC2(CCC2)O1 53582,C1(NC(Cn2c(C)ncc2)=O)CC(C)N(C(=O)C(C)O)C1 53583,c1(C(=O)NCCC(C(=O)N2CC(C#N)(CCF)C2)OC)ccc2nccn2c1 53584,c1(C(=O)NC2C(CC)N(C(=O)Cc3nc[nH]n3)CC2)cnn2c(C)cccc12 53585,c1(C(NNC(c2cccc(-n3cc(C(=O)O)nn3)n2)=O)=O)occ2c1CCCC2 53586,c1(C(=O)NC2CCC(CNC(c3cnc(Cl)nc3)=O)CC2)ccc(I)cc1Cl 53587,C(=O)(CCCC(F)(F)CO)N1C(CNC(c2cc3n(n2)CCCCO3)=O)CCC1 53588,C(CCCCC(=O)O)C1C(c2cn(C)nc2)C1.C1(N)CCCC1(C)O 53589,c1(C(C)C)cccc(NC(C2CC2CNC(c2cccc(SCCO)c2)=O)=O)c1 53590,c1(C(=O)NC2(CC=C)CN(C(C3SCCC3C)=O)C2)ccn2ncc(C)c2n1 53591,C1(CC(=O)N(CCNC(C)=O)C2CC2)CN(C(=O)CCC2CC2C)CCO1 53592,C1(C(=O)NCC(C)(C2CC2)NC(=O)CSC(F)(F)F)CC1[N+](=O)[O-] 53593,C1(C(=O)NC(c2ccccn2)C(=O)O)C2Cc3ccc(Cl)cc3C12 53594,N1(C(C2C(CC)CC2)=O)CCCN(C(c2c(OC)cccc2C)=O)C(C)C1 53595,O(C1(OCC)c2cccnc2CCC1NC(c1csc(N)c1)=O)CC 53596,N1(C(CC2(C)CC2(Cl)Cl)=O)CC2C3CCC(C2C1)N(C(=O)CN1CCCC1=O)C3 53597,N1(C(C=CC=CCC)=O)CC(N=[N+]=[N-])CC1C(=O)NC1CCC(CCO)CC1 53598,Cn1[nH]nnc1=NC1CC2CCC1N(C(=O)Cc1cc(F)c(F)cc1F)C2 53599,C1(CNC(CC=CC(C)(C)C)=O)CC2CCC1N(C(=O)CSc1ccccc1)C2 53600,C1(OC)CC(NC(=O)Cn2ccc([N+](=O)[O-])n2)C12CCN(C(=O)C(F)=C(C)C)CC2 53601,c1(CN(CC(=O)NCCCN(C)C)C)ccc([N+](=O)[O-])o1 53602,C1(NC(C=C(C)C)=O)CCOC(CNC(c2ccc(F)cc2)=O)C1 53603,C(CCCC(C)(C)C(=O)NNC(=O)C(C)(C#N)CC)OC(CS(CC)(=O)=O)=O.C1(CC=C)CC(C)C1 53604,Cc1cc(C#N)ccc1C(N1CCC(C(=O)NCCS(C)(=N)=O)C(O)C1)=O 53605,N1(C(C2C(C)N(C)CC2)=O)CCCC(C)(NC(=O)CCc2ccc(Cl)nc2)C1 53606,Nc1c(-c2noc(CCN3CCCCC3)n2)cnn1Cc1ccc(F)cc1 53607,C(C(O)C(=O)N(C)CC1CCCN1C(c1cc(C(C)(C)C)on1)=O)SC 53608,N1(C(CC2(OC)CC2)=O)CCC(C2CC2C(=O)NC2(CC(F)(F)F)CC2)CC1 53609,N1(C(Cc2c(SC)cccc2)=O)CC(C)CN(C(=O)C=C(C)C)C(C)C1 53610,C1(CC(=O)Nc2ncn(CC)c2)CN(C(C2(CF)CC(=O)C2)=O)CC1C 53611,c1(C(c2nnnn2C)NCC(CCC)C)cc(S(N)(=O)=O)ccc1F 53612,c1(C(N(C(C)CC2CC2)C)=O)cc(CNC(C2(C3CC3)CCC2)=O)ccn1 53613,C1(NC(CC(=C)Br)=O)CCC(C)N(C(=O)CCC=CC)C1 53614,N1(C(c2n(CCC)ccc2)=O)CC(C(=O)NC2(CCOC)CC2)CC(C)C1 53615,C1(CCNC(CC(OC)OC)=O)CCCN(Cc2ccnn2C)C1 53616,C1(OCC=C)CCN(C(c2cnn(-c3ccccn3)c2)C(=O)NCC(=C)C)C1 53617,C1(C)(CC)CC(C(N2CCCC2(C)CNC(=O)C(C)CC2CCC2)=O)CCO1 53618,C(C(CCCC)NC(=O)CNS(=O)(=O)N(C)C)NC(CC=C)=O 53619,S(=O)(=O)(CC(=O)NC1(C)CN(C(=O)C(C)(C)N2CCCC2)C1)NC 53620,N1(C(C2C(OCC)C2C)=O)CC2(CCN(C(C3CC4(C)CC3CO4)=O)C2)C1 53621,CCCCC(C(=O)NCCC1(C(C)(C)O)CC1)N(C)C.C12(CC1)C(=O)NC2 53622,Cc1cc(C(N2CC(C(C)NC(=O)CN(C)Cc3ccc(Cl)s3)C2)=O)c(C)s1 53623,C(=O)(C(F)C(=O)NC(C)(C)CC(=O)N1CCC(NC(C)=O)C1)OCC 53624,c1(C(=O)NC(CC)CNC(c2c[nH]c(=N)o2)=O)sc2cccc(F)c2c1Cl 53625,c1(N2CCN(C(C3CC(NC(C4(Br)CCC4)=O)C3)=O)CC2)nc2ccccc2[nH]1 53626,N1(C(CC2(C)CC2)=O)CCC2(CNC(c3ccccc3C3CC3)=O)CCCCC12 53627,Cc1ccc2ccnc(NCc3nc(C(=O)O)c(C)s3)c2c1 53628,N1(C(C=CCN)=O)CCCC(F)(CO)C1.CC(C)(O)CC=O 53629,c1(CN2CCCC(NC(=O)Cn3cccn3)CC2)ccc2c[nH]nc2c1 53630,N1(C(C(CC)NC(C)=O)=O)CCC(C(=O)O)C1NC(=O)C(F)(F)F 53631,C(=O)(C(O)C1=CCCCC1)N(C1(C(=O)NCCC(CCCCC)O)CC1)C 53632,C1(C(N2CCC(C)(NC(CCC(=O)NC)=O)C2)=O)CCC(=O)C(C)C1(C)C 53633,c1(C(=O)NCC(C)N(C(C(C)n2ccnc2)=O)C)cc(S(N)(=O)=O)sc1Cl 53634,C12(C(N(C3CCC3)C)=O)CCCC(CN1C(=O)C(O)CN1CCCC1)C2 53635,C1(CN(C(CC=CCC)=O)C)COCCN1C(=O)CC1CCCC(C)O1 53636,N1(C(C(CC)OC2CCCCC2)=O)CCCC2(CCCN2C(C)=O)C1 53637,C1(NC(c2ccc(F)cc2O)=O)C2COCC1CC(NC(C1CCCCS1)=O)C2 53638,c1(C(=O)NCC(CNC(=O)CNS(=O)(=O)C2CC2)OC)cccc(C)c1C#N 53639,C1(NC(CC2(C=C)CCC2)=O)(CO)CCN(C(C2CN(CC)CCO2)=O)CC1 53640,N1(C(C(CC2CCCC2)OC)=O)C2CCC1CC(CNC(C1(Cl)CC1)=O)C2 53641,C1(CCNC(C2(C)CC(=C)C2)=O)CCCN(C(c2cc(CCC)[nH]n2)=O)C1 53642,N(C(=NCCN(C)C)NCc1ncccc1N(C)C)CC(C)(C)OCC 53643,N1(C(c2cc(C)n(C)n2)=O)CCCN(CCNC(C2CC2CF)=O)CC1 53644,CC1(CCCC(=O)NCC2(O)CCN(C(=O)Cc3cccs3)C2)NC(=O)NC1=O 53645,c1(-c2occ(C(N3CC(CCC)C(CO)C3)=O)n2)cccc([N+](=O)[O-])c1 53646,C12(C(N3CC(N(C(CCc4ccc(CC)cc4)=O)C)C3)=O)CC(C)(C1)OC2(C)C 53647,C1(NC(c2c(CC)nco2)=O)CC2(C1)CC2C(=O)NC1(C(F)(F)F)CC1 53648,C1(NC(Cc2nnc(C)o2)=O)CCC12CN(C(C1CCCN1C1CC1)=O)C2 53649,C(=O)(C(F)CC(CC)CC)NC1(C(=O)NC(CCC)c2nn[nH]n2)CC(F)C1 53650,N1(C(C(c2ccc(OC)cc2)(C)C)=O)CC2CC(C)N(C(=O)CSC(C)C)C2C1 53651,N1(CC(C)NC(=O)NC(C(=O)OC)C)CCN(S(=O)(=O)Cc2ccccc2)CC1 53652,c1(CCC)cc(C(=O)N(CCNC(=O)C(C)SC)CC2CC2)no1 53653,C1(C(=O)NC)CCCCN1C(=O)CC=CCNC(=O)CC1(CSC)CC1 53654,c1(C(=O)NC23CC2CN(C(=O)COCC2CCCO2)C3)ccc(OCF)c(F)c1 53655,CC1c2ccccc2CC1NC(=O)NCc1cn(-c2cccc(Cl)c2)nn1 53656,Cc1cc(C)c(CC(N2CCC(NC(=O)C(F)(F)C(C)O)CC2)=O)c(C)c1 53657,Cc1nncc(C(=O)NCC2CCCCN2C(C2CC(=O)C2C(C)(C)C)=O)c1C 53658,N1(C(c2cc(CC)sn2)=O)CC(C(=O)NC(C(C)C)C(C)C)C2(CC2)C1 53659,c1(C(=O)NCCCC2OCCN(C(C3(CC)CC3)=O)C2)cc2nccnc2[nH]1 53660,CCC(CC(=O)NCC(O)CNC(C12CC(C)(CO1)C2)=O)C1CC1 53661,C(=O)(C(C)CC(C)(C)C)NCc1c(CN(C)CC2CCC(C)C(C)C2)cccc1 53662,N1(C(c2c(OC)nccn2)=O)CCC2CN(C(=O)C=Cc3ccnn3C)CC12 53663,c1(C(N2CC3CSCC3(C)C2)C(=O)NC(C(=O)OC)C)cn2cc(F)ccc2n1 53664,C(CCCC(=O)N1CC(NC(c2scc(OC)c2OC)=O)C(C)C1)(OC)OC 53665,C(CC(C(C)(C)C)NC(=O)Cc1nc([N+](=O)[O-])n[nH]1)N(C)C(C1CCSC1)=O 53666,CC1(C)CC=CCN(C(C2(CF)CCN(C(=O)CC3(C#N)CC3)C2)=O)C1 53667,C12(C(=O)OC)CCC(C(=O)N(C3CN(C(=O)Cc4sccc4C)C3)C)(C1)C2 53668,C(c1cncn1C)=CC(N1C(C2(NC(c3c(C)n[nH]c3)=O)CC2)CCC1)=O 53669,C1(C(CNC(=O)NOC2CCC2)O)CCCCO1 53670,c1(C(C(=O)NCCCCCNC(=O)CSC(C)(C)C)N(C)C)ccccc1Cl 53671,Cc1cc(C(=O)NC2CC(C)CN(C(=O)CC3(C)CCC3)C2)nc(O)c1 53672,c1(OC)cccc2cc(C(C)NC(c3cnc(C)cc3C)c3nnnn3C)oc12 53673,C1(C2CC2)(CNC(C2CCC(C)(C)O2)=O)CCN(C(=O)C(Cl)=CCl)C1 53674,C(C1=NOC2CCCC12)NC(CCC1CCN(C(C2CCC(=C)CC2)=O)C1)=O 53675,C(=O)(CC(C)C(C)C)NCC1(CNC(CCC(=O)NCC)=O)CC1(F)F 53676,CCC(C(=O)OC)C(=O)N1CC(c2ccccc2)(NC(C2CC(F)CN2C)=O)C1 53677,c1(CNCC(C)CC2CCCCC2)cnn(CCF)c1 53678,CC1(CNC(C2CC2CC(=O)CNC(=O)NC2CC2)=O)CC2(CC2)C1 53679,C1(NC(c2c(C)nc[nH]2)=O)CC(C2CCN(C(c3csc(S(C)(=O)=O)c3)=O)C2)C1 53680,c1(OC)nccc(C(=O)NC(C)(C)CN(C)C(c2occc2Br)=O)n1 53681,N1(C(c2ncn(C)n2)=O)CCCC2C1CCCN2C(c1csc(CO)n1)=O 53682,n1(CCC)cccc1C(=O)NCC(O)C(=O)NC1(C(N)=O)CC1 53683,C1(C(=O)NCC(CC(C)C)(C)NC(c2cnc(Cl)s2)=O)CC(=O)CC12CCC2 53684,c1(NC(=O)NCC(c2ccoc2)C)ccc(OCC2CCC2CO)cc1 53685,C12COC3(C1)CN(C3)C2=O.c1(NC(C(N2CCC(C)C2)=O)=O)ccc(C#N)[nH]1 53686,N1(Cc2c(O)ccc(C)c2)CCC2(CC1)CC(NC(c1cncc(Br)c1)=O)CO2 53687,C1(NC(C(C)n2ccnc2)=O)CCCC12CN(C(=O)C1CC1)C2 53688,N1(C(CSCCCC)=O)CCOCC(NC(=O)NC2CCCC(CC(N)=O)C2)C1 53689,C(CCF)(C(=O)NCCC1CC(C)C1)NC(C1CC(OCC)C1)=O 53690,C1(CC(=O)OC)CN(Cc2ncc(SC)s2)C2(CC2)CO1 53691,c1(C(=O)NCCC2CN(C(CSCC)=O)CC2C)cc2c(C3CC3)cccc2[nH]1 53692,N1(C(C2(C#N)CC(=O)C2)=O)CCC(C2(NC(C3CC3C3CCCC3)=O)CC2)CC1 53693,C1(C(=O)NCCOCCNc2coc(Cl)n2)CCCN(Cc2cccc(F)c2)C1 53694,c1(CC)cc(Br)c(C(c2nnnn2C2CCCCC2)NC2CCC2C(F)(F)F)s1 53695,c1(CCC)ccc(C(=O)NC2CC2NC(C2(C3CC3)CCOCC2)=O)cc1N 53696,CCCC(C)CC(=O)N(CCNC(=O)CC1CCCCC1(F)F)CCOCCO 53697,N1(C(C2C3CC2N(Cc2ccc(C(=O)O)[nH]2)C3)=O)CCC2(CCCO2)C1 53698,N1(c2c(C)cncn2)CC2CC1CN2C(C1(C)CC=CCC1)=O 53699,C(CC(N)CC(=O)NCC1CC2CCC1C2)SC 53700,C1(NC(C2CCCC23CC3)=O)CCCN(C(=O)Cc2cscc2Br)CC1 53701,C(CCC(=O)NC1CCC(CNC(=O)C(F)=CC2CC2)C1)OCC 53702,c1(CC)ccc(C(=O)N(CCNC(c2ccc(C)o2)=O)CC2CC2)c(F)c1 53703,C1(CN(C(=O)Cc2csc(C3CC3)n2)CC)CCCN(C(=O)CN2CC=CC2)C1 53704,CCC1=NOC(C(=O)NCCCCC(C)NC(c2cc(C(C)C)no2)=O)C1 53705,C(=O)(CCC(=O)NC)NCC1(C=O)CC1.C(CCCCN(N1CCOCC1)C)OCC 53706,CC1CCN(S(C)(=O)=O)CCN1C1C2CCC1(c1ccc(F)cc1)C2 53707,C(C(=O)NNC(=O)CCNC1CCCCC1)c1c(C)n[nH]c1C 53708,C1(C(=O)NC(CNC(c2cnc(CC)[nH]2)=O)C(C)C)CCC(F)(F)CO1 53709,N1(C(c2nccc(SC)n2)=O)CCN(C(C2CCC(C)=C(C)C2)=O)CC(C)(F)C1 53710,c1(C(=O)NCCC(CNC(C2C(=C)C2)=O)O)ccc(OC)c(S(=O)(=O)N)c1.C1N=N1 53711,CCC(CC)C(F)C(=O)N1CC(C(=O)NCC2CCC(F)(F)C2)C2(CCC2)C1 53712,c1(C(=O)NCCC2CCN(C(c3ccc(CC)o3)=O)C2)cncc2ncn(C)c12 53713,C1(NC(C=CCN(C)CC)=O)CC(NC(C2CC(F)(F)C2)=O)C12CCOCC2 53714,C1(CC=C)(NC(=O)CCC2CC2)CCCN(C(=O)CC(N2C(=O)CCC2=O)C)C1 53715,C12C3C=CC4(CN(C(=O)C14)C2)O3.c1(C(N(CCC=C)C)=O)ccccc1 53716,c1(C(N2C(CN(C(C3(OC)CS(=O)(=O)C3)=O)C)COCC2)=O)ccc(O)nc1Cl 53717,C(c1cnn(C)c1C)=CC(=O)NCC(CNC(CN(C)CC)=O)C 53718,c1(CNC(C(C)Cc2ccccc2)=O)ccc(-c2cc(N(C)C)ccn2)cc1 53719,C1(NC(Cn2nnc(C)n2)=O)CN(C(C2CCCCC2(F)F)=O)CC12CCC2 53720,O=C1C=C(c2cnc3cc(C(=O)NCCN4CCOCC4)ccn23)CCC1 53721,c1(C(N2CCC(CNC(C(CC#C)C)=O)(OC)C2)=O)cc(C(=O)CC)ccc1F 53722,c1(C(=O)NC)ccc(CC(=O)NCC(C)NC(c2cnn(C)c2C(C)C)=O)cc1 53723,N1(C(c2ccn(C(CC)CC)n2)=O)CC(CNC(=O)Cc2cc(OC)no2)C2CC12 53724,c1(CN2C(C(=O)Nc3ccnc(OC)c3F)COCC2)n[nH]c2ccc(C)cc12 53725,C(=O)(CCCCNC(C)=O)NCCN(C(C(C)(C1CCOCC1)OC)=O)C1CC1 53726,C(c1ncco1)=CC(=O)NCC1CCN(C(c2ccoc2C2CC2)=O)C1 53727,CC(C)(C)C1=NOC(C(=O)NCCOCCNC(=O)C(F)CC2CCOC2)C1 53728,C1(OC)CN(C(=O)C2=NOCC2)CC1C(=O)N(C)OCC(F)(F)F 53729,Cn1cc(C(=O)NCC2CCCCC2NC(=O)CSC(F)(F)F)c2sccc2c1=O 53730,C1(CC(N)=O)(NC(c2c(C)cc(C)[nH]2)=O)CCN(C(c2sc(F)cc2C)=O)CC1 53731,C1(C(=O)NCC2=CCCCC2)C2CCN(C(c3ccsc3Cl)=O)CC12 53732,C1(CC)(NC(c2coc(C(C)(C)C)n2)=O)CCCN(C(C2CSCCS2)=O)C1 53733,c1(C(C)=O)ccc(C(=O)NC(CNC(=O)CCC(F)F)CC(F)(F)F)cc1F 53734,C1(C(=O)NCC(C2CCCC2)NC(C(CN(CC)CC)F)=O)CCC(C)CC1 53735,N1(C(c2cnn(C(CC)CC)c2C)=O)CCC(C)C(NC(c2csc(=N)[nH]2)=O)C1 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53896,C1(CN(C(=O)Cc2cccs2)CC)CCN(C(=O)C(F)COCCN(C)C)CC1 53897,Cc1nsc(C(N2CC(F)(C(=O)NCCSC(F)F)C2)=O)c1N 53898,O(C1CCc2c(Br)cccc21)C(=O)C(c1ccc(F)c(F)c1)=O 53899,N1(C(C2(F)CCN(C(C(C=CC)O)=O)C2)=O)CC(C)OC(C)(C)C1C 53900,C(=O)(CS(=O)(=O)CC(=O)N1CCCC1CNC(=O)C(=Cc1c[nH]cn1)F)OC 53901,c1(C(=O)NC2C(c3ccc(C)cc3C)CCCC2)cc(N)cc(O)c1Br 53902,c1(C(=O)NCCC2(CNC(C3CC3C(=O)O)=O)CC2)cc2c(cn1)CCCC2 53903,Cc1nsc(Br)c1C(=O)N(C)CC1CCCCN1C(=O)CCC1(C)CC1 53904,N1(C(CN(C(C(C)OCCOC)=O)CC#N)=O)CCN(C2CCCC2)CC1 53905,Cc1c(NC(c2nnnn2CC2CCCCO2)C2CCOCC2)ccc(Br)c1Cl 53906,C1(CNC(CCCCC#C)=O)CCCC2CN(C(=O)Cc3ccc(F)nc3)CC12 53907,n1(CC(=O)N(C2CN(C(=O)COCCN(C)C)CC2F)C)cnc2ccccc12 53908,Cc1cnn(CC(=O)NC2CC(C(C)NC(=O)C(C)Oc3cccnc3)C2)c1 53909,CCC(CC(=O)NCC1OCCC1C(=O)N(C)Cc1cc(OC)no1)C(F)F 53910,N1(C(CCN(C(=O)CCCC#N)CC#C)=O)C2CCC1CC2 53911,N1(C(CC2C(C)C2)=O)CC2CCCC(C1)N2C(=O)CC(C)c1ccco1 53912,C1(C(=O)NC(CCNC(Cc2ccn(C)c2)=O)(C)C)CCNC(=O)C1 53913,C(=O)(C1=Cc2ccccc2C1)N(CCC(=O)NC1COCCC1O)CC=C 53914,C(=O)(C1=C(Cl)CCOC1)NCc1ccc(C(N2CC(C#C)OCC2)=O)cc1 53915,N1(C(CN(CCC)C)=O)CCC2(NC(C3CCN(C(C)=O)CC3)=O)CCCCC12 53916,C=C(C)C1CN(C(C2COCCN2C(=O)C=Cc2ccncn2)=O)CCO1 53917,N1(CC(=O)CCC2CC2(F)F)CCC(NC(=O)C(c2ccc(Br)cc2)(F)F)CC1 53918,c1cc[nH]c(=N)n1.C1(N(CC)CCNC(=O)CCCC2CC2C)CCCCCC1 53919,Cc1ccc(CNC(C2CCN(C(=O)COCC3CCCOC3)CC2)=O)c(C)c1 53920,N1(C(c2c(CC)nc[nH]2)=O)CC2CCC(C1)C2CNC(=O)C(C)NC(=O)COC 53921,C12(C(=O)NCC(C(C)C)O)CCC(NC(=O)CC(C)O)(CC1)C2 53922,CC(C)CC(CNC(=O)C1=CCCOCC1)C(=O)N1CCc2nn[nH]c2C1 53923,C(=O)(CC(O)CNC(C1CCCC1O)=O)NCC(=O)N(CC)CC 53924,Cn1nc(C(N2CCC(C)(NC(C3CCCC3)=O)CC2)=O)c2cc(F)ccc12 53925,c1(CC)ccc(C(C)C(=O)N(C)CCN(C(=O)CC(C)C2CCCO2)C(C)C)cc1 53926,C(=O)(C(CC(C)C)N(C)C)NCC1(OC)CCN(C(c2ccn(C3CC3)n2)=O)C1 53927,C(=O)(C1=CCCC1(C)C)N1CC2C(NC(C3C(C(=O)OC)C3)=O)(CC2)C1 53928,c1(C(N(CCCNC(=O)Cc2ccnn2C)CC)=O)cnc(Cl)c(F)c1N 53929,c1(COCC)nnc(N2CCCC2CCNC(=O)C2CC2)s1 53930,CC1CC(NC(c2cc(C#N)n(C)n2)=O)CCN1C(=O)Cc1cnc(C2CC2)[nH]1 53931,C=CCN(OC)C(=O)CCC1CCCN(C(=O)CC2CC(F)(F)C2)C1 53932,C1(NCC(CNC(=O)C=CC(=O)OC(C)(C)C)OC)CC2CCC(C1)C2(F)F 53933,Cn1ccc(-c2cc(C(=O)NCC3CCN3C(=O)CC3CCCO3)n[nH]2)c1 53934,c1(OC)cc(C(=O)N(C(C)CN(C)C(c2cccn2C)=O)C)cc(C(F)(F)F)c1 53935,C1(C(=O)NC(c2nccn2C)CC)CCCN(C(c2nn(C)cc2C)=O)C1 53936,C1(N(C)C)(C(=O)NC2CCCC(NC(=O)C=Cc3ncc[nH]3)C2)CCCCC1 53937,c1(C(=O)NCCN(CCC)C(C2(C)CC(C)=NO2)=O)nc(C)n(C)n1 53938,Cc1nc(CC(=O)NC(Cc2cn[nH]c2)C(=O)NC2(C)CC2)n[nH]1 53939,C1(NC(CCc2nc(C)c(C)[nH]2)=O)CN(C(=O)CC2CCCCC2)CCC1C 53940,c1(-c2cc(NC(C3CCCCCC3)C)sc2)ccc(F)cc1 53941,c1(C(=O)NC(C)CNC(C2CCN2S(C)(=O)=O)=O)cnc2n1CCS2 53942,C1(CNC(C2(C(C)C)COC2)=O)C(C2CC2)CCN1c1nccn2nnnc12 53943,CCCCC(CC)CC(=O)NC1CCC(C)N(C(=O)C=CS(=O)(=O)CC)C1 53944,c1(CC(C(=O)N(CCOCCNC(C2(CC)CCOC2)=O)C)C)ccccc1Cl 53945,C1(C(=O)NCC2N(C(c3cc(C)sc3C)=O)CC(F)C2)CCCC2(CC2)C1 53946,C1(NC(c2csc(F)c2)=O)C2CCC(C2)C1C(=O)NC1CCC=CCC1 53947,C1(N(CC)Cc2ccccc2OCC(F)(F)F)CC(C)CN(C(=O)C=CC(C)C)C1 53948,Cc1cc(Br)ncc1NC(=O)CCC1CCCN1Cc1cnn(CCF)c1 53949,N1(CC)CCC(O)C(C(N2CCCN(CC3CCCCC3)CC2)=O)C1 53950,c1(NC(C)C)ncccc1C(=O)NC1CCCC1NC(C1CCOC1C)=O 53951,c1(C(N2C(CNC(c3ccn(C4CC4)n3)=O)CC(OC)C2)=O)cc(C)ncc1C 53952,Cc1cc(F)ccc1CNC(C1C=CCN1C(=O)CCC1CCOC1)=O 53953,C(C)(C)(CC(F)C(=O)N(C1CCOC(C)(C)C1)C)NC(C1C(C)OC(=O)N1)=O 53954,CC1(C)CC=C(C(=O)NCC(C)(C)NC(c2ccc(O)nn2)=O)CC1 53955,C1(CNC(CN(C2CN(C)CCO2)C)=O)CCN(C(c2ccccc2)=O)C12CC2 53956,C1(N(C(CCN(C(=O)C(C)Cn2cccn2)CC)=O)C)CC1C1CC1 53957,N1(C(c2c(CC)noc2)=O)CCCC2(CCN(C(C3(C4CCCO4)CC3)=O)C2)C1 53958,C1(CNC(=O)OCc2onc(C(=O)OC)n2)CCCCN1C(=O)OC(C)(C)C 53959,C1(CNC(N2CC(CC)OC(C)C2)=O)CC2(CO1)CC1(C2)OCCO1 53960,C1(CCCC)CN(C(c2sc(C3CC3)nc2C)=O)CCN1C(=O)C(C)C(C)(C)O 53961,S(=O)(=O)(CC(=O)N(C)CCOCCCNC(=O)CC1(C)CCCC1)NC 53962,C1(NC(=O)CSCC(N2CCCC2)=O)CC2CC1N(C(C1C3CCCOC13)=O)C2 53963,CN1CC(C(=O)NCC(C)(C)NC(=O)COC(F)F)c2ccccc2C1=O 53964,C1(NC(C2N(C)CC(F)C2)=O)CC12CCN(C(C1CCc3nn[nH]c3C1)=O)CC2 53965,N1(C(CSS(C)(=O)=O)=O)CCC2(CC2)CC1C(N1CCCC(CN=[N+]=[N-])C1)=O 53966,C1(NC(c2c(F)ccnc2F)=O)CC1C1CCCN(C(=O)C2=C(Cl)CC2)C1 53967,N1(c2nc(OC)nc(OC)n2)CC2CCCC(C1)C2C(N1CCCC(F)C1)=O 53968,C(=O)(C1=C(C)CCCC1(C)C)N(CC)CC1CCCN1C(=O)Cc1cccc(N)c1 53969,c1(C(N2CCN(C(c3ncsc3C3CC3)=O)C(CF)C2)=O)ccc(F)cc1Cl 53970,Cc1nc(CNC(=O)CCC(=O)N(C)C)oc1C(=O)NC(c1nc[nH]n1)(C)C 53971,C1(COC)CN(C(c2cc[nH]c2C2CC2)=O)CCN1C(C1CC(C)(C)CN1C)=O 53972,Cc1cc(C(N2CC(F)(F)CC2CNC(=O)CCc2cnc[nH]2)=O)cc(N)c1O 53973,C1(NC(C(C)OCC=C)=O)C2CCC1N(C(c1nc(C)n(C)n1)=O)C2 53974,c1(N(CC(=O)NCC(N(C(=O)C(C)(C)C)C)C2CC2)C)ncnc2[nH]cnc12 53975,N1(c2ncnc(Nc3c(C#C)nccc3)c2C)CCOCCc2ccc(F)cc21 53976,C(C(=O)NNC(=O)c1ccccc1CC(F)(F)F)C1(C)CC1(F)F 53977,c1(C(=O)NCCC2(C)CCN(C(C3C(C)CCO3)=O)C2)coc2ccc(F)cc12 53978,Cc1cccc(F)c1CC(=O)NC1CC1CNC(=O)C(C)(C)CF 53979,C(C(C)CN=c1cc(C)nc(CO)[nH]1)NC(C=Cc1cccc(OCC)c1)=O 53980,c1(OC)cccc(OC)c1S(=O)(=O)NC1C2CCCCCCC12 53981,C1(CNC(C2CC(F)(F)C2)=O)CC2(CCC2)CN1C(c1cccn2nnnc12)=O 53982,CC12COC(C(N3CCC(O)(CNC(c4ccns4)=O)C3)=O)(C1)C2 53983,c1(N2C(CN(C(C(CCC)N(C)C)=O)C)COCC2)ccc([N+](=O)[O-])cc1 53984,c1(C(C)NC(=O)NCCn2cccc2)cc(Br)ccc1I 53985,c1(C(N2C3CC(NC(CCC=C(C)C)=O)C2CC3)=O)nn(C)c2c1CSCC2 53986,Cc1nn(C)c(Cl)c1C(=O)NC12CC(CNC(c3ncccc3O)=O)(C1)OC2C 53987,N1(C(CSCCCC)=O)CC2(CNC(c3[nH]c(O)nc3C)=O)CCC1CC2 53988,c1(OCCN(C(=O)CCCn2cc(CN)nn2)CC)ccc(C)c(C)c1.C(CO)O 53989,c1(OC)cc(O)c(CN2CC(C)(C(=O)Nc3cncnc3Br)C2)cc1Br 53990,C1(CNC(C2(C(N)=O)CCC2)=O)CC2COCC2N1C(=O)C(c1ccccc1)F 53991,Cc1c(C(N2CCN(CCNC(=O)C=CC(F)(F)F)CC2)=O)cnn1C1CCC1 53992,C(=O)(Nn1ccccc1=O)C1CC(NC(C(C2CC2)OC)=O)C1 53993,N1(C(C2C(C)CC2)=O)CC(C(N2CC(n3ccnc3)C2)=O)CC1(C)C 53994,C(C(N=[N+]=[N-])C(=O)N1CC(F)(CNC(=O)CCc2c(Cl)cccc2Cl)C1)OCC 53995,c1(C(=O)NCC(C2CCCCC2)NC(C(C)SC(C)C)=O)cccc(N(C)C)n1 53996,C1(C(N2CCC(NC(=O)Cc3ccc(Cl)s3)C(F)C2)=O)CN=C2N=CNN2C1 53997,N1(C(CCCCC2CN(C(=O)CC3CCC4CC34)C2)=O)CCOC(CC2CC2)C1 53998,C(CCCCCF)NC(=O)COC(=O)C(=CC(F)(F)F)F 53999,Cc1cn2c(CC(N3CCCC(NC(C4(C5CC5)CC4)=O)CC3)=O)csc2n1 54000,Cc1nn(CCO)cc1C(N1CCC(NC(=O)C(O)Cc2ccccc2)CC1)=O 54001,c1(CC)cc(C(=O)NC(CSC)Cc2ccccc2Br)cc(Cl)c1 54002,N1(C(c2cc(C)cc(C)c2C)=O)CCOC2(CCN(C(C3CCN3C)=O)C2)C1 54003,c1(CCC(N2CC(NC(=O)Cn3ncnn3)CC(C)C2)=O)ccc2ncsc2c1 54004,c1(C(N2CCN(C(C3CCC(C)CC3)=O)CC2)=O)cc2cc(Cl)ccc2n1C 54005,c1(C(N2CC(C(C(N3C(C(=O)OC)C=CC3)=O)OC)C2)=O)ccnnc1C 54006,S(=O)(=O)(c1c[nH]c(C(=O)NCC(C)(C(C)C)NC(C2CC(F)(F)C2)=O)c1)NCC 54007,C(=O)(CCCCNC(=O)C(C)C1CCCO1)NCCSCCOC 54008,N1(C(C(CCC)C)=O)CCN(C(c2ccc[nH]2)=O)CC1c1cn[nH]c1 54009,N1(C(C(CSC)C)=O)CCC(C)(C(=O)NCc2cn(-c3ccccc3C)nn2)C1 54010,N1(C(c2cc(CC(C)C)on2)=O)CCN(C(=O)C=CC2CCC2)C(C)C1C 54011,C12(NC(Cc3ccc(C#C)cc3)=O)CCN(C(=O)CC(C)CCC)CCC1C2 54012,N1(C(C2C(C(C)C)C2)=O)CC(C)(CNC(c2onc3c2CCCC3)=O)CC1(C)C 54013,CC(C)CC(C)CC(=O)NC12CCCC1CN(C(=O)CSc1ccccc1Cl)C2 54014,c1(OC)cncc(C(=O)NC2CCCC(C(N3CCC(F)CC3)=O)C2)c1 54015,C1(NC(C2C(OC)C2)=O)C2CC(O)C1N(C(=O)CNC(c1cscn1)=O)C2 54016,c1(NC(C2CN(c3ccncn3)CCO2)=O)ccc2c(=O)[nH]ccc2c1 54017,c1(C(N2C(CC(N3CCC(C#C)CC3)=O)CCC2)=O)cc(Br)c(O)c(Br)c1 54018,C1(NC(C)=O)CN(N(C)CCCSC(C)(C)C)CC1c1noc(C2CC2)n1 54019,C1(S(N)(=O)=O)(C(=O)NC(C)CN(C(=O)CCC#N)C)CCCC1 54020,CCCC(CNC(=O)CC1(O)CCCC1)NC(=O)CC1CCOC1C 54021,C(=O)(C(CNC(=O)C=CC(=O)N(C)C)NC(C)C)N1CC(CC(=O)OC)C1 54022,N1(C(NC2CCc3cccnc32)=O)CC2(CCOCC2)c2ccccc21 54023,c1(C(CC)N(C(c2n[nH]c(C)n2)C(=O)NC2CC2)C(C#C)C)ccccc1 54024,C(=O)(C1=CCCCO1)NC(C)CNC(C1(Oc2ccccc2)CC1)=O 54025,CCCCC(CNC(=O)CCOC(C)=O)NC(=O)CN1CCCCC1=O 54026,c1(C(C(=O)N(C2CCN(C(=O)CO)C2)CCC)N(C)C)c(F)cccc1F 54027,N1(C(C(c2ccc(Br)cc2)C)=O)CCC(F)C(NC(C2CS(=O)(=O)C2)=O)C1 54028,c1(C(=O)NC2CC(CNC(CC(CCC)O)=O)C2)cc(F)cc2nccnc12 54029,c1(CCC(=O)N(C)CC2N(C(CCSC)=O)CCC2)ncc(F)cn1 54030,N1(C(c2c(CC)noc2)=O)CCN(C)C(C(=O)NCC2CCCCS2)C1 54031,O=S1CCCCC12CN(Cc1ccn(CBr)c1)CC2 54032,C(=O)(C(CCNC(=O)C(C1CC1)SC)OC)N(CCC)CC1CC1 54033,c1(C(=O)NCC(CO)NC(=O)CC2(O)CCC2)cccc(-n2ccnc2)c1 54034,c1(C(=O)NC2CCC(N(C)C(c3ccccc3Cl)=O)CC2)cc(F)ccc1F 54035,c1(CN(CCNC(=O)NCC2CC(CC(C)C)OCC2)C)ccc(Cl)cc1Cl 54036,CC(C)CC(C(=O)NC1CCN(C(=O)C(C)SCC#N)CC1)N1CCCCC1=O 54037,N1(C(CC(CN(C)C)(C)C)=O)CCC2(C=C(C(=O)N3CCCCC3CF)C2)C1 54038,C1(C(N2C(CF)CC(OC)C2)=O)CC2CCC(C1)N2C(=O)Cc1cnns1 54039,N1(C(C(CCCC)O)=O)CCCC(C2CCCN(C(=O)CC3CC(OC)C3)C2)C1 54040,c1(C(=O)NCC2C(CNC(CCC(=C)Br)=O)C2)cc2ccccc2n1C 54041,N1(C(C2CC3C=CC2CC3)=O)CC2CCN(C(c3cnc4cccnn34)=O)C2C1 54042,C(=O)(CCCC(=O)N1CCC(CNC(=O)C(C)(Cl)Cl)C1)c1n(C)cnc1 54043,c1(CC)onc(C)c1C(=O)NCC1(F)CN(C(c2cc(CO)ccn2)=O)C1 54044,N1(C(C2(F)CCOC2)=O)CCC2(CC1)CC(NC(C13CCC(CO)(CC1)C3)=O)C2 54045,c1(C(=O)OCCC2CCC(C)O2)ccc(F)c2[nH]ccc12 54046,C12(NC(CC(=C)C)=O)CCC(CNC(=O)CCCOc3ccccc3F)(C1)OC2 54047,c1(-c2cn(CC(N3C(c4ccc(C)s4)CCC3)=O)nn2)cn2ccccc2n1 54048,C1(NC(COCCCCC)=O)CCN(C(=O)CC(O)C(C)C)CC1O 54049,C(c1cn(C)cn1)=CC(=O)NCCC(C)NC(=O)C=Cc1ccncn1 54050,C1(CNC(C2CN(C)C(=O)C2)=O)CC(C(=O)NCc2cn[nH]c2)=NO1 54051,CCCC(CC(=O)Nc1cc(C)cnc1OCC)NC(C1CN2CCC1C2)=O 54052,CCCCCCC(C)N(CCC(C)NC(C1CN(CC(=O)OC)C1)=O)C 54053,C1(CC(N2CC3C(NC(CC4N(CC)C(=O)CC4)=O)C3C2)=O)CC2C=CC1CC2 54054,c1(-c2scc(C(C(=O)NCc3ccco3)N(CCCC)CC)n2)cccc(C)c1 54055,c1(CC)c(C(=O)NC2CN(C(=O)CCc3ccn(C)c3)CC23CC3)cccc1C 54056,C1(CNC(CN(C(COC)=O)C)=O)CCC2(CN(C(c3c(C)n[nH]c3C)C)C2)O1 54057,N1(C(Cc2c(C)occ2)=O)CC(NC(c2cocc2C(N)=O)=O)CC(F)C1 54058,c1(C(=O)NCC2C(NC(C(=O)NCC)=O)C2)ccc(F)cc1Br 54059,c1(C(=O)NCCNC(C(C)O)=O)ccn(CC(F)(F)F)c(=O)c1 54060,N1(C(c2cc(C)ns2)=O)CCCN(C(C2CCn3nccc3C2)=O)C(C)C1 54061,c1(C(N2C3CN(C(c4ccc(C(N)=O)cn4)=O)CC2C3)=O)ccc([N+](=O)[O-])cn1 54062,N1(CC(=O)NCC(C)N(C(c2c[nH]c(=N)s2)=O)CC)CCCCCC1 54063,N1(C(C2C(CNC(C(C)O)=O)CC2)=O)CC(C)c2ncccc21 54064,N1(C(CC2CCC(C)(O)CC2)=O)CC2(CCCC(CNC(C3(Cl)CC3)=O)O2)C1 54065,N1(C(CC2ON=C(C)C2)=O)CCC(O)(CCNC(c2cc(C(F)F)cs2)=O)CC1 54066,CC(C)CCCCC(=O)NCCCC(O)C(=O)NCc1cc(Cl)ccn1 54067,C1(NC(CCN(CC=C)C(C2CC2(C)C(C)C)=O)=O)C(O)CC1O 54068,c1(CC(C(=O)NCCC(O)C2CC2)NC(c2c(CC)ccs2)=O)ccccc1Br 54069,c1(NC(=O)NCC2CCCC2NC(=O)C(Cl)(Cl)Cl)cnncc1Cl 54070,C(=O)(CCCCCCCCN)N1CCN(CC(=O)Nc2c(OC)cccc2)CC1 54071,c1(C(=O)NC2CCN(C(C3CCC(NC(C)=O)CC3)=O)C2)ccc(O)cc1O 54072,CC1(NC(c2c(OC(F)(F)F)cccc2O)=O)CCN(S(N)(=O)=O)CC1 54073,C1(CNC(COCC)=O)CN(C(=O)C(C2CC2)SC)CCC1(C)C 54074,C1(C(=O)NC2CC(NC(c3n(CC)ccc3)=O)C2)Cc2cc(F)ccc2O1 54075,Cc1c(C(=O)NCC(C)CNC(=O)C(C(C)C)NS(C)(=O)=O)ccc2c1CCC2 54076,N1(C(CCc2nc(C)sc2)=O)CCN(C(=O)C(C2CCCCC2)O)C2(CCC2)C1 54077,c1(NC(c2cc(-c3cnc(C)s3)ncc2)=O)ccc(C(F)(F)F)cc1[N+](=O)[O-] 54078,C1(CCNC(c2cnc(Cl)s2)=O)CCCN(C(c2cnc(Br)s2)=O)C1 54079,c1(CNC(c2cnn(C)c2C)c2n(CC)nnn2)cn(C)c2ccccc12 54080,C1(NC(c2c(CC)nn[nH]2)=O)CC(CNC(=O)CSCCOC)C1(C)C 54081,N1(C(CCN(C(C)=O)C)=O)CCN(C(=O)C(Cl)=CCl)CCC1C 54082,C#CCC(C(=O)NCC(C)C(=O)OCC)NC(c1cc(CC)nn1C)=O 54083,c1(SC)cccc(F)c1C(=O)NCC1COCCN(C(c2cnccn2)=O)C1 54084,C1(CC(=O)NC2C(NC(c3cc(=N)[nH]cc3)=O)C2)CCC2(CC1)OCCO2 54085,c1(C(C(=O)NCCCCCN(C(C2CC(C)C2)=O)C)O)ccc(F)c(Cl)c1F 54086,c1(C(N(C2CN(C(C3(S(N)(=O)=O)CCC3)=O)C2)C)=O)ccccc1C#N 54087,C(=O)(N1OC2CCC1CC2)C1(C#C)CCNCC1 54088,Cc1cc(NC(C2(Oc3ccccc3C)CC2)=O)ccc1NC(c1cc[nH]n1)=O 54089,CCCCC(CC)C(=O)NC1CCCC1NC(=O)C(C)(C)c1cnc[nH]1 54090,c1(C(CC)CC)cc(C(N2CCC(CN(C(=O)CCn3cnnn3)C)C2)=O)on1 54091,C=CCC(C)(O)C(=O)NCC1(OC)CCN(C(=O)C(C)NC=O)C1 54092,c1(-c2ccc(N3C4(C#C)CC(C3)C4)cc2)nc2ccccc2c(=O)n1SC(F)F 54093,c1(N2CCOCC(CNC(Cc3cccc(OC)n3)=O)C2)cc2nncn2cn1 54094,C1(NC(C2C(C)C2)=O)CN(C(=O)C(C)S(C)(=O)=O)CCC12CCC2 54095,CC1(C)CCC(C)(NC(C2(NC(c3sccc3F)=O)CC(CO)C2)=O)C1 54096,Cn1nc(CNC(=O)C(C2CCOC2)NC(=O)OC(C)(C)C)cc1C(F)(F)F 54097,N1(C(CC2(C(C)C)CN(C(=O)Cc3cccnc3O)C2)=O)CCS(=O)(=O)CC1 54098,C(=O)(C1=CC(O)C(NC(C2CC3(CCC3)CO2)=O)C1)N1CC(C2(C)CC2)C1 54099,C(C(C)C)(C(O)C(=O)NC(C(N1CC=CC1CN(C)C)=O)c1ccoc1)OC 54100,c1(C(N2CCCCC2c2ccccc2)C(=O)N(CC=C)CC)cn(C(C)C)nc1Br 54101,CCCCC(C(=O)NC1(C2CN(C(=O)C3=CCOC3)C2)CC1)N(C)C 54102,C1(CC(=O)NCC2N(C(C(F)OC)=O)CCC2)CCCN(C(C)C)C1 54103,Cc1cccc(C(N2CC=CC(NC(C3CC(N=[N+]=[N-])C3)=O)C2)=O)c1F 54104,C(=O)(CCCC(C)(F)F)N(C1CCCN(C(C(C=CCCC)O)=O)C1)CC 54105,N1(C(C(C)SC)=O)C2CCC1CC(CNC(C1(N3CCOC3=O)CC1)=O)C2 54106,C(=O)(CC(C)(C)CC(F)(F)F)N1CCC(COC)(NC(=O)C(F)=C(C)C)C1 54107,C1(NC(c2cc(CC)n(CCO)n2)=O)CN(C(C2CC(=O)N(C)C2)=O)C(C)(C)C1 54108,N#CCCCC(=O)N1CC(F)CC1CNC(c1cccnc1-n1nccn1)=O 54109,c1(OC)c(Cl)ccc2[nH]c(C(N3CCCC(CNC(=O)C4=CCCS4)C3)=O)cc12 54110,C=CC1(CC(=O)NC2(C)CCN(C(c3c[nH]c(=N)nc3C)=O)C2)CCCCC1 54111,CCC(CO)CN=c1cc(C)[nH]c(=NCCN2CCC(F)(F)CC2)[nH]1 54112,c1(C(N2CC(NC(C(C=C)(C)C)=O)C(C)C2)=O)c(C)ccn1C 54113,C1(C2CCC2)(CNC(C(CSC)OC)=O)CCN(C(c2ccncn2)=O)CC1 54114,N1(C(C2CN(C)C2)=O)CCC2(NC(=O)C3=COCCO3)CCCCC12 54115,N1(C(C2OCCN(CC)C2)=O)CC2(CCN(C(=O)CCC(C)C)CC2)CC1C 54116,CC1CCCCN1C(=O)CN(C(=O)C(=O)NC1CC1)CC1CC1 54117,N1(C(C(F)=CC)=O)CCN(C(=O)C(CC(F)F)c2ccc(F)cc2)C(CCC)C1 54118,c1(CC)cc(NC(=O)CC2(OC)CCOCC2)nc(CC)n1 54119,C(C(C)C(C)C(=O)N1CC(C(=O)NCCNS(C)(=O)=O)C(C(C)C)C1)OC 54120,C(=O)(CC(C)CC(C)C)NCCC(C(=O)N(CCCOC)C)(C)C 54121,c1(CC)cc(C(=O)NC(c2cccc(C)c2)CNC(=O)C(C)OCC)ccc1Cl 54122,N1(C(CNC(=O)NC)=O)CCC(C)(C)C(CNC(=O)C(C2CCCCO2)OC)C1 54123,N1(C(C2(C)CCCO2)=O)CC2(NC(=O)CCC3(C#N)CCC3)CC1C2 54124,C(C(=O)N1CCN(C(=O)C2=CCCC2)C2CC12)(c1ccccc1)=C(C)C 54125,C1(CN(C(=O)CN(C)C(C)C)CC)CCN(C(=O)CC2CCC(C)(C)O2)CC1 54126,c1(C(=O)NC(CC(C)NC(c2c(C)ccnc2C)=O)C)n[nH]c2cccnc12 54127,c1(C(=O)OCC)nc(=NC(C)CNC(=O)Cc2cc(O)nc(O)n2)cc[nH]1 54128,C12(CNC(C(CC#C)(C)C)=O)CCCC(CN1C(=O)CNC(=O)OCC)C2 54129,C1(CCC)CN(C(=O)Cn2cnc(C#N)n2)CC1C(=O)N(C12CC(C1)C2)C 54130,C1(C(=O)NC(C(C)C)(C)CNC(=O)Cc2cnn(C(F)F)c2)CC2(CCC2)CO1 54131,C1(C(N(CC(C)NC(Cc2c(OC)cccc2)=O)C)=O)CCCC1S(C)(=O)=O 54132,CC1COCCN1C(C1CC1c1cccc(Br)c1)=O 54133,C1(NC(C2CC=CCO2)=O)CCOC12CCN(C(=O)Cc1ccccc1F)CC2 54134,C12(CC(=O)N(C3CC4CCC3CC4)C)CCC1CN(C(c1cc(Cl)c[nH]1)=O)C2 54135,C#CC1(C(N2CC(OC)CC(NC(c3cccc(F)c3C)=O)C2)=O)CCOCC1 54136,c1(NC(CCC)=O)nc2ccc(CC(=O)NC)cc2[nH]1 54137,c1(OC)ccc(OC(=O)N(CC(c2ccccc2OC)O)C)c([N+](=O)[O-])c1 54138,c1(CC(=O)NC(c2cnn(C)c2)C(=O)NCC(CSC)(C)C)ccc(C)c(C)c1 54139,N1(C(C2CCN(CC)C2)=O)CCN(C(=O)COc2ccc(F)cc2F)CC1CF 54140,N1(C(c2c(CC)c[nH]n2)=O)CC(O)CC1(C)C(=O)NCC(C)C(C)(F)F 54141,N1(C(CC(C)C)=O)CC2CCN(Cc3c(F)cccc3Br)CC2C1 54142,C(=O)(C(O)CCS(C)=O)NCCCCCNC(C(C)Cc1cccc(Cl)c1)=O 54143,c1(NC(CCN(C(=O)CC(C)=C(C)C)CC#C)=O)ccc(CSC)c(F)c1 54144,CC1(C)CCCC(CCN2CCC(c3ccccc3)(C(F)(F)F)C2)O1 54145,C1(C(=O)NOCCCN(Cl)Cl)CN(C(C2CCOC2)=O)CC1F 54146,c1(N2CCC(c3scc(CC)n3)CC2)ccc(S(=O)(=O)N2CCCCC2CC)cn1 54147,c1(C(=O)NC2C(CNC(C3N(C)CCC3)=O)COC2)cnc2c(c1)CNC(=O)N2 54148,c1(C(=O)NC2CC(CCNC(C3(CC)COC3)=O)C2)scnc1C(F)F 54149,c1(COC)ccc(C(=O)NC(CNC(=O)CC2CC2(Cl)Cl)C2CC2)o1 54150,C1(CC(C)NC(c2cncc(F)c2)=O)CC2CCC(C1)N2C(C1CCCCCO1)=O 54151,N1(C(C2CCCOCC2)=O)CCOC2(CCN(C(C3CCS(=O)(=O)CC3)=O)C2)C1 54152,c1(CC)cccc(C(N2CCN(C3CN(C(C4(C)CC4(F)F)=O)C3)CC2)=O)c1N 54153,O=C(C1=COCCO1)NCCC1COCCN1C(C1CC1C(F)(F)F)=O 54154,Cc1nonc1C(=O)NC1(C(=O)NC2CSC2)CCSC1 54155,N1(C(CC2CC(OCC)C2)=O)CCC(C)C(CNC(c2ccc(O)nc2C)=O)C1 54156,C1(CCNC(C=CCNC(COC(CC)C)=O)=O)COCC1O 54157,C(=O)(C1=C(Cl)CCCC1)N(C(C)CN(C)C(c1ccsc1-n1cnnn1)=O)C 54158,c1(CN2C(C(=O)NCc3c(C(N)=O)nccn3)C(O)CC2)nc2ccccc2[nH]1 54159,C1(n2cc(SCC)nn2)CCCN(C(=O)C=CC2CCC2)C1.C12CC(C1)NC2=O 54160,c1(OC)ccc(F)c(CC(=O)NC2CCN(C(=O)CCF)CC2O)c1 54161,C1(C(=O)NCCC(C)N(C)C(c2cnc(C(F)(F)F)s2)=O)CCCOC1C1CC1 54162,C1(C(=O)NCC(CNC(c2ccc(C(N)=O)cc2)=O)O)CC12CCS(=O)(=O)CC2 54163,c1(CCC)cc(C(=O)NCCC(C)(C)NC(C2CCC2(OC)OC)=O)n[nH]1 54164,C1(CNC(CCN(CCC)C)=O)CCCCC1NC(c1cccc(C(F)F)n1)=O 54165,C#CC1(O)CC(C(=O)NCCOCCC(=O)NC(C#C)C2CCC2)C1 54166,C1(C(N(CCCNC(=O)CCc2nccs2)CC)=O)CNC(=O)CC12CCOC2 54167,c1(C(C)OC(c2c[nH]nc2-c2cccc(Br)c2)=O)ccc(F)c(F)c1F 54168,Cc1cn2cc(C(N3CCC(F)C(NC(c4ccc(O)cc4F)=O)C3)=O)sc2n1 54169,CCC(C)(C(=O)NCC(CC)(CC)NC(C1CCN(C)C1)=O)C(N)=O 54170,N1(C(c2n[nH]cc2C)C(=O)NCCC)CCSC2COCCC12 54171,CCC(C)C(O)C(C)C(=O)NCCCN(C(=O)CSCC(N)=O)C1CC1 54172,C1(NC(C=CC=CCC)=O)C2CN(C(c3ccc(-c4ccc(F)cc4)[nH]3)=O)CC12 54173,CC1CN(C(=O)Cc2ccncc2OC(=O)C(C)(F)F)CC1Cc1ccccc1 54174,C#CC(C)(CC)NC(=O)C(CC)NC(=O)Cc1sccc1C 54175,n1(CCOC)cc(C(=O)N(C2CCN(C(=O)C=Cc3cncs3)C2)C)nn1 54176,C#Cc1ccnc(C(N2CC3(C2)CN(C(=O)CC(F)(F)Br)C3)=O)c1 54177,S(=O)(=O)(c1ccc(C#N)cc1)NC(CC1(C)CN(CC2CNC(=O)O2)C1)=O 54178,N1(C(c2c(N)cccc2F)=O)CCN(C(=O)CC2CC3(CCC3)CO2)CC(O)C1 54179,c1(C(=O)NC2CN(C(C(C3CCCOC3)OC)=O)C2)nonc1N 54180,C1(NC(=O)CC2CCC(F)(F)C2)CN(c2ccncc2[N+](=O)[O-])CCC12CCC2 54181,C1(Cc2ccc(CC)o2)(CO)C(OCc2ccc(F)cc2)CC1OC 54182,C1(F)(C(=O)NC(C2CN(Cc3c(OC(C)C)cccc3)C2)C)CCC(F)(F)CC1 54183,C(=O)(N=c1ccn(CCCO)[nH]1)C1N(C(c2ccc(COC)cc2)=O)CC=C1 54184,C1(C(=O)NC2CCC(Cn3cc(Cn4cccn4)nn3)CC2)(CC)CCCCO1 54185,N1(C(CC2(C)CCOC2)=O)C(C(N2CCC([N+](=O)[O-])CC2)=O)C2CC(O)C1C2 54186,C(=O)(CC(CNC(c1c[nH]cc1C(C)C)=O)C1CCC1)NC(COC)CO 54187,c1(OC)ccc(C(=O)N(CC(C)NC(=O)CCCOC)C)cc1Br.C(C)(=O)O 54188,C(=O)(C1=CCC(C)(C)CC1)NCC(CNC(c1c(C)c(C(N)=O)ccc1)=O)O 54189,C1(CNC(c2ncc(C3CC3)cc2F)=O)CC12CCN(C(c1cocn1)=O)CC2 54190,C1(C(=O)NC(CC(=O)N(CC#CC)C)C2CC2)Cc2ccccc2C1 54191,c1(NC(N2CC(OC3CCCCC3CC(F)(F)F)C2)=O)ccc(F)nc1 54192,c1(C(=O)NCC2OCCN(C(c3cc(C)nc(O)c3)=O)C2)coc(S(C)(=O)=O)c1 54193,C1(NC(CNC(C(CC)C)=O)=O)CCCCN(C(C2(C)CC2C)=O)C1 54194,Cc1cc(C(N2CC3C(CNC(C4CCC(=O)N4)=O)C3C2)=O)c2sc(=N)[nH]c2n1 54195,CCC(C)CN(C)N(CCCNC(C1CCCC1)=O)CC(=O)OC(C)(C)C 54196,N1(C(Cc2c(C)noc2Cl)=O)CCC(NC(c2c(F)cncc2Cl)=O)C(F)C1 54197,c1(CCOCC(=O)NCCCN(C(=O)CC2C=CCCC2)C(C)C)ccccc1 54198,Cc1cc(Cl)c(C(N2C3CCC2C(NC(=O)C(C)O)C3)=O)cc1N 54199,C1(C(=O)NCC(C=C)O)CC(O)C(O)CC1CNC(C1CC(O)C(F)C1)=O 54200,CCC(CC(C)C)C(=O)N1CC2CC(NC(=O)CNC(=O)CC(C)C)CC2C1 54201,C(C)(CN=c1[nH]c2c(c(=NCCCN=c3cc[nH]c4ccccc34)[nH]1)SCC2)SC 54202,C(=O)(CCCCCO)NCCOC1(CNC(C2CC(C)OC2)=O)CCOCC1 54203,CCC(C)(C(=O)N1CCCC(COC)(NC(c2ccc(Cl)c(C)c2)=O)C1)C(N)=O 54204,C1(C(N2CCC(NC(c3ccnn3C3CCC3)=O)(CF)C2)=O)CN2CCC1CC2 54205,c1(OCC(C)C)cc(N)ccc1-c1cccc(-c2nccn2C2COC2)c1 54206,N1(C(C(=Cc2cn[nH]c2)C)=O)CCCC2(CCCCC2NC(=O)CC(C)C)C1 54207,c1(C(N2CCC(CC(=O)NCc3ccc(F)cc3F)C2)=O)cc(Br)ccc1CO 54208,c1(C(N2CC(N(C(C(Cc3c(C)nc[nH]3)O)=O)C)C2)=O)cc([N+](=O)[O-])cn1C 54209,N1(C(CCCC(C)=O)=O)CC2(CC(NC(=O)C(N3CCP(C)(=O)CC3)C)CO2)C1 54210,C1(NC(CN(C(CCOCCC)=O)C(C)C)=O)CCOC(CC)C1 54211,C1(C(=O)NC(CNC(C(CC(=O)OC)C)=O)C)Cc2cccnc2C1 54212,c1(N2CC3C(CNC(c4c(OC)cc(C)s4)=O)C3C2)nc(C)nc2n[nH]cc12 54213,N1(C(=O)Cn2cccc2)CCC(C(N2CC3CC3C2)=O)C(O)C1 54214,c1(C(=O)NC(C(C)NC(C2(O)CCCCC2)=O)CO)ccc(Cl)c(C#N)c1 54215,CC(C(=O)NC1CCN(C(=O)CNC(=O)CN(C)C)C1)C(C)(C)C 54216,Cc1cc(C(=O)NCCCCNC(c2cncc(C(N)=O)c2)=O)sc1Br 54217,C1(C2CCC2)(C(=O)NC2C(NC(C3(C(F)F)CCCO3)=O)CCC2)CC1 54218,N1(C(C(C)OC)=O)CCCN(C(c2cc(C)n(C(C)(C)C)n2)=O)C(C)C1 54219,CC(C)C(CC(=O)NC12CC(NC(c3ccnc(S)c3)=O)(C1)C2)C(C)C 54220,C1(N(C)C(c2cnc[nH]2)=O)CCCN(C(C2NC(=O)OC2(C)C)=O)CC1 54221,O=C(CCN1C(=O)CSc2ccccc21)NCCNC(c1cccn1C1CC1)=O 54222,c1(CNC(CCCN(C(C(CSC)C)=O)C)=O)nn(C)cc1C 54223,c1(C(=O)NC(C2CCCCC2)CNC(C(C=C)(C)O)=O)nccc(C)c1F 54224,C1(C(=O)NCC2(O)CC(CNC(c3cc(COC)sc3)=O)C2)CC(=O)N(OC)C1 54225,N1(C(C23N(C(CC(C)n4ccnc4)=O)CCC2C3)=O)CCc2nnnn2CC1 54226,c1(C(N2C(CC)C(NC(c3scnc3C(F)F)=O)CC2)=O)csc2nccn12 54227,c1(SC)ccc(C(N2CCN(C(c3ncccc3F)=O)C3CC23)=O)cc1[N+](=O)[O-] 54228,c1(C(=O)NCC(CCNC(Cc2cn(C)nc2)=O)(C)C)c[nH]c2ncccc12 54229,C1(NC(CCC2C(C)C2)=O)CCN(C(c2ccc(OC(F)(F)Cl)cc2)=O)C1(C)C 54230,N1(C(c2ccn(CC(F)F)n2)=O)CCN(C(c2cnc(O)o2)=O)C(C2CC2)C1 54231,c1(NC(COC)=O)cccc(NC(=O)NC(c2ccn(C)c2)C)c1 54232,c1(CC(C)C)cc(C(N2CCC2CNC(C2(C3CCCO3)CCC2)=O)=O)n[nH]1 54233,CCCC(CC)CC(=O)NC1CCN(C(c2ccc(C)cc2)=O)C1 54234,C=C1CC(C(=O)N(C2CC(C)C2)C)(CNC(c2cc(Cl)cs2)=O)C1 54235,N1(C(C(C)Nc2ccc(SC)cc2)=O)CC(O)CCC(F)(F)C1 54236,c1(NCCC(C)(C)SC)cc(C)c(S(=O)(=O)NC(c2ccncc2)CCO)cn1 54237,C#Cc1cccc(C(N2Cc3[nH]nc(CNC(=O)Cn4ccnn4)c3C2)=O)c1C 54238,C1(CNC(=O)CSc2ccccc2)OCC2CCN(C(=O)CC(F)F)CC12 54239,CC(F)(F)C(C)(C)CC(=O)NC(CNC(c1ccncc1Cl)=O)C(C)(C)C 54240,c1(C(N2CCN(C(c3cc(C)nn3C)=O)CC(O)C2)=O)cc2cc(Cl)ccn2n1 54241,C#CCCC(O)C(=O)NC1COCCN(C(c2ncc(C(F)(F)F)cc2Cl)=O)C1 54242,C(CCCCNC(c1c[nH]nc1-c1ccco1)=O)NC(C=CCOC)=O 54243,N1(C(C2CC(C#C)(O)C2)=O)CC(NC(c2c(C)ccnc2C)=O)C(N=[N+]=[N-])C1 54244,C1(C(=O)NC2CC=CC2)CC(O)CN1C(=O)CCc1csnn1 54245,C(C1CCCN1C(=O)CC1CC(OC)C1)=CC(=O)N(C)CC1CCN(CC)C1 54246,C(N=c1ccc(Br)c(S(=O)(=O)NCCC(C)O)[nH]1)c1nccc(C)c1F 54247,C(c1ccc(F)cc1Cl)=CC(N1C(CC)CN(C(c2noc(C)c2C)=O)CC1)=O 54248,C1(C(=O)NC(C)CC(N2CCCC2(C)CO)=O)CC1C1CCOCC1 54249,c1(C(=O)NC(C(=O)N(C2CCOCC2)C)CC2CC2)cccc(CC#N)c1 54250,N1(C(CC(C)C)C(=O)NCCN2CCOCC2)CC(C)(C)OC2(CCCOC2)C1 54251,c1(C(N2CC3(CN(C(CC(=O)NCC#C)=O)C3)C2)=O)cc(S(N)(=O)=O)cs1 54252,N1(C(CCC(CC)C)=O)CCCN(C(c2cnc(CC3CC3)s2)=O)CCC1 54253,N1(C(c2cc(CCC)n(C)n2)=O)CCC(C)C(NC(c2ocnc2CCC)=O)C1 54254,c1(-c2cc(C)c(OC(C)C)nc2)ccc2[nH]c(C(=O)NCCC3CC3)nc2c1 54255,C1(C(=O)NCc2cnsc2)(CNC(CC(C)n2ccnc2)=O)CCCCC1 54256,C(=O)(C(F)CC(C)(C)NC(c1ccns1)=O)NC1CCN(C)C1=O 54257,c1(C(N2CCC(N(C(C3CC3c3cnc[nH]3)=O)CC)C2)=O)ccc(Cl)c(F)c1 54258,c1(OC)ccc(F)c(C(F)(F)F)c1.C12(CC1C(=O)OC(C)(C)C)CNC(=O)OC2 54259,Cn1cc(Br)c(CC(=O)NCC2(O)CN(C(=O)C=Cc3ccccc3)C2)n1 54260,Cc1ccnc(C2(NC(=O)N(C(C)CS(C)=O)C)CCC2)n1 54261,CC1CCC(NC(c2cc(Cl)no2)=O)CN1C(=O)C(N1CCN(C)CC1)C 54262,[N-]=[N+]=NCCCOCC(=O)NC(C(=O)NCCC(O)C1CCC1)C1CCC1 54263,C(=O)(CCCCC(=O)N1CCN(C(c2cccc(OC)c2)=O)CC1C1CC1)NC 54264,CCCC(C)(O)CC(=O)N1CCCCC(CCC(=O)N(C)CC2CCOC2C)C1 54265,N1(C(c2nnn(C)c2N)=O)CC2CCN(C(C3CCCOC3)=O)C2C1 54266,CCCCCC=CCC(=O)NC1CCC1NC(CN(CC(=O)NC(C)C)C)=O 54267,n1(CC(N2CC(N(C)C)C2)=O)cc(CNC(=O)C(O)c2ccsc2)nn1 54268,N1(C(C(=O)Nc2ccc3nc(C)[nH]c3c2)=O)CCC2C(CCCN2C(C)C)C1 54269,n1(CCS(CC)(=O)=O)cc(C)c(=NC(=O)NCc2ccccc2N2CCOCC2)[nH]1 54270,c1(CC(N2C(CNC(C3CC(=C4CC4)C3)=O)CC2)=O)ccc(O)c(F)c1 54271,C1(NC(CSCC)=O)CCN(C(=O)CCCN2C(=O)CCC2=O)CC1O 54272,C1(N(C(=O)COCC2CCC2)CC#C)CCN(C(=O)Cc2csnn2)CC1 54273,C1(NC(CCCC=C)=O)CCN(C(C2CC3CCC2C3)=O)C(c2ccccc2)C1 54274,c1(CN(C(c2cccc(-c3nc(=O)o[nH]3)c2)=O)CC)c(F)cccc1Cl 54275,C(CCCC(=O)NCC1CN(C(C2CC2C(C)(C)C)=O)CCO1)SC 54276,CC1CC2CC2CC1C(=O)NC1CCC(C)N(C(=O)CCC2CCCOC2)C1 54277,C1(N(C(CC(=O)NCC)=O)C)CS(=O)(=O)C12CCN(C(C1CCCCC1)=O)CC2 54278,N1(C(c2ccc(OC)o2)=O)CCN(C(=O)C(C)SC(C)C)C(c2cccnc2)C1 54279,C(=O)(C1=NOC2(CCC2)C1)NCC(CC)NC(=O)Cc1ccc(Cl)nc1F 54280,C(CCCCCCNC(C1(CC)CCC1)=O)n1cc(COC(C)C)nn1 54281,C1(C(N2CCC(CC(C)NC(C(C=C)O)=O)CC2)=O)Cc2ccccc2C1 54282,c1(CC)cc(N)ccc1C(=O)NCC1CCC(NC(c2cnoc2C2CC2)=O)C1 54283,C(=O)(C(F)CC(C)(C)NC(=O)CC(C)(C)CN(C)C)Nc1c(CC)noc1 54284,C1(c2cc(C)cc(C)c2)CC1N=c1[nH]c(=NCCC(C)O)[nH]c2c1COC2 54285,c1(C(=O)NCC2N(C(CCC(C)OCC)=O)CCC2)ccc(S(N)(=O)=O)cn1 54286,C1(C(=O)NCC2CC(F)CN2C(C23CC(F)(C2)C3)=O)CCN(C2CC2)CC1 54287,N1(C(CSCCOC)=O)CCCCC(C2CN(C(c3cc(C(C)=O)cs3)=O)C2)C1 54288,Cc1n[nH]c2cc(C(=O)NC3CCCC3NC(c3ncccc3F)=O)ncc12 54289,c1(NC2CC(NC(c3ccc(F)c4occc34)=O)C2)c(Cl)cncc1[N+](=O)[O-] 54290,CC1CCN(CCOC(C2(c3ccccc3)CC3(CC3)C2)=O)CC1 54291,c1(CN(C)Cc2cc(C)no2)nc2c(c(=NCc3ncn(C4CC4)n3)[nH]1)CCC2 54292,Cc1cc(N2CC(F)(F)CC2CNC(C2CCC3CC3CC2)=O)ncc1C#N 54293,C1(C(=O)NC(CC(C)C)c2ccccc2)(CF)CCN(C(=O)OC(C)(C)C)CC1 54294,C1(OC)CN(C(=O)C(O)CNC(C2CC2C(F)F)=O)CC12CC2 54295,C(=O)(C1NC(C)(C)Cc2ccccc21)OC.c12ccc(cc1OC)C(=O)NNC2=O 54296,N1(C(=O)Nc2cc(C(N)=O)cc(Br)c2F)CCc2c(F)cccc2C1 54297,N1(C(COC)=O)CCC2(CCC(C(=O)NCC3(N4CCOCC4)CCCC3)C2)C1 54298,N1(C(C2C(C)CCC2)=O)CCCC(CCNC(=O)COCC2CCOCC2)C1 54299,c1(C(N2C3CC(NC(c4cncc(C)n4)=O)C(C3)C2)=O)cc(F)c(C)cc1Cl 54300,c1(NC)ncccc1C(N1CC(NC(=O)Cc2ccsc2Cl)C(C)C1)=O 54301,C#CC1(C(=O)Nc2ccccc2OC)CCN(C(c2ccnnc2)=O)C1 54302,C1(NC(c2ccc(C(N)=O)s2)=O)CC(NC(C2CCCC(CF)C2)=O)C12CCC2 54303,N1(C(C2C(C)C2C2CC2)=O)CC2CC3CC2C1C3NC(C1COCCN1C)=O 54304,n1(C(C)C)ncc(C(=O)NCC(C2CC2)NC(C2(O)CC2)=O)n1 54305,c1(CSCC(N2C3CC(NC(CSC)=O)C(C3)C2)=O)cn2cc(C)ccc2n1 54306,c1(C(=O)NCC(C2CCOCC2)(F)F)cc2c(s1)CCCNC2=O 54307,CC1CN(C(=O)CCOCCNC(=O)CC#N)CC1CO 54308,C(C(C(=O)NCC12CCC(CC1)CC2)C(C)C)NC(C(C(C)C)OC)=O 54309,N1(C(C(C)SCC)=O)CC2(CNC(c3cc(Cl)nc(Cl)c3)=O)CC1CO2 54310,c1(C(=O)NCC(CNC(c2cccs2)=O)OC)cc2ccc(F)cc2o1 54311,c1(OC)ccc2[nH]c(C(=O)NCC3CCN(C(=O)CC#N)CC3C)c(C)c2c1 54312,N1(C(Cc2n(C)ncc2Br)=O)CC(NC(c2cc3sccc3[nH]2)=O)CC(F)C1 54313,C1(NC(CCN(C(CCCOCCOC)=O)CC2CC2)=O)CCCN(C)C1C 54314,CC(C)CC(C(=O)NC(CC(C)(C)C)C(=O)N(C)Cc1ccnn1C)C(C)C 54315,C1(C(=O)NCCN(CCC)C(C2CC(OC)C(OC)C2)=O)CC(=O)N(C(C)C)C1 54316,c1(C(=O)NCCO)nc(Cc2c(C(=O)NCC(=O)Nc3ccco3)scc2)cs1 54317,C1(N(S(=O)(=O)Cc2ccc(F)cc2)Cc2ccccc2)CCc2ncnn2C1 54318,CN1C(=O)C(F)CC1C(=O)NCC1(NC(=O)CN2CCC(F)CC2)CCC1 54319,C1(NC(=O)C2CC2)CC2(CCN(C(C34CC(CO3)C4)=O)CC2)C1 54320,C1(C(=O)NC(C)CC(C)NC(=O)C(C)Oc2cccnc2)CCN(C(N)=O)CC1 54321,c1(-c2cnc(CC(=O)Nc3n(CC)ncc3)nc2)ccc2cncn2c1 54322,C1(O)(CNC(CC(CC)(F)F)=O)CCCN(C(C2CCCCCC2(F)F)=O)CC1 54323,O=C(CCCC(F)(F)F)NC1CN(C(C2(CO)CC2(F)F)=O)CC12CC2 54324,C(C1=CCCN(C)C1)NC(C(C(C)NC(c1cnc(N)cn1)=O)C)=O 54325,C1(N(C(Cc2nc(CC)sc2)=O)C)CCN(C(c2csc(=N)[nH]2)=O)CC12CC2 54326,N1(C(c2n(C(C)C)ncc2)=O)CCC(NCc2ncc[nH]2)C(F)C1 54327,CC1CC(C)N(C(c2nn3c(c2Br)CCC3)=O)CCN1C(=O)C1=CCCC1 54328,c1(N(C2C(OC)COCC2)C)ncnc2c([N+](=O)[O-])cccc12 54329,C1(c2nnnn2CCOC)(NCCOC(CC)(C)C)CCC(C(C)C)C1 54330,c1(C(CO)NC(C2(NC(COCC(=O)OC)=O)CC2)=O)cccnc1 54331,C(c1cn(C)nn1)=CC(=O)NC1(CNC(C2C(C)C2)=O)CC1 54332,C=C(C)C1CCC(C)=CC1CC(=O)NC1CCN(C(c2ccc(Cl)cc2F)=O)C1 54333,C(=O)(C1=CC(c2ccc(F)cc2)=NS(=O)(=O)N1)N(CC(=O)OC)C 54334,C1(O)(CNC(C2CCC2)=O)CCN(Cc2cccc(-c3ccccc3)n2)CC1 54335,C=C=CCCC(=O)NC(C1CCN(C(=O)Cc2cc(C)cs2)C1)(C)C 54336,N1(C(COC)=O)CCCC(C2N(C(=O)CN(c3n[nH]c(O)n3)C)CC2(C)C)C1 54337,n1(CC)cc(C(=O)NCC2(CC(=O)NCC3CC34CCC4)CC2)nn1 54338,Cc1ccc2c(C(=O)NCC(C)CNC(=O)CCc3ccc(F)nc3)coc2c1 54339,c1(C(N2C(CNC(=O)C3=CC(C)(C)C3)CCC(C)C2)=O)ccc2c(c1)CCC2 54340,Cc1cc(C(=O)NCCN(C(=O)C=Cc2cc[nH]c2)C2CC2)cnc1C 54341,C(=O)(C(C)(F)C(C)(C)F)N1CC(CN(C)C(c2cn3cnnc3cn2)=O)OCC1 54342,n1(CC)cc(Cl)c(C(=O)NCC2CCCN2C(c2sc(C)cc2C)=O)n1 54343,c1(C(=O)NCCCC2CCCN2Cc2sccc2Br)cc2ccccc2o1 54344,C(=O)(C(Cc1ccoc1)NC(c1ccc(CO)o1)=O)NC(C)CCN1CCCC1 54345,C1(=O)CCCCC(=O)N1.N1(C(CCC2(CCC#C)N=N2)=O)CC2(CO)CCC1C2 54346,CC(C)CC(C(=O)N1CCOCC1CC)ONC(c1ccc(CC2CC2)s1)=O 54347,C1(NC(c2ccc(Cl)s2)=O)CN(C(=O)C=Cc2cnc[nH]2)CC2CC12 54348,N1(C(C2(NC(C(COC(C)=O)C)=O)CCN(C)C2)=O)CCC2OCCC2C1 54349,CC1CC(C(N2CCCC2CNC(c2cccc(C3CC3)n2)=O)=O)CC(C)C1 54350,c1(CC(N2C(CNC(CC(C)SC)=O)C(C)CC2)=O)c(C)cc(C)cc1C 54351,C1(N(C(C(C)OCCOC)=O)C)CN(C(=O)Cc2ncc(Cl)s2)CCC1O 54352,C(c1cncc(F)c1)=CC(=O)NCC(C)N(C(=O)CC1CCS(=O)(=O)CC1)C 54353,CC(C)C(C)(CNC(c1cnc(S)n1C)=O)NC(=O)C(c1ccc(Cl)s1)C 54354,c1(CCC(=O)NCC(C)(C2CCC2)NC(C(C)OCCCC)=O)c(C)n[nH]c1C 54355,c1(COC)cnn(C)c1C#N.C(=O)(CC(O)CC1CNC1=O)OCC.[nH]1cc(CO)nn1 54356,C(CC(C)C)(C(=O)NC1CC2(C1)CC2NC(=O)CC1(CS(C)(=O)=O)CC1)OC 54357,C1(C(N2CC(CNC(c3ncccc3F)=O)C3(C2)CC3)=O)CC2(C1)CC(F)(F)C2 54358,N1(C(C(C)N(CC)CC)=O)CCC(NC(=O)C(CO)OC)C1C 54359,N1(c2nc(C)c(=O)n(C)n2)CCCC2(CCCO2)CC1 54360,C(CN=C(NCCN1CCCC1)NCc1ccco1)c1c(C)nccn1 54361,C(C1=CCN(C(c2cncc(Br)c2)=O)CC1)NC(C1(N(C)C)CCC1)=O 54362,C(=O)(C1CCCn2cnnc21)NC(CN(C(c1ccc(CC)nc1)=O)CC)C 54363,C1(C(N(CC(=O)OCC)C)=O)CC2CC2N1C(=O)CCc1nc(=N)[nH][nH]1 54364,Cc1nn(C)cc1C1CCCN1C(c1cnc(N(C)CC2CC3CCC2O3)s1)=O 54365,c1(C(=O)NC(C2N(C(Cc3c(C)n(C)nc3)=O)CCC2)C)nn(C)c2c1CCC2 54366,C(C(C)C)(C(O)C(=O)N1CCC(CF)(NC(=O)CN(CC(C)(C)C)C)C1)OC 54367,C1(C)(C(N(CCCC(=O)NCC(CC)(C)Cl)C)=O)CC(F)(F)C1 54368,C(=O)(C1=CC2CCC(C1)C2)NC(C)CC1CN(C(C2CC3CC3C2)=O)C1 54369,C1(C)(CNC(C(C)NC(c2cc[nH]c2)=O)=O)CCCC1 54370,Cc1ncccc1C(=O)N(CCCNC(C12CC(O)C1C2)=O)C 54371,N12CC(C3CCCCC13)CC2=O.C(=O)(C(O)CC1CC1)NC(C)(C)C 54372,CC1=C(CNC(=O)C(c2ccco2)NC(=O)OC(C)(C)C)S(=O)(=O)CCO1 54373,S(=O)(=O)(c1c(Cl)cc(Br)cc1Cl)N1CC(C)(C(=O)Nc2cc(Cl)cc(Cl)c2F)C1 54374,C12CC(C)(C1)NC2=O.C(=O)(C(N)=O)NCCCN(C)C 54375,N1(C(C2C(CCOC)C2)=O)CC23CCCC2(C1)CN(C(C1CCC(OC)C1)=O)C3 54376,C1(OCC)CCN(S(=O)(=O)N2CC=CC(N)C2)CC1 54377,c1(C(=O)NCC2N(C(C(C(=O)OC)C)=O)CC(C)(C)C2)cccc2c1cnn2C 54378,C1(C)(C(N(CC(=O)NCc2ccccc2)C)=O)CC(C#N)C1 54379,c1(NC(C(=O)NC(CC=C)CO)=O)ccc(OC(F)(F)F)c(Cl)c1 54380,N1(C(C(Cn2ccc(C)n2)C)=O)CCN(C(c2ncccc2O)=O)CC1C1CC1 54381,C(=O)(C(C)(C)C(N)=O)N1CCC(CN(C(c2c(NC)cncc2)=O)C)C1 54382,CCC(C)C(C)C(=O)NC1(C)CC(NC(c2cnn(CCO)c2N)=O)C1 54383,N1(C(C(C)SCC)=O)CCC2CN(C(=O)C=Cc3cnccn3)CCC12 54384,c1(C(=O)OC)cccc(C(=O)NCC(C)(C)CNC(=O)CCF)c1C 54385,c1(C(=O)NCC(C)N(C(c2nc(COCC)sc2)=O)C)ccc(C)c(F)n1 54386,CCC(C)(C)CCCC(=O)N(C1(C(=O)NCCOCCC2CC2)CC(O)C1)C 54387,C1(n2nc(C(N(CC(C)CNC(=O)CCF)C)=O)c(O)c2)CCC(F)(F)CC1 54388,c1(C(c2nnnn2C(C)CC)NCC(COCC)C)c(C)cc(Br)cc1C 54389,CCC(CNC(=O)CN1CCCS1(=O)=O)(CC)NC(=O)CC1C=CS(=O)(=O)C1 54390,CC(CNC(c1ccccc1O)=O)C(F)C(=O)NCc1c(F)cncc1F 54391,N1(C(C(C)=C2CCC2)=O)CC2CCC(CNC(c3n[nH]c4c3NCCC4)=O)(C2)C1 54392,C1(OC)(CNC(C2CC(CC(F)F)C2)=O)CCN(C(c2cnc(SC)n2C)=O)C1 54393,n1(CC(CC)NCC(C)CCCO)cccc([N+](=O)[O-])c1=O 54394,CCCCCC(F)C(=O)NCCCN(C)C(C12CC(C)(C1)OC2(C)C)=O 54395,CC1(C)CC(CCNC(=O)C(CC2CC2)NC(c2cncnc2)=O)CO1 54396,C1(C(=O)NCC2(NC(=O)Cn3cc(Br)cn3)CC2)CCC(=O)N2CCCC12 54397,Cc1coc2ccc(C(=O)N(CC(C)NC(c3cc(Cl)cc(F)c3F)=O)C)cc12 54398,c12nnc(N(C3COCC3F)C)n1C2.c1(CC)ccccc1 54399,N1(C(C2(C)CCN(C(c3cc(C)oc3C)=O)C2)=O)CCCC2C(O)CC12 54400,Cc1[nH]c2ncccc2c1CNC1COCCC1(O)CCCl 54401,C1(CCOC)(NC(=O)C(C)Cc2cnco2)CCN(C(=O)CSS(C)(=O)=O)CC1 54402,C1(C(=O)N(CC(C)C)C)(CC)CCN(C(=O)CCC2CCOCC2)C1 54403,c1(C(N2CC(C)(NC(C(C)CC(F)(F)F)=O)C2)=O)c(N)c(F)cc(F)c1F 54404,C(C(C)C)(C(O)C(=O)NC1CC(N(C(=O)CCc2cc(C)no2)C)C1)OC 54405,N1(C(c2ccn(CC)c2C)=O)CC(N(C(=O)CP(C)(C)=O)C)C2(CC2)C1 54406,C1(C)(C(N(CC=C)CCOC)=O)CN(C(C2CCC(C(N)=O)C2)=O)CC1C 54407,n1(CCC)nnnc1C(c1cc(C)[nH]n1)NCCc1cnoc1 54408,CC(CNC(=O)COCC1CC1)C(=O)NC(CO)CCC1CC1 54409,C1(C(=O)NCC(C)SC)C2CCC(C2)C1NC(C1(O)CC1)=O 54410,CCC(CC(=O)N1CC(=CCNC(=O)NC)OC(C)C1)C(F)F 54411,CCCC(CC)C(=O)N1CC2CC2(NC(c2cc(C(C)(C)C)c[nH]2)=O)C1 54412,C1(NC(CCSC)=O)CCN(C(c2ccc(CF)cc2)=O)CC1C 54413,C(=O)(C(CCCC(C)(F)F)N1CCC2CCOCC2C1)NCCOCC 54414,C(=O)(CN=c1cc[nH]cc1)N1C(C(=O)NCC2N(C(C)=O)CCC2)CCCC1 54415,C(=O)(C(C)C(=O)NC(C)C(=O)Nc1cncnc1O)OC 54416,C(=O)(C1CNC(=O)c2ccccc21)N1C(CNC(C2(C(C)C)COC2)=O)CCC1 54417,C(=O)(CCCCCS(N)(=O)=O)NC1C(NC(c2ccnc(OC)n2)=O)CCC1 54418,C1(CNC(c2ccc(F)cn2)=O)CN(C(=O)CNc2nccs2)C2CCN1C2 54419,c1(C(=O)NC2(C)CC(NC(c3ncc(OC)cn3)=O)C2)cc(C)cc(O)c1 54420,CC(CCCCCO)N=c1[nH]c(=NCCN2CCC2)c2ccccc2[nH]1 54421,c1(C(=O)NCC2CCN(C(C(CC)F)=O)C2)cc2cscc2s1 54422,Cc1c(Br)cnc(O)c1CNC(=O)NCc1cn(-c2ccccc2)nn1 54423,C(CCCCCF)NC(c1cncc(F)c1)=O.C12CCOC1CNC2=O 54424,c1(C(C)C)ncc(Cl)c(C(=O)NCC2CCN(C(C3CCC3C(F)F)=O)CC2)n1 54425,N1(c2ncc(C(=O)OCC)nc2)CCC(CNC(c2csc(NC)n2)=O)C(C)C1 54426,C1(NC(CC(C)NC(CCCCC)=O)=O)CCCCCC1F 54427,CC1=C(C(=O)NCCCCCCNC(c2ccc(F)c(C)c2)=O)CCC(C)(C)C1 54428,C1(C(=O)NC(C2CC=CCC2)C(=O)NC(CCCCC)C)CC(=O)CC(=O)N1 54429,C1(F)(CN(C(=O)Cc2cccnc2O)CC2CS(=O)(=O)C2)CCCCCC1 54430,CC1CCN(CC(=O)NC2CCCC(NC(C34CCCC3(C(N)=O)C4)=O)C2)CC1 54431,C(=O)(C(C)(C)C(=O)N1CCC(F)(C(=O)NC(C)CN(C)C2CC2)CC1)OC 54432,Cc1cc(C(=O)N(C2C3CN(C(C4CN(C)CCO4)=O)CC23)C)c(Cl)cc1F 54433,CC1Cc2ccc(C(=O)NCCC(=O)Oc3ccc(C#N)cc3)cc2CO1 54434,c1(C(=O)NC2N(C(C(C)Oc3ccc(C)cc3)=O)CC3CC32)cc(C#N)cn1C 54435,C1(C(N2CCN(C)C(=O)C2)=O)CC(C)(C)CCN1C(C1CN2CCC1CC2)=O 54436,N1(C(C(C)(C)C2CCCO2)=O)CCC=CC1C(=O)NC1(c2ccc(O)nc2)CC1 54437,N1(C(=O)Cn2cc([N+](=O)[O-])cn2)CC2(CCN(C(c3csc4nnsc34)=O)C2)C1 54438,C1(CC=C)(NC(c2c(C)noc2C)=O)CCN(C(=O)COCCOCCCC)C1 54439,c1(C(=O)NCC(CNC(=O)CCc2ncco2)OC)cnc[nH]c1=N 54440,N1(C(c2c(CC)cc(Cl)cc2)=O)CCC12CCCN(C(=O)C(C)NC=O)C2 54441,c1(-c2c(C(=O)NCCNC(C(COC)(C)OC)=O)cn(C)n2)cc(Cl)ccc1Cl 54442,CCC(C)C(O)CNC(=O)COC1CC(NC(C2(CC)CCCCO2)=O)C1 54443,N1(C(C)=O)CCOC(CCCC)C1.C12CN(C1)C(=O)CCNC1(CC1)C(=O)N2 54444,CC(C)CC(CC(C)C)C(=O)N1CCC(O)C(NC(C2CC(F)C(=O)N2)=O)C1 54445,c1(C(=O)NCC(CNC(c2cncc(C)c2)=O)C)sc2[nH]c(C)nc(=O)c2c1C 54446,CC1(C(=O)NCCCC2CCCN2C(c2cnc[nH]2)=O)CCCC1(F)F 54447,C1(C(C)C)(C(=O)NC2CN(C(c3coc(-c4ccsc4)c3)=O)C2)CCCO1 54448,c1(CCC)onc(C)c1C(N1C(C(=O)Nc2ncccc2OC)CC2CC12)=O 54449,C1(CC(=O)NC(C)C(C)NC(c2ccccn2)=O)CCCCC12CC2 54450,Cc1[nH]nc2c1CC(C(N1CCCC(F)(CNC(=O)C(C)(C)C(F)F)C1)=O)CC2 54451,N1(C(CN2CC(C)(OC)C2)=O)CC=C(C(=O)NCC2CCN(C(N)=O)C2)CC1 54452,c1(C(=O)NC(CNC(c2n[nH]c(C)c2Br)=O)CO)cccc2[nH]ccc12 54453,c1(C(N2CC3C(NC(CCCCSC)=O)(CCC3)C2)=O)cccc(S(N)(=O)=O)c1 54454,N1(C(C2CC(CCC)C2)=O)CC(C2CCN(C(C3CCCN(CC)C3)=O)CC2)C1 54455,c1(OC)csc(C(=O)NC2CCC(CNC(=O)CCCc3cccnc3)C2)c1 54456,CC#CCCCC(=O)NC(CNC(c1nnsc1C(F)F)=O)CC(C)C 54457,c1(C(=O)NCCCC2CCCN2C(C2CCC(F)(F)C2)=O)cccn2nncc12 54458,N1(C(C2CCC(C)(C)C2)=O)CCc2[nH]nc(CNC(C3CCOC3)=O)c2C1 54459,CC1CCc2onc(C(=O)NC3CC4C3CCN4C(c3cn[nH]c3)=O)c2C1 54460,c1(OC)cc(OC)nc(NC(C2CCN(C)C(=O)C2)=O)n1.N12CCC1C2=O 54461,c1(CC(=O)NCCC2CCN(C(CCCc3onc(C)n3)=O)C2)cccc(F)c1 54462,N1(C(C)=O)CCOC(C(=O)NC2CCC(N(C(=O)C=CBr)C)CC2)C1 54463,Cc1nn(C)c2c(N(C)CCn3cncn3)nc(=NC3CCCOC3)[nH]c12 54464,C1(CC2CC(CC)OCC2)C2CC3CC1CC(C(c1nnnn1C)OC)(C3)C2 54465,C(=O)(CC(C=C)CCC)N1CCC(N(C(=O)C(C)(C(C)C)OC)CC#C)CC1 54466,C1(C(=O)Nc2c(C)ccnc2)CN(C(c2cccc(Cl)c2I)=O)CC(F)(F)C1 54467,C1(CCC)CCCN(C(=NCCC2CCOC(C)C2)NCC2CC2)C1 54468,c1(C(N2CCCCC2CC=C)C(=O)NCC=C)ccccc1Br 54469,N1(C(C(c2cccc(F)c2)=O)=O)CCCC(CO)(NC(C2CC3C=CC2O3)=O)C1 54470,c1(C(=O)NCC(CC(C)C)NC(=O)CC2CN(C)C2)ccnc(C(F)(F)F)c1N 54471,Cc1[nH]c(C)c(C(=O)NCCN(C(=O)CCC(=O)N(C)C2CC2)CC(C)O)c1C 54472,N1(C(C(CCCC)F)=O)CCC2(CC(C(=O)N(C3CC(C(N)=O)C3)C)C2)C1 54473,N12CCCN(CC1)CCn1cc(nn1)NC(C)C2=O.C(C)(C)(CCCO)C(=O)O 54474,C1(NC(Cc2nc(C)sc2)=O)CCCN(C(=O)C(C)OC2CCCC(C)C2)C1C 54475,CCCC(CCC)CC(=O)NC1CC2CC1N(C(c1ccc(F)c(C)c1)=O)C2 54476,N1(C(CN(CCCC)C(C2(N3CCCC3)CC2)=O)=O)CC(C(=O)OCC)CC(O)C1 54477,C1(C(=O)NCCN(C(C(CCCC)O)=O)C(C)C)Cc2nccnc2C1 54478,c1(C(=O)NC2C(C)CN(C(c3cc4scnc4[nH]3)=O)C2)cnc2ccncc2c1 54479,c1(N2CCC(=CC)C2)cc(C)c(S(=O)(=O)N2CCOC(c3ccccc3)C2)cn1 54480,C1(CNC(CN(CCOC)C)=O)(NC(=O)C(C)CO)Cc2ccccc2C1 54481,CC(C)CC(CNC(=O)CC1CC2(CCC2)C1)NC(=O)CCc1cccc(Cl)c1 54482,N1(C(C2CC(C)(C)C2)=O)CCN(C(C2CCC(C(F)(F)F)CC2)=O)CC(O)C1 54483,N1(CCC(N2CCC(C)(NC(CC(CC)O)=O)C2)=O)CCSC(C)(C)C1 54484,Cc1cccc(CCC(=O)NCC=CCNC(C2CCCN(C)C2)=O)c1 54485,N1(C(c2cn(CC=C)nc2)=O)CCC(N(C(=O)C(N2CCCCC2)C)C)C(C)C1 54486,N12CC(C3(CC3)C1)C2.c1(SC)ccc(C(=O)N(CCC2CC2)C(C)=O)o1 54487,CC(C)C(CNC(C1CNC(=O)C1)=O)C(=O)NC1CCCCCC1CO 54488,c1(C(=O)NC2C(NC(C3C(OC)C3)=O)CCC2)csc2ccc(Br)cc12 54489,c1(C(c2nnnn2CCCSCC)NCCC(CC)C)nc(C)[nH]c1Br 54490,Cc1cc(C(=O)NCCOC2CCN(C(=O)CC(C)C)C2)c(C)n1C1CCOC1 54491,n1(CC)ncc2c1CC(CN(C(c1nn(C)cc1Cl)=O)C1CC1)CC2 54492,c1(OC)cc(OC)nc(C(=O)NC2CC3CC(NC(=O)C=C4CCC4)CC23)n1 54493,C1(CNC(CNC(c2cn(C)nc2)=O)=O)COC(CNC(c2ccsc2Cl)=O)C1 54494,N1(C(c2n[nH]c(CC)c2Cl)=O)CC(C)C(NC(=O)CN(S(=O)(=O)CC)C)C(C)C1 54495,C1(NC(=O)NCC23COC(C(c4ccc(C)s4)C4CC4)(C2)C3)CC1C1CCOCC1 54496,c1(-c2n(C)cnc2)cccc(F)c1C(N1CC(NC(C2CCO2)=O)CC(F)C1)=O 54497,CCC(C)C(O)C(C)C(=O)N1CC(OC)CC1C(=O)NCc1ccc(F)c(Cl)c1 54498,S(=O)(=O)(c1ccsc1C(=O)O)N.c1(CC2(Cl)C(C)(C)C2)ccc(NC)cc1 54499,C(CCC)(C(=O)N1CCCC1C(N1CCCC1CCCC)=O)=CCC 54500,c1(CNC(C(COC)O)=O)nc(CNC(=O)C(C)Cn2ccc(C)n2)cc(O)n1 54501,C1(CCC(=O)NC2CN(C(C(N)=O)=O)C2)CCC(=O)NC1 54502,c1(Nc2cccc(-c3ccc(C)cn3)c2)cc(N2CC(F)C(F)C2)nc(C)n1 54503,c1(-c2ccnc(N(C)Cc3n(CC)ccn3)n2)ccc(O)c(C)c1C 54504,N1(C(CN2CCN(CC)CC2)=O)CCC2CCN(C(C3CC=CC3)=O)CC2C1 54505,C#CCC(C(=O)NC(c1nn(C)cc1O)C)NC(=O)CCCCN(C)C 54506,Cc1nc2ccccn2c1C(=O)NCCC(C)NC(c1nc[nH]c2ncnc1-2)=O 54507,c1(C(=O)Nc2ccc(NC(C(COCC)C)=O)c(C)c2)c(C)[nH]c2ccccc12 54508,c1(C(=O)NCC2CCC2NC(=O)C(O)C2CCC2)ccc(Cl)c2cccnc12 54509,N1(C(c2cc(CCC)on2)=O)CC(NC(C2CCCC2(C)C)=O)C2(CCCC2)C1 54510,c1(C(=O)NCC(C2CCOC2)NC(c2cnccn2)=O)ccn2ccccc12 54511,C1(C(=O)NC(CC)CNC(C2(CC)CCC(O)CC2)=O)CCC2C(C1)C2(F)F 54512,C1(CNC(c2cnc(-c3ccccc3)[nH]2)C)CCCN(Cc2ccccn2)C1 54513,c1(C(=O)NCC(CCCC)NC(C2CC3(CC3)CO2)=O)ccc(O)c([N+](=O)[O-])c1 54514,C(C(C)CC(=O)NC1COCCC1NC(c1snc(Cl)c1Cl)=O)OC 54515,C1(C(=O)NCC2(COC)CCCN2C(C2CC(C)(F)C2)=O)CNC(=O)CC1C 54516,N1(C(Cc2ccc(C)c(C)c2)=O)CCC2CN(C(=O)CC(C)(C)O)CC2C1 54517,N1(C(CC(C=C)C)=O)C2CCC1CC(O)(CNC(=O)CC1=CCCC1)C2 54518,c1(C(N(CCCNC(C2(C)CC2Br)=O)CC)=O)c[nH]cc1COC 54519,C1(CC(=O)NCCC2CN(C(=O)C(C3CC3)SC)CCO2)(CO)CCOCC1 54520,c1(CC(=O)NCC(C)(C)NC(C2CCC(C(=O)OC)C2)=O)cc(F)ccc1OC 54521,CC1(C)CN(C(=O)C(C2CCCO2)NC(=O)OC(C)(C)C)Cc2ccccc21 54522,c1(OC)ccc(CCC(=O)NC2CCN(c3ccccn3)CC2)cc1 54523,C1(CC(=O)NCC2CN(C(c3c(C)snc3)=O)CC2C)CC(C)CC(C)(C)C1 54524,Cc1ccc(S(=O)(=O)NCC(N2CC3(C2)CN(C(C2CNC(=O)N2)=O)C3)=O)cc1 54525,C1(CC)CN(C(=O)COC2CCN(C)CC2)CCN1C(=O)C=Cc1ccc(C)o1 54526,C1(c2nnnn2C2CC(OC)C2)(NCCc2ccn(CC)n2)CCC1C1CCC1 54527,C12(C(N3CC(C)C(NC(c4cnn[nH]4)=O)C3)=O)CCC(C1)C2(C)C 54528,c1(OC)cc(CC(N2CCC(CN(C)C(C3C(C)CC3C)=O)CC2)=O)ccn1 54529,C1(NC(c2csc(S)n2)=O)CC(C2CCN(C(c3cccc4c3OCC4)=O)C2)C1 54530,C1(CNC(=O)COCCn2cccn2)COCCN(C(C2CC2CF)=O)C1 54531,C12(C(N3CC(CNC(Cc4cncc(OCC)c4)=O)C3)=O)CCCN(CC1)C2 54532,C1(NC(CCOCC)=O)CC2C1CCN2C(c1ccc(C(C)(C)C)c(Cl)c1)=O 54533,N1(C(c2c(CC)cc[nH]2)=O)C(C(=O)NC(c2snnc2C)C)CCC1C1CC1 54534,CON=CC(=O)NCC(O)CCNC(c1cn(CCCC#N)nn1)=O 54535,C1(C(=O)NCCOC2CN(C(=O)CO)C2)CC1C1CC(F)(F)C1 54536,c1(SC)ccc(OC(F)(F)CNC(c2cncc(C)n2)=O)cc1 54537,c1(C(=O)NCC2(C)CCCN2Cc2cccs2)c(Cl)cc(Cl)cc1Cl 54538,C1(C(=O)OC)(C(=O)NCCCC(C)NC(c2cccnc2CO)=O)CCCCC1 54539,N1(C(c2cc(CC)on2)C(=O)NCC(F)F)CCC(NC(C)=O)CC1 54540,CC1(C)CC(=O)N(CC(N2CCN(C(=O)CC3CS(=O)(=O)C3)CC2CCO)=O)O1 54541,c1(C(=O)NCCN(C)C(C2(c3ccccc3)CC2(F)F)=O)cc2cccn2cn1 54542,C(C(CO)CC(C)C)NC(C1(C)N(C(c2cc(C)sc2N)=O)CCC1)=O 54543,Cc1nc(NC(C)(CNC(C2(CC3CC3)CCCO2)=O)C2CC2)cc2nncn12 54544,C1(CNC(=O)CCc2cccs2)CCCN(C(C2CCC(F)(F)CO2)=O)CC1 54545,c1(OC(C(N2C(CNC(COC(C)C)=O)CC2)=O)C)ccc(Br)cn1 54546,c1(C(=O)NCC(CN(C(=O)CCC2CNC(=O)N2)C)(C)C)cn2ccccc2n1 54547,N1(C(c2nn(CC)c(O)c2)=O)CC(NC(=O)CNC(c2ccsc2)=O)CCC1C 54548,Cc1cc[nH]c1C(=O)NCCCCc1cn(C2CCCC2N)nn1 54549,c1(CC)ccc(C(N2CCC(CNC(c3coc(Br)c3)=O)C(C)C2)=O)cc1N 54550,Cc1nc(CNC(c2sccc2CNC(=O)C(c2ccnn2C)C)=O)[nH]c1C 54551,S(=O)(=O)(c1cccc(=NCc2nc(C(F)F)nn2C)[nH]1)NC1C(OC)C(C)(C)C1 54552,C1(C)(CC)CC(NC(c2c(OC)cccc2O)=O)CN1C(c1cnc(S)nc1)=O 54553,N1(C(C(C)(C)C2CCC2)=O)CCCC(C2CCN(C(C3(F)CC=CC3)=O)C2)C1 54554,C12(NC(c3cc4oc(Cl)cc4[nH]3)=O)CCCN(C(c3cc(Cl)on3)=O)CC1C2 54555,c1(-c2ccc(CNC(c3nccnc3Cl)=O)cn2)cnc2sccc2c1 54556,CC1COC2(CCC2)CN1C(=O)CSCCNC(=O)C(O)Cn1cncn1 54557,c1(CCOC)cc(C(=O)NCC2(CN(C(=O)CC3CCOC3)C)CC2)no1 54558,C(=O)(C1=C(Cl)CCOC1)N1CCC(C)(NC(c2cc(C)cc(O)n2)=O)C1 54559,C1(C2CC2)(C(N(CC(C)N(C)C(c2cc(C(N)=O)[nH]n2)=O)C)=O)CC=CC1 54560,c1(NC(C2N(C(C=CC=CC)=O)CCOC2)=O)ncc(I)nc1Cl 54561,CS(=O)(=O)CCC(=O)NCCC1(O)CCCN(C(C2CCC(C(F)F)CC2)=O)C1 54562,N#CC1(NC(c2ccc(I)cc2O)=O)CCN(C(c2ccc(Cl)nc2Cl)=O)C1 54563,c1(C(=O)NC2C(NC(CCCOCCOC)=O)C2)occ2c1CCC2 54564,Cn1ncc2nc[nH]c(=NC3CC(C(N4CCC(c5ccccc5)C4)=O)C3)c12 54565,CC(C)(CCC(=O)N1CC(C)(C(=O)NC2CCCCC2(F)F)CC1(C)C)[N+](=O)[O-] 54566,CC1CC(NC(=O)Cn2nnc(C3CC3)n2)CN1C(=O)CC1COCCO1 54567,c1(CC)cc([N+](=O)[O-])cc(S(=O)(=O)NC(c2cc3ccccc3o2)C)c1 54568,c1(OCC(=O)N(C(C(=O)NC2(CCOC)CC2)C)C)ccncc1 54569,C(C(C(=O)NCCc1cccc(C)c1)C(C)(C)C)NC(C(C)=C1CCC1)=O 54570,C(CC1CC1)(C(=O)NCCN1CC=CC1)NC(C1C(C)C1C)=O 54571,C(=O)(C(F)C(C)CC(C)(C)C)NCC1N(C(c2c(CC)occ2)=O)CC(C)(C)C1 54572,C(=O)(C1CCc2cccc(=O)n21)N1C(CNC(c2cn[nH]c2)=O)CCCCC1 54573,N12CC3C(C3C1)C2=O.c1(NCc2cnc(CC)s2)ccc(Cl)cn1 54574,N1(C(COC2CCCC(C)C2)=O)CCN(C(C23COC(CCO2)C3)=O)C(C)C1 54575,c1(C(N(C(C)C)CC2CCSC2)=O)cccc(NCc2nccn2C)n1 54576,C1(C(N2CC(=C)C2)=O)CC2CCCC2N1C(C1CS(=O)(=O)C1)=O 54577,c1(C(=O)NC(CNC(Cc2nnc(C)s2)=O)C(C)C)c(Cl)cnn1C 54578,c1(CC)cc(C(=O)NCC(C)CNC(=O)CCCC2CCOCC2)ccn1 54579,c1(-c2nn(CC=C)c(-c3cn(CC(F)(F)F)nn3)n2)cc[nH]c(=NCC)c1 54580,C(CC(=O)NC12CC(CNC(=O)C(c3cccc(C)c3)F)(C1)C2)(C(F)(F)F)OC 54581,c1(CNC(=O)NCc2n(COC)ncc2)cccc([N+](=O)[O-])c1C 54582,C1(C(=O)NCC=CCNC(C2(c3cccs3)C(C)C2)=O)CCC(F)(F)CC1 54583,C=Cc1cncc(C(N2CCC(NC(c3ncncc3F)=O)C(F)C2)=O)c1 54584,C=Cc1ccc(C(=O)NC2CC2CNC(=O)Cn2nnc(-c3ccco3)n2)cc1 54585,c1(N2CC(OC)(CNC(=O)CCc3nc(C)cs3)C2)cc(=O)n(C(C)C)c(O)n1 54586,N1(C(c2cc(OC)c(Br)cc2)=O)CC2(CCC(S(=O)(=O)C3CC3)C2)C1 54587,c1(Oc2c(CNc3cccc(OC)n3)cccc2)ccc(S(N)(=O)=O)cc1 54588,c1(OCC)nc(Cl)ccc1C(=O)NC1CCN(C(C2CC3(CCC3O)C2)=O)C1C 54589,c1(C(=O)NCC2CC(NC(C(C(C)O)N(C)C)=O)C2)cccc(OC(C)C)c1F 54590,C12(C(=O)NC(C(C)NC(C3CN(CCC)C(=O)C3)=O)(C)C)CCOC(C)(C1)C2 54591,C(=O)(CCCCC(=O)N1CCC(NC(=O)CCn2nc(C)c(C)c2C)C1)NC 54592,c1(C(N(CC(CNC(c2n(C=C)nnc2)=O)C)C)=O)cc(Br)ccc1O 54593,N1(C(=O)CC2CC2(Cl)Cl)Cc2ccccc2C(Nc2ncc([N+](=O)[O-])cc2Br)C1 54594,n1(C(C)C)cnc(C(=O)NCC2C(CNC(=O)C=Cc3ccsc3)C2(F)F)c1 54595,C=CCC(C(=O)N(CCCNC(c1cc(F)ccc1C(F)(F)F)=O)CC)C(C)C 54596,Cc1ccc(C(N2CC(NC(c3ccsn3)=O)C(O)C2)=O)cc1O 54597,Cc1cccc(C(=O)NCC2CCC(NC(=O)CSc3nncs3)C2)c1 54598,N1(C(C2C(C)CC(C)O2)=O)CCC2(CC1)CCN(C(c1cc(C#N)ccn1)=O)C2 54599,c1(OC)ccc(Cl)c(Cl)c1C(=O)NCC1CCN1C(C1CC1c1cccs1)=O 54600,O=C(C#CC1CC1)NC1CCCC1NC(c1cccnc1)=O 54601,C1(C)(C(=O)NCCN(C(=O)C(C(C)C)NC(N)=O)CC)CCC(C)=C(C)C1 54602,N1(C(CC2CCN(C)C2)=O)CCN(C(c2cnoc2-c2ccco2)=O)CC(O)C1 54603,N1(C(C)C)CCC(C(=O)NCC2CCCC2NC(=O)C2=CCOC2)CC1 54604,C1(NC(c2c(CC)cno2)=O)CN(C(c2c(Cl)cncc2Cl)=O)CCC1C 54605,N1(C(c2ccc(OCC=C)cc2)=O)CCC(F)C(NCc2ccc(I)cc2)C1 54606,C(CC1=CCN(C(C2CCOC2C)=O)CC1)NC(c1cc(C)sc1)=O 54607,C=C1COCCN(C(=O)C=CC(C)NC(=O)CC(C)n2cccn2)C1 54608,O=C(C1=CC2C=CC(C1)C2)NCC1CC(F)CN1C(=O)CSc1cccs1 54609,c1(C(=O)NCC2(NC(=O)COc3ccncc3)CC2)cnn(C2CC2)c1Cl 54610,C1(NC(=O)CCc2cccs2)CC2(C1)CC2NC(=O)CCCc1ncco1 54611,C(C(=O)NC(CC(=O)N(C)Cc1cc(OC)no1)C1CC1)(C(C)C)OCC 54612,c1(C(=O)NCC(C)CNC(=O)C(CO)N(C)C)cc2c(C(F)(F)F)nn(C)c2s1 54613,c1(C(C)NC(C2(O)CCN(C(c3cnc(Br)o3)=O)C2)=O)ccc([N+](=O)[O-])cc1 54614,C1(C)(NC(c2n(CCC)nnn2)c2ccc(Br)o2)CCC2(CC1)CC2 54615,N1(C(C(CC(F)F)NC(C(CSC)OC)=O)=O)CCC(F)(F)C(F)C1 54616,C1(C(N2CC(N(CC=C)C)C2)=O)CC(=C)CCN1OCC(=O)OC.C1(=O)CO1 54617,N1(C(CN(CCC)C)=O)CCOCC1CN(C(=O)C(F)C(C)C)C 54618,S(=O)(=O)(c1cccnc1C(F)(F)F)NC(CCN1C(C)C(C)N(C)CC1)(C)C 54619,O=C(C1=CCCOC1)NCC1CC1CNC(C1C(C2CC2)C1(F)F)=O 54620,N1(C(C(C)NS(CCC)(=O)=O)=O)CCC2(CC(NC(=O)CC3CCCCC3)C2)C1 54621,c1(C(=O)NCC(CC(C)C)NC(C(C)(CO)NC(C)=O)=O)cnc2cc[nH]c2c1 54622,C1(NC(c2onc(C)n2)C2CCOCC2)CCn2nnnc2C1 54623,C1(C(N(C2CCN(C(c3c(Cl)cn(CC)n3)=O)C2)CCO)=O)CC12CCCCC2 54624,c1(C(N(CCCCCNC(C2CCOC(C)(C)C2)=O)C)=O)cc2ccncc2[nH]1 54625,CC1(C)CCC(C(=O)NC2(CO)CC2)CN1C(C1CN(C2COC2)C1)=O 54626,c1(NC(CC)CC#N)ccc(S(=O)(=O)NCc2nocc2C(C)C)cc1C#N 54627,C1(C(N2C(CCCNC(CN3C(C)CC3)=O)CCC2)=O)CN2CCC1CC2 54628,C1(NC(C2CN(C(N)=O)C2)=O)CN(C(c2ccc3n[nH]cc3n2)=O)CC2(CC2)C1 54629,N1(C(c2n(CC)cc(Cl)c2)=O)CCC2(COC)CCCC12 54630,C1(CNC(c2cncc(Br)c2)=O)CCCCC1Nc1ncc(I)cn1 54631,O=S(=O)(c1ccc(=NCc2cccn3ccnc23)[nH]c1)NCC1(SCCO)CCC1 54632,C12(NC(C=CC(C)(C)SC)=O)CC(CNC(=O)C=CC(=O)NC)(C1)OC21CCC1 54633,C1(CNC(c2c(CC)[nH]nc2Cl)=O)CC2(CCC2)CN1C(c1ccncc1F)=O 54634,C(=O)(CS(=O)(=O)NC)NC1(CCN(C(C2(CCC=C)CC2)=O)C)CC1.COC 54635,C(=O)(C(C#N)C(C)(C)C)NC(C(NOCC(=O)OC)=O)C 54636,c1(C(N(C(C)C)CCN(C)C(c2cc(Cl)cnn2)=O)=O)ccc2c(c1)N(C)CC2 54637,C1(C)(C(=O)NC(CCNC(c2c(C)oc(C3CC3)n2)=O)C(C)C)CCCS1(=O)=O 54638,N1(C(CC(C)C)=O)CC2CCC(NC(c3occ4c3CCOC4)=O)CC2C1 54639,N1(C(c2ccc(Cc3nn[nH]n3)o2)=O)CCOCC1c1cccnc1O 54640,C1(CC)CC(C(=O)NC2COCC(C)(C)C2)CCN1C(C1CCC(=O)C1)=O 54641,C1(F)(C(=O)NCC2C(NC(C=NOC)=O)C2)CCCOC1 54642,CC1C(O)CC2CCC1N2C(=O)N(C1(c2cccc(Br)c2)CC(C(=O)O)C1)C 54643,c1(C(=O)NC(C(=O)NC(C=C)COC)Cc2cnc[nH]2)cc(C)nn1CC 54644,c1(OCC(=O)NCC2N(C(C(CC)=CC)=O)CCOC2)ccc(Cl)cc1Br 54645,c1(C(=O)NCC2N(C(C3N(C(C)=O)CC(O)C3)=O)CCC2)ccc(N)cc1Cl 54646,CON(C(=O)CCC1CCCN1C(C1C(C)(C)C1(F)F)=O)C1CCC1 54647,CCC(CC)(CO)C(=O)NC1CCN(C(=O)C(c2ccc(F)cc2)C)CC1 54648,C(CNC(=O)Cc1cc[nH]n1)(C(=O)N1CC(C(=O)NC2CC2)C1)N(C)C 54649,C1(CN(C(CC(C)N2CCOCC2)=O)C)CCN(C(=O)C(C)(C)C#N)CC1 54650,C(C(C)(C)C(=O)NC1CCCC1NC(=O)C(=C1CCCCC1)F)OC 54651,c1(C(N2CC(F)(CNC(C(CCC#C)O)=O)C2)=O)cc(F)c(F)c(Cl)c1F 54652,Cn1ncc(NCc2cccnc2P(C)(C)=O)c(Cl)c1=O 54653,c1(C2C(C(=O)NCCC(=C)CNC(C3CC3F)=O)CC2)ccc(Cl)c(Cl)c1 54654,c1(C(N(C2CCN(C(=O)C=CC(=O)OC(C)(C)C)C2)CC)=O)cc(=O)n(C)cn1 54655,C1(C(=O)NC2CN(C)CC2(C)C)CC2(CCCCC2)N1C(=O)OC(C)(C)C 54656,C1(COCC)CCN(C(c2nonc2C)C(=O)NCc2ccccc2)C1 54657,N1(C(=O)NCc2ccn(C(C)C)n2)CCN(C2CCCOC2)CC1 54658,N1(C(Cc2ccc(C)s2)=O)CC=CCC1C(N1CCCC1CCO)=O 54659,N1(C(c2ccc(CC)s2)=O)CCCC2CN(C(=O)Cc3ccc(C)c(C)c3)CC12 54660,c1(CC(N2CCC(N3CCN(c4nncs4)CC3)C2)=O)ccccc1Cl 54661,c1(C(C(=O)NC2C(NC(Cc3c(C)scc3)=O)C2)C)ccc(F)cc1 54662,c1(CCN=C(NCC2OCC(C)C2)NCc2ccccc2)c[nH]c2ccccc12 54663,C1(C=O)CC(OC)C1.c1(CNC(=O)N(C)C)csnn1.C1(=O)N(CCOC)CCN1.CO 54664,C1(CCC)CCCCC1NC(=O)C(C)(C)C1CCN(C(c2ccco2)=O)C1 54665,c1(OC)cc(C(N2CC3(CC(C(N4CC5C(C4)C5(F)F)=O)C3)C2)=O)cc(F)c1F 54666,C(C(C)C(F)C(=O)NCCCC1CC(C)C1)NC(c1c(C)cc[nH]1)=O 54667,C(=O)(C(CC)(CC)CC)NC1CCC(C(=O)NC(CCC=C)C(=O)OC)CC1 54668,N1(C(c2n(CC)ccc2)=O)CCCC(C)(NC(=O)Cc2ccc(OC)cc2C)C1 54669,c1(CC(=O)NCCn2ccc(NC(C3(OCC)CCC3)=O)c2)cnccc1C 54670,c1(C(N2CC(C)C(CNC(=O)Cc3csc(Cl)c3)C2)=O)cc(Cl)cc(F)c1N 54671,CC1CCCCC1CC(=O)NCC1(C)CC(C)(C)C1.C12CC(C1)NC2=O 54672,N1(C(C(CCSC)O)=O)CCOCC(C(=O)N(CCC(C)C)CC(C)C)C1 54673,C(c1cccc(Cl)c1)=CC(=O)NC(C(C)NC(COCC(=O)OC)=O)C 54674,C1(NC(C2(CC#C)CC2)=O)COCCC1C(=O)NC(c1ncc(C)cn1)C 54675,n1(CCN(C)C(=O)NC2C3CCC2(C)C3(C)C)cc(C#N)ccc1=O 54676,c1(C(=O)NCC2CN(C(CCCOC(C)C)=O)C2)ccc2ccc(Br)cc2n1 54677,N1(C(C2(C(=O)O)CCC(F)(F)CC2)=O)CCN(C2=NCCCN2)CC1 54678,C(C)(CCC(=O)N1CCC(C)(CCNC(c2cc(F)n(C)n2)=O)C1)SC 54679,C#CCCCC(C)C(=O)NCC(C(C)C)NC(=O)Cc1cccc(SC)c1 54680,C1(NC(CC2CN(C(C)=O)C2)=O)CC12CC(NC(c1cccc[n+]1[O-])=O)C2 54681,N1(CC2C(CCc3c(C)cccc3)CCC2)C(=O)NC2(CCC2)C1=O 54682,C(=O)(NNC(=O)C(C)OC(c1cn2c(OC)cccc2n1)=O)c1ccc(COC)o1 54683,C1(CC)CN(C(=O)CC2CC(C)=NO2)CC1NC(C1CCC(N(C)C)CC1)=O 54684,C1(NC(=O)Nc2c(N(C)C)ccc(C(N)=O)c2)CCNC12CCOCC2 54685,N1(C(CSC)=O)CCC(C)(CNC(c2c(C)coc2C)=O)C1 54686,C(=O)(CN=c1cc[nH]cc1)N1C(CCNC(C2(O)C(C)(C)OCC2)=O)CCCC1 54687,CC(C)C(O)C(C)C(=O)NC1CC(Cn2cc(-c3ccc(F)cc3)nn2)C1 54688,CC1(O)COCCN(C(c2cc(CNC(=O)C(c3ccccc3)F)no2)=O)C1 54689,N1(C(CCC#CC)=O)CC(NC(C2(SC)CCOCC2)=O)C(C2CC2)C1 54690,Nc1c(C(=O)NCCOCCCNC(C2CC23CC3(F)F)=O)cccc1Cl 54691,Cc1[nH]nc(Cl)c1NC(=O)N(C)Cc1cnn(C2CC2)c1C 54692,Cc1c([N+](=O)[O-])c(C(N2CC(NC(=O)C(=O)N(C)C)CC3(CC3)C2)=O)nn1C 54693,C1(CNC(=O)CCc2ccccn2)C(C2CC2)CCN1C(=O)Cn1cccn1 54694,c12ccc(c(C)c1)OC2.C(COC(=O)NC(C)(C)C)(CNC(=O)O)OC.OC 54695,C(=O)(C(=O)NNc1ncncc1Cl)NCc1[nH]c2cc(C)oc2c1 54696,c1(C(N2CCC(NC(CC(C=C)C)=O)(COC)C2)=O)nc2cccnc2s1 54697,C1(C2CC2)(CNC(c2ncc(Cl)cc2F)=O)CCN(C(C2(O)CCOCC2)=O)C1 54698,N1(C(c2ccc(N)c(C)c2C)=O)CCN(C(C23CCCCC2C3)=O)CC(C)(C)C1 54699,C(C(CC(=O)N1CCCC1CN(C)C)NC(=O)CC(C)CN(C)C)OC 54700,N1(C(c2cc(CCC)c(C)s2)=O)CC(NC(=O)CCNC(C)=O)C(C)(C)C1 54701,C1(c2noc(C(C3CCOCC3)OCc3ccccc3)n2)(OCC)CCCC1 54702,N1(C(C(CCC)CC)=O)CCCC2(C1)CN(C(C1(CCO)CC1)=O)C2 54703,C1(NC(C(CSC)O)=O)CC2CCC1CN(C(C1(F)CCCCC1)=O)C2 54704,c1(C(=O)NC(CC)CNC(=O)CCOC(C)=O)cnoc1CC(C)C 54705,N1(C(CC2N(C(C3ON=C(C(C)C)C3)=O)CC(O)C2)=O)CCCN(C=O)CC1 54706,O=C1NC2(CCO1)CN(C(=O)C(c1ccoc1)NC(C1CCC=CCCC1)=O)C2 54707,C1(C)(C(=O)NC2(CC)CC2)CC(O)CN1C(=O)C(CC1CCC1)OC 54708,CN1CCCC(CNC(C2CC(NC(c3cc(F)n(C)n3)=O)C23CCC3)=O)C1=O 54709,C(=O)(C(C)(F)C(=O)OC)NCC1(F)CC(NC(C(CC=CC)C)=O)C1 54710,C1(NC(CC2C=CC(NC(c3c(C)n[nH]c3)=O)C2)=O)CN(C(C)C)CC1C 54711,C(=O)(C(CO)C(C)(C)C)NCCC(C)(C)NC(CN(C)C(c1ccoc1)=O)=O 54712,c1(N2CC(O)(CNC(C(CCC)OC)=O)C2)ncc(C)c(SC)n1 54713,Cc1sc(C(N2CCC(CCC3CCCNC3)CC2)=O)c(Br)c1C 54714,c1(OC)cc(C(C(=O)NC(C)(C)C)N(C2CCC(=O)NC2=O)C(C)C)cc(F)c1 54715,c1(C(C)C)nccc(C(=O)NC(c2cccc(Cl)c2)CNC(C2CC2C)=O)n1 54716,NS(=O)(=O)c1ccc(C(=O)Nc2ccc(Br)c(C(F)(F)F)n2)cc1 54717,c1(C(N2CC(C(=O)Nc3cccc(O)c3Cl)C2)=O)c(O)ccc2ccccc12 54718,c1(CC)nc(C(=O)N(CCCNC(C2CC(F)CN2C)=O)C)c2ccccn12 54719,c1(C(N2C(C(C)NC(C3(C)CCC(=O)N3)=O)CCC2)=O)cc2nc[nH]c2cn1 54720,N12CCC(C(C)C1)Nc1c(cccc1)C2=O.N1(CCC=O)CCC(O)CC1.CN 54721,C(C(CNC(=O)CCc1cnn(C)n1)CO)NC(C1CN(C(C)=O)C1)=O 54722,N(C1CCCc2c(I)n[nH]c21)C(c1coc(C(F)(F)Br)n1)=O 54723,CC1(C)CCCC(C(=O)NCCCc2cn(C3CCCC=C3Br)nn2)C1 54724,c1(OC)cc(-c2csc(CO)c2)ccc1OC(F)F 54725,N1(C(c2nnc(C(C)C)s2)=O)CCN(C(=O)C2=CC3CCCC23)CCC1C 54726,C12(NC(C3C4CN(C)CC43)=O)CCC(NC(C3(C#N)CC4CC4C3)=O)(CC1)C2 54727,C(=O)(CCC(=O)C1CC1)NCC(C(C)NC(c1n[nH]cc1C1CC1)=O)CO 54728,c1(C(N(CC(N2CCN(C(C(C)C(C)O)=O)CC2)=O)C)=O)cc(F)c(Cl)cc1Cl 54729,C1(C(=O)NC(C2(CNC(C34CC(C)(C3)C4)=O)CC2)C)CCCC(C(F)(F)F)C1 54730,c1(C(=O)NC(CCNC(C2C(C=C)CC2)=O)(CC)CC)cnc2[nH]cc(C)c2c1 54731,c1(CC(=O)N(CC(O)C(=O)N2CC(OCC(F)F)C2)C)ccc(O)cc1 54732,c1(CCCSCCNC(N2CSCCSC2)=O)ccc2ccccc2c1 54733,N1(C(c2cc(C)sn2)=O)CCC2(CCN(C(c3cc(F)c4cn[nH]c4c3)=O)C2)C1 54734,c1(CNC(C(C)N(C(=O)CSC)CCC)=O)ncc(C)cc1C 54735,c1(N(CCNC(=O)CC(C)C2CCCCC2)CC)ncnc(Cl)c1Br 54736,N1(C(c2c(C)cccn2)=O)CCCC(NC(C2CSCCS2)=O)CC1 54737,N1(C(C(=O)N(CCC(C)C)C)C)CCC(NC(c2cnco2)=O)CC(C)(C)C1 54738,C12(C(N3C(CCNC(Cc4nc(C)oc4)=O)CCC3)=O)CCC(F)(CC1)C2 54739,C1(C(=O)NCC(N(C(=O)CO)C)C2CC2)C2CC3C(C2)C13 54740,c1(C(=O)NC2C3CN(C(CC4(C)CCCO4)=O)CC2C3)c[nH]c2nccc-2c1 54741,C1(NC(c2n(C)c(=O)ccc2)=O)COC2(CCN(C(=O)C=Cc3cscn3)C2)C1 54742,C1(CN(C)CCC2C(CC)CCCC2)CC12CCOCC2 54743,n1(CC=C)nnnc1C(c1csc(Br)n1)NC(c1nnc(CO)s1)C 54744,c1(C(=O)NCC2N(C(c3cc(C)c(N)cn3)=O)CC2)ccc(S(N)(=O)=O)cc1 54745,O=C(CS(=O)(=O)C1CC1)NC1COC2(C1)CN(C(c1cnc3cccnn13)=O)C2 54746,Cc1nc(NCCC2CCSC2)cc(=NCC(C(C)(C)C)N(C)C)[nH]1 54747,C#CCCCCCNC(=O)C(CCC1CCC1)NC(C1CC1C(N)=O)=O 54748,S(=O)(=O)(c1ccc(NCCCCn2cnnc2)cc1Br)N(CCCC(=O)NC)C 54749,C(=O)(CC(O)(c1ccccc1)C1CC1)N1CC(n2cc(CC(C(C)C)O)nn2)C1 54750,N1(C(C2N(C(C(CC)C(F)(F)F)=O)C3C(C2)C3)=O)Cc2ccnn2CC1C 54751,CC1(C)C(NC(=O)CC(F)(F)F)C(C)(C)C1NC(=O)CC1(C(F)(F)F)CCC1 54752,C1(C(=O)NC(C)(C)CS(C)(=O)=O)CN(C(=O)CCC2CCOC2)CC12CC2 54753,CC1(C(=O)NCC2CCN(C(=O)CCCc3ccccc3Br)C2)CC(F)(F)C1 54754,Cc1c(N2CCOCC2)ncnc1N1CCC(NC2COCC2C)CC1 54755,C1(C(=O)Nc2cccc(OC)c2)CCCN(C(=O)C=CCF)C1C 54756,C1(COC)(CNC(C2CCC(C)CC2)=O)CCCN1C(=O)CCOC1CCOC1 54757,c1(NC(C(CCOC)NC(=O)C(=O)N(C)C)=O)cn(CC)nc1C#N 54758,c1(C(N2CC(C(C)NC(c3cc(C)ns3)=O)C2)=O)c(C)ccnc1O 54759,c1(C(N2CCC(CC#N)C2)C(=O)NC)cccc(Cl)c1F 54760,S(=O)(=O)(CCC(=O)NCC1C=CC(NC(=O)C(c2ccccc2)O)C1)NC 54761,c1(CNC(c2c(CC)cc[nH]2)=O)ccc2c(c1)CCN(C(c1c[nH]nc1C)=O)C2 54762,c1(NC(C2CC2C(N2C3COCC2C3)=O)=O)cnc(I)cn1 54763,N1(CCC)CCCC(C(=O)NC(C)CCNC(c2cc(CC)no2)=O)C1 54764,C(N=c1[nH]c(=NC2CCCCCC2F)c2ccccc2[nH]1)c1nc(C)c(C)[nH]1 54765,c1(C(=O)NCCC2N(C(CCC#CC)=O)CCC2)ccc2c(c1)OCCO2 54766,Cc1nc([N+](=O)[O-])cn1CCC(N1CC(NC(C2(C)CC(C)(C)C2)=O)CC1C)=O 54767,c1(C(=O)NC2C(OC)CN(C(c3ccc(F)c(N)c3)=O)C2)cc2c(s1)CCCC2 54768,Cc1cn2c(CC(N3CCC(CNC(C4(C)C(C)(C)C4(C)C)=O)C3)=O)csc2n1 54769,c1(C(N2CCCC(C(C)NC(C(COC)NC(C)=O)=O)C2)=O)cnc(Cl)c(N)c1 54770,c1(C(N(C)CC2CCN(C(CCCC#CC)=O)C2)=O)cnc2c(c1)CCCC2 54771,C1(CNC(CCC(=O)N(C)C)=O)CC2CCCC2N1C(=O)CSCc1ncc[nH]1 54772,Cc1cc(C)c2[nH]c(C(=O)NC3CC(NC(=O)COCC4CCCO4)C3)cc2c1 54773,c1(C(=O)NCCCN(C(C2(O)CCC(CC)C2)=O)CC)cccc2c(C)[nH]nc12 54774,c1(C(=O)NC(c2c(C(N3CCC(C(C)C)C3)=O)con2)C)ccc(O)nn1 54775,C1(=CC(=O)NC(C2(O)CN(C(=O)C=CCCc3ccccc3)C2)C)CCSCC1 54776,c1(C(=O)Nc2nc(Cl)ccc2Br)c[nH]c2cc(-c3cnn(C4CCC4)c3)cnc12 54777,C1(NC(c2cc(CNC(C(CC)=CCCC)=O)no2)=O)CC(C)(C)OC1=O 54778,Cc1ncc(Cl)c(C(N2CCC(NC(c3cc(O)ncn3)=O)CC2C)=O)n1 54779,c1(COC(F)(F)F)c([N+](=O)[O-])cnn1C.c1(CC(=O)N)cncn1C1CC1.CC1CN1 54780,C1(C(=O)NC2(C(N(CC(CC)(C)OC)C)=O)CC2C)CC(C#N)(OC)C1 54781,Cn1cc(C2=CCCC2)cc(C(N2CC(CO)CC(F)(F)C2)=O)c1=O 54782,C1(C(N2CCC(C)C2CNC(c2cn(C)cc2C(F)(F)F)=O)=O)CC2(C1)CC2(F)F 54783,C1(C(N2CC(CCCNC(c3c(OC)n[nH]c3)=O)OCC2)=O)OCCN(C)C1=O 54784,n1(CC(=O)NC2C=CCN(C(c3n(CC=C)ccn3)=O)C2)ncc2ncccc12 54785,c1(OC)c(F)cc(C(=O)NC(C)(C)C(C)NC(=O)CC2CC=CCC2)c(N)c1F 54786,c1(C(=O)NC23C(CN(C(c4cc(C)n(C)n4)=O)C2)CC3)coc2c1C(=O)CCC2 54787,c1(C(N2CCC(C(C)NC(c3cc(CCO)on3)=O)CC2)=O)ccc(O)cc1Cl 54788,C1(NC(C(C=C)(C)O)=O)CN(C(c2ccncc2N2CCCC2)=O)CC(C)(C)C1 54789,c1(CC)ccc(C)c(NC(C2CCC(C)N2C(=O)CCC2CC2(F)F)=O)c1 54790,N1(C(CCN(C(CCC(C)CN(C)C)=O)CC2CC2)=O)CCOCC(C)(O)C1 54791,CCC(C(=O)N1CCC(CNC(=O)CC2CCC(F)(F)CC2)C1(C)C)C(C)(F)F 54792,C(N=c1[nH]c(N2CCCC3(CC2)CC3)nc2cc[nH]c12)C1(F)CC1 54793,C(C1CCCN1C(=O)CC1CC1)=CC(=O)NCC(C)C1CCC1 54794,c1(OCCC)ccc(CNC2(CC)CCNC2)cc1C 54795,C1(C(=O)NCC2(NC(=O)C(c3ccc(F)cc3)F)CC2)CC2CCCC(C1)C2 54796,N1(C(C2C(C)CCO2)=O)CCC(F)(C(=O)NC2(C)CCCC2O)C1 54797,Cn1cc(C=CC(c2ccc(OC(F)F)cc2)=O)cn1 54798,C1(CNC(c2ccc(F)cn2)=O)C(C2CC2)CCN1C(=O)COCC(F)F 54799,c1(C(=O)NC2CCC(NCC3CN(S(C)(=O)=O)C3)C2)cc(OC(F)F)nc(Cl)c1 54800,C(C1c2ccsc2CCN1C(=O)COCC(C)C)NC(CCCCCCC=C)=O 54801,C1(CC)(CC)CCC(NC2(c3nnnn3C)CCOC2)CC1 54802,C1(N(C(=O)C(F)CC2CN(C(C)=O)C2)CC)CCCN(C(=O)Cc2cn[nH]c2)C1 54803,Cc1c(CNC2C=CC(C(=O)Nc3ncccc3F)C2)[nH]c2ccccc12 54804,C(=O)(C1=NOC(C)C1C)NCCCC(C)NC(c1ccc(C)cn1)=O 54805,C1(CC(=O)NC(C)CC2CC2)CCN(C(C23C(=O)C4CC2C3C4)=O)C1(C)C 54806,C1(C(C)C(=O)NCC2(O)CN(C(C3CCCC(F)(F)C3)=O)C2)CCC(C)(C)CC1 54807,N1(C(C2CCC(CC)CC2)=O)CCC2CCN(C(C3CC(F)C3)=O)CC12 54808,c1(C(=O)NCC(C(=O)N(C2CC2)C2CC2)OC)ccc(CO)cn1 54809,C(CC(=O)N1CCC(n2ccnn2)C1)(CC(C)C)NC(CC(CCC)C)=O 54810,Cc1csc(CN(C(=O)C(c2ccnn2C)NC(=O)CCOCC(F)F)C)c1 54811,N1(C(C(CO)OC)=O)CCC(C(=O)NC2CC3CCC2C3)(C(C)C)C1 54812,C(=O)(CCCCC(C)CC)Nc1c(CC)cc(C(F)(F)F)cc1.N12CC(C1)C2=O 54813,c1(C(=O)NCC(CN(C(=O)C=CCN2CCCC2)C)O)cc2sc(Cl)cc2s1 54814,c1(C(N2CCCC(CNC(C(CC)CN(C)C)=O)C2)=O)ccc(C)nc1C 54815,c1(C(N2CC(O)(CNC(c3cc(Cl)cc(Cl)n3)=O)C2)=O)cc(Cl)cc(Cl)c1O 54816,c1(C(N(C(CNC(C=C(CCC)C)=O)C2CC2)C)=O)ccnn1CC 54817,c1(-c2cn(-c3ccc(NC(C(C)CN)=O)cc3)nn2)cc(F)ccc1Cl 54818,CC1(CNC(=O)CCN(C(c2ccc(C3CC3)o2)=O)CC2CC2)CCCCC1O 54819,c1(C(N2CCN(C(C3CCC(OC(F)F)CC3)=O)C3CC23)=O)nnc(O)cc1O 54820,Cc1c(C(N)=O)cccc1C(N1CC2(CCC2NC(C2C3CC4C(C3)C24)=O)C1)=O 54821,N1(C(c2cc(CNC(CCCN(C(C)C)C)=O)on2)=O)CCOC2CN(C)CC12 54822,N1(C(c2ccc(CCCC)cc2)=O)CC2CCN(C(=O)CCC3CC3OC)CC2C1 54823,CC(C)(C)CC(O)CC(=O)NCCC1(O)CN(C(c2cc(CCO)on2)=O)C1 54824,CCC(CC)(CCNC(=O)CC1CC2(CC2)CO1)NC(c1cnn(CCF)c1)=O 54825,C1(CNC(CC=CC=C)=O)(CO)CCCN(C(=O)C(F)C2CCOC2)C1 54826,C1(N(CCC(=O)Nc2csnc2CC)C(c2c(CCC)nco2)=O)CCCCCC1 54827,C1(CCC(N2C(CNC(c3c(C)coc3)=O)CCC2)=O)CCCCN1C 54828,CCC(C#N)C(=O)N1CC(F)CC1CN(C(=O)COCCF)C 54829,N1(C(CSCC)=O)CCC2(C1)CN(C(=O)C(C)C(C)O)CCO2 54830,n1(CC)cc(C(=O)NC2CCC(CCNC(=O)Cc3cc[nH]c3)C2)nn1 54831,N1(C(Cc2n(C)ccn2)=O)CCC2CN(C(C3OCC4CCCCC34)=O)C2C1 54832,Cc1nc2ccc(C(N3CC4(CC(C(=O)N(CC(N)=O)C)C4)C3)=O)cc2o1 54833,N1(C(CNc2nccc(OC)n2)=O)CCOCC(NC(C2CCOC2C)=O)C1 54834,CCC(C)(CC)C(=O)NC(C1CCN(C(=O)C(=O)Nc2cccc(C)c2)CC1)C 54835,C1(NC(N2CC(COC)OC(C)(C)C2)=O)CCc2cc(OC)ccc2C1 54836,CCC(CCC(=O)N(CCC(=O)NC1CCN(C(C)C)CC1)C1CC1)OC 54837,c1(CC)cc(C(=O)NC2CCCC2CC(=O)NC2(CC)CCC2)on1 54838,C1(NC(C23OCC(COC)(C2)C3)=O)CCCCN(C(=O)C(C(C)O)N(C)C)C1 54839,N1(C(CCc2ccc(C)nc2)=O)CCC2(CC(NC(C3(C)CCOCC3)=O)C2)C1 54840,c1(CC)nn(C)cc1CNC(=O)Cc1nncs1 54841,N1(CCCNC(C=C(CC)C)=O)CCN(C(c2ncoc2C2CCCO2)=O)CC1 54842,C1(NC(c2cnc(C(C)(C)C)s2)=O)CC(F)(F)CC1NC(=O)C1=CCSC1 54843,Cc1cc(CC(=O)NCC2(F)CC(NC(=O)C(C)(C)NS(C)(=O)=O)C2)n(C)n1 54844,O(NC(=O)CCCN(C(=O)C(C)CNC(N)=O)C(C)C)CC=C 54845,c1(-c2cn(CC(CCN(C(CC)C(=O)OC)CC)F)nn2)c(C)cccc1Cl 54846,N1(C(c2cccc(C#C)c2)=O)CCC(NC(=O)C(CO)NC(N)=O)C(F)(F)CC1 54847,N1(C(C(C(=O)NC)(C)C)=O)CCN(C(=O)CCNC(C2CCCO2)=O)CC(O)C1 54848,CCCC(CC)CC(=O)N1CCN(C(c2c[nH]nc2-n2cnnn2)=O)CC1C 54849,C1(O)(C(COC)C)CCCN(C(=O)NCCCc2nc3c(s2)CCC3)C1 54850,C(N=c1nc2c(cnn2C)c(NC2CC(N(C)C)C2)[nH]1)c1cc(C)c(Br)cn1 54851,N1(C(C2C(CC)CCO2)=O)CC(S(=O)(=O)N2CCN(C(C3CC3(F)F)=O)CC2)C1 54852,c1(C(=O)NCC(CC)NC(=O)C(F)NC(C)=O)ccc2c(c1)CCCN2C(C)=O 54853,N1(C(C23C(CN(C(C4(C(=O)OCC)CC4)=O)C2)C3)=O)CCCC(OC)CC1 54854,N1(C(c2nc(CC)[nH]n2)=O)CCC(C2CCCCN2C(c2scnc2Cl)=O)CC1 54855,c1(C(=O)NC2CC(F)(CNC(C3CC(C)N(C)C3)=O)C2)cccc(S(N)(=O)=O)c1 54856,Cc1c(C(=O)N(CC(C)NC(=O)COc2ccc(OC)cc2)C)cc(O)cc1N 54857,C1(C(N(CC(N2CCC2C2CCCC2)=O)C(C)C)=O)CCCC(=O)N1 54858,C1(C(=O)NC2CC2CNC(=O)C=CC2CCCC2)(COC)CC=CC1 54859,C1(N(C(Cn2cc(-c3cccc(C)n3)nn2)=O)C)CCCCC1(C)C 54860,C1(CN(C2CCCN(C(C)=O)C2)C(=O)C=Cc2cncs2)OCCOC1(C)C 54861,n1(CC(=O)NC2CCN(C(C(C)CF)=O)CC2O)nc2n(c(=O)c1=O)CCOC2 54862,c1(C(=O)NCCSCC(=O)NC(C(CC)(F)F)(C)C)cc2ccccn2c1 54863,C(CNC(=O)Cc1csc(Cl)c1)(C(C)C(C)C)NC(Cc1cnc(C)[nH]1)=O 54864,C(=O)(CCCC(C)NC(=O)CCc1cccs1)NCC1N(CC)CC1 54865,c1(OC)cccc2c(NC3CCC(OCc4ccccc4)C3)c([N+](=O)[O-])cnc12 54866,N1(CC(=O)NC)Cc2ccccc2C1=O.C1(=O)C(CC2CC2)ON1C 54867,C1(NC(c2nc(C)oc2)=O)C(C)(C)C(NC(c2ccc(O)c(C)c2C)=O)C1(C)C 54868,C(C)(CC(C)NC(=O)Cc1cncs1)NC(CN(CCOC)C)=O 54869,C1(NC(C(COC)(C)C)=O)CCN(C(c2cccc(CCN(C)C)c2)=O)C(C)C1 54870,C=C(C)CC(C(=O)N(C)Cc1cccnc1O)NC(=O)Cn1cccc1 54871,Cc1nsc(N)c1C(=O)NCC1(C)CCCN1C(=O)Cc1nc(C)c(C)[nH]1 54872,C1(NC(C(=Cc2cn[nH]c2)C)=O)CC(C)N(C(c2nnsc2N)=O)C1 54873,Fc1ccsc1C(c1cn[nH]c1)NCc1cccs1 54874,N1(C(c2n(C(C)C)ccc2)=O)CCN(C(=O)CCc2nccn2C)CC12CC2 54875,c1(NC(c2cccnc2)CC)nc(N2CCN(CCO)C(C)C2)nc2sccc12 54876,c1(C(N2CCN(C(C(C)SCC)=O)C(CCOC)C2)=O)cc2ccsc2c(O)n1 54877,CC(C(=O)NC1CC(CCn2cc(-c3ccncc3F)nn2)C1)C(F)F 54878,N1(C(C2N(C)CCC2)=O)CCCC2C1CCN2C(c1cc(Cl)ccc1[N+](=O)[O-])=O 54879,c1(N(CCC(=O)NC2CCN(C)CC2)C)cc(Cl)ccc1-c1nn[nH]n1 54880,C1(CC(=O)NC(CN(C(=O)CC2CCC(=O)NC2)C)(C)C)NC(=O)CNC1=O 54881,N1(C(c2c(CC)nccn2)=O)CCCN(C(=O)C(O)Cn2cncn2)C(C)C1 54882,CCCC(C)(CCC)C(=O)NC1COCC1CNC(=O)C=Cc1ccoc1 54883,C(C1=CCCN(C)C1)NC(COC1CCN(C(c2cc(OC)ns2)=O)C1)=O 54884,CCC(F)(C(=O)OC)C(=O)NC(CCNC(=O)CCC(=O)N1CCCC1)C(C)C 54885,C(=O)(CCCC(F)(F)F)N1CC(CC(=O)Nc2cn(CC)nc2)(OC)C1 54886,C(CC1=CCN(C)CC1)C(=O)NC(C(N(OC)C)=O)C 54887,C1(C(N(CCN(C(c2c(CC)nc[nH]2)=O)C)C(C)C)=O)C2CCCCCCC12 54888,CC1(C)CC(CNC(c2cnc(=N)[nH]c2)=O)N(C(=O)C(N)=O)C1 54889,C1(C(N(CC(N)=O)C)=O)CC2(CCC2)CN1C(C1CSCC(=O)N1)=O 54890,C(=O)(C#CC1CCC1)NCC(CC=C)NC(=O)Cc1cccc(C(N)=O)c1 54891,C1(NC(CC=C=C)=O)CN(C(c2nn(C)cc2C)=O)CC1C(F)(F)F 54892,N1(C(CSC(C)(C)C)=O)CCCC1C1CCCN1C(c1ccc(F)s1)=O 54893,N1(C(C23CC(NC(CC4CC(=C)C4)=O)(C2)C3)=O)CC(C)CC(C)(C)C1 54894,CCC(C)(C(=O)NC1CC(C)N(C(=O)C(=O)NOC)C1)c1ccccc1 54895,Cc1onc(-c2ccccc2)c1C(=O)OCCn1cnc(C#N)n1 54896,C1(NC(CC(C(F)F)NC(C=CC(C)C)=O)=O)CCn2ncnc2C1 54897,c1(OC(C(N2CC(O)(CN(C(c3c(CC)cco3)=O)C)C2)=O)C)ccc(O)cc1 54898,c1(C(=O)NC(C(=O)NC(CCC)C)C2CCOC2)oc(C)nc1CC 54899,c1(C(=O)NC2CC(C)(NC(C3CN4CCN3CC4)=O)C2)cccc([N+](=O)[O-])c1N 54900,C1(C(N2CCC(N(C(Cc3ncc(CC)[nH]3)=O)C)CC2)=O)CCCCNC1=O 54901,N12CC(O)CC1(C)C1CC1C2=O.C(C(C)(C)[N+](=O)[O-])n1cc(C2(C(C)OC)CCC2)nn1 54902,C1(NC(C(CC)C#N)=O)(CO)CCCN(C(C2CC3CC(=O)C2O3)=O)C1 54903,c1(CCC(=O)NC)cn(C)nn1.C(=O)(CCOCCCCCN(CCO)CC)N 54904,C1(COCCC)(CNC)CCN(C(C2CC(OC(C)C)C2)=O)C1.C1CCC(=O)O1 54905,N1(C(C(C)OCC(C)C)=O)CC2CC(NC(c3ccncc3)=O)CC1C2 54906,c1(C(CC(=O)NCC(CNC(c2c(CC)occ2)=O)(C)F)O)cccc(F)c1 54907,C12(NC(CC3(C=C)CN(C(c4cnn(C(C)C)c4)=O)C3)=O)CCC(CC1)C2(C)C 54908,C1(C(N(CCNC(=O)CSC2CC2)CC)=O)CC(=O)C1C 54909,Cn1cc(-n2cc(C3(O)CN(C(=O)CNC(c4ccc(Cl)s4)=O)C3)nn2)cn1 54910,C1(NC(C2C(CC)OCC2)=O)CC2CCC1CN2C(C1CCC(C)CC1)=O 54911,c1(CC(=O)N(CC(C)NC(COCCC)=O)CC)ccc(C)nc1 54912,c1(C(N2C3CN(c4nccc(C)n4)C(CC3)C2)=O)cc(Br)c2ccccc2n1 54913,C(=O)(C1CN(C)C(=O)c2ccccc21)NC(C)CNC(=O)C=CCF 54914,c1(NC)cnccc1C(=O)NCCCN(CCO)C(C1CCC1OC)=O 54915,C1(C2CCN(C(c3ccc(S(C)(=O)=O)o3)=O)C2)(NC(CS(CC)=O)=O)CC1 54916,C1(NC(C(C=C)(C)CC)=O)CC2CN(C(=O)C(CCC)C(C)C)CC2C1 54917,C(C1=CCCN(C(c2ocnc2C2CC2)=O)C1)NC(C1CCC(C)(CC)O1)=O 54918,CN1CCCN(C2CC3CC2CN3C(c2cccc(C3CC3)c2)=O)CC1 54919,C(CNC(c1c(C)n[nH]c1C)=O)(C(C)(C)C)NC(C(C)OCCC#C)=O 54920,C12(C(=O)NCCN(C(C3C4CCC3(c3cscn3)C4)=O)CC)CCC(OC)C1C2 54921,C(C(O)(C(F)(F)F)C1CCC1)NC(NC(CC)C)=NCSC1CC1 54922,N1(C(CCCC=C)=O)CCN(C(c2ccc(-c3ccccc3)[nH]2)=O)C(CCC)C1 54923,Cc1cccc(C(=O)NCC2(C)CCCN2C(=O)COc2ccccc2)c1F 54924,Cc1cc(C(N2CCN(C(C3C4CC5C(C4)C35)=O)CC2CC(F)F)=O)nnc1C 54925,c1(C(=O)NC2COCC2NC(C)=O)c(F)ccc(C)c1Cl.C1CC(O)CC(=O)N1 54926,C1(CCC)CN(C(=O)CC#N)CC1C(N1CC(CC(F)(F)F)C1)=O 54927,c1(OC)cc(C(=O)N(C2CCC(NC(c3[nH]ccc3C)=O)CC2)C)cc(F)n1 54928,CS(=O)(=O)c1cc(C(N2CCN(C(=O)C3=CCCC3)C(C3CC3)C2)=O)ccc1F 54929,c1(OC)c(Cl)cc(C(=O)N(CC(C)(C)NC(C2CC(C)C2)=O)C)cc1Cl 54930,CCCC(CNC(c1cnn(C2CC2)c1)=O)C(=O)NCc1ncccc1O 54931,c1(CNC(CN(C(=O)C(COC)NC(C)=O)CC)=O)ccc(C)c(C)n1 54932,C(=O)(CCC(N)C(=O)O)N1CCN(Cc2c(OC)cccc2)CC1C 54933,Cc1ccc2c(c1)N(C(=O)N(CC1=CCCOC1)CCO)CCC2 54934,c1(C(=O)NCC(N(C(CCOC(C)C)=O)C)C2CC2)cc(Br)c2cccnn12 54935,N1(C(c2ccn(CC)c2C)=O)CCN(C(c2cnn3ccsc23)=O)C2CC12 54936,CC1CC(CNC(c2cc(CN(C)C)no2)=O)CN1C(=O)CCn1cncn1 54937,N1(C(C(CC)(F)F)=O)C(CNC(c2ccnc3ccsc23)=O)CC2COCC12 54938,C1(C2CN(C(=O)CCc3nc(O)n[nH]3)C2)(NC(C2N(C)CC(O)C2)=O)CC1 54939,C(N=C(NCC1CCCO1)N1CCC2(C1)CC2(F)F)c1cc(C)cc(C)n1 54940,c1(NCC(=O)Nc2cccc3[nH]ccc23)cc(F)c(N2CCCCC2)c(F)c1 54941,C1(NC(COCCCC)=O)CC2CCC1N2C(=O)C(C(C)C)SC 54942,C1(CC)(NC(c2nccn2C)=O)CCN(C(c2c[nH]nc2C)=O)CC1 54943,N(C1CCc2c(OC)cccc21)C(=O)NCc1c(C(=O)OC)sc2ccccc21 54944,CC(O)C(C(=O)NCC(C)(C)CNS(C)(=O)=O)N(C)C 54945,C1(CCC(=O)NC2C(C(=O)OCC)CC2)CCCN1C(=O)CCCN(C)C 54946,CCS(=O)c1ccc(-c2ccc3nnc(C(=O)NCC(C)O)n3c2)cc1 54947,C1(Nc2cccc(OCC#N)c2)CCCC2CNCCC12 54948,Cn1nccc1C1OCCC1C(=O)NCC(C1CCC1)NC(C1CC(F)(F)C1)=O 54949,C1(C(=O)NCC(C)NC(C(=O)NCC)=O)CCC(C)(C)CC1 54950,N(C(=NCCC1CCCN(CCOC)C1)NCc1cnccc1Cl)C(C=C)C 54951,CCC1=C(C(=O)NC2(CNC(=O)C#CC3(C)CC3)CC2)SCCO1 54952,c1(NC(C2C3(CN(C(=O)OC(C)(C)C)C3)CCC2)=O)nc(O)c2ncnc-2[nH]1 54953,C1(NC(c2cn(CC(C)C)nc2)=O)CCCCCN(C(=O)CC(C)F)C1 54954,CC1(C(=O)NCC2(F)CN(C(C3CC3CF)=O)C2)CC(c2ccccc2Cl)=NO1 54955,CC1(F)CC2(CN(C(C3CC=CCN3C(c3c[nH]ccc3=O)=O)=O)C2)C1 54956,CCC(F)(F)CC(=O)NCC1CN(C(=O)C(C2CCCCC2)N(C)C)CCCO1 54957,c1(C(N2CC(OCC)C(NC(=O)CC3CCC(=O)C3C)C2)=O)c(O)cccc1F 54958,C1(OCC(=O)NC(C2CCCCN2C(=O)C2=CCSC2)C)CCCCC1C 54959,c1(C(=O)NCC(C)(C(C)C)NC(C(CCOC)C)=O)nc[nH]c2ncnc1-2 54960,C1(C(N(C)CC2CN(C(=O)Cc3cncn3C)CCO2)=O)C2(CCC2)C12CCC2 54961,CCCCCCCCC(=O)NCC1(OC)CN(C(C2(n3cncn3)CC2)=O)C1 54962,C1(CN(C(C2C(C(N(CC#C)C)=O)C2)=O)C)CCN(C(c2cnc(S)[nH]2)=O)CC1 54963,C1(C(=O)NCC(C)C(=O)NC2CC(CO)(CO)C2)CCCCC1(F)F 54964,c1(NC(C(C(C)CNC(=O)CC2(C)CCC2)F)=O)cccc(N=[N+]=[N-])c1 54965,c1(C(=O)NCC(CC(C)C)(C)NC(C2CC=CC2)=O)cc2c(cn1)COCC2 54966,C(=O)(CCC1CCc2ccccc21)NCCCn1cc(C(C(C)C)O)nn1 54967,C#Cc1ccc(C(=O)NCC(C)(C2CC2)NC(=O)C(CC)OCC)nc1 54968,C(=O)(CCC(C)(C)NC(c1cnn(CCO)c1)=O)NCc1cn(C)nc1 54969,C(=O)(C(CO)C(C)(C)C)NCCC(C(C)C)NC(c1c(OC)cccc1)=O 54970,c1(C(N(C)CC2C(NC(CCCN(C)C)=O)CCC2)=O)cc(O)cc(F)c1 54971,C1(NC(CCCCC=CC)=O)CCOC2(CCN(C(=O)CCCCC)CC2)C1 54972,Cc1ncc(CNC(C2(NC(=O)CCCn3cncn3)CC2C)=O)o1 54973,N1(C(C2CCC3(CCC3)C2)=O)CCCC2(CCCN2C(=O)CC2CCCOC2)C1 54974,C1(N(C(=O)C(C2CCC2)OC)CC)CCCN(C(c2c[nH]nc2C(C)C)=O)C1 54975,Cc1cc(NC(C2CCCN2C(=O)CC2CCC(C)(C)C2)=O)cc(O)c1 54976,C1(CC)Cc2ccccc2CN1Cc1cccc(OC)c1 54977,n1(CC(N2CC(C(C)NC(Cc3c(C)occ3)=O)C2)=O)ccc2c(C)cccc12 54978,C(=O)(C1(C)OC(=O)c2ccccc21)NCC1CCc2c(cnc(C)n2)C1 54979,C#CCCCCC(=O)N1CCC1C(N1CCCC(CCCO)C1)=O 54980,C(=O)(C(C(C)(C)C)NC(=O)CCOCCC)NCC(CCC=C)O 54981,c1(CC(=O)NCCCCC(C)NC(C23CCCC2C3(F)F)=O)cccc(Cl)c1F 54982,c1(C(N2CC(CNC(c3ccc(SC)o3)=O)C2)=O)ccc(N)c2c1CCCC2 54983,Cc1c2cccc(NC(C3CC3C(=O)NCC3CCCOC3)=O)c2nn1C 54984,c1(NCc2cc(N3CC(C)OCC3)ncc2)cc(OC)ccc1F 54985,CC(C)(O)C(C)(C)C(=O)N1CCC(C(=O)NC2CCCC(F)(F)C2)CC1 54986,c1(N2CCC(C)(NC(C(C)Oc3ccccc3)=O)C2)ncc(Br)c(N(C)C)n1 54987,C1(CNC(CN(C2CCC2)C)=O)CC(NC(=O)C(C)(C)CF)CC1O 54988,O=C(CCC(=O)N1CCOCC1)NCCCN(C(c1ccsn1)=O)CC1CCCC1 54989,N1(C(CC(C)(C)N(C(c2nn(CC)c(C)c2)=O)C)=O)CCC2CCN(C)C2C1 54990,N(C(=NCC1CCCC12CC2)Nc1ccccc1Cl)CCNS(CC)(=O)=O 54991,N1(C(C2CC(SC)C2)=O)CCCC2(CNC(=O)COCC(=O)OC)CCCC12 54992,c1(C(=O)NCC(CCCC)NC(C2CCC(OCC)C2)=O)c(CC)nn(C)c1Cl 54993,c1(C(CN(CCOC)C(C)C2CC2)O)cccc(Cl)c1 54994,N1(C(C2C(C)=CCS2)=O)CCC2(CC2NC(C2CC2c2ccccc2)=O)C1 54995,N1(C(c2ccc(OC)c(O)c2)=O)CC2(CC(NC(c3ccc(F)o3)=O)CO2)C1 54996,C1(NC(C(CN(C(C2(CC)CCOC2)=O)C)C)=O)CCCCCC1C 54997,N1(N2CC(n3c(C(=O)OCC)ncn3)C2)CCC(CO)C2CCC12.C=O 54998,Cc1nc2ncc(C(=O)NCC3CCCN(C(C4CC4(Cl)Cl)=O)C3)c(=O)n2[nH]1 54999,c1(N2CCC(CCNC(CCNC(=O)C=CCl)=O)CC2)ccn2ccnc2n1 55000,C1(C)(CC)CCN(C(=O)CCN2CCC(NC(=O)CN3CCOCC3)CC2)C1 55001,c1(C(N2CCC(O)(CC(C)NC(COCCCC)=O)C2)=O)nc(Cl)c(=O)[nH]c1N 55002,CC(C)(F)C(=O)N1CCC1CNC(c1cc(C2(O)COC2)on1)=O 55003,c1(C(N=S(N(C)C)(C)=O)=O)cccc2c1CN(C)C2 55004,c1(C(=O)NCCCNC(c2c(C#C)c[nH]n2)=O)cccc2c1ccn2CCOC 55005,c1(C(C)C)cc(C(=O)NC2CC(NC(C3CCN(C)C3)=O)C2)on1 55006,n1(CCC)cc(C(=O)NC(c2cn(-c3ccc(Cl)cc3)nn2)C2CC2)c(C)n1 55007,c1(NC(C2(CC#C)CCCO2)=O)cccc(CNC(=O)C(C)C(F)F)c1 55008,Cc1nn(C)c(C)c1CC(=O)NCC1C(C)CCCN1C(c1cnco1)=O 55009,c1(C(=O)NCCN(C(=O)C(C)c2cc[nH]n2)CCOC)nc(O)sc1C 55010,C1(NC(COC)=O)CC2CCC1N2C(=O)CCNC(c1ncccc1O)=O 55011,c1(CC2(CNC(N(CC(C)C(C)C)CCOC)=O)CCC2)cccc(Cl)c1 55012,Cc1snnc1C(=O)N(C)CCN(C(=O)C(F)C1(NC(=O)OC(C)(C)C)CC1)C 55013,Cc1ccc(Br)nc1C(=O)NC1C2CC3C(C2)C13C(=O)O 55014,n1(CC)c(SC)nc2c(C)csc2c1=O.C1(C)CC(C)N1.C(C)(C)(C)OC=O 55015,c12ccc(cc1)[nH]c2=O.c1(CSCCC(=O)Nc2cc(CO)[nH]n2)ccccc1 55016,N1(C(=O)C=Cc2ccco2)CCCC(C2CN(C(=O)C3=CC4CCCC34)C2)C1 55017,N1(C(c2ccccc2)CC)C(C)CN(C)CC1C.C1(C=O)CC2(C1)CC1(CNC1)C2 55018,N1(CC(=O)N(C2C3CN(C(CC(C)OC)=O)CC32)C)CCCCS1(=O)=O 55019,N1(C(c2ccc(SCC)nc2)=O)CCC(NC(C2(CCF)CC2)=O)C(C)C1 55020,N1(C(CN2CCC(=O)CC2)=O)CC(NC(=O)CCc2cnn[nH]2)C(C2CC2)C1 55021,C(=O)(C(C1CN(C(c2cscn2)=O)C1)OC)N(CC(C)C)CC 55022,N1(CC(=O)NC2(C)CN(C(C3(C(F)F)CCCO3)=O)C2)CCC(F)(F)C1 55023,c1(C(C(=O)NCC2(CC(=O)NCCOCCC#C)CC2)F)ccccc1 55024,c1(OC(CC(=O)NC(CCNC(C=CC(CC)=CC)=O)C)C)cc(Cl)cc(Cl)c1 55025,N1(C(C(=O)NC(C)C)C2CC=CC2)CCOC2(CCCS(=O)(=O)C2)C1 55026,c1(C(N2CCN(CC)C(C)C2)C(=O)NCC2CCOC2)ccc2c(n1)OCCO2 55027,c1(SCC(=O)N(CCCN(C(C2CN(S(CC)(=O)=O)C2)=O)C)C)ccccc1O 55028,CC(C)C(C(C)NC(=O)Cc1csc(-c2nc[nH]n2)n1)NC(=O)Cc1ccsc1 55029,N1(C(c2c(CC)ccs2)=O)CC(NC(C2CN(S(C)(=O)=O)C2)=O)CC(F)C1 55030,C(=O)(C#CC1CCOC1)N1C2(CCCC2)C(F)(F)CSCCC1.C1(OC)CCCC1 55031,C1(C)(CCNC(C2C(C)CC2)=O)CCN(C(=O)CC2CC2)CC1 55032,N1(CCC2CC(C(=O)OCC)C2(C)C)CC(N2CCCC2)CC1CC 55033,N1(C(c2c(CC)nns2)=O)CCC(OCCCNC(=O)C(F)C(C)C)CC1.C(=O)OC 55034,Cc1nc2n(n1)CC(C(=O)NCCCCC(CO)NC(c1ccsc1C)=O)CC2 55035,N1(C(C(C2CC2)NC(N(C)Cc2ccccc2)=O)=O)CC(C)(C)NC(C)(C)C1 55036,c1(C(N2CC(C(C)NC(C(CCCC)(C)F)=O)C2)=O)nc2cc(F)ccc2s1 55037,c1(C(N2CC3C(NC(c4ccc(C(=O)OC)cn4)=O)(C3)C2)=O)cc(C)c(C)cn1 55038,C1(CNC(c2c(C(C)C)noc2)=O)CC2COCC2N1C(=O)CC1CCC2CC12 55039,C(=O)(C1Cc2ccccc21)NCC1C(NC(c2c(O)nc(CC)c(C)c2)=O)CCC1 55040,C(=O)(C(CO)C(F)(F)F)N1CCC(CC=C)(C(=O)NC(c2ncc[nH]2)CO)C1 55041,c1(C(N2CC(OC)C(C(N3CCCC3CC3CC3)=O)C2)=O)c[nH]c2nccc-2c1 55042,N1(C(c2c(C)nco2)=O)CCC2(CCC2NC(C2CC23CCCCCC3)=O)CC1 55043,C(=O)(C(CC(F)F)C1CCC1)NCC1CC(NC(=O)CCc2nc(O)n[nH]2)OC1 55044,C1(c2n(CCOCC)nnn2)(NC2(C)COC2)CC2C=CCC12 55045,c1(COC)nc(C(=O)NC2(CO)CN(C(=O)C(C)C3CCOC3)C2)co1 55046,C(=O)(C(O)CC(F)(F)F)N(CC)CC1CCCN(C(=O)CCn2cnnn2)C1 55047,C1(C(=O)NCC2C(C(=O)NCC3CC(O)C3)CC2)CCCC1F 55048,N1(C(COC2CC(NC(C(CCCC#C)C)=O)C2)=O)CCN2C(=O)OCC2C1 55049,C1(NC(c2cc(C)c(C)o2)=O)CC2(C1)CC(CNC(=O)C(C1CC(C)(C)C1)N)C2 55050,Cc1c(C(N2CCC3CN(C(=O)C=CS(C)=O)CC23)=O)ccc2cncn12 55051,c1(C(CC)(C)O)cn(Cc2ncoc2C2CN(C(c3ccc(F)s3)=O)C2)nn1 55052,C1(CNC(c2c(C)onc2)=O)CN2CCCCC2CN1C(=O)C1=CCOCC1 55053,C1(NC(Cc2c(C)cccc2)=O)CC(C)CN(C(C23CCC(CC2)OC3)=O)C1 55054,c1(-c2cc(OC)c(F)cc2F)cnn2c1CN(Cc1c(Cl)ccc(F)c1Cl)CC2 55055,Cc1c(CC(N2CC3CC3(CNC(C3CCCC3(C)C)=O)C2)=O)ncn1C 55056,c1(C(N2CCCC(N(C(C3C(C=C)OCC3)=O)C)C2)=O)cnc(CC)nc1O 55057,c1(CC)ccc(C(C)(C)C(N2CC(NC(c3cnc(O)n3C)=O)C(O)C2)=O)cc1 55058,C(=O)(C(C)(C)n1cc(NCc2ncnn2C2CCOCC2)cn1)OC 55059,C1(CC(=O)NCC(C)OCC)(CC2CCCC2)OCCO1 55060,N1(c2c3ncn(C(CCCC)(C)CO)c3ncn2)CCc2cc(C)ccc2C1 55061,Cc1cccc(O)c1C(=O)NCC1(F)CC(NC(=O)COCCc2cccs2)C1 55062,Cc1cc(C)c([N+](=O)[O-])cc1N(C1CCN(C(=O)OC(C)(C)C)C12CC2)C 55063,C=CCC(C)(C)CNC(=O)C(=O)NCC1CCOC1C 55064,Cc1cccc(CC(=O)N(CCCNC(=O)C(C)Cn2cccn2)C2CC2)c1Cl 55065,C12(CC(N3C(C)CC(CNC(C4(F)CCC4)=O)C3)=O)CC3CC(CC(C3)C1)C2 55066,Cc1cc(N2CCC3CN(C(=O)C(C(C)C)N(C)C)CC23)ncc1[N+](=O)[O-] 55067,Cc1cc(Cl)cc(Cl)c1OCC(=O)N(C)CCNC(c1ncn(C)n1)=O 55068,C1(C(N2CCCC(NC(c3nc(CC)oc3)=O)(CO)C2)=O)CCCCCS1(=O)=O 55069,c1(C(=O)NC(CC)CNC(c2cc(N)cc(F)c2)=O)ncc([N+](=O)[O-])cc1Br 55070,N1(c2cc(C)ncn2)CCC(NC(C2CCC3(C2)CC3(F)F)=O)C12CCC2 55071,c1(CNC(=O)NCCC(=O)Nc2c(CC)cccc2)cc(Br)cnc1C 55072,N1(C(=O)NC(CCC)C(F)(F)F)CC(N(C)CCOC)CC12CCC2 55073,Cc1cc(C(N2CCOCC(NC(c3cc(N)ccn3)=O)C2)=O)c2c(c1)CCO2 55074,C1(C(=O)NCCCCC=C)CCC2(CC2)N1C(=O)Cc1n[nH]c(C)n1 55075,CCC(CC)C(F)C(=O)N1CCCC1CC(=O)N(C1CN(C(C)C)C1)C 55076,CCCC(C(=O)N1CC(C)(OCCNC(=O)Cc2n[nH]cc2Br)C1)OC 55077,c1(C(=O)NCC2(NC(C(c3ccc(Cl)s3)C)=O)CCCC2)cn2c(n1)COCC2 55078,c1(NCC(N(C(c2cnc(C)o2)=O)C)C2CC2)nc(Cl)nc2[nH]c(O)nc12 55079,N1(C(C(CC=C)C)=O)Cc2ccc(CNC(c3cc(COC)no3)=O)cc2C1 55080,c1(C(N2CC(O)CCC(NC(CC(COC)C)=O)C2)=O)ccc2c(c1)OCCN2 55081,C1(O)(CCNC(c2ccn(C(C)C)n2)=O)CCN(C(C2CCCCC2F)=O)CC1 55082,C=CC(C)CC(=O)NCC1CC(CNC(C2C=CCC2)=O)C1 55083,CC1(NC(=O)CNc2nccs2)CC(NC(c2csc(-c3ncccn3)n2)=O)C1 55084,N1(C(CNC(C)=O)=O)CCC2(CCN(C(=O)CN(C3CCSC3)C)C2)C1 55085,N1(C(C(CCNC(=O)CSC(F)F)OC)=O)CC2(CNC(=O)C2)C1 55086,c1(CN(C)C)cccc(C(=O)Nc2nc(C3C4COCC34)cs2)c1 55087,C1(OCCC)CCCCC1C(=O)N(C)CCN1CCN(C(=O)CC(C)(F)F)CC1 55088,CC1CCCC(C(=O)N(CCCNC(=O)CC23CC(O)(C2)C3)C)C1 55089,CCCC(C(O)C(=O)NCC(C)(O)C(C)C)NC(c1ccc2c[nH]nc2c1)=O 55090,c1(OC)cc(C#N)ccc1CNCCC(C)(C)C(=O)Nc1ccccc1N(C)C 55091,Cc1ccc([N+](=O)[O-])cc1C(=O)NC(c1ccc(F)cc1)c1cccs1 55092,Cc1cccc2ncc(CN3CC(C4(C)OCCO4)CCC3C3CCNCC3)n12 55093,N(C(=NCC1CCC1)N1CCCC(O)(c2ccc(Cl)cc2)C1)C(C(C)C)C 55094,c1(C(=O)NC2CCC(N3CCOCC3)C2)ccnc(Cl)c1O 55095,Nc1ccc(CNC(Cc2cn(CC3(O)CCCCC3)nn2)CC(=O)O)cc1F 55096,C1(CNC(C2CC23CCCC3)=O)CN(C(c2cnc(S)nc2)=O)CCC1(F)F 55097,C12(C(=O)NC3CCCN(C(C4C5CC(F)(F)CC45)=O)C3)CCCCCC1OCC2 55098,c1(C(=O)NCCN(C(CCSCC)=O)C2CC2)cccc(F)c1 55099,C12(CNC(C3(C)CC=CCC3)=O)CCC(CNC(C3CC(F)(F)C3)=O)(CC1)CO2 55100,N1(C(CN(C)CC)=O)CC2CCC(C1)N2C(=O)C=Cc1ccc(OC)c(C)c1 55101,C1(CC(=O)N(CC(C)NC(=O)C(C)(C)c2cccs2)C)CN2CCN1CC2 55102,CN1CCCC1CCCNC(C1(CC(F)F)CCNC1)=O 55103,N1(C(C(C)=CC)=O)CCC2(CCN(C(=O)CC3COC(=O)C3)C2)C1 55104,N1(C(C(C)C2CC2)=O)CCC(F)(CNC(=O)CNC(=O)C=Cc2cccnc2)C1 55105,N1(C(C(C)C)=O)CC(NC(=O)C(C)Oc2cccnc2)C(C#N)C1 55106,CCCCC(C)(CO)NC(C1CC=CC(NC(=O)CCc2cscn2)C1)=O 55107,c1(SC2CCC(CCN(C(C(=Cc3cnc[nH]3)C)=O)C(C)C)C2)cccc(Br)c1 55108,C1(C(=O)NCCC#C)CN(C(C2(CN(C)C)CC2)=O)CCO1 55109,C1(NC(C(CC=C)(C)C)=O)CC1C1CCCN(C(C2CCCC(O)C2)=O)C1 55110,c1(OC)c(CN2CCCC(C(=O)Nc3c(C)ncnc3C)CC2)cc(Cl)cc1Cl 55111,Cc1nncn1NC(=O)C1c2c[nH]nc2CN1C(=O)C1CCc2ccccc21 55112,c1(OC)ccc(CN(C(=O)C(=O)Nc2csnc2C2CC2)C)c(C(F)(F)F)c1 55113,C(=O)(CC(=O)NC1(CNC(=O)CCn2cncn2)COC1)NCC#C 55114,C1(C(N2CCC(C#CC)C2)=O)N(C(=O)CCCCC(N)=O)CCCC1(C)C.C1CO1 55115,CCC(C)(CO)C(=O)NCCCC(C1CCN(C(=O)COCP(C)(C)=O)CC1)O 55116,C1(F)(C(=O)NC2(C(=O)NCC3(CC=C)CCCC3)CSC2)CCOC1C 55117,N1(C(c2nncc(OC)c2)=O)CC(NC(c2cc(C(F)F)[nH]n2)=O)CC12CCC2 55118,C12(CNC(C(CO)NC(c3c(C)non3)=O)=O)CCN(CC1)CC2 55119,C1(NC(c2ccc(=O)oc2)=O)CC(F)CN(C(c2cnn(CC3CC3)c2)=O)C1 55120,c1(CC(C(=O)OC)NC(C2OCC3CCCC2C3)=O)c(F)c(F)c(F)c(F)c1F 55121,Nc1c(F)cc(C(N2CC3CC2C3NC(c2csc(C(F)F)c2)=O)=O)c(F)c1F 55122,C#CCCCC(=O)NCCC1CSCCN1C(=O)COC(C)(C)CC 55123,CC1C(O)CCCN1C(c1n[nH]cc1CNC(c1ccc(=O)n(C)c1)=O)=O 55124,c1(C(=O)NC2C(CNC(CS(CC)(=O)=O)=O)CCCC2)cc2cccc(C)c2s1 55125,c1(C(N2Cc3[nH]nc(-c4ccnnc4)c3C2)=O)ccn2ncc(Br)c2n1 55126,C12(NC(Cc3c(C)scc3)=O)CCC(CNC(=O)C(n3cc(Cl)cn3)C)(C1)OC2 55127,S(=O)(=O)(c1cc(Br)c(F)cc1F)N1CCC(C)C2(C1)CCCCC2 55128,c1(CC(=O)NC(CC)CNC(=O)CCC2CCC2)cccc(OC2CCOC2)c1 55129,N1(C(C(c2cccs2)SC)=O)CCCN(C(=O)COC(C)=O)CCC1 55130,c1(NC(C)C)cccc(C(N2CCC(CN(C(=O)CCc3cnc[nH]3)C)C2)=O)c1 55131,C1(C(N2CC(NC(C3CCN4CCCC4C3)=O)(CF)C2)=O)CCc2cnnn2C1 55132,CCC(C)(F)C(=O)N1CCCC(CN(C)C(c2cccc(F)c2)=O)C1 55133,N1(C(C2(C=C)CC2)=O)C2CCC1CN(C(C1(C3CC3)CCC1)=O)C2 55134,C(=O)(CC(CC)C1CCC1)N(CCCN(C)Cc1onc(CCC)n1)C 55135,O=S(=O)(c1ccc(-n2cc(-c3cccc(F)c3Cl)nn2)cc1)C(F)(F)F 55136,CCCCC(C(=O)N1CC2CC1CN2C(c1n[nH]cc1C)=O)N1CCCS1(=O)=O 55137,CCCCCCCCC(=O)NC1CCC(CCC(=O)NC(C)COCCOC)C1 55138,C(=O)(C1=NOC2COCC12)NC(CNC(c1nn(CCCC)c(=O)cc1)=O)CC 55139,O=C1Cc2c(N3CCC3C(=O)Nc3ccc4nncn4c3)ncnc2N1 55140,c1(CNC(C2(C)CCN(C(C(CCC)OC)=O)C2)=O)cccc(F)c1F 55141,n1(C2CC(O)C2)nc(CN2CCCc3[nH]ccc3C2)c2c1CCCC2 55142,C1(CC(=O)NCCCCC2C(C)C2)(NC(C2CC3CCC3C2)=O)CCCCC1 55143,N1(C(c2ccn(C(C)C)n2)=O)CC2CN(C(c3ccnc(S)c3)=O)CC(C1)O2 55144,C1(C(N(CCCNC(C2CC=CCO2)=O)C)=O)CC2(CCCCC2)S1(=O)=O 55145,c1(C(=O)NCC2(CNC(C(C3CCC3)OCC)=O)CCCC2)ccc(N)c(Cl)c1 55146,C1(C(=O)Nc2c(C(=O)OC)csc2)CCN(C(c2cc(OC)n[nH]2)=O)CC1O 55147,C#CC1(C(=O)NC2CCCC2CCOC)CN(C(C2CCC(F)C2)=O)C1 55148,c1(C(=O)NCC2C(CNC(C3CCC(COC)C3)=O)C2)ccc(C(F)(F)F)nn1 55149,c1(C(=O)NC(CNC(c2onc(C)c2C)=O)C2CCC2)cc2c(nc1N)CCC2 55150,N1(C(c2n(CC)ncc2)=O)CC2CCCC(C1)N2C(c1cc(N)c(Cl)c(O)c1)=O 55151,c1(CN2CCN(CCC(=O)NC3CN(C)C3)CC2)c[nH]c2cccc(F)c12 55152,N1(C(C(C2CCN(C(CN(C)CC)=O)C2)F)=O)CCC12CC(CC(N)=O)C2 55153,c1(CCC(=O)NCc2cn(CC(C)(C)C)nn2)ccc([N+](=O)[O-])cc1 55154,CCC(CNC(C1CCCOC1CN)=O)(CC)NC(C1CC(F)(CO)C1)=O 55155,C(=O)(CCS(C)(=O)=O)NCCN(C(C1CC(CC)OCC1)=O)C1CC1 55156,c1(C(=O)NCC(C)N(C(CCC(C)OC)=O)C)ccn2c(C(F)(F)F)nnc2c1 55157,CC1CCN(C(C23CCCCC2OCC3)=O)C(C)C1NC(C1CC=CCN1C)=O 55158,N1(C(c2c(CC)non2)=O)CCC(NC(=O)C=C2CCCC2)C(F)C1 55159,CC(C)CCN=C(NCC(C)(C)C1(O)CCC1)NC1CC1C 55160,C(=O)(C1=CC2CCC(C1)C2)N(C1CCC(NC(C(C(C)C)C)=O)CC1)C 55161,N1(C(Cc2cc(C)no2)=O)CC(C)N(C(=O)CSc2cc(Cl)ccc2Cl)CC1C 55162,O=C(C1=CCCCC1)NC1C=CCC(C(=O)NCC(Cl)Cl)C1 55163,C1(C(=O)NC(CC#C)CC)CNC(=O)CN1C(=O)C(COC)N(C)C 55164,CC(C(=O)NCCCC(=O)N1CC(C(N)=O)(N(C)C)C1)C(F)F 55165,C1(NC(CCCCC=C)=O)CN(C(=O)C=Cc2ncc(C)[nH]2)CC12CCC2 55166,N1(CCC(CC)CO)CCC2(CC1)CC2n1cc(-c2ccc(N)cc2CC)nn1 55167,c1(C(N2CC(CNC(C3(C)CCOCC3)=O)C3C2C3)=O)ccc(Cl)nc1N 55168,C1(C(=O)NC(CCC)C(=O)OC)CCCN(c2nnc(CC(C)C)s2)CC1 55169,N1(Cc2nc(CCC)sc2)CC=C(CNC(C2CC2(C)C(C)C)=O)CC1 55170,CC1(CC(=O)NC2CC(C(F)C(=O)NCc3conc3C3CC3)C2)CCCCC1 55171,c1(C(=O)OC)c(S(=O)(=O)NC2CCOC23CCCC3)n[nH]c1C 55172,c1(CCC(=O)N(CC(C)C)Cc2c(C)cccc2)nc2ccccc2c(=O)n1C 55173,C(=O)(C(O)CNC(=O)C(C)CNC(C)=O)NCC1CC(C(=O)OC)C1 55174,c1(N(C(C(CCSC)NC(C(C(=O)OCC)C)=O)=O)C)ccc(C#N)cc1F 55175,c1(CC)nc(C(N2CCC(C(C)C(=O)NCC(O)CF)CC2)=O)c(N)s1 55176,C(=O)(C(CNC(C1CC2(C1)CC(C)C2)=O)C(C)C)N1CCN(C(CC)C)CC1 55177,Nc1cc(F)cnc1-n1cc(CC(CC(=O)O)NCn2cc(C3CC3)cn2)nn1 55178,c1(NCCOC)cccc(-c2cn(CC(C)NC(=O)CCCCC3CC3)nn2)c1 55179,N1(C(C=CC(=O)OCCCC)=O)CCC2CN(C(=O)CC3CC3C3CC3)CCC12 55180,c1(C(=O)NCC(C)C2CC2)cc(-c2ccncc2)n[nH]1 55181,c1(CC)onc(C)c1C(=O)NCC1CC1NC(=O)CCCN1C(=O)CCC1=O 55182,c1(C(C(=O)NC(C)C(=O)OC)N(C(C)(C)C)CC=C)cc([N+](=O)[O-])c(C)s1 55183,Cc1cc(C)c(C(C2CC2)NC2CCC2)cn1 55184,CCCC(C(=O)N1CCC(NC(c2cnoc2CC(C)C)=O)C1)N(C)C 55185,Cc1nc(C)n(CCCC(=O)NC2CCC(NC(=O)Cc3sc(O)nc3O)C2)n1 55186,c1(C(N(CCNC(C2CC3(CCO2)CC3)=O)CC)=O)cnc2ccncc2c1 55187,N1(C(c2nn[nH]n2)CCOC)CCC(C#N)(c2ccc(C)cc2)CC1 55188,c1(C(C(=O)NC)N(C2CCC3(CC2)CC3)C)cc2cnccc2o1.c1ccccc1 55189,CC1(C)CN(C(c2c(F)cncc2F)=O)c2cc(-c3cccc(O)c3)cnc21 55190,CC(C)CC(C(=O)NCC1CCN(C(c2cn(C)c(=O)n2C)=O)CC1C)C(C)C 55191,N1(C(C2C(C(C)C)OCC2)=O)CC=CC(C(=O)NCCCC2(C)CC2)C1 55192,Cc1nscc1CCNC(=O)C(=O)NCC1CC2CC2C1 55193,c1(CN(c2nnc(CC3C(OC)COCC3)n2C)C)ccnc2ccsc12 55194,C1(CC)C(NC(c2ccn(C)c2C)=O)CCCN1C(c1ccc(=O)n(C)n1)=O 55195,C1(C(=O)NCC2(NC(=O)C=CCO)CCC2)CNC(=O)N1 55196,c1(CN2CCC(F)(C(=O)NC(C)C3CC3)CC2)cnc2ncccn12 55197,C1(NC(c2c(Cl)cc(C)s2)=O)C2CC(CN(C(c3cc(CF)on3)=O)C2)C1CO 55198,C1(F)(CNC(C2(C)CC=CCO2)=O)CC2CCC(C1)N2C(c1cnc(C#N)s1)=O 55199,CCC(C)CC(=O)C(=O)N1CCCC(C(=O)NCC2(SC)CCC2)C1 55200,C(C1CCOC1)=CC(=O)NC1CC(C(=O)NCC(=O)NC(C)C)C1 55201,c1(C(N2CC(C(=O)NCC3(O)CCC3)C(O)CC2)=O)ccc2occc2c1 55202,C(c1csc(S(=O)(=O)N2CCCC2)c1)=CC(N1CC(C(=O)O)(CO)C1)=O.C1(N)CC1 55203,C(=O)(C1=C(C)OCCS1)N1C2CN(C(c3c(Cl)ccc(OC)n3)=O)C(C2)C1 55204,c1(OC)ccc2ccnc(C(C)NC(c3cc(F)ccc3C(=O)O)=O)c2c1 55205,C1(CC(=O)Nc2cc(C(C)(C)C)no2)CCN(c2ncncc2I)CC1 55206,N1(C(c2cc(OCC)no2)=O)CCCCC1C(C)(C)CNC(c1cnsc1)=O 55207,CC1(C=CC(=O)NCC2(O)CCN(C(C3(C)CCC(=O)N3)=O)C2)CCOCC1 55208,Cc1ccc(CC(=O)NCC2(C)CCCN2C(=O)C=Cc2ccncn2)cc1C 55209,c1(C(=O)NC2CN(C(C(CC)(C)C)=O)CC2C#N)c(Cl)ccc(OC)c1F 55210,C1(C)(CNC(CC2CC(OC)C2(C)C)=O)CCN(C(c2ccn(C)c2C)=O)CC1 55211,N1(C(c2c(C)nc(O)[nH]2)=O)CC2CCCC2(NC(c2cccc3ccnn23)=O)C1 55212,CC(O)(C(=O)NCCCOCCNC(=O)CC1CCC1)C1CCC1 55213,C1(NC(c2ccn(CC3CC3)n2)=O)CCOCC1NC(C1(CF)CCOCC1)=O 55214,C1(C(N(C(C2CCCCC2)C)C)=O)CCN(C(=O)C(O)CC2CCCC2)C12CC2 55215,N1(C(C(CC)C)=O)CC(O)(C2(CNC(C3CCC(N(C)C)C3)=O)CC2)C1 55216,C(=O)(CCCCCF)NC1(CNC(c2c(C)cc(CC)o2)=O)CCC1 55217,N1(C(C(CCCC)N(C)C)=O)CCCCCC(NC(=O)CC2(C)CC2)C1 55218,C1(CC=C)(NC(=O)C(C)CN(C)C(c2csnc2OC)=O)CCOC1 55219,N1(C(CCC=C=C)=O)CCCCC(CNC(C2CCCOC2)=O)C1 55220,C1(NC(CC(=C)Br)=O)CCN(C(=O)CNS(=O)(=O)N(C)C)C12CCC2 55221,C1(NC(c2cn(CC)nn2)=O)CN(C(c2coc(C(N)=O)c2)=O)CC1O 55222,C12(C(=O)NCc3ncc(CC)[nH]3)CCC(NC(c3cnsc3)=O)(CC1)C2 55223,c1(C2CN(C(=O)NCCCC(C)NC(=O)OC(C)(C)C)C2)ccc(Cl)c(F)c1 55224,c1(C(=O)NCCCOCCCNC(C2(SC)CC(O)C2)=O)cc(Cl)c(C)cn1 55225,C=CCC(C(=O)N(CC(=O)NCC1CCC1)C1CCC1)NC(C)=O 55226,C(=O)(CC(CN(C)C)C(F)F)N1CCN(C(c2nn(CC)c(C3CC3)c2)=O)C(C)C1 55227,c1(C(=O)NC(CC#C)C(=O)NCCCC2CCCCC2)cc(C)ccc1O 55228,c1(C(NNC(C(=O)OC(C)(C)C)=O)=O)nc(=NCc2ccco2)[nH]cc1Cl 55229,C(C1OCCc2ccccc21)N1C(=O)CN(Cc2c(OC)nccc2)C1=O 55230,Cc1nn(CC(=O)NC(C)(CNC(C2(Cl)CC2(C)C)=O)C2CC2)cc1[N+](=O)[O-] 55231,c1(NC(C2N(C(CC(C)O)=O)CC(C)C2)=O)cc(Br)cc(F)c1C#N 55232,Cc1nc(Cl)ccc1CC(=O)NC(C)C(C)(C)NC(c1ncoc1C)=O 55233,C(=O)(C1=CNS(=O)(=O)N=C1C)N1CC(CNC(CC(C(F)(F)F)OC)=O)OCC1 55234,c1(CNCC2OCCN(C(C3N(C)CCC3)=O)C2)ccc(Br)cc1C#N 55235,S(=O)(=O)(C(F)F)N1CC(C(=O)NCCC2CC(C(F)(F)F)C2)C1.C12CN(C1)C2=O 55236,N#Cc1cnn(CC(=O)NCCCCCNC(c2cc(C3CC3)on2)=O)c1 55237,C(=O)(CCC(C(C)C)NC(=O)C(F)C(C)(F)F)NC(CC)CCCO 55238,N1(C(CC2N(Cc3ccc(OC)cc3F)CCOC2)=O)C2COCC1CC(F)C2 55239,c1(CNC(C2CCCN(C(C)C(=O)NC(C)(C)C)CC2)=O)cn(C)c(=O)nc1O 55240,C1(NC(c2cncc(OC)n2)=O)CN(C(=O)C2=COCCC2)CC(F)(F)C1 55241,c1(OCC(=O)NCC2C3CN(C(c4cc(O)cs4)=O)CC23)cccc(F)n1 55242,CCCCC(=O)C(=O)NC(C)(CNC(=O)C=CS(C)=O)C1CC1 55243,CCC(C(=O)N1CCCC1CCNC(=O)C=CI)C(C)C 55244,c1(CC2N(C(c3csc(C)c3C)=O)CCC2)ccc(S(C)(=O)=O)cc1 55245,N1(C(C=CC=CC)=O)CCC(C2(O)CN(C(=O)C3=CSCS3)C2)CC1 55246,c1(OCC(=O)NCCCNC(=O)CC(O)c2ccccc2)ccc(Cl)cc1Cl 55247,c1(C(=O)NC2CCN(C(C(C)C3CCCO3)=O)C(C)C2)cccn2nncc12 55248,CC(C)CC(C)CC(=O)N1CCC(C(=O)NCCc2c[nH]nc2O)CC1 55249,S(=O)(=O)(c1c(C)nn(C(C)(C)C)c1C)N1C(C(=O)N(n2ccccc2=S)C)CCC1 55250,C1(CC)CN(C(=O)COC)CCN1C(c1cn(CCN2CCOCC2)nn1)=O 55251,c1(CC)cncc(C(=O)NC(C)CC2CCN(C(=O)C(C)(C)C3CCC3)CC2)c1 55252,N1(C(CC)C(=O)OC(C)(C)C)CC2(CC2C(=O)NCC(N2CC(C#N)C2)=O)C1 55253,C1(C(=O)NC2CC(OC)C2)C2CN(C(C3CCC4(CC4)C3)=O)CC12 55254,N1(C(CCC#CC)=O)CCCC(CO)(CNC(=O)C=NOC)C1 55255,C1(NC(C2C(OC)CC2)=O)CCN(C(C2CC(SC)C2)=O)CC1(C)C 55256,C(CC1=CCN(c2cc(CNC(C)=O)ncn2)CC1)NC1CN(C(C)=O)C1 55257,N1(C(c2c(CCC)[nH]cc2)=O)CCC(C)N(C(c2c[nH]nc2C)=O)CC1 55258,c1(C(=O)NC2CC(C)(NC(C3C=CCC3)=O)C2)cccc([N+](=O)[O-])c1O 55259,N1(C(c2c(C)nc(C)c(C)n2)=O)CCC2(C)CN(C(c3nn(C)cc3C)=O)CC12 55260,c1(C(=O)NCC(C)(C)NC(C(C(C)SC)O)=O)oc2ccccc2c(=O)c1C 55261,CC1CN(C(C2COCCN2C=O)=O)CCCN1C(=O)CCC(C)(C)F 55262,N1(C(C2(COC)CN(C(C3CC4COCC4C3)=O)C2)=O)CCc2nncn2CC1 55263,C1(C2CN(C(=O)COC(F)F)C2)(NC(=O)COc2ccc(Br)cn2)CC1 55264,c1(C(=O)NCCC(CNC(C2CC2(C)C)=O)OC)ccc(C(C)C)cn1 55265,CC1C=C(C(=O)NCCCCCN(C)C(C2(C)CS(=O)(=O)C2)=O)C1 55266,C1(C(N2C(CNC(C(CC)(C)CO)=O)C(C)CC2)=O)C2CCC1(C)C2(C)C 55267,c1(C(C)C)ccoc1C(=O)NCC1COCC1NC(C1CCCN1C1CCCC1)=O 55268,C1(F)(CNC(CCCC=C)=O)CCC(CNC(=O)CC2(CO)CC2)CC1 55269,Nc1nc2ncccc2cc1C(N1CC2(NC(C3CCC(=O)NC3)=O)CC1C2)=O 55270,C1(CCNC(c2c(C)onc2CO)=O)CC2CCC(C1)N2C(=O)C(C#N)C1CC1 55271,Cc1ccc(C)c(CN2CCC(C(C)NC(=O)CN3CC(=O)N(C)C3=O)C2)c1 55272,c1(CNC2(CC(=O)Nc3c(C)cccc3)CCC2)cccc2cccnc12 55273,c1(CNC2CCC(C(=O)Nc3c(C#N)cc(F)cc3)C2)ccc(Cl)c([N+](=O)[O-])c1 55274,S(=O)(=O)(c1ccc(NCc2ccncn2)c(Cl)c1)NC(c1cc(C)cc(C)c1)C 55275,Cc1cc(C(N2CCOC(CNc3ccncn3)C2)=O)c(C(F)(F)F)o1 55276,c1(OC)ccc(C2(CSC3CCC(NC4(C(=O)OC)CC4)C3)COC2)cc1Cl 55277,C1(NC(c2ccc(C(C)C)o2)=O)C=CCN(C(=O)CNC(=O)CCCCO)C1 55278,N1(CC(=O)N(CC(CC)NC(c2ccn(C)n2)=O)C)C(=O)NC(C)(C2CC2)C1=O 55279,Cc1cnc(O)n1-c1cccc(NC(=O)C(=O)N(C)CCN2CCCC2=O)c1 55280,c1(OCCC)ccc(-c2cc(C(=O)OCCNC(C)=O)ccn2)cc1 55281,CC(Cc1ccncc1)N=c1cc[nH]c(=NCCCc2ccccc2)[nH]1 55282,c1(OC)nc(=NCCC2CCCOCC2)[nH]c(OC)c1[N+](=O)[O-] 55283,C(=O)(C1CCc2nccn21)NC1CN(C(C2(SC)CC2)=O)CC1C 55284,C1(C(=O)NC(C)CCNC(=O)Cc2cccnc2Br)CC2CCC1CC2 55285,c1(C(N(C)CCOCCNC(C2CCCC(C#N)C2)=O)=O)cnc2ccccn12 55286,C=C1CCCN(C(=O)CSCCNC(c2ncn(CC)n2)=O)C1 55287,C(=O)(CCCCC(C)C)N1C(CNC(CCCc2onc(C)n2)=O)CC(C)(C)C1 55288,C(=O)(CC1CCc2ccccc21)NC1CCC(NC(CCNC(=O)OCC)=O)C1 55289,C12(C(=O)NC3C(C)N(C(c4ccc(CO)o4)=O)CC3)CC=CC(C1)OC2 55290,N1(C2CCC(NC(c3cc(C4CC4)on3)=O)C2)CCN(C(=O)C2=CCSC2)CC1 55291,Cc1ccc(CC(=O)NCCC(C)(C)NC(=O)CC2CC(C3CC3)C2)cc1Cl 55292,c1(CCC(=O)NCC2CN(CC(O)COc3cccs3)C2)ncc(F)cn1 55293,c1(-c2c(C)noc2)cnc2cc(C(=O)NCCc3ccsc3)ccn12 55294,Cc1ccn2cnc(C(=O)NC3C=CCN(C(C4(CC(F)(F)F)CC4)=O)C3)c2c1 55295,C1(CNC(C2CC(NC(C(C)n3cncn3)=O)C2)=O)CCOCC1(C)C 55296,C(CCC(=O)NNc1ccc(F)cc1Cl)n1cc(CNC(=O)NC)nn1 55297,C1(N(C(C2CCCN(C(C3C(C(C)C)OCC3)=O)C2)=O)C)CCCC(C)C1C 55298,C12(CNC(C3N(C(=O)NC)CCC3)=O)CCC(NC(c3sccc3F)=O)(CC1)CO2 55299,C=C=C(C)CC(=O)NCCN(C(=O)C(CC)NC(=O)OC)CC 55300,C1(C(C)(C)C)(C(=O)NCCOC2CN(C(CC3C(C)CCC3)=O)C2)CCCCC1 55301,c1(C(C)=O)cc(C(=O)NC(C(=O)NCCS(C)(=N)=O)C2(O)CCC2)no1 55302,c1(CNc2c(CC(=O)Nc3ncc(C)c(F)c3)cccc2)ccc(F)c(C)c1Cl 55303,c1(CC(=O)NCC(C)(CC)NC(C(CCC)O)=O)ccc(S(N)(=O)=O)cc1 55304,c1(C(N(CC(CNC(CNC(CC)=O)=O)(C)C)C)=O)c[nH]c2cc(OC)ccc12 55305,c1(C(N(CCC(C)NC(c2ncoc2C(F)(F)F)=O)C)=O)snc2ccccc12 55306,c1(NC(CN(C(=O)NC2C(OC)CC2)C2CC2)=O)ccc(C(N)=O)cn1 55307,C1(NC(C2N(CC)CC2)=O)C2CC1N(C(=O)C(C)(C)CC1CCC1)C2 55308,CCC1=C(C(=O)N2CC(NC(c3cc(S(C)(=O)=O)c(C)o3)=O)C(O)C2)CCCO1 55309,c1(OC)cccc2ccc(CNC(=O)CC3CCCN3C)nc12 55310,S(=O)(=O)(c1ccc(C(F)(F)F)cc1)N1CC2C(c3nnc(C(C)C)o3)(CC2)C1 55311,C(=O)(C(F)C(C)CC(C)(C)C)N1C(C(C)NC(=O)C(=O)N=S(C)(C)=O)CCCC1 55312,S(=O)(=O)(c1ccc(NCC=CBr)c(Br)c1)Nc1ccc(OCC)nc1C 55313,c1(CC(C(=O)N(CC)CC2CCC2)NC(c2cc(C)no2)=O)cnn(C)c1O 55314,C=CC1CN(C(=O)CCCn2ccnn2)CC1NC(=O)CC1CNC(=O)C1 55315,c1(N2CC(N(C)C(c3cc4cccnc4s3)=O)C2)ncnc2cc(Br)ccc12 55316,Cc1nc(C)c(C(C)NC(N2CCC(CCc3nn[nH]n3)CC2)=O)s1 55317,Cc1cc(C)c(CN2CCN(C(=O)C=Cc3ccoc3)C3CC23)cc1C 55318,C(c1ccc([N+](=O)[O-])o1)=CC(=O)Nc1cccc(-c2ccc(C)o2)c1 55319,c1(C(=O)Nc2c[nH]nc2C(=O)Nc2cc(F)ccc2I)cc2sccc2[nH]1 55320,c1(C(N(CC(C)(C)CNC(c2cc(C(F)F)[nH]n2)=O)C)=O)cccc(F)c1Cl 55321,C(=O)(C(CC)C(F)(F)F)N1C(CC)C(C(=O)NC(CCOC)C(N)=O)CCC1 55322,C(=O)(C(C)(C)Cc1cn(CC(=O)NC(C)C)nn1)NCc1ncc(CC)o1 55323,N1(C(CC=C)=O)CCC2CCC12Cn1cc(C(=O)NCC2CC2)nn1.c1ccccn1 55324,N1(C(CC)C(=O)O)CCC2(CC1)CC2(C)C(=O)NC1CCOC(c2cccs2)C1 55325,c1(CCC)c(C(=O)NCCCN(C(=O)C(c2ccccc2)C)C)cnn1C 55326,c1(C(C)NCc2cc(C3CCC3)no2)coc2ccccc12 55327,c1(C(=O)NC(CCCC)CNC(c2cc(Cl)no2)=O)cc2cccn2cn1 55328,c1(NC(C(CC)C)C)nc(N2CCCC3(C2)CC(OC)(OC)C3)nc2sccc12 55329,CN1CCC(C#N)(C(=O)NCC2(C)CCCN(C(C3(C)CCCCO3)=O)C2)CC1 55330,C1(C(=O)NC(C)Cc2cnn(C)c2)CC2CCC(C1)O2.C12CCC(CC1)C(=O)N2 55331,c1(C(=O)NCC(CC(C)C)NC(=O)CSC(C)C)cc(O)c2ccccc2c1 55332,C(=O)(CS(=O)(=O)C(C)C)NC(c1ccccc1)C1(N(C(C(CC=C)(C)C)=O)C)CC1 55333,CN1CCN(C(=O)Cc2csnn2)CC1CNC(=O)COc1ccon1 55334,N1(C(C(=O)NCCCC)CC2CCC(C(C)(C)C)CC2)CCC2C(O)C(C)(C)C12 55335,C(=O)(C#CC1CCCC1)NCCCCC(C)NC(C1(c2cccc(O)c2)CC1)=O 55336,C(=O)(C(C(C)CC1CC(F)(F)C1)NC=O)NC1CCN(CCCOC)CC1 55337,c1(C(N(CC(CNC(C2C(C)OCC2)=O)O)C)=O)ccc(N(C)C)cc1F 55338,c1(C(=O)NC(C)C(CO)NC(=O)C#CC2CCCO2)cccc2sccc12 55339,C1(NC(c2n(CCC)ccc2)=O)CCN(C(c2cn[nH]c2)=O)C1(C)C 55340,C#Cc1nc(C(=O)N(CC(N2CCN(C(=O)CCCCOC)CC2)=O)C)cs1 55341,N1(C(c2c(C)cno2)=O)CCC2(C1)CN(C(c1nc(CN(C)C)no1)=O)C2 55342,CC(=O)CCCC(C)C(=O)NC(CC(=O)N1CCCC(O)(CN(C)C)C1)CC(C)C 55343,CC1(C)COCC(C(=O)NC2C=CCN(C(c3cncc(CO)c3)=O)C2)O1 55344,CCC(CC)C(C(=O)NCc1ccc(C(N2CC(S(N)(=O)=O)C2)=O)nc1)OC 55345,N1(C(c2ccc(C(C)C)o2)=O)CCCC(C)(CNC(c2cnc(O)c(Cl)c2)=O)C1 55346,Cc1cc(CN(c2nnnn2CC2CCS2(=O)=O)C)cc(C)c1Br 55347,C#CC(C)(C)C(=O)NC1(CNC(c2nnc(C(C)C)s2)=O)CC1 55348,C1(C(=O)NCC(CC(=O)N(CCCO)CC)O)CC2C(C1)C2(C)C 55349,N1(C(CCC2CC(C)C2)=O)CCCC(CO)(CNC(=O)CS(C)(=O)=O)C1 55350,C(=O)(C(C)(C)CCCNC(C1CCC(=O)C1)=O)NCC(n1ccnn1)C 55351,C1(CC(=O)NC)CN(C(C2CCC2(C)C)=O)CCN1C(C1CCC=CCC1)=O 55352,C#CC(CNC(=O)C(Cn1cncn1)NC(=O)CN1CC(C)(C)C1)CC(C)(C)C 55353,n1(CC)nc(C2CC2)cc1C(N1CC(NC(=O)CCCc2cccs2)C1)=O 55354,C(=O)(C(O)P(C)(C)=O)N(CCCNC(=O)CCCc1cncs1)C 55355,c1(CN(c2ccccn2)CC)ccc(CNC(=O)NCCCCOCCOC)cc1 55356,N1(C(=O)NCC(N2CCCCCC2)C)C2CCCC1CN(C)C2 55357,CC(C)CC(CCO)N=c1[nH]c2c(c(=NCC3C(F)(F)C34CCC4)[nH]1)CCCC2 55358,C1(C(N2CC(C(C)(C)O)(CNC(C3(SC)CCC3)=O)C2)=O)CC2(C1)CC(F)C2 55359,Cc1ccc2nc(C(=O)NC3CN(C(=O)CS(C)(=O)=O)CCC3CO)cn2c1 55360,c1(C(N2CCN(Cc3cccc(C)c3C)CC2)=O)ccc2c(c1)OC(C)C2 55361,Cc1nccc(Cl)c1C(=O)NCCN1CCCN(C(C2CC2Cl)=O)CC1 55362,C12(C(N(C)CC3CN(C(C4COC5(CCC5)C4)=O)C3)=O)CC3CC(CC(C3)O1)C2 55363,CC1(CNC(c2cnc(C3CCC3)s2)=O)CCCN1C(C1CCC(C(N)=O)C1)=O 55364,C#CCC(CC#C)C(=O)NCCCCN(C)C(c1csc2c1CCCC2)=O 55365,C1(OC)CC=C(C(=O)N2CC(N3CCN(C(c4occ5c4CCC5)=O)CC3)C2)C1 55366,CC#CCCC(=O)N(CCNC(c1cncnc1-c1ccccc1)=O)C1CC1 55367,c1(SC)cncc(C(=O)NC2CC(NC(=O)C=CC3CCOC3)C2)c1 55368,N1(C(C2(C)CS(=O)(=O)C2)=O)CCC(C2CCN(C(=O)CC#N)C2)C1 55369,C1(C(N(C(CC)C(=O)NC(C)(C)CCCF)C)=O)CN2CCC1CC2 55370,N1(C(CCC=CC(C)C)=O)CCC(C)(NC(=O)C(C)CC2CCCCC2)C1 55371,n1(CC(=O)Nc2c(C)cc(NC(=O)CSCC(N)=O)cc2)cnc2c1CCCC2 55372,C(C)(C)(CC(=O)NC1CCN(C(C2CCC3CCC23)=O)C1)SC 55373,C1(c2cccnc2)(C(=O)NCC2N(C(C3CC3(Cl)Cl)=O)CCC2)CC2(CCC2)C1 55374,c1(NC(C(C(C)C)NC(C(CCC)NC(N)=O)=O)=O)cc(C#N)ccc1O 55375,N1(C(Cc2c(C)ocn2)=O)CCN(C(=O)Cc2csc(C(C)C)n2)CC1 55376,S(=O)(=O)(c1cccc(=NC2CCC=CCCC2)[nH]1)NC1CN(C)C2(C1)CCOCC2 55377,c1(N2CCC(N(C(=O)C(O)CCSC)CCC)C2)cc(C)c(C#N)cn1 55378,CC1CC(C(N2CCC(C(C)NC(C3(C4CC4)CCC3)=O)C2)=O)CCC1C 55379,c1(C(N2CCC(C3N(C(C(F)OC)=O)CCC3)C2)=O)ccc(F)nc1F 55380,C1(CC(=O)N(C(C=C)C)C)CCN(C(c2cc[nH]c2CCC)=O)C1 55381,CC(CC(=O)c1cccc(Br)c1)C(=O)NCC(O)(C(=O)O)c1ccccc1 55382,C1(NC(c2scc(OC)c2)=O)CS(=O)(=O)CC1NC(=O)C=CSC 55383,C(C)(C)(CC(F)C(=O)NCc1ccc(C)s1)NC(CCC(CC)OC)=O 55384,N1(C(C(C)OCCCC)=O)CC2(CCC(NC(C3C=C(C)CS3)=O)CC2)C1 55385,S(=O)(=O)(C=Cc1ccccc1)N1CCN(C(=O)C=Cc2ccccc2)C2C1C2 55386,n1(CC)ncc2c(O)nc(=NNC(=O)Cc3ccncc3OC)[nH]c12 55387,C(=O)(NN1CCCC1C(=O)NC1(C(O)CO)CC1)c1cc(C(=O)OC)[nH]c1 55388,N1(C(C(C)NC(=O)NC)=O)CCCC(CO)(NC(=O)CC2C=CS(=O)(=O)C2)C1 55389,C1(NC(c2ccc(C(F)F)o2)=O)C=CC(CC(=O)NC2CC=CCC2)C1 55390,C1(NC(C2C(NC(CCCC3C(C)C3)=O)CCC2)=O)CCOC1(C)C 55391,C1(C(=O)NCCC2(CNC(=O)COC3CC(F)(F)C3)CC2)CCCCCS1(=O)=O 55392,c1(C(=O)NCCN(C(=O)CC2OCCCO2)CCC)coc(OC)n1 55393,C1(C(=O)NC(C)C(=O)O)CC=CC(n2cc(-c3ccc(F)cc3)nn2)C1 55394,c1(C(=O)NCCCCNC(C#CC(C)(C)C)=O)cc2n(n1)CCCC2=O 55395,C1(CNC(C(=O)N(C)CC2CC2)=O)CCN(C(C2CC(=C3CC3)C2)=O)C1 55396,C12(NC(C(CC#C)O)=O)CCOCC1CN(C(c1cn[nH]c1)=O)C2 55397,CCC(c1ccnc(Cl)c1)=CC(=O)NC(C)CCC(=O)OC 55398,N1(C(C(C)(C)OCC)=O)CCOCC(CNC(c2nc(C)n(C)n2)=O)C1 55399,C=CC1OCCC1C(=O)NC(C)CCNC(=O)CCc1nncn1-c1ccccc1 55400,N#CC1CN(C(c2ccc(N3CCC3)cc2)=O)CCN1C(C1CCOC1)=O 55401,N1(C(CCC#C)=O)CCCC2(CCC(NC(=O)C(=Cc3cccc(Cl)c3)C)C2)C1 55402,c1(CC(C(=O)OC)NC(c2c[nH][nH]c2=N)=O)cccnc1F 55403,c1(N2CCC(NC(CC(CC)O)=O)C(O)C2)c(Cl)cccc1[N+](=O)[O-] 55404,C(=O)(CC(C(F)F)NC(c1ncc[nH]1)=O)Nc1cccc(C(C)C)c1 55405,c1(NC(N2CCC(CC)C2)=O)cncc(OC)n1 55406,C1(CC)C(NC(C2CCC(CC)CC2)=O)CCCN1C(=O)CCn1cnnn1 55407,n1(CC(=O)N(C)CC2CCN(C(C3(COC)CCCC3)=O)C2)ncn(C)c1=O 55408,N1(C(=O)CSC2CCOC2=O)CC(C2CCN(C(=O)CCOC3CCC3)CC2)C1 55409,N1(C(CCC=C)=O)CCC(C(=O)NCC2(c3ccnc(Cl)c3)CC2)CC1 55410,Cc1ccc2c(c1)CCC(C(=O)NCC1CCCCC1NC(c1csnn1)=O)O2 55411,C(=O)(C#CC1CCOCC1)NC(CC=C)CNC(c1cnn(C)c1OC)=O 55412,N1(C(C2C(C)CC=CC2)=O)CCC(F)CC1C(=O)NCC1(C#N)CC(C)(C)C1 55413,C(=O)(C(C)CC(C)C)N(CCNC(CN(CC)CC)=O)CCOCCCF 55414,CCC(CN(C)C)CC(=O)N1CC(O)(CNC(=O)CCCC(=O)OC)C1 55415,c1(COC)cccc(CC(=O)NC2CCC2CNC(c2cccc(CO)n2)=O)c1 55416,C1(CC)CN(C(c2cc(=O)n(C)o2)=O)CCN1C(C1CCCOCC1)=O 55417,c1(OC)ccc(CNC(=O)NNC(C)Cc2ccccn2)c(F)c1Br 55418,C1(C(=O)NCC(C2CCN(C(C3(C)CCC(=O)N3)=O)CC2)C)CCS(=O)(=O)C1 55419,Cc1cc(C(N2CCC3(NC(=O)C(F)C4CCCC4)CC3C2)=O)cc(C)c1O 55420,C1(CC)COC(C)CN1C(=O)CCNC(C1C=CC1C(=O)OC(C)=O)=O 55421,OC1COC2(CCN(c3ncc(-c4nn[nH]n4)cc3Cl)CC2)C1O 55422,c1(C(=O)Nc2cc(C)c(NC(c3c(C)n[nH]c3C)=O)cc2)ccn2cncc2c1 55423,C(CCC(=O)NC1CC(C)(NC(c2cc(C(N)=O)cs2)=O)C1)OC(C)C 55424,O=C(C1=CCOC1)NCCCCNC(C1CCS1(=O)=O)=O 55425,CCCCCCC(CC)C(=O)N1CCCCC1Cn1cc(CNC(N)=O)nn1 55426,c1(C(N2CC3CC3(C(=O)NCCO)C2)=O)cn2c(Cl)cccc2n1 55427,C1(CN(C)C(=O)N(C(C)(C)C)C)CC1C1CC1 55428,c1(C(N2CCC(O)(CCNC(C(C)(C3CC3)OC)=O)C2)=O)nc(Cl)c(=O)[nH]c1N 55429,Nc1ccc(C(=O)NC2(c3nnnn3CCO)CCC2(C)C)c(O)c1.C(CCCO)S 55430,c1(C(=O)NCC(CNC(C(COC)(F)F)=O)F)cccc2c1ncn2C 55431,Cn1cc([N+](=O)[O-])cc1C(=O)NCC1(F)CN(C(c2cc(F)n[nH]2)=O)C1 55432,c1(OC)cc(C)c(C(=O)NC2COCC2NC(c2ccc(Cl)cc2C)=O)cn1 55433,c1(C(C)C)ccc(OC(C)C(N2CCC(OC(C3CC(C#N)C3)=O)CC2)=O)cc1 55434,C1(C)(CNC(CN(C)C)=O)CCCN1C(c1ccc(C(=O)O)nn1)=O.C(C)(C)C 55435,C1(n2cnnn2)(C(=O)NC2(C)CN(C(c3cc(C4CC4)no3)=O)C2)CCOCC1 55436,N1(C(c2c(OC(C)C)n[nH]c2)=O)CC(NC(C23CCCC2C3)=O)C2(CCC2)C1 55437,c1(C(=O)NCC(CC)NC(C2C(CCC)CCC2)=O)ccc(C)cc1O 55438,Cc1nccc(C(=O)NC2CC(C(=O)N(CCO)CCO)C23CCC3)c1C 55439,c1(C(=O)NC(C(C)O)C(=O)N(C)C)cnc(F)c(F)c1 55440,CC1(C(=O)NCC2(C)CCN(C(c3c(N)cnn3C)=O)C2)CC(C2CC2)=NO1 55441,C1(CC)(NC(=O)CN2CCSCC2)CCCN(C(c2ccc(Cl)c(OC)c2)=O)C1 55442,c1(C(=O)NC(CN(C(=O)C=CCF)CC)C)cc2c(OC)cc(OC)cc2[nH]1 55443,CC1(C(=O)NC2(C3CCC3)CC2)CCN(C(=O)C=CCN2CCC2)CC1 55444,Cc1cc(C)c(C(=O)NC2(C)CN(C(C34COCC3C4)=O)C2)cc1C 55445,N1(C(CN(C)CC)=O)CCC12CN(Cc1[nH]c(C)c(C(=O)OC)c1C)C2 55446,CC(C)C(C(=O)NC1CCN(C(C2CCS2(=O)=O)=O)C1C)Sc1ccccc1Cl 55447,c1(C(=O)NCC2N(C(C(C=C)O)=O)CCN(C)C2)ccc2[nH]ccc2c1F 55448,c1(NC(C)=O)ccc(C(=O)NCC2(O)CC(NC(C3CCC3(F)F)=O)C2)s1 55449,c1(C(=O)NC(C2CCN(C(C3CCOC(=O)N3)=O)C2)C)ccnc(C(F)(F)F)c1 55450,Cc1cc(C(N2CCCC(N(C(=O)C(C)C3=CCCC3)C)C2)=O)cc2nc[nH]c12 55451,c1(C(=O)NC2C(CC)N(C(C)=O)CCC2)c(Cl)ccc(O)c1Cl 55452,N1(C(CCC(C)C)=O)CCc2cc(C(=O)NC3CNC(=O)C3)cnc2C1 55453,C(=O)(C1=CCCC1C)N1C(C(N(CC(C)C)C)=O)CC(=O)C1 55454,C(=O)(C1=CC=CN2CCS(=O)(=O)N=C12)NC(CN(C(=O)CCC#N)CC)C 55455,N1(CCN(C(=O)CC2CC=CCN2C)C)CCN(C(c2ccns2)=O)CC1 55456,C1(NC(CCc2ccc(CC)cc2)=O)CCC(C)N(C(C2C=CCCC2)=O)C1 55457,C(=O)(CC(C)n1cccc1)NCCCN(C(C1CC(O)C1)=O)CC 55458,N1(C(c2cc(COC)sc2)=O)CCC2C(CCN2C(c2ccn3ccnc3n2)=O)C1 55459,Cc1cc(Br)c(N)cc1C(=O)NCCN(C(=O)CCCC(F)(F)F)C 55460,c1(C(=O)NC(CCNC(c2cn(C)[nH]c2=N)=O)(C)C)cccc2nsnc12 55461,N1(C(c2ccc(C(N)=O)s2)=O)CCC2(CC1)CC(NC(C1C3CC4C(C3)C14)=O)C2 55462,c1(C(=O)NC2(C)CC(NC(=O)CC3(C(F)F)CC3)C2)ccc2c(c1)C(=O)C(=O)N2 55463,C1(NC(C(CCOC)C)=O)COC2(C1)CN(C(=O)C=Cc1cn[nH]c1)C2 55464,c1(C(N2C(CNC(=O)C(O)c3cnc[nH]3)CCC2)=O)cnn2cccc(Cl)c12 55465,N1(C(c2cc(C)[nH]c2)=O)CCN(C(=O)CC(C)C(F)(F)F)CCC1C 55466,c1(C(=O)NCC(CNC(c2ncc(C)cn2)=O)O)c(N)sc2ccccc12 55467,c1(C(=O)NC2CCC(CNC(C3CC4CCCC34)=O)C2)ccc2n[nH]cc2c1Cl 55468,c1(NC(CC)C(=O)N(C)CC2(NC(=O)C(N)=O)CC2)cccnc1Cl 55469,C(=O)(C1=CCN(C(c2cnnc(O)c2)=O)C1)NC(C(C)C)CO 55470,N#Cc1ccc(C(N2CCCCC2CCNC(C2CC(=O)N(O)C2)=O)=O)c(O)n1 55471,Cn1cc(C(=O)NC2CCCCC2CNC(=O)C(C)(C)c2cscn2)n(C)c1=O 55472,C1(NC(CCCOC(C)=O)=O)CCOCC1NC(=O)CCc1ncco1 55473,C1(C(=O)NC(Cn2ncc(C)c2)C)CC(C)(C)CN1C(c1cc(C)c(F)cn1)=O 55474,CC(C)CC(C(=O)NCC1(C)CN(C(=O)CC2CCOCC2)CC1C)N(C)C 55475,C(=O)(C1=CC2CCCCCC12)NC1CN(C(C2CN(C(C)=O)C2)=O)C2(C1)CCC2 55476,N(C(=NCCCSC)NCC1CC(=O)N(CC)C1)Cc1ccc(OCCC)cc1 55477,C(=O)(C(CC(C)C)n1ccnc1)NC(CC=C)CNC(C1(CN(C)C)CC1)=O 55478,c1(C(N(CCNC(C2(C)CC3CCC2O3)=O)C2CC2)=O)ccc(Cl)c([N+](=O)[O-])c1 55479,c1(C(N(C2CCCCN(C(=O)C(C)(C)C(F)F)C2)C)=O)cn2ccc(F)cc2n1 55480,CCCCC(CNC(=O)CCCN(C)C(=O)OC)NC(C1CC(CC)C1)=O 55481,C1(C(=O)OC)CC1C1CCN(C(N2CCC(C#N)(SC(C)(C)C)CC2)=O)CC1 55482,Cc1nc(C(N2CCOC(CNC(=O)CC3CCC(F)(F)C3)C2)=O)[nH]c1C 55483,C1(CCC)(CO)CCN(C(=O)C=CC(C)NC(=O)C(C)C2CCC2)C1 55484,c1(C(=O)NCC2N(C(c3c(C)coc3)=O)CCC2)ccc([N+](=O)[O-])cc1Br 55485,c1(CC(C)(C)O)ccc(C(=O)NCC(O)CNC(=O)CCn2ccnn2)s1 55486,Cc1ccc(C)n1CC(=O)NCC1CCN1C(=O)CCc1cccnc1Br 55487,Cc1onc(Br)c1C(N1CC(CNC(c2ccc(O)nn2)=O)C(C)C1)=O 55488,c1(NC)cccc(C(=O)NC2(CNC(=O)CCn3cccnc3=O)CCOC2)c1 55489,c1(C(N2CC(CC(=O)N(C(C)C3CC3)CC)OCC2)=O)ccn2ccnc2c1 55490,Cc1cc(C(=O)NCC2CC(NC(c3cc(Cl)sc3Cl)=O)C(O)C2)cn(C)c1=O 55491,C(=O)(CCC(C)(C)[N+](=O)[O-])NC1(CNC(CN(CC(C)(C)C)C)=O)CC1 55492,C1(NC(=O)CSCC2CCCCO2)CC2(CCCN(C(c3cccnc3)=O)C2)C1 55493,N1(C(C(c2ccccc2)C)=O)CCOCC1(C)c1cn(CCCCCO)nn1 55494,C(=O)(C(CO)C(C)(C)C)NCCCN(CCC)C(c1ccc(CC(C)C)s1)=O 55495,S(=O)(=O)(C(F)(F)F)CCC(N1CC(C2CCCO2)(OC)C1)=O 55496,c1(NCc2n(C)c([N+](=O)[O-])cn2)nc2c(c(=NCCS(C)=O)[nH]1)CSC2 55497,c1(CCC=C)ccc(C(=O)N(CCNC(C2(c3ccc(F)cn3)CC2)=O)CC)cc1 55498,N1(CC(=O)NC(=O)NCC)C2CCC1CC(CNC(=O)C=Cc1cncn1C)C2 55499,C12(c3onc(-c4cc(C(C)C)oc4)n3)CCC(CC1)N(CC(F)F)C2 55500,C1(C(=O)NC2CCC(N(C)C(c3cnsn3)=O)CC2)OCC2CCCC1C2 55501,C1(CC(=O)NC(C(=O)OC)(C)C)CC(C)NC(=S)N1.c1(C(N2C(=O)C2)=O)cccs1 55502,c1(OC)cc(C)cc(C(=O)NCC(C)N(C(=O)CC(O)C(C)C)C)c1N 55503,c1(CCC(=O)NCC(CC)NC(C2CCC(C(F)(F)F)O2)=O)c(F)cccc1F 55504,CC1(C)CC(C(N2CCN(C(=O)CCCF)CC(O)C2)=O)CC(C)(C)C1 55505,Cc1cc(C(=O)NC(C(=O)N2CC(C(C)(C)O)C2)C2CCOC2)nn1C 55506,Cc1ncc(C(N2CCN(C(c3ccnc(CO)c3)=O)CC2C(F)F)=O)cc1N 55507,N1(C(c2c(CSC)cccn2)=O)CCC(CNC(=O)CCCNC(N)=O)C(O)C1 55508,C12(C(=O)NC(C3CCN(C(c4cc(F)ccc4O)=O)C3)C)CCCCN1CCC2 55509,CC1CC(NC(=O)CCC2(C)CC2(F)F)CCN1C(c1coc(O)n1)=O 55510,C1(NC(CSc2ccc(C#N)cc2)=O)CN(C(=O)CCC(N)=O)CC12CCC2 55511,N1(CNC(=O)O)CC2(C(=O)NCCNC(C(C)(C)C)=O)CCC1C2.c1(N)cscn1 55512,C(=O)(C1CC=Cc2ccccc21)NCCNC(C=CC(=O)OC(C)(C)C)=O 55513,C(=O)(CCCC(C)(C)C#N)NCC(CNC(C(C(=O)OCC)C1CC1)=O)O 55514,c1(C(=O)NC(C2CCCN(C(=O)CCc3cnn[nH]3)C2)C)cc2ncccn2n1 55515,CCCC(C(F)(F)F)NC(=O)CSCCNC(=O)Cc1ccoc1C 55516,C1(C2CCN(C(=O)CC(C)SC)CC2)(NC(C2C(C#C)C2)=O)CC1 55517,n1(CC(C)NCC(CO)C2CC2)ccc(NC(=O)OC(C)(C)C)c1.c1nncn1C 55518,N1(C(c2cccc(OC)c2N)=O)CCC(NC(=O)Cc2ccsc2)C12CCCC2 55519,C(CCC(=O)N1CCCC1CC(N1CC(N(C)C)C1)=O)N(C(C)=O)C 55520,C1(NC(=O)COCc2cn(Cc3ccc(C(=O)O)o3)nn2)CC2CSCC(C1)C2 55521,N1(C(C=C(C)C)=O)CC(NC(C2CCOC2c2cccnc2)=O)CCC(O)C1 55522,C(c1ccc(O)c(OC)c1)=CC(=O)NC(CC)CN(C)C(c1csnc1Cl)=O 55523,C(=O)(CCCC1CCC1)N(CCOCCNC(C(C1CCOC1)OC)=O)C 55524,CC(CNC(c1cc(C(O)C2CC2)ccn1)=O)CC(=O)N(C(C)C(C)C)C 55525,CCCC(CNC(C1CCN(OC)CC1)=O)C(=O)NCCN1CC(C)(O)C1 55526,C1(C)(C(N(CCC)CCO)=O)CCN1C(=O)C(C1(O)CCCC1)F 55527,c1(NC)nc(N(CCCNC(CCCC#CC)=O)C)nc(C)c1OCC.C(=O)OC 55528,C1(C)(NCc2cc(CC)[nH]n2)CCN(c2ccnc(-c3cc(OC)ccn3)n2)C1 55529,C12(C(=O)NCCN(C(Cc3cc(OC)no3)=O)C3CC3)CC(C)(CO1)C2 55530,c1(CCC(=O)NCC(C)NC(=O)C(C)OC2CCCCCC2)nnc(O)nc1O 55531,C(C)(C(=O)NCCC(=O)N1CCCC1)(C(F)(F)F)NC(C(CC)N)=O 55532,N1(C(CCC2(C)CN(C(c3cc[n+]([O-])cc3)=O)C2)=O)CCC(C)(O)C(O)C1 55533,C1(C(N(C2CCC2O)C)=O)CC12CCN(C(=O)Cc1cn[nH]c1)CC2 55534,CCC(C)CCCC(=O)N(C1CCCN(C(c2snc(Cl)c2Cl)=O)C1)CC 55535,c1(C(=O)NCC(CN(C(c2c(C)cncc2)=O)C)O)c(Cl)cccc1[N+](=O)[O-] 55536,c1(C(=O)NC(CCNC(c2c(C)nc(C)[nH]2)=O)(C)C)cccc2oc(C)cc12 55537,c1(C(=O)NC2CC(C)(CNC(c3n(CC)ccn3)=O)C2)ccc(F)cc1C 55538,c1(C(=O)NCC2C3CC2N(C(=O)C(O)C(F)(F)F)C3)cc2c(F)c(F)ccc2[nH]1 55539,c1(CNC(=O)CCc2cnc[nH]2)cc2ccccc2[nH]1 55540,C1(NC(c2c(CC)csc2)=O)CC2CN(C(=O)CC(F)(F)CC)CCN2C1=O 55541,C1(NC(CCC(C)OC)=O)CCCCCC1CNC(=O)CC1(O)CCC1 55542,CCC(C)(CCNC(c1nn(C)cc1Cl)=O)NC(c1ccc(CC=C(C)C)cc1)=O 55543,C(=O)(C1=NNC(=O)CC1)NCC1CCC(F)(CNC(C=CC(CC)C)=O)CC1 55544,c1(C(=O)NC2C(NC(=O)C=CI)CC2)ccc(Cl)s1 55545,N1(C(C(C(=O)OC)OC)=O)CCCN(C(=O)C(C)CC(F)F)CC1 55546,CCC(O)C(C)C(=O)N1CC(C(=O)NCCNC(=O)C2=C(C)OCC2)C1 55547,c1(CN2C(C)(C(N(CC)Cc3ccccn3)=O)CC2)cccc(C(F)(F)F)c1Cl 55548,C(=O)(C1=CC2(CN(C(C3(C)CC(=O)N(C)C3)=O)C2)OC1)NCCCOC(C)C 55549,N1(C(CC2(C(=O)N(C(CC(C)C)C)C3CC3)CC2)=O)CCNC(=O)CC1C 55550,CC1(C)CN(C(=O)CC2CCCCO2)CCC1NC(c1coc(C#N)c1)=O 55551,CC1(C)CCOC1C(=O)NC1C=CCN(C(c2cnc(-c3ccccc3)s2)=O)C1 55552,CC(C)C(=O)C(=O)N1CC(C2CCCN(C(c3ccc(C#N)s3)=O)C2)(O)C1 55553,N1(C(c2cc(COC)oc2C)=O)CC2CC(NC(=O)C3=CCCC3C)C1C2 55554,C1(NC(c2ccco2)C)CCCCN1S(=O)(=O)N1CCCC(C#N)C1 55555,N1(C(C2CN(C(CC(CC)O)=O)C(C)(C)C2)=O)CC(O)C(N=[N+]=[N-])C1 55556,C(CS(=O)(=O)CC(=O)NCC1(C)CN(C(c2ccc(O)cn2)=O)C(C)(C)C1)OC 55557,C(=O)(C(C)(C)C(C)NC(C1CCOC1)=O)Nc1cncc(C)c1 55558,C1(C(=O)NC(CCOC)C(N2CC3(CCOC3)C2)=O)CC2(CCC2=O)C1 55559,O=C(C=CSc1ccccc1)NCCCCNC(=O)COc1ccsc1 55560,C1(C)(CNC(C=CCCC)=O)CN(Cc2cccc(OCCC)c2)CCO1 55561,C(CCF)(C(=O)NCC1CC1(Cl)Cl)NC(Cc1cn(CC)nn1)=O 55562,C(=O)(C#CC(C)(C)CNC(=O)CC1CCC(C)O1)N1C2CC(OC)C2CC1 55563,CC(C)C(F)C(=O)NC1CCCCC1NC(=O)CCSc1ccccn1 55564,Nc1ccnc(C(=O)NC2CCCC2NC(C2CC2C2CCCO2)=O)c1Cl 55565,c1(C(=O)NC2C(NC(C(C)OCC3CC3)=O)CCC2)cc(F)cc(S(N)(=O)=O)c1 55566,c1(C(=O)NC(CNC(C2(NC(N)=O)CC2)=O)CO)cc2n(n1)CC(F)C2 55567,c1(CC)ncc(C(=O)N(C(CNC(c2ccnnc2O)=O)CC)C)cn1 55568,CC(C)CC(C)(CNC(=O)CC1CC1)NC(c1ccc(N2CC=CC2)cc1)=O 55569,N1(C(CCC(=O)N(CC)CC)=O)CCCCC(CNC(=O)C(F)CC2CC2)C1 55570,C1(CNC(C2N(C(C)=O)CCC2)=O)CC2(CO1)CN(C(c1sccc1C)=O)C2 55571,C12(C(=O)NC3CCN(C(=O)CC4CC5C=CC4O5)CC3)CCC(O)(CC1)CC2 55572,CC(C)CC(C(=O)N1CC(NC(C2(C)CCN(C)C2=O)=O)CC(F)C1)C(N)=O 55573,Cn1c(C(=O)NC2COCCC2NC(=O)CCc2cccs2)cc2ccsc12 55574,N1(C(c2c(C)ocn2)=O)CCC(NC(=O)Cn2cc(CO)nn2)C12CC2 55575,c1(N(C)C)cccc(C(N2CCC2CNC(C2CCN(C)C2=O)=O)=O)n1 55576,N1(CC(c2nc(Cl)ccc2Cl)=O)C2CCC1C(F)C(Nc1cc(Cl)ccn1)C2 55577,C=CCC(C(=O)NCC1CC1CNC(C1CC2(CC2)CO1)=O)C(C)C 55578,c1(OCC(=O)NCCC(C)(C)NC(C(COCC)C)=O)cccc(F)c1F 55579,O=S1(=O)CCC2(CCN2CCC(F)(F)C(F)(F)Br)C1 55580,C(N=c1cc(C)[nH]c(=NCCN2CC(C)CC(C)C2)[nH]1)c1ncc(C)nc1 55581,CC1(CC(=O)NCCCN(CCCNC(=O)CCc2cscn2)C)CCCC1 55582,C1(O)(CC(N2C(C(CC)O)CCC2)=O)CCN(C(C2CCCC2O)=O)CC1 55583,CC(C)(C)C(CNC(c1ccc(=N)[nH]c1)=O)C(=O)NC1CCC2(CC2)C1 55584,CCCC(O)C(=O)NC1CC(F)(CNC(=O)CC2CC2)C1 55585,C(=O)(C(F)(F)CCn1cc(CCC(=O)N(C)C)nn1)N(CCC(C)N(C)C)C 55586,c1(C(=O)NC2CCC(NC(CN(S(C)(=O)=O)C)=O)C2)cnn2cccc(Br)c12 55587,Cc1cc(CC(=O)NC2CN(C(c3cccnc3C)=O)CC2C)cc(O)n1 55588,C1(NC(C2CCC(C)O2)=O)CC1C1CCCN(C(C2(CO)CC2)=O)C1 55589,c1(CCCC(N2CC(O)(CCNC(CC(C)O)=O)C2)=O)ccc(CN(C)C)cc1 55590,N1(C(C2(CC)CC2(F)F)=O)CCCN(C(=O)CC2CCC2(C)C)CC1 55591,N1(C(C2(C)CCOC2)=O)CCN(C(c2cc(CO)on2)=O)C(CCO)C1 55592,CC(c1cccnc1)=CC(=O)NC1(C)CCCN(C(=O)CC2C=CS(=O)(=O)C2)C1 55593,Cc1ccc(OCC(=O)NCCCC(C)NC(C2(S(C)(=O)=O)CC2)=O)cc1 55594,C1(C(=O)NC(CC)CNC(C2CCSC(C)C2)=O)Cc2ccccc2N1 55595,c1(C(=O)NCC(CC=C)NC(=O)C(C)S(C)(=O)=O)coc2cc(F)ccc12 55596,C(=O)(CC1CCOc2ccccc21)N1CCC(C(C)Nc2ncccc2C#N)C1 55597,C(N=c1nc(N(N2CCOC2=O)C)c2ccc(C)cc2[nH]1)C1C=C(C)C1 55598,c1(CC(N2CC(OCCNC(C3C(C)CC=CC3)=O)C2)=O)cnn2ccccc12 55599,C1(C(=O)NC2C(NC(C34CC(C(C)(C)C)(C3)C4)=O)COC2)COC(=O)N1C 55600,N1(C(c2cnc(-c3ccco3)s2)C(=O)NC)CC2(CCCC2)C1c1ccco1 55601,c1(C(=O)NC(C)(C)CC2CCC2)ccc(CNC(C23CCCCC2C3)=O)cn1 55602,Cc1cc(Cl)c(Cl)cc1C(N1CC2CC2(C(=O)Nc2ccnc(O)c2)C1)=O 55603,C1(NC(CC2C(C)C2)=O)CC2(CCN(C(C3(Nc4cccs4)CC3)=O)CC2)C1 55604,CC(C)(C)C(=O)CCC(=O)NCC1CCCN(C(C2(C)C=CCC2)=O)C1 55605,CC1ON=C(C(=O)NCC2CCN(C(=O)CCSc3cc(O)nc(O)n3)C2)C1C 55606,c1(-c2cc(-n3cc(C4(C)N(C)CCC4)nn3)n[nH]2)cnc(N)c(N)c1 55607,C=CC1(CC(=O)N(CC(C)O)CCNC(=O)C(C)CC2CCC2)CCOCC1 55608,C(c1ccccc1)=C(C(=O)NC(COC)CNC(C1(CO)CCCC1)=O)C 55609,C(=O)(CS(=O)(=O)C1CCCC1)NCCCC(C)NC(c1c(OC)csc1)=O 55610,Cc1nc(=N)[nH]c(=NCC(C)NC(c2ccc(F)o2)=O)[nH]1 55611,C(=O)(CC(C)(C)CC(F)F)N(C1CCCC1)C(C1CCCC1)CC 55612,c1(OC)ncc(CNC2CCC(C(=O)Nc3cnc(C)nc3)C2)cn1 55613,c1(CC)cccc(C(=O)NC2CC23CC(NC(=O)CCNC(=O)CC(C)C)C3)c1 55614,C1(CNS(=O)(=O)Cc2ccccn2)CCCN(C(=O)CCCCBr)C1 55615,c1(CC(=O)NC2CCN(C(=O)C(F)CC3CCC3)C2)ccn(C(CC)CC)n1 55616,CC(C)CC(C(=O)NC1CN(C(c2cnn(C)c2C#N)=O)CC1O)NC(N)=O 55617,CC1(C)CN(C(c2ncoc2CN)=O)CC(CNC(=O)CCC2(C)CC2)O1 55618,Cc1nc2cc(C(=O)NCC(C)N(C(=O)CC3CC(O)C34CCC4)C)ccc2o1 55619,c1(C(=O)OCC)ccc(C2CCCCN2C(C2COC(C)C2)=O)n1C 55620,C(=O)(C1(C)CCc2ccccc21)N1CC(F)CC(NC(COCC(=O)OC)=O)C1 55621,CC(O)C(C)(C)C(=O)N1CSCC1C(N1CC2CSCC2C1)=O 55622,C(=O)(C1CCc2ccccc21)NC1CC(CNC(c2cn(C)nn2)=O)CC1O 55623,C(C(=O)NN1CCCC1CO)c1n(CC)cnn1.N12CC(CC(C)(C)C1)NC2=O 55624,S(=O)(=O)(c1ccc(Cl)cc1F)NC1C(C#N)CN(C(=O)Cc2cccs2)C1 55625,c1(SCCNC2OCCN(C(c3ccccc3)C)CC2)c[nH]c2cc(F)ccc12 55626,C(CCc1ccccc1)(C(F)(F)F)NC(C(n1ccc(C2CC2)n1)C)=O 55627,Nc1cc(F)cnc1C(=O)NC1CC(CCNC(c2sccc2C2CC2)=O)C1 55628,N#Cc1ccsc1C(=O)NCc1ncccc1C(=O)NOCC1CCCCC1 55629,N1(C(C=Cc2ccc(CC)o2)=O)CC(NC(c2cnn3ccsc23)=O)CC1(C)C 55630,C(=O)(C(CC(C)(C)C#N)N1CCSC2CCC12)NCCCSC 55631,C1(CCC)CN(C(=O)Cc2nccn2C)CC1NC(c1nscc1C)=O 55632,C(=O)(C1(C)CCn2ccnc21)NC1CC(CNC(c2cc(OCC)ncc2)=O)C1 55633,c1(C(N(CCNC(CC=CCC)=O)CCC)=O)cc(Cl)cn1CC 55634,N1(C(=O)Nc2c(NCCN=[N+]=[N-])ccc(Cl)c2)CCC2(CC1)CC2c1nn[nH]n1 55635,C1(NC(CCCCCC)=O)CN(C(c2cnn(C)n2)=O)C2(CCOC2)C1 55636,C1(C(N2C(C(=O)NC3C(C(C)(C)C)C3)C(O)CC2)=O)CC2CC(=O)C1O2 55637,CC1(C)CC(NC(C2(CF)CCC2)=O)CN1C(C1CCCCC1O)=O 55638,C(=O)(C1c2c[nH]nc2CN1C(C1CC12CCCCC2)=O)NC1CC(CC(=O)OC)C1 55639,c1(C(=O)NC2CC(C)(NC(=O)CC3CC=CCC3)C2)cc(F)ccc1F 55640,C=CCCCCC(=O)N(CC(C)N(C)C(C1CCN(CC)CC1)=O)C 55641,C1(C(=O)NCC(C(C)C)NC(C2CCN(C3CCCCC3)C2)=O)CCCC2CC12 55642,c1(C(=O)NCC2C(NC(C(CCSC)O)=O)C2)occ2c1CCOC2 55643,c1(C(=O)NC2C(NC(C=NOC)=O)COC2)cnc2c(c1)NC(=O)CS2 55644,N1(CC(=O)NC2C(NC(C3(OC)CCCOC3)=O)COC2)CC(=O)N(C)C1=O 55645,C(=O)(CC(C)C(F)(F)F)N(CC(C)N(C(CSc1nnc(C)o1)=O)C)C 55646,c1(C2(C(=O)NC3C(NC(C(C)C=Cc4ccccc4)=O)C3)CC2)cc(F)ccc1F 55647,N1(C(C(N2CCSCC2)C)=O)CCCOC(CCNC(=O)CC(C)CN(C)C)C1 55648,C=CCCC(C)(C)C(=O)N1CC(CNC(=O)CC(C)N(C)C)C(O)C1 55649,C1(C)(NC(C=CCCC)=O)CCN(C(=O)Cc2c[nH]c(=N)nc2O)CC1 55650,C(=O)(C(O)C(C)(C)C)Nc1cc(C)sc1C.C12CC1C(=O)N2 55651,c1(C(N2CC3(CCCN(C(C(C)C(F)F)=O)C3)C2)=O)cn(C)c(=O)c2cncn12 55652,c1(C(N2CCC(NC(C3C(CC(C)C)C3)=O)CC(O)C2)=O)ccc(F)c2occc12 55653,c1(C(=O)NCC2CCN(C(C=CC)=O)C2(C)C)cc([N+](=O)[O-])cc2c1OCCO2 55654,CC1c2ccsc2CCN1CCOc1cc(F)ccc1N 55655,N1(C(C(C(=O)OCC)F)=O)CCN(C(c2cc(C(C)(C)C)on2)=O)C(COC)C1 55656,c1(C(=O)NCC2N(C(C3(C)CCC(=O)NC3)=O)CCC2)cc(F)cc2nc[nH]c12 55657,C12(C(=O)NC3CC(C(C)C)OC3)CC(CN(C(c3cc(C#N)n(C)n3)=O)C1)C2 55658,C12(NC(c3ccc(OC)nn3)=O)CCC(CNC(=O)C(O)C3CCC3)(CC1)OC2 55659,C(=O)(C(=O)C(C)CC)NCC(CNC(CCCOCC=C)=O)(C)OC(C)=O 55660,C(C)(C)(C(=O)NO)NC(C=CC(C)NC(c1ccnnc1O)=O)=O 55661,N1(C(CCC2OCC(C)(C)C2)=O)CCOCC(NC(c2cccc(Cl)c2Cl)=O)C1 55662,c1(C(=O)NC2CC3(C(NC(CC(CC)SC)=O)C3)C2)ccc(OC)cc1F 55663,C(C1=CCCSC1)(c1n(CC(=C)C)nnn1)SCCNc1ccc(CC)c(Cl)c1 55664,c1(C(N(C)CC2N(C(C3ON=C(CC)C3)=O)CCOC2)=O)ccc2ncnn2c1 55665,S(=O)(=O)(c1ccc(N2CCC(C)C2)cc1Cl)NCc1cccc(OC)n1 55666,C(=O)(CC(C)C(F)F)NCc1c(C(N2CCCC(C(=O)NC)C2)=O)nco1 55667,CC1c2c[nH]nc2CCC1C(=O)NC1CCN(C(=O)CC(C)(F)F)CC1F 55668,c1(C(N(CC(C)NC(C(C(C)C)OCC)=O)C)=O)ccc(Cl)cc1[N+](=O)[O-] 55669,C(CCC(C)C(=O)N(C1C2CN(C(=O)COCC3CCCO3)CC12)C)OC 55670,C(=O)(C1SCc2cccnc21)N1CC(CNC(CN(C)CC)=O)C(F)(F)CC1 55671,c1(OCC(=O)NC2CN(C(=O)Cc3cc[nH]n3)C2)ccc2c(c1)CCCC2 55672,C(CC(C(=O)N(C)Cc1ccoc1)NC(c1c[nH]nc1C)=O)OCC 55673,N1(C(COc2cccc(C)c2)=O)CC(NC(=O)CC(F)F)CC(C)C1 55674,c1(OC)ccc(C(=O)NC2CCN(C(c3nc(C)ccc3C)=O)CC2C)c(F)n1 55675,C(=O)(C#CC1CCCOC1)N(C)CC1(C)CCCC1NC(=O)CCC(F)(F)F 55676,C1(OC)CN(C(=O)COCc2nc(=O)n(C)[nH]2)CC1NC(c1nc[nH]n1)=O 55677,c1(OC)cc(CC(C)NCC(C)OC(C)(C)C)ccc1O 55678,CCCCC(C(=O)N1CCN(C(C2OCCCO2)=O)C(COC)C1)C(C)C 55679,C(=O)(CCC(N)=O)NCC(C(=O)NC(COC)(C)C)OC 55680,CC1OCCC1C(=O)NC(C1(CNC(c2ccc(CC3CC3)s2)=O)CC1)C 55681,Cn1ncc2cc(C(N3C4CCC3C(NC(=O)CCC3CCCC3)C4)=O)ccc12 55682,N1(C(C2(C(F)(F)F)CCOCC2)=O)CC2CC(C1)C2N=c1[nH]ncs1 55683,N1(C(c2cnn(CC)c2Cl)=O)C2CCCC1CN(C(C13CCCN1CCC3)=O)C2 55684,N1(C(C(Cc2ccc(OC)cc2)C)=O)CCN(C(=O)C=CCBr)C(C(F)(F)F)C1 55685,c1(CC)c(C(=O)N(C)CC2CCN(C(=O)CNC=O)C2)nnn1C 55686,N1(C(c2cc(C(C)C)no2)=O)C(C(=O)NCCOC(F)(F)F)CC2CCCC12 55687,C(C(N=[N+]=[N-])C(=O)N1CC(NC(C2CC2(C)Br)=O)CCC1C)OCC 55688,CN1CCc2[nH]nc(C(=O)NC3CCC(CCNC(=O)C=CC4CCC4)C3)c2C1 55689,C(CC(=O)N=c1ccn(CCF)[nH]1)(C(F)(F)F)NC(C1(C(C)C)CC1)=O 55690,c1(NCc2ccccn2)ccc(-c2cncnc2)cc1 55691,Cc1ccc(C(=O)NCC2CCCCN2C(c2cnsc2)=O)c(N)n1 55692,c1(C(=O)NCC2N(c3nccc(OCC)n3)CCOC2)cc(F)cc(Br)c1C 55693,CCCC(CCC)=CC(=O)NCCOC1CCN(C(C2C3(CC3)C23CC3)=O)C1 55694,CC(C)C1=NOC(C(=O)N(C)CC2(O)CCCN(C(=O)C=CC(C)(C)SC)C2)C1 55695,Cc1ccnc(C(=O)NCC2CCCC(NC(=O)COCc3nc(C)no3)C2)n1 55696,C12(C(N3C(C(=O)OC)C(C)CC3)=O)CCN(C(C3C4CC(=O)CC34)=O)CCC1C2 55697,N1C(=NCCC(F)F)NCC(F)=C2CCN(C2)Cc2cccc(c2)C1.CCC=C.SC 55698,C1(NC(c2nc(-c3ccc(C)o3)sc2)=O)CN(C(C2(O)COC2)=O)CC1C(F)F 55699,c1(C(=O)NCCC(CNC(CCc2cc(C)on2)=O)O)cccc(CC#N)c1 55700,C(CCN=c1[nH]c2ccc(Br)cc2s1)OCCNC(C1CC2C=CC1C2)=O 55701,c1(C(N2CC3C(C(=O)OC)C3C2)=O)ccc2cccc(OC)c2n1 55702,CC1(CNC(c2cc(O)cs2)=O)CCCN1C(c1nc(Cl)c(Cl)s1)=O 55703,C#Cc1cnc(C(=O)N(CCC(C)NC(c2cccc(CC)c2F)=O)C)c(C)c1 55704,n1(CC=C)c(=O)c2ccccc2n2c(=S)n(CN3CCCC3(C)C)nc12 55705,c1(NCC(=O)NCc2ccc(N(C3CCCC3)CC)cc2)cccc(F)c1[N+](=O)[O-] 55706,C1(CC)(CC)CC(NC(=O)C(=O)N(C)C)CN1C(=O)C(C)Oc1cccnc1 55707,c1(CNC(C(CNC(c2cc(CC)oc2C)=O)N(C)C)=O)nn(C)c(=O)n1C 55708,c1(C(=O)NC(C(=O)N(CCO)CC)c2ccco2)cccc(O)c1F 55709,C12CCN(C1C)C2=O.C1(OC)CCN(C(=O)C(N)=O)CC1 55710,C1(C(N2CC(C(=O)NCC3CC(OC)CN3C(C)=O)C2)=O)Cc2nccnc2C1 55711,C(=O)(C(C)CCCOC)N1C(CC(NOCC(CC)C)=O)CCC1 55712,C1(CNC(CCOCC#C)=O)CC2(CO1)CN(C(=O)C(C)(C)CC=C)C2 55713,C1(CNC(CNC(=O)OC)=O)CCC2(CO1)CC(NC(C1(C)COCCO1)=O)C2 55714,C1(C(N(C)CC2CN(C(CC=CC)=O)C2)=O)CCC(C)C1 55715,C12(CNC(C3CC(C#C)(O)C3)=O)CCCC1N(C(=O)Cc1occc1C)CCC2 55716,c1(NC(=O)NC2CC2c2ccc(-n3cnnn3)cc2)ccc(C(F)(F)F)cc1 55717,n1(CCOC)nc(CSc2ccccn2)nc1-c1ccc(CCC(C)C)nc1 55718,C(CCCC(C)NC(C1CC12CC2)=O)NC(C1(CCOC)CC1)=O 55719,C=C1CON(C(=O)CC2CCN(C(=O)Nc3ccc(C)cc3)C2)C1 55720,N1(C(C(COC)(C)O)=O)CC(NC(c2ccc(OCCF)cc2F)=O)CC(O)C1 55721,N1(C(=O)NC(CC(C)C)c2ccccc2)CCc2cc(Cl)ccc2C1 55722,CC1(C)CC(NC(=O)CC2Cc3ccccc3N2)CN1C(C1CNC(=O)C1)=O 55723,C1(NC(C(c2cn(CC)nc2)=O)=O)CCCCC1CCNC(C1CC1CF)=O 55724,N1(C(CN2CCCC(CC)C2)=O)CCN(C(c2ccc(O)cn2)=O)C2(CC2)C1 55725,C1(C(=O)NCCN(CC(C)O)C(c2ccn(C3CC3)n2)=O)CC12CC(F)(F)C2 55726,C1(O)(C(C)NC(Cc2n(C(C)C)cnn2)=O)CCN(C(=O)C=CC2CCOC2)C1 55727,CC(CC(=O)N(C)CC1CCCCN1C(C1CCCO1)=O)P(C)(C)=O 55728,CC(C)C(CNC(C12CCC(CC1)C2)=O)C(=O)NC1CCCC(O)C1O 55729,CCCC(CCC)=CC(N1CCC(CNC(=O)Cc2nc[nH]n2)(OC)C1)=O 55730,CC(C)CC(O)CC(=O)NC(C1CCCN1C(=O)C(C)CO)C 55731,C12CCN(CC1)CC(=O)N2.C1(CN(C(=O)OC(C)(C)C)C)CC1(F)NC(C)(C)C 55732,C(=O)(CCCCCO)N1C(C)CC(NC(c2ccc(C(=O)CF)cc2)=O)C1 55733,N#Cc1c[nH]cnc1=NCC1(F)CC(NC(c2ccnc(Cl)c2Cl)=O)C1 55734,C1(CNC(C2(C=C)CCC2)=O)CC2CCC(C1)N2C(c1ccnn1C(F)F)=O 55735,C1(C(CN([N+](C)(C)C)CC)O)CS(=O)(=O)CCO1 55736,c1(C(C(=O)NC2CCCC2)N(CCOC)C)cc(OC)c(F)cc1F 55737,N1(C(C(=CC2CCCC2)C)=O)CCCC(CCNC(c2cc(C)ccn2)=O)CC1 55738,c1(C(=O)NCC2N(C(c3c(C)cn(C)c3)=O)CCC2C)cc2c(C)n[nH]c2cn1 55739,C12(C(=O)NCC(CC)NC(c3cc(C(C)=O)n[nH]3)=O)CC(c3ccccc3)(C1)C2 55740,c1(CN2C(C(=O)Nc3ccc(CCO)cc3)CC(F)(F)C2)cc(Br)c(O)cc1O 55741,C#CCC(C)(C)C(=O)N1CCC(COC)(NC(C2CC2CC(C)C)=O)C1 55742,c1(CC(N2C(C)(CNC(C(C)OCCC#C)=O)CCC2)=O)cc(F)cc(Cl)c1 55743,c1(C(=O)NCC(CNC(CC2CC(=O)NCCC2)=O)O)ccc(F)c2ccsc12 55744,c1(NCC(C(C)C)O)ccc(S(=O)(=O)NC2CC3OCCCC23)c(Br)c1 55745,N1(C(C(C)N(C)C)=O)CCN(C(c2cncs2)=O)CC1c1cc(F)ccc1F 55746,C(=O)(CC1CCCc2c1[nH]c1ccccc21)OC(C1C(OC)C2C1CC2)=O 55747,C1(CSC2CCOCC2)CN(C(=O)C(F)=C(C)C)CCN1OC 55748,C1(CC(N2CCOC(CNC(C3(F)CCOC3)=O)C2)=O)C=CS(=O)(=O)C1 55749,N1(C(CC(=O)N(C)C)=O)CCCC(O)(CNC(c2ccc(=O)n(C)c2)=O)CC1 55750,C1(OC)CC2CC(=CC(=O)NCC(CCNC(C)=O)(C)C)CC12 55751,N1(C(CCOCCOC)=O)CCC2CN(C(c3nccc4[nH]ccc34)=O)CC12 55752,C1(C(N2CC(CCC)C(NC(C3CCOC3(C)C)=O)C2)=O)COCC(C)(C)O1 55753,N1(C(COC(CC)C)=O)CCCCC1CN(C)C(c1sc(F)cc1Br)=O 55754,c1(CC)ncoc1C(=O)NC1CC(CNC(=O)CN(C)C(=O)OC(C)(C)C)C1 55755,c12cc(cc(Cl)c1)C2.C1(CCn2cc(CCN)nn2)CCS(=O)(=O)N1 55756,C1(NCC(c2ccccc2)OC)CN(C(=O)C(=O)NC2CC2)CC1CC(C)(C)C 55757,C1(NC(CC2(C)CC2(Cl)Cl)=O)CC2CC(C1)N(c1ncc(Br)c(O)n1)C2 55758,Cn1cncc1C(=O)NCc1ocnc1C(=O)NCCC1CC1C1CC1 55759,Cc1cc(-c2nc(Cc3ccc(F)cc3)nn2CC2CC2C)oc1Br 55760,C1(O)(CNC(=O)C(O)C2CC2)CN(C(=O)CC2CCOC2=O)C1 55761,C(C(CC(C)C)C(=O)N1CCCC(NC(c2cn(C)c(=O)cn2)=O)C1)OC 55762,c1(C(=O)NCC(C)N(C(c2cccc(CC)c2)=O)CC)cnc2n1CCC(C)C2 55763,Cc1cnc(C(N2CCCC(CC(N3CCCC(OC(C)C)C3)=O)C2)=O)cn1 55764,C(=O)(C1(C)OCCc2ccccc21)NCC(C(C)C)(C)NC(C12CC(CO1)C2)=O 55765,c1(C(N2CCC(O)(CNC(C3C(OC)C3)=O)CC2)=O)cc([N+](=O)[O-])ccc1Cl 55766,c1(CN(C)CC2CCC(C)(C)CC2)cc(=O)c2cc(Br)ccc2[nH]1 55767,c1(CC(=O)NCC23CC(CC)(C2)C3)ccc(O)cc1.N1(C2CC2)CCC1C(=O)N 55768,c1(OC(C)C)cncc(C(=O)NC(C)C(C)NC(=O)C(C)(C)c2ccccn2)c1 55769,CCCCC(O)C(=O)NC(C1CCN(C(c2cccc(CN(C)C)c2)=O)C1)C 55770,C1(CNC(c2cnco2)=O)COCCN(C(C2(CC(F)F)CC2)=O)C1 55771,N1(C(C2(CC)CCCN(C(=O)CC3CC4CCC3O4)C2)=O)CC(C)CCCC1C 55772,c1(C(C(=O)NCC(=C)C)N(CCC=C)CSCC=C)nccc(Cl)c1F 55773,c1(C(C(=O)NC(C)C)N(CC=C)Cc2cccnc2)c(Cl)c(C)nn1C 55774,c1(CC(=O)NC(c2noc(C)n2)CC)ccoc1C 55775,c1(C(=O)NCC2CN(C(=O)C(F)(F)CC3CC3)CC2(F)F)cccc2c1CCO2 55776,N1(C(C(c2ccccc2)C)=O)CCC(CCCNC(C2CC2C)=O)CC1 55777,C(=O)(C(C)C1=CCCC1)N1CCCCC(N(C(c2cccc(C#C)c2)=O)C)C1 55778,CC(C)CCN=C(NC1CN(C(=O)OC(C)(C)C)C1)NC1C(O)CC1(C)C 55779,CCC(C)C(C)NC(C1(CCNC(=O)C(C)c2cccs2)CC1)=O 55780,CCC1=NOC(C(=O)NCC2CC(C)N(C(=O)CCc3cnccn3)C2)C1 55781,c12ccc(nc1)[nH]c2=O.CCC(C(=O)NCC(C)(O)C1(C)CC1)NC(C)=O 55782,c1(C(=O)N)cc[nH]n1.C1(=O)CCN1.C1(=O)COCC(=O)NCC(C2CC2)N1C.CN 55783,C(CC(C)C(=O)N1CC(OCCNC(c2cnc(C(C)OC)s2)=O)C1)OC 55784,c1(N2C(=O)CC(C(N3CCC(OC)C3)=O)C2)ccc(Cl)c(F)c1 55785,c1(CC(N2CCC(C(C)NC(C3(CC=C)CCC3)=O)CC2)=O)ccc(F)c(C)c1 55786,CCCCCCC(CC)C(=O)N1C2CCC1CN(C(C13CCCC(CO1)C3)=O)C2 55787,CC(Cc1ccnn1C)C(=O)OC1COCC1N(C)C 55788,c1(N2CC(C)C(CO)CC2)nc2c(c(=NCCN(C)C)[nH]1)CCCCC2 55789,c1(CNC(C=C2CCC(C)CC2)=O)cc(O)nc(CNC(=O)CC2OCCC2C)n1 55790,Cc1ccc2c(c1)C=C(C(=O)NC1CCOC(CNC(C3CC3F)=O)C1)CO2 55791,N1(C(C(CCC)O)=O)CC2CC(C1)CN(C(=O)C(F)C(F)(F)F)C2 55792,C(=O)(C(CC1CCCCC1)C(C)C)N1CCC(N(C(CCC)=O)C)CC1 55793,C(CC(F)CN=[N+]=[N-])NC(C(CC=CC)NC(C1OC2CCC1C2)=O)=O 55794,c1(OC)[nH]c(=N)ccc1C(N1CCN(C(C)CNC(C2(CO)CCC2)=O)CC1)=O 55795,N1(C(CC2C(C)C2(F)F)=O)CCC(CNC(c2cc(C(C)(C)C)n[nH]2)=O)C1(C)C 55796,CC1CN(C(=O)CC(F)F)CC(CCNC(=O)C(c2ccccc2F)(C)C)O1 55797,CCC(C)C(O)C(=O)N1CCCCC1CCNC(=O)CN1CCCC(CC)C1 55798,CC(C)C(CCC(=O)NC(C)(C)CF)NC(=O)Cc1cn(C)cn1 55799,C#CC1(C(=O)NC(C)COCC)CCN(C(=O)C2=CCCSC2)CC1 55800,c1(C(C)=O)ccc(C)nc1NCC(C)CNC(C1CCOC(C)(C)C1)=O 55801,C1(C(=O)NCC=CCNC(=O)C(Cc2cccc(Cl)c2)=NO)CCC2CCC(=O)N12 55802,C1(F)(CNC(=O)CCF)CC2CCC(C1)N2C(=O)C=Cc1nccs1 55803,C(=O)(C(F)C(F)(F)F)N(C(CNC(c1cccc(CC)n1)=O)C)CC 55804,C(=O)(C1=NNC(=O)CC1)N(CC(CC)NC(c1ccc(Br)c(N)c1)=O)CC 55805,C=CCC(C(=O)NCCC1(CNC(=O)CN=S(C)(C)=O)CC1)C(C)(C)C 55806,CC1=C(C(=O)N2CC(NC(C3(C)CCCS3(=O)=O)=O)C(F)C2)SCCO1 55807,N1(C(C(CC)CO)=O)CCC(NC(C2(O)CCSC2)=O)C(C)C1 55808,[N-]=[N+]=NCC(C(=O)NCCOC1CCCC1)NC(C1CC2(CC2)CO1)=O 55809,c1(CNC2C3CN(C(c4occ(C(C)C)n4)=O)C2C3)cnc(N(C)C)c(Cl)c1 55810,N1(C(CCC=C)=O)CCC2(CC1)CN(C(=O)C(C)CCCOC)C2C(C)C 55811,c1(OC)ccccc1CC(=O)N1CCC1CNC(c1oncc1C)=O 55812,c1(CC)cc(C(N2CCC(=CC=CCNCC(=O)O)CC2)=O)c(C)nn1 55813,CCC(CC)C(=O)NCC1CC(NC(c2cncc(C(=O)OC(C)(C)C)c2)=O)C1 55814,C1(CC(=O)NC2(C#C)CC2)COCCN1C(=O)Cc1cnoc1 55815,C1(CC=C)(NC(c2cccc(C3CC3(F)F)c2)=O)CCN(C(C2CCSC2)=O)C1 55816,N1(C(c2cn(CC)nn2)=O)CCC2CN(C(=O)Cn3c(C)cc(O)cc3=O)CC12 55817,c1(C(N(C2CN(C(C3(CC=C)COC3)=O)CC2F)C)=O)ccc(=O)n(CCF)n1 55818,CC1(C)CC(c2nnnn2C2(C)CC2)(C2CC2)N=C1C(=O)CC(C)(C1CC1)CO 55819,C(CCCCC(=O)N1CC2CC(C1)C2NC(c1ncc(N)cc1Cl)=O)OC 55820,N1(C(C2N(C(C)=O)CC(O)C2)=O)CC2CCC2(NC(C2CC3CC3C2)=O)C1 55821,CC1(C)CCN(C(C2CCN(C(=O)CC3CCC(=O)N3)CC2)=O)CC1 55822,c1(CC(=O)N(C)CCNC(C2(Cc3cc[nH]c3)CC2)=O)ccc([N+](=O)[O-])cc1Cl 55823,C(C(=O)N1OC2CCC1CC2)N1CCN(C(=O)Cc2ccon2)CC1 55824,Cn1nc(C(N2CC=C(CNC(=O)Cc3cccnc3)CC2)=O)c2c1CCSC2 55825,C(=O)(CC(CC)C(C)(C)C)NC(CNC(CCCOCC=C)=O)C(C)(C)C 55826,CC1(C)C2CCC1(CC(N1CCN(C(=O)C#CC3CC3)CC1C(F)F)=O)CC2 55827,N1(C(C(CC)SC)=O)CCCCC(N(C(c2ccoc2C(F)(F)F)=O)CC)C1 55828,c1(NC(C2CC23CCN(C(c2cc(Br)cc(I)c2)=O)C3)=O)cc(I)ccc1CO 55829,N1(C(CNC(CCC)=O)=O)CCC(C)C(NC(c2ccc(C3CC3)c(Cl)c2)=O)C1 55830,c1(C(=O)NCC2(C)C(C)CN(C(c3ccncc3F)=O)C2)nnn2c1CSCC2 55831,N1(C(c2ccnc(C)c2C)=O)CCOC2(CCN(C(c3[nH]cnc3C#N)=O)C2)C1 55832,N1(C(C2CCC(N(N3CCOCC3)CC(F)(F)F)CC2)=O)CCCC(CO)CC1 55833,C=CCC(CNC(=O)CCn1cncn1)C(=O)Nc1ccc(O)nc1 55834,c1(C2(C(=O)NC(C)CCNC(C34COCC3C4)=O)CC2)c(Cl)cccc1Cl 55835,C1(CNC(c2scc(C)c2Cl)=O)CC2(CC2)CN1C(=O)CCc1nnc(S)n1C 55836,c1(C(=O)NCC2CC(OC)CN2C(c2cnccc2Cl)=O)ccc(=O)n(C)n1 55837,CC(C)CCCC(=O)N1CC(O)CCC1C(=O)NCc1cccnn1 55838,Cc1cc(C(=O)NC2CC2C(=O)NCCCOc2ccc(Br)cc2)c(C)n1C 55839,c1(C(=O)NC(C(C)C)(C)CNC(C2(O)CC2)=O)ccn2cnnc2c1 55840,c1(CNC(c2c3c([nH]n2)CC(C)CC3)=O)cc2c(cc1O)OCO2 55841,c1(NC(c2nc(C)sc2)C)nc(N2CCc3sccc3C2)nc2sccc12 55842,C(=O)(CCCCC(N)=O)NC1CCCC(NC(COc2c(C)cccc2Cl)=O)C1 55843,C(C(CC(F)(F)F)NC(C1(CO)CCOCC1)=O)NC(c1cnc(OCC)nc1)=O 55844,C(C)(CNC(=O)Cc1cnc(C(F)(F)F)s1)(CO)NC(C(C)OCCC(C)C)=O 55845,C1(CNC(C2CCCC2c2nc[nH]n2)=O)CCCCN1C(c1ccsc1Cl)=O 55846,Cc1coc(C)c1CNC(C)(CNC(=O)CCC1CCC(C)O1)C1CC1 55847,C1(NC(CSCCC)=O)CN(C(c2cnn(CC)n2)=O)CCC1c1ccccc1 55848,c1(OCC)nc(C(=O)NC(CNC(c2ccn(C3CCOCC3)n2)=O)CC)ns1 55849,c1(CC(=O)NC2CN(C(CCNC(=O)Nc3cccs3)=O)C2)cccc(F)c1 55850,c1(CC)cc(Cl)ccc1NC(=O)N(C(C)(C)CC)C(c1cccc(Cl)c1)C 55851,N1(C(C(CCCC)O)=O)CCC(C2CCN(C(c3c(C)noc3C)=O)C2)CC1 55852,c1(C(=O)NCC(C)(C)CNC(c2cncc(C3CC3)c2)=O)ccc(CCO)cc1 55853,C12(CNC(C(C)C3CCOC3)=O)CC(CO1)N(C(c1scnc1Cl)=O)C2 55854,C(=O)(CCC(C)CN(C)C)NC(C(N1C(C)(C(=O)NC)CCC1)=O)C 55855,CC1(C)CN(C(=O)C#CC2CCOC2)CCC1NC(c1ccccc1)=O 55856,C#CCCN=C(NCc1cnccc1O)NC(C)CC 55857,c1(C(N2C(CNC(C3(C)CCOC3)=O)CC2)=O)ccc(Cl)cc1C(N)=O 55858,C1(C2CC2)(C(N2CCC(NC(c3sccc3F)=O)CC2)=O)CC=CC1 55859,c1(C(=O)NCC2(CCNC(CC)=O)CC2)cccc(C2(S(C)(=O)=O)CC2)c1 55860,C(=O)(C(CNC(=O)CCC1CCC1)CC(C)C)NCCc1ccc(C)s1 55861,C(=O)(C(CO)C(C)(C)C)NC(CCC)C(=O)NCC1(C)CCCC1O 55862,N1(C(C(=O)Nc2cccc(C)c2)=O)CCN(C(c2cnc(C)n2C)=O)C(C)C1C 55863,Cc1cc(F)ccc1CNC(=O)C(c1ccncc1)N1CCCC1C1CCCC1 55864,c1(C(=O)NC2C(C)CN(C(=O)CSC(F)F)C2)cccc(C#CCC2CC2)c1 55865,C12(CNC(C3(N(C(=O)Cc4cnns4)C)CC3)=O)CCCC1CCC2 55866,c1(CNC(=O)Cc2cnoc2)ccnc(C(=O)NC2CCS(=O)CC2)c1 55867,C(CN=c1[nH]c(N2CC(C(=O)NC)CC(C)C2)nc2ccccc12)=CC 55868,N1(C(C(C)NS(C)(=O)=O)=O)CCOCC1CN(C)C(c1csnn1)=O 55869,c1(NCC(C)S(C)(=O)=O)ccc(S(=O)(=O)N2CCN(CC(C)(C)F)CC2)cc1Cl 55870,O=C1CN(CC2CC2C2CCCC2)C(=O)N1Cc1cnsc1 55871,CC(C)C(C(=O)NCC(C(C)C)NC(=O)COc1cnn(C)c1)NS(C)(=O)=O 55872,C1(CCNC(C(C=C)(C)O)=O)CN(C(=O)C(C)OC2CCOC2)CCCO1 55873,N1(C(C(CSC)O)=O)CC2(CCN(S(=O)(=O)c3cc(C)ccc3F)CC2)CC1C 55874,C1(CCN(C(C(Cn2ccc(C)n2)C)=O)C)CCN(C(=O)CSCC(N)=O)CC1 55875,CCC(C)CC(C)C(=O)NC(CNC(c1ccccc1CO)=O)(CC)CC 55876,c1(NCC2(C)CN(Cc3sc(C)c(Br)c3)C2)ccnc2ccnn12 55877,N1(C(=O)COCC2CCCO2)CCCN(C(C2COC3CC2C3)=O)CC1 55878,N1(C(c2c(C)cn(C)c2)=O)CCCC(O)(CCNC(=O)CC2COCCO2)C1 55879,C12(CNC(c3nc(C)nc(O)c3)=O)CCCC1CN(C(=O)C(F)(F)CC(C)C)C2 55880,C(CC(N)=O)(C(=O)NCC1(O)CCCC1(C)C)NC(CCC1CC(OC)C1)=O 55881,C1(C#N)(C(=O)NCCN(C(C2CCCS2)=O)CC)CC1 55882,c1(NC(c2nnn(C)n2)c2n(CC3CC3)nnn2)ccc2c(c1)CC(O)C2 55883,C(N=c1[nH]cnc2[nH]cc(C(F)F)c12)C1CCCN(C(c2ccc(F)s2)=O)C1 55884,C=C=CC(C)C(=O)N1CCC(OCCNC(C2CCC(=O)N2CC)=O)C1 55885,Cc1nn(CC(=O)NC2CC(NC(=O)C(C)CN(C)C)C(O)C2)c(C)c1[N+](=O)[O-] 55886,c1(NC2C(C)COCC2)[nH]c(=NCc2sncc2Br)nc2c1ncn2C 55887,c1(C(N2CC(C)(C)C(NC(=O)C3=CCCS3)C2)=O)ccn2ncccc12 55888,CC(C)(CNC(=O)C=CCO)CC1CN(C(c2cnc(C(F)F)s2)=O)C1 55889,CCCCCC(=O)NC1COCCC1NC(c1cnc(C2CC2)[nH]1)=O 55890,C1(CC(N2CCC(O)(CNC(C3CC(OC)C3)=O)C2)=O)CC2(CCC2)CO1 55891,c1(CC(=O)NCCNc2cn(CC(=O)N(C)C)nn2)cccnc1O 55892,C1(CC=C)(NC(c2cnn(C)c2OC)=O)CCN(C(=O)CC2CC2C)C1 55893,C(=O)(C1=NOC(C)C1C)NC(C1N(C(c2ccc(OC)cc2OC)=O)CCC1)C 55894,C(CC(C)(C)C)(C(=O)NCCC1CC(C(=O)N(C)Cc2cn(C)cn2)C1)OC 55895,c1(C(N(C)Cc2ccc(C)cc2Br)=O)n[nH]c2cccc(F)c12 55896,C1(NC(CCc2cn(C)nc2)=O)CN(C(C2CCCS(=O)(=O)C2)=O)CCC1F 55897,Cc1ccc(C=CC(N2CCC(NC(=O)CC3(C)CCCO3)CC2)=O)s1 55898,C(CN=c1[nH]c(=NC2CCC(C3CC3)CC2)[nH]c2c1SCC2)C1(OC)CCC1 55899,C1(C(N(CCCNC(c2ccnc(OC)c2F)=O)C)=O)COc2ccccc2O1 55900,CN1C(=O)CCC1CC(=O)NC1CC(CC(=O)NCC(F)F)C1 55901,CC(C(=O)NC1(C)CCN(C(c2ccccc2OC2CCCCC2)=O)C1)C(F)F 55902,C(C(=O)NCCCN(C(=O)CO)C(C)C)(C1CC1)SC 55903,C1(C)(C(N2CCC(C)(NC(c3cnc(C#N)s3)=O)C2)=O)CC(C2CC2)=NO1 55904,N1(C(C(CC=CCC)C)=O)CCC2(CC2C(=O)NC2CCNC(=O)C2)C1 55905,c1(C(=O)NCC(CCCC)NC(=O)C(O)C(C)(C)CC)cccc2ccncc12 55906,Cc1c(C(=O)NC(C)C(C)CN(C)C)ccn1CCO 55907,c1(C(N2C(CNC(CC(C)N(C)C)=O)CC3(CC3)C2)=O)cccc2nccn12 55908,C1(NC(c2c(C)cc[nH]2)=O)CN(C(=O)Cc2ccccc2CS(N)(=O)=O)CC1O 55909,N1(C(C(C)N(C(CC(=O)NCC)=O)C2CC2)=O)CCOC(C)(C2CC2)C1 55910,N1(CC(=O)NC(CC)CNC(=O)C(F)(F)c2cnnn2C)CCN(C)C(=O)C1 55911,N1(C(C(COC)C)=O)CC2(CCN(C(=O)C(C)Cc3ccncc3)CC2)C1 55912,N1(Cc2cn(CC(C)C)nc2)CCC(C)(CNC(c2ccc(I)c(O)c2)=O)CC1 55913,c1(COC(C)(C)C)nc(-c2cc[nH]n2)nn1CC(C)(C)O 55914,C(C)(C(CC(=O)NCCC(C(C)C)OC)NC(C1CN2CCC1CC2)=O)OC 55915,Cc1cnc(CC(=O)N(C2CCN(C(C3CCSC3)=O)C2)CCO)s1 55916,N1(C(C2CC=C(C)CC2)=O)CCCC(CCNC(=O)C=CC(C)C)CC1 55917,C1(C(=O)NCCOC)CC2(CC(C(=O)Nc3cc(-c4c(C)n[nH]c4C)[nH]n3)C2)C1 55918,C1(C(C)NC(=O)C(C)(C)c2cccnc2)CN(C(C2CCC(F)C2)=O)CCO1 55919,C(CC(C(=O)NCCC(F)Cn1cc(C2CC2)nn1)OC)OC.N(CCO)(CCO)C 55920,Cc1c(C(=O)NC2CN(C(=O)COCC(F)F)CC2C)cnn1C1CCOCC1 55921,Cc1c(C(N2CCC(CN(C(=O)C(C)NC(C)(C)C)C)C2)=O)sc(Cl)c1Cl 55922,C1(C(=O)NC(CC)CSC)CN(C(c2ccc(CO)cc2)=O)CC(C)(C)C1 55923,C1(O)(CN(C)C(C2(C(F)F)CCCO2)=O)CCN(C(c2cnc(C3CC3)s2)=O)C1 55924,c1(C(=O)NCCN(C(C2CC3OC(=O)OC3C2)=O)CC)nn(C)c2c1CCC2 55925,C1(NC(c2cc(C)[nH]c2)=O)CCCCC12CCN(C(c1cnc(F)c(C)c1)=O)C2 55926,C(=O)(C1CCCc2cccnc21)N1CCC(C)C1CNC(=O)CC1(O)CCCC1 55927,N1(C(c2c(C)nc(O)cc2)=O)CC(CNC(=O)C(C)n2cnnn2)CC(C)(C)C1 55928,C1(NC(=O)COCC2CC2)CCC(NC(=O)Cn2cnccc2=O)CC1 55929,N#Cc1ccc(C(N2CCOC(CC3CC3)C2)C(=O)NC2CCCC2)c(Br)c1 55930,c1(C(CCN(CC)Cc2ccc(Cl)c(Cl)c2)=O)nc2ccccc2s1 55931,N1(C(c2ccc(C)c(C)c2)=O)CCC(NC(c2cnc[nH]2)=O)C(CO)CC1 55932,C1(NC(C(C)SCC)=O)C2CCC1N(C(c1c(Cl)cncc1Cl)=O)C2 55933,CN1CC(CC(=O)NCC(O)CN(C(=O)C(O)C2CC2)C)C1 55934,N1(C(c2c(SC)ccs2)=O)CCCC(CN(C)C(c2ccc(C)c(O)n2)=O)CC1 55935,c1(C(=O)NC(c2cccc(C)c2)CNC(=O)C=CC2CCC2)cccc(O)c1F 55936,C1(C(=O)C)C2CN(Cn3cc(C4CC(CO)C4)nn3)CC12.C1(OCC)CCCOC1 55937,N1(C(C(CC)(C)F)=O)CCC(C2(NC(=O)C(=Cc3ccc(F)cc3)C)CC2)C1 55938,c1(C(N(C(CNC(c2cc(C(=O)OC)no2)=O)C)C)=O)noc2c1COCC2 55939,C1(CC(=O)NC(CCC)CO)CN(C(=O)Cc2ccsc2)CCC1C 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55957,CCCCC(C)(F)C(=O)N1CC2CCCC2(NC(c2cccc(C)n2)=O)C1 55958,c1(-c2cc(N(CC)CC)ncc2)c[nH]c2cc(C(=O)NCCSC)ccc12 55959,C(=O)(C(C)S(N)(=O)=O)NCC1(C(N)=O)CN(C(c2c(C)cc(SC)o2)=O)C1 55960,c1(CC)ccnc(C(N2CCC(C(=O)N(C)CC3(O)CCC3)C2C(C)C)=O)c1 55961,C1(CN(C(C2C(C=C(C)C)C2(C)C)=O)CC)CCCCN1C(c1n[nH]cc1Cl)=O 55962,CCC(CC(=O)NCC(CO)NC(c1cnc(C2CC2)s1)=O)C1CC1 55963,N1(C2CCN(C(C(C3CCCCC3)=O)=O)C2)CCN(C(=O)CCC2CCC2)CC1 55964,c1(NC(C2CN(C(c3cccnc3F)=O)CC2O)=O)ccc(I)c(Br)c1 55965,C=C1CC2CCC(C1)N2C(=O)C(F)C(C)CNC(C1(C(N)=O)CCC1)=O 55966,c1(-c2cn(CC(C)(C)O)nc2)ccc2[nH]c(C(=O)NC3CCS(=O)(=O)C3)cc2c1 55967,C1(CCNC(C2(OC)CCC2)=O)CCN(C(c2cc(C)ns2)=O)CCC1(F)F 55968,C1(O)(CC(N2C(C)(CC(=O)NCCc3ccc(O)nc3)CC2)=O)CCCCCC1 55969,c1(C(N2CCCC(n3cccn3)C2)=O)ccc(-c2ncc(C(F)F)s2)cc1 55970,CC1(C)CC(NC(c2ccn3ccnc3n2)=O)CCN(C(c2cnc(Cl)s2)=O)C1 55971,C1(C(N2CCC(CC=C)(NC(c3sc(F)cc3C)=O)C2)=O)C2CCCCCC12 55972,C1(CC)CC2CCC(C1)N2C(c1ccc(F)cc1C(F)(F)F)=O 55973,c1(CSC)ccc(C(=O)C(C)C)cc1.C1(=O)CN(CC)CCN1CCS.CCCCCC 55974,c1(CN(C(C2CC(CC)OCC2)=O)C)c(C)nn(C)c1Cl 55975,C=C(C)CN=C(NCC1COCC(C)(C)O1)N1CCC(F)(F)C(C)C1 55976,C1(CC(=O)NC(CNC(C=C(C)Cl)=O)C2CC2)CC(=O)c2ccccc2C1 55977,c1(C(=O)NCC23N(C(C=C4CCC(C)C4)=O)CC(C2)C3)cc2c(s1)CCC2 55978,c1(C(N2CC(CNC(c3ccccc3OCCF)=O)C2)=O)nccc2n[nH]cc12 55979,C(c1ccc(O)cc1)=CC(=O)NC1(C)CCN(C(C(C)OCCN(C)C)=O)C1 55980,C1(NC(C(COC(C)C)NC(c2ccc(CC)o2)=O)=O)COCC1C1CC1 55981,c1(C(c2n(C(CC)C)nnn2)NCc2noc(C)n2)c(C)cccc1Cl 55982,C1(CCCNC(COC(CC)C)=O)CN(C(=O)CCCCN(C)C(C)=O)CCO1 55983,C(=O)(CC(O)C(C)C)NCC1(OC)CN(C(c2ccnc(-n3cccn3)c2)=O)C1 55984,Cc1nsc(C(N2CCC3C(NC(c4ccnc(S)c4)=O)C23)=O)c1N 55985,c1(COC)ccnc(C(=O)NC(C2CCOC2)CNC(=O)CP(C)(C)=O)c1 55986,C(=O)(C(O)(C(F)(F)F)C1CC1)NCC1(C)CC=CC1 55987,C1(C(=O)NCC(C(C)C)(C)NC(=O)C(C)CO)CCC(F)(F)CC1 55988,C1(CNC(c2c(C)nc(C)[nH]2)=O)CC(C(C)(C)C)CN(C(=O)CC(C)C2CC2)C1 55989,C1(CC=C)(C(=O)NC2CCN(C(=O)Cn3cc(C#N)cn3)C2CC)CCCCC1 55990,CCC(C(=O)NCC1CCCC1NC(=O)C(C)(C)F)NC(N)=O 55991,C1(C(=O)NCC2(NC(C(C(C)C)OC)=O)CCCC2)CCC(F)(F)CO1 55992,C(=O)(C1=C(C)CCCC1)N(C1CCCCN(C(CCCC(=O)NCCC)=O)C1)C 55993,CCS(=O)(=O)C=CC(=O)NC1(CF)CCN(C(c2ccc3ncnn3c2)=O)C1 55994,C(C(=O)N(CC(=O)NC(c1cnn(C)c1C)C)C1CC1)(C(C)C)OCC 55995,CCCCCC(O)C(=O)NCC1CCN1C(C1C(=C)C1C(=O)OC)=O 55996,N1(C(CCC(C)OCC)=O)CCC(C)(C)C(NC(c2cc(C(F)(F)F)no2)=O)C1 55997,Cc1nc2cccc(C(N3CCN(C(C4COC(=O)O4)=O)C(C4CC4)C3)=O)c2[nH]1 55998,N1(C(C(=O)NCC(C)(Cn2cccn2)OC)=O)CCC(n2cccn2)CC1 55999,C1(CN(C)C(c2csc(Cl)c2)=O)CCCN(C(=O)CN(C)C2CC2)C1 56000,c1(CNC(C23C(CN(Cc4nc(C(C)C)on4)C2)C3)=O)nc2ncc(Br)cn2n1 56001,N1(C(CCCCC=C)=O)CC2CN(C(=O)C(n3c(C)cc(O)cc3=O)C)CCC12 56002,C1(O)(C(=O)NCCC(C)NC(c2ccc(CO)o2)=O)CCCC(C)(C)CC1 56003,N1(C(c2cc(C)nn2C)=O)CC(C)CN(C(c2cccnc2C(F)F)=O)CC1C 56004,C1(CC(=O)N(C)CCN(C)C(c2cc(C)c(C)s2)=O)(OC)CCCCC1 56005,C(=O)(N=c1nn[nH]n1-c1ccc(F)cc1)NCCCCC1C(C)C1 56006,c1(C2C(C(N(CC(C)NC(C3COCCO3)=O)C)=O)C2)cccc(Cl)c1 56007,c1(CC(=O)OC)occc1C(N1CCCC1C1CCN(C(c2csc(Cl)n2)=O)C1)=O 56008,C(=O)(CC1=CCOCC1)N1CCC(CNC(c2c(Cl)c(C)n(C)n2)=O)C(C)C1 56009,C(=O)(CCCC(CC)NC(=O)CCCCCC)NC(C1CCOC1)C#C 56010,N1(C(C(CC)F)=O)CC2C(CNC(=O)CCc3nnc(C(F)F)o3)C2C1 56011,N1(C(c2csc(Br)n2)=O)CCC2CCN(C(=O)C=CC3CCCC3)C2C1 56012,N1(C(Cc2ccc(C)cc2)=O)CCN(C(c2ccc(=O)n(C)c2)=O)CC1C 56013,Cc1cc(N)c(C)nc1C(=O)N(CCC(C(C)(C)C)NC(=O)CC(C)C)C 56014,c1(-c2c(C(=O)NCC(C)C)cc(OCC)nc2)nc2ccc(CO)cc2s1 56015,NS(=O)(=O)c1cncc(NC2(c3cc(F)cc(F)c3)CC2)c1 56016,N1(CC)CC(C(=O)NC2CCC(CNC(=O)C(F)(F)CN(C)C)CC2)CC1=O 56017,N1(C(CCC#C)=O)CCC(C)C1CNC(=O)CCSc1nnnn1C 56018,CON(C)C(=O)c1conc1CNC(=O)Cn1cnnc1 56019,C(CS(=O)(=O)CCCN1CCCC(NC(=O)C(c2ccccc2)O)CC1)OC 56020,C1(NC(c2cncnc2)=O)CN(C(=O)CCN2C(=O)CCC2=O)C2(CCOC2)C1 56021,c1(SCC#C)cccc(C(=O)N(C2CCC(NC(C3(O)CCOCC3)=O)C2)C)c1 56022,C1(C(N(C)CC2(O)CN(C(=O)CN3CCSCC3)C2)=O)SC2C=CC1CC2 56023,C1(C(=O)NCCC(CNC(CCCN(C)C)=O)O)OCCOC12CCC2 56024,Cc1coc(C(C)C)c1C(=O)NC1CCN(C(C23CCC(C2)OC3)=O)C1 56025,Cc1cc(C(c2nnnn2C(C)C)NC(C)Cn2cnnc2)c(Br)cc1F 56026,c1(C(N2CC(SC)C(NC(=O)CCC3CC(F)(F)C3)C2)=O)n[nH]c2c1CSCC2 56027,N1(C(=O)OC(C)(C)C)CCC(NS(=O)(=O)NCC2CC2c2ccncc2)CC1 56028,C1(CNC(C(CC)N(C)C)=O)CC2(CCN(C(=O)C(O)CCSC)C2)CO1 56029,C#CC1CCN1C(=O)C(Cn1ccnn1)NC(=O)CCSC 56030,CCC(CCC(=O)Nc1cccc(C(C)F)c1)NC(c1ccc(CO)nc1)=O 56031,C1(NC(C2CC2[N+](=O)[O-])=O)CC2C1CCN2NC(c1ccnc(S)c1)=O 56032,N1(C(=O)COCC(F)F)CCC(O)(CCNC(C2(c3ccc(F)cn3)CC2)=O)C1 56033,N1(C(C=CCN(C)CC)=O)CCN(C(=O)Cc2coc(C)n2)C2CS(=O)(=O)CC12 56034,N1(C(CC(=O)OCC)=O)CCC2(CC1)CC(CNC(=O)Cc1cccc(O)c1)C2 56035,C1(C)(NC(CCOCCC)=O)CCCN(C(c2[nH][nH]c(=N)c2Br)=O)C1 56036,C(CCN(C)C)(C(=O)NC1CCCCC1)NCc1nc(NC(C)=O)sc1 56037,CC(C)C(C)(O)CNC(C1CC(n2cc(-c3cc(C4CC4)no3)nn2)C1)=O 56038,CC1CN(C(c2ccnc(C(C)(C)C)c2)=O)CCC1NC(c1cc(=O)cc[nH]1)=O 56039,C1(C(=O)OC)CCC(C(N2CCC(CCNC(=O)CC=C(C)C)C2)=O)CC1 56040,N1(C(=O)C(F)C2CCCC2)CC2CC1CN2C(C1(F)CCC1)=O 56041,N1(C(c2c(CC)nco2)=O)CC(C)OC2(CCN(C(=O)CSCC(C)C)C2)C1 56042,c1(CC=C)ccccc1C(N1CCC(N(C(C2COCCN2CC)=O)CC)C1)=O 56043,C1(F)(CNC(Cc2ccn(C)n2)=O)CCN(C(C2CN(C3CCC3)C2)=O)CC1 56044,C1(CCC)CN(C(=O)CSc2n[nH]c(O)n2)CCN1C(=O)C(C)NC(=O)CC 56045,C(N1CCC(F)(F)CC1C)Cc1cn(CCC(CC)(F)F)nn1 56046,c1(-n2c(CC3(C)CCCCO3)nc(C3CC34CC4)n2)ccc2nc[nH]c2c1 56047,CCC(O)C(C)C(=O)NC12CC(NC(=O)OCc3ncc(C)[nH]3)(C1)C2 56048,C1(O)(CC)CCN(C(=O)C(C)(C)CN(C(=O)CCC(C)SC)C)C1 56049,N1(C(CCNS(CC)(=O)=O)=O)CCC2(COCC(CNC(c3cnco3)=O)O2)C1 56050,Cc1ncc2n1CC(C(=O)NC1CN(C(C3CCOC(C)(C)C3)=O)CC1C)CC2 56051,N1(C(C(c2ccnn2C)C)=O)CC(NC(=O)Cc2nc[nH]n2)CC12CCCOC2 56052,C1(CCC(=O)NCC(CC)(C)NC(=O)COC(C)(C)C)CCC(O)CC1 56053,N(C(=NCC=C1CCOCC1)N1CCC(c2nncs2)C1)CCOC(C)(C)C 56054,c1(NC(=O)NC)cccc(C(=O)NC(C)C(CO)NC(C2(C)CCCC2C)=O)c1 56055,S(=O)(=O)(c1ccc(F)cc1Cl)NC(c1ccc(S(C)(=O)=O)cc1)C 56056,N1(C(C2C(OC)C2)=O)CCC(C)C(CNC(=O)C=CC=C(Cl)Cl)C1 56057,C1(CC(=O)NC(CC(C)NC(COCCOCCOC)=O)C)CCCC12CC2 56058,c1(OC)c(Cl)nc[nH]c1=NCC1(CNC(=O)CNC(N)=O)CC12CCC2 56059,C1(CC)C(C(=O)NC(CCSC)C(=O)NC2(C)CS(=O)(=O)C2)CCN1C 56060,Cc1ccn(C(C)CC(=O)NCC2(C)CC(NC(c3cc(F)cs3)=O)C2)n1 56061,N1(C(C(CC=CC)NC(=O)CN2CCCC2C)=O)CC(C)N(CC)C(C)C1 56062,C#CCCC(O)C(=O)NC1CC(NC(c2cccc(=O)n2C)=O)C1 56063,C1(CNC(C2C(C(C)NC(Cc3c(C)n[nH]c3)=O)C2)=O)CC2(CCC2O)C1 56064,c1(C(=O)NC2CC2C(N2CCn3ccnc3C2)=O)ccc([N+](=O)[O-])cc1I 56065,CCCC(C(=O)NC(C)(C)CNC(c1cc(Br)cc(N)c1C)=O)C(C)C 56066,CC1=C(C(=O)N2CCC(C3(NC(c4sccc4F)=O)CC3)C2)CCCC1 56067,c1(C(N(C(CNC(C=C(C)C(C)C)=O)C)C)=O)cc(F)cc(Cl)c1O 56068,C(c1cc(C)cc(C)c1)=CC(N1CC(C)(NC(c2cccc(OC)c2F)=O)C1)=O 56069,N1(CC(=O)NCc2ncoc2C(F)(F)F)CCCCC1 56070,CCCCC(CNC(C1CC(CCNC(C23CC(CO)(C2)C3)=O)C1)=O)CC 56071,c1(-c2n(C)c(O)nn2)ccc2ccccc2c1Br.N1CC(O)CC12CCC2 56072,C1(NC(C2CC3CCC2O3)=O)C=CCN(C(=O)CCc2ccsc2)C1 56073,CC1(C)CC(NC(c2ccc(-c3cc[nH]n3)cc2)=O)CN(C(=O)COC2CC2)C1 56074,c1(CCC(=O)NC(CNC(CCOCC(C)C)=O)(C)C)cc(Cl)no1 56075,N1(C(Cn2cc(CNC(C(C)SCCCC)=O)nn2)=O)CCCC(C)(N(C)C)C1 56076,c1(OC)ccc(C(N2CCC(N(C)C(c3cc(C(F)F)ncn3)=O)CC2)=O)cn1 56077,CC(CC(C)(C)C)C(=O)N1CCOC(C)C1C(=O)NCCc1noc(=O)n1C 56078,c1(C(=O)NC2C3CN(C(c4c(C)nc(C(C)C)s4)=O)C2C3)cnc2ncccn12 56079,c1(C(N(C2CN(C(c3c(C)nc(Cl)cc3)=O)C2)C)=O)ccc2c(c1)CCCCN2 56080,N1(C(C)=O)CC2CC1CCC2NC(c1ccc(OCC2CC2)nc1)=O 56081,Cc1c(Cl)c(C(N2CC(CNC(=O)Cc3ccc(O)cc3)CC2C)=O)nn1C 56082,C(=O)(CCCCC(=O)N(CCC(=O)NCCCC1CC(C)C1)C1CC1)OC 56083,N1(CC(=O)NC(CC)CNC(=O)CC2(CS(C)(=O)=O)CC2)CCCCCC1 56084,c1(NC(=O)NCc2c(CC)onc2C)ccc2c(c1)C(C)(C)CC(=O)N2 56085,c1(C(N2CC(C(=O)Nc3cn(CC)nc3C)C(F)C2)=O)cnc(C)cc1C 56086,C(=O)(CCc1ccsc1)NCCN(C(=O)COC)CCC.C1(=O)CCN1 56087,Cc1nc(C)c(C(=O)NC23CCCC2N(C(=O)C(C2CC2)C2CC2)CC3)nc1C 56088,CC(C)C(CNC(=O)CCCSC(C)(C)C)NC(=O)Cc1cnn(C(F)F)c1 56089,Cn1cc(S(N)(=O)=O)cc1C(=O)C(=O)NCCC1CCCCN1C(=O)CC(F)F 56090,c1(OCC(=O)NC2CC(C)N(C(C3CC4CC3C3CC43)=O)C2)ccccc1C#N 56091,CCCCC(O)C(C)C(=O)NC(c1cnn(C)c1)C(=O)NC(C1CCOC1)CO 56092,c1(C(N(C2CN(C(Cc3cnc(C)o3)=O)CC23CC3)C)=O)ccn2cccc2c1 56093,C12(CC(=O)NC3CC(NC(C4CCCCO4)=O)CC3O)CCC(CC1)OC2 56094,Cc1cccc(CC(=O)NC2CC2NC(=O)C(C)C2CCCC2)c1 56095,N1(C(Cc2n(C)nnc2)=O)CCC2(CCOC2)C(CNC(C2(CCO)CC2)=O)C1 56096,C(N=c1cc(C)c(S(=O)(=O)N2CC(O)C(C)(C)C2)c[nH]1)C1(OCC)CCOC1 56097,C1(NC(c2cc(C)cc(C)c2)=O)CC2CC(C1)N(CCOCC(C)C)C2 56098,N1(C(C2CCN(CC)C2)=O)CC(OC)C(NC(=O)CSCC(=O)NC)C1 56099,C1(NC(C(C)(C)c2ccccc2)=O)CC2CN(c3nc(C(F)(F)F)ns3)CC2C1 56100,C1(NC(c2ccccc2Cl)=O)CN(C(C2CCC3(CCC3)OC2)=O)CC2(CC2)C1 56101,Cc1c(C(=O)NC2CCCC(NC(=O)C(F)=C3CCCC3)C2)sc2ccccc12 56102,c1(S)ccnc2cccnc12.S(=O)(=O)(CCCCF)NCc1nnc(CC)n1N 56103,N1(C(CC#C)=O)CC2CCCC2(NC(=O)Cc2cc(OC)cc(Cl)c2)C1 56104,O=C(C#CC1CC1)N1CCCCC1C1CCCN(Cc2cc[nH]n2)C1 56105,C1(C(=O)NC(Cc2cn(CCOC)nn2)C(=O)OC)CCC2(CC1)CC(O)C2 56106,C1(NC(CNC(=O)OCC)=O)CN(C(C2CCCCC(=O)N2)=O)C2(CCCC2)C1 56107,C(=O)(CCCCC#N)NCCC1CC(NC(C2(C)COCCO2)=O)C1 56108,N1(C(c2c(CC)cncc2)=O)CC(C(=O)NC(c2n[nH]c(CO)n2)C)CC(C)C1 56109,C1(C#N)(C(=O)NCC(C)(C)NC(C(F)=CCC)=O)CC2C=CC1C2 56110,C(CN=c1[nH]c(=NCc2c(C)nn(C)c2Cl)[nH]c2c1COC2)OCCC=C 56111,c1(C(N(C2C3CN(C(C4ON=C(C)C4)=O)CC32)C)=O)ncc2c(F)cccn12 56112,C=CCCC1C(=O)NCc2csc(c2)C(c2nnnn2C2CC2)N1.C(C)(C)OC 56113,C1(NC(C2C(C)(C)C2)=O)CCCCCC1C(=O)NCC1(C(C)(C)O)CC1 56114,C1(CNC(c2c(C)nsc2)=O)CCCC(NC(C2OCC2(C)C)=O)C1 56115,C1(NC(c2ccc(CSC)o2)=O)CC2CCC1N(C(=O)C(C)n1cnnn1)C2 56116,C(=O)(CC(C(F)(F)F)n1ccnc1)N1CCC(Sc2cc(C(C)=O)nn2C)CC1 56117,C1(C(=O)NC2(C#C)CCOC2)CCC2(CC2)N1C(C1CN2CCN1CC2)=O 56118,c1(OC)ccc(CCC(N2CC=CC2CNC(C2CCCO2)=O)=O)cn1 56119,N1(C(c2cc(OC)ns2)=O)CC(C(N2CCNC(=O)C2C(C)C)=O)CC(C)(C)C1 56120,Cc1cccc(Br)c1C(C(=O)NC1(C)CC(C)OC1=O)NC(C1CC=CCO1)=O 56121,C=CC(C)(O)C(=O)NCC1(CN(C)C(c2csc(-c3cocn3)n2)=O)CC1 56122,CN1CCOCC1C(N1CCC(C(F)C(=O)NCC2(CO)CCCO2)C1)=O 56123,c1(C(=O)NCC(C2CCC2)NC(C2C(CC(C)C)C2)=O)nsnc1O 56124,C1(C(=O)NC(C2CC(CCO)C2)=O)CN(C(C2(COC(N)=O)CCC2)=O)C1 56125,C(C)(C)(CCCCC(=O)NC1CCN(C(c2ccc(Cl)c(Cl)c2)=O)CC1)OC 56126,Cc1cnnc(O)c1C(=O)NCC1(O)CC(C(N2CCC(C)C2CO)=O)C1 56127,CC(CN=c1nc(N2CC3C(C)C3C2)c2c([nH]1)CCCCC2)Sc1ccccc1 56128,C1(C(=O)NCC2(C)N(C(C3OCCN(C)C3)=O)CCC2)CC(C)(C)CN1C 56129,c1(C(N2CC3C(CN(C(C(C=C)O)=O)C)C3C2)=O)cc(C)cc(C)c1 56130,CCCCC(C)(C)NC(=O)C(Cc1ccc(C)cc1)NC=O 56131,CC1CC=C(C(=O)NCC2CCC2NC(=O)CSc2nnnn2C2CC2)CC1 56132,Cc1ccc2c(CC(=O)NCCC(C)(C)CNC(C3(O)CC3)=O)c[nH]c2c1 56133,c1(CNC(C(c2ccnn2C)C)=O)ccoc1C(=O)NC(C)Cn1cccn1 56134,C(C1=C(C(=O)O)C(c2ccccc2)NC(=O)N1C)N1CCC(CCC)CC1 56135,N1(C(C(C(=O)NCC)(C)C)=O)Cc2occ(C(=O)N(CCCN(C)CC)C)c2C1 56136,N1(C(C2C(C)CCC2)=O)CCC2(CC(NC(c3cccs3)=O)C2)C1 56137,CC1CN(CC2CC2)CCN1C(=O)C(c1ncc(-c2ccc(Cl)cc2)o1)C 56138,C(=O)(C(C)N=c1cc[nH]cc1)N1CCC(N(C(=O)C2=CCC(C)CC2)CC)CC1 56139,C1(N(C(c2cc(CC)no2)=O)C)CC2CC1N(C(=O)C(C)(C)CN(CC)CC)C2 56140,N1(C(C2(F)CCN(C(c3cc(C)ncc3C)=O)CC2)=O)CCCC12CCCOC2 56141,N1(CCS(C)(=O)=O)CCOCC1c1cn(CCO)nn1 56142,c1(C(N2CCC(CC3CN(C(c4cnco4)=O)C3)CC2)=O)ccn2ccnc2c1 56143,CC1(C)CN(C(=O)CC2(C(F)(F)F)CC2)CCC1NC(c1cc2ccsc2s1)=O 56144,C(=O)(CCCCCC#N)NC(C(=O)NC(C#C)CC(C)(C)C)(C)C1CCC1 56145,Cc1cc2nc(-c3nc(CC(C)C)nn3CC3CCCCC3)ccc2c(=O)n1C 56146,C=CCCCCC(=O)N1CCN(C)C(C(=O)NCCNC(=O)CC)C1 56147,Cc1cc2c(cc1C)OC(C(N1CCN(C(=O)CC3(CO)CCC3)C(C)C1)=O)C2 56148,C(=O)(C(C)C(=O)NCc1cc(C(=O)NC(C)C(C)n2cncn2)no1)OC 56149,c1(CC(=O)N(CCN(C(=O)CSc2cccs2)CC)CC)ccc2c(c1)COC2 56150,CC1CCC(C(N2CCC(CN(C(=O)C(C)(F)F)C3CC3)CC2)=O)CC1C 56151,N1(C(C2(NC(C3C(C)C3)=O)CCCCC2)=O)C2CCC1CN(C)C2 56152,N1(C(C2(CC)CCN(C(C3CC34CCCC4)=O)C2)=O)CCC(C)(C2CC2)C1 56153,Cc1nc2n(n1)CC(C(=O)NCC1CN(C(=O)CCn3cncn3)CC1O)CC2 56154,c1(OC)cc(C(=O)Nc2ccc(C(=O)Nc3csc(C#N)c3)cn2)ccc1Br 56155,c1(C(C)C)[nH]nc(CNC(N2CC(O)CC2C(C)C)=O)c1Br 56156,CN1CC(F)CC1C(=O)NCCCNC(c1ccc(F)cc1)=O 56157,S(=O)(=O)(CC(=O)N(CCCNC(=O)Cc1cnn(CC)c1)CCO)NCC 56158,Cc1ccc(C(F)F)cc1C(N1CCC1CNC(c1cccc(C#N)c1)=O)=O 56159,CC1CCC(CO)CN1C(C1(F)CCN(C(=O)C=CC2CCCCC2)C1)=O 56160,c1(OC)cccc2c(N3CCCC(CC(C)C)C3)ccnc12 56161,c1(N(C(c2cnc(C(C)C)[nH]2)C)C)ccc(CN(C)C)cc1 56162,C=C1CCC(NC(C2(CNC(=O)C(C)OCC(C)C)CCC2)=O)CC1 56163,C(C(O)CC(=O)NC1CN(C(=O)C(C)(C)N2CCCCC2)CC1F)N(C)C 56164,C(=O)(CCS(N)(=O)=O)N1CCC(CC=C)(NC(C2CCOC2C)=O)C1 56165,C(=O)(CCCC(C)(C)NC(=O)C(C#N)C(C)(C)C)NC1CCN(CC)C(C)C1 56166,Cc1ccc(C)c(C(N2CC(CCNC(C3CC(C(C)C)=NO3)=O)C2)=O)c1 56167,c1(N2CCC(C)C2)ncnc2c1ncn2CC1CCCCC1O 56168,CC1(C)COC1C(N1CCCC1CNC(=O)Cc1cc[nH]c1)=O 56169,Cc1scc(C(=O)NCCN(CCCN(C)C)C(=O)CC2CC3CC3C2)c1C 56170,N1(C(CNC(CCC)=O)=O)CCC2CCN(C(=O)Cc3cccc(OC)c3)C2C1 56171,C1(CNC(CC(CC)(C)C)=O)CC2CCC(C1)N2C(C1(COC)C=CCC1)=O 56172,c1(C(C(=O)NC)NC(C2CCCC(OC)C2)=O)ccc(NC)cc1 56173,N(C1CCCc2c(I)n[nH]c21)C(=O)NCc1cn(C(C)(C)C)nn1 56174,CC1CCN(C(=O)C(=O)NC2(CNC(=O)CC3(C)CC3F)CC2)CC1 56175,C(=O)(C1=NOC(C)(C)C1)N1CCCC(C(=O)NCCC(C(C)C)OC)(CO)C1 56176,c1(NC(C)=O)nnc(S(=O)(=O)NC2CCC(F)(F)C(C)C2)s1 56177,C12(CNC(CCCCCC)CC)CNCC(=O)N1CCOC2 56178,c1(CC)cc(NC(=O)COC2(C)CN(C(=O)CNC=O)C2)cc(C)c1 56179,C1(CC(=O)NC(CCNC(CC=CCC)=O)(C)C)CCCC(C)(C)C1 56180,c1(NC(NCC(NOCC)=O)=NC)cc(NCC)cc(CO)c1 56181,C1(CCC)(NC(=O)Cc2cccc(C)c2)CCN(C(C2COCC2(C)C)=O)CC1 56182,c1(NCc2ccn(CC)n2)[nH]c(=NCc2ccc(OC)o2)nc2scnc12 56183,N1(C(C(CC(C)C)(C)O)=O)CC2(C=C(C(=O)NCC3CCSC3)CO2)C1 56184,CC(C)(CCC#N)C(=O)N1CCN(C(c2sc(C(F)(F)F)cc2Br)=O)CC1 56185,N1(C(c2c(CC)non2)=O)CC2CCN(C(c3cc(O)cc(O)n3)=O)CCC2C1 56186,C1(NC(C=C=C(C)C)=O)CC12CCN(C(=O)C(F)C1CCCC1)C2 56187,C1(NC(C(c2cc(C)oc2C)C)=O)CCCCN(C(=O)C(F)(F)c2nccs2)C1 56188,C1(NC(c2c(CC)occ2)=O)(CO)CCN(C(C2(C)CSC2)=O)CC1 56189,C1(NC(c2cc(CC)on2)=O)(CO)CCCN(C(C2(C)CCCO2)=O)C1 56190,c1(C(CNC(C2N(C)CC(F)C2)=O)NCC2(CO)CCCO2)ccc(F)cc1F 56191,C(=O)(C(F)(F)CC(C)C)N(C(C)CNC(=O)COc1c(F)cccc1Cl)CC 56192,c1(C(=O)NC(CC)CN(C)C(c2cc(C)cs2)=O)cc(N)c(Cl)c(O)c1 56193,C1(C(=O)N)CCCCC1CNC(=O)C(C(C)C)N(C)C.N1(CCC)CCCC1CO 56194,C1(C(N(C(CF)CF)C)=O)CC1C1CN(C(C2CN3CCC2CC3)=O)C1 56195,C1(CC(=O)NCC(CNC(C2(C)CC=CC2)=O)CO)CC(C)(C)CCO1 56196,N1(C(C2C(C)C2)=O)CCCCC1CNC(=O)CCc1cnn(C)n1 56197,N1(C(Cc2c(C)cnn2C)=O)CC(CNC(C2CCCC23CCC3)=O)C(C)(C)C1 56198,C(=O)(C(C(C)OC)N(C)C)NCC(CC)N(C)C(C1CC(OC)C1)=O 56199,C(=O)(CS(=O)(=O)c1ccccc1Cl)NC1CCC(NC(C23OC(C)C(C2)C3)=O)C1 56200,c1(C(=O)OCC)ccc(CCNC(=O)NCC2CC(C(F)(F)F)CO2)cc1 56201,C1(C(C)C)(C(N2CCC(C(C)(C)O)C2)=O)CCN(C(=O)CSCC(F)F)C1 56202,O=C(C(O)CC(F)(F)F)NC1CCN(C(=O)C=Cc2cccc(O)c2)C1 56203,Cc1nnc2n1CC(C(=O)NC1CCC(C)(C)NC1)CC2 56204,O=C(N=S1(=O)CCNC(c2ccccc2)C1)c1cc2c(s1)CCCCC2 56205,c1(C(N2CC3C(CNC(COCCCCCC)=O)(C3)C2)=O)nccc(Cl)c1C 56206,C(=O)(CCCC1CCCC1)NCC1(CNC(C(C)OCC=C)=O)CC1 56207,N1(C(Cn2ccc(OCC)c2)=O)CCC(CN(C2CNC2=O)C)C12CC2.CCC.OC 56208,N1(C(c2ccsc2Cl)=O)CCOCC1CCNC(C12CCC(C1)C2)=O 56209,C(CC)(C(=O)N1CCC(c2ncco2)C1)N(C(CSCC)=O)C 56210,c1(OC)noc(C(N2CC=CC2CNC(C2CC(F)C2)=O)=O)c1Br 56211,c1(C(=O)NCC(C)CN(C)C(c2nccn2C)=O)cc([N+](=O)[O-])n[nH]1 56212,C1(C(=O)OC)CCN(C(=O)C2CCC3(CC3)N2C(=O)CCN2CCCCC2)O1 56213,C1(C(C)NCc2ncnn2CC2CC2)CC(=O)N1.C1(C(=O)OC)(C(N)=O)CC1C 56214,C1(COC)CC(COC(c2cc(C(=O)OC)no2)=O)CC(CC(=O)OC)C1 56215,c1(CNC(N2C(C)CSCCC2)=O)c(Br)ccc(Cl)c1F 56216,CC(CC(C)(C)C)C(=O)N1CC2CC(C1)N(C(=O)CNc1ncccn1)C2 56217,C(=O)(C(C)CN1CCOCC1)NCC1CCN1C(c1noc(C(C)(C)C)n1)C 56218,Cc1c(C(=O)N(c2nccc(Cl)n2)C)cccc1C(F)(F)F 56219,C1(C(=O)NCC2CC3(CCC3O)C2)CCN(C(C2CCC(O)CC2)=O)C12CC2 56220,c1(OC)ncc(C=CC(=O)NC2CCCN(C(C3CCCN3C)=O)C2C)cn1 56221,c1(NC(=O)NCC(COC)OC)ccc2c(c1)NC(=O)C1(CCCCC1)OCO2 56222,c1(C(N2CCN(C3CCCC3)C(C)C2)C(=O)NC(C)C)cc(C(N)=O)cc(Br)c1 56223,C(=O)(CC=C(Cl)Cl)NCCOC1CN(C(C2(C(=O)OC)CC2(F)F)=O)C1 56224,N1(CCN(C(CCC)C)C)CC(C)OC(C)C1 56225,n1(CC)cc(CN(C)C(C2CC(N(C(=O)C(C)CO)C)C2)=O)nn1 56226,CC1CC(CCNC(c2cc(Cl)no2)=O)CCN1C(=O)Cc1ccc(F)nc1 56227,N1(C(c2ccc(CC)[nH]2)=O)CC(NC(C2CC(OC(F)F)C2)=O)CC1C 56228,N1(C(CC(C)CF)=O)C2CCC1CC(NC(=O)CN1CSCCSC1)C2 56229,CC(CCCCNC(=O)Cn1cccnc1=O)NC(C1(CC2CCC2)CC1)=O 56230,C1(NC(c2c(Cl)cn(CC)n2)=O)CN(c2ccnc(C3CC3)n2)CC1(C)C 56231,C1(CC(=O)N(C2CCN(C(C(CC)F)=O)CC2)C)CCCC(C)(C)O1 56232,c1(C(N(CC(CN(C(=O)CCc2cnc[nH]2)C)O)C)=O)cnc(C(F)F)s1 56233,CC1CCCc2cc(NC(N3CCSc4ccccc43)=O)nn21 56234,CC1CC(NC(=O)C(C)(C)NC(=O)CCCCC2CC2)CCN1C 56235,C=C(C)CC(C)C(=O)NCC(CC)NC(=O)C(C)(C)C(F)F 56236,N(C(=NCCc1ccccc1F)NC(C)(C)CF)C1(C)CCC1 56237,C(c1cncnc1O)=CC(=O)NCCC1CN(C(CCNC(=O)CO)=O)C1 56238,CC1CN(C(C2CCC3(CC2)N=N3)=O)CCC1NC(C1SCCCS1)=O 56239,Cc1cc(N)c(C(N2CCC(O)(C(C)CNC(c3ccc(Br)o3)=O)C2)=O)c(F)c1 56240,C1(C(N2CCC(C)(NC(=O)CC3COC(=O)C3)C2)=O)C2Cc3ccccc3C12 56241,C(=O)(CC(C)CC(=O)NC1CN(C(c2cc(C3CC3)no2)=O)C2(CCC2)C1)OC 56242,c1(C(=O)NCC2(NC(c3c(CC)nc(C)o3)=O)CCCC2)ccc(OC)nc1Cl 56243,Cc1cn(C)nc1C(=O)NC(c1cnn(C)c1)C(=O)N(C)Cc1cnn[nH]1 56244,c1(OC)c(C(N2CC(NC(c3occc3C)=O)CC(O)C2)=O)cccc1Br 56245,c1(CC)cscc1NC(=O)C(C)(C1CCC1)NC(C1CC1(F)Cl)=O 56246,C=CCCCCCCCC(C(=O)OC)N1CC2CCCN2CC1CC 56247,CC(CCC(=O)N(C(C)C(=O)NCC(C)(C)C)C)OCCO 56248,CC(C)CCCCC(=O)NC1C=CCN(C(=O)Cc2ccns2)C1 56249,NS(=O)(=O)c1cccc(C(=O)NC2C3CC2CN(C(c2ccc(CO)o2)=O)C3)c1 56250,N1(C(C2CN(C(C)C)C2)=O)C(C(=O)Nc2cnc(Cl)nn2)CCC1C 56251,CCC(CO)(C(=O)NCC(C1CCC1)NC(c1cnc[nH]1)=O)OC 56252,C1(NC(=O)NC2CC23CCCC3)CNCCC12CCOCC2 56253,C1(O)(CNC(CC2C(C)CC2)=O)CCN(C(C2(CO)CC2)=O)C1 56254,N1(C(c2n(C)nnc2)=O)CC(NC(C2CCOC2)=O)C2CCCC2C1 56255,c1(CNC(=O)NC2C(C(=O)OC(C)(C)C)OCC2)nc(Cl)ccc1Cl 56256,N1(C(CC#C)=O)CC2COCC2(C(N2CCCC2C(C)(C)O)=O)C1 56257,c1(C(C)OC)ncc(C(=O)NC2CC(N(C)C3CC3)C2)s1.c12cn(nn1)[nH]c2=O 56258,N1(CC(=O)NC)CC(O)CC2(CCNCC2)C1.C12(CC1)C(=O)N2 56259,CCC(CC(C)C)C(=O)NCC1(C(N2CCC(OC(C)C)C2)=O)CCCCC1 56260,C1(N(C(C(CNC(c2nc(C)sc2)=O)N(C)C)=O)C)COC(C)(C)C1 56261,CCCCN=C(NCc1ccc2c(c1)OCO2)NCc1ncnn1CC 56262,N1(C(C2N(C(c3c(C)ncc(Cl)c3)=O)CCSC2)=O)Cc2cccc(O)c2C1 56263,N1(C(CCS(N)(=O)=O)=O)CCC2CCN(C(C3(O)COC3)=O)CC12 56264,CC(C)CC(C(=O)N1CCC(O)(CC2CC2N)CC1)ONC(c1ccccc1)=O 56265,C1(CNC(C2C(=C)CC2)=O)CC2(CCN(C(c3ncccc3N)=O)CC2)CO1 56266,C1(n2cc(SCC)nn2)CCCN(C(c2cnn(C3CCS(=O)(=O)C3)c2)=O)C1 56267,C(C(=O)NC1CCCCC1NC(=O)C#CC1CC1)(C(C)C)(C(C)C)NC(C)=O 56268,Cc1ccccc1C(=O)N(C)CCOCCN(C(=O)CC(C)N(C)C1CC1)C 56269,CCC(C)(CO)CN=c1cc(NC(c2csc(C3CC3)n2)C)nc(C)[nH]1 56270,C1(NC(=O)NC(C)(C)CC2CCOCC2)CCC2C3CCC(C3)C12 56271,CC(C)CCC(F)C(=O)N1CCC(O)(CCNC(C2CCCCCC2)=O)CC1 56272,c1(OC)cc(NCC2(OC(C)=O)CC(c3nnnn3CC(F)F)C2)cc(O)c1 56273,c1(C(=O)NC2CCCC(NC(CN(C)C)=O)C2)ccc(Cl)c(N2CCCC2)n1 56274,c1(NC(C)=O)ccc(F)cc1C(N1CC2CCC1C2NC(=O)CC1(C)CC1)=O 56275,C1(c2nnc(N3CCCC(CSC)C3)n2C)C(C2CC2)CCN1NC(=O)C1CC1 56276,C1(C(=O)OCC)CCOCCN1C(C1CC(=O)N(c2ccc(C)cc2OC)C1)=O 56277,c1(C(=O)OC)cc(C)cc(NC(N2CCCC2c2cccs2)=O)c1C 56278,c1(C(C(=O)NC2CC(CNC(C=CC=CC)=O)OCC2)(C)C)cccc(C#N)c1 56279,N1(C(C(C=C)(C)C)=O)CCC(C(F)(F)F)C(NC(c2nnc(C)cc2O)=O)C1 56280,CC(C)CCC(O)C(=O)N1CCC(n2cc(CNC(C3COC(=O)N3)=O)nn2)C1 56281,c1(CC(=O)N(CC(CC)NC(c2ccnc(O)c2)=O)CC)cc(Cl)ccc1OC 56282,c1(OC)ccc(-c2nc(C(=O)NCC3CCC(NC(C4CSC4)=O)C3)cs2)cc1 56283,c1(-n2c(C)ncc2)ccc(CN2CCC(N(CCCn3ccnc3)C)CC2)cc1 56284,N1(C(Cc2c(C)scc2)=O)CCN(C(=O)CS(=O)(=O)C2CC2)C2COCC12 56285,c1(C(=O)Nc2ccc(C)nc2Br)cc(-c2ccc(C)cc2)n2cnc(C(N)=O)c2n1 56286,C1(C(=O)NCCN(C(=O)COC2CCCOC2)C(C)C)OCC2COCCC12 56287,C1(C(=O)NCC(C)N(C)C)CN(C(C2CCC2C)=O)C(C)(C)C1 56288,c1(OC)cc(C2(C(=O)NC3CCC(CNC(=O)CC4CC=CC4)C3)CC2)ccc1C 56289,c1(CC)nc(C)c(C(=O)N(C(C(=O)NOCCCOC)C2CC2)C)o1 56290,N1(C(CCCC#C)=O)CCC(NC(C2CCCN(C(C)=O)C2)=O)C1(C)C 56291,CCC(C)(C)C(C(=O)NC1(CNC(c2cscc2C)=O)CCOCC1)OC 56292,C1(C2CC2)(CNC(C=C(CCC)C)=O)CCN(c2cc(C(F)(F)F)nc(C)n2)C1 56293,c1(CNC2CCCC(C(=O)NCC=C)C2)ccc(F)c(Br)c1F 56294,C1(NC(=O)Nc2ccnc(N3CCOC3=O)c2)CCc2cc(Br)ccc2C1 56295,N1(C(C2=C(C)OCC2)=O)CC2(CCC(NCc3cc(F)cc(Br)c3)C2)C1 56296,C12(NC(c3csc(-c4ccoc4)n3)=O)CC1CN(C(c1cc[nH]c1C1CC1)=O)C2 56297,N1(C(C(N2CCCC(O)C2)=O)=O)CC2(C1)OCC1CC21 56298,Cc1cc(C)cc(C=CC(N2CCCC2CN(C(=O)CCSCC(N)=O)C)=O)c1 56299,N(C1CCNC(=O)c2[nH]ccc21)C(C1CCC(C(=O)OC)CC1)=O 56300,c1(OC)ccc(OCC(=O)NC(C)C(C)(C)NC(C23CCCC2(CO)C3)=O)cc1 56301,C1(C(N2CCN(Cc3cc(C4CCCC4)no3)CC2)=O)CC2(CSC2)C1 56302,c1(C(N(C2CCN(C(C(COC)C)=O)C2)C)=O)c[nH]c(=N)c(C)c1 56303,C1(C(=O)NC2(n3cncn3)COC2)C2CC1N(C(c1cnc(Cl)s1)=O)C2 56304,C12(NC(c3cc(C)sc3)=O)CCCC1CN(C(c1cc[nH]n1)=O)C2 56305,C1(CNC(CC(C=C)(C)C)=O)CN(C(=O)CCc2nc(C)no2)CC2(CCC2)O1 56306,C1(CC#C)(C(=O)NCc2snnc2C)CCN(C(c2cccc(C)n2)=O)C1 56307,CCC(CC(=O)N(C)CC1C2CN(C(=O)CC3CC4(CCO3)CC4)CC12)C(C)C 56308,c1(C(=O)NCC23CC(CO2)N(C(=O)CC=C(Cl)Cl)C3)c(F)ccc(Cl)c1F 56309,C1(NC(c2c(CC)occ2)=O)CC(C2CCN(C(c3ncnc(C)c3C)=O)C2)C1 56310,C1(N(C(=O)C(C2CCOC2)C2CC2)C(C2CC2)C2CC2)CCC(F)(F)CC1 56311,C(C)(C)(CN=c1[nH]nc(C#N)s1)C1CCN(C(COc2c(C)cc(Cl)cc2C)=O)C1 56312,C12(NC(C3ON=C(CC)C3)=O)CCCC1CN(C(=O)Cc1csc(C)n1)C2 56313,Cn1cc(CCC(N2CCC(c3ccco3)C2)=O)cn1.C12CC1C(=O)N2 56314,c1(-n2c(C(=O)Nc3c(O)n[nH]c3-c3ccccc3)ccn2)ccccc1F 56315,CC1CC(N(C(=O)C(C)(C)CN(C(=O)Cc2cncnc2)C)C)CC(C)O1 56316,N1(C(C2(c3cccc(OC(F)F)c3)CCC2)=O)CC(NC(=O)C2CC2)CC(O)C1 56317,N1(C(CC(N)Cc2ccc(OC(F)(F)F)cc2)=O)CC2NCCOC2C1 56318,C(=O)(C(C)CC(C)C(C)=O)NC1C(C(=O)NCC2(CC(=O)OC)CC2)CC=CC1 56319,CCCC(CC)C(=O)NCCCNC(=O)C(O)Cc1c(F)cccc1Cl 56320,C(CN=c1[nH]c(=NC(C)c2ccccc2F)c2cc(Cl)ccc2[nH]1)NC(=O)NC 56321,c1(OC)cc(NC(C2CC2NC(c2cc(Br)ccc2C)=O)=O)cc(C#N)c1 56322,c1(C(=O)NCC(c2cccc(Cl)c2Cl)F)cc(Cl)c([N+](=O)[O-])[nH]1 56323,n1(CC)c(Sc2nccc(NC(=O)CN(C)C)n2)nc2ccc(Br)cc12 56324,N1(C(Cc2cc(C)[nH]n2)=O)CC(NC(C2CC3(CCCO3)C2)=O)CCC(O)C1 56325,c1(OC)ccc(C(=O)OC(c2cnn(C)c2C)=O)c(OCCN(CCC)CC)c1 56326,c1(C(N2CCC(F)(C(=O)Nc3ncc(Cl)nc3Br)CC2)=O)cc(Cl)cc(Cl)c1O 56327,C=CCC(C(=O)N(C)CCN(C(=O)C(O)c1ccsc1)C)C(C)(C)C 56328,C(=O)(C(C)(C)S(=O)(=O)C1CC1)NCC(CNC(CCc1c(C)cccc1)=O)(C)C 56329,C1(C#CC(=O)N2CC(O)CC2C(N2CCCCC2CO)=O)(CC)CC1 56330,N1(C(c2c(C)nc(O)s2)=O)CCN(C(=O)CCc2cn(C)nn2)CC(C)C1 56331,N1(C(C=COCC)=O)CC(NC(c2cnc(OCC(F)F)cn2)=O)CC2(CC2)C1 56332,c1(C(=O)Nc2cnccc2Cl)n[nH]c2c1CN(Cc1cn3ccccc3n1)CC2 56333,C1(C(NOC(C)C)=O)CCC(NC(=O)COCCF)CC1 56334,Cc1cncc(CC(=O)N(CCC(=O)NOC(CO)C(C)C)C2CC2)c1 56335,CC1=C(Br)CN(c2ccnc(NCc3ccc(C4CCCOC4)cc3)n2)CC1 56336,c1(C(=O)NCCN(C(=O)C(C)N2CCC2)CC)cc(C(=O)OC)c[nH]1 56337,c1(OC)cc(Cl)c(CN2CCCN(C(C3CCCN3C(C)C)=O)CC2)c(Cl)c1 56338,c1(C(N2CC3C(C(=O)Nc4c(C)cc(Cl)nc4)C3C2)=O)ccc(F)c(C#N)c1 56339,c1(SC)cc(C(=O)NCC2CC(F)(CNC(=O)CCc3csc(=N)[nH]3)C2)c(C)o1 56340,c1(CCN2C3CCN(C(=O)OC(C)(C)C)C3CCC2)ccc2cc(O)ccc2c1 56341,C1(NC(CC2N(C(C(C)OCCC=C)=O)CC(O)C2)=O)CCC(C)(C)CC1 56342,Cc1cc(NC(=O)CSCCNC(C2CC3(C2)CC32CC2)=O)c(F)cc1F 56343,C(CC(C(=O)N(C)CCO)NC(=O)CSCCNC)SC 56344,C(=O)(CS(=O)(=O)CC(=O)OC)NC1C(NC(C(COC)C)=O)CCC1 56345,CC1CC(C(=O)NCC2(F)CN(C(c3cc(O)cc(O)n3)=O)C2)Cc2nn[nH]c21 56346,C1(C(=O)NC2CC(CO)C23CCC3)(CC)CCCN(C(=O)CC(C)F)C1 56347,N1(C(c2cc(C)nc(C(F)(F)F)n2)=O)CC2(CCCN(C(=O)C(C)C3CC3)C2)C1 56348,C1(C)(NC(c2ccc(C(C)C)nc2)=O)CCN(C(C2CCC(F)C2)=O)CC1 56349,CC1CC(=O)NC(C(=O)NC(C2CC2C(=O)NCC=C2CCSCC2)C)C1 56350,C(C(C)(C)C#CC(=O)NC1CS(=O)(=O)C1)NC(Cn1c(C)ccc1C)=O 56351,Cc1cnc(C(=O)NC2CCC2NC(c2cc(Cl)nnc2O)=O)cc1Cl 56352,C1(CNC(C(C)NC=O)=O)CCN(C(=O)C(C(C)(C)C)N(C)C)CCC1(F)F 56353,c1(C(=O)NC2C(NC(C(=Cc3cccs3)C)=O)CCC2)cc(Cl)ccn1 56354,N1(C(C2(NC(c3ccncc3O)=O)CC(OC)C2)=O)CCC2(C1)CC2(F)F 56355,N1(C(c2c(CC)[nH]cc2)=O)CCN(C(=O)C(C)NC(C)=O)CC1C(F)F 56356,Cc1cncc(C)c1C(N1CCOC(CCNC(C2CCC(C)(C)OC2)=O)C1)=O 56357,CC1CC(NC(=O)C(c2ccccc2)NC(=O)CCn2cnnn2)CCO1 56358,C1(NC(CCC#CC)=O)CCN(C(c2c(C)noc2CCC)=O)CC1C 56359,C1(O)(CNC(C2CC(N(C)C)C2)=O)CN(C(=O)COc2ccon2)C1 56360,C1(OC)CCC(C(N2CC(N(C)C(c3cnn(C(C)C)c3F)=O)C(O)C2)=O)CC1 56361,c1(OC)cc(CN(CCCNC(c2csc([N+](=O)[O-])c2)=O)C2CC2)c(OC)cc1C 56362,CCC(C)(CO)C(=O)N1CC2(CCN2C)C1 56363,CCCCCC(F)C(=O)NC1CC=C(C(=O)N2CC(O)CC2CC(C)C)C1 56364,C1(NC(C(=Cc2cccc(Cl)c2)C)=O)C(C)CCN(C(=O)C(C)CO)C1C 56365,C1(CCC(=O)NCCC(C)(C)F)CCCCN(C(=O)C=CC2CCOCC2)C1 56366,CC1CN(C(=O)CC2(O)CCCCC2)CC1(C)CNC(=O)C=CBr 56367,C(CC(C)C(=O)N(C(C)C(=O)N(C1CC(C)(C)C1)C)C1CC1)=CCC 56368,CC(O)CC(C)(C)CNC(C1CN(C(c2ncncc2N)=O)CC1(F)F)=O 56369,c1(C(N(CC(CC)NC(c2coc(Cl)c2)=O)C)=O)ncc2[nH]ncc2n1 56370,Cc1ncccc1NC(=O)C(C)CN(C(=O)C(C)O)C 56371,C1(C(=O)NCCC=CCCC)C=CCN(C(C2CC=CC(O)C2)=O)C1 56372,N1(C(C2(CCOC)CCC2)=O)CCC(NCCCC2CCOC2)C(C)C1 56373,C(CC(C)C(=O)NC(c1cccnc1)C(=O)NCc1cnc[nH]1)=CCC 56374,c1(C(=O)NCC2N(C(C(CC#C)C)=O)CCC(C)C2)ccc2nc[nH]c2c1F 56375,C(=O)(C(CC)CC(F)(F)F)N1CCC(CNC(c2cc(CC)on2)=O)C12CC2 56376,c1(C(N2C3C(NC(C4(C)CC5CC5C4)=O)C(C3)C2)=O)cc2cnccc2[nH]1 56377,c1(N2CCC(NC(C(N3C(=O)CCC3=O)C)=O)C(F)C2)ncc(C#N)cc1Br 56378,C(=O)(C1=C(C#N)CCC1)N1CC(N(C(c2ccc(-c3nc(C)on3)cc2)=O)C)C1 56379,c1(OC)cccc(CNC2C(C(=O)C(F)(F)CSC)CC2O)c1 56380,N1(C(c2cc(C)oc2)=O)CCN(C(c2ncc3[nH]ncc3n2)=O)CC2(CC2)C1 56381,CC1CC(C(N2CC(C)(NC(=O)C(c3cccc(F)c3)C)C2)=O)CC(C)O1 56382,c1(CCC(=O)N(CCCNC(C2CC3(F)CC2C3)=O)C)ccc2c(c1)CCO2 56383,C1(C)(C(N(CC(=O)N(CCC#C)CCO)CCOC)=O)CC2CCC1C2 56384,Cc1ccnc(CNC(=O)CC2CN(C(=O)OC(C)(C)C)CC2C)n1 56385,C=CC(C)(C)CC(=O)NCC1CN(C(=O)C=Cc2cncs2)CC1O 56386,c1(NC(C(C)(C)C)=O)ccc(NC2(c3cccc(Br)n3)CCC2)cc1 56387,C1(CNC(CCCN(C(C)=O)C)=O)CCCCN(C(c2cocc2C(N)=O)=O)C1 56388,C1(F)(C(=O)OCC)CN(C(=O)CC(c2cccc(F)c2)O)CC12COC2 56389,N1(C(CN(C(=O)COCC(C)(C)C)CCOC)=O)CCC(CO)(CO)C1 56390,c1(C(=O)NC2C(CNC(C(CCCOC)C)=O)C2)cccc2c1OC(C)(C)CC2 56391,Cc1csc2c(C(N3CCCCC3CNC(=O)CC34CCCC3C4)=O)cccc12 56392,C(=O)(C(C)CC(C)(C)C)NCC(CC)N(C(=O)CSC(F)F)C 56393,c1(C(N2CCCC(N(C(c3nc(C)c(C)s3)=O)CC)C2)=O)nc(C)ccc1F 56394,C(=O)(C(F)CC(C)C)NC1(CCOC)CCN(C(CCC=C)=O)C1 56395,C1(C)(CC(=O)NCC(C)Cn2ccnc2)CCN(C(=O)CC2CC(C)(C)C2)C1 56396,c1(C(=O)NCc2cc(C(=O)NC(C(=O)OC(C)C)C)ncc2)ccc(=O)n(C)n1 56397,N1(C(C(C)OCC)=O)CC2(CCCC(CNC(c3nn(C)cc3[N+](=O)[O-])=O)O2)C1 56398,C(N=c1[nH]c(=NCC(=O)N2CCCO2)c2c(F)cccc2[nH]1)c1scc(CC)n1 56399,Cc1cc(C=CC(=O)NCC2(O)CCCN(C(c3ccccn3)=O)C2)ccc1F 56400,N(C(=NCc1ncn(C)n1)NCC(C1CCOCC1)(F)F)C1CC1.C(C(C)(C)C)NC 56401,C=C(CNC(=O)Cc1ccsc1)CCNC(C1CCN1C(C)=O)=O 56402,C=C(C)C(C)(C)C(=O)NC1CCC(C)(CNC(=O)CNC(C)=O)CC1 56403,C(c1ccccc1F)=CC(=O)N(C(C)CCNC(C1(CF)CCOCC1)=O)C 56404,c1(OC)cc(C(=O)NC2CC(C)(NC(=O)CN(C)CCO)C2)cc2c1OCCO2 56405,c1(C(=O)NC2C(CNC(CC(=O)N(C)C)=O)CCC2)cc2cc(Cl)c(Cl)cc2[nH]1 56406,C1(NC(CC(C)(C)C)=O)CCN(C(=O)CCCOc2ccccc2Cl)CC(O)C1 56407,C1(N(C(c2c(C)cns2)=O)C)CN(C(c2ccsc2)=O)CCC1O 56408,N1(CC(N2CCC(OCC(=O)OC(c3ccncc3)C)C2)=O)CCCC(CO)C1 56409,c1(C(=O)NC23C(NC(c4cnns4)=O)CC(CC2)C3)cc2sccc2cn1 56410,c1(N(CC)Cc2ccco2)ccccc1C 56411,C(=O)(CCCCCC#N)N1C(CNC(=O)C=Cc2ccccc2)CC(COC)C1 56412,Cc1cnsc1C(=O)NC1CCC(N(C)C(c2cn(-c3ccccc3)cn2)=O)C1 56413,N1(C(CCCC2(NC(C=CC(C)C)=O)CCC2)=O)CC(S(C)(=O)=O)C1 56414,c1(C(N2CC=CC(NC(C(C=C=C)C)=O)C2)=O)cc([N+](=O)[O-])n[nH]1 56415,N1(C2CCN(C(CCNC(=O)OC)=O)C2)CCN(C(C2CCCSC2)=O)CC1 56416,N1(C(c2cnc3n2CCC3)C(=O)NC2(C)CC2)CCC(O)C2CCCCC12 56417,C1(CC)CN(C(=O)COCC2CC2)CCC1NC(C1CC(O)(C#N)C1)=O 56418,CCCC(C(=O)N(CCNC(=O)C(c1ccccc1)F)CCOCC)NC(N)=O 56419,c1(C(N2CCC(CC(N3CC(F)C(F)C3)=O)C2)=O)cnnc(Cl)c1 56420,C1(NC(CN(C)Cc2nnc(C)n2C)=O)CC2CC1N(C(C1(C)CCCC1)=O)C2 56421,N1(C(CC2C(C)(C)CCCO2)=O)CC2CC(C1)CN(C(C1C3CCCCC13)=O)C2 56422,Cc1ccccc1N=c1[nH]c(N2CCC(CC3CCN(C)C3=O)CC2)nc(=N)[nH]1 56423,c1(CNC(=O)Nc2ccc(-c3n(CC)cnn3)cc2)nc(C)c(C)c(C)c1C#N 56424,Cc1nc2sccn2c1C(=O)NC1(C2CCCN2C(C2COCCO2)=O)CC1 56425,CC1(C(=O)NCC(c2ccc(O)c(O)c2)O)CCCN(CCN2CCCCC2)C1 56426,c1(C(=O)NC2C(NC(C(COCC)(C)C)=O)CCC2)ccc(P(C)(C)=O)nc1 56427,c1(C(C2CC2)OC)nc(C2CCCc3ncnn32)n(-c2ccc(C(C)C)cc2)n1 56428,c1(C(N(C2CCCN(C(=O)C(F)=CCCF)C2)CC)=O)cnc(C2CC2)nc1O 56429,CCN=c1ccc(C(=O)NC(CO)C(C)NC(c2ccc3c(c2)COC3)=O)c[nH]1 56430,c1(CC)nccnc1C(=O)NC1(CNC(=O)COc2cccc(F)c2)CC1 56431,C1(C(=O)NC(C)C(=O)NCCF)(CC)CCN(C(=O)C(CO)OC)C1 56432,N1(C(c2c(SCC)nccn2)=O)CCN(C(=O)C2=CCCC2)C(C(C)C)C1 56433,C1(C(=O)NCCC(C)NC(c2c(C)onc2CO)=O)CCCCN1S(N)(=O)=O 56434,C1(NC(Cc2cc(CC)nn2C)=O)CC(O)CN(C(=O)CCC2(CO)CC2)C1 56435,c1(C(=O)NC(CNC(CN(CCC)C)=O)C(C)C)cc(C)c(C)c(S(N)(=O)=O)c1 56436,c1(OCC(=O)NC(CN(C(c2cnc(C(=O)OC)s2)=O)C)C)ccc(F)cn1 56437,CCC(C)C(O)C(C)C(=O)NCCC1(NC(=O)C(C)=C(C)C)CCCC1 56438,CC1C(NC(=O)C=Cc2nccs2)CCCN1C(=O)CC(C)c1ccccc1 56439,Cn1ncc(C(N2CCCC2CNC(c2cnn(C3CCC3)c2)=O)=O)n1 56440,c1(OC)c(Cl)ccc(C(=O)NC2CC(CNC(c3nnc(Cl)cc3N)=O)C2)c1F 56441,C1(C(N2CCCCC2C2CNC2)=O)CC(F)(F)CCO1 56442,N1(C(C(C(=O)OCC)F)=O)CCC(NC(c2ccc(CO)cc2F)=O)C12CC2 56443,C(CCN=c1[nH]c(=NC(C)c2ncc3ccccn23)[nH]c2c1CSC2)OC 56444,C(C)(CC(C)NC(=O)CNC(c1cscn1)=O)NC(C1(CCOC)CCC1)=O 56445,N1(C(CN(C(C)=O)C)=O)CC(O)CC1CNC(=O)C(CO)c1ccccc1 56446,c1(OC(F)F)ccc(-c2ncn(C3CCC3)n2)cc1.C1(C2CC2)CCCO1 56447,C1(NC(c2cc(C)cc(F)c2)=O)CCC(O)CN(C(=O)COCC(F)(F)F)C1 56448,N1(C(c2cc(CC)oc2C)=O)CCC(CNC(=O)CC23CCCC2C3)C(O)C1 56449,N1(C(c2csc(C)c2C)=O)C(C)CC2CN(C(=O)CCC3(C)CC3(F)F)CC12 56450,Cc1ccc2oc(C(=O)NC3(C)CC(NC(=O)COC4CCCCC4)C3)cc2n1 56451,CCC(CC)(CC)C(=O)N1CCN(C(c2nc(C(C)(C)C)no2)=O)C(C)C1 56452,N1(C(C23CC(OC)C2C3)=O)CCN(C)C(CNC(c2ccc(O)nc2)=O)C1 56453,C(=O)(CCCN=[N+]=[N-])NCC(C)CNC(c1cc(C2CCCN2C)[nH]n1)=O 56454,C(N=c1[nH]c2cc(Cl)c(S(=O)(=O)NCC(Cl)(Cl)Cl)cc2s1)C1C(C)OCC1 56455,C1(NC(c2c(CC)ncs2)=O)COC2(C1)CN(C(C1(C)CCC(C)CC1)=O)C2 56456,C1(F)(CNC(C2CCC(=C)CC2)=O)CCCN(C(C2(F)CC=CCC2)=O)CC1 56457,N1(C(c2cccc(C)c2Br)=O)CC(NC(C2CC(O)C2)=O)CC12CCCC2 56458,c1(Nc2ccc(C(N3CCCC3CCO)C(=O)NCCO)cn2)ccc(F)cc1 56459,C1(CN(C(C(CC)F)=O)C)CCCCN1C(=O)CCCSC 56460,C1(CNC(C2CC3CCC2O3)=O)CN(C(=O)CSc2ccccc2O)CC1(F)F 56461,c1(C(N2CC(C)C(NC(C3CCN(C)C3=O)=O)C2)=O)cnc2c(Cl)cccn12 56462,N1(C(C(C)SC(C)C)=O)CCCCC(C(=O)NCC2CCCOC2(C)C)C1 56463,c1(C(c2cccnc2)N2CC(CNC(CCN(S(C)(=O)=O)C)=O)C2)ccc(F)cc1 56464,N1(C(=O)OC(C)(C)C)CCC2CCN(CC(c3ccccc3)O)C2C1 56465,CCS(=O)(=O)CC(=O)N(C)CCn1cc(-c2ccc(Cl)c(F)c2)nn1 56466,c1(CC(N2CC(CC(C)NC(c3occc3F)=O)C2)=O)ccc(Br)cc1F 56467,C1(C(N(CCC(=O)Nc2c(CC)c[nH]c2)C(C)C)=O)(N)CCCCC1.CC 56468,c1(C(=O)NC2C(NC(C=CCC)=O)CC2)cc2ccc(Cl)cc2c(=O)o1 56469,Cc1c(C(N2CCC(O)(C(C)NC(=O)C(C)(C)CO)C2)=O)cc(Br)cc1N 56470,C(=O)(CC(C)(C)Cc1ccc(Cl)cc1)NC(CC)(C)CNC(c1cccnn1)=O 56471,n1(CCCCSC)nnnc1C(c1cccn1C1CC1)NCCC1(C)CC1 56472,c1(C(N2CCCC(CCC(=O)NCCCNC(=O)OC)C2)=O)ccc(C)c(O)n1 56473,C12(C(=O)OC)CC1CN(C(=O)C(Cn1cncn1)NC(=O)C(C(C)C)SC)C2 56474,CCCC(C(=O)NC(C(=O)NC)C1CCCC1)NC(c1cnn(C)n1)=O 56475,c1(N2CC=C(CNC(C3C(C4C(C)C4)C3)=O)CC2)nc(Cl)nc2c1ncn2C 56476,C#CC1CN(C(=O)CC2CCCCC2C)CCN1C(c1cccc(C(C)=O)c1)=O 56477,c1(-c2cn(CCN(C(C=C(CC)CC)=O)C)nn2)c(F)cccc1F 56478,C1(NC(Cc2nc(C)sc2C)=O)CC2(NC(=O)C(C)n3ccnc3)COC1C2 56479,Cc1cc(=NCCCC(C)(C)NC(c2ncc(F)cn2)=O)[nH]c(C(F)(F)F)n1 56480,C1(C(C)C)CCN(C(=O)C(C#N)C2CC2)CC1.C(=O)(CC(C1CC1)C1CC1)N 56481,C1(C(N2CC(O)(CC=C)C2)=O)CC2C=CC1N(C(C1(CC=C)CCCC1)=O)C2 56482,C(=O)(C(F)C1=CCCCC1)NC1(C)CN(C(=O)C(c2cccc(F)c2)(C)C)C1 56483,c1(C(=O)NC2C(NC(C(Br)=C(C)C)=O)CC2)cc2ncccc2o1 56484,N1(C(Cc2cc(C)no2)=O)CC2CCCCN2CC1CNC(c1oncc1C)=O 56485,N1(C(C)=O)CC2CCC1C1CN(C(c3c(F)cc(F)cc3F)=O)CC21 56486,C1(OC)COCCC1CNC(c1csc(CNC(=O)CCOCC(F)F)c1)=O 56487,c1(C(=O)NC(C)CCCNC(=O)CC2CCCS2(=O)=O)ncccc1C#N 56488,O=C(C(F)CC1CC1)NC1CCCC1NC(c1cnn(CC2CC2)c1)=O 56489,C(=O)(C(C)C(C)CC)N1CC(CCCCNc2ccc(OCC#C)cc2)C1 56490,c1(C(=O)OC)ccc(C(=O)NC2CCC2NC(C2CCCN(CC)C2)=O)cc1Cl 56491,N1(C(c2ccc(OCC)cc2)=O)CCN(C(C2(C)CC2C)=O)CC1c1cn[nH]c1 56492,CCC(c1ccc(C)cc1)=CC(=O)NC(C)CNC(c1n[nH]cc1OC)=O 56493,c1(C(N(C)CCOCCN(C)C(C2(C)CC2F)=O)=O)ccc2c(c1)OCC2 56494,N1(C(c2ccc(C3(C)CC3)cc2)=O)CC2(CCN(C(C3(C)CCCN3C)=O)C2)C1 56495,C(=O)(CCC(=O)NC(C)(C)CC(=O)NCCC1(COC)CCC1)NCC 56496,CC1(CNC(=O)NC2(c3cccc(O)c3)CCCC2)CCCCCC1 56497,C1(SC)CN(C(c2c(C)noc2C(F)F)=O)CC1NC(=O)CCC(N)=O 56498,c1(SCC)ccccc1-n1nc(C(C)OC)nc1-c1cccc(C2CCOC2)c1 56499,c1(C(c2nnnn2CC(F)F)NCCCc2n(C)ncc2)snc(OC#N)c1Br 56500,N1(C(CC(CC)(C)C)=O)CCC2(CCCN2C(c2sccc2C)=O)C1 56501,C1(C(=O)NC2CCCC2NC(C2(CO)COC2)=O)CC12CC(F)(F)C2 56502,CCCCC(C(=O)NCC1(F)CCN(C(=O)C(O)(C2CC2)C2CC2)C1)C(C)C 56503,N1(C(C(F)=CC)=O)CCC(C2CCCN(C(c3n[nH]c(CC)c3Cl)=O)C2)C1 56504,C12(NC(C3CCCOC3c3ncc[nH]3)=O)CC1CN(C(C1(O)CC1)=O)C2 56505,C1(CNC(COCCC(C)C)=O)COCCN(C(C2OCCOC2C)=O)C1 56506,c1(C(N2CCSCC2(C)c2ccccc2)C(=O)NCCC)cc(Cl)c(Cl)c(Cl)c1 56507,C1(C(=O)NC(CC)(C)CC)N(C(c2c[nH]c(=NC)o2)=O)CCCC1(C)C 56508,N1(C(CC2C(C(=O)O)C2)=O)CC2(CNC(C34CCCC(O)(CC3)C4)=O)CC1CCO2 56509,Cc1nc(Cc2ccccc2)oc1C(=O)NCC1CCN1C(C1CC1F)=O 56510,C1(NC(CC(CC)O)=O)CC2CCC(C1)N2C(=O)C(c1ccc(F)cc1F)C 56511,C(C#N)(c1ccccc1)=C1CCCN(C(CCc2scc(C)n2)=O)C1 56512,c1(C(=O)NC2CCCN(C(C(CCC)=CCC)=O)C2)cc2ccc(Cl)cn2c1 56513,C(CNC(=O)C=CC(F)F)(CC(=O)NCC1COC(C)(C)C1)OC 56514,C1(NC(CCNC(=O)NC)=O)CCN(C(c2c(C)ccoc2=O)=O)CCC1(F)F 56515,c1(C(N2CC(C(C)(C)O)(CNC(C3C(OCC)C3)=O)C2)=O)nn(CC)nc1C 56516,c1(OC)cc(C(=O)NCC(COC)NC(C2(C)CCCCC2C)=O)cnc1C 56517,N1(C(C2C(C)(CC)CCC2)=O)CC2(C(=O)Nc3cn(C)nc3C#N)CCC1CC2 56518,c1(CNC2C(c3ccc(OC)cc3)C2)ccc(C)nc1O 56519,N1(C(CCSCCCC)=O)CC2CC(N=c3[nH]nc(C(N)=O)s3)CC1C2 56520,N1(C(c2cn(C)c(=O)cn2)=O)CC2CCN(C(=O)CC=C(Cl)Cl)CCC2C1 56521,CC1NC(=O)CCC1CNC(C1(CNC(c2ccncn2)=O)CCCO1)=O 56522,c1(CN2CC=C(CNC(C3C(C)C3C)=O)CC2)cccc2cc[nH]c12 56523,C1(SC)CCN(C(=NCC2SCCS2)NCC(=O)NC(C)C)C1 56524,N1(C(CCc2cc(OC)no2)=O)CC(NC(=O)C=CCO)C2(CC2)C1 56525,c1(C(=O)NCC(C)NC(C2CC3C(C2)C3(F)F)=O)ncc2[nH]ncc2n1 56526,N1(C(C(C)=C(C)C)=O)CCC(NC(C2(C)CC2(F)F)=O)C(C)C1 56527,C1(OC)CN(C(C2CC3(CCC3)C2)=O)C(C)(CNC(c2ccc(F)cc2Cl)=O)C1 56528,N1(C(c2c(C)cns2)=O)CC(NC(=O)Cn2cc(C#N)cn2)C(C(F)F)C1 56529,CC1CCC(Cl)=C(C(=O)N(c2ncnc3cnccc23)C)C1 56530,C(=O)(C1CCCc2scnc21)NCC1CCN(C(C2C(C(=C)C)OCC2)=O)CC1 56531,N1(C(C(C(C)C)OC)=O)CCC(CNC(=O)C(C)(C)O)C(F)(F)CC1 56532,c1(-c2c(C(=O)NCCN3CCN(CC(C)OC)CC3)cn(C)n2)ccc(F)c(C)c1 56533,N1(C(CC2(C)CCOC2)=O)CCC2(CC2)CC1C(=O)NCC1(C#N)CCCCC1 56534,CC(C)C(O)CC(=O)N1CC(F)CC1CC(=O)Nc1ccc(Cl)nc1 56535,Cc1ccc(C(=O)NCC(=C2CN(C(c3ncccc3Cl)=O)C2)F)cn1 56536,C1(CC(N2C(COC)CCC2)=O)(NC(=O)Cn2nccn2)CCCCC1 56537,c1(NC2CC(C)N(C(c3cccc(OCCF)c3)=O)C2)ccccc1[N+](=O)[O-] 56538,C(c1cnc[nH]1)=CC(=O)NCC1(C(F)(F)F)CCCC1.c12ncoc1CNC2=O 56539,c1(CC(=O)NC2CCN(C(CCCCCC)=O)CC2O)ccc2cccnc2c1 56540,c1(OC)ccc(SC(C)C(=O)NC2(C)CC(NC(=O)CNC(C)=O)C2)cc1 56541,CN1N=C(CC(=O)N2CCC3(NC(c4ccnc(Cl)c4Cl)=O)CCCC23)CC1=O 56542,CC(C)(F)CCC(=O)NCC1CCC(NC(=O)CC2COC(C)(C)CO2)CC1 56543,O=C1NCc2cc(CNC3CCCCC3Nc3ncncc3F)ccc21 56544,C1(COC)(NC(=O)CSCC(N)=O)CCN(C(=O)C=CCN2CCOCC2)C1 56545,C1(NC(c2ccccc2CO)=O)CN(C(=O)CC2CCNC2=O)CC(F)(F)C1 56546,C1(C(N2CC(N3CCC3)C2)=O)CCC(O)CN1C(C1CC2(CSC2)C1)=O 56547,N1(C(C(C)OC)=O)CC2CCC(C1)C(NC(c1cccc(OC(C)C)c1)=O)C2 56548,N1(C(c2nc(C)c(C)[nH]2)=O)CCCC2CN(C(=O)CSC3CCOC3=O)CCC12 56549,C1(C2CCN(C(=O)Cc3ccsc3)C2)(NC(c2cncc(C=C)c2)=O)CC1 56550,CC1(C)CN(C(c2ccc(=N)[nH]c2)=O)CCC1NC(c1ccc(C(N)=O)cn1)=O 56551,C(=O)(C(F)CC(C)C)N(C(C)Cc1ccc(OC)cc1OC)CCOC 56552,N1(c2c(Cl)cnc(OC)n2)CCC(C)C(NC(c2cn(C3CCC3)nn2)=O)C1C 56553,Cc1ccc(C2=CCC(C#N)CC2)c2[nH]c(C(=O)NCCc3ccnn3C)cc12 56554,Cc1[nH]c2ncccc2c1C(=O)NC1CN(C(c2nn[nH]c2Cl)=O)C(C)(C)C1 56555,C=CC1(C(N2CCOC(C#N)C2)=O)CCN(C(c2cc(CC)no2)=O)CC1 56556,C(=O)(CCCOC(C)(C)C)N1CC(C(C)NC(C=C(C)C(F)F)=O)C1 56557,C(=O)(C(C)(Cc1ccncc1)N1CCN(C)CC1)OC 56558,N1(C(C(C2CCCOC2)OC)=O)CCCC2C1CCN2C(=O)CN1CCS(=O)CC1 56559,C(CCCCC(=O)N1CCCC(NC(=O)COCC2(F)CC2)C1C)SC 56560,c1(CC)ccc(C)cc1C(=O)NC1CN(C(c2cc(Cl)n(C)n2)=O)CC1C 56561,N1(C(Cc2c(C)noc2)=O)CCC2CN(C(c3cccc(=O)n3C)=O)CCC2C1 56562,C#Cc1cc(C(=O)NCCC2CCN2C(=O)C(=CC2CCCC2)C)ccc1C 56563,C(CCO)(C(C)(C)C)NC(CCC(C)NC(=O)CCc1ncccn1)=O 56564,c1(NC(=O)NCC(=O)NCCC2CCCN2Cc2cccnc2)ccc(F)cc1 56565,c1(C(N2CCC(C(C)(C)NC(C(C)O)=O)CC2)=O)cc2occc2s1 56566,c1(C2C(C(=O)NCC3C(CNC(C(N)=O)=O)C3)C2)ccc(F)c(F)c1 56567,c1(CC)nnsc1C(=O)NCC(C)(O)CNC(=O)CCC1CCCOC1 56568,C(=O)(C(C)(O)CC(F)F)NCC(CN(C(CCn1c(C)nc(C)n1)=O)C)(C)C 56569,c1(C(C(N2CCC(NC(Cn3c(=N)nc[nH]3)=O)(CF)C2)=O)=O)ccc(F)cc1F 56570,O(NC(=O)C(CC(N)=O)N(CCF)C1CC1)CCC(C)C 56571,CC(C)(CC(=O)NCC(C1CCOC1)NC(=O)Cn1nnc(=N)[nH]1)CC(F)F 56572,c1(CC)ccc(C=CC(=O)NCC2CC(C(F)(F)F)CN2C(C2COC2)=O)cc1 56573,Cc1ccc(-n2cc(C(C)N(C)C(C3CCN(C)C3)=O)nn2)c(Br)c1 56574,C(=O)(C(O)CC(F)(F)F)NCC1(C(C)(C)C)CCN(C(=O)C(C)(C)C(F)(F)F)C1 56575,C1(NC(=O)Cc2ccnc(Cl)c2F)C2CCC1N(C(=O)CC1CCCC1(F)F)C2 56576,c1(NC(C2(CCC=C)CN(C(=O)CN3CCC(C)C3)C2)=O)cnc(C)c(C)c1C 56577,C=CCCCCC(=O)NCc1csc(CCC)n1 56578,C1(C(N2CC3CC(NC(=O)CCc4cnn[nH]4)C2C3)=O)(CC)CCC(F)(F)CC1 56579,C(=O)(N=c1[nH]c(S(C)=O)nc(Cl)c1Br)NC(c1cccc2cc[nH]c12)CC 56580,N1(C(Cc2c(C)cco2)=O)CCc2sccc2C1CNC(=O)C(Cl)=CCl 56581,N1(c2nccc(OCC)n2)CC2(C)CN(C(c3ccncc3)=O)CC2(C)C1 56582,CC1CC(C(=O)NCC2CC(C(=O)NC3(C)CC=CC3)C2)CCS1 56583,C1(N=c2cnc3cc(F)c(F)cc3[nH]2)(CC)CCN(C(C2CCC(C)O2)=O)CC1 56584,C1(CC=C)(C(=O)NCC(N2CCOC2=O)C)CCCN1C(=O)COCC(F)F 56585,C1(CC(N)=O)(NC(Cc2ncc(C)[nH]2)=O)CCN(C(=O)Cc2ccco2)CC1 56586,S(=O)(=O)(c1cccc(CN2C3CCC2CC(OC(F)F)C3)c1)N1CCN(C)CC1 56587,N(C1CCc2ccccc2-n2ccnc21)C(c1ccc(CC(N)CO)cc1)=O 56588,C1(COC)(NC(=O)C(C)CC(N)=O)CCCN(C(=O)Cc2cccc(C#N)c2)C1 56589,c1(CC)ccc(C(c2nnnn2C2COC2)Nc2ccc(C)nc2)c(C)c1 56590,N1(C(COCCC=C)=O)CCC(Nc2nccc(CC#N)n2)C(C)C1 56591,Cc1nc(C(N2CC(NC(c3cn(C)c(=O)n3C)=O)C3CC23)=O)c(C)n1C1CC1 56592,C(=O)(NN1CCCC1C(=O)NCCCN(C)C)c1c(C)ncs1 56593,CC(C)CC(C(=O)NCC1(C)CSC1)ONC(c1ccc(N)cn1)=O 56594,C(=O)(C(O)CC(C)C)N1CC(NC(c2c(OC)noc2C)=O)C(n2cccn2)C1 56595,c1(C(=O)NC2C(NC(C3(CCOC)CC3)=O)CCOC2)cnc(O)c(Br)c1 56596,N1(C(C(CCSC)(C)C)=O)CC2(CCC(NC(=O)CCNC(=O)COC)CC2)C1 56597,c1(C(=O)NCC2C(NC(CCOC)=O)CC2)ccc(CN2CCCCC2=O)cc1 56598,c1(NC)c(C(N2CCCC(CCF)C2)=O)sc2nccnc12 56599,C1(NC(C(=O)NCc2nc(C3CC3)cs2)=O)CCOc2ccccc2C1 56600,C1(C2(O)CCOCC2)(C(=O)NC2CC3CC(NC(C(CC=C)C)=O)C2C3)CC1 56601,C=CCC(CC(=O)NCCCC)NC(=O)NCC(=O)NC(CN(C)C)C1CC1 56602,N1(C(CCCCC(=O)OC)=O)CCC2C(CCN2C(c2ccc(Br)cc2I)=O)C1 56603,C1(C(=O)NCC(O)C(=O)NC2CC(CO)C2)CCC(O)CC1 56604,CN1CCN(C(C2(CO)COC2)=O)CC1CNC(=O)CSCc1ccncc1 56605,Cc1nc(C2CCC2)ncc1NC(C1CC1Br)=O 56606,C(=O)(C(CC(N)=O)NC(=O)CCn1cncn1)N(C(CC(C)C)C)C 56607,C1(c2nnnn2C)(NCC2(C(C)C)CCC2)CCCN(C)C1 56608,C(=O)(C1=CCCN(C(C2CCN(C(c3ccc[n+]([O-])c3)=O)CC2)=O)C1)OC 56609,c1(CONC(c2ccc(CNC(CC(C)(C)O)=O)o2)=O)ccc2c(c1)CC2 56610,c1(C(=O)NC2CC(O)(CNC(C3C(C)(C)C3C(F)F)=O)C2)cnc2[nH]nnc2c1 56611,CC1(CC(N2CCC(OCC3CC3)C2)=O)CN(C(=O)CCc2ccco2)C1 56612,c1(C(N2CCN(C(C(CC)C)=O)C(c3ccccn3)C2)=O)ccn2cncc2c1 56613,c1(CC(=O)NCC(N(C(=O)CCn2cncn2)C)C2CC2)cccc(C(F)F)c1 56614,N1(C(C)C)CCN(C(C23CC(CN2C(=O)C(F)(F)CO)C3)=O)CC1 56615,c1(N2C(CN(C(=O)CSc3ccccc3)C)CCC2)ncc(S(C)(=O)=O)cc1Cl 56616,C1(NC(C(C)Cc2cccnc2)=O)COCCN(C(c2cc(F)ccc2N)=O)C1 56617,c1(C(=O)NC(CN(C)C(C2(Cl)CC2(C)C)=O)(CO)CO)ccc2ccoc2c1 56618,C(=O)(C1=NOC(C)(C)C1)NCC1(C)C(C)CN(C(c2ccc[n+]([O-])c2)=O)C1 56619,c1(NC2C(Cn3cc(-c4n(CC)ncc4)nn3)CCC2)ncccc1OC 56620,C(=O)(C(O)C(C)C)NC(C(N1CC(O)(CC=C)C1)=O)CO 56621,c1(CN(C(=O)CC2(c3ccccc3)COC2)CC=C)cccc(F)c1F 56622,c1(C(N2CC(NC(=O)NC3CCN(CC)CC3)C2)=O)ccc(OC)c(F)c1 56623,N1(C(c2c(C(C)C)cnn2C)=O)CCC(C)C(NC(=O)C=CCO)C1 56624,CN1CCC(Nc2cc(NCc3nc(C(F)(F)F)n[nH]3)ncn2)CC1=O 56625,c1(C(=O)O)ccc(C(N2CC(Cc3ccc(Cl)c(F)c3)C2)=O)c(F)c1 56626,c1(C(N2C3C(NC(c4c(CC)onc4)=O)CC(C3)C2)=O)c(C)ccc2n[nH]cc12 56627,C(CCNC(=O)COC1(C)CCCC1)(C(=O)N1CCC(CN(C)C)CC1)OC 56628,N1(C(CC=CCNC(CCCNC(=O)OC)=O)=O)CC2CC1C1CC21 56629,C1(C(=O)NCC23CC(CNC(=O)CCn4cccc4)(OC2)C3)CC2OC1C1CC21 56630,S(=O)(=O)(c1cc(F)c(F)cc1[N+](=O)[O-])NC(c1ccc(C(F)C(F)(F)F)cc1)=O 56631,N1(C(c2cc(C)c(F)cc2Cl)=O)CC(C)CN(C(c2ccc(N)cc2)=O)C(C)C1 56632,N1(Cc2cc(OC)c(Cl)cc2)CCC(F)(F)C(C(=O)Nc2ncc(Cl)cc2Br)C1 56633,c1(NC(c2ccccn2)=O)nc(NCCN2CCN(OC)CC2)cc(O)n1 56634,c1(C(=O)NC2C3CCN(C(CN(C4CC4)CC)=O)C32)cc2ccc(OC)cc2[nH]1 56635,C1(NC(COc2cccc(C)c2C)=O)CN(C(c2cc[nH]n2)=O)CCC1(F)F 56636,c1(CC(=O)N(C(C)CN(C(=O)C(O)c2ccco2)C)C)ccccc1C1CC1 56637,CC1CN(C(=O)CC(=O)NC2CC2)CC1CC(=O)NCC1(C)CCCO1 56638,C1(C(=O)NCCC(C)O)(OC)CCN(C(=O)C(O)C(C)C)C1 56639,N1(C(CCOCCOC)=O)CCC(CC(=O)NC2COCC2F)C1(C)C 56640,C(=O)(C1=CCCCCC1)N1C(CNC(C2CC(OCC)C2)=O)C(C)CC1 56641,N1(C(C(C=C=C)C)=O)CCC(C2CCN(C(c3ccc(=O)n(C)c3)=O)CC2)CC1 56642,C1(C(CC)CC)CC(C(N2CCN(C(=O)CCO)CC2)=O)CCO1 56643,c1(NC(C(Cc2cc[nH]n2)NC(CCC(CC)=O)=O)=O)cn(C)c(=O)cc1C 56644,C1(NC(c2ccc(C(C)C)s2)=O)CC2CC(NC(C3(c4cc[nH]n4)CC3)=O)C2C1 56645,C1(C(=O)NCC(CC)(C)C(N)=O)CC(C)(C)CCN1C(=O)C=C1CCCCC1 56646,C1(N(C)C)CCCN(C(=O)CN(C(=O)CCCc2cnn[nH]2)CC2CC2)C1 56647,N1(C(c2c(COC)cc[nH]2)=O)CCN(C(=O)Cc2ccc3c(c2)CC3)C2(CC2)C1 56648,CCC(CC(F)(F)F)C(=O)NCC1C(C2CC2)CCN1c1nnc(C)s1 56649,Cc1ccc(C(N2CCC(O)(C(=O)Nc3nc(Cl)c(C)c(Cl)n3)C2)=O)c(I)c1C 56650,C=CC(C)CC(=O)NCC(O)CNC(c1sc(Br)cc1C)=O 56651,CCCC(O)CC(=O)NC1(CO)CCN(C(=O)CN(CC)Cc2ccccc2)C1 56652,c1(N(C)CC2CCC3CC23)ccc(S(=O)(=O)NCC(F)Br)cc1Cl 56653,c1cc(=NC2CCCSCC2)[nH]c(NCC2CCCOCC2)n1 56654,C(C)(C)(C(=O)N1CC(C(C(=O)NCC2(COC)CCC2)OC)C1)OC 56655,c1(OC)ccc(OCCC(N2CC(O)(CN(C(=O)C(C)=C(C)C)C)C2)=O)cc1 56656,N1(C(CN2CC(=O)NCC2)=O)CCN(C(C2CCC3CC23)=O)C2(CC2)C1 56657,S(=O)(=O)(c1ccc(C(=O)NCC23CCC2CN(C(=O)C=CCO)C3)o1)NC 56658,c1(N2CCN(CC)CC2)nc(C(F)F)nc(=N)[nH]1.C1(=O)CC(=O)N2CCC(C2)N1 56659,CC1(NC(c2cccc(CS(C)(=O)=O)c2)=O)CCN(C(C2CC23CCC3)=O)CC1 56660,C(C(C)C(F)C(=O)NCCC(F)(F)C(C)C)NC(c1cc(C)ns1)=O 56661,C1(N(C(CCC(=C)Cl)=O)C)CCCN(C(c2nocc2Br)=O)CC1 56662,CC(=O)C(C)(C)CC(=O)NCCOCCCNC(c1cc(C(N)=O)c[nH]1)=O 56663,C(=O)(C1=CCS(=O)(=O)C1)N(CCF)Cc1cn(-c2cccc(C(C)C)c2)nn1 56664,c1(C(=O)NC2CC(NC(=O)CC3CCCC34CC4)C2)cc2ccc(Cl)c(F)c2o1 56665,C(=O)(C(CC(F)F)N(C)C(C1CCOC1C(C)C)=O)NCC(=C)CC 56666,C1(N2C(=O)C2C2CCCC2)CCSCC1.c1(CC2CCOC2)ccccc1 56667,C(=O)(C(C)(C)CC(C)C)N1CC(OCCNC(C(F)=CC)=O)C1 56668,Cc1ncc(C(=O)NC(C)C(C)(C)C(=O)NC2CN(C(N)=O)C2)c(=N)[nH]1 56669,C(=O)(CCC(F)(F)C(F)(F)F)N(CCC)CCNC(C1(C)CCOC1)=O 56670,C1(NC(C2N(C(CCC)=O)CCC2)=O)CC2CC1N(C(c1cc[n+]([O-])cc1)=O)C2 56671,c1(C(=O)NCC2C(C)CN(C(C3C=CCC3)=O)CC2)cc2cc(F)ccc2s1 56672,c1(NC(CC)=O)ccc(C(=O)NCCCN(C(=O)C(C)CN(C)C)CCO)cn1 56673,N1(C(CCOCCOCC)=O)CCC2CCC12CNC(=O)C=Cc1cn(C)nn1 56674,C1(NC(CCNC(CN(C(COC)=O)CC2CC2)=O)=O)CCOC(C)C1 56675,N1(C(C(=O)NC(C)C)CC2CCC2)Cc2c(Cl)cccc2C(C)C1 56676,c1(OC)ccc2c(c1)CCC2NC(c1cccc(Cn2nc(C)cc2C)c1)=O 56677,Cc1cc(C(=O)NC2CCCCC2NC(=O)CCC(F)F)c(F)cc1F 56678,C1(C(N(CCCO)CC#C)=O)(OC)CCN(C(C2(C#N)CCCC2)=O)C1 56679,c1(CC(=O)NCc2c(CCNC(C(C)OC)=O)ocn2)c(F)cccc1C#N 56680,CC1CCCC(C(=O)NCCOC2CCN(C(=O)CCCC3CCCC3)C2)C1 56681,CCC(CC)CC(=O)NCc1ncoc1C1CN(C(=O)C(C)(C)C(C)C)C1 56682,Cc1cccc(C(=O)NCCOC2CN(C(C3(C(C)(C)O)CC3)=O)C2)c1F 56683,c1(C(=O)NC2CCN(C(Cc3cncc(C)c3)=O)C2)ccc2c(c1)CCC2=O 56684,C1(C(=O)NCCC(C)N(CCC)C)C=CCCN1C(=O)Cc1ccsc1 56685,C(c1ccc(Cl)cc1Cl)=CC(N1C(C(=O)Nc2ccc(Cl)cc2O)CC(F)C1)=O 56686,N1(C(COCC(=C)C)=O)CCCC(N(C)C(c2ccc(Cl)s2)=O)CC1 56687,c1(NC(=O)CCc2ccc(-c3nn[nH]n3)cc2)ccc(F)cc1O 56688,c1(COC)cccc(C(=O)NC2CCCC(NC(=O)CSC(C)(C)C)C2)c1C 56689,C1(C)(NC(C(C)CC2CCC2)=O)CCN(C(=O)CCCF)C1 56690,CC1(C)CC(C(N2CCCC(O)(CNC(c3ccsc3)=O)C2)=O)CC(C)(C)S1 56691,C1(C(=O)OC)CC12CCC(NC(c1sc(SC)cc1C)=O)CC2 56692,c1(CC(=O)NC2(CCNC(Cc3cc(C)n(C)n3)=O)CC2)ccc(Cl)c(Cl)c1 56693,C12(CNC(=O)COC3CC3)CCC(CC1NC(=O)C(C1CCOCC1)O)C2 56694,c1(OC)cc(F)cc(F)c1S(=O)(=O)NC(C)(C)Cc1cc(F)cc(F)c1 56695,c1(-c2ccc(CC)cc2)cccc2c(C(N3CCC(N(C)C)C3)=O)[nH]nc12 56696,N1(C(c2cc(CC)[nH]n2)=O)CCC12CCN(Cc1cc(C)cnc1Cl)CC2 56697,C1(C(N(CC(=O)OC)CC#C)=O)CC12CCN(C(=O)CC(C)(F)F)CC2 56698,c1(C(=O)OC)cc(C(=O)NCC2(NC(c3conc3C)=O)CCOC2)cn1C 56699,c1(C(c2n(CC)nnn2)(C)NCCC(CC)(F)F)nnc2n1CCOC2 56700,c1(C(=O)NCC2(F)CC(CNC(C(=O)NCCC(N)=O)=O)C2)csc2nccn12 56701,c1(C(=O)NCC2(COC)CN(C(C3CC4CC4C3)=O)C2)cnc2n1CCCC2 56702,C(CC(C(=O)NC(c1cn[nH]c1)C)NC(c1[nH]ccc1C)=O)OCC 56703,C(=O)(C(C)(F)C(=O)NCC(C)(F)CNC(C1CC1CC(C)C)=O)OC 56704,S(=O)(=O)(c1ccc(I)cc1)N1CCN(C(c2ccc(NC)cc2)=O)CC1C 56705,N1(C(C2CCS(=O)(=O)C2)C)CCCC(NC(=O)Cn2cccn2)C1=O 56706,C1(NC(c2c(C)nccn2)=O)(CNC(C2CCCC2C)=O)CC2CCC1CC2 56707,N1(C(C(CC=CC)C)=O)CC(NC(=O)C(C2(O)CCOCC2)(F)F)CC(C)C1 56708,C(C(C)(O)CC(=O)NCC1CC(C)(C)CN1C(=O)Cc1cc(C)ns1)OC 56709,Cc1ccc(CC(C)C(N2CC(NC(=O)C(C)(C)CO)CC2CO)=O)cc1 56710,c1(C(=O)NCC(c2ccccc2)N(C(C(C=CC)O)=O)C)cccc(C(F)F)n1 56711,C(=O)(C1c2c[nH]nc2CN1C(c1cc(CO)on1)=O)N(CCCC)CCO 56712,S(=O)(=O)(c1ccccc1N)Nc1ccc(N(C)Cc2ccccc2)cc1 56713,CC(O)(CNC(c1coc(CNC(C2CC23CCCC3)=O)n1)=O)CCO 56714,c1(C(N(c2ccc(OC)c(Cl)c2)C)=O)ccc2c(n1)CCC2.C1(=O)C(C)O1 56715,C1(NC(=O)C=Cc2ccoc2)CN(C(c2cnc[nH]2)=O)CC12COC2 56716,c1(C(N(C)CC2(CNC(C3CCC4CCC34)=O)CC2)=O)ccc(S(N)(=O)=O)s1 56717,N1(C(C2CCN(C)C2=O)=O)CCC(C)(NC(c2cc(O)nc(Cl)c2)=O)CC1 56718,O=C(CCC(=O)c1cccs1)NCC1(O)CN(C(=O)CCOc2cccnc2)C1 56719,c1(C(=O)NCCCCNC(C2C(C)CCOC2)=O)c(F)ccc(Cl)c1[N+](=O)[O-] 56720,C1(O)(C(C(=O)NC2CCC(C(=O)NC(C3CCCCC3)C)C2)N(C)C)CCCCC1 56721,C(C(=O)NC1CCC1NC(c1csc(-c2ccc(C)n2C)n1)=O)(C(C)C)SC 56722,C1(NC(c2c(C)coc2C)=O)C2CCC1N(C(c1cscc1Br)=O)C2 56723,n1(CC)nnnc1C(c1nc(C(=O)OC)cs1)NC1CC1c1ccccc1 56724,C(C(=O)C1(NC(c2nc(COCC)oc2)=O)CC1)(C(C)C)NC(C(CC)SC)=O 56725,Cn1nccc1C=CC(=O)NC1CC(NC(c2ccsc2C#N)=O)C1 56726,N1(C(c2c(CC)nccc2)=O)CC(O)CC1(C)C(=O)NC1CC(N2CCCC2)C1 56727,N1(C(C2(CC)CCCCC2)=O)CC2(CC(NC(C3(O)CCC3)=O)c3nccn32)C1 56728,CC1(C)CC(C(=O)NCC(O)(CO)CO)CN(C(=O)Cn2cnnc2O)C1 56729,c1(-c2cccc(OCC)c2F)c(C(=O)NCc2cccn2C)[nH]c2ccccc12 56730,C(=O)(C(F)C(C)CNC(=O)CC1CC(NC)C1)N1CC(CSC)C1 56731,CC1CC(NC(C2COCCOC2)=O)CN(C(c2ccsc2)=O)C1 56732,N1(C(C2CCCCC2)=O)CC2(C=C(C(=O)N3CCOC4C(O)CC34)CO2)C1 56733,Cn1ccc(CNC(c2n[nH]cc2NC(=O)C(C)(C)c2ccccc2)=O)n1 56734,CCCC(C)(C)CC(=O)N1CC(CNC(=O)C(C)(C)c2ccccn2)C(F)(F)C1 56735,N1(C(C(C)=CCC)=O)C2CCC(C2)C1CC(N1CCOC2CC12)=O 56736,N1(C(=O)C(F)F)CCCC2C(CCCN2C(c2cc(F)c[nH]2)=O)C1 56737,C1(NNC(NCc2ccc(C(=O)OC)o2)=NCC2CC2)CC(OC)C12CCC2 56738,C(=O)(C#CC1(C)CCCO1)NC(C1CCCN1C(c1cnccc1Cl)=O)(C)C 56739,c1(C(N2CC=CC(NC(C3CC(OC)C3)=O)C2)=O)ccc(Cl)c(F)c1N 56740,c1(NC(C2N(C(c3ncc(C)nc3)=O)CCC2)=O)cccc(Cl)c1O 56741,C(CCN=c1[nH]cnc2c(F)cccc12)N(C(C(C)(O)C(F)(F)F)=O)Cc1cccs1 56742,Cc1snnc1C(=O)NCCC1CCC(NC(c2cnoc2-c2ccco2)=O)C1 56743,N1(C(c2n(CC)ncc2)=O)CC2(C(=O)NC(COC)C(C)C)CCC1CC2 56744,C1(NC(C(C)(CO)NC(C(CN(C)C)N(C)C)=O)=O)CN(C)CC1(F)F 56745,C(C(C)(F)C(C)C)NC(c1c(CNC(CCCCC)=O)cco1)=O.C=CCCS 56746,n1(CC=C)nc(-c2ccc(Cl)cn2)nc1C1CC(C)Cc2c[nH]nc21 56747,C1(CC(=O)NC(C)CC2CCC(O)(c3ccccc3)C2)CC(C)CC(C)(C)C1 56748,N1(C(c2sc(C)cc2C)C(=O)NCCC(=O)OCC)CCC(C#N)CC12CC2 56749,C1(CC(=O)N(C)CC2CCCN2C(=O)Cn2cc(Br)cn2)COCC(C)(C)O1 56750,c1(CNC(C2CC(=C)CN2C(=O)CCc2ccc[nH]2)=O)cc(CC)cc(Cl)c1 56751,C1(CNC(CCCOCCOCC)=O)CN(C(C2CCNC2=O)=O)CC1C 56752,c1(C(=O)NCCCOCCN(C)C(c2sccc2C2CC2)=O)nn[nH]c1Cl 56753,C=C(C)CCC(=O)N1CCC(NC(C2CC(C)=NO2)=O)C1CC 56754,C1(CNC(C2CCCC2)=O)COCCN(C(C2CCCOCC2)=O)C1 56755,Nc1cc(C(=O)NC2CC3(C2)CC(NC(c2ncncc2F)=O)C3)cc(F)c1O 56756,N1(C(c2c(C)n(C3CC3)nc2)=O)CCC(NC(=O)C2=COCCO2)CC1C1CC1 56757,C(=O)(C(F)CC(C)(C)NC(c1cccnc1)=O)N(C(C)CCO)C 56758,C(CNC(=O)CCn1c(C)csc1=O)(C(C)(C)C)NC(CCSCCC)=O 56759,C(c1cccc(F)c1F)=CC(N1CCC(NC(c2cc(=N)[nH]cc2)=O)(CO)C1)=O 56760,N1(C(c2ccn(CC)n2)=O)CCCN(C(=O)CN(C)S(=O)(=O)N(C)C)C(C)C1 56761,c1(CCC(N2CC(NC(C(CC)N(C)C)=O)C(F)C2)=O)cnc2ccccn12 56762,Cc1cc(Br)cnc1C(N1CCC(CN(C(=O)Cc2cccc(F)c2)C)CC1)=O 56763,C1(NC(CN2CCN(C)CC2)=O)CCSC12CN(C(c1n[nH]cc1Cl)=O)C2 56764,CC1Oc2ccc(C(=O)OCC(=O)N(C)Cc3ccccc3F)cc2NC1=O 56765,c1(C(N2CCC(O)(CNC(C3(C)CC=CCO3)=O)C2)=O)nnn2c1CCC2 56766,c1(C(=O)NCC2C(NC(COCC)=O)COC2)cc2ccccc2cc1OC 56767,C1(C(=O)NC(C2CN(C(c3c(CC)c(C)sc3)=O)C2)C)CCC(N=[N+]=[N-])C1 56768,N1(C(C2C(C)C2)=O)CC(CNC(=O)Cc2nc[nH]n2)C2(CCC2)C1 56769,c1(-c2nc(-c3c(C(=O)OC(C)(C)C)cc(Cl)cn3)on2)cc(Br)c(O)cc1O 56770,C(=O)(C1CCc2nccn21)NCC1(C)CCN(C(COCC(=O)NC)=O)CC1 56771,C(=O)(C1=NOC(CNC(=O)CCc2ccco2)C1)N1C(C#C)CCC1 56772,c1(C(=O)NC(C2CN(C(c3c(NC)cncc3)=O)C2)C)ccc2nc(O)cn2c1 56773,Nc1nonc1C(=O)NCC1(CC(N2CCC(F)C2)=O)CC1 56774,C1(CC#N)CCCN(c2ccnc(NCC3CC3c3cccnc3)n2)C1 56775,CCN(CC1CCN(Cc2ccccc2)CC1)N1CCCCC12CCS(=O)(=O)CC2 56776,N1(C(=O)OC)CC2C=CC1C(C(N1CC(C(=O)NCC3CCCCC3O)C1)=O)C2 56777,c1(CC(N2C(CN(C(C(F)=C(C)C)=O)C)COCC2)=O)c[nH]c2ccc(Cl)cc12 56778,Cc1cn(C)cc1C(N1C(C(N2CCOC(CN=[N+]=[N-])C2)=O)CCC1C(C)C)=O 56779,C(CCCCN)N(C=O)C.C12(CC(=O)NCC3(C(C)(C)OC)CC3)CCCC1C2 56780,c1(C(N2C(C=CC(=O)N(CC(C)(O)C3CC3)C)CCC2)=O)cccc2ccnn12 56781,c1(CCC(=O)NCCc2ccc(OCCC)cc2)ccc(Cl)cc1Cl 56782,N12CCCN(CC1C)C(=O)c1nc(C)c(s1)C2=O.C1(OCC)(COCC)CCC1 56783,c1(C(C)(CO)N(C(c2cn(C3CC3)nn2)=O)CC2CC2)c(F)cccc1F 56784,c1(C(=O)NC23CN(C(C(C=C)O)=O)C(C2)C3)ccc(C#N)cc1F 56785,C1(CC(=O)NC(C2CCN(C(c3ncoc3C3CC3)=O)C2)C)CC(=O)NC(=O)C1 56786,Cc1cc(C(=O)Nc2cnc(F)cc2C(=O)NC2CC(F)C2)nc2ccccc12 56787,N1(C(C2(NC(C)=O)CCC2)=O)CCC(CO)(CNC(C2CC(=O)N(O)C2)=O)CC1 56788,CS(=O)(=O)c1ccc(F)c(C(=O)NCC2(F)CC(NC(=O)C(F)F)C2)c1F 56789,c1(C(N(C2CCN(C(=O)C(O)CN3CCCC3)C2)CC)=O)ccc(=O)oc1 56790,C#CC1CC2(CC(C(N3CCN(C(=O)C(C)(C)NC(C)=O)CC3CO)=O)C2)C1 56791,CC(C)CC(C)(CNC(C1(Cl)CC1(C)C)=O)NC(c1cccc(C2(C)CC2)c1)=O 56792,Cc1cc(C(=O)NCCOC2CCN(C(=O)Cn3cccc3)C2)cc2ccsc12 56793,CCC(C(=O)N1CCC(C(=O)N(CC(C)(C)O)C2CC2)C1)C(C)(C)CC 56794,c1(OCC)cccc(C(N2CC(NC(C3CCC3(F)F)=O)CC2CO)=O)c1N 56795,C1(C(=O)NCCOCCC=C)CC2(CCC2)CN1C(=O)C(F)C1CCC1 56796,c1(C(=O)NC(C(C)NC(c2c(C)sc(C(F)(F)F)n2)=O)C)cc2n(n1)CCOC2 56797,N1(C(c2nn(C)cc2I)C(=O)NCCC)CCCCC1C1OCCO1 56798,N(C=CC(=O)C(F)(F)F)C(C1CCCCN1C(c1cc2ncsc2[nH]1)=O)=O 56799,CC(C)CC(C)CC(=O)N1CCN(C(=O)C2=CCCC2C)C2(CC2)C1 56800,C1(NC(C(CN(C(c2n(CC#C)cnn2)=O)C(C)C)O)=O)CCC2(CCC2)C1 56801,C#Cc1cccc(C(=O)NC2CC(CNC(c3cc(OC)n[nH]3)=O)C2(C)C)c1F 56802,c1(C2(C(=O)Nc3c(CC(=O)OCC)onc3)CC(N)C2)cccc(F)c1 56803,N1(C(C2CCC(C)C2)=O)CCOC2(CCN(C(c3cc(Cl)ccc3N)=O)C2)C1 56804,C1(CC(=O)NC2(C(N(CCOC)C)=O)CC2)CCC(C#N)C1 56805,c1(NC(C2CCN(CCNC(CCCCOCC)=O)CC2)=O)ccc(F)c(N)c1 56806,CCCC(C(=O)N1CCC(NC(c2cncs2)=O)C(O)C1)C(C)C 56807,N1(C(c2c(C)ncs2)=O)CCC2(CCCC2NC(c2cc(O)nc(O)c2)=O)CC1 56808,N1(C(CC)=O)C2CCC1CN(C(c1c(C3CC3)cccc1C1CC1)=O)C2 56809,c1(SCC(=O)NC2CCC2NC(C2CNC(=O)N2)=O)c(F)cccc1F 56810,c1(OCCC(=O)NC2(C)CCN(C(=O)CC3CC3)C2)ccc(F)cc1Cl 56811,c1(C(N2CCC(NC(CC3(OC)CCCC3)=O)C(C)C2)=O)csc2cccnc12 56812,C1(C(C)C#N)CCN(C(=O)C(C)N(C(c2ccccc2)=O)C2CC2)CC1 56813,CCC(CCOC)C(=O)N1CCCC(CC(=O)NCC2C=CCOC2)C1 56814,C1(F)(CNC(c2ccn(C)n2)=O)CCN(c2nc(Cl)ncc2C2CC2)CC1 56815,C1(C(NOCC(=O)NCc2cc(Cl)cs2)=O)CC2(C1)CC(O)C2 56816,N1(CC(N2C(CN(C(c3cncnc3C)=O)CC)CCC2)=O)CCn2nccc21 56817,c1(CCC(N2CC(C(C)NC(=O)C(O)c3ccco3)C2)=O)cccc(O)c1 56818,Cc1cc(=NCCc2ccc(C)c(F)c2)[nH]cc1S(=O)(=O)NC1CCS(=O)C1 56819,C1(c2n(C)cnn2)CCC(C(=O)NCC2CCN2C(CCC2=CCCC2)=O)CC1 56820,C1(NC(C2CC(F)CN2C(=O)Cn2cnnc2O)=O)CCn2ncnc2C1 56821,C#CCC(CC(F)F)C(=O)NC(CNC(c1nccnc1C(N)=O)=O)CC(C)C 56822,Cc1cccc(CC(C)N(C(=O)C(Cc2ccccc2)n2cnnn2)C)n1 56823,N1(C(C2(C)CCCCO2)=O)CCC2(CC1)CCN(c1ncc(Br)c(O)n1)CC2 56824,C(=O)(CC(C)(C)NC(C1COCCC1C)=O)NCC1(OCC)CC1 56825,c1(CC(=O)NC2CC(CC)(CC)N(C(=O)CN(C)C)C2)cnn2ccccc12 56826,Cc1nn(CCO)cc1C(=O)N(CC(C)N(C(=O)C(C(C)C)N(C)C)C)C 56827,Cc1ccnc(C(=O)NCC2CCC2NC(=O)C(F)C2CCCC2)c1N 56828,c1(C(=O)NCC2C(C)CCN2C(=O)CC2(C)CCCCC2)ccn2c1CSCC2 56829,Cc1cncc(C(=O)NCCN(C(=O)Cc2cnc(C3CC3)[nH]2)C2CC2)c1 56830,S(=O)(=O)(c1cccc2nsnc12)NC(C(C)C)C(N1CCC2C(O)CC2C1)=O 56831,N1(C(C(N2CCNC2=O)C)=O)CCN(C(=O)COCC2(F)CC2)C(C)C1 56832,CCCC(C(=O)NC1CC2C(NC(c3[nH]nnc3C(F)F)=O)C2C1)OC 56833,C=C1COCCN(C(=O)C(CN(C)Cc2ccccc2)NC(C2CC2Cl)=O)C1 56834,S(=O)(=O)(c1cc(C(F)(F)F)ccc1Cl)NC1CCN(C(c2cscn2)=O)CC1F 56835,N1(C(CC(C=C)C)=O)CCN(C)CC1CNC(c1ccn(CCF)n1)=O 56836,c1(OC)ccc(F)c(N)c1C(N1CCC(C(C)NC(C2C(C)(C)C2(C)C)=O)C1)=O 56837,N1(S(CCOCC)(=O)=O)CCC(O)C(C(=O)Nc2cnc(C(F)(F)F)c(F)c2)C1 56838,C(=O)(C(C)(C)CC(C)(C)C)NC(C)C(C)C(=O)N1CC(F)(CF)C1 56839,C(CCNC(C1(C(C)(C)O)CC1)=O)(C(=O)NC(c1ccncc1)C)OC 56840,CCCCCCC(F)C(=O)N1CCOC(C2CN(C(c3ccc(=O)n(C)n3)=O)C2)C1 56841,S(=O)(=O)(c1ccc(NCc2cccnc2)c(F)c1)N1CCC(OC)CC1(C)C 56842,CCCCCC(O)CNC(=O)CC(CNC(c1c[nH]nc1C(C)C)=O)C1CCC1 56843,C1(NC(C2C(OC)CN(C(=O)CC(=O)N(C)C)C2)=O)CN(C)C(C)(C)C1 56844,N1(C(=O)NCc2scc(CC)c2)CCC(O)C(CC(C)C)C1 56845,N1(C(c2ccccc2F)=O)CCC2CCCC12C(=O)NCC1C=CCC1 56846,C1(CC)CN(C(C2CCOC2CNC(c2cccnn2)=O)=O)CCCO1 56847,c1(C(N2C(CCOC)CN(C(=O)C(C)(O)C3CC3)CC2)=O)cc2ccccn2c1 56848,C1(C(=O)NCCN(CCCCCC)C(C)=O)(Cc2ccccc2)CCNC1=O 56849,C1(CC#C)(C(=O)N(CC(=O)N(CC(F)Cl)C)CC2CC2)CCOC1 56850,C1(c2c(C)n(C)nc2)C(C(=O)N(C)Cc2cnco2)CC(=O)N1C 56851,C(C)(C(CC(=O)NCC1CCCC1(C)C)NC(C1CCOC1)=O)OC 56852,c1(C2CCN(C(c3sccc3CC)C(=O)NCCOCC)C2)cccc(Br)c1 56853,C1(CN(CCCC)C(=O)NCCCC)CCCN(c2cc(O)ncn2)C1.CCCC 56854,c1(CCCC(N2CC(O)(CNC(CCCOCC)=O)C2)=O)cccc(C(F)F)c1 56855,C(=O)(C(CC)C(C)C)NC(C(=O)N(CCOCC#C)C)CCC1CC1 56856,C(=O)(C1=NOC(C)C1C)NCC(CNC(c1ccc(C(C)C)c(Cl)c1)=O)OC 56857,C1(CNC(CCCC(C)(C)C)=O)CN(C(=O)CCC2(C)N=N2)CCC12CCC2 56858,N1(C(C(=O)NCc2c(OC)cc(C#N)cc2)=O)C2CC3CC(C2)CC1C3 56859,N1(C(CSCCCC)=O)CCC(NC(=O)CSCC(=O)OC(C)(C)C)CC1C 56860,C(C(C)(CO)NC(c1sccc1NCC=C(C)C)=O)NC(C)=O.S(C)(=O)(=O)N 56861,C1(CNC(c2cn(CC)nn2)=O)CN(C(C2CCCCNC2=O)=O)C2(CCC2)C1 56862,c1(CCC(=O)NCC(CC)(C)NC(=O)C(C)CF)ccc(Cl)c(C)c1 56863,N1(C(C(C)=CC2CC2)=O)CCC(NC(c2ccnn2C2CCC2)=O)C(CO)C1 56864,C12(CNC(c3cc(COC)no3)=O)CCCC1N(C(C1(CCF)CC1)=O)CCC2 56865,C(CC1=CCN(C2CCNC2=O)CC1)NC(CCC(C)OC)=O 56866,c1(OC)cc(C(=O)NCCc2ncc[nH]2)ncc1-c1ccc(C)nc1C 56867,C(=O)(CC(O)CC(C)C)N1CC(O)CC(NC(C=CCC)=O)C1 56868,c1(NC(C2CCCCN2C(=O)C=Cc2cncs2)=O)cncc([N+](=O)[O-])c1 56869,C(=O)(C1CCCc2c1ncn2C)NC1CC(C)(NC(CC=C(C)C)=O)C1 56870,c1(C(=O)NCC(CNC(C2CC2C(C)(F)F)=O)OC)cnc[nH]c1=N 56871,N1(C(c2n(C)nc([N+](=O)[O-])c2)=O)CCC2(CC1)CC(CNC(c1cocn1)=O)C2 56872,CCCCC(C(=O)NCCOCCOCC)N(C)C.c1(=O)c(=O)[nH]1 56873,N1(C(C=CC)=O)CCC2(CC1)CC(CNC(C1CC(=O)N(CCC)C1)=O)C2 56874,c1(C(N(CC(CC)NC(=O)Cc2n[nH]c(C)n2)C)=O)cc(C2CCOCC2)on1 56875,N1(C(c2cc(CC)[nH]n2)=O)CCC(C)(C)C(C(=O)NC(C)Cc2cc(C)[nH]n2)C1 56876,C(=O)(C1=CC(O)CCC1)NC(C)C(C)(C)NC(C1SCCCS1)=O 56877,C1(C(=O)NCC2(C#N)CC2)CC2C=CC1N(C(C1CCCC(=O)C1)=O)C2 56878,C1(N(C(CCC(=O)NC)=O)C)CCCN(C(c2ccc(O)nn2)=O)CC1 56879,c1(C(=O)NCC2C(NC(C(C)n3cnnn3)=O)C2)coc2cccc(O)c12 56880,Cc1c(CN2CC(C)CC2c2ccccc2F)cccc1F 56881,N(C1CCc2cc(Cl)ccc21)c1ccnc(NCC2CCN(C(=O)OC)C2)n1 56882,N12CCC(c3ccccc3)(C1)C(=O)C2.N=c1sccn1CC1CC2CC2C1 56883,CCCC(C)(CCC)C(=O)NCC(O)CNC(C1CSCN1C(C)=O)=O 56884,N12CC(CC(F)(F)C1)C2=O.N1(C(c2cc(C(C)=O)[nH]n2)=O)CCCC(N(C)C)CC1 56885,c1(C(N2CCCC(CC(N3C(CC(C)C)CC3)=O)C2)=O)ccc([N+](=O)[O-])o1 56886,c1(OC)ccc(Cn2cc(C(C)N(C)C(C3CC3(Cl)Cl)=O)nn2)cc1.C1C(=O)O1 56887,CC1CC(C(=O)NCC(C2CCN(C(=O)CC3CC3(Cl)Cl)CC2)O)=NO1 56888,Cc1c(CC(=O)NCC2(CNC(C3CC3C(N)=O)=O)CC2)cnn1C 56889,c1(C(=O)NCC2CC(NC(C(CCC)C#N)=O)C2)[nH]c2cc(Cl)ccc2c1C 56890,CCCC(C(O)C(=O)N1CCC(O)(CO)C1)NC(c1cc(C)c(CC)o1)=O 56891,C(=O)(C(C(C)CC1CCCCC1)N(CC(=O)OCC)C)NCC(=C)C 56892,c1(C(=O)NC(C)C(=O)NCC2CC3(CCCO3)C2)cc(F)cnc1O 56893,S(=O)(=O)(C(F)(F)F)N1CC(NC(=O)CCc2cnc[nH]2)C1 56894,N1(C(CC(C)(C)O)=O)CC(NC(c2csc(Cl)c2)=O)CC(O)C1 56895,C(C(N=c1[nH]c2c(F)cc(Cl)cc2s1)C1CC1)NC(c1c(C)[nH]nc1C(C)C)=O 56896,N(C(=NCCC1COC(C)(C)O1)NCC1CCC1)CC(=O)Nc1ccc(OC)cc1 56897,CC1CCCN(C(c2cnccn2)=O)C1CNC(=O)C(=O)Nc1ncc[nH]1 56898,N1(C(C2(S(N)(=O)=O)CC2)=O)CC(NC(=O)Cn2cc([N+](=O)[O-])cn2)C(C2CC2)C1 56899,N#Cc1ccc([N+](=O)[O-])c(SCC(=O)Nc2cncs2)c1 56900,C(=O)(CC(C)(F)F)NC(CN(C(=O)Cc1ccnc(C(F)(F)F)c1)CC)C 56901,C=CCCC(F)(F)C(=O)N1CC2CC(NC(=O)C(C(C)(C)C)OC)C1C2 56902,C(=O)(CCC(C)(C)C#N)NCc1ccc(OC)cc1.C12CC(C13CCC3)C(=O)N2 56903,C(C(C)C)(C(O)C(=O)N1CC2(CC2)CC1CC(=O)NC1CN2CCCC1C2)OC 56904,Fc1ccc(Cl)c(F)c1CNCc1cc(I)c(Cl)cc1F 56905,c1(OC)ccsc1C(=O)NCC(F)CNC(c1ccn(CC(F)(F)F)n1)=O 56906,C(=O)(CC(C)(C)C)NCC1(CC(=O)N(C)CCc2cnccn2)CC1 56907,c1(OC)cccc2c1CN(C(C1C3CC(CC3F)N1Cc1ccc(C)s1)=O)C2 56908,C1(OC)CN(C(=O)C(O)CSC)CC1C(=O)N(C1CC(N(C)C)C1)C 56909,c1(OC)ccc(C(=O)NCC(CNC(C2(C)SCCCS2)=O)CO)cc1N 56910,Cc1c(C(N2CCOCC2CCNC(=O)CC(C)N(C)C)=O)cccc1Cl 56911,c1(C(C)(C)C)nsc(OC)n1.c1(CC=O)csc(C2CC2)n1 56912,C1(C(=O)NCC)CCCN(S(=O)(=O)CC)C1.C1(=O)C(=O)N(CC)CCCN1 56913,N1(C(COCCOC)=O)CC2=C(C1)CN(C(c1cc3ccccn3c1)=O)C2 56914,C(=O)(C(CCCOC)NC(=O)CC(O)C1CC1)NC1(CC)CC1 56915,C1(COC)(CNC(c2coc(C(C(=O)NC)N(C)CCC3CC3)c2)=O)CC=CC1 56916,C1(NC(C2(NC(CC(C)O)=O)CC(O)C2)=O)CCN(C)C1=O 56917,Cc1c(C(=O)NCC(C)CNC(=O)COCC2CCOC2)ccc(F)c1F 56918,CC(C)C(F)(CNC(=O)CCc1ccncn1)C(=O)NC1C(O)C2CCOC12 56919,C=CC1(C(=O)NC(C)CN(C(C2C=C(C)CS2)=O)CC)CCOCC1 56920,c1(NC(C2CCN(C(C3CCN(C)C3)=O)C2)=O)ccc2c(c1)CCN(C)C2 56921,N1(C(C2C(C(=O)OC)C2)=O)CC(CNC(=O)CC(C)(C)SC)OC(C)(C)C1 56922,C1(CC)C(C(=O)NC2(CF)CN(C(c3cnc(C)nc3)=O)C2)CCN1C 56923,N1(C(C2N(C(CCC)=O)CCCC2)=O)CC2(NC(C3CCC3C)=O)CCC1CC2 56924,c1(C(=O)NCCCC(C)NC(C2C3CCCC23)=O)cc2c[nH]cnc-2n1 56925,CCC(CC)(C(=O)NC1CN(C(=O)Cc2ccccc2OC)CCC1C)OC 56926,N#Cc1cc(Cl)cnc1N1CCCC(C(N2CCCC2c2ccncc2)=O)C1 56927,C1(NC(C(n2c(C)ncc2)C)=O)CN(C(c2scnc2C(C)C)=O)CCC1F 56928,Cc1cc(CNC(c2cnn(CCNC(=O)C(O)C(C)(C)C)c2)=O)cnc1F 56929,N1(C(c2c(Cl)cc(C)s2)=O)CC(C)CCC1CNC(c1ccc(F)s1)=O 56930,CCC(C)CC(=O)NCC(O)CNC(C12CC(CC(=O)OC(C)(C)C)(C1)C2)=O 56931,C(CSC(C)(C)C)(C(=O)N1CC(CNC(c2csc(C)c2)=O)C1)NC(C)=O 56932,c1(COC)nc(C(=O)NCC(C2CCCCC2)NC(=O)COCC2CC2)cs1 56933,C=CCC(C)C(=O)NC1CCN(C(c2cn(-c3ccc(C)cc3)nn2)=O)CC1 56934,C(=O)(C(C)CCCC(C)=O)N1C(CC(N2CCC(CC#C)CC2)=O)CC(C)(C)C1 56935,c1(NC(C2CC(NCc3ccc(C)cc3Br)C2)=O)ccc(C#N)c(Cl)c1 56936,N1(C(c2nc(C(C)C)sc2)=O)CC(NC(=O)C2=CCSC2)C2(CCC2)C1 56937,C1(NC(c2cc(CNC(CC(C)C)=O)[nH]n2)=O)CCCC1(C)C 56938,N1(C(CC(=O)c2ccncc2)=O)CCC(F)(C(=O)NOCCCO)C1 56939,C(CC)(CC)(CCNC(c1cccc(Cl)c1F)=O)NC(C(CC)n1ccnc1)=O 56940,N1(C(CC(=O)NCC#C)=O)CCC(C)(C)C1C(N1CCC1(C)CCO)=O 56941,c1(NC(C(C(C)C)NC(C=CC)=O)=O)cnc(Cl)nc1C 56942,C1(OC)CN(C(=O)CC2CCOCC2)C(C)(CO)C1.c1(C=O)cc(C(N)=O)[nH]n1 56943,C(C(C1CCCCC1)NC(=O)CCF)(C(C)C)NC(c1ccc(SC)s1)=O 56944,C=CCC(C)(CC)C(=O)NC1CN(C(C2(O)CCOCC2)=O)CC2(CC2)C1 56945,N#Cc1ccc(CCNCc2nnco2)cc1 56946,c1(NCC(c2ncc[nH]2)C)[nH]c(=NCC2CC(C(F)(F)F)C2)nc2c1ncn2C 56947,n1(CC)cc(C(=O)NCC23CC(CN2C(=O)CSC)C3)c(C(C)C)n1 56948,c1(COCC(=O)NCC)cn(CCCNC(c2cnn(C(F)F)c2)=O)nn1 56949,c1(CC)[nH]ccc1C(=O)NC(CC1CC1)C(=O)NCC1CC1(F)F 56950,c1(C(=O)NCc2cc(NC(C(=CC3CCCC3)C)=O)no2)ncnc2sccc12 56951,c1(C(=O)NC2C(OC)CN(C(=O)C(CO)N(C)C)C2)cc2cc(Cl)ccc2n1C 56952,n1(CCC#C)cc(C=CC(=O)OCC)cn1.C1(C)CO1 56953,c1(COC)ccc(NC(C2CN(C(=O)CCc3ccc(F)nc3)CCS2)=O)cc1 56954,c12cnc(c(Cl)c1)N1CCCC1NC2=O.c1(NC(C)=O)ncncc1Cl 56955,N1(C(CCCOCC)=O)CCCC(CN(C(=O)C(n2cc(Cl)cn2)C)C)C1 56956,N1(C(CC(C)C)=O)CCCC(C2CN(C(C3CCc4n[nH]cc4C3)=O)C2)C1 56957,c1(N2C(C3CCN(C(c4ccns4)=O)C3)CCC2)nc(Cl)nc2[nH]ccc12 56958,C1(CCC)C(=O)NCCN1C(=O)NCCc1ccncn1 56959,C1(CCOC)(NC(=O)CC(C)(C)C2CC2)CCN(C(c2conc2C(C)C)=O)C1 56960,N(C(=NCc1coc(C)n1)N1CCC(Cc2ccccc2)C1)C(C=C)C 56961,Cc1cc(N2CCN(C(=O)C=CC(C)(C)C)C(C)C2)nc(-c2cccnc2)n1 56962,C12(C(=O)N(CC)Cc3cccnc3)CC(CNC(C=CC=CCC)=O)(C1)C2 56963,C1(CNC(c2nnnn2C2CCC2)C2C(c3ccoc3)C2)CC2(CCC2O)C1 56964,N1(C(N)=O)CCC(CNC(=O)Nc2cccc(SC3CC3)c2)CC1 56965,c1(C(=O)NC(CN(C(COCCC=C)=O)C)(C)C)cc2ccccc2nc1O 56966,Cc1cc(C(=O)NCC2CC(F)(CNC(C3(C)CC3(F)Cl)=O)C2)ccn1 56967,c1(OC)ccc(C(=O)C(N2CC3CC3C2C(=O)NOCC(O)CO)=O)cc1Cl 56968,c1(C(C)C)ccc(C(N2CC(NC(=O)CC3CCS(=O)(=O)C3)C(O)C2)=O)c(Cl)n1 56969,CC1COCCN1CCNC(C1CC12CC(NC(=O)Cc1ccc(O)cc1)C2)=O 56970,CP(C)(=O)C(O)C(=O)N1CCC(CCCCNC(C2CCC(=O)O2)=O)CC1 56971,NS(=O)(=O)CCCC(=O)N1CCN(C(=O)CCCN2CCCCC2)C2CC12 56972,c1(OCC)cc(Cn2nccc2NC(c2ccc(C)cc2Cl)=O)ccc1OC 56973,c1(C(N2CCN(Cc3ncc(Cl)cc3O)C3CC23)=O)c(F)cccc1Cl 56974,N1(C(C2(C3CC3)CN(C(C(C3CC3)SC)=O)C2)=O)CC(C2=NOCC2)C1 56975,CC12CCCC1N(C(C1C3CCN(C(C4CC5CC4CC5O)=O)CC13)=O)CCC2 56976,c1(OC)c(C(=O)NC23COC(COC(C)C)(C2)C3)nc(O)nc1O 56977,C1(=CC(=O)NC2CCC(CNC(Cc3ccn(CC)n3)=O)C2)CN2CCC1CC2 56978,C1(C(N2C(C3CCN(C(c4ccc[n+]([O-])c4)=O)C3)CCC2)=O)OC2CCC1CC2 56979,C(=O)(C(F)(F)C(F)F)N1CCC(CNC(c2ccsc2)=O)CC1 56980,c1(C(=O)NC(CC)CNC(=O)C(C)N(CC)CC)cc(F)ccc1C(F)(F)F 56981,C#CCC(CCCO)NC(C1CCCC1NC(C1CC2(C1)CC21CC1)=O)=O 56982,c1(CC(=O)NCCCN(C(C2C(SC)CCC2)=O)C)ncn2c1COCC2 56983,c1(SCC(=O)NC2CCN(C(C3CCCC3O)=O)C2)n[nH]c(O)n1 56984,C(=O)(CCC(=O)NC1C2CC1N(C(=O)C(C1CCCCCC1)C)C2)NCCC 56985,C1(CC(=O)NCCN(C(CCOCC)=O)CC)CC(C)CC(C)(C)C1 56986,c1(NC(N2CCC(CC3CCC3)C2)=O)ccc(C(F)(F)F)cc1O 56987,CCCC(CC(C)C)C(=O)NC1CCC(CNC(=O)C(F)(F)c2cncs2)C1 56988,c1(C(=O)NC2(CNC(C(CC)C)=O)CCCCC2)ccc(F)cc1C 56989,CN1CCN(C(=O)CCCc2nncn2C)C(CNC(c2ncc(Cl)s2)=O)C1 56990,C=CCC(CNC(=O)CCC(=O)NC(C)CC)C(=O)NC(C)C 56991,c1(C(=O)NCC(CC)NC(=O)C(c2cccnc2)O)nn(C)c(Cl)c1Br 56992,N1(C(C2CCN(C)S2(=O)=O)=O)C2CCC1CN(C(C1CC(CCO)C1)=O)C2 56993,Cn1cc(Cl)c(C(N2CCC(Oc3cnccc3CNC(=O)C(C)(F)F)C2)=O)n1 56994,N1(C(C23CC(C)C2C3)=O)CC2CC2(CNC(c2cc(C(F)(F)F)ncn2)=O)C1 56995,CC(C)C1=NOC(C(=O)N(C)CCOCCNC(=O)Cn2cc(Br)cn2)C1 56996,Cc1cc(C(=O)NC(Cc2cn(-c3cccc(=O)o3)nn2)CC(=O)O)c(C)s1 56997,CC1CCC=C1C(=O)NCCn1ccc(C(=O)N(C)CC2CC(F)(F)C2)c1 56998,c1(CNC(C2C(C(C)C)CCO2)=O)cnn(C)c1C(=O)NC(C(C)C)C1CC1 56999,C1(C(N2CC(F)(C(=O)NC3(C(N(OC)C)=O)CC3)C2)=O)CC12CCOC2 57000,N1(C(c2ncnc(C)c2C)=O)CC2CCCC1C2CNC(c1ccc(F)cn1)=O 57001,c1(-c2nc(COC)nn2-c2c(C(F)F)cc(Br)cc2C)noc2c1CC(C)CC2 57002,CC1(C)CCC(C(N2CCCC(CC(=O)Nc3cccc(CO)c3)C2)=O)C1 57003,C(=O)(CCCCCCCBr)NC1C(C(=O)Nc2c(C(=O)OC)cccn2)CCC1 57004,C(C)(C)(C(C)CC(=O)N1CC(C)CC(O)C1)NC(C(C)OCCN(C)C)=O 57005,C1(CNC(=NCCC)NCCC2CCOCC2)CCC2(CCCC2)O1 57006,CC(O)CCCNC(=O)CC1CCCC1NC(=O)Cc1ccsn1 57007,c1(C(N2C(CNC(Cc3c(C)con3)=O)CC2)=O)cn(C)c(=O)cc1Cl 57008,N1(C(C(CC)SC)=O)CCCC2(CCN(C(C)C(=O)N(C)C)C2)C1 57009,c1(C2CCN(C(C(N)Cc3cncs3)=O)C2)cccc(OCO)n1 57010,c1(C(=O)NC(CNC(CSCC(=O)OC)=O)CO)ccc2c(c1)CCCS2 57011,C(=O)(C(O)CC(C)C)N1CCCC(CN(C(C2CN(c3nncs3)C2)=O)CC)C1 57012,c1(N2CCN(CC3(C(=O)OC)CCCO3)CC2)ccc(F)c(OC)c1 57013,C1(c2cn(Cc3c(CC)ccs3)nn2)C(C)CCN1C(=O)C(C)N1CCC1 57014,c1(C(=O)NC(C2CCOC2)CNC(C2(CC)CC2)=O)ccnc2ccc(F)nc12 57015,N(C1CN(C(C2CC=CCO2)=O)Cc2ccccc21)C(CCS(=O)(=O)NC)=O 57016,c1(C(N(C2CCN(C(=O)CC3(c4ccon4)CC3)C2)C)=O)ccc2occc2n1 57017,C1(CC(=O)NC(C2(C(=O)NCC(C)Cn3ccnc3)CC2)C)CCCCO1 57018,Cc1cc(-c2cc(C)ccc2OC(F)(F)F)ccc1CC1CCCCNC1 57019,CC1CCN(C(c2n[nH]c3c2COC3)=O)CCN1C(=O)C(C1CCOCC1)F 57020,C(=O)(C(C)C(C)CC(=O)O)N1CC(C(F)(F)C(=O)O)(OC)C1.c1(CO)cn(C2CC2)nn1 57021,C(=O)(C(O)C(C)(C)CC)N(CCNC(C1N(CCC)CCC1)=O)C(C)C 57022,C1(CC=C)N(c2ncnc(NCCC(O)C(C)C)c2C)CCCC1(C)C 57023,Cn1ncc2nc(Cl)nc(N3CCC(C)(CNC(=O)CCF)CC3)c12 57024,C1(NC(C2C(CNC(C3(CCC)CCC3)=O)CCC2)=O)CCC(O)C(O)C1 57025,C(=O)(C(C)C(C)(C)C)N1CCC(C2N(C(C(C)SC)=O)CCCC2)C1 57026,c1(C(=O)NCC2CC(NC(C3C(C)C3)=O)C(O)C2)cc([N+](=O)[O-])c(F)cc1N 57027,CC1CCN(C(=O)C(F)CC2CCC2)CCN1C(c1cnc2n1CCOC2)=O 57028,c1(C(N(CCC(C)NC(C2(CO)CCOC2)=O)C)=O)cc(Cl)ccc1N 57029,C(=O)(C#CC1CCCCC1)N1C2CN(C(c3c(NC)cnnc3)=O)C(C2)C1 57030,C1(NC(C2(CNC(C3CCCCC3O)=O)CC(=C)C2)=O)CCC2CCCC1O2 57031,N1(C(C2CCC(NC(C3CCC(C)(CC)O3)=O)C2)=O)CC2CCCCC12C 57032,c1(-c2c(C(=O)NC(C(C)NC(CCCC)=O)C)c[nH]n2)ccc(Cl)cc1 57033,N1(C(C2(CC)CCC2)=O)CCC2(CCOC2)C(CNC(=O)CCC2(O)CCC2)C1 57034,C(=O)(CCCCCn1cc(CN2CCCC2CO)nn1)NCCCC(=C)C 57035,CCC(CC(=O)N1CCCC1CNC(=O)C=C1CCC1)SC 57036,C#CCC(CO)NC(c1n[nH]cc1CNC(c1c[nH]cc1CC)=O)=O 57037,C1(CC)CCCN1C(=O)CNC(=O)Cn1cc(NC(=O)Cc2cnsc2)nn1 57038,N1(C(C(CC)OCC)=O)CCC(NC(C2(C)CCCS2(=O)=O)=O)C(F)C1 57039,C1(C(=O)NCC2(SCC)CC2)CNC(=O)CN1C(=O)C=CC1CCCN1C 57040,C(=O)(CS(=O)(=O)CC(=O)N1CCN(C(=O)C(C)N(C)C)CC1CF)OC 57041,C(=O)(C(C#N)C(C)C)NCc1c(C(=O)NC(CC)C(=O)OC)n(C)nc1 57042,C1(CNC(=O)COC2CCC2)CC2(CO1)CN(C(C1CCC(=O)O1)=O)C2 57043,c1(CN(CC(=O)N(C)CC2CCN(C(CCSC)=O)C2)C)ccc(Cl)cc1 57044,CN=c1[nH]cc(C(N2CC(O)CC2C(=O)NCC2C=CCOC2)=O)o1 57045,C1(NC(C2CCC(CCC)CC2)=O)CN(C(=O)C(C)(C)O)CCC1(F)F 57046,C1(C(=O)NC2CN(C(c3ccn(C)c3)=O)CC23CC3)CCC2(CC1)CNC(=O)C2 57047,C(=O)(CC(C)C(=O)N1CCC(CNC(c2cnc(S)n2C2CC2)=O)CC1C)OC 57048,C1OCCCC1(C)C.C1(C2CC2)C(=O)N1.C12(CC1)CC(=O)N2.CN(C)C 57049,N1(C(C)=O)CCCC1CC(N1CCCC1C(C)NC(=O)CN(C)CCO)=O 57050,Cc1ccc(S(=O)(=O)N2CC(NC(c3c(C(F)(F)F)cccc3F)=O)C2)cc1C 57051,CCC(O)C(C)(C)C(=O)NCCCN(C)C(c1csc(-c2ccc(Cl)cc2)c1)=O 57052,C(=O)(C(C)(CO)NC(C1CC(C#N)(OC)C1)=O)NCc1n(CC)ncn1 57053,Cc1nc(C2CCCO2)sc1C(=O)NC1COCC1NC(c1ccccc1O)=O 57054,N1(C(=O)NCC=C)CCN(C(=O)Nc2ccc(C(=O)OC(C)C)cc2)CC1CC 57055,c1(NC(=O)CC2CNC(=O)O2)cc(Cl)ccc1OC(F)(F)F 57056,C12CCC(CC1)C(=O)N2.N1(C(C#C)=O)CCC(C(C(=O)NC)NC=O)C1 57057,C1(O)(CNC(C=C(C)C(F)F)=O)CC2CCC(C1)N2C(c1cnc(S)nc1)=O 57058,N1(c2ccnc(NCc3ccc(F)c(C)c3F)n2)CCCC2(CC1)CNC(=O)C2 57059,N#Cc1cc(S(=O)(=O)N2Cc3c[nH]c(=N)nc3C2)ccc1NCCC1CCCO1 57060,C1(C)(NC(C(C)C2CCCO2)=O)CCN(C(c2cc(N)cc(O)n2)=O)CC1 57061,C1(N(C(c2cn(-c3ccc(OC)cc3)nn2)=O)C)CN(C(=O)CCF)CC12CC2 57062,CC1OCCN(C(C2CC(=O)CN2C(=O)CCc2ccoc2)=O)C1C 57063,N1(C(C(C)OC2CCOC2)=O)CC2CC1CN2C(C1CC(C)(C)CN1C)=O 57064,C1(CC(=O)NCC(CC=C)NC(c2sccc2C)=O)CCCC(C)(C)CC1 57065,C1(NC(c2ccc3c(c2)OCC3)=O)CCC2(CC1)CC2NC(C1CC1(Cl)Cl)=O 57066,Cc1cccc(C)c1CC(N1CCC(CO)C(NC(c2[nH]c(O)nc2C)=O)C1)=O 57067,N1(C(C(C(CC)C)O)=O)CCN(C(=O)CCCNCc2cccs2)C2(CCC2)C1 57068,N1(C(Cc2c(C)n[nH]c2)=O)CCC(C)C(CNC(c2cc[n+]([O-])cc2)=O)C1 57069,N1(C(C(C)C#N)=O)CCOCC1CC(=O)N(C)CC1(O)CN(C)C1 57070,C1(NC(CCCC)=O)CCCN(C(=O)C=CCOCC(F)(F)F)C1 57071,C1(C)(CCCC(C2CCN(Cc3c(C)cncn3)CC2)=O)NC(=O)NC1=O 57072,C12(CNC(C(C)(C)F)=O)CN(C(c3ccc(OC(F)F)cc3F)=O)CC1CCO2 57073,c1cc2c(NCCCC3CCOCC3)[nH]c(=NCCC(O)C3CCCC3)sc-2n1 57074,n1(CC(=O)NC2CCCN(C(C3N(CC)CCC3)=O)C2C)ncc2cccnc12 57075,C(c1ccc(C2CC2)cc1)=CC(N1CCNCC1C1CCCC1)=O 57076,N1(CC(=O)NC(C(=O)OC)C2CCC2)CCN(c2cc(Cl)ncn2)CC1 57077,N1(C(CC(C)(C)O)=O)CCC2(CCCC2NC(c2[nH]nc3ncccc23)=O)C1 57078,CCCC(CN=c1ccc(Br)c(S(=O)(=O)NC(c2nccnc2C)C)[nH]1)OC 57079,c12ncc(cn1)[nH]c2=O.C1(CC)(NC(=O)COC(C)C)CC(F)(F)C1 57080,CC(C)C(CNC(=O)CCC1CCCCO1)NC(=O)CCCN(C)C 57081,C1(C(CC)O)CCCN1C(=O)C=CCNC(=O)CC1(COC)CC1 57082,c1(OC)cccnc1-c1cn(C2(C(=O)NC(C)CC3CCOC3)CCC2)nn1 57083,N1(C(CSS(C)(=O)=O)=O)CCCN(C(=O)C2CC2)CCC1.C12CC(C1)C(=O)NC2=O 57084,O=C1CCOC(C(N2CCCC2c2cn(CC3COCCO3)nn2)=O)C1 57085,C1(NC(=O)OC)CCCN(CCC(=O)CCOc2ccc(C(C)(C)C)cc2)C1 57086,C1(CCC)CN(C(=O)C(C#N)CC)CCN1C(c1ccnc(O)c1)=O 57087,N1(C(C2(CCC=C)CN(C(=O)C(O)C(C)C)C2)=O)CC(C)(C)C1COC 57088,N1(C(C=C(C)C)=O)CCN2CCN(C(=O)CCc3ccccn3)CC2C1 57089,CC1(CNC(=O)CCC2CNC(=O)N2)CCCN1C(c1cc[nH]n1)=O 57090,c1(C(=O)NCC2N(C(C(COC)C)=O)CC2)nc(-n2cccc2)sc1C(C)C 57091,CC(C)C#CC(=O)NCCCCNC(=O)CC(C)NC(C1CCCC1)=O 57092,C1(NC(C2(C)CCC(=O)C2)=O)C2CC3C1C3C2C(N1CCOC(C2CCC2)C1)=O 57093,C1(C(N2CC(NC(c3cn(CC)nc3)=O)C3C(C2)C3)=O)CN2CCCN1CC2 57094,c1(N2CCCC(C(C)NC(=O)CCCNC(N)=O)C2)ccc(C#N)cc1[N+](=O)[O-] 57095,Cc1ncc(Br)c(N2CCC(C(N3CC(O)C(O)C3)=O)C2)n1 57096,C(=O)(CCCCC(=O)NC)N1CC2C(NC(c3cccc(SCCC)c3)=O)(C2)C1 57097,Cc1nscc1C(N1CC=CC1CNC(c1cc(C(C)(C)C)n[nH]1)=O)=O 57098,C1(NC(Cc2c(C)non2)=O)CN(C(c2csc(C)n2)=O)CC1C(F)(F)F 57099,c1(COC(CNC2C(C)CCC2)=O)cccc(COCC(=O)O)c1 57100,C1(C(=O)NC2C(C(=O)OC)CCC2)CCCCN1C(=O)Cc1ccoc1 57101,C(=O)(CC(C)CC(=O)N1CC(=O)CC1C(N1CCOC(C2(C)CC2)C1)=O)OC 57102,C1(C(=O)NCCC(COC)(C)C)CCC(C)(C)N(C(=O)Cc2ccsn2)C1 57103,c1(C(N(c2cc(C)cc(F)c2)C2CCNCC23CC3)=O)cnc2ccccc2c1 57104,C1(CC)(NC(=O)CCC2CCCO2)CCCN(C(c2ncc(OC)cc2F)=O)C1 57105,CC1=C(C(=O)N(C2CN(C(C3CCCC3CN(C)C)=O)C2)C)S(=O)(=O)CCO1 57106,Cc1nnc(O)c(C(=O)NCC(O)CN(C(=O)Cc2cn3ccsc3n2)C)c1C 57107,CC1(C)CC(CNC(C2CCN(C3CCCCC3)C2)=O)N(C(=O)CO)C1 57108,c1(CCC(N2CCC(N(C(CC)=O)C)C2)=O)c[nH]c2c(C)cccc12 57109,CC1CCN(C(c2cccc(SC(F)F)c2)=O)CCN1C(C1CCCC(=O)N1)=O 57110,c1(CCC(=O)NC(CNC(c2c(CC)cc[nH]2)=O)(C)C)c(F)cccc1F 57111,C(=O)(CC(C)(C)C#N)NCC1C(C(=O)NC2CCN(CC)CC2)C1 57112,N1(C(c2nc(OC)c(C)s2)C(=O)NC)CCC(C)C(C)(C)C1 57113,CC(c1ccccc1F)=CC(=O)NC1CC(NC(C2(F)CCCC2)=O)C12CCC2 57114,N1(C(=O)Cn2cccnc2=O)CCC2C(CCCN2C(=O)C=CC2CC2)C1 57115,c1(C(N2C(CNC(C(C)SCCCC)=O)CC2)=O)ccccc1[N+](=O)[O-] 57116,CC(C)C(C(C)NC(=O)CCn1cnccc1=O)NC(=O)Cc1cnoc1 57117,CN1CCN(C(C2(C#N)CCSCC2)=O)CC1CNC(=O)Cc1cncs1 57118,CC1(C)CCC(O)(CNC(c2ccc(CNC(=O)CC3CCCSC3)nc2)=O)C1 57119,C(=O)(C(C)(C)C(=O)NCC(C)(O)CNC(C1CC2CC2C1)=O)NC 57120,c1(N(C2CC(N)C2)C(c2ccc(C)cc2Cl)=O)ncc2ccsc2n1 57121,N1(C(C(C)NC(=O)OC)=O)CC2C(CN(C(=O)CN3CC4CC4C3)C)C2C1 57122,c1(C(N2C3(CCC(C(=O)NCC)C2)COC3)=O)[nH]c2cc(OC)ccc2c1C 57123,c1(C(=O)NC(C2CCCN2C(=O)CN(C2CCSC2)C)C)nnnn1C(C)(C)C 57124,Cc1[nH]c2ccccc2c1C(=O)NC(C)CN(C(=O)CC1CC(F)C1)C 57125,C1(C)(C(=O)NCC(CNC(c2ccc(CC)nc2)=O)O)CC(C(C)C)=NO1 57126,C(=O)(C1CCCn2cncc21)Nc1c(OC)cccc1 57127,Cc1ccc(C(=O)NC2CCN(Cc3nc(O)n[nH]3)C(C)C2)cc1CO 57128,N1(C(CS(=O)(=O)NC)=O)CC2(CCN(C(C34CCN(CC3)CC4)=O)CC2)CC1C 57129,Cc1cc2[nH]c(C(N3CCCC(NC(c4cc(F)n(C)n4)=O)C3C)=O)cc2o1 57130,c1(CS(CCN(c2ccc(C(=O)OC)nc2)C)=O)c(SC)nc2ccccc2c1C 57131,C(CCCCNC(=O)Cc1cncnc1)NC(c1cnn(C(F)F)c1)=O 57132,C1(C)(C(C)NC(c2ccccc2)C(c2ccccc2)O)CC2(CC2)C1 57133,c1(C(=O)NC2CCC(NC(Cc3cc(C)ns3)=O)C2)ccc(-n2cncn2)cc1 57134,CCCC(CC)CC(=O)NCCCN(C(C12CCC(N=[N+]=[N-])C1C2)=O)C1CC1 57135,c1(CNC(C(CCC)(C)CC)=O)cccc2c1CN(C(=O)C(C)OC(C)(C)C)C2 57136,c1(CCCC(=O)NCCN(C(C2C(C=C)C2)=O)C)ccccc1Br 57137,Cc1nn(C)c(Br)c1C(=O)Nc1cccc(NC(C23CC(F)C2C3)=O)c1 57138,C(=O)(CCCC(C)(C)CC)N1CC2C(CNC(c3ccc(C=C)cc3)=O)C2C1 57139,C1(NC(C2C(C)(C)C2)=O)C2CC1CN(C(C1CCN(c3nccs3)CC1)=O)C2 57140,c1(C(=O)NC(C2OCCN(C(c3[nH]cc(CC)c3)=O)C2)C)nccc(Cl)c1Cl 57141,c1(CC)cc(C(=O)N(CC(O)CN(C(=O)CN2CC(=O)NC2=O)C)C)ccc1C 57142,C1(CNC(C2CC(F)(CO)C2)=O)CCN(C(=O)Cc2ccsc2)CCC1(F)F 57143,N1(C(=O)C=CCF)CCC(O)(CN(C(=O)CN2CCSCC2)Cc2ccccc2)C1 57144,O=C(C1=CC2(CCOC2)C1)NC(Cc1cc(F)c(Cl)c(F)c1)C(=O)O 57145,C1(NC(C2(OCC)CCSCC2)=O)CN(C(=O)CSc2cnn(C)c2)CCC1F 57146,C1(C)(C(c2ccc(CC#N)s2)NC)CCCN1C(=O)CC1CCCC1C(=O)OC 57147,n1(CC)cnc2c(NC(C)CC(C)C(F)F)[nH]c(=NCc3nccs3)nc12 57148,CC(C)CCCC(C)NC(C1CC2(C1)CN(C(=O)Cc1noc(C(C)C)n1)C2)=O 57149,C1(CNC(C(C)OCCC(C)C)=O)(CNC(=O)C(N)=O)CC1(F)F 57150,CCCCCCCC(=O)N1C2CCC(C2)C1CNC(C1CCCS(=O)(=O)C1)=O 57151,CCCCCCCCC(C(=O)NC1COC1)N1CC2CSCC2C1 57152,C=C(C)CC(C(=O)N1CCC2(CC2C(=O)NCc2cccc(Cl)c2)C1)OC 57153,C(CS(=O)(=O)CC(=O)NC1C2CC1N(C(C1CCc3nc[nH]c3C1)=O)C2C)OC 57154,c1(C2C(C(=O)NCCCN(C(C3CC3F)=O)CC)C2)ccccc1F 57155,c1(C(=O)NCC2CC(NC(c3c(CC)cno3)=O)C2)ccc(Br)c(N)c1 57156,C1(CC(=O)NCC(CNC(c2c(C(=O)OC)csc2)=O)CO)CC=CCN1C 57157,CCC(C(=O)N1CCC(CF)(NC(=O)CCc2ccccc2Cl)C1)C(C)C 57158,c1(OC)ccnc(F)c1C(N1CC(CNC(=O)C(C)SC(F)(F)F)(OC)C1)=O 57159,N1(C(c2c(COC)ccs2)=O)CCN(C(=O)C(F)C(C)(C)O)CC12CCC2 57160,CCC(CCCO)NC(=O)CCSc1cccc(OC)c1 57161,CCC(CC)(CO)C(=O)NCC1(NC(C2CCC3(C2)CC3(F)F)=O)CC(F)(F)C1 57162,N1(C(C2C(=C)C2C(=O)OC)=O)CCCN(C(C2CC2(Cl)Cl)=O)CCC1 57163,Cc1cc(C(=O)NCC(=O)NCC2(C(N)=O)CN(C(=O)C(C)(C)CF)C2)c(C)o1 57164,c1(CC(=O)NC2CC(C(N3CC(C)OCCC3)=O)C2)cnc2ccccn12 57165,c1(CC(N2CCC(CCNC(C3C(=O)OCC3)=O)C2)=O)c[nH]c2ccc(F)cc12 57166,C1(N(C(C2C(OCC)C2C)=O)C)CCCN(C(=O)C(C)O)C1 57167,C(=O)(CC1=NNC(=O)C1)NCC1N(C(CCc2ccnc(C)n2)=O)C2C(C1)C2 57168,C1(NC(CN(S(CC)(=O)=O)C)=O)CCN(C(C2CC2C2(C)COC2)=O)C(C)C1 57169,N1(CC(=O)NCC2(NC(C3C4CC5C(C4=O)C35)=O)CCCC2)C(=O)CCCC1=O 57170,C(=O)(C(C)S(C)(=O)=O)NC1(CCCC(=O)Nc2cccc(C(C)C)c2)CCC1 57171,C1(CNC(C(C)OC)=O)CCN(C(=O)CC(C)(C)C)CC1 57172,N1(C(C(CCC)F)=O)CCC(C)CC1CNC(c1ccc(CSC)o1)=O 57173,N1(C(CCCSC(C)(C)C)=O)CCCC2(CNC(c3ccc([N+](=O)[O-])o3)=O)CC12 57174,N1(C(C(CSC)O)=O)CCC12CN(C(=O)CC1(C)CCOCC1)C2 57175,c1(OC)c(Cl)cc(C(=O)NCC23CC(CCO2)N(C(=O)CSC)C3)cc1Cl 57176,CS(=O)(=O)CCC(=O)NCC(C1CCOC1)NC(c1cocn1)=O 57177,C(N=c1cc(NCC2CC3CCC3C2)nc[nH]1)C1(COC)CCC1 57178,n1(C2C(C(=O)OCC(C)Cc3cccs3)C2)cnc2ccccc12 57179,CCC(C)CCC(=O)NC(Cn1cccn1)C(=O)N(C1CCCC1C)C 57180,N(C(=NCCC(=O)NC)NCC(F)F)Cc1cccc(C)n1.C(C)(C)C 57181,c1(CC)cccc(C(N2C(C(=O)NCC3(F)CCCCC3)CCC2C2CC2)=O)n1 57182,C12(C(=O)NCC3CCN(C(C(CC)c4cccnc4)=O)C3)CC(CN1C1CC1)C2 57183,C(=O)(CC(C)(C)CNC(C)=O)N1CC(OC)C(NC(=O)C(C2CCCCC2)F)C1 57184,C1(C(=O)NC(CC)C(=O)c2ccccc2)CCc2nc(C(C)(C)C)ncc2C1 57185,n1(CC(=O)NC(C)CCNC(=O)CC2CCC23CCC3)nc2ccccn2c1=O 57186,Cc1cc(C(=O)NCC2CC(NC(c3ccc(SC(F)(F)F)s3)=O)C2)nc(C)n1 57187,Cc1n[nH]c(C)c1C(N)=O.C12CCCN(C1)Cc1c(con1)CNc1cn2nn1 57188,CCCCC(O)C(C)C(=O)NC(C)CN(C)C(c1ncc[nH]c1=O)=O 57189,C1(CC)CN(C(c2cccc(OC)c2C)=O)CCC1NC(=O)C=C(CC)CC 57190,n1(C(C(=O)N(C(CNC(c2c(C(C)C)n[nH]c2)=O)C)C)C)cnc(C#N)n1 57191,C(=O)(C(C#N)CC)N(CC(=O)NC(C=C)(C)CC)CCC 57192,CC1CC=C(C(=O)N2CC(NC(=O)CCOC3CC3)CC3(CC3)C2)CC1 57193,C1(CNC(CC#N)=O)CCC2(CO1)CC(NC(=O)CCC1CCCCCC1)C2 57194,Cc1[nH]nc2c1CC(C(N1CC(CNC(C3CCCN3N=O)=O)CC1C)=O)CC2 57195,N1(C(C(C)NC(c2ccoc2)=O)=O)CC2(CC(NC(c3cnccn3)=O)CO2)C1 57196,Cn1nc(C(=O)NCCCCCC(=O)NCCc2csnn2)cc1C#N 57197,c1(C(=O)NCCCOCCNC(C2(C)CCCS2)=O)cn2cccc(F)c2n1 57198,C1(NC(CCCN2C(=O)CN(C)C2=O)=O)CC12CCN(C(C1CC1(F)F)=O)CC2 57199,c1(C(=O)NC2C(CNC(CC3(COC)CC3)=O)C2)cc(C#N)ccc1C 57200,Cc1ccc(C(=O)N(CCCC(C)O)C2CCCC2)c(C)c1.c12ccccc1S2 57201,N1(C(C2(OC)CCCOC2)=O)CCC(NC(=O)CCn2nc(C)nc2C)C(O)C1 57202,Cc1cc(C(=O)NCC2CCC(C(=O)NC(C)C(=O)NC(N)=O)CC2)c(C)o1 57203,c1(C(=O)NCC(CC)NC(=O)Cc2csc(C)c2)cnn(C2CCCC2)c1CC 57204,N1(C(CC2CCCC(OC)C2)=O)C2CCC1CC(CNC(c1ccc(Cl)s1)=O)C2 57205,O=C(N=c1[nH]nco1)C12CC(C=O)(C1)C2.N1(CCn2ccnc2)CCC(O)CC1 57206,CN1CCC(CO)(CNC(C23CC2CCN3C(=O)C(O)C2CCCC2)=O)C1 57207,C12(C)CCCN(C1)C2=O.C12CCN(CC1)C(=O)N2.c1(COC)ccc(C#N)s1 57208,N1(C(c2n(CC=C)ccn2)=O)CC2CCCC(NC(C34CCC(C3)OC4)=O)C2C1 57209,Cc1cccc2c1OCC2C(=O)NCCOC(C)(C)CNC(=O)CC1CCOC1 57210,C1(COC(=O)N(C)C)(CO)CCOCC1.c12cn(nn1)CC(=O)NC2C(C)C 57211,C12(COC)COC(C(=O)NCC3C=CCN3C(c3cc(C(C)(C)C)n[nH]3)=O)(C1)C2 57212,Cc1cc(NC(=O)CC2C3CN(C(=O)C=Cc4ccccc4)CC23)cc(C)c1F 57213,CCC(CCOC)C(=O)N1CCCCC1CCCNC(=O)C=C1CC1 57214,c1(CC)nc(N2CCC(NC(C3(n4cncn4)CC3)=O)C(F)C2)cc(C)n1 57215,N1(C(c2ccc(C)o2)=O)CC(C)N(C(c2nc(N)sc2Br)=O)CC1C 57216,C1(CNC(c2cccc(C3CCC3)c2)=O)C2CCC(C2)N1C(=O)CC1(O)CCC1 57217,Cc1cc2cc(C(N3CCC(NC(=O)C(C)(C)F)C4(CCC4)C3)=O)oc2cc1C 57218,CCC(C)C(=O)C(=O)N1CC(C)(CCC(N2CCCCC2CC)=O)C1 57219,C(=O)(CCCC(=O)N(C)C)NCC1C(C(=O)NC(CCC=C)C)CCCC1 57220,c1(C(N(C(C)CC(=O)NCCCCC2CC2C)C)=O)cc(F)ccc1F 57221,C(CCC(C(=O)N1CCCCCCC1)NC(C1CC2CCCC2C1)=O)OC 57222,c1(C(N(CCNC(C2C(Cl)(C(=O)OCC)C2)=O)CC2CC2)=O)c(Cl)c(C)nn1C 57223,C(=O)(C#CC(C)(C)C)NCC(c1ccc(C)cc1)NC(C(CC)OC)=O 57224,c1(C(N(CCCN(C(C(C)C(C)C(C)(C)C)=O)C)C)=O)cc([N+](=O)[O-])ccc1Cl 57225,C1(OCC)CN(C(=O)C=C(C)C2CC2)CC12CC2 57226,CC(C)C(F)C(=O)NC1CCN(C(C)C(N2CCCC(C)C2)=O)CC1 57227,c1(C(=O)NC2C(NC(CCC)=O)C2)cccc(N)n1 57228,c1(CC(=O)NCCN(C(=O)CN(C(=O)C(C)C)C)CC)csc(-c2ncccn2)n1 57229,c1(CNC2CN(C(COC)=O)CC2C)cccc(CNC(=O)OC(C)(C)C)c1 57230,C1(C(N2CCC(COC)(NC(=O)CCC(F)F)C2)=O)OC(C)(C)OC1(C)C 57231,CCC(C)CC(C)C(=O)N1CC2CC(C1)N2C(C1(Cl)CC1)=O 57232,N1(C(C(C(C)C)NC(N)=O)=O)CCCN(C(C2SC3C=CC2CC3)=O)CC1 57233,c1(CNC(C(CSCC)NC(C2CSC2)=O)=O)ccccc1O 57234,Cc1n[nH]c(C)c1CCC(=O)NC1(CNC(c2c(C(C)C)cnn2C)=O)CCC1 57235,CC1(C)COC(CC(=O)NCCOCCNC(C2(c3ccns3)CC2)=O)C1 57236,C1(NC(CCOCC#C)=O)CCCN(C(c2cc(N)nc(Cl)c2)=O)C1C 57237,c1(C(=O)OC)ccc(CC(=O)NC(C)CCNC(C2CC(OC)C2)C)cc1F 57238,c1(C(N2CCCC(CCCCNC(CC=C=C)=O)C2)=O)c(OC)cccc1Cl 57239,CC1=C(C(=O)NCC2CC(NC(c3ccc(Cl)c(Cl)c3)=O)C2)CCCC1 57240,N1(c2nc(C#N)cc(C)n2)CCC2C1CCCN2C(=O)C(C)(C)C 57241,C1(NC(c2c(CC=C(C)C)cccc2)=O)CC2(CCCCN2C(=O)CCF)C1 57242,N1(C(=O)OC(C)(C)C)CCCC(CO)C1C(=O)NCC#Cc1cn[nH]c1.C(=O)C1CC1 57243,c1(CC)cn2c(n1)CC(C(N1CC(OCCNC(=O)C(O)C(C)(C)C)C1)=O)CC2 57244,CCCCC(C(=O)OC)NCC1CN(C(=O)OC(C)(C)C)C(C)(C)C1 57245,c1(CC)oc2ccccc2c1CC(=O)NCC(C)N(C)C(c1ccnc(O)c1)=O 57246,C12(NC(C3CCC(C)C3)=O)CCCC1N(C(c1cnc(C#N)s1)=O)CCC2 57247,c1(C(c2n(C(CC)C)nnn2)NCCOc2cccc(C)c2)cc(Cl)c(Br)cn1 57248,N(C1COc2cc(Cl)ccc21)C(=O)Nc1cc(C2CC2)ncn1 57249,N1(C(=O)NC(C)Cc2ccccc2)CCC(N)CC1.c1(-c2ccccc2)ccncc1 57250,C1(n2cc(CCOC)nn2)(C(=O)NC(C)COCc2ccccc2)CCOCC1 57251,C(=O)(C(C)C(=O)NC1CCCC(NC(=O)C(Cl)=CCl)C1)OC 57252,c1(CNC(c2n(C(CC)C)nnn2)CCCc2ccccc2)ccc(F)cc1Br 57253,c1(-c2c(SC)cccc2)c(C(N2CCOC(C)C2)=O)nn2c1CCCC2 57254,c1(CC)cn2cc(C(N3CCC(N(C(=O)COC(F)(F)F)C)C3)=O)cc(F)c2n1 57255,C1(C(=O)Nc2cc(O)ccc2F)CCCCCCN1C(c1cc2occc2[nH]1)=O 57256,C1(C(=O)NCC(C)N(C)C(c2csnc2Cl)=O)CCCCC12CCC2 57257,C1(C(N2CCC(N(C(=O)CCOc3cccc(F)c3)C)CC2)=O)COCCOC1 57258,C1(NC(C2N(C)CC2)=O)CCCC(C(=O)NCCC(Cl)Cl)CC1 57259,CC1(C(=O)NCc2ccc(CCNC(C3CNC(=O)C3)=O)cc2)CCCCCC1 57260,N1(C(c2sc(C=O)c(Br)c2Br)=O)CCC2(CC1)CC(C(N1CNC(=O)C1)=O)CO2 57261,C12(C(N(C(C)CNC(=O)CCC3CC3)C)=O)COC(C(F)(F)F)(C1)C2 57262,C(C(CC(=O)N(C1CCOC1)CCO)NC(=O)CCc1cc(C)on1)OC 57263,C1(NC(c2cc(O)ncn2)=O)C2CCN(C(=O)CCCC3CCCCC3)C12 57264,c1(NC(CCN(C(=O)CCOC2COC2)C)=O)cncc(C(F)F)c1 57265,C(=O)(C(F)CC(C)(C)NC(c1ccc(CO)s1)=O)N(C1(C#C)CC1)C 57266,C1(F)(CNC(C(=O)NCC)=O)CCC(NC(=O)C=C(C)C)C1 57267,N1(C(c2cc(CC)c(F)cc2)=O)CC(C)N(C(=O)CC(F)(F)CC)CC1C 57268,N1(C(=O)CC2CCC(C3CC3)O2)CCN(C(=O)C(O)C2CCCC2)C(C2CC2)C1 57269,C(=O)(C(CCNC(C1(O)CCCC1)=O)OC)NC(C#C)CC1CCCC1 57270,C=C(C)C(C)(O)C(=O)NC1CCC(NC(c2ccc(CNC(C)=O)cc2)=O)CC1 57271,C1(C(=O)NCc2c(C)ccc(C)c2)CC2CCCCC2N1C(c1conc1C)=O 57272,C1(C(N2CCCC(CNC(C(C)C3CCOC3)=O)C2)=O)CCCCC12OCCO2 57273,C1(CNC(C2CC(CC)C2)=O)(OC)CCN(C(=O)C(O)Cc2cnn(C)c2)CC1 57274,C1(OC)CC(C(N2CC(C(C)C)C2)=O)N(C(=O)Cc2ccns2)C1 57275,c1(C(=O)NCC(CC)NC(C2(C)C=CCCC2)=O)cc2n(n1)CC1(CC1)C2 57276,C(=O)(C(C)(CC)C(N)=O)N(C)Cc1ccccc1CNC(c1nn(C)cc1Cl)=O 57277,N1(C(C(CCCCC)O)=O)CC2(CCCCN2C(C23CC(C)(C2)OC3(C)C)=O)C1 57278,c1(CC)nnc(N2CCC(C)(c3ccccc3)C2)n1CC(C)CC1CCOCC1 57279,C1(F)(CNC(c2n(C=C)ncc2)=O)CCCN(C(c2ccc(C(F)F)o2)=O)CC1 57280,N1(C(C2(CNC(CC(C)n3cccc3)=O)CC2)=O)CCC(C2(C)CC2)CC1 57281,c1(C(=O)NCC2CCN(C(C3(C)C(C)C3)=O)C2)ccc2oc(O)nc2c1 57282,C=CCCC(C)NC(=O)C(C)=CCNC(=O)CCc1cnn[nH]1 57283,Cc1cc(=NC(Cc2ccccc2)C(=O)NCCCOC(=N)O)[nH]n1C 57284,C1(C(=O)NCc2cccc(OCC)c2)C2CC3C(C2NC(=O)C2=CCCCO2)C13 57285,c1(NC(C23CC2CN(Cc2cnn(C4CC4)c2)C3)=O)cc(F)ccn1 57286,Cc1ccc(O)cc1C(=O)NC(CC1CC1)CC(=O)N1CCC(C(F)(F)F)C1 57287,c1(C(C)C(N2CCC(N(C(=O)CC(F)(F)F)C3CC3)CC2)=O)cccc(C#N)c1 57288,C(=O)(C1CCc2ccccc21)NCc1cc(C(=O)NCCCC2CCC2)no1 57289,CCC(C)(CC(=O)Nc1cnn(CC2CCC2)c1)NC(=O)COCC(C)C 57290,c1(C(N(C2CCN(C(=O)CC(C)(C)C)C2)CC)=O)cccc2ncnc(O)c12 57291,CC1(C)CN(C(=O)CNC(N)=O)C(CNC(C2SCCS2)=O)CO1 57292,C1(O)(C(C)CNC(=O)Cc2cnns2)CCN(Cc2cc(-c3ccoc3)[nH]n2)C1 57293,C1(S(C)(=O)=O)(C(=O)NCC(CC)(C)NC(C2CCN(C)C2C)=O)CCC1 57294,C1(C(=O)NCCCCC=C)CCC2CCC1N2C(c1cnn2c1CCC2)=O 57295,Cc1ccc(NC(C2(C)CCN2Cc2cccc(Cl)c2C)=O)cc1OC(F)F 57296,C(=O)(CCC(=O)N(C(C)CNC(C12CCC(CC1)O2)=O)C)NCC 57297,c1(OC(C)C)ccccc1C(=O)NCCC(C)NC(C1CCCN1C(C)C)=O 57298,N1(C(=O)COc2ccc(Cl)c(Cl)c2)CCC2(CC1)CN(C(C1C=CCC1)=O)C2 57299,c1(C(=O)NCC(C)CN(C(=O)CC2CC23CC3)C)c[nH]c(C(N)=O)c1 57300,C1(C(=O)NC(C2CCC2)C)CCCN(C(c2cccnc2S)=O)C1 57301,C1(NC(C2CC(C)(C(=O)OC)C2)=O)CCC(NC(c2ccc(=O)oc2)=O)CC1 57302,c1(C(=O)NCc2c(CCNC(C(CC)C(C)C)=O)ocn2)cc(S(C)(=O)=O)co1 57303,C12CCCN(C1)C2=O.C1(NN(C(=O)COC2CCN(C)CC2)C)CCC(CO)CC1 57304,c1(C(c2nnnn2C2CCC2)NSC(F)(F)F)cccc(Br)c1 57305,C(=O)(CCCC(CC)NC(=O)CCOC(C)C)NC(CCC)C(C)(C)C 57306,CCC(F)(C(=O)OC)C(=O)N1CCC(O)(CCNC(=O)C(C)OCC2CC2)CC1 57307,N1(C(Cc2c(C)n[nH]c2)=O)CCC2(CCN(C(=O)CNC(C3CC3C)=O)CC2)C1 57308,N1(C(C2CCC(CC)O2)=O)Cc2[nH]nc(C(N3Cc4c[nH]nc4C3)=O)c2C1 57309,C1(C(N(CCOc2ccccc2C)CC)=O)CCCN(Cc2nc(C)cs2)C1 57310,C1(NC(C2CCC(CNC(C3C(C)=CCS3)=O)O2)=O)CC(=O)N(O)C1 57311,N1(C(c2nc(C)oc2)=O)CCCN(C(=O)CCn2ccc3cccnc23)CC1C 57312,C(c1c(Cl)nc2ccccn12)=CC(N1CCCC(F)(CNC(C2C(C)C2)=O)C1)=O 57313,C(CCC(=O)N1CC(OCC(=O)NCC2CC2[N+](=O)[O-])C1)SC 57314,c1(C(=O)NC2(CCNC(c3ccon3)=O)CCC2)cc(O)cc(F)c1 57315,C1(CN(C)C(C2C3CCCCC23)=O)CCCCN1C(=O)CCC1CCOCC1 57316,N1(C(C(CSCC)NC(c2ccco2)=O)=O)CCCN(C)CC1CC 57317,Cc1c(F)ccc(N)c1C(=O)NCC1(NC(=O)C(c2cccnc2)O)CC1 57318,CC1CN(C(c2cnc(O)c(F)c2)=O)CC2(CCN(C(C34CCC(C3)C4)=O)C2)O1 57319,C1(CC(=O)NC2C(CC)N(C(C3CNC(=O)C3)=O)CC2)CCC2(CC1)OCCO2 57320,CC(C)CCC(O)C(=O)N1CCC2(CC2NC(=O)C2=CCC2)C1 57321,c12cc(n[nH]1)C(=O)NC2.N1(C(C2C(=C)C2C)=O)CC(COC)(OCC)C1 57322,c1(C2C(C(N3CC(n4cc(-c5cc(F)ccn5)nn4)C3)=O)CC2)ccc(F)cc1 57323,N1(C(c2nccc(CC)c2)=O)CC(C(N2CC3CCCC23)=O)CC(C)(C)C1 57324,CC1CC2CN(C(=O)CCc3cccc(OC)c3)CC2N1C(=O)COC(F)(F)F 57325,C=C(F)C1(CC(N2CCCCC2CCN(C)C(c2nc(C)c(C)s2)=O)=O)CCC1 57326,CC(C)C(C(=O)N1CC(CO)(NC(=O)CCN2CCNC(=O)C2)C1)NC(N)=O 57327,Cc1cnc(Cl)c(C(=O)N(C)CC2CCCN2C(=O)C(=O)C2CCCC2)c1 57328,c1(NC(C2C(NCc3ncc(C)c(Br)c3)CCC2)=O)ccc2oncc2c1 57329,C(=O)(CC1=CCN(C(c2ccsc2C#N)=O)CC1)NCCC(C)N(C)C 57330,C1(CNC(COCC(=C)C)=O)CN(C(=O)CCOC2CCCC2)C2CC12 57331,C(=O)(CCN(OC)C(=O)C1CS(=O)C1)Nc1c(OC)cccc1 57332,c1(C(=O)NCc2ccc(C)o2)cccc(Cn2ccnc2)c1 57333,C(C(C)C(F)C(=O)N(CC(N1CCCC1)C)C)NC(c1cnc(C)n1C)=O 57334,CCCCC(CN(C)C(C1CCN(C(C2(CCOC)CCC2)=O)CC1)=O)CC 57335,Cc1cccc(C(N2CC(O)(C(C)(C)CNC(=O)C(O)C3CCC3)C2)=O)c1F 57336,N12CCC3(CC1)CC3C2=O.C1(=CC(=O)NC2C(C(C)(C)C)C2)CCSCC1 57337,N1(C(c2c(C)nncc2)=O)CCC2C(CCCN2c2ncnc3c(C)csc23)C1 57338,C1(C(=O)NCC2CCSC2)(CC)CCCN(C(c2cnccc2C)=O)C1 57339,CCCCC(C(=O)NC1CC1CC)NC(=O)C(C)(C)C(=O)NCC 57340,c1(CC(=O)NCC2N(C(CSCC#C)=O)CCN(C)C2)cccc2c1OCCO2 57341,C=CCC(CC)C(=O)NCCC1(NC(=O)Cc2csc(-c3ccoc3)n2)CC1 57342,C1(C(=O)OC)CC(C)CN(C(=O)Cn2cc(-c3cc(Br)ccc3OC)nn2)C1 57343,C(CC(O)CNC(c1cn(Cc2ccccc2)nn1)=O)NC(C1(F)C(C)C1)=O 57344,Cc1scc(C(=O)NC2CC3C(NC(=O)CCc4nccn4C)C3C2)c1C 57345,N#CC1CCC(CC(=O)N(CCC(=O)N2CCC2CF)CCO)C1 57346,n1(CC(=O)NC2CC(NC(C34CCC(CC3)C4)=O)C2)nc2n(c1=O)CCOC2 57347,C(c1cn(C)c(=O)n(C)c1=O)=CC(N1CC(NC(c2c(C)ccs2)=O)C(C)C1)=O 57348,c1(C(N2CC(NC(=O)CSc3ccc(Cl)cc3)(CO)C2)=O)cccc(F)c1O 57349,C(N=c1[nH]c(=NCCC(C)(C)CO)[nH]c2c1SCC2)C1(N(C)C)CCCC1 57350,c1(C(=O)NC(c2nc(C3CC3)no2)C)cc2n(c1)CCS(=O)(=O)C2 57351,CC(C)(CNC(C1CCC2(CCC2)C1)=O)CC(=O)NC(C)(C)C(C)(C)CO 57352,N1(C(C(c2cccc(Cl)c2)C)=O)CC2CCN(C(=O)Cn3cnnc3)CC12 57353,CC(C(=O)N1CC(N(C)C(c2coc(C3CCCC3)n2)=O)C(C)(C)C1)S(C)(=O)=O 57354,Cc1nc2sccn2c1C(=O)NCC(F)CNC(=O)COCC(C)(C)C 57355,c1(C(=O)NCC(CC)NC(=O)CC2NC(=O)CNC2=O)cc2c(C)ccc(F)c2o1 57356,C(=O)(C(C)S(N)(=O)=O)NCCn1ncc(C(=O)NC(COC(C)C)(C)C)c1 57357,O=C1CNc2cc(C(N3CCCC(NC(C4C=CCCC4)=O)CC3)=O)cnc2N1 57358,C1(NC(=O)C(CO)c2ccccc2)CCCCCN(C(c2nccc(Cl)c2F)=O)C1 57359,C1(C(=O)NC2CCC(CNC(c3ccnnc3Cl)=O)C2)CCC=CCCC1 57360,CC(C)(C)C(O)CC(=O)N1CCC2(CC1)CC2NC(=O)OC(C)(C)C 57361,c1(C(=O)NC(C2CCN(C(c3n[nH]cc3Br)=O)C2)C)cccc(CO)c1 57362,C(=O)(C1CNC(=O)c2ccccc21)N1CCCCC(CNC(C2(C#C)CC2)=O)C1 57363,c1(C(=O)NC2CCCC2C(=O)NCc2cnccc2Cl)cc2n(n1)CCC2 57364,c1(CC)occc1C(N1CC(NC(C2CCC2c2ccccc2)=O)C1)=O 57365,N1(C(CCC(C)C)=O)CC2(CC(NC(=O)CC3CCOCC3(C)C)CO2)C1 57366,N1(C(COC(C)=O)=O)CCC2(CC1)CC(C)N(C(=O)C=Cc1ccccn1)C2 57367,N1(C(=O)OCC(=O)NC2C(C)SCC2)CCN(C(=O)C(c2cnccn2)=O)CC1 57368,C1(C)(CNC(c2cc(COC)[nH]n2)=O)CCN(C(c2snnc2C)=O)C1 57369,Cc1cc(C(N2CC(CC(C)NC(C3C=CCCC3)=O)C2)=O)ns1 57370,C1(OC)CCC12CC(C(=O)NCCCC(C)(C)NC(=O)CCc1ccnn1C)C2 57371,N1(C(CCS(N)(=O)=O)=O)CCCCC12CC(NC(=O)C(=Cc1cccnc1)F)C2 57372,c1(CC(=O)NCC(CCNC(=O)C(C)Cc2cnc[nH]2)OC)cncnc1O 57373,N1(C(CNC(=O)OC)=O)CC(CCNC(=O)C=C2CCN(C)C2)C(C)C1 57374,c1(C(=O)NC(CCCC)CNC(=O)C(=O)NCC2CC2)cn(C)c(C)cc1=O 57375,Cc1cc(C(=O)NCC2(F)COCCOC2)c(C)nc1C 57376,N1(C(C2COCCN(C(Cc3ccn(CC)n3)=O)C2)=O)CCCN(C)C(=O)C1 57377,C1(NC(C(C)OCc2ccc(C)cc2)=O)CN(C(=O)C2=COCC2)CCC1F 57378,C=CC1(C(=O)N(C)CCOCCCNC(=O)CCS(C)=O)CCOCC1 57379,Cc1c(C(=O)N(C2CC(NC(c3cccc(N)n3)=O)C2)C)cnc2ccccc12 57380,CC#CCC(C(=O)N(CCC(=O)OCC)C)NC(=O)CCc1cn[nH]c1 57381,c1(CC(N2CCC(C)C(NC(c3ccon3)=O)C2)=O)ccc2cccnc2c1 57382,N1(C(C(=O)NCC)=O)CCCC2(NC(=O)CSc3c(C)n[nH]c3C)CC2C1 57383,C1(CCNC(C(C)OCCOC)=O)(NC(CCCCOC(C)(C)C)=O)CCCC1 57384,c1(CC#N)c(F)cc(NCc2ccc(-c3cncnc3)cc2)cc1F 57385,c1(C(N(C2C(C)CC2)C)=O)coc2c1CN(C(=O)CCc1nccn1C)C2 57386,N1(C(C2CCC(C(N)=O)C2)=O)CCCC2(CCN(C(c3cccnc3F)=O)C2)C1 57387,C(=O)(CCCC(F)(F)CO)N1CCCC(C(C)NC(c2nccc(C)n2)=O)C1 57388,C1(C)(C(=O)NC(C(C)O)CO)CCCN(C(=O)CCC2CC2C)C1 57389,c1(C(=O)NCCOCC#C)ccnc(CNC(=O)C(C)C2CCCO2)c1 57390,C1(C(N2CCC(CN(C)C)CC2)=O)C2CCC(C2)N1C(C1CC2COCC2C1)=O 57391,c1(N(C)C)cncc(NC(=O)C=CC(=O)NC2CC2)c1.N12CC3CC1(C3)C2=O 57392,c1(CC)sc(=N)[nH]c1C(=O)NCC1CC1CNC(c1cn(C)c(C)n1)=O 57393,CC12CN(C(=O)Cn3cnc4c(N)ncnc34)CC1CN(C(C1(CO)CC1)=O)C2 57394,c1(C(=O)NCC2CN(C(C3(c4cccs4)CCOCC3)=O)C2)ccn2ncnc2c1 57395,C1(Cn2cc(CNC(CCC)=O)nn2)CCCC(NC(=O)C(F)(F)CC)C1 57396,CC(C(=O)NCCC1CN(C(=O)CCN2CCN(C)CC2)CCCO1)C(C)(F)F 57397,C=C1CC(C(=O)N(C)CC2COC(=O)N2)(CNC(c2sccc2CC)=O)C1 57398,C1(CC)CNC(=O)CN1C(=O)C(C)(C1CC1)N(C)C(c1cc([N+](=O)[O-])n[nH]1)=O 57399,c1(N2C(C)(C(=O)NC(c3ncccn3)CC)CC2)ncnc2c1ncn2C 57400,CCC(C)CC(=O)N(C1CC(NC(=O)CCOc2ccccc2F)C1)C 57401,c1(C(=O)NC(CCN(C(C(CCC)CC)=O)C)C)ccc([N+](=O)[O-])cc1CC 57402,N1(C(c2ncc[nH]2)=O)CCCC(C2CCN(C(C3(C(F)F)CCC3)=O)C2)C1 57403,CCCCCCC(=O)N(C)CC1CCN(C(C2(C(=O)OC)CC2)=O)CC1 57404,C1(NC(=O)CCc2cscn2)COC2(CCN(C(C3CCCS3)=O)CC2)C1 57405,C(C1CCC(C)CC1)=C(C(N1CCC(N(C(C2CCN(C)C2=O)=O)CC)C1)=O)C 57406,C1(C(N2CCCCCC(NC(CC)=O)C2)=O)COc2cc(OC)ccc2C1 57407,C(=O)(CS(=O)(=O)C(C)C)N1CCN(C(c2snc(C)c2N)=O)C(CC(F)F)C1 57408,C(=O)(C(C)(CC)C(N)=O)N1C(CNC(c2c(SCC)ccc(Cl)c2)=O)CC=CC1 57409,c1(C(N(CCCCCNC(c2n(CC)ncn2)=O)C(C)C)=O)occ2c1CCC2 57410,N1(C(CSC)=O)C2CCC1CN(C(C1CCOC(C(C)C)C1)=O)C2 57411,C1(C(=O)OC)N(C(=O)CCC(C)NC(c2coc(CO)c2)=O)CC1(C)C 57412,N1(C(CC(C(C)C)NC(=O)Cn2cnnc2)=O)CCN(C)CC(C)C1 57413,CN(C)NC(=O)CCC(=O)N1CCC1CNC(c1ccccc1-n1cnnn1)=O 57414,C(=O)(C(C(=O)NC(C)Cn1cc(-c2ncccc2F)nn1)OC)OC 57415,C1(C(N(CC(C)O)CCNC(c2cnn[nH]2)=O)=O)CCOC(C)C1 57416,C1(NC(c2cc(Cl)cs2)=O)CCN(C(=O)C=CCn2cncn2)C12CC2 57417,c1(CCC(=O)NCC(CO)NC(c2c(C)nccc2)=O)cccc(F)c1Br 57418,N1(C(c2cc(OCC)n[nH]2)=O)CC(NC(=O)C(C2CCCCC2)F)CC1CO 57419,N1(C(CCc2cnc(C)s2)=O)CCCC(CNC(C2CC2(F)F)=O)CC1 57420,c1(CC(=O)N(C2CC(CNC(=O)Cc3ccns3)C2)C)ccc(Cl)cc1 57421,C(=O)(C1Cc2c(Cl)cccc21)NCC1CC2N(C(C3CCN(C)C3)=O)C(CC2)C1 57422,C1(c2nnnn2C2CCCC2)(NCCCC(=O)OCC)CCCC(C=C)C1 57423,CC1CCC(NC(C2CNC(=O)C2)=O)C1 57424,N1(C(C2(C(C)C)CCN(C(CCC(CC)=O)=O)C2)=O)CCCC(C2CCC2)C1 57425,c1(C(=O)NCC2CCC(C3CC3)O2)ccc(Cn2cc(C3CCCC3)nn2)o1 57426,C1(n2cc(CCNC(=O)CCOC3CCOC3)nn2)(CN)CCOCC1 57427,C(CCCC(=O)NCC1CC(CCC)C1)N(C(CSCC#C)=O)C 57428,Cn1[nH]c(C(=O)NCCC2CCN(C(=O)COC3COC3)CC2)nc1=O 57429,Nc1ncccc1C(N1CCC(N(C(=O)CC2CS(=O)(=O)C2)CC2CC2)CC1)=O 57430,c1(C(=O)NC2C(NC(CC3CC(=O)NCC3)=O)C2)cc(F)cc(Cl)c1 57431,C(=O)(CC(C)(C)c1ccccc1)NCC(Cn1cc(CCCSCC)nn1)(F)F 57432,C1(F)(C(=O)NCC(CC)(CC)OC)CCCN(C(c2ccc(C)o2)=O)C1 57433,C1(CCC(=O)NCC(C(N2CC(O)(COC)C2)=O)C)CC2CCC(C1)C2 57434,c1(-c2cccc(COC)c2)cccc2nc(C(=O)NCCN3CC4CC4C3)cn12 57435,Cc1cnn(C)c1-c1cn(C(C)(C)CC(=O)NCCC(=O)NC2CC2C)nn1 57436,C1(C(=O)NCC2OCC(C(=O)NCc3c(CC)n[nH]c3)C2)CC(=O)NC(=O)C1 57437,C(c1ccc(O)cc1)=CC(=O)NCCC1CCN(C(C2CC(F)(F)C2(F)F)=O)C1 57438,n1(CCC(=O)NC2C(NC(C3ON=C(CC)C3)=O)CCC2)cc(S(N)(=O)=O)cn1 57439,C1(S(N)(=O)=O)(C(=O)NCc2cn(CC(=O)NCCCOC(C)C)nn2)CC1 57440,n1(CC(=O)N(CC(C)NC(c2sccc2-n2cccc2)=O)C)cc(CO)nn1 57441,c1(C(=O)NC(C)Cc2cccs2)ccc2nn[nH]c2c1O 57442,C1(CC)C(O)CCN1C(=O)C(C)(C)CC1CC1 57443,c1(C(=O)NC(CNC(c2ccn(CCCC)n2)=O)C2CCC2)cn(CC)nc1C 57444,N1(C(C2COC(C)C2)C(=O)NCCCOC)CCc2ccc(Cl)cc2C1C 57445,C(=O)(CC1=NNC(=O)C1)N(C(C)CNC(c1ccc(CO)c(F)c1)=O)CC 57446,C1(C(=O)NC(CC(C)NC(CC2(OC)CCOCC2)=O)C)CC12CCCCC2 57447,N1(C(C(C(C)C)C2CCC2)=O)CCCCC(C(=O)NOCCC(F)F)C1 57448,C(CCCC(=O)N(C1CCC1(C)C)C)N(C(C(C)N(C(C)=O)C)=O)C 57449,O(NC(=O)C(CNC(=O)CCCCCSC)C(C)(C)C)CC(CC)C 57450,N1(C(=O)NC2C(=O)NCC2)CCN(C(=O)CC2COCCOC2)CC1 57451,c1(C(=O)NC2CC(NC(c3cnco3)=O)C2)cncc(-c2ccccc2)c1 57452,C=CCC(CNC(c1ccc(SC)s1)=O)NC(c1cscc1SC)=O 57453,c1(CC(=O)NC2(CC)CN(C(=O)CC3(OC)CC3)C2)cn2ccccc2n1 57454,N1(C(C2C(CCC)CN(C(=O)CCn3cncn3)C2)=O)CCN(C)C(=O)C1CC 57455,c1(C(=O)NC2C(NC(CC(=C)C)=O)CCC2)cn2cc(Br)cc(C)c2n1 57456,C(c1ccc(F)cc1)=CC(=O)NCC(C)(C1CCC1)NC(c1ccc(CO)o1)=O 57457,C1(C(N(CC(C)C)C)=O)CCCN(C(C)Cc2ccc(C(C)(C)C)cc2)C1 57458,CS(=O)(=NC(=O)CCC1CC2(CCC2)C1)c1ccc(Br)cc1 57459,N1(C(CCN(C(C2CCC(=O)CC2)=O)C2CC2)=O)CC2(CCC2)CC1CO 57460,c1(OCCNC(c2cnsn2)C)ccccc1F 57461,c1(C(=O)NC(CC)CNC(c2ccc(-c3ncc[nH]3)cc2)=O)cc(=N)[nH]c(Cl)n1 57462,CC1CC2(CO1)CC(c1nnnn1CC(F)F)(NCC13CCCC1CCO3)C2 57463,Cc1ccc(NNC(=O)Nc2cnc(O)c(F)c2)nn1 57464,N1(c2cc(C)[nH]n2)CCCN(C(=O)CC23CCCC2C3)CC1 57465,N1(C(C2CCN(C(C)=O)C2)=O)CC2CCC(C1)N2C(=O)C(C)(C)C1CCCCO1 57466,c1(C(CC)(C)C)n[nH]c(=NC2CN(C(=O)CN3CCCCC3)CC2C)o1 57467,c1(C(=O)NC(CC)C)ccc(CC2(c3ccccc3)CC2)cc1 57468,c1(C(N(CCC(=O)NCC2C(OC)CCC2)C(C)C)=O)csc(C)c1C 57469,c1(CC)cc(C(N2CC(CNC(c3scnc3COC)=O)C(C)C2)=O)cc(N)c1 57470,C(=O)(CC1=CCOCC1)N1C(C(=O)NCc2c(CC)nn(C)c2)CC(F)CC1 57471,CC1(C)CCCN(C(=O)Cc2nnc(O)s2)C1CNC(c1cnc(Cl)s1)=O 57472,c1(OC)ccc(C(C)C(=O)N(C(C)CCNC(=O)C(C)(F)F)C)c(C)c1 57473,C1(CC(N2CCC(N(CCCOC)CCO)CC2)=O)CCn2cncc2C1 57474,N1(C(C2C(NC(C(C)C(F)(F)F)=O)C=CCC2)=O)Cc2n[nH]cc2C1CO 57475,CN1CCC(CC(C(=O)O)NC(C2CCCC2CF)=O)CC1 57476,C1(NC(c2nc(COCC)sc2)=O)CC2CCC1N2C(c1cn(C)ccc1=O)=O 57477,C#CCCCCC(=O)N1CC(NC(=O)COCC#C)C(C)(C)C1 57478,N1(C(c2ccc(C(=O)OC)o2)=O)CC2CCC2(CCNC(=O)C=C(C)C)C1 57479,C(=O)(CS(=O)(=O)C1CC1)N(CCCCCNC(c1ncn2c1CCC2)=O)C 57480,c1(C2OCCN(C(CC(C)P(C)(C)=O)=O)C2)cc(F)c(Cl)cc1[N+](=O)[O-] 57481,CC1=C(C(=O)NC2CCCC2NC(=O)CC2CC=CCN2C)CCC1 57482,Nc1ccc(C(=O)NCC(C2CC2)NC(C2(O)CC2)=O)cc1OCCO 57483,C1(NC(c2c(C)ncs2)=O)CN(C(C2CCNC(=O)C2)=O)C2(CCCCC2)C1 57484,S(=O)(=O)(c1ccc2c(c1)N(C(=O)Nc1ccc(S(C)=O)cc1)CCC2)N(C)C 57485,c1(C(=O)NC(C)CNC(C2CCCCCCC2)=O)cccc(S(=O)(=O)CCO)c1 57486,N1(c2snc(C(=O)OC)n2)C2CCC1C(CNC(=O)C=CCOC)C2 57487,c1(CC(=O)NCC(F)CNC(c2cc(F)n[nH]2)=O)nccc2ccccc12 57488,CC(C)C(C(=O)NCC1(CNC(c2ccccc2)=O)CC12CCC2)N(C)C 57489,C(=O)(C1OCCc2cc(OS(=O)(=O)NCC34CC5CC(CC(C5)C3N)C4)ccc21)OC 57490,C1(C#N)(CC(=O)Nc2cnc(CC(C)C)[nH]2)CN(C(=O)OC(C)(C)C)C1 57491,c1(C(N)=O)ccc([N+](=O)[O-])cc1NC(C1CN(Cc2nc(Br)cs2)CCC1O)=O 57492,c1(C(N2CC(CNC(CC(CC)(C)C)=O)(COC)C2)=O)cc2cccnc2nc1O 57493,C1(CC(=O)NC2C(NC(c3c(OC)c(Cl)sc3)=O)C2)CCCCC12CC2 57494,Cc1cc(CC(=O)NC2CC(CCNC(=O)C=CCO)C2)cc(C)c1 57495,c1(C(CNC(C(C)CC2CC2)=O)NC(=O)CN(C)C)cccc(Cl)c1Cl 57496,CC1OC(C)C(C(N2CCN(C(=O)CC3(C)CC3(F)Cl)C(CCO)C2)=O)C1C 57497,COn1cnc(C)c1C(=O)NC1COCCN(C(=O)CCCC(C)C)C1 57498,c1(C(=O)NC(C)CNC(c2ccc(CO)cn2)=O)cc2cccnc2nc1N 57499,N1(CCCC)CCCCC1C(N1CCC(CF)(NC(c2nc(O)sc2C)=O)C1)=O 57500,C(=O)(CC(C)(C)CC)NCC(C)NC(CCCOCCC)=O 57501,N1(C(c2cc(CCCCC)[nH]n2)=O)CCCC(NC(C2(C)CCOCC2)=O)C1 57502,N1(C(C2C(COC)C2)=O)CCC(C(C)(C)NC(=O)C(=CC2CCCC2)C)C1 57503,CC(F)(F)C(C)(C)CC(=O)N(C1CCCCC1)CCNC(=O)C1CCSC1 57504,C1(CNC(C2C(C)CC(=O)CC2)=O)CC2COCC2N1C(=O)C1=NOC(C)C1 57505,NS(=O)(=O)c1ccc(C(N2CCC(F)C(NC(=O)CCc3cscn3)C2)=O)nc1 57506,C(=O)(C(F)(F)C(F)(F)F)NC1(C2N(C(C(C)NC(C3CCCC3)=O)=O)CCC2)CC1 57507,C(CS(=O)(=O)CC(=O)NC1COCCC1C(=O)NCc1cc(Cl)ccn1)OC 57508,c1(C(=O)NC2CCN(Cc3nccc(C)c3)CC2F)cc2cnccc2nc1C 57509,C1(CNC(c2ccc(COC)[nH]2)=O)CCN(C(=O)CSCC2CCCO2)C12CC2 57510,C1(C(=O)NCC(C(N2CCC(NC(CC)=O)C2)=O)N(C)C)CCC2(CCC2)O1 57511,c1(C(=O)NCC(CC)NC(C2CCC(N(C)C)CC2)=O)csc2c(F)cccc12 57512,N1(C(C2(CC)CN(C(=O)CC3CC=CCC3)C2)=O)CCC(C)(O)CC1 57513,O=C1CCC(CCC(N2CCCC2C2(NC(c3ccncn3)=O)CC2)=O)CN1 57514,N1(C(Cc2c(C)nsc2)=O)CC2CC2(CNC(=O)C(C)n2ccnn2)C1 57515,c1(C(=O)NCC2CC(NC(C3C(=C)C3)=O)C(O)C2)ccn2c(C)cc(C)nc12 57516,C1(CCNC(c2c(C)con2)=O)CN(C(C2CC2(Cl)Cl)=O)CCO1 57517,N1(C(C(C=C)(C)C)=O)CCC(NC(c2oc(C)cc2C)=O)C(F)(F)CC1 57518,N1(C(C(C)C#N)=O)CCC2CCN(C(=O)CN3CC4CC4C3)CC2C1 57519,N1(C(C(C)OC)=O)CCOCC(NC(C2CSCCS2)=O)C1 57520,CC1(C)CCCN(C(=O)C(=O)NCCCc2ccccc2N)C1 57521,N1(C(CCN(C(Cc2cccc(C#C)c2)=O)C2CC2)=O)CCOCC2(CC2)C1 57522,C1(C(=O)NC2C(NC(c3n[nH]c(C(C)C)c3Br)=O)C2)CCCCCN1C 57523,Cc1cc2[nH]nc(CNC(=O)NC(c3ccc(C#N)cc3)C)c2o1 57524,C(C(C)(O)CC(=O)NCc1c[nH]nc1C(=O)NC1CCCCC1)OC 57525,Cc1cc(=O)c(C(N2CCC(C(=O)NCC34CC(F)(C3)C4)(CO)C2)=O)c[nH]1 57526,c1(-c2c(OC)c(F)ccc2)cccc2sc(C(N3CC(F)(F)CC3OC)=O)cc12 57527,C(=O)(C(CNC(C1(C)COC1)=O)C(C)(C)C)NCC(CC)C(C)C 57528,C1(C(=O)NC2C3CC2N(C(=O)CN(C)C2CC2)C3)(OC)CCOCC1 57529,n1(CC)c(C)cc(C(=O)NC2COCCC2NC(=O)C(C)(F)C(=O)OC)c1C 57530,CC1CCN(CC(=O)NC2CCCC2NC(=O)COCCc2ccccc2)C1 57531,Cc1c(Br)ccc(N2CCN(CCNC(C3CC4CC4C3)=O)CC2)c1[N+](=O)[O-] 57532,Cn1nc(C(N2CC(NC(c3cscc3F)=O)CC(O)C2)=O)c(Cl)c1Cl 57533,C12(CNC(=O)NCCN3CCOCC3)CC(c3ccccc3)(CO1)C2 57534,CCC(C)CCCC(=O)NCC(CC)(CC)NC(c1cc(C(=O)OCC)no1)=O 57535,CCC(CNC(=O)C(CC1CCCC1)NC(=O)CN1CCNC(=O)C1)C(C)C 57536,c1(OCCNC(=O)NC2CCCC(C(=O)OC)CC2)ccc(Br)c(F)c1F 57537,C(CC(=O)N(CC(=O)NC(CO)C1(O)CC1)C)SCC 57538,N1(C(CN(C(=O)OCC)C)=O)CCC2CC12C(=O)NCCCn1cccn1 57539,C1(NC(C)=O)CN(C(=O)Cc2csc(Cl)n2)CC1c1ccccc1 57540,c1(COC)nn(C)c(Cl)c1C(=O)NC(CCNC(C1CCC1(F)F)=O)CC(C)C 57541,C1(C(=O)NCCN(C(C=C(C)CN2CCOCC2)=O)C)CCCN1CC(C)C 57542,C1(NC(c2ncn(CC)c2)=O)C2CN(C(C3(OCC)CCSCC3)=O)CC12 57543,C(C)(CO)(C(=O)N(C)CCN1CCCCC1)Nc1ccc(C(=O)OC)o1 57544,CC1=CCC=CC1C(N1CC(C)(CC(=O)NCC2(N(C)C)COC2)C1)=O 57545,C1(C(N2CC(C)(NC(c3c(C)n(CC4CC4)cc3)=O)C2)=O)CC(C2CCC2)C1 57546,C1(CC)CN(C(c2ccc(C3CC3)o2)=O)CCC1NC(=O)C(C)SC(F)(F)F 57547,N1(C(C(C)OCCCC)=O)CC2CCCN(C(c3cc4ccccn4n3)=O)C2C1 57548,C(=O)(C(C(C)C)C(C)C)N(C1CCN(C(=O)C(c2cncn2C)O)C1)CCC 57549,c1(-c2nnc(C(c3ccccc3)C)o2)ccc(OC(F)F)cc1 57550,c1(C(=O)NC2CC(NC(C(CC)OCC)=O)C2)ccnc(F)c1N 57551,C1(NC(c2cc(CCNC(c3ccn(C)c3)=O)on2)=O)C2CCCOC12 57552,C1(C(=O)NCCNC(CC2C(C)CCC2)=O)CCC(C)(F)CC1 57553,C(=O)(C(F)(F)CCn1ccnn1)NCC(C)CN(C)C(c1cc(Cl)cn1C)=O 57554,Cc1cc(C(N2CC3CC2C3C(N2CCCC(O)C2C)=O)=O)ccc1Br 57555,Cc1nc(C)c(C(C)NC(=O)C(C2CC2)NC(=O)CCC(C)N(C)C)[nH]1 57556,c1(C(N2CC3C(N(C(c4cc(COC)on4)=O)C)C3C2)=O)cc(O)cc(C#N)c1 57557,CC1(C)CN(C(=O)NCC2CCC3(C2)OCCO3)CC2(CCOCC2)O1 57558,c1(C(N2CCC(C)(NC(C3C(C)CCCC3)=O)C2)=O)cnc2n1CCS2 57559,c1(C(N2CC(OCCNC(C3(Cl)C(C)(C)C3)=O)C2)=O)ccc(C2CC2)nc1 57560,c1(C(C(=O)OC)NC(=O)CCn2cc(-c3cnsc3)nn2)ccc(F)cc1C 57561,C#CCC(C)(CC)C(=O)N1CC(NC(=O)C(c2cnn(C)c2)C)C1 57562,C(=O)(C(C(C)C1CCOC1)N(C)Cc1cccc(Br)c1)NCCCSC 57563,C(C1=C(C)OCCS1)NC(NC(COC)C)=NCc1conc1C(F)(F)F 57564,N1(C(C(C(=C)Cl)(C)C)=O)CCCC(NC(=O)C2=C(Cl)CC2)C(F)C1 57565,N1(C(CN(CCOC)C)=O)CCCC(O)(CNC(=O)CC(C)c2cccnc2)C1 57566,C(=O)(CCCCCN(C)C)NC(C(C)C)C(C)NC(C1CCCCS1(=O)=O)=O 57567,N1(C(C2C(C)(C)CCCO2)=O)CC2(CC(C(=O)N(CCO)CCO)CO2)C1 57568,c1(N2CCC(C(=O)OC)(COC)C2)ncc(S(C)(=O)=O)cc1Cl 57569,c1(C(=O)NCC2CCN(C(C(CC)(C)OC)=O)CC2)cc(O)cc(F)c1F 57570,CC1=C(C(=O)NC2CC(Nc3ncc4ccnc-4[nH]3)C23CCC3)CCS1(=O)=O 57571,C1(NC(c2c(C)c[nH]c2)=O)CCN(C(c2ncc(Br)cc2C)=O)CC1C(C)C 57572,c1(C(N2CCCC2C2(O)CNC2)=O)ccc(Cl)cc1Cn1ccnc1 57573,c1(C(=O)NC2(C)CCN(C(C(COC)(F)F)=O)C2)ccc2nnn(C)c2c1 57574,C(=O)(C(C)CC(=O)NCC(CO)NC(C1CN(C(C)=O)C1)=O)OC 57575,C1(C(N2C(CC=C)(C(=O)NCC(C)C(C)O)CCC2)=O)CN(C)CCN1C 57576,O=C1CCCC(C(N2CCC2C(=O)NCC=Cc2ccccc2)=O)C1 57577,N1(C(c2cc(OC)n[nH]2)=O)CC(C)CN(C(C2CC3(COC(=O)N3)C2)=O)C(C)C1 57578,CC1(CNC(=O)C2CC2)COCCN(C(=O)C2=NOC(CC3CCCCC3)C2)C1 57579,Cc1cnsc1C(=O)NCCC(O)CNC(C1C=CCCC1)=O 57580,C1(CCNC(C2CCOCC2)=O)CCN(C(=O)CC2CS(=O)(=O)C2)C1 57581,N1(C(COCCC)=O)CCN(C(=O)C(c2cccc([N+](=O)[O-])c2)C)CC(O)C1 57582,C1(C(=O)NC(CN(CC)CC)C)CCC2CCC1N2C(c1cncn(C)c1=O)=O 57583,C1(NC(c2nc(C(C)(C)C)oc2)=O)CC2CCCC(C1)N2C(=O)C(F)CC1CC1 57584,C1(CNC(c2ccc(CC(C)C)cc2)C)CC2(C1)CC(C#N)C2 57585,c1(N(C)C)ccccc1CC(=O)NC1CC1C(=O)Nc1ccsc1 57586,C1(N(C(=O)C(C(C)C)N(C)C)CC)CCCCN(C(c2ccc(C)c(F)c2)=O)C1 57587,N1(C(CC(C=C)CC)=O)CCC(C)(C)C(C(=O)NCCc2cnn(C)c2)C1 57588,N1(C(CCSCCCC)=O)CCC(C)C(N(C)C(c2sc(C)cc2C)=O)C1 57589,c1(C(=O)NCC(=C)CCNC(=O)C=Cc2cnccn2)nncc2c1CCCC2 57590,C1(C(=O)NC2C3CCN(C(c4ncc(N(C)C)nc4)=O)C32)OCCCC1(C)C 57591,C1(N(C(=O)Nc2c(C)cccc2)C)CCCN(C(C)C(N)=O)CC1 57592,C1(C(=O)NCC2(C)CCCN(C(CC3(C)CCCO3)=O)C2)CNc2ccnn2C1 57593,Cc1cc(C(C)(C)C(N2CC3CC3C2CNC(=O)CC2CC2)=O)ccc1Br 57594,C(=O)(C1c2c[nH]nc2CN1C(=O)C=CCN(C)C)NCCCN(C)C1CC1 57595,C(C)(CNC(=O)COCCC(C)C)(CNC(=O)CCc1nncs1)OC 57596,N1(C(C=C(C)Cl)=O)CCC(NC2CCCC2NC(=O)C(C)(C)CN(C)C)CC1 57597,c1(C(C(=O)NCCC2CC2)N(C2CCCS(=O)(=O)C2)C)ccn2ncnc2c1 57598,n1(CC(=O)NCC(CCCC)NC(CCSCC)=O)ncc(=O)c2ccccc12 57599,N1(C(C(CNC(C2(OC)CC(C)C2)=O)N(C)C)=O)CCc2ccc(C#N)cc21 57600,C1(CC)CCN(C(C2CN3CCC2C3)=O)C1CNC(=O)C(C1CC1)OC 57601,C1(NC(=O)Cc2cscn2)CCC2(CCN(C(=O)C3=CC4(CCOC4)C3)C2)C1 57602,CCC(C)(C)CC(=O)N1CCC(CO)C(NC(=O)COCc2cccc(Cl)c2)C1 57603,C1(NC(C(Cc2cn(C)nc2)O)=O)COCCN(C(=O)CN2CSCC2=O)C1 57604,c1(C(=O)NCC(CC)(C)C(=O)NCCn2ccccc2=O)cccc2ccnn12 57605,C(=O)(C(C)(C)c1ncco1)N1CC(CNC(C(C2CCC2)OC)=O)C1 57606,Cc1cc(CC(=O)NC2CN(C(=O)CCc3cncs3)CCC2CO)cc(F)c1 57607,C(CCN(C(=O)C(c1ccc(C)cc1)=O)C)(C(C)(C)C)NC(C(CC)COC)=O 57608,C1(COC)(NC(=O)C(n2nccc2C)C)CCN(C(=O)CSS(C)(=O)=O)CC1 57609,C1(C(N)=O)(OC)CN(C(=O)CNC(=O)OC(C2CCCCC2)c2ccco2)C1 57610,c1(NC2CCCN(C(c3ncncc3Cl)=O)C2)ccnc2ncnn12 57611,N1(C(CC2C(C)(C)CC2)=O)CC(CO)C2(C1)CN(C(=O)C(C)(C)c1ccsc1)C2 57612,N1(C(c2sc(C)c(C)c2C)=O)C2CCC1CC(F)(CNC(=O)Cc1ccco1)C2 57613,N1(Cc2ccc(C)cc2Br)C2CCC1CC(NC(c1c(C)ccnc1O)=O)C2 57614,C12(C(=O)NC3(CCO)CN(C(c4ccc(OC)cc4)=O)C3)CCCCC1C2(F)F 57615,CCCCC(C)CCC(=O)NCCCC1(NC(c2ccn(C)c(=O)c2)=O)CC1 57616,c1(CC)sc(C(=O)NC(C)(C)CN(C)C(c2ccccn2)=O)cc1C 57617,C=CC(C)(C)CCNC(C1(OC)CCN(C(=O)COCC(C)(C)C)C1)=O 57618,c1(OCC(=O)NC(CCNC(CC=CC=C)=O)(C)C)cc(F)cc(F)c1 57619,c1(C(c2n(C)ccn2)=O)ccc(NC(=O)CNC(=O)Cc2ccc(Br)s2)cc1 57620,N1(C(c2cnc(NC(C)=O)o2)=O)CC2(CC(NC(C3CCCN3C=O)=O)CO2)C1 57621,C12(NC(c3ccoc3)=O)CN(C(c3cnsn3)=O)CC1CS(=O)(=O)C2 57622,N1(C(CC2(OC)CC2)=O)CCN(C(C2CC2(C)C(F)F)=O)C(CC(C)(C)C)C1 57623,c1(C(=O)OC)sc(C(=O)N(C2CCN(C(C3(CCF)CC3)=O)C2)C)cc1N 57624,C1(CC(=O)NC2(CC=CCC(=O)NCC3CC(OC)C3)CCC2)CCN(C)CC1 57625,C1(Nc2cc(C)n(-c3c(C)cccc3)c2C)Cc2ccc(C#N)cc2C1 57626,N1(C(C2=CC(C)(CC)C2)=O)CCCC(C2CCN(C(=O)CNC(=O)OC)C2)C1 57627,CC(C(=O)N1CCCCC1CCN(C)C(C1(F)CCC1)=O)C(F)F 57628,C=CCC(C)(CC)C(=O)N1CCC(CNC(=O)CN2CCN(C)C(=O)C2)C(O)C1 57629,c1(C(=O)NC(CC)CN(C(=O)C(CSC)OC(C)C)C)cnncc1OC 57630,N1(C(COCCCCC)=O)CC(CNC(c2c[nH]nc2OC)=O)CC1COC 57631,N1(C(C(C(C)O)N(C)C)=O)CCC2(CC1)CC(NC(=O)Cc1cn[nH]c1)CCO2 57632,c1(C2N(C(C3CC(C(=O)OC)C3)=O)CCOC2)c(C)nn(C)c1C 57633,c1(OCCC)cccc(CN2CCNCC2C(=O)NCC)c1 57634,C(=O)(C(F)(F)C(F)F)NCC(N1CCN(C(C(C)=CC2CC2)=O)CC1)C(F)(F)F 57635,c1(C(N2CCC(O)(C(C)NC(C(CC)CC)=O)C2)=O)cc(C)c(C#N)cn1 57636,c1(COC)cncc(C(=O)N(C2CCCC(N(C(=O)CSCCOC)C)C2)C)c1 57637,C(C1c2ccsc2CCN1C(=O)C=Cc1ccccn1)NC(CCP(C)(C)=O)=O 57638,Cc1cnc(F)c(C(=O)Nc2snc(C)c2Cl)c1 57639,C(=O)(CCCC(C)(F)F)N(C1C(C)CN(C(C2CC(O)(C(F)(F)F)C2)=O)CC1)C 57640,C1(C)(C(=O)NCCC(CNC(c2ccc(CN(C)C)o2)=O)O)CC2CC2C1 57641,C1(NC(C2(COC)CC2)=O)CN(C(=O)CC2CCN(C)CC2)CCC1C(F)(F)F 57642,N1(C(c2ccc(CN(C)C)[nH]2)=O)CCCCC12CC(NC(C1CN(C)C1)=O)C2 57643,c1(CC(COC)C(=O)NC2CC(C(=O)OC(C)(C)C)C(O)C2)ccc(F)cc1F 57644,C#CCC(O)C(=O)NCC1C=CC(NC(c2conc2C(F)(F)F)=O)C1 57645,C1(CN(C(CCCOC)=O)C)CN(C(=O)COc2c(Cl)cccc2Cl)CC12CC2 57646,c1(N2CCCC(CNC(C=C(C)C3CC3)=O)C2)nc(C)nc2sc3c(c12)CCC3 57647,C1(CC(=O)NCCCCCNC(C2C(C)=CCS2)=O)C=CS(=O)(=O)C1 57648,C1(C(N2CC(NC(C3(CC=C)CCC3)=O)C2)=O)CC(=O)N(CCC)C1 57649,n1(CC(=O)NCC2CC(NC(c3cc(Cl)c(Cl)[nH]3)=O)C2)cnc2c1CCCC2 57650,C(N=c1[nH]c2c(c(=NCc3cccc(N)c3C)[nH]1)CCCC2)C1N(CC)CCC1 57651,C1(NC(C(C)CC2CC2)=O)C2CC3CN(C(c4ccc(N)cc4O)=O)C1C3C2 57652,N1(C(CS(=O)(=O)NC)=O)CCCCC1C1CCCN1C(=O)CN1CCCNC1=O 57653,C1(CCNC(C2CC2CF)=O)CCN(C(C2CCCC2c2nc(S)n[nH]2)=O)CC1 57654,C(=O)(C(CCN(C)C)NC(=O)C(C)C#N)N1CC(C(CC)CC)C1 57655,N1(C(c2c(OC)c(C)cs2)=O)CCN(C(c2cc(CO)[nH]n2)=O)CC1C1CC1 57656,c1(CC)c(C(=O)NCC2CC(C)(C)CN2C(=O)C(C)OCCC(C)C)cccc1C 57657,C(COC)(CC(=O)N1CC(c2cccc(C#N)c2)C1)NC(C(OCCOC)OC)=O 57658,CS(=O)CCC(O)C(=O)NCCCNC(=O)Cc1cccc(CC(F)(F)F)c1 57659,Cc1ccc(C2CCCN(C(=O)NCCNc3ccc(OC(F)F)cc3)C2)cc1 57660,N1(C(c2cncc(C(C)C)c2)=O)CCCOC(CNC(=O)C(O)C2CCCC2)C1 57661,Cc1cc(N(C2CCN(C(C)C)C2)C)nc(=NCCOc2c(F)cccc2Cl)[nH]1 57662,n1(CCC)cccc1C(N1C(C(=O)N(C)CCc2ncccn2)CC1C)=O 57663,CC(C)(CNC(N1CCOC(CCO)C1)=O)C(N)=O 57664,N1(C(C2CC(CNC(c3c(C(C)C)nco3)=O)C2)=O)CC2CC(C)C2C1 57665,Cn1nccc1CC(=O)NCC1CC1CNC(C1CCCCC1)=O 57666,N1(C(C=NOC)=O)CC2=C(C1)CN(C(=O)Cc1ccsc1C)C2 57667,C1(CNC(c2ncc(C)nc2)=O)CC2CCC1N(C(=O)CC1CC(C)(C)CO1)C2 57668,C1(c2nnnn2C)(NC(c2ccn(C)n2)CC)CCOC2(CCCC2)C1 57669,S(=O)(=O)(c1ccc(-c2ccccn2)s1)NCC1CC(C)NC1 57670,N1(C(C2CCCO2)=O)CCCC(C2CCCN(CC=C3CCCCC3)C2)C1 57671,C1(CN(C(=O)CN(C)C(=O)C2CC2)C)CN(C(=O)C=Cc2cccnc2)CCO1 57672,N1(C(c2c(C)[nH]cc2)=O)CCC(O)C(NC(=O)CSc2nnnn2C2CC2)C1 57673,CC1CN(C(c2cscc2C(F)F)=O)CCN1C(=O)CCSc1nnnn1C 57674,CC(C)(C)CC(O)CC(=O)N1CC(O)CC1CC(N1CCNC(=O)CC1)=O 57675,c1(N2CCCC(C)(C)CC2)nc(N2CCCOC(C(C)(C)C)C2)c2ncsc2n1 57676,C1(CNC(C(C(=C)Cl)(C)C)=O)C(C2CC2)CCN1C(=O)CCc1cnc(C)s1 57677,C1(C2(O)CN(C(c3ccc(CO)o3)=O)C2)(CNC(c2ccnnc2)=O)CC1 57678,N1(C(C(C)c2cccs2)=O)CC2CCC(NC(c3ccc(C#N)s3)=O)(C2)C1 57679,C12(C(=O)OC3CCC(c4n(C)ccn4)CC3)CCC(=O)N1CC1(CC1)C2 57680,c1(NCc2cn(CC)nc2C2CC2)ccc(Br)cc1C(C)(C)C 57681,C1(CN(C(c2ccon2)=O)CC)CCCN(C(=O)CN2CCC(C)(O)C2)C1 57682,C1(C(=O)NCC2C(NC(CC(C)C)=O)CCCC2)CS(=O)(=O)CC(=O)N1 57683,N1(OC(=O)CCNC(N(c2ncc(SC)s2)CC)=O)CCC2(CC1)OCC(O)C2O 57684,c1(CC)cc(C(N2CCC(O)(CN(C(=O)C(CO)N(C)C)C)C2)=O)c(C)o1 57685,Cc1c(Cl)c(C(=O)NC2CCCN(C(=O)C(c3ccccn3)O)CC2)nn1C 57686,N1(CCC(=O)NCCN(C(CC2C(C)C2)=O)C)CCOC1=O 57687,C12(CNC(=O)OC(C)(C)C)CC(CO)(CCO1)C2.c1(C=O)cnccc1C(=O)O 57688,Cc1cc(O)nc(CNC(C2CCCC2C(C)C)=O)n1 57689,S(=O)(=O)(c1ccc(-c2cccc(C(F)F)c2)cc1)NC1CCC(=O)NC1 57690,O=C(CC1NC(=O)c2ccccc21)NCC1CCN(C(c2coc(O)n2)=O)C1 57691,N1(C(CSCC#C)=O)CCc2ccccc2C(NC(C2CCC(F)C2)=O)C1 57692,CCCC(C)CC(=O)NC12CN(C(c3cccc(OC)c3N)=O)C(COC)(C1)C2 57693,C1(C(=O)NC2C=CCN(C(C(n3cc(C)nc3)(C)C)=O)C2)CC2CCCC2C1 57694,N1(C(CS(CC)=O)=O)CCC2CN(C(=O)CC(=O)N(C)C)C(C)C12 57695,c1(C(C)NC(c2ccc(-n3c(C)cc(C)n3)cc2)=O)nc2ccccc2[nH]1 57696,C1(CCC(=O)N(CCC#N)Cc2cscc2Br)CCc2ccccc2C1 57697,c1(C(C)SCC)nc(COC2CCCN2C2CCCC2)n(-c2ccnnc2)n1 57698,CCCC(C)=CC(=O)N(CCCNC(=O)CSC(F)(F)F)CC 57699,C1(C(N(C)CCC(=O)N)=O)CCS(=O)(=O)N1.C(=O)(CCNC(N)=O)OCCCO 57700,C1(NC(CSCCC(C)C)=O)CC2(CCN(C(C3CCC(C)S3)=O)CC2)C1 57701,N1(C(=O)NC(C)Cc2cccnc2)CCc2ccn(C(=O)OC(C)(C)C)c2C1 57702,N1(C(c2csc3nccn23)=O)CCC2(CCCN2C(c2cc(O)cs2)=O)C1 57703,C1(NC(c2c(C)sc(Cl)n2)=O)CCN(C(c2nccnc2Cl)=O)C12CCC2 57704,c1(CCC(c2n(CCC)nnn2)NC2C3COCC23)ccccc1Br 57705,c1(C(=O)NCC2CC(NC(c3c(CC)ccs3)=O)C2)ccnc(C)c1 57706,Cc1ccc(Br)c(C(=O)NC2CCCCC2NC(C2CN(C)C2)=O)n1 57707,CN1CC2CC2(CNc2cccc(COc3ccc(F)cc3F)c2)S1(=O)=O 57708,C(=O)(C(C)(F)C(=O)NCC1CC(O)CN1C(C1(Oc2cnn(C)c2)CC1)=O)OC 57709,C(CCCCCCC(=O)NCC(C)(CO)c1ccccc1)NC(C)=O 57710,Cc1ccnc(C(=O)NCC#CCNC(C2CCCN(CC(F)(F)F)C2)=O)c1 57711,N1(C(C2C(C(C)(C)C)CC2)=O)CCC(N(C(=O)CCCc2ccccn2)CCO)C1 57712,N1(C(c2c(CC)n(CC)nc2)=O)CC2(CCC2)CC1CNC(C1OCC1(C)C)=O 57713,CCCC(C)CCCC(=O)NC1(CCOC)CCN(C(=O)CSc2cccs2)C1 57714,CC#CCC(C(=O)NC1CC2CC(O)C1C2)NC(c1ccnc(C)c1)=O 57715,N1(C(CNC(=O)OC)=O)CCCC1C(C)NC(=O)CCc1cncn1C 57716,C(=O)(C(C(=O)OCC)C(C)(C)C)NC1(C)CCN(C(c2ccn(CC)n2)=O)CC1 57717,CC1CN(c2nnc(Cc3ccccc3)n2CC2CN(C)CCCN2)CC(C)O1 57718,c1(C(=O)NC2C(C)CN(C(=O)C3=CCCO3)CC2)cnn2c1CC(C)CC2 57719,C12(C(N3CC(NC(=O)COc4nc(O)nc(O)n4)C3)=O)CCCCC1OCC2 57720,c1(C(=O)NCCCC(C)NC(C(C(C)(C)C)SC)=O)cc([N+](=O)[O-])ccc1C 57721,c1(C(=O)NC2CN(C(=O)Cc3ccoc3)CC2O)cnc2ccccc2c1 57722,Cc1c(C(=O)NCC(F)CNC(=O)C(c2ccn(C)c2)C)cnn1CC(F)F 57723,N#Cc1cc(CN2CCC(C(=O)Nc3cc(F)c(Cl)cn3)CC2)ccc1O 57724,C1(CC(=O)NCCCC2(NC(C3C(C)C3)=O)CC2)COC2CC1C2 57725,Cc1ccc2c(=NCC(=O)N=S(C)(C)=O)[nH]c(=NCc3cccc(Cl)c3)[nH]c2c1 57726,n1(CC)cc(C(N2CCC(C(C)(C)NC(c3cc(C)cn3C)=O)C2)=O)c(C)n1 57727,N1(C(c2c(C)cc(Cl)cc2)=O)CC(C)(C)OC2(C1)CN(C(c1cocc1C)=O)C2 57728,C(=O)(CCCCCC#N)NCc1cc(C(=O)NC(CC(=O)OCC)C)ncc1 57729,N1(C(c2cccc(COC)c2)=O)CCC(C2CCN(C(=O)C=C3CCC3)C2)CC1 57730,C1(NC(=O)C=C2CCSCC2)CC2CN(C(c3ncc(F)cc3F)=O)CC12 57731,C1(NC(C(N2CCC(O)CC2)C)=O)CCN(C(C2CC(C)(C(C)(C)C)C2)=O)CC1 57732,C(=O)(C(F)CC(C)(C)NC(=O)Cn1cccn1)N1CC(C#C)C(OC)C1 57733,Cc1cccc2cc(C(=O)NCC3CN(C(=O)COCC(F)F)CCC3C)oc12 57734,C(CCCCCC(=O)N1CCC(NC(C2CC(OC(F)(F)F)C2)=O)C(O)C1)SC 57735,c1(COCC(=O)NC2CC(C)(NC(C3C(C)CC3)=O)C2)ccccc1 57736,n1(CCC(N2CCCC(CNC(C(F)=C(C)C)=O)C2)=O)cnc2c(N)ncnc12 57737,CC1(C(=O)NC2CCCC2CNC(=O)CC2(O)CCC2)C=CCCC1 57738,c1(C(N(CCN(C(=O)Cc2cc(C(C)C)no2)CC)CC)=O)cncc(C)n1 57739,CCC(C)C(C(=O)N1CCC=CC1C(=O)NCCOCCN=[N+]=[N-])OC 57740,N1(C(C=CCC)=O)CC2CCCC(NC(C3C4CC5C(C4)C35)=O)C2C1 57741,CC(CS(C)=O)C(=O)N1CC(CCNC(=O)CC2=CCCC2)C1 57742,C1(N(C(C(C)(C)C)=O)CCF)CCCN(C(=O)CCOC(C)=O)C1.C(C(F)(F)F)O 57743,CC1(C)CCc2sc(C(c3nnnn3C3CC3)NCCC3CCOCC3)cc2C1 57744,CC(C)(CNC(C1CCNC1=O)=O)CC(=O)N1CCC1CN=[N+]=[N-] 57745,C(=O)(C1=CCOC1)N1CC(O)(CNC(CC(c2ccc(Cl)cc2)N(C)C)=O)C1 57746,C1(N(C(C2(CSC)CC2)=O)C)CCC(NC(=O)CN2CCOCC2)C1 57747,C1(C(=O)NCC(C(C)O)C)CCOCCN1C(C1CCC(O)CC1)=O 57748,N1(C(C2(C)CCCCC2)=O)CC(NC(=O)CC2CC2)C(C2CC2)C1 57749,CCCCCCC(C)CC(=O)NC1(COC)CN(C(c2c[nH]nc2[N+](=O)[O-])=O)C1 57750,c1(C(=O)NC2CC(NC(C(c3cccs3)SC)=O)C2)cc(-c2cccnc2)[nH]n1 57751,C(=O)(CCCC(=O)OCc1csc(C(N2CCC(OC)C2)=O)c1)OC 57752,CC(C)CC(C(=O)NC(CNC(=O)Cc1nccn1C)C1CCC1)n1ccnc1 57753,C(C(C)(C)C(C)C)N(CC(C)C(=O)OCC)C(CN(CCOC)C1CC1)=O 57754,C1(NC(=O)CN2C(=O)CCC2=O)CCN(C(=O)Cc2ccc(F)c(F)c2)CC1F 57755,c1(C2(C(N3CC(C)(NC(c4c(Cl)cn(C)n4)=O)C3)=O)CCC2)ccccc1C#N 57756,C1(OC)CCCC1C(=O)N(C(C)CCNC(c1cn(C)cn1)=O)C 57757,C(C(CO)CC(C)C)NC(C1(CCNC(C(C)=C2CC2)=O)CCC1)=O 57758,N1(C(c2c(CNC(c3nc(CCC)oc3)=O)c[nH]n2)=O)CC(O)CC1C1CC1 57759,c1(OC)cnc(C(=O)NC(C)(CNC(C2CCCC2O)=O)Cn2cccn2)cn1 57760,C1(NC(c2c(C)coc2)=O)CCCC(CN(C)C(c2nn(C)cc2Cl)=O)C1 57761,C(=O)(C1CCCc2cc(C#N)ccc21)NCCN(C(C(CN(CC)CC)F)=O)C 57762,C=CC(C)CN=C(NCC1CCCO1)NCC1(C(C)(F)F)CCOCC1 57763,Cc1c(C(=O)NCC#CCNC(c2[nH]c3ccccc3c2Cl)=O)nc2sccn12 57764,N1(C(=O)Cc2cccc(O)c2)CC2CN(C(=O)C=Cc3cnccn3)C2C1 57765,C(CCC(O)CO)N(C(=O)CCn1cc(CCN2CCNC(=O)C2)nn1)C 57766,C1(CNC(C(c2ccc(C)s2)C)=O)CN(C(=O)CCc2cncc(F)c2)CC1C 57767,c1(C(=O)NC2CN(C(c3ccc(C(=O)OC)[nH]3)=O)C3C2C3)ccccc1[N+](=O)[O-] 57768,c1(NCC2CC(O)(CNC(c3c(CC)scn3)=O)C2)cc(C)nc2ncnn12 57769,c1(OC)cc(F)c(F)cc1C(=O)N(CCNC(=O)Cc1cnn(CC)c1)C(C)C 57770,C1(OC)CN(C)C(C)(C(=O)N(CCCNC(c2ccoc2CC(N)=O)=O)C)C1 57771,C#CCC(CCOC)NC(C1COCCN1C(=O)CCS)=O.NCC 57772,CC1Oc2c(C(N3CC4(CCC4NC(=O)COCCF)C3)=O)cccc2NC1=O 57773,C1(N(CCCCCC)C(=O)CN(c2ccncc2)CC)CCS(=O)(=O)C1.C(=O)(CC)O 57774,c1(SCCC(=O)N(C(C)CN(C(=O)Cc2ccoc2)C)C)ccccn1 57775,c1(CNC(C2CCN(C(=O)OC(C)(C)C)C2)C)ccc(Cl)cc1C(F)(F)F 57776,N(C1CCCOc2c(F)cccc21)C(c1ccc(SC(F)(F)F)c(F)c1)=O 57777,C(=O)(C(O)CCCNC(c1c[nH]c(=NC)s1)=O)N(CC=C)CCOC 57778,c1(OC)ccc2ccccc2c1CC(=O)NCC1CN(C(c2csc(Br)n2)=O)C1 57779,C1(C2CCCC2)(C(N2CC3(CC(NC(C4CCOC4C4CC4)=O)C3)C2)=O)CCC1 57780,CC1(C)CC1(c1cn(CCC(F)(F)Cl)nn1)C(=O)O.C1(=O)CSCCN1 57781,c1(NC2C3N(C(c4cc(C(C)C)[nH]n4)=O)CC(CC3)C2)ncc(Cl)cc1[N+](=O)[O-] 57782,N1(CC(C)NC(=O)C(C2CCN(C(c3cc(O)cs3)=O)C2)F)CCCCC1 57783,N1(C(C2C(=C)C2)=O)CCC(C)C(NC(c2cc(C3(O)COC3)on2)=O)C1C 57784,c1(CN2C(C(=O)NCc3nc(Cl)ccc3F)CC(O)C2)ccn2ccnc2c1 57785,N#Cc1cncc(OCC(O)CNC(C2CCCCC2c2ccccc2)=O)c1 57786,Cc1cc(C)c(C(=O)N(C)CC2CCCCN2C(=O)C2=CC(C)C2)cn1 57787,C1(C(N(C)CC2CCCN(C(C3(CO)CCC3)=O)C2)=O)CC2(CCOCC2)CO1 57788,C12(NC(CCCn3cc(C(C)(C)NC(C)C)nn3)=O)CC3CC(C1)CC(C)(C3)C2 57789,c1(CC)ccc(N)c(C(=O)NC23CCC(NC(C4CCCO4)=O)(CC2)C3)c1 57790,N1(C(C)COC2CCCCC2)CCCC(NC2CC2)C1 57791,N1(C(c2c(C)nc[nH]2)=O)CC(C)CCC1CNC(=O)COc1ccsn1 57792,N1(C(c2c(C)nsc2)=O)CCC(CNC(=O)CC=Cc2ccccc2)C12CCC2 57793,C#CCC(O)C(=O)N1CCC(C(=O)NCc2cnn(CC#C)c2C2CC2)C1 57794,S(=O)(=O)(c1ccc2c(c1)CCCO2)NCc1c(COC)cccc1 57795,N1(C(c2c(C)nns2)=O)CC2C(CNC(c3ccc(CN(C)C)o3)=O)C2C1 57796,C1(=O)C(C(C)(C)C)N1.N1(CCC)CCCCC1C(=O)N(C)CCN(C)C1CC1 57797,c1(C(N2CCC(S(N)(=O)=O)C2)C(=O)NCC(C)C)noc2c(Cl)cccc12 57798,N12CC3CC1(C3)C2.c1(C(C)NCC2CC(CN=[N+]=[N-])C2)csnn1 57799,c1(C(N(C2CCN(C(=O)C=C(C)C3CC3)C2)CC)=O)ccc(S(N)(=O)=O)c(C)c1 57800,CC1ON=C(C(=O)N2CC(CNC(=O)CN3CCCCCCC3=O)C(O)C2)C1C 57801,c1(C(N2CC(C)(C)C(NC(=O)C(F)C(C)(C)O)C2)=O)cccc2c1CNC2=O 57802,CCCCC(C)C(=O)NC(CNC(C1(CSC)CC(F)(F)C1)=O)CC 57803,CCC(C)C(O)C(=O)NCC1CC2CN(C(c3cc(N)ccc3Br)=O)CC12 57804,C(=O)(C(C)C(C)C(C)(C)C)N(CC)CC1CCN(C(c2ccc(C)n2C)=O)CC1 57805,C(=O)(C1CC=Cc2ccccc21)N1CCC(C)C(NC(C2CC(C)(F)C2)=O)C1 57806,C(CCC(C)C)(C(=O)N(C)Cc1cc(C)cs1)NC(C(C=C)C)=O 57807,N1(C(c2c(CC)onc2)=O)CCC(NC(=O)C=NOC)C(F)C1 57808,C(=O)(C(CC(C)C)NC(C1CC2CCC1N2C(C)=O)=O)NCCOC 57809,c1(C(N2C(C(C)NC(C=C(C)Cl)=O)CCC2)=O)cnc(C)cn1 57810,c1(-c2nn(C(C)C)c(CCCCN(C)C)n2)ccc(OC(F)(F)F)cc1Cl 57811,c1(C(N(CCNC(CC(C)OC)=O)C)=O)cc2cc(Cl)sc2[nH]1 57812,C(CCC(C)(C)C(=O)NC1CCn2nnnc2C1)NC(C(COC)C)=O 57813,c1(C(N2CC(OC)C(NC(=O)C3=CC(C)CC3)C2)=O)ccc(C(F)(F)F)c(N)c1 57814,C1(NC(CN(C)CC)=O)CCCC1(C)CNC(=O)Cn1cc(C(F)F)cn1 57815,C(=O)(C(COC)CC(C)C)NCC1(F)CC(CNC(C(CC)N(C)C)=O)C1 57816,CC1CC(NC(c2cc3n(n2)CCO3)=O)CCN1C(c1cc[n+]([O-])cc1)=O 57817,c1(OCC)ccccc1OCCNCC1COCC1(C)C 57818,N1(C(C(C)NC(C)(C)C)=O)CCCC1CCCNC(=O)Cn1cc(Br)cn1 57819,C1(NC(CN(C2CC2)CC)=O)CN(C(C2(c3ccsc3)CC2)=O)CC1C1CC1 57820,C12(NC(c3ccc(=O)n(CCF)n3)=O)CCCC1N(c1ncc(Br)cn1)CC2 57821,c1(C(N(C(CNC(c2cc(C)cc(F)c2)=O)C)C)=O)cc(Br)cc(C)c1C 57822,CC(C)CC(C)(CNC(C1CC1C)=O)NC(c1cc(CC2CCC2)c[nH]1)=O 57823,c1(N(CC=C)CCF)[nH]c(=NC2CC(N3CCC3)C2)nc2scnc12 57824,c1(C(C(=O)NC(CC)(C)C)N(C)C(C2CCCO2)C)ccc(-c2cnn(C)c2)o1 57825,N1(C(C2(CC)CCCCC2)=O)CCCCC(CNC(c2nccc(Cl)c2C)=O)C1 57826,C1(CNC(=O)CCOCC2CCCO2)CCN(C(C2CC(=C(F)F)C2)=O)CC1 57827,C(CN=c1ncc(F)c[nH]1)C1CCC(NC(c2cc3ccsc3s2)=O)C1 57828,CC1(C)CC(C(=O)NC(C)(C)CCCNC(=O)CCc2nc[nH]n2)=NO1 57829,C1(CN(C(c2c(COC)noc2)=O)C)CCCC(NC(C2CCC2)=O)C1 57830,C12(NC(CC(=C=C)C)=O)CCCCCC1N(C(C1CC3(C1)CS(=O)(=O)C3)=O)CC2 57831,C1(CCC)CN(C(C2CC2[N+](=O)[O-])=O)CCN1C(=O)COCc1cccc(C)c1 57832,c1(C(N2CC(C(C(N3CC(COC(C)=O)C3)=O)O)C2)=O)csc(C)n1 57833,N#CC1(C(=O)NCC2CC(F)(CNC(=O)Cc3ccsc3Cl)C2)CCC1 57834,c1(C(=O)NCC(CC=C)NC(=O)Cc2c(C)cnn2C)ccc2c(c1)CCC2=O 57835,C1(NC(C(CO)OC)=O)CN(C(c2oncc2C)=O)C2CCCC12 57836,c1(C(=O)NCC(C)N(C(CC(C(=C)C)O)=O)C)ccc2c(c1)NCCC2 57837,C(C(CC(C)C)C(=O)NC1CN(C(=O)CCOC2CCC2)CC12CC2)OC 57838,N1(C(C2OCCC2NC(C2(n3nccn3)CC2)=O)=O)CC2CC3CC2C1C3 57839,C(=O)(CC(C)C(=O)NCC(C)CC(=O)NC(c1cncn1C)CO)OC 57840,C1(NC(c2c(C)noc2)=O)CN(C(=O)C=C2CCCCC2)C2CCCC12 57841,c1(OC)c[nH]c(C(N2CCN(C)CC2CNC(=O)CC2CCC(=O)O2)=O)cc1=O 57842,Cc1[nH]c(=NC(C)c2nccs2)sc1S(N)(=O)=O 57843,c1(C(N2C3(CNC(C=COCC)=O)CC(C2)C3)=O)c(C)cc(Br)cc1Cl 57844,CC(CO)(C(F)F)NC(=O)CC1CC1CNC(=O)C(N)=O 57845,C1(C(N(CC(C)CNC(=O)CC2(C)CCC2)C)=O)OCCN(C)C1=O 57846,c1(C(=O)NC2(C(=O)NCC(C)CN(C)C)CCCOC2)cc(O)cc(F)c1F 57847,C1(NC(c2n(C)ccc2)=O)CC(NC(c2ccc(-c3cccs3)[nH]2)=O)C(O)C1 57848,N1(C(CN(C)C(c2cnns2)=O)=O)CCN(C(=O)C(C)(C)CC2CC2)CC1 57849,Cc1ccc2[nH]c(=NCC3CC4(CC(NC(=O)CC5CCC6CC56)C4)C3)sc2n1 57850,C(CC(O)CO)NC(C(c1ccccc1)NC(CCOC(C)=O)=O)=O 57851,CCC(N=c1cccc(S(=O)(=O)NC(CC2CC2)CO)[nH]1)c1cc(C)ccc1C 57852,C(=O)(C(C(C)C)OCC)N(CCNC(CC=CC)=O)CCC 57853,CC12CC1CCN2c1nnc(-c2ccccn2)o1 57854,N1(C(C(CC=C)C)=O)CCC2(CNC(c3c(F)cc(F)cc3F)=O)CCCCC12 57855,n1(CC(=O)NC2CC(O)(CSC)C2)nc(C)cc1C.C1(c2cccs2)C(=O)N1 57856,CCC(C)(CNC(C1CN2CCC1C2)=O)C(=O)N1CCC(OC(C)(C)C)C1 57857,C(c1ccc(O)cc1)=CC(=O)NCC1CCC(NC(C(C2CCCC2)OC)=O)C1 57858,c1(C(=O)NC2CN(C(C=Cc3ncc(C)[nH]3)=O)C(C)C2)cnc2ccccc2c1 57859,c1(NC2(C(=O)NC(CCCNC(C3C(OC)CC3)=O)C)CC2)ccc(C)c(C)c1 57860,C#CC1(C(=O)NC2COCC2CN(C)C)CCN(C(=O)C(n2cc(C)cn2)C)C1 57861,N1(C(CC(C)C2CC2)=O)CCCC(C)(NC(c2ccc(CO)cn2)=O)C1 57862,c1(C(=O)NC23CCCC(NC(c4n(CC)nnc4)=O)(C2)C3)csc2ccccc12 57863,C1(CNC(CNS(NC)(=O)=O)=O)CN(C(=O)CN2CCCC2CO)CCO1 57864,N1(C(C(C)=O)=O)CCCCC(Cn2cc(-c3ccc(N)c(F)c3)nn2)C1 57865,N1(C(c2c(C)c(N)ccc2)=O)CCC(C2CCCN(C(c3occc3Br)=O)C2)C1 57866,CC(C(C)(C)O)N(C)C(c1nc(Cn2cc(Br)cn2)cs1)=O 57867,C1(OCC=C)CCN(C(=O)CC2CC(NC(=O)C(F)F)C2)C1 57868,c1(C(=O)NC2C(CNC(C3N(C)C(=O)CCC3)=O)C2)cc(F)c2ccccc2c1 57869,c1(C(=O)NC2CC2)ccnc(-n2cc(C3CC34CCC4)nn2)c1 57870,N1(CC)CCCCC1C(=O)NC1CC(CC(=O)NCC2CC(=O)N(CC)C2)C1 57871,c1(C(N(C)CC2CCCN(C(COCCCC#C)=O)C2)=O)cc(F)c(F)cc1O 57872,N1(C(C2ON=C(CC)C2)=O)CCN(C(c2cc(Cl)no2)=O)CC1C(C)(C)C 57873,N1(C(c2ccc(=N)[nH]c2)=O)CCC(F)(CNC(=O)CC2CNC(=O)C2)CC1 57874,c1(C(=O)NCC(CNC(c2cc(C)c(C)nc2)=O)CO)ccc2cn(C)nc2c1 57875,CC1CN(Cc2cn(CC(F)CCNC(=O)CC=C(Cl)Cl)nn2)CCO1 57876,C(=O)(C1=CCCC1(C)C)N1CCCC(N(C(c2cnn(C(F)F)c2)=O)CC)C1 57877,C1(CCNC(C(C)=CC)=O)CCCN(C(=O)CC2CC2)C1.C1(N)CC(N(C)C)C1 57878,c1(NC(c2cncc(-c3cc(C)cc(F)c3)n2)=O)cc2nc[nH]c2nc1C 57879,c1(C(C)C(N2CCC(c3cn(CCCCC(=O)O)nn3)CC2)=O)cccc(C#N)c1 57880,c1(C(N2C(C(=O)Nc3cc(SC)n[nH]3)CSCC2)=O)cc(Cl)nc(Cl)c1F 57881,CC1(C(=O)NC(CNC(C2CCCCN2C2CCCC2)=O)CO)CCCCO1 57882,Cc1nc(N2CCC3CC(NC(C4CC4(F)F)=O)CCC3C2)ncc1[N+](=O)[O-] 57883,Cc1nc(=O)n(C2CCN(C(C3CCN(C4CCSCC4)CC3)=O)CC2)[nH]1 57884,C1(C(N2CCC(C(=O)NCC(c3cnn(C)c3)C)CC2)=O)C2CC3C(C2=O)C13 57885,C1(CC=C)(C(N2CCC(C)(N(C)C)C2)=O)CCN(C(=O)CN2CCN(C)CC2)C1 57886,C1(C(N(C2CN(C(=O)C=Cc3cnn(C)c3)CC2C(F)F)C)=O)C(C#N)C1(C)C 57887,C=C=CCCC(=O)N(C)CCOCCC(N1CCCCC1C(C)(C)O)=O 57888,c1(C(C)C)ccc(C(=O)NCCCC(C)NC(=O)CCOCC2(F)CC2)s1.C1CC1 57889,n1(C2(C(=O)NCC3CCOC3)CC2)ccc(C2CC2)n1.C12CC(C1)NC2=O 57890,c1(Sc2ccc(C(=O)OC(CNC(C(=O)OC)CO)(C)C)o2)ccc(C#N)cc1 57891,C(=O)(CCCCC(F)F)NCCC(C)N(C(C(C)Cc1ccc(Cl)cc1Cl)=O)C 57892,c1(N(CC(C)SC)C)ncc(C)cc1S(=O)(=O)N1CCCC(CCO)CC1 57893,c1(C(=O)NCCCC(C)C)coc2c1CN(C(c1cc3n(n1)CCO3)=O)C2 57894,c1(C(=O)NC2CCC(CNC(c3c(C)ncs3)=O)C2)cc(F)cnc1O 57895,N1(C(C2(NC(c3nccc(C)c3N)=O)CCCC2C)=O)CCCC2CCCCC12 57896,Cc1cc(C(=O)NCC2CC2CNC(c2ccsc2)=O)c(C)s1 57897,C1(CNC(C2(CF)CCC(=O)C2)=O)CC(C(=O)N2CCC2)=NO1 57898,c1(CN(C(C2C(NC(C(C)=C(CC)C)=O)COC2)=O)C)cccnc1O 57899,n1(CC=C)nnnc1C(C=CC=C)NCC.C12CCC(C1)C(=O)OC2=O 57900,c1(CC)onc(C(=O)NC2CCOCC2NC(=O)CC(C)n2ccnc2)c1C 57901,CCC(C)(C(=O)NCc1ccccc1CN(C(=O)C(C)C(=O)OC)C)C(N)=O 57902,c1(CCC(=O)NCC2CC2NC(C23CCCC2C3)=O)cccc(Br)c1F 57903,Cc1nc(-c2ccc(Cl)s2)sc1CN(C(=O)NC)CCc1ccccc1Br 57904,C(=O)(CC1=CCCC1)NC1C(NC(C(N2CCC(O)CC2)C)=O)C1 57905,N1(C(Cc2ccn(C)n2)=O)C(C(=O)Nc2nc3c(s2)CCC3)C2CC(F)C1C2 57906,N1(C(=O)OC(C)(C)C)CCCC(NC(C2CCC(=O)N(C3CC3)C2)=O)CC1 57907,Cc1cnsc1C(N1CCC1CNC(=O)CCNC(c1cnccn1)=O)=O 57908,N1(C(C(=O)N(CCC#C)CC)C)CC2CCC1C1CN(C(=O)CCCOC)CC21 57909,N1(C(C=CC(C)(C)C)=O)CCN(C(=O)COc2ccc(F)c(Cl)c2)C2CCC12 57910,CP(C)(=O)CCC(=O)N1CCCCC1C1(NC(c2[nH]ccc2C2CC2)=O)CC1 57911,C1(CC(N2CCC(C)(CCC)C2)=O)CC(C)(C)CN1C(=O)CC(C)(C)C 57912,C(=O)(C1CC(=O)c2ccccc21)NCC1CN(C(c2ccc(C)o2)=O)C(C)CC1 57913,c1(C(=O)NCC(C)NC(C2C(C)C2C)=O)cc(S(=O)(=O)NCc2ccco2)c[nH]1 57914,Cc1[nH]nc2ncc(C(N3CCN(C(=O)C(CO)NC(N)=O)C(C)C3)=O)cc12 57915,c1(NC(C2C(NCc3cc(C)sc3C)CCCC2)=O)c(C)ccc2n[nH]cc12 57916,N1(C(c2n(C=C)nnc2)=O)CC(C)CN(C(=O)C=Cc2cn(C)nn2)C(C)C1 57917,c1(C(=O)NC(C)CCCCNC(c2cccc(CO)n2)=O)cc(Cl)c([N+](=O)[O-])[nH]1 57918,c1(SCCC(=O)NC(C)CCN(C(=O)CCc2cnn[nH]2)C)ccc(F)cc1 57919,c1(C(N2CCC(NC(CSC(C)C)=O)C(F)C2)=O)ccc(Cl)c2ccccc12 57920,CC1C(N(C(=O)CCC2CCC(NC(c3cc(C#N)cs3)=O)C2)C)CCCC1C 57921,c1(N2CCC(C(N3CC(S(C)=O)C3)=O)CC2)cc2ccccc2s1 57922,Cc1ccc(C(N2CCOCC2CCNC(=O)CCC(C)(F)F)=O)c(C)n1 57923,c1(OCC)cnc(C(=O)NC(C2(O)CCN(C(=O)Cc3ncc(C)o3)C2)C)cn1 57924,N1(C(C(C)(C2CCC2)NC(C2CCOC2=O)=O)=O)CCC2(CC1)N=N2 57925,c1(C(=O)NCCCNC(c2ccc(N)c(F)c2)=O)ccc2c(c1)S(=O)(=O)NC2 57926,c1(C(N2C(CNC(CC3(C=C)CC3)=O)C(C)CC2)=O)cnc(OC)nc1C 57927,N(C1c2ccccc2CC1NC(=O)C(C)N(C)C)C(c1n(C(CC)C)ncc1)=O 57928,N1(C(CC(CC)CC)=O)CC2CCC1CN2C(=O)C(C(C)(C)C)c1cc[nH]n1 57929,C=CC1(CC(N2CCC(C(C)C)(CO)C2)=O)CN(C(c2ccncc2NC)=O)C1 57930,C(CO)(CN=c1cc(NCCCN2CCC(CO)CC2)nc[nH]1)OC 57931,C1(C2CCN(C(c3cc(N)cnc3Cl)=O)C2)(NC(CC2C(C)C2)=O)CC1 57932,C1(CC(N2CC3C(NC(c4ccc(C(N)=O)[nH]4)=O)C3C2)=O)CCCC2(CC2)C1 57933,c1(C(=O)NCC2COCC2NC(C2CC2(Cl)Cl)=O)cc2c(nc1O)CCCC2 57934,C(=O)(C(CCC)S(N)(=O)=O)NCCCN(C1CCCC1)C(CC1CC(=C)C1)=O 57935,C1(CC(=O)NCC=CC(=O)NCC2(OC)CCOC2)CCCCC1O 57936,C1(NC(C2(NC(C)C)CC2)=O)CCC(CNC(C2(F)CCOC2)=O)CC1 57937,Clc1ccc(-c2noc(-c3noc(C4CCC45CCC5)n3)n2)cc1 57938,N1(C(C2CC3(CC(NC(C4C5CCC(=O)C45)=O)C3)C2)=O)CCC2(CCCC2)CC1 57939,c1(C(=O)NCC2(F)CC(NC(=O)CC3CC34CC4)C2)nn2cccnc2c1Cl 57940,c1(C(=O)NCC23C(CN(C(C(C)CC(N)=O)=O)C2)C3)ccc(Cl)c(O)c1N 57941,N1(C(c2ccc(C)nn2)=O)CCN(C(=O)C(C(C)(C)C)n2ccnn2)CC1C 57942,c1(OC)cc(F)c(F)cc1C(N1CCC(CN(C)C(c2cnc(C)n2C)=O)C1)=O 57943,c1(C(=O)NCCc2cc(OC)cc(C)n2)cnn2ncccc12 57944,C12(NC(=O)Cn3cccn3)CCCC1N(C(c1ncccc1O)=O)CC2 57945,c1(C(=O)NCC(C)NC(=O)CCc2cnn(C)n2)cccc2c1OC(C)C(=O)N2 57946,C(C(CC)(CC)C(=O)NCCCCCCOC)NC(C(C)SCC)=O 57947,c1(NC(C)=O)cccnc1C(=O)NCC1CC1CNC(=O)CCn1ccnc1C 57948,N1(C(C2(S(N)(=O)=O)CC2)=O)CCCC(C2(NC(=O)CC(O)C3CC3)CC2)C1 57949,c1(C(=O)NC2C(NC(c3ccc(C)c(F)c3)=O)COC2)cccc2c1OCCC2 57950,N1(C(C2N(C(C)=O)CCC2)=O)CC23CCCC2(C1)CN(C(=O)C(C)S(N)(=O)=O)C3 57951,C#CCC(O)C(=O)N1CCCC(OCc2cn(-c3nc(C)ccn3)nn2)C1 57952,N1(C(CN(C(=O)OC(C)(C)C)CC2CC2)=O)C2CSCC1C2 57953,n1(CC)c(C(C)OC(C(C)NCC(CC(C)C)OC)=O)nc2ccccc12 57954,C1(NC(CC2C(C)CC2)=O)CC2CC(NC(c3cnn(C)c3C(F)F)=O)CC12 57955,N1(C(CC2CC(CC)C2)=O)CC=C(CNC(C2CC23CCCCC3)=O)CC1 57956,c1(C(C(=O)NCC(c2c(C)cccc2)C)(C)C)ccc([N+](=O)[O-])cc1F 57957,C(C)(C(C(=O)NCC=CC(C)(C)C)NC(c1cc(CO)n(C)n1)=O)OC 57958,c1(C(N2C(C(N3CCOC(CCO)C3)=O)CC2)=O)cncc(C(F)F)c1 57959,C1(C(=O)NCC(C)NC(C2CC(O)C2)=O)CCCC1O 57960,C1(C(C(=O)NC(C)(C)C)N(C)CC2(CC(C)C)CC2)CC(C)CC(C)C1 57961,N1(COC)CC2(C1)CN(c1nc(CC3CC3)n(-c3cnc4sccn34)n1)CC2CO 57962,n1(CC)nc(C)c(COC(c2ccc(N3CCCC3)nc2Cl)=O)c1C 57963,c1(CSC)ccc(C(CCCCSC)OC)cc1[N+](=O)[O-].N12CCCC(CC1)C2 57964,CC1(CNC(C2CCC(=O)N2)=O)CCC(NC(=O)Cc2ccc(F)cc2)CC1 57965,c1(C(N(CCN(C(c2n(CC)ncc2)=O)C(C)C)C)=O)cnnc(Cl)c1 57966,Cc1ccc2c(CC(=O)NC3(C)CCN(C(=O)C4=CCCCO4)C3)coc2c1 57967,CC1(C)C(NC(C2(c3cccs3)CC2)=O)CC1CNC(=O)Cc1nnc(O)s1 57968,Cc1cnccc1CCNC(=O)CC1CCCN(C(c2cnn(C)n2)=O)C1 57969,N1(C(C(CCC)N(C)C)=O)CC2CCC1CN2C(=O)C(O)CC(C)C 57970,N1(C(c2c(Cl)cc(C)s2)=O)CC2(CCC(CNC(C3(F)CCCOC3)=O)O2)C1 57971,c1(CC)nn[nH]c1C(=O)NCC(C)(C)CNC(c1ncn(CC)n1)=O 57972,c1(C(=O)NCC2(O)CC3CCC2CC3)cc2cc(Cl)ccc2cn1 57973,CCCCCCCC(F)C(=O)N1CCC(NC(c2ccc(Cl)c(Cl)c2)=O)C1CC 57974,N1(C(C=CCN(C)CC)=O)CC(CNC(c2cccc(N3CCCC3)n2)=O)CC1C 57975,C1(NC(c2c(C)n[nH]c2)=O)CN(C(=O)CC2(C)CC(F)(F)C2)CC12CCC2 57976,n1(C(C(=O)NCCCCNC(COCC=C)=O)C)cnc2ccccc12 57977,N1(C(C(C)CC2CC2)=O)CC(CO)C2(C1)CN(C(c1ccc(C(F)(F)F)[nH]1)=O)C2 57978,c1(CC)cncc(C(N2CC=CC(C(=O)NC(C3CCC3)C3CC3)C2)=O)c1 57979,c1(NC)cccc(C(=O)NC(C(C)NC(=O)CCCc2ccccc2)C(C)C)n1 57980,C(=O)(C(O)C(F)(F)F)N(CC=CC(=O)NC(C#C)CCC)C 57981,CC1(C)COCCC1CNC(C12CC(NC(c3sccc3CO)=O)(C1)C2)=O 57982,c1(C(=O)OC)csc2c1CCN(Cc1ccc(NC(C)=O)cc1C#N)C2 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58018,C1(C(N2CC(C)(CCO)C2)=O)(NC(=O)COCCF)CCOCC1 58019,C1(NC(c2nnnn2Cc2cccc(F)c2)(C)C2CC2)CC(=O)N(C(C)(C)C)C1 58020,c1(C(=O)NCC2OCCN(C(C3CCC(C)CC3)=O)C2)c(F)ccc2ccoc12 58021,c1(OC)cccc(C(=O)NC2CN(C(C3(CF)CC3(F)F)=O)CCC2O)c1F 58022,N1(C(c2c(C)cc(C(F)(F)F)s2)=O)CC(C2CN(C(=O)CC(C)(F)F)C2)C1 58023,c1(COC)nc(C(=O)NC2CN(C(=O)C(C)CN(C)C)C2)cs1 58024,N1(C(C2N(CC)CCC2)=O)CCC(C(F)F)(CNC(c2coc(N(C)C)n2)=O)C1 58025,Cc1c(NC=O)cccc1F.C(CCC(C)(C)C)N1CCCC1c1ccccc1Cl 58026,C1(CNC(c2nccc(C)n2)=O)CCCCN(C(=O)C(C)n2cncn2)CC1 58027,C12(c3ccn(CC(=O)OC)n3)CCC(CC1)N2C(=O)CN1CC2CC2C1 58028,N1(C(C(=O)NC(c2c(C)nn(C)c2C)C)=O)CC2CCCOC2C1 58029,c1(C(N2CCC(C)(NC(=O)C(F)C3CCOC3)C2)=O)cnc2c(c1)OCCN2 58030,Cc1ncc(C(=O)NC2CN(C(=O)CC3CC(NC(C)(C)C)C3(C)C)C2)n1C 58031,N1(C(c2c(OC)cncc2)=O)CCN(C(c2cc(CC3CC3)on2)=O)C(CO)C1 58032,c1(C(=O)NC2CCC(NC(c3cc(Cl)ncc3Br)=O)C2)cccc2nccn12 58033,C12(NC(c3cc(C)n(CCO)n3)=O)CCCN(C(=O)C(C)(C)CO)CC1C2 58034,c1(C(N2CC(NC(C(CC)(C)OC)=O)C(F)C2)=O)ccc2c(c1)CCO2 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58053,S(=O)(=O)(c1ccc(NC2C=CCC2)cc1Cl)NC(c1c(C)nns1)C 58054,C1(C(N(C)CC2CCCN(C(c3ncc[nH]c3=O)=O)C2)=O)CS(=O)(=O)CCO1 58055,N1(C(CCCOCCOC)=O)CC2(C1)CN(C(c1cnc(C)n1C)=O)C2 58056,C1(NC(CC=C(C)C)=O)CC2(CCN(C(C3CC3Br)=O)CC2)C1 58057,C1(CNC(C2CC(N(C)C)C2)=O)CCN(C(=O)CN2CC3CC3C2)C1 58058,c1(CN2CCCC(NC(=O)NC(CC)C(=O)N(C)C)C2)nc2ccccc2n1C 58059,c1(C(=O)NCC(CC)NC(=O)C(C)C(C)C)nn(C)c(Cl)c1Cl 58060,c1(CNC(CN2CCN(C(c3ccccc3CO)=O)CC2)=O)ccc([N+](=O)[O-])o1 58061,C1(C)(C(NC(Cc2ccn(CC)n2)=O)CC)CC(F)(F)CN1c1nc(C2CC2)ns1 58062,Cc1c(NC(=O)C(C)OC(F)F)cc(F)cc1CO 58063,Cc1cc(C(=O)NC(CC(=O)NCC(F)(F)Cl)C2CC2)cnc1O 58064,CCCC(CNC(c1[nH]nnc1C)=O)C(=O)NC1CC12CC(OC)C2 58065,c1(-c2c(C(=O)NC(CC(=O)O)C(=O)O)cn(C)n2)ccc([N+](=O)[O-])cc1 58066,C1(CCC)CN(C(C2CC2C)=O)CCN1C(=O)CNC(=O)C(F)(F)F 58067,c1(C(=O)NCC2CCN(C(CC)=O)CC2C)cc2c(C)nn(C)c2nc1C 58068,C1(C(=O)NCC(C)N(C(Cc2cc(C(C)C)no2)=O)C)CCC([N+](=O)[O-])CC1 58069,N1(COC(C(CC)C)C)CCC(CCn2ccnc2-c2ncc(F)cn2)CC1 58070,C(c1ccc(Cl)cc1)=CC(=O)NCCC(C)N(C(=O)C(=O)NCC1CC1)C 58071,C1(NC(CCc2cc(OC)c(F)cc2)=O)CCC(O)CN(C(C2CCCS2)=O)C1 58072,c1(N(CC(N2CCC2c2ccccc2)=O)C)ccc(F)cc1F 58073,CCC(C)CC(C(=O)NC)NC(c1cnn(C)c1NC(=O)CCN1CCOC1=O)=O 58074,C1(NC(c2ccoc2)=O)CN(C(c2cccc(OCC(F)F)c2)=O)CC1O 58075,C12(C(=O)NCCCCN(C(CC3CC(C(C)C)OCC3)=O)C)CCC(F)(CC1)C2 58076,c1(NC)ccc(C(=O)NCCn2cc(C(=O)NC3CCC3(C)C)cn2)cc1 58077,C1(CC#C)CCN(c2nnc(CS(C)=O)n2CC(C)CCC)CC1 58078,C1(NC(CN(C(C(C)C)=O)C)=O)CCN(C(C2CC3CCC2O3)=O)CC(C)(C)C1 58079,N1(C(CSc2cn(C)nc2)=O)CCC2CCN(C(=O)CC3CC3(C)C)CC12 58080,Cn1ccc2c(c1=O)CCN(C(=O)Cn1cc(Cc3ccc(C#N)cc3)nn1)C2 58081,c1(C(=O)NCC(C(=O)NCCCCC)N(C)C)cc(C)c(C)cn1 58082,N1(C(CC(C)F)=O)CC2(C1)C(NC(c1cc3ccc(Cl)cc3[nH]1)=O)CCS2(=O)=O 58083,c1(C(C)C(=O)NCC2CN(C(c3c[nH]c(=N)s3)=O)CC2O)ccc(F)c(F)c1 58084,C1(NC(CCC)=O)CCCC(N(C)C(C)=O)C1.C(=O)(CCO)NCC(C)(C)C 58085,C(CNC(C)C)(C(=O)O)N(C(CCSCC)=O)C 58086,C1(C(N(C2CN(C(Cc3c(C)nn(C)c3C)=O)C2)C)=O)CC2(C)CCC1(C)O2 58087,C(=O)(C(CC)(CC)CC)NCc1c(C(N2CCC(OCC=C)CC2)=O)scc1 58088,c1(NC(N2CCCC(C#C)(C)C2)=O)ccc(S(=O)(=O)C2CC2)nc1 58089,C=C(Cl)C(C)(C)C(=O)NC1CCC(NC(c2cc(Cl)c[nH]2)=O)CC1 58090,Cc1cc(C(=O)NCCC(C)N(C)C(C2C(C3CC3)C2(F)F)=O)nc(C)n1 58091,C1(NC(c2scc(C)c2Cl)=O)CCC2CCN(C(C3CC3(F)F)=O)C12 58092,c1(C(N2CCC(C(C(=O)NC(C)CCF)F)C2)=O)cc(O)cc(F)c1 58093,C12(CNC(c3n(C)ncc3)=O)CC3CC(CC(NC(=O)CSC(F)(F)F)(C3)C1)C2 58094,CC(CNC(=O)CN1CCCC1=O)C(F)C(=O)NCC1(CF)CC1 58095,Cc1cc(C(N2CC(CNC(C3CC3c3ccn(C)n3)=O)C2)=O)n(C2CCC2)n1 58096,c1(CC(=O)NC(CNC(C(CC)OCC)=O)C(C)C)cccc(C(F)(F)F)n1 58097,N1(C(CN2C(=O)CCCC2)=O)CC2OCCN(C(=O)CC3CC4(CCC4)CO3)C2C1 58098,c1(C(N2CC(NC(c3sc(CC)c(C)c3)=O)C(F)CC2)=O)c(F)ccc(F)c1O 58099,C=C1CCN(C(c2cn(C)nc2OC)=O)C(C(=O)NCCCF)C1 58100,C1(C(=O)NCc2c(C)nn(C)c2C)CC(N=[N+]=[N-])CN1C(=O)C(C)C1CCC1 58101,S(=O)(=O)(c1ccc(O)c([N+](=O)[O-])c1)NCCCCCC(=O)Nc1c(C)cccc1 58102,c1(N(C2CCN(C(c3ccsc3C(F)(F)F)=O)C2)C)cc(F)ncn1 58103,c1(OCC)ccc2c(C(=O)NCC(=O)OC(C)(C)C)c[nH]c2c1 58104,CC#CCCCC(=O)NC1COCC1C(N1CC(OC)CC(C)C1)=O 58105,Cc1cc(C)c(C(=O)N(C2CCC(CNC(=O)C=Cc3ccccn3)CC2)C)o1 58106,CN1CC(NC(C2CSC(C(F)(F)F)C2)=O)CC1=O 58107,c1(NC)cccnc1C(=O)NC(C)CC(C)NC(=O)COC(C)(C)C 58108,C1(O)(CN(C(C=CC(CC)=CC)=O)C)CCN(C(=O)CC2(O)CCC2)C1 58109,N1(C(C)=O)CC2CC2(C(=O)NC2(c3cccnc3)CC2)C1.N12CC(C1)C2=O 58110,c1(C(=O)NC(C)C(c2ccccc2)NC(=O)COCC(F)F)ccc(N)cc1O 58111,c1(NC(C)CN(C(=O)C2=CCSC2)C)ncnc2c1nnn2C1CC1 58112,c1(C(=O)NCC2(C)C(C)CN(C(=O)CC3CC(F)C3)C2)cc2c(s1)CCOC2 58113,N1(C(c2cc(C)sc2)=O)CCCOC(CNC(C2CCCN(C)C2)=O)C1 58114,O=S(=O)(c1ccc(=NCC2CCOC(C3CC3)C2)[nH]c1)NCC12CC(CCO1)C2 58115,c1(CC)noc(C)c1NC(=O)Cc1csc(NC(c2ccc(OC(F)(F)F)s2)=O)n1 58116,N1(C(Cc2cc(C)sc2)=O)CC2(C1)CN(C(=O)C(C)OCC(F)(F)F)CC2CO 58117,C(=O)(C1=CCCS1)NCC(CCOC)NC(=O)CCc1cccc(OC(C)C)n1 58118,c1(OC)ncc(F)c(CNC(=O)NC(CC)CCO)n1 58119,c1(N2CC(C)(C)C2C2CC2)ccc(C#N)c(CNS(C)(=O)=O)n1 58120,CC12CCC(C(=O)NCC3CCN3C(=O)CCCOc3ccccc3)(CC1)CO2 58121,c1(CN(C)Cc2cc(F)ccc2Br)cc(F)c2c(c1)CCC2 58122,c12ccnn1CCOC2.c1(C(c2nnnn2CCCF)N)csc(Br)c1.C1(C)CC1 58123,C1(NC(C(CC=C)CC)=O)CN(C(=O)CCc2nc(C3CC3)no2)CC1C1CC1 58124,c1(CC)[nH]c(C(=O)NC2CC(CO)N(C(c3sc(F)cc3C)=O)C2)nc1Cl 58125,c1(C(N2CC(NC(C(CSC)O)=O)C(C)C2)=O)coc2c(C)cccc12 58126,C1(NC(=O)NCC2C(C)CCC2)CC(=O)N(CC2CCC2)C1 58127,C(c1ccc(F)cc1)=CC(=O)NCC1CC(NC(=O)C2=CCOC2)C1 58128,c1(C(=O)OC)c(C)ccc(NC(N2CCOC3CC23)=O)c1C 58129,N1(C(CCc2cn(C)nc2)=O)CC2CC3CC2C1C3NC(=O)C(O)C(F)(F)F 58130,C(=O)(C1CCCc2nccn21)N1CC(NC(c2ncc(OC)cn2)=O)(CO)C1 58131,c1(C(N(CCCOCCNC(C(C)C(F)F)=O)C)=O)n[nH]c2cccnc12 58132,c1(C2(C(N(CCN(C(C(CC)C)=O)C)CC)=O)CCC2)cc(OC)cc(OC)c1 58133,CC1CC(C(N2CC(CC(C)(C)CNC(=O)CC3CCCCC3)C2)=O)C(=O)O1 58134,CCCC(C(=O)N1CC(NC(=O)Cn2ccnc2C(C)C)C(C)C1)OC 58135,C1(CNC(=O)C2=CCOC2)CC2CCC(C1)N2C(C1CC12CCOCC2)=O 58136,C(=O)(CS(C)(=O)=O)NC(C)C(CO)NC(=O)CCC(=O)c1ccc(Cl)s1 58137,c1(NC(C2CCN(Cc3cnc(Br)o3)CC2O)=O)cc(C(F)F)cc(Br)c1 58138,C1(CNC(c2ccncc2F)c2n(CCC)nnn2)OCCOC1(C)C 58139,N1(C(C(C)CCN(C)C)=O)CCCC12CCN(C(C1(O)COC1)=O)CC2 58140,N#Cc1cc(Cl)c(C(=O)NC2CCCC2CNC(c2cc(Cl)nnc2O)=O)s1 58141,c1(C(=O)NC(CNC(c2cn(CCC=C)nn2)=O)CC)noc2ncccc12 58142,c1(NC(C2N(Cc3c(C)nn(C)c3)C3C(C2)C3)=O)cccc2ccccc12 58143,C=CC1(NC(C2CC23CCN(C(=O)Cn2nccn2)C3)=O)CCOCC1 58144,N1(C(CC)=O)CCC(C2CCC2)(CNC(C2CCn3c(C)nnc3C2)=O)CC1 58145,N1(C(C(C(C)C)n2ccc(C)c2)=O)CCCCC(N2CCCC2)C1 58146,C(=O)(CCCCCCCC(=O)N1CCC(N(C(=O)C(F)C2CC2)C)CC1)OC 58147,c1(CC(=O)NC(CNC(C(C)=CC2CC2)=O)C)cccc(F)c1 58148,c1(C(N2CC3C(NC(CSCCCC)=O)(C3)C2)=O)c(OC)ccc(Cl)c1F 58149,CC(C)(C)C(O)C(=O)NCC1CCCCN1C(=O)Cc1n[nH]c(=N)s1 58150,c1(C(=O)NCC2CCN(C(C=CCCC)=O)C2)ccc(F)c(C(C)(C)F)c1 58151,N1(c2cccc(C)c2)N=C(C(=O)NC2CC2NC(c2ccns2)=O)CCC1=O 58152,c1(N(CCC)CCNC(c2coc(C)c2)=O)ncccc1[N+](=O)[O-] 58153,C1(CNC(NCC(CCC)Oc2ccco2)=NC)CCCCN1CC(C)C 58154,C(=O)(C(C)(C)CS(N)(=O)=O)N1CCC(N(C(c2coc(C3CC3)n2)=O)CC)CC1 58155,c1(C(=O)NCC(CNC(C(C)=C2CCC2)=O)(C)C)n[nH]c2ccc([N+](=O)[O-])cc12 58156,C12(CNC(c3c(SC)cccn3)=O)CCC(CC1)N2C(=O)Cc1ccco1 58157,CN1CCOCC1C(N1CCC(C2CCCN2c2nc(C(F)(F)F)ns2)CC1)=O 58158,C1(C(N2C(C3CCN(C(=O)Cn4cnnn4)C3)CCC2)=O)CC2(CCCO2)C1 58159,N(C(=NCCCF)NCc1ccccc1)CC1(O)CCCOC1 58160,c1(C(N2CCC(N(C(CC(C)SC)=O)C)CC2)=O)ccc(C)c(C)c1F 58161,C12CCCN1C2=O.C1(C(=O)NC(CC2(CSC)CCC2)=O)COC(C2CC2)C1.C1(C)CC1 58162,C1(CNC(C(Cc2ccc(OC)cc2)=O)=O)C(C)CCCN1C(c1cnns1)=O 58163,C(N=c1[nH]c(=NC(C)c2ncc(C)cn2)c2c(ncn2C)[nH]1)C1(OC)CCSC1 58164,S(=O)(=O)(c1c(Br)cccc1[N+](=O)[O-])N1C(C)CC(C(F)(F)F)C1 58165,C1(OC)CCN(C(C2CCOCCN2C(C2CCSCC2)=O)=O)C12CCC2 58166,C12(CNC(=O)C3CC3)CCCC1N(C(=O)CCc1ccnc(Cl)c1)CC2 58167,c1(C(=O)NC23C(NC(c4ccn(C)c4)=O)CC(CC2)C3)ccc2c(n1)OCCO2 58168,c1(N2C(C(C)(C)NC(C(C)Cn3ccnc3)=O)CCC2)ncc2c(n1)CCOC2 58169,C1(C(N2CC3C(NC(c4cc(F)ccc4F)=O)C3C2)=O)CC2CCC(C1)C2(F)F 58170,c1(C(=O)NC(CC)CNC(=O)CC2CC2CC)cccc(COC)n1 58171,c1(C(=O)Nc2c(C(=O)OC)ccc(OC)c2)ccc2c(c1)N(C)C(=O)C2 58172,C1(C2(O)CN(C(=O)CN3CCCC3C)C2)(CNC(c2ccc(C)cn2)=O)CC1 58173,C=CC(C)C(C)C(=O)N1CCC(CNC(c2cccc(Br)c2N)=O)CC1 58174,N1(C(C=C(C)C(F)F)=O)CCC2(CC1)CN(C(C1CN(C)CC1C(F)(F)F)=O)C2 58175,c1(OC)ccncc1C(=O)NCCC1(C)CCN(C(=O)CCc2n[nH]c(=N)s2)C1 58176,C1(C(=O)NCC2CN(C(C3CC(CC)C3)=O)CC2O)C2CCC3(COC(=O)C13)O2 58177,c1(OC)cccc(NC(=O)C(=O)NCCCOCCNC(=O)CC(C)(C)C)c1 58178,CC1(C(=O)NCC2CC(C(=O)NCCn3ncccc3=O)C2)C=CCCC1 58179,C1(CN(C(=O)COc2cccc(Br)c2)C)CCCN(C(=O)C=CC(F)(F)F)C1 58180,C1(C2C(C)(C)C2C(=O)NC2CN(C(=O)C3CC3)C2)CCN(c2cnccn2)CC1 58181,N1(C(C2C(Cl)(C(=O)OC)C2)=O)C2CCC1CC(CCNC(=O)C(C)=C(C)C)C2 58182,C12(C(N3CC4C(CNC(C(CCCC)C)=O)C4C3)=O)CC3CC(CC(C3)C1)C2 58183,CC1(C)C(NC(=O)CCc2cccnc2Cl)CCN1C(=O)C(F)C(F)(F)F 58184,C1(C(N(CC(O)C(F)(F)F)C)=O)CC2CCC(C1)N2CC1CCC(=O)O1 58185,CCC(CNC(C1CCNC1=O)=O)(CC)C(=O)N(C1CC(C)C1)C 58186,C(=O)(C(CO)C(C)(C)C)NC(CSC)C(=O)NOCCN(C)C 58187,c1(C(=O)NC2CCN(C(CCCSC)=O)C(C)C2)ccc2c(c1)CC(=O)NC2 58188,C1(NC(CCOC(C)C)=O)CCN(C(c2cnc(-c3cccs3)o2)=O)CC(O)C1 58189,C1(N(C)C)CC(C(=O)NC(C(=O)NCCN2CCC2)C2CCCC2)C1 58190,c1(C(C(N2CCC(n3ccnc3)C2)C)=O)ccc(F)cc1 58191,n1(CC=C)cc(C(=O)NC2CCCC2NC(C2CCCN2C)=O)nn1 58192,C1(F)(C(N2CC3(CCN3C(=O)Cc3c(Cl)cccc3Cl)C2)=O)CCCC=C1F 58193,CC(C)CCC(C(=O)NCc1cnn(C2CC2)c1)NC(=O)C(C)NC(N)=O 58194,C(=O)(C(C)(C)S(C)(=O)=O)NCCC(C)N(C)C(c1coc(N(C)C)n1)=O 58195,CS(=O)C1CN(C(=O)COCCNC(c2ccccn2)=O)C1 58196,c1(CC(=O)NC2(CCOC)CCN(C(C(CC)SC)=O)C2)cccc(Cl)c1Cl 58197,N1(C(C2CC(C(=O)OC)C2)=O)CCCCC1CC(=O)NCCN(C)C 58198,CC12CCOC(C(=O)NC3CCN(C(c4scnc4C(C)(C)C)=O)CC3O)(C1)C2 58199,C1(=CC(=O)NC(C2CC(NC(C3CCCC3F)=O)C2)C)CCCCC1 58200,N1(c2scc(C)n2)CCC(C(N2CC(NC(C3CC=CCO3)=O)C(F)C2)=O)CC1 58201,c1(C(=O)NC2CC3CN(C(C#CC(C)(C)O)=O)C2C3)cccn2cncc12 58202,C1(OC)CN(C)C(C)(C(=O)NCC2CN(C(=O)CCc3cnn[nH]3)CCC2C)C1 58203,C(=O)(CCCCC(C)(C)C)N1CC2CCC(N(C(Cc3cc(C)on3)=O)C)C2C1 58204,Cc1cccc(C(C)NC(c2cccc(Br)c2Cl)C)c1C 58205,N1(C(CSC(C)C)=O)CCC(C)(C(N2CCC(O)C(C)C2)=O)CC1 58206,CC(CS(C)(=O)=O)C(=O)NCC1CN(C(=O)Cc2cocn2)CC(C)(C)C1 58207,c1(CC(=O)NCCCCC2CN(C(C3C(C)C3)=O)C2)cnc2n1CCCC2C 58208,N1(CC2C(Cc3ccccc3)CCC(C)C2)CCC(CC(N)=O)C(C2CC2)C1 58209,Cc1cccc2c(C(=O)NCC3CCCN(C(C4CC(C)CO4)=O)CC3)cnn12 58210,C=C(C)CC(C(=O)N1CC2CC1C2NC(=O)C(CC1CCCC1)OC)NC(C)=O 58211,C1(O)(CNC(CCCC#CC)=O)CCCN(C(=O)CCC(=O)N2CCCC2)CC1 58212,N1(C(C(C)C)=O)CCC(C(=O)NCc2ccnc(Cl)c2)CC1 58213,N1(C(=O)NCCC2CCC(C)O2)CCN(Cc2ccccc2)c2ccccc21 58214,N1(c2nc(N3CCOCC3)nc(N(CC=C)C)n2)CCC(O)C(C)(C)C1 58215,C1(C(N2CCC(C3(C)N=N3)C2)=O)(NC(C2N(C(C)C)CCC2)=O)CCN(C)C1 58216,c1(C(=O)NCCCNC(C(CC2CCC2)NC(C)=O)=O)ccncc1NC(C)=O 58217,CCC(C)(C(=O)N1CCC(CN(C(C2COCCC2(F)F)=O)CC)CC1)C(N)=O 58218,c1(C(C(=O)NCCC(C)NC(c2cn(C)cn2)=O)C)c(F)cccc1F 58219,CC1(C)CC(C)(CNc2nccc(NCc3cccc(OC(F)(F)F)c3)n2)C1 58220,C12(CNC(=O)CCc3cnc[nH]3)CC(CO1)N(C(=O)Cn1nnc(C3CC3)n1)C2 58221,c1(CCCNCC2(CC#C)CCOCC2)cc(OC)ccc1O 58222,c1(C(=O)OC)c(Br)cc(Br)c(NC(=O)C(=O)NC2CCC(N(C)C)C2)c1C 58223,N1(C(C2CCCCO2)=O)CCC2CN(C(=O)C(c3ccccc3F)O)CC2C1 58224,CS(=O)C=CC(=O)NC1CC(CNC(C2(C(F)F)CCOCC2)=O)C(O)C1 58225,c1(C(N2CC3C(CNC(C4C(C(C)C)CCC4)=O)(C3)C2)=O)n[nH]c2c1COCC2 58226,C(=O)(CCC(C)(C)[N+](=O)[O-])NCc1cccc(-n2c(C)nc(C)n2)c1 58227,C1(C(=O)NC2(C(=O)NC(c3cccs3)C)CC(O)C2)CCC2(CCC2)O1 58228,c1(C(=O)NC(C)CC2CN(C(C3(n4cc(Br)cn4)CC3)=O)C2)cnn(C)c1 58229,Cn1ccn2ncc(C(=O)NC3CC(CNC(c4cccnc4O)=O)C3(C)C)c12 58230,CCC(CC)(C(=O)NC1CCC(C)(CNC(=O)CN2CC(C)(OC)C2)C1)OC 58231,N1(C(Cc2cc(C)[nH]n2)=O)CCC(CCNC(=O)CCNC(=O)C=CCl)CC1C 58232,c1(C(N(CCC(=O)NCc2scc(C)c2)CCCO)=O)cc(F)cc(F)c1 58233,CC1CN(C(c2cnc(F)c(Cl)c2)=O)CCC1CNC(C1(C(N)=O)CCC1)=O 58234,C1(CCC(=O)N(C2C3CN(C(C4(C)CCCOC4)=O)CC23)C)CCCCCC1 58235,C1(F)(C(=O)NCC2(F)CC(NC(CN(S(CC)(=O)=O)C)=O)C2)CC2(CCC2)C1 58236,N1(C(c2c(C)occ2)=O)CCC2(C)CN(C(C3C4CC5C(C4)C35)=O)CC12 58237,c1(C(N2C(C)C(NC(c3ncncc3Cl)=O)CC2)=O)cc2n(n1)CCCC2O 58238,N1(C(C23CC(OC)C2C3)=O)CC(C2(NC(=O)CSc3ccc(Cl)c(Cl)c3)CC2)C1 58239,CC1CCC(CNC(=O)Cc2ccc(F)nc2)CN1C(c1cncn1C)=O 58240,C1(C(=O)NCCOCCC)CCOC1CNC(=O)C=C(C)C(C)(C)C 58241,CC1(C)CN(C(=O)C(N2CCC3(c4cccnc4)CC3C2)=O)CCC1C(F)(F)F 58242,C1(NC(c2csc3cncn23)=O)CC2CN(C(c3ccc(F)c(Cl)c3)=O)CC12 58243,c1(C(=O)NC(CC)CNC(C2CC(O)(C(F)(F)F)C2)=O)cc[n+]([O-])cc1 58244,C1(C(N(CC(=O)N(C(CC)CC)CCC)C)=O)CCCN1C(C)=O 58245,c1(C(=O)NCC2(C(C)(C)O)CN(C(CC)=O)C2)cnc2c(Cl)cccn12 58246,N1(C(C2C(C(C)C)C2)=O)CCN(C(=O)Cc2c(Br)cnn2C)C(CCO)C1 58247,c1(N(C2CC(C)C2)C)nnc(-c2ccc[nH]2)n1CCc1ccccc1F 58248,C12(NC(=O)CCn3cncn3)CCCC1(F)CN(C(C13CCC(F)(CC1)C3)=O)C2 58249,N1(C(c2nc(OC)sc2)=O)CCOC(C2CN(C(c3cc(C)oc3C3CC3)=O)C2)C1 58250,N1(C(COC2(C)CCOCC2)=O)CC=C(CCNC(C2CCC(=O)O2)=O)CC1 58251,Cc1nc(C(=O)NNC(=O)C(C)C2CCCOC2)cn(C)c1=O 58252,c1(C(C(=O)NCCN(C2CCCCC2)C(c2cnc(C)[nH]2)=O)O)ccccc1Cl 58253,C12(C(=O)NC(C)CC3CCN(C(C4(C)CCCC4O)=O)CC3)CCC(CC1)CC2 58254,N1(C(C2CCC(=O)N2)=O)CCCOC(CNc2nccc(-c3ccnn3C)n2)C1 58255,C1(NC(CC2(C)OCCO2)=O)C2CN(C(C3CCCN(C(N)=O)C3)=O)CC12 58256,CC(C)C(O)C(C)C(=O)NCCCC(C)CO 58257,C1(CC(C)(C)C)CN(C(=O)CCC(=O)c2cccs2)CC1NC(=O)COC(F)(F)F 58258,C1(CC(C)NC(=O)N(CC2CC2)CC2CC2)COCCO1 58259,c1(C(=O)NCC#CCNC(C(CC)CCOC)=O)c(Cl)cc(Cl)cc1Cl 58260,C1(NC(c2cc(C)sn2)=O)CCC12CCN(C(c1cc(Cl)c(F)cc1Cl)=O)CC2 58261,CC1=NN(C)C(=O)C1CC(N1C2CCC1C(NC(c1cccc(F)c1Cl)=O)C2)=O 58262,C1(n2cc(C3C(C(=O)OC)C3)nn2)CCCN(C(C2(C3(C)CC3)CC2)=O)C1 58263,c1(C(=O)NC(CNC(C(CC)O)=O)C2CCC2)cc(C)cc([N+](=O)[O-])c1 58264,c12cc[nH]c1C(=O)NC2.C1(C(=O)OC)CC(C(N2CC(N3CC(O)C3)C2)=O)C1 58265,N1(C(C(C)SCC)=O)CC(CNC(=O)C(Cl)=CCl)(OC)C1 58266,CC(CCCCO)NC(=O)C(CCF)NC(c1cncc(O)c1)=O 58267,c1(C(N2CCCC(Br)C2)=O)ccc(NCc2ccncc2Cl)cc1 58268,C1(C(N2CC(CNC(C(COC)C)=O)CC2(C)C)=O)CN2CCCN1CC2 58269,N1(C(c2c(SC)c(Br)ccc2)=O)CC(CC(=O)O)OC2(CCOC2)C1 58270,c1(CCC(=O)NC(C2CN(C(C3CCCCO3)=O)C2)C)cccnc1Cl 58271,C1(COC)CCCCN(C(=O)CC(C)CNC(=O)CC(C)O)C1 58272,c1(C(N(CCNC(CCN(CCCCC)C(C)C)=O)C(C)C)=O)cccnc1O 58273,Cc1ccc(O)c(CNC(C2C=CCN(C(C3(C)CC4(CCC4)C3)=O)C2)=O)c1 58274,C12(C(=O)NCC(C3CC3)SC)CC(C)(CN1C(=O)CCn1ccnn1)C2 58275,N1(C(C=CCC)=O)CCC2(CCCC2NC(c2cnn3c2OCC3)=O)CC1 58276,C1(C(N2C(C)CC(NC(C3N(C(C)=O)CCC3)=O)C2)=O)Cc2cccnc2C1 58277,N1(C(CCCSCC)=O)CCN(C(C2CCN2C2CCCC2)=O)CC1COC 58278,N1(C(C2(C)CCCO2)=O)CCC(C2CN(C(C3CCC3(F)F)=O)C2)CC1 58279,c1(C(CC(=O)NCc2ccc(CCCCCCC)cc2)O)ccc(O)c(O)c1 58280,CC1CCC(NC(c2ccc(CO)c(Cl)c2)=O)CN1C(=O)CCC1CCC1 58281,C(=O)(C(F)C(C)(C)O)NCC1N(C(c2nn(C)c(Br)c2)=O)CC(O)C1 58282,[N-]=[N+]=Nc1ccccc1CCC(=O)NC1CC2CC1N(C(=O)CCC(N)=O)C2 58283,c1(CCC)ncoc1C(=O)NCC1CC(CNC(=O)CC(=O)N(C)C)CO1 58284,Cc1cccc(Cl)c1C(=O)NC1CC1NC(=O)C1=C(Cl)CC1 58285,Cn1nc(O)cc1NC(C1CC1C(=O)Nc1ncco1)=O 58286,Cc1cnc(C(=O)NC2CCC(C(=O)NCc3ccnn3C)C2)cc1C 58287,c1(C(=O)NC(CNC(C23CCC(=O)N2CCS3)=O)CO)cc(=O)n2nccc2[nH]1 58288,N1(C(C(C)=CC)=O)CCN(C(CNC(c2ccsc2)=O)C(F)F)CC1 58289,c1(C(=O)NCC2C(NC(c3coc(Cl)c3)=O)CCC2)ccc(F)c(Br)c1 58290,C1(NC(c2ccc(OC)o2)=O)CCCC(NC(c2ccnc(C(F)F)c2)=O)CC1 58291,Cc1cc(C(=O)NCc2cnn(C)c2)cc(C)c1O 58292,C(=O)(C1=Cc2ccccc2C1C)NCCN1CCCN(C(CCCCOC)=O)CC1 58293,CC1CCN(C(c2c[nH]nc2C(F)F)=O)CCN1C(=O)CCc1ccccc1F 58294,Cc1ncc(C=CC(=O)N(CC[SH]=S(C)C)Cc2cc(F)c(O)c(Cl)c2)c(O)n1 58295,N1(C(c2c(CC)cco2)=O)C2CCC1C(C(=O)NCc1nc(C)co1)C2 58296,CC1(C)CC(CNC(=O)C2=CSCS2)CN1C(=O)COc1ccccc1 58297,Cc1cncc(C(=O)NC(C2CC2C(N2CCOC(CN=[N+]=[N-])C2)=O)C)n1 58298,S(=O)(=O)(c1cnc(Cl)nc1)N1C(C(=O)Nc2c(OC)cccc2)CC(O)C1 58299,C1(N(C(c2cnc(CC)s2)=O)C)CN(C(C2CC2C(C)(F)F)=O)CC1(C)C 58300,c1(C(N2CCC(N(C(C3CCCO3)=O)CC)C2)=O)cc(C)n(C)c(=O)c1 58301,O=C1NCc2cc(C(N3CCOC4(C3)CN(C(C35CCCC3C5)=O)C4)=O)ccc21 58302,c1(OCC)cnc(C(=O)NC2CC(NC(=O)C(S(C)(=O)=O)C3CC3)C2)c(Cl)c1 58303,CCCCC(C(=O)N(C(=O)C(C)(O)C1CCC1)CC)NC(C1CN(C(N)=O)C1)=O 58304,c1(NC(CCC)CC)cc(NCCc2scnc2C)nc(C)n1 58305,C1(O)(C(C)NC(=O)Cn2cnnn2)CCN(C(=O)C(F)CC2CCCCC2)CC1 58306,C1(NC(CCOCC#C)=O)CC2(CCCN(C(=O)C(CC(C)C)NC(C)=O)C2)C1 58307,C(c1cccs1)=C(C)C(N1CCC(CN(C)C(C2CC2CF)=O)C1)=O 58308,Cc1cc(=NC(=O)C(=O)NC2CC3CC2N(C(c2cc(C(N)=O)cs2)=O)C3)[nH]o1 58309,CCCC(C(=O)N1CCC(C(C)NC(c2ccc(N)cc2CC)=O)C1)S(N)(=O)=O 58310,C1(C(N(CC(N2CCCC2)=O)C)=O)CC12CCN(C(=O)CCc1cn[nH]c1)CC2 58311,c1(OC)c(F)cc(S(=O)(=O)N2CCCC2CCCN(C)C)cc1F 58312,CC1(C)CC(O)(CC(=O)NCCCCCCNC(c2cc(N)cnc2Cl)=O)CO1 58313,C(=O)(C(C)(C)CCNC(=O)CC1CCCNC1=O)N(CCC(O)CO)C 58314,C1(C(N2CCC(=CC)C2)=O)CCN(C(=O)Nc2ccccc2O)CC1 58315,CC#CCCC(=O)NCC(COC)NC(c1oc(C)nc1CC)=O 58316,c1(OC)nc(C(=O)OCC(=O)N(C)CC2CCCCC2)sc1C 58317,C12(C(=O)Nc3c(OC)ccc(C)c3)CCCC1CCN2C(C1CCC1C)=O 58318,CCC(CC(C)C)C(=O)NCC1CC2CCC1N2C(=O)CCn1ccnn1 58319,c1(OC)ccc(C2CC2)c(C(=O)NCC2CC(CNC(=O)CC(C)F)C2)c1 58320,C1(C(=O)OC)CC12CN(C(C13CC1CCN3C(c1cc(C)sc1C)=O)=O)C2 58321,C12(C(=O)NCC3CN(C(c4n[nH]c(C)c4Cl)=O)CC3(F)F)CCCCN1CCC2 58322,C(CC(C)C)(C(=O)NC(C)CC(C)O)NC(c1ccc(C)n1C)=O 58323,c1(C(=O)NCC(CN(C(CCOCC)=O)C)C)occc1F 58324,Cn1ccc(=NC(=O)CCOCCNC(=O)C2=NOC3CCCC23)[nH]1 58325,C1(C(N2CC(CC)(CC)C2)=O)CN(C(=O)C=C(C)C(F)F)CC(C)(C)C1 58326,C1(C(=O)OC(C)(C)C)CCCCC1NC1CC(NC(=O)NC2CC=CCC2)C1 58327,n1(C(COC)C)nc(-c2ccccc2)nc1CC(C)CC(C)C 58328,C1(F)(CNC(CC2CCC(C)C2)=O)CCN(C(=O)Cc2csc(C(C)C)n2)CC1 58329,c1(C(N(C2CC3CCC(C2)N3C(C2CNC(=O)C2)=O)C)=O)cc(Cl)cc(Cl)c1Cl 58330,c1(C(C)C)ccc(C(=O)NC2C3CN(C(C4CCC(=O)N4C)=O)CC23)cc1 58331,C1(C(=O)NC(CNC(C=C(C)CN2CCOCC2)=O)(C)CO)CCC(F)(F)C1 58332,c1(C(N2CC(F)CC(NC(C=C(CC)C)=O)C2)=O)cccc2nccnc12 58333,C1(C(=O)NC2(CNC(CC3C(C)C3)=O)CCCCCC2)CCn2cnnc2C1 58334,N1(C(C(c2ccccc2)NC(Cc2n(C)ccc2)=O)=O)CCC2(CNC(=O)N2)C1 58335,N1(C(C(COCC)C)=O)CCC2(CCC(CNC(c3ccc(C)n3C)=O)O2)CC1 58336,C1(C)(C(=O)NCCOCCCNC(c2c(C)snc2)=O)CCCC1O 58337,Cc1ccc(Cl)cc1NNC(=O)NCC1COc2ccccc2O1 58338,c1(N(c2ncc(C#N)s2)CCC(C)(C)C2CC2)cnc2cc(C(=O)O)ccn12 58339,C(CCCC(CO)NC(=O)Cc1nnc(O)s1)NC(c1c(OCC)cccc1)=O 58340,c1(C(=O)NC(C(C)NC(c2cc(CO)[nH]n2)=O)CO)cc(Br)c([N+](=O)[O-])[nH]1 58341,c1(C(=O)NCCCN(C(c2cccc(C)c2C)=O)C(C)C)ccc2nc[nH]c2n1 58342,N1(C(C(CCC=C)(F)F)=O)CCC2(CC(NC(=O)COC3CCOCC3)CO2)C1 58343,C(c1ccc2c(c1)OCCO2)=CC(=O)OC(c1ncc(C)[nH]1)C1CC1 58344,C(CC(C)(C)CC(=O)NC1CC1CNC(=O)C(n1cc(Cl)cn1)C)OC 58345,C1(CNC(C2CC(C)(C)C2)=O)CN(C(C2CCCC2(F)F)=O)CCCO1 58346,Cc1noc(C)c1S(=O)(=O)N(C1CC2CC1CN2)C(C)CO 58347,C(=O)(CCC(CF)CF)N(C(C)CNC(C1CCOC1)=O)C 58348,CC(CC(F)(F)F)C(=O)N1CCCCC(NC(c2snnc2C2CCC2)=O)C1 58349,c1(OC)c(NC(=O)Cc2csc(NC(c3cn(C)cn3)=O)n2)cccc1F 58350,CC(C)CC(O)C(=O)N1CC(CNC(C23CC(C2)C(C)O3)=O)C1 58351,c1(NC(COC(c2c(C)nc(C3CCOC3)s2)=O)=O)csc2nccn12 58352,N1(C(CC(CC)SC)=O)CCC2C(CCCN2C(C2(C)CCN(C)CC2)=O)C1 58353,C12(NC(CCc3c(C)noc3)=O)CCC(C(=O)NCc3cc[nH]n3)(CC1)C2 58354,c1(N2CCCC(COC)C2)nc(N2CCC=C(Br)C2)c2ccc(C)cc2n1 58355,c1(C(=O)NCC(=C)C)cnc2ccc(-c3cc(OC)cc(C)c3)cc2c1Cl 58356,Cc1ccc([N+](=O)[O-])cc1C(=O)NCC1CN(C(=O)CCOCC(F)F)CC1O 58357,C1(NC(CC(=O)OCC)=O)CCN(C2CCN(C(=O)CSC(F)(F)F)C2)CC1 58358,CC1CN(C(c2ccnc(Cl)c2)=O)CC1NC(c1cc(O)no1)=O 58359,N1(C(C(CC)(C)CO)=O)CC2(CC(NC(c3ncccc3Br)=O)CO2)C1 58360,N1(C(CN(C)C)=O)CCC(F)(F)C(CNC(c2cnccc2C(C)(C)C)=O)C1 58361,N1(C(CC2CCCC(C)C2)=O)CCC(F)(C(N2CC(C)(N(C)C)C2)=O)CC1 58362,C(C(=O)N1CCCCO1)(c1cn(C)nn1)NC(C(OCC)OCC)=O 58363,c1(NCCN(CCC)CCC)ccc2c(c1)C(=O)N(CC(C)C)C2 58364,N#Cc1ccc(C(F)(F)F)c(N2CCC(CCC#N)CC2)c1 58365,Cc1c(C(=O)NC(CO)C(=O)NCC(c2cnn(C)c2)C)cccc1C#N 58366,C(C(=O)Nn1cnn(C)c1=S)C1CC(C)N(C(=O)CCc2cncn2C)C1 58367,CC(CNC(c1n[nH]c(=N)[nH]1)=O)CC(=O)N(C(C)C(C)(C)O)C 58368,N1(C(c2c(COC)cco2)=O)CCC(C)C1CNC(=O)CCOc1ccccc1 58369,C1(C)(OCC(=O)N(C)CCN(C)C(=O)Nc2conc2C2CCC2)CCOCC1 58370,c1(C(N2CCC(n3cccn3)C2)C(=O)NC(C)C)cc(F)cc(F)c1Br 58371,C1(NC(c2c(CC)nns2)=O)CC(CNC(=O)CCc2c[nH]c(=N)[nH]2)C12CCC2 58372,C1(C(=O)NC2C(C#C)CCCC2)CCCCN(C)C1=O 58373,N1(C(COCCC(C)C)=O)CCCCC(NC(=O)CCCC(C)O)C1 58374,N1(C(Cc2cnc(C)s2)=O)CCC(C)C(NC(c2ccc(-c3ccco3)o2)=O)C1 58375,Cc1cc(C(=O)N(CC(C)NC(C2CC2C2CCC2)=O)C)cc2c1CCC2 58376,CCC(C(F)(F)F)NCC1CC(CC)(CC)CO1 58377,C(c1cccc(Cl)c1Cl)=CC(=O)NCCC(C)N(C(=O)CC1NC(=O)NC1=O)C 58378,CC(C)C(C)(CNC(c1nsnc1O)=O)NC(C1C=CCC1)=O 58379,c1(C(N2CC3CC(NC(C4(O)CC(C)(C)C4)=O)C3C2)=O)cncc2ccsc12 58380,CC(C)(C)C#CC(=O)N1CC(NC(C2CS(=O)(=O)C2)=O)C(c2ccc(F)cc2)C1 58381,c1(OC)ccc2cccnc2c1COC(C1CCC2(CC2)C1)=O 58382,N1(C(c2c(CCC)n[nH]c2)=O)CCCCC(C(=O)NCCC(CCC)C2CC2)C1 58383,c1(OCC(=O)NCC(n2cc(C3C(C)C=C(C)CC3)nn2)C)ccccc1[N+](=O)[O-] 58384,c1(OC)nc(=NCCc2nc(-c3ccccc3)n(C)n2)[nH]c(C)c1F 58385,Cn1cnnc1CNC(c1n[nH]cc1CNC(C1(F)CCOC1)=O)=O 58386,CC1OC(C)C(C(=O)NCC2(C)CCCN2C(c2ccc(C(N)=O)s2)=O)C1C 58387,C1(NC(C(c2n(C)cnc2)O)=O)CCN(C(=O)CCN2CCCC2=O)CC1 58388,N1(C(COCC(=O)NC)=O)CCOCC1CN(C)C(C1(C)CCCCO1)=O 58389,CC(O)CCCNC(=O)CCNC(C1(C(C)(F)F)CC1)=O 58390,CC(C)(O)C(F)(F)C(=O)N1CC(F)(CNC(C2CCCC(C(F)(F)F)C2)=O)C1 58391,C1(CNC(C(C)CF)=O)CCCN(C(=O)CCN2CCCC2=O)C1 58392,c1(C(=O)NC2C(CC)CN(C(c3cnn(C)c3N)=O)C2)cc(SC)cc(Cl)c1 58393,C1(NC(CCc2cc(C)no2)=O)CC2C1CCN2C(C1CC2CC(=O)C1C2)=O 58394,N1(C(CCCCCNC(CNC(CC)=O)=O)=O)CCC2(CCOC2)CC1 58395,CCC(F)(F)C(C)(C)C(=O)N1CCN(C(c2ccc(C(C)C)o2)=O)CC1C 58396,C1(C(C)C)CCOCCN1C(=O)COC1(C)CN(C(=O)C(C)Cn2ccnc2)C1 58397,c1(OC)ccc(C(=O)N(C(C)CNC(=O)C(C)(C2CC2)OC)C)cc1S(C)(=O)=O 58398,CN1CCN(C(=O)Cc2csc(S)n2)CC1CNC(C1CN(C)CCO1)=O 58399,NS(=O)(=O)c1nc(C(N2CCC(NC(=O)CCF)C(CO)C2)=O)n2ccccc12 58400,CN1C(=O)c2ccccc2C1C(=O)N1CCCCC1CCNC(C1CC1(C)C)=O 58401,CC#CCCCC(=O)NCCCC1(C)CN(CC2CCC(C#N)CC2)CCO1 58402,O=[N+]([O-])c1cccc(Br)c1CN1CCC2CCNCC12 58403,S(=O)(=O)(c1cccc(=NCC(C)c2nccs2)[nH]1)N(C(C=C)C1CC1)C 58404,N1(c2nnc(CCC)s2)CCCC(CO)(NC(c2ncoc2C)=O)C1 58405,c1(NC(C(C2CN(C(C(CC=C)NC(C)=O)=O)C2)OC)=O)cc(C)c(C)cc1F 58406,c1(C(N(C2CN(C(C(F)OC)=O)C2)C)=O)n[nH]c(C)c1C 58407,N1(C(COCCSC)=O)CCCC1CC(=O)NC(C12CC(CO1)C2)C 58408,N1(C(CN(CC)CC)=O)CC2C3CCC(C2C1)N(C(C1CCC(C)S1)=O)C3 58409,CON1CCC(C(N2CC(NC(=O)CC3CCN(C)C3)CC(F)C2)=O)CC1 58410,C12(NC(C(CSC)OC)=O)CCC(CN(C(c3cc(CO)on3)=O)C1)C2 58411,c1(C(C2(O)CN(C(C3CCN(C(=O)C4CC4)C3)=O)C2)C2CCCO2)ccc(Cl)cc1 58412,N1(CC=C(C)C)CCCC(C(=O)NC(CC2CC2)CO)C1 58413,c1(NS(CC)(=N)=O)ccc(OC)c(OC)c1OC 58414,c1(OC)cc(C(=O)NC2CCCCC2NC(=O)C2=CCC2)c2c(c1)CCO2 58415,c1(C(=O)OCC(=O)N(C2CCOC2=O)C)coc2cccc(F)c12 58416,N1(C(C=CC(C)(C)SC)=O)CC=CC(C(=O)N(C)Cc2sccc2C)C1 58417,c1(OC(C)C)cncc(C(=O)NC2(CNC(c3cc(C#N)c[nH]3)=O)CC2)c1 58418,C(C)(CCC(=O)NC1CCC1C(=O)NCC(O)Cn1cccn1)OC 58419,N1(C(CN(CC(C)(C)C)C)=O)CCCC1(C)C(=O)NCC1(C#N)CCC1 58420,n1(C(CC)C)ncc(C(=O)N(CCCN(C)C(c2snnc2C2CC2)=O)C)c1C 58421,N1(C(c2c(OC)nsc2OC)=O)CCC(C)C(NC(c2cc(Cl)on2)=O)C1 58422,CC(C)(CF)C(=O)NC1CCCCC1NC(=O)C=CC(=O)NCc1ccncc1 58423,CCC(CN(C)C)CC(=O)NC1CN(C(c2cc(C(C)=O)on2)=O)C(C)(C)C1 58424,c1(C(=O)NC2CC(NC(c3ncncc3Cl)=O)C23CCC3)cccc2sccc12 58425,N1(C(C2CCC(OC)CC2)=O)CCC(NC(=O)C#CC2(C(F)(F)F)CC2)C1(C)C 58426,N1(C(C2(C)CS(=O)(=O)C2)=O)CC(CNC(c2ccc(F)s2)=O)C2(CC2)C1 58427,C1(CC(=O)OC(C)C(=O)N(c2cccc(F)c2)C)CC(O)CN1C(C)C 58428,N1(C(=O)CC2NC(=O)NC2=O)CC2CCN(C(C34CC5CC3C4C5)=O)C(C2)C1 58429,c1(C(=O)NC2C(C)CN(C(C3(C)CCC3)=O)CC2)cnc2[nH]ccc2n1 58430,N1(C(CC(C)(C)C)=O)C2CCC1C1CC1(NC(C1CC3CCC1O3)=O)C2 58431,C1(CNC(CCOC)=O)CN(C(=O)CCNC(=O)CC(C)C)CC(C)(C)C1 58432,C1(C(N2CCC(O)(CCNC(C3CC3(F)F)=O)C2)=O)CC(C2CC2)=NO1 58433,C=CC(CCC)CC(=O)N1CC(C(O)C(=O)NC2CC(C(=O)OC)C2)C1 58434,C1(C(=O)OC)(NC(c2cc(C)c(OC)c(Cl)c2)=O)CC(O)C12CCC2 58435,C(=O)(C#CC1(C)CC1)NCC1(OC)CCN(C(c2ccc(CN(C)C)o2)=O)C1 58436,Cc1cc(C(=O)NCC2CCC(NC(C3CC4CCCC34)=O)C2)c(N)c(F)c1 58437,Cc1cnc(C(N2CC(C(N)=O)(CNC(C3CSCCS3)=O)C2)=O)cn1 58438,c1(C(N(C)CC2N(C(C=CC=CC)=O)CCC2)=O)cccn2ncnc12 58439,C1(C(N2CC(CCC#C)C2)=O)CC(NC(=O)Cn2ncnn2)CCO1 58440,C(=O)(C(C(C)C)C(C)C)NC1CC(CNC(C(C(C)(C)C)NC(C)=O)=O)C1 58441,c1(C(N2C(CCNC(c3cc(C)no3)=O)CCC2)=O)ccc(C)c(Br)c1 58442,c1(-c2ccc(C#N)s2)cc(C(N2CCC(O)(CF)CC2)=O)cc2[nH]ncc12 58443,N1(C(C(CCCCCC)F)=O)CCOC2(CCCN(C(=O)CCC3CC3)C2)C1 58444,CN=c1nc(N2CCN(CC(F)(F)Cl)CC2)[nH]c(=NC2CCCCCCC2)[nH]1 58445,c1(C(=O)NCC(C2CCOC2)NC(c2sccc2F)=O)c(F)cccc1[N+](=O)[O-] 58446,C1(C(N(C)CC2CC(=C)C2)=O)CC2CCC1N2C(=O)Cn1nnc(C)n1 58447,c1(C(=O)NC(C)CN(C)C(c2ncc(F)cc2F)=O)cc(F)cc(Br)c1F 58448,c1(CNC(C)Cc2ccco2)cc(Br)c(F)cn1 58449,C(=O)(CS(=O)(=O)CC(=O)NCC1CC(O)CN1C(=O)Cc1ccc(C)s1)OC 58450,C1(CCNC(CSS(C)(=O)=O)=O)CCN(C(=O)CCOC2COC2)C1 58451,C1(NC(C(N2CCCCCC2)C)=O)CCN(c2ccncc2C#N)CC1O 58452,C1(C(=O)OC)CC2CC(C(=O)NC3CC(OCc4ccc(C)cn4)C3SC)CC12 58453,C1(C(=O)NC(CNC(CC(CC)C2CCC2)=O)(C)C2CCC2)CC(=O)NC(=O)C1 58454,Cc1cc(O)ccc1CC(=O)NCC1COC(CNC(C2CC(C)(C)CO2)=O)C1 58455,c1(CC)nn(C)c(Cl)c1C(N1CC(CNC(=O)C(C)(O)C2CCC2)C(C)(C)C1)=O 58456,CCCCCCC(CC)NC(C1CC(CCNC(=O)CC(C)n2cccc2)C1)=O 58457,Cc1cc(C(N2CCC(C3CC3)C2CNC(=O)CC(C)(C)O)=O)cc2nc[nH]c12 58458,C=CCCC(C(=O)N(CC(=O)NC)CC)NC(c1ccc(C)cn1)=O 58459,N1(CC(CNC(c2cc(C)sc2)C2CN(c3nnnn3C)C2)(C)C)CCN(C)CC1 58460,c1(C(=O)NCC(CNC(c2nc(CC)[nH]n2)=O)C)cc(C)ccc1[N+](=O)[O-] 58461,C1(C(N2CC(CNC(C3CCN(C)C(=O)C3)=O)C2)=O)CCc2nn[nH]c2C1 58462,c1(C(=O)NCCNC(c2c(C(N)=O)cccc2)=O)cnc2nccn2c1 58463,c1(C(=O)NC2CC(CNC(CCC3CC(C)C3)=O)CC2O)ccc(F)cc1C#N 58464,C1(CCONC(C2CN(CN3C(=O)CNC3=O)CC23CC3)=O)CCC(F)(F)CC1 58465,c1(C(N2CC(CNC(c3nc(CC)oc3)=O)C3C2C3)=O)cc(C)ccc1[N+](=O)[O-] 58466,c1(C(N2CCC(NC(C=CCN(C)CC)=O)C2)=O)cncc2c[nH]nc12 58467,N1(C(C2CCCN2C(c2ccco2)=O)=O)CCCCC1CC1CC=CC(O)C1 58468,N1(c2nc(OC)c(F)c(C)n2)CCC2(CC1)OCCC2NC(=O)C1=C(C)OCC1 58469,C1(C(N(C2CC(NC(CCSC)=O)C2)C)=O)CCOCC1C 58470,c1(C(N2C(C(=O)NCC3(O)CCCC3)CC(O)C2)=O)c(F)cncc1Br 58471,N1(C(CC(C)(C)O)=O)CCN(C(=O)CCCc2ccccn2)C(CO)C1 58472,c1(CC(N2C(CN(C(C(C)SC(F)(F)F)=O)C)CCC2)=O)ccccc1Cl 58473,n1(CC(=O)NC2C(CNC(C(C)Cn3cccn3)=O)C2)sc2ccccc2c1=O 58474,c1(C(=O)NC2CC(CCNC(c3[nH]c(=N)sc3)=O)C2)n[nH]c2c1CC(F)(F)CC2 58475,c1(C(=O)NCCCN(C)C(c2cc[nH]c2C2CCCC2)=O)cccc(CO)n1 58476,CC1CCN(C(c2c(C(F)(F)F)cnn2C)C(=O)NCCCC2CC2)CC1 58477,C1(NC(CC=C)=O)CCC(CCNC(c2cn(C(C)C)nn2)=O)C1 58478,C1(C(=O)NCC(=O)NCC)CCC(O)CN1C(c1cn(CC)nc1C)=O 58479,N1(C(c2cn(CC)nc2)=O)CCCOC(CCNC(c2nccc(C)n2)=O)C1 58480,N(C(=NCCCNC(c1cccs1)=O)N1CCN2C(=O)NCC2C1)CCOCC 58481,C1(CC=C)(NC(C2C=CCC2)=O)CCN(C(c2ccc(C(N)=O)cn2)=O)C1 58482,c1(C(N2CCC(C(C)(C)C)(CNC(C3N(CC)CC3)=O)C2)=O)sc(C)c(C)c1C 58483,N1(CC2CN(C(C=CC=CCC)=O)C2)CCN(C(c2cnsn2)=O)CC1 58484,C1(NC(CCC2(NC(CC(C)C3CC3)=O)CCC2)=O)COCCC1(F)F 58485,N1(C(c2cn(C)nc2Br)C(=O)N(CCC(=O)OCC)CC)CC=CCC(C)(C)C1 58486,c1(-n2ncc(C(=O)NCCCOCCCNC(C3C(C)C3)=O)c2)cccc(O)c1 58487,n1(CC)ncc(Cl)c1C(=O)NCC(C)CNC(=O)Cc1cc(C)[nH]n1 58488,C1(N(C(CNS(NC)(=O)=O)=O)C)CCN(C(=O)CC2CCCCN2C(C)=O)CC1 58489,C1(C(=O)NCC(CNC(c2cc(O)ccc2F)=O)O)CCC2(CCC2)O1 58490,C(C(F)(F)C(F)(F)F)OCCC(=O)NCC(C)N(C(=O)CSCC#N)C 58491,N1(C(CCC)=O)CCC(C)(C(=O)NCc2ccsc2)C1 58492,C1(C(N2CC(OC)C2)=O)CCC=CC1NC(C1CCCN(C)C1)=O 58493,n1(-c2c(C(=O)NCCN(C)C(C3(C)C=CCC3)=O)cccc2)ccc([N+](=O)[O-])n1 58494,c1(C(C)(C)C)ccc(CONC(=O)NC(c2ccccc2)CO)cc1 58495,Cc1ccnc(CN(C2CC2c2ccccc2)C(=O)NCCCN2CCCCC2)n1 58496,c1(C(C)NC(=O)CC2CSC2)nocc1C(=O)NCC1CCC(C)C1 58497,C=CCN(CC=C)N1CCC(CC(=O)N(CCCO)C)CC1 58498,CC(C)(C#Cc1cn(CCOCCNC(C2CC2C(N)=O)=O)nn1)SC1CCCO1 58499,C#CCCC(O)C(=O)NCC(C1CCN(C(C2CCS(=O)(=O)N2)=O)CC1)(C)C 58500,Cc1nc(N2C3CCC2CC(NC(=O)C2=NOC(C)(C)C2)C3)c2ccsc2n1 58501,C#CC1(O)CCN(C(C2CC(C)CN(C(C3(C#C)CC3)=O)C2)=O)CC1 58502,C1(C(CNC(C(C)OCC=C)=O)(C)C)CCCCN1C(=O)CN(CC)CC 58503,Cc1ncn2ccc(C(N3CC(CNC(=O)C=CC(C)C)C4(CC4)C3)=O)cc12 58504,c1(C(=O)NC2CCCN(C(c3cc(CC)oc3C)=O)C2)cc(C)cc(Br)c1 58505,CC(C(=O)NCC(C1CC1)NC(=O)CNC(=O)C(F)(F)F)C(C)(F)F 58506,CCCN=C(NCC1(C)CCCc2ccccc21)N1CCC(OCC(C)C)C1 58507,CC(C)C(C)CC(=O)NCC(n1cc(CC2(O)CC(C(=O)O)C2)nn1)C 58508,C(CC(C)(C)C(=O)NCC1(F)CCN(C(C2(C)CC(C#N)C2)=O)CC1)OC 58509,c1(C(=O)NCc2cnc(CSC)n2C)ccc(=O)n(CCC#N)c1 58510,C(=O)(CCCC(C(=O)NCC(N)=O)C1CCC1)Nc1cccnc1 58511,C(=O)(C(C)CN(C(=O)C(C1CCOCC1)O)C)NC(COC)CO 58512,C(=O)(C(C)CC(F)F)NCC(CC)(CC)NC(=O)COc1ccc(C(C)=O)cc1 58513,c1(C(C)=O)cc(C(=O)N(C(C)CCNC(=O)C#CC(=O)N(C)C)C)oc1C 58514,c1(C(C(=O)NCC(O)CNC(C2(O)COC2)=O)N(C)C)c(F)cccc1Cl 58515,C1(C(N(C2CCN(CC)CC2)C)=O)CC(C)CN(C(=O)CN2CC=CC2)C1 58516,N1(C(C(C)OCCCC)=O)CC2CCC2(CNC(=O)C=Cc2cnc(C)s2)C1 58517,c1(CCC(=O)NCC2CC(NC(C(CC)SC)=O)C2)cn(C)nc1C 58518,C1(COC)(NC(=O)C=Cc2ccnn2C)CCN(C(=O)CC(C)(C)OC)CC1 58519,c1(C(N2C(C(N(CC(F)(F)F)C)=O)CC(F)(F)C2)=O)cc2ccc(Br)cc2s1 58520,N1(C(CC=C=C)=O)CCC2(NC(=O)CCc3ccc(OCC)cc3)CCCC12 58521,C=CC1(CC(=O)NCC(c2ccccn2)C)CN(C(=O)COCCCN=[N+]=[N-])C1 58522,C=CCC(CC=C)C(=O)N(C1CCN(C(C2CC3C=CC2C3)=O)C1)CC 58523,C1(CNC(C2(C#N)CC(C)C2)=O)CCN(C(c2cnnc(Cl)c2)=O)C1(C)C 58524,C(=O)(C(F)(F)CCC1CC1)NC1CCC(CNC(c2ccnc(OCC)n2)=O)C1 58525,C=CC1(c2nn[nH]n2)CCN(C(=O)C(N)Cc2cnc3c(c2)CCC3)CC1 58526,Cc1cc(CN(C)CCN(C(=O)CCc2conc2C)C)cc(C)c1Cl 58527,C#Cc1ccc(OCC(=O)NCCN(CCC)C(c2conc2C(C)C)=O)cc1 58528,Cc1cc(C(N2CCN(C3CC3)CC2C)C(=O)NCCC2(C)CC2)cnc1C 58529,C(=O)(C(C)CN(C(=O)Cc1cnn(C)c1)C)N(C(CC)CSC)C 58530,n1(CC)ncc(Cl)c1C(=O)NCC1CCCC1NC(C1(O)CC(C)(C)C1)=O 58531,c1(OC)cc(C(=O)NC2CCCCC2NC(=O)CCS(C)=O)cc(C)n1 58532,C1(C(=O)NCC(CO)C(F)(F)F)CC2CCC(C1)N2C(C1(F)CCCCC1)=O 58533,N1(C(C2(C)CC2Br)=O)CCc2nc[nH]c2C12CCN(C(C1CCCCS1)=O)C2 58534,c1(C(=O)NC(CC)CN(C(=O)C(C)C2=CCCC2)C)oc2ccc(C)cc2c1C 58535,c1(C(=O)NCCCN(CCCNC(C2CC(O)C2)=O)C)n[nH]c2c1CCCC2 58536,CC1CCC=C1C(=O)N1CCCCC1CCNC(=O)C(=Cc1cn(C)cn1)F 58537,CC1CN(C(CC2(C#N)CC2)C(=O)NCC2CCOC2)CC(=O)N1.C 58538,c1(N(C)C)ccc(C(=O)NCCC2(NC(=O)C(O)CN3CCCC3)CCC2)cc1 58539,C12(c3cn(CC(CC)C)nn3)COC(CN1C(c1nocc1Br)=O)C2 58540,c1(C(N(C2CN(C(=O)CCCN3C(=O)CNC3=O)C2)C)=O)n[nH]c2ccccc12 58541,N1(C(C(C2CCCCC2)NC(C(C=C)CC)=O)=O)CCCC(O)(C2CC2)C1 58542,c1(C(=O)NCCOCCNC(CS(CC)(=O)=O)=O)cc2sc(=O)n(C)c2s1 58543,C1(CCC)(C(=O)OC)CCCN1C(C1(c2ccccc2)CC(F)(F)C1)=O 58544,Cc1ccc(Cl)c(O)c1C(=O)NC1CCN(C(=O)CC(F)(F)F)C1C1CC1 58545,C1(C(=O)NC2CCN(C(COC)=O)CC2CO)C2CC3CC(C2)CC1C3 58546,C(=O)(C(C(C)(C)C)NC(=O)OC)N1CCC(F)(CNC(c2cn(CC)nc2)=O)C1 58547,CC1(C)OCC2CC12NC(C1(NC(c2cc(Cl)n[nH]2)=O)CC(F)(F)C1)=O 58548,C1(c2nc(-c3ccccc3I)no2)(OC)CCCCCC1 58549,CC(C)(CCNC(C1CCC(F)C1)=O)NC(=O)COCCN(C)C 58550,c1(C(=O)OC)ccc(C(=O)NC(C)CCNC(=O)C(=O)NC(C)C)c(Br)c1 58551,c1(OC)ccc(C(c2nnnn2C(C)(C)C)NCC2CC(C)C2)cc1OC 58552,Cc1ccc(O)c(C)c1NC(C1CCC(CNC(=O)COCC2CC2)C1)=O 58553,c1(C(N(CCNC(=O)CC2CN(C)CC2O)CC)=O)ccc2c(c1)OC(C)(C)C2 58554,N1(Cc2c(C(=O)OC)c(C)sc2)CC2CS(=O)(=O)CC2(C#N)C1 58555,CNS(=O)(=O)NCC(=O)N(C1CN(C(=O)Cn2nnc(-c3ccco3)n2)C1)C 58556,C12(C(N3CCN(C(c4c(C)coc4)=O)CC3CO)=O)CCC(N(C)C)(CC1)CC2 58557,C1(C(=O)NC(C#C)C(C)C)CCN(C(c2ccsc2OC)=O)C12CCC2 58558,N1(C(CCCC(C)C)=O)CC(NC(=O)CCC2(C)CC2)C2CCCC12 58559,C(=O)(C(C)(C(F)(F)F)Nc1ccccc1)N1CCCN(C(C(CC)(C)O)=O)CC1 58560,CC1(C)CN(C(=O)C=Cc2ccsc2)CC1CNC(c1sccc1C#N)=O 58561,CC(C(=O)N(C)CC1CCN(C(C2CCCC2)=O)C1)C(C)(F)F 58562,CCCC(C(=O)OCC)N1CCN(C(=O)C(C2CCCCC2)N)CC1 58563,C1(OCC)CC2CCC1(NC(C1N(C(c3cnn(C(C)C)c3Cl)=O)CCC1)=O)C2 58564,c1(C(N2CC(OC)(CNC(=O)C(CO)OC)C2)=O)ncc(Cl)cc1F 58565,c1(C(=O)Nc2cncc(Cl)n2)ccc(=O)n2c1COCC2 58566,C1(C)(CNC(C(COC)O)=O)CN(C(=O)C(C)(C)OCC(F)(F)F)CCO1 58567,C=C(Cl)CC(C(=O)N1CC(CO)C2(CC2)C1)NC(c1cc[nH]c1)=O 58568,N1(C(CC(C)F)=O)CCN(C(c2cc(Br)cn3ccnc23)=O)CC2(CC2)C1 58569,C(=O)(C1=CCN(C(c2cn(C)c(=O)cn2)=O)C1)NC1CC2CC(OC)C2C1 58570,N1(C(c2ccc(-c3ccc(S)cc3)cc2)=O)CCCC2CNCCCC12 58571,c1(C(C(=O)NCCN(C(=O)CCc2cnoc2)CC(C)O)O)ccc(Cl)cc1 58572,N1(C(C=Cc2cnc(C)s2)=O)CC2OCCN(C(=O)COCCCN(C)C)C2C1 58573,c1(CC)nn(C2CC2)cc1C(=O)NCCNC(c1cncnc1)=O 58574,c1(OCC)ccc(C(=O)N(C(C)CCNC(c2cscc2CC)=O)C)cc1C 58575,Cc1nc2ccccc2cc1C(=O)N(C1CCCC(N(C)C(C2COC2)=O)C1)C 58576,N1(C(c2cc(C(CC)C)no2)=O)CC2CCC2(CNC(c2ccc(OC)o2)=O)C1 58577,C=C(C)CCCC(=O)NCC(C)N(C)C(c1ccn(C(C)C)n1)=O 58578,Cc1ccc(C(=O)NCC2(O)CCCN(C(c3nnc(O)nc3O)=O)C2)c(N)n1 58579,N1(C(CC(CCC)CC)=O)CC(CO)C2(C1)CN(c1nccc(C(C)(C)C)n1)C2 58580,C1(C(N2CCC(COC)(CNC(c3cnc(O)s3)=O)C2)=O)CCC(C)=C(C)C1 58581,C(CCC(C)(C)C(=O)N1CCC(O)(C=C)C1)C1CN(C(C(C=C)CC)=O)C1 58582,C1(c2n(C(CC)(C)C)nnn2)(Nc2ccc3c(c2)OCO3)CCCC(C2CC2)C1 58583,c1(C(=O)NC2CC3(C(NC(c4occ(C)c4)=O)C3)C2)ccc2c(c1)C(=O)CCC2 58584,CCC(C)(CNC(C1CC(F)CN1C)=O)C(=O)NCCCc1cn[nH]c1 58585,N1(C(CCCC2C(C)C2)=O)C(C(=O)NC(C)(CO)C(C)(C)O)CCC12CC2 58586,C1(NC(C2(C(=O)NC)CC2)=O)CCCN(C(c2ccnc(C(C)C)n2)=O)C1C 58587,C=CC1CN(C(=O)CC2CCCCCCC2)CC1NC(C1CC(C(F)F)(OC)C1)=O 58588,CC1(C)C=C(C(=O)NCC(CNC(C2CC3(CCCO3)C2)=O)CO)C1 58589,C1(NC(=NCCC)NCCCc2ccccc2F)CCc2cnn(CCOC)c2C1 58590,C(C)(c1ccc2ccnn2c1Cl)=CCCC 58591,C1(CNC(c2cn(CC=C)nn2)=O)CN(C(C2(C(=O)NC)CC2)=O)CCC1C 58592,C#CC1(NC(C2C(CNC(=O)C(O)CCCCC)C2(C)C)=O)CCC(C)(C)C1 58593,N1(C(CC#C)=O)CCC2C(CCN2C(C2COc3ccccc3O2)=O)C1 58594,C1(C(=O)NC2CCN(C(c3nocc3C3CC3)=O)C2)C2CCCOC12 58595,C=C(Br)CC(C)(C)C(=O)NCC1CCC(NC(=O)COc2ccon2)CC1 58596,C12(NC(C(c3ccccc3)C)=O)CC(C1)N(C(=O)C(C)N1CCCC1)C2 58597,C(=O)(C1Cc2ccc(F)cc21)NCC1CC(N)(COC)C1 58598,C=CC(C)(CCOC)C(=O)NCCCCC(C)NC(=O)COC 58599,N1(C(c2c(F)ccc(OC)n2)=O)CCCCCC(NC(c2cncc(F)c2)=O)C1 58600,c1(C(=O)Nc2ccc(C(=O)NCc3n(C)ccc3)cn2)c(F)cc(O)cc1F 58601,c1(C(=O)OC)nc2c(s1)CCN(Cc1ccc(OC(F)(F)F)c(F)c1)C2 58602,Cc1nccn1CCCNC(c1nnnn1C1(C)CC1)C1CCCCC1 58603,CC(C)CC(CNC(c1cc(C(N)=O)co1)=O)C(=O)NCC(O)CC1CCCC1 58604,c1(C(=O)NCCN(C(=O)Cc2cc[nH]c2)C)ccc2c(c1)C(=O)NC2=O 58605,N1(C(C(C)CO)=O)CCCC2(NC(C3(CN(C)C)CC3)=O)CC2C1 58606,FCCCN=C(NCc1ccc(Cl)cc1)NCC1CC(=C2CCC2)C1 58607,C(=O)(C(C)C(C)NC(=O)CC1CN(C(c2cncn2C)=O)CC1C)OC 58608,C1(C(=O)NCC(=C)C(F)(F)F)CC(NC(=O)CCC#CC)C12CCC2 58609,c1(C(N(CC(C)NC(=O)Cc2cccnc2)CC)=O)nc2ccccc2s1 58610,c1(C(=O)NCCC(=O)N2CC(OCC(=O)NC3CC3)C2)ncncc1Cl 58611,Cc1oc(CNC(C2CCCC(F)C2)=O)nc1C(=O)NCc1ccc(O)cc1 58612,CC1(NC(=O)CC2CCCC2(F)F)CCCN(C(c2cnc3c[nH]nc3c2)=O)C1 58613,Cc1nc(N(C)CC2CCCN(C(c3ccco3)=O)C2)cc2nncn12 58614,C1(CC(=O)N(CC=C)CC)(OC)CN(C(=O)CCc2nc(C)no2)C1 58615,c1(CC(=O)N(C(CN(C(C=C(C)Cl)=O)C)C)C)cccc(OCC#N)c1 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58723,CC1CC(NC(=O)C(=O)NCC2CC2)CN1C(c1cnc(C(F)F)nc1)=O 58724,CC(C)C(CN(C)C)NC(=O)N(C(C(=O)O)c1cccs1)Cc1ccncc1 58725,N1(C(c2ncn(-c3ccn(C)n3)c2)=O)CC2CCN(C(c3csc(=N)[nH]3)=O)CC12 58726,c1(CC(N2CCCC(NC(c3cc(C)ns3)=O)C2C)=O)cc(Cl)c2c(c1)OCO2 58727,N1(CCNC(C2CC=C(C)CC2)=O)CCN(C=O)CC1=O.N1(CC)C(=O)CSC1=S 58728,N1(C(C(c2ccoc2)NC(c2ncc(F)cc2F)=O)=O)CC2CC1CC2O 58729,C1(F)(CNC(Cc2ccc(C)s2)=O)CCN(C(=O)CCC2CCCCO2)C1 58730,N(C1CCCc2cc(F)ccc21)C1CCC(C(F)F)CC1 58731,C1(N(C(Cc2c(C)non2)=O)CCO)CCCN(C(=O)C(F)CC2CC2)C1 58732,c1(C(=O)NCC2CC(NC(C(C(CC)C)C)=O)C2)c(C)ccc2ncccc12 58733,Cc1nnc(CCCC(=O)N(CC(O)CNC(c2ccc(CO)cn2)=O)C)n1C 58734,Cc1nc(CC(=O)NC(CO)C(C)NC(=O)C(C)Sc2nncn2C)n[nH]1 58735,C(=O)(CC(C)C(=O)NCc1cc[nH]c1C(=O)NCc1ncnn1C1CC1)OCC 58736,N1(C(C2CNC(=O)N2)=O)CC(NC(c2csc3cncn23)=O)C2CCCCC12 58737,C(=O)(CC(C)(C)C(C)(F)F)NCCNC(C1N(C(C)C)CCC1)=O 58738,c1(C(=O)NCC23N(C(=O)C(COC)OC)CC(CC)(C2)C3)ccc2ncnn2c1 58739,c1(CCN(C)C(=O)OC(C)(C)C)cnn(C)c1.c12cnc(s1)NC2 58740,N1(C(c2nc(CC)sc2)=O)CC(N(C(=O)CN=S(C)(C)=O)C)C2(CC2)C1 58741,C1(CCNC(C2C(CC)C2)=O)CCCCN1C(=O)C(=O)NCCOC 58742,C(=O)(C#CC1CCC1)NCC1(C)N(C(C(CC)CC2CCCC2)=O)CCC1 58743,N1(C(CC(C)C)=O)CCCC2C(CCCN2C(c2cc(C3(Cl)CC3)n(C)n2)=O)C1 58744,c1(C(=O)NCC(CNC(C2C(CC)C2)=O)O)ccc2nn[nH]c2c1 58745,CC(CC(C)Nc1csc(C(c2ccccc2)O)n1)NC(=O)C(F)(F)C1CC1 58746,N1(C(c2ccc(C=C)cc2)C(=O)NCCC)c2ccccc2C(C)C1C 58747,C(CNC(=O)Cc1ccc(F)cc1F)(CC(F)(F)F)NC(c1c(C)[nH][nH]c1=N)=O 58748,C1(CNC(CSCC)=O)CCCCCN1C(c1oc(CC2CC2)nc1C)=O 58749,N1(C(C(CCN(C)C)O)=O)CC2CC(NC(=O)CCc3cnccn3)CC1C2 58750,c1(OC)nc(-c2ccco2)ccc1C(=O)Nc1cnnn1C 58751,C1(C(=O)NCCCOCC#C)CCC2CCC1N2C(c1cccc(=O)n1C)=O 58752,C1(CCNC(CNS(NC)(=O)=O)=O)CN(C(c2cnccn2)=O)CCO1 58753,c1(C(=O)NCCNC(=O)CNC(=O)CC(n2cnnn2)C2CC2)ccc(Cl)cc1 58754,c1(NC(C2(CNC(C=Cc3ccc(C)s3)=O)CC2)=O)ccc(C)c(Cl)c1 58755,C(=O)(C(CNC(C1CC(N2CCCC2)C1)=O)Cc1ccc(O)cc1)OCC 58756,N1(C(C2(COC)CCCC2)=O)CCC(CNC(=O)CC2COCCO2)(OC)C1 58757,c1(NS(C)(=O)=O)cc(NC(=O)NCCCn2cnnc2)ccc1F 58758,N1(C(C2N(CC)CCC2)=O)CCC(CC(=O)NC2CCC(=O)N(C)C2)C1(C)C 58759,CN1CC(C(=O)NCCC2CN(C(c3cnn(C(F)F)c3)=O)C2)CC1=O 58760,N1(C(=O)OC(C)(C)C)CCOC(C(=O)N(CC#N)Cc2ccc(Cl)cc2)C1.N1(C)CCCC1 58761,CSC1=C(C(=O)NC2CCC(CNC(=O)CN3CCSCC3)C2)CCCC1 58762,Cc1cc(C(=O)NCC(C)(O)CNC(=O)Cc2ccn(C)n2)ccc1C(N)=O 58763,C1(C(=O)NCCc2n[nH]cc2C(=O)NC(C)C(C)SC2CC2)(CC)CCOC1 58764,C(=O)(C(C(C)NC(c1ncncc1Cl)=O)C(C)C)NCc1nccc(C)n1 58765,N1(C(CC2CCC(C)CC2)=O)CC2(CCC2NC(=O)C=Cc2cn(C)cn2)C1 58766,Cc1cccc(O)c1C(N1CC(N(C(=O)C(C2CCOCC2)C)C)C(C)(C)C1)=O 58767,S(=O)(=O)(c1ccc(NCCc2cc(C(F)(F)F)co2)c(Cl)c1)NC1CC(C)C1 58768,C(CC(=O)N(C)CCNC(=O)C(C1(C)CC1)NC(=O)C(C)C)OCC=C 58769,C1(O)(CNC(c2n(C(C)C)ncc2)=O)CCN(C(=O)CN2C(=O)CCC2=O)C1 58770,N1(C(C(C(C)C)SC)=O)CCC(C2CCN(C(=O)COC(C)C)C2)CC1 58771,C1(NC(=O)C=CSCc2ccco2)C2CC1N(C(=O)Cn1nnc(C3CC3)n1)C2 58772,CC(CN(C)C)C(=O)NC1CCC(CNC(C2(C)CC2Br)=O)C1 58773,C1(C(=O)NCC(CCNC(c2cnc(C3CC3)[nH]2)=O)OC)C(C#N)C1(C)C 58774,N1(C(C2(O)CCN(C(C3C=CC=CC=C3)=O)C2)=O)CC2OCC(CO)C2C1 58775,c1(NC(N2CCCC(NCCc3sccc3F)C2)=O)cccc(C(F)(F)F)c1F 58776,c1(C(=O)NC2(C(COC)O)CC2)nscc1Br 58777,C1(C(=O)NC(c2cnc(C)s2)C)(CC)CCN(C(=O)CCNC(=O)NC)CC1 58778,N1(C(C(C=C)OC)=O)CCCCC2(CCN(C(c3cnn(C4CC4)c3Cl)=O)C2)C1 58779,c1(C(C(=O)N(CC(C)O)CCNC(C2(OC)CC2)=O)OC)ccccc1 58780,Cc1ncccc1CC(=O)NC(COC(C)C)C(=O)NCC1(C(N)=O)CC1 58781,C1(CC(C)NC(C2(Cl)CC2(C)C)=O)CCN(C(c2c[nH]cc2Br)=O)CC1 58782,C(=O)(C(F)n1ccnc1)NCCCN(C(C1CCSC1)=O)CC 58783,C#CCC(C)(CC)C(=O)NCCC1CCN(C(=O)Cn2[nH]cnc2=N)CC1 58784,CCC(CC(=O)NC12CC(C(=O)NC3CC(OC)C3)(C1)C2)CC(C)C 58785,c1(C(=O)NCC(C)N(C(=O)CC(C(F)F)n2ccnc2)C)cc(O)ccc1OC 58786,Cc1cnc(F)c(CNC(C23CC(NC(=O)C(F)(F)CN(C)C)(C2)C3)=O)c1 58787,C1(NC(C(COC)C)=O)(COC)CCN(C(=O)COCC(C)(C)C)C1 58788,C#CCC(C)(C)C(=O)NCC1(O)CC(C(N2CCCCCCC2)=O)C1 58789,C1(OCC)CC2(C1)CC2C(=O)NCCCNC(=O)CCc1ncc(C(C)(C)C)o1 58790,Cc1c(F)cccc1S(=O)(=O)N1CC(NC(=O)Cc2ccccc2I)C(C#N)C1 58791,Cc1csc(CCCC(=O)NCCC2CC(NC(C3(C)CCOC3)=O)C2)n1 58792,C1(C(N2CC(NC(Cn3ncc(C#C)c3)=O)CC(C)C2)=O)(OC)CCC(C)(C)C1 58793,C1(C(N(C2C(C)COCC2)C)=O)CCOCCN1C(=O)CC(O)CN(C)C 58794,N1(C(CSCCC)=O)CCC(CNC(C2CC(O)(CCC(C)(C)C)C2)=O)C1 58795,c1(OC)cccc(C(N2CC(n3cc(CC(C)O)nn3)C(C)C2)=O)c1F 58796,N1(CC2(CC#C)CC2)CCC(NC(C2(CC#C)N=N2)=O)C(c2cnn(C)c2)C1 58797,C(=O)(C1=CCCOC1)N1CCC(COC)(NC(=O)CC2CCCN2C)C1 58798,c1(-c2ccn(CC)n2)cnc(NC(c2ccsc2C(F)F)=O)c(O)c1 58799,C(CNC(=O)CCC1CCCN1C)(CC(F)(F)F)NC(C(C)=C(CC)C)=O 58800,CCC(C)C(O)C(=O)NCCC1(NC(=O)CCCN(C)C(C)C)CCOCC1 58801,c1(C(C(=O)NCC2N(C(c3ccnc(C)c3N)=O)CC2)O)cc(F)c(F)cc1F 58802,C12(CNC(c3c(C#N)scc3)=O)CCC1CN(C(=O)CC1CC=CCC1)C2 58803,c1(NC(=O)C=CC(=O)OCC)ccc(C(N2CCC(CCC=C)C2)=O)cn1 58804,c1(COC)nc(N2CCCC2C2(NC(c3cnc(C)o3)=O)CCC2)cc(C)n1 58805,c1(C(=O)NC2C(NC(c3cc(C)sc3)=O)CCCC2)cc(F)cc(F)c1F 58806,c1(NCC2C(C)CCN(C(C3CCCSC3)=O)C2)cccc(F)c1[N+](=O)[O-] 58807,CC(N=c1[nH]c(N2CCOC(C3CCCC3)C2)nc2c1SCC2)c1ccncc1 58808,C1(NC(c2c(C)cno2)=O)CN(C(=O)C(C)(O)CC(C)C)CC12CCOCC2 58809,C1(OCCC)CCCN(C(C2(C(C)NC(c3cnc(C)o3)=O)CC2)=O)C1 58810,c1(C(c2nnnn2CC)NCC=C=C)ccc2ccccc2c1Br 58811,CC(C1=CCCCC1)n1ccnc1-c1ccc(-c2nn[nH]n2)cc1 58812,CC1(C)CN(C(=O)NC2CCCC3CC23)Cc2cccc(OC)c2O1 58813,C1(C(=O)Nc2cc(C(=O)OCC)no2)CCC2CCC1N2C(=O)CC=C(C)C 58814,C1(NC(C)CNC(C2CC2C2CCCC2)=O)CN(C(=O)OC(C)(C)C)CCN1C 58815,C1(CNC(C(COC)O)=O)CCCC12CCN(C(c1cn(C)ccc1=O)=O)CC2 58816,C1(C)(N(C)C)CCN(C(=O)C(Cc2cn[nH]c2)NC(=O)C2=CCCCO2)CC1 58817,C1(CCc2n(CC=C)nc(-c3ccccc3Cl)n2)CC(OCC)C12CCC2 58818,c1(CC(N2CCCC2c2cn(CC3(F)CCOC3)nn2)=O)c(F)cccc1Cl 58819,Cc1nc[nH]c1CC(=O)NCCOCCN(C(=O)CC1CS(=O)(=O)C1)C 58820,c1(C(=O)NC(CC)CNC(=O)Cc2cn(C)nn2)c(C)noc1C 58821,C1(C)(C(=O)NC(CNC(CC2N(C)CCCC2)=O)C2CC2)CCC2CC2C1 58822,N1(C(CC(C)C)C(N2CCS(=O)(=O)C(C)C2C)=O)C(=O)c2cccnc2C1=O 58823,C1(NC(c2cn(CCN(C)C)nn2)=O)CC(CNC(C2C=CCCC2)=O)C(O)C1 58824,c1(C(N2CC(CNC(=O)COCC3CC3)C(F)(F)C2)=O)cnn2cccc(Cl)c12 58825,C(CNC(c1cc(Cl)no1)=O)(CCNC(=O)C=C(C)C(F)F)OC 58826,C1(NC(COC(CC)(C)C)=O)CC2CCC(C1)N2C(c1csc(Br)c1)=O 58827,C1(CN(C2CC(O)(C(F)(F)F)C2)C)CCC2(CCCOC2)O1 58828,C1(C2CCN(C(=O)CC3CCC4CC4C3)C2)(NC(c2oc(C)c(CO)c2)=O)CC1 58829,N1(C(CC=CC=C)=O)CCCC2CN(C(c3cc(Br)ccn3)=O)CCCC12 58830,Cc1ccnc(C)c1C(=O)NC1CCCCC1NC(C1(C(F)F)CCCO1)=O 58831,N1(S(CC(=O)OCC)(=O)=O)CCC(F)(F)C(C(=O)N=c2[nH][nH]cc2CC)C1 58832,CC(C(=O)NC1CN(C(c2ccc([N+](=O)[O-])cc2Cl)=O)CC1O)C(F)(F)C(F)F 58833,Cc1cn2cccc(C(=O)N(C)CC3(NC(c4cnoc4C4CC4)=O)CC3)c2n1 58834,c1(C(N2CC(NC(C(CC)n3ccnc3)=O)C(C)CC2)=O)ccc2scnc2c1 58835,C1(CC(N2C(C)(CCC)CC2)=O)CN(C(c2cc(F)ccc2O)=O)CC12CC2 58836,CC(CC(C)(F)F)C(=O)NC1COCC1NC(c1cccc2c1COC2)=O 58837,C(=O)(CCC(C)(C)[N+](=O)[O-])N1CCC(CNC(c2c(C)con2)=O)C1(C)C 58838,Cc1cccnc1CC(=O)NC(CCC1CC1)C(=O)NC1(CO)CC(O)C1 58839,N1(C(c2c(C)nc[nH]2)=O)CCC(C2CCN(C(C34CSC(C3)C4)=O)CC2)CC1 58840,c1(SC)cscc1C(=O)N(CC(C)CNC(=O)CC(C)O)C 58841,N1(C(C#C)C)CCN(C(C2(CNC(=O)CN=[N+]=[N-])CC(=C)C2)=O)CC1 58842,N1(C(COc2cccc(C)c2C)=O)CCC(C2CC2NC(=O)CC(C)(C)F)CC1 58843,C12(C(N3CC(NC(COCCOC)=O)C3)=O)CC(c3ccccc3)(C1)C2F 58844,C1(C2CCN(C(C3(C)CC3(F)F)=O)CC2)(NC(CCc2ccn(C)n2)=O)CCC1 58845,C1(CCC)CN(C(=O)COC2CCOCC2)CC1NC(=O)CCc1nc(C)cs1 58846,N1(C(COCCN(C)C)=O)CCCC1CN(C)C(c1csc(C2CCCO2)n1)=O 58847,C1(C(=O)NC(CCC(=O)N(C)CC)C)CC(=O)C12CCC2 58848,C1(NCc2cccc(C)c2)CC(NCc2c(CC(=O)O)nn(C)c2)C12CCC2 58849,C1(CN(CC(=O)NC(c2ccccc2)CCC)C)CCCCC1C1CC1 58850,N1(C(C(Cn2cccn2)OC)=O)CC(C(N2CCC(O)C2)=O)C(C(C)C)C1 58851,c1(C(=O)NCC(C)(C2CC2)NC(C(C)SC)=O)cc(Br)c(C)o1 58852,CC1(F)CN(C(c2ccoc2Br)=O)CCN(C(c2cnccc2Cl)=O)C1 58853,CCC(C)C(O)C(=O)N1CCCC(CO)(NC(=O)CC2(C3CC3)CC2)C1 58854,C1(C(N2C(C)(CC)CC2)=O)CSCCN1C(c1ccc(COC)o1)=O 58855,N1(C(c2cc(C)oc2C)=O)CCC(NC(=O)C(C)Oc2cccc(N)c2)CC1C 58856,N1(C(CP(C)(C)=O)=O)CCOCC(CNC(C2CC(n3ccnn3)C2)=O)C1 58857,c1(SC)cccc(C(=O)NC2CCC(CNC(C3(C)COC3)=O)C2)c1Cl 58858,CC1(NC(c2nccnc2Cl)=O)CCN(Cc2ccccc2)CC1 58859,CC1CC(c2cn(-c3ccncc3)nn2)CCN1C(=O)CSC1CC1 58860,C(=O)(CCC(C)C#N)N1CCC(N(C(c2sc(CCC)c(CC)c2)=O)CC)CC1 58861,CC1CN(C(C2CC(=O)N(C3CN(Cc4cc(Cl)cnc4F)C3)C2)=O)CCN1C 58862,CC1(C)CC(C(=O)NCCOC2CCCC2)CN1C(CCC1CCC1)=O 58863,c1(NC(N2C(C(N3CCCC(C(F)F)C3)=O)CCC2)=O)cc(F)ccc1F 58864,C1(NC(=O)CCOCC(F)F)CC2CCC(C1)N2C(c1cc2c([nH]1)CCC2)=O 58865,c1(NC(C2(C)CCN(Cc3cn(CCC)nc3)C2)=O)cncc(Br)c1C 58866,c1(C(N(CCN(C(c2ccc(C#C)o2)=O)C)C)=O)ccc(C(F)(F)F)cc1O 58867,N1(C(CN(C(C)=O)C)=O)CCCCC1C1CCN(C(=O)C(C)CC2CC2)CC1 58868,N1(C(c2c(CC)cc(N)cc2)=O)CC(NC(=O)C(O)CC(N)=O)C(C2CC2)C1 58869,C1(NC(C2C(NC(C(C(C)O)N(C)C)=O)CC=CC2)=O)CCCC(O)C1O 58870,C12(C(N3CCC(CNC(C(C)SCC)=O)C3)=O)COCC1CS(=O)(=O)C2 58871,N1(C(c2cn(CCC)nn2)=O)CCC(NC(c2cn(C)cc2C)=O)CC1C1CC1 58872,C12(C(N3CC4C(NC(c5cccc(C)c5F)=O)C4C3)=O)CCCCC1OCC2 58873,Cc1oc(C)c(CN(C(=O)NCc2nc(-c3cccnc3)no2)CC2CCCO2)c1C 58874,C(=O)(C#CC1CCCCO1)NC1CCC(NC(c2sc(C)c(C)c2C)=O)CC1 58875,c1(C(=O)NC(C2(CNC(c3c(C)c(Cl)cnc3)=O)CC2)C)ccn2cncc2c1 58876,S(=O)(=O)(c1ccc(Br)cc1F)N1C2CCN(C(c3ncccc3Cl)=O)C2CCC1 58877,CCC(F)(F)CC(=O)NCC1CN(C(c2coc(C3CC3)n2)=O)CCCO1 58878,c1(C(N2C3CC(NC(C(C)P(C)(C)=O)=O)C2CC3)=O)cc(=O)n2nccc2[nH]1 58879,CC(CC(=O)NCC(CNC(=O)C=CC=C(Cl)Cl)CO)c1cnn(C)c1 58880,c1(N2CC3CC(NC(C=C(C)c4ccco4)=O)C3C2)ncc2c(n1)CCCC2 58881,N1(C(C(C)OC)=O)CCCC(O)(CNC(=O)CSC(C)(C)C)CC1 58882,c1(C(N2CCN(C(C3(CC=C)CC3)=O)CC2C2CC2)=O)ccc2c(c1)CCC=C2 58883,C12CCCC(C1)C(=O)NC1(C)CN(C1)C(=O)C2.Cc1nc[nH]c1CC(=O)N(C)C 58884,c1(CN(C2CCN(C(c3nn(CC)c(C)c3)=O)C2)C)cccc(C#N)c1 58885,C12CS(=O)(=O)CC1CNC2=O.c1(CCOCC(=O)NC2CCSC2)ccccc1 58886,C1(CNC(c2ncn(C(C)C)n2)=O)CC(C)CCN1C(=O)CP(C)(C)=O 58887,C(=O)(CC(C(F)(F)F)NC(=O)CC(C)C1CC1)NCCN(CCOC)C 58888,Cc1cc(C(=O)N(C2CN(C(=O)CCc3cnn(C)n3)C2)C)cn1C(C)C 58889,C1(C(N(C2CCCN(C(c3ccsc3)=O)CC2)C)=O)CC(F)(F)C12CCC2 58890,CCC(CN(C)C)CC(=O)NCC(CNC(c1ccc(N)c(F)n1)=O)S(C)(=O)=O 58891,c1(CNc2c(F)cc(C(F)(F)F)cn2)ccc2ncc(Br)cc2c1 58892,c1(C(CO)NC(C(C)C#N)=O)ccc(F)c(Cl)c1 58893,N1(C(CNC(CC)=O)=O)C2CCC1C1CC1(NC(=O)CC1COCCOC1)C2 58894,C(=O)(C(C)(CO)NC(C1CC(n2cncn2)C1)=O)OC 58895,C1(CC(=O)NCC(C2(O)CN(C(C(C=CC)O)=O)C2)(C)C)CCCC12CC2 58896,C(=O)(C(O)CC(=O)OC(C)(C)C)NCCCN(C(COCC#C)=O)C(C)C 58897,N1(C(C2(CC3CCC3)CC2)=O)CCCC(O)(CNC(C2(F)CCS(=O)(=O)C2)=O)C1 58898,c1(-c2cc(-c3nc(CCCCCC)nn3CCOC)ncc2)cc(F)cc(Cl)c1 58899,c1(C(N2C(C)C(NC(c3cccnc3S)=O)CC2)=O)ccc(F)c(S(N)(=O)=O)c1 58900,C1(N(C(=O)C=CCNC(=O)Cn2ccnn2)C)CCCCCC1O 58901,N1(C(c2cn(C)nc2C2CC2)=O)CCS(=O)(=O)C(CCNC(=O)CC(C)(F)F)C1 58902,CCC(CC)(CCNC(c1nnn(-c2ccc(Cl)cc2F)c1C(F)F)=O)OC 58903,n1(CC)ccc(C(=O)NCC2CN(C(c3cscc3OC)=O)C2)cc1=O 58904,C1(C(N(CCC(=O)NCC(C#C)CC2CC2)CC=C)=O)C2CCCCCC12 58905,N1(C(c2n(CC)ccc2)=O)CC(C)OC2(CCN(C(=O)C(=O)CC(C)CC)C2)C1 58906,CCCC(C)(C)CC(=O)NC1CC(C(F)C(N2CC3(CC(CO)CO3)C2)=O)C1 58907,N1(C(C2(CNC(CCN(C)C)=O)CCCO2)=O)CCSC(C)(C)C1 58908,C1(OC)CCC12CC(C(=O)NC1CC1NC(c1c(C)noc1C(F)F)=O)C2 58909,c1(OCCCC(=O)NCC2(O)CCN(C(C(=O)NCC)=O)C2)ccc(C)c(C)c1 58910,c1(OC)cc(C(N2CC3CC2CCC3NC(=O)CCS(N)(=O)=O)=O)c(O)c(Cl)c1 58911,C1(NC(C(C)N(C(c2cnn(CCO)c2)=O)CC)=O)CCCCCCC1 58912,c1(C(=O)NCC(CN(C(CCC(=O)NC)=O)C)O)ccc(OC)c(S(N)(=O)=O)c1 58913,C1(NC(c2c(OC)cncc2)=O)CCN(Cc2ccc(Br)[nH]2)CC1O 58914,C1(C(=O)NC(CNC(c2c(C)nn(CC(C)C)c2Cl)=O)(C)C)CN(CP(C)(C)=O)C1 58915,C#Cc1ccc(C(N2CCOC(C(C)NC(=O)C=CC(=O)OCC)C2)=O)cc1C 58916,C(CCC(c1ccccc1)(c1nnnn1C(C)C)NCc1ccc(C)nc1)OC 58917,c1(C(=O)NCCC2(CNC(CCC(C)OC)=O)CC2)cnn2ccncc12 58918,c1(C(=O)NC2(CCNC(C(CC#C)C3CC3)=O)CC2)ccc(C)cc1C 58919,C1(CNC(C2CC(SC)C2)=O)CCCCN(C(c2c[nH]c(=N)s2)=O)C1 58920,C1(C(C)(C)C)(CNC(C2(C)CCCS2)=O)CCN(C(c2ccc(F)s2)=O)C1 58921,c1(C(=O)NCC2OCCN(C(CCc3scc(C)n3)=O)C2)cc(O)c(F)cc1N 58922,CC(=O)CC(C)(C)CC(=O)N1CCCC1CCNC(=O)C#CC1CCCOC1 58923,CON(CC1CC1)C(=O)C(F)(CNC(c1cnnc(C)c1C)=O)C(C)C 58924,Cc1ccc(C(=O)NCC2CCC(NC(c3cnns3)=O)C2)cc1C 58925,N1(C(C(CC=C)C)=O)CC(C)(C)CC1CC(=O)NC1CCC(O)(CC)CC1 58926,C1(C2CC2)(C(=O)NC(CNC(C(C=C)O)=O)Cc2ccccc2)CCC1 58927,c1(C(N2CCN(C(C)=O)CC2c2cccc(F)c2)=O)cccc2ccn(C)c12 58928,Oc1c(CN2CCC(O)(CO)C2)cc(Br)cc1Cl 58929,N1(C(c2ncc(-c3ccc(C)nc3)cc2C)=O)CCC2(CC1)SCC(=O)N2C 58930,C1(C(=O)NCCNC(c2cc(CC)no2)=O)CC1C1CCC1 58931,C=CCN=C(NCc1nccc(C(F)F)n1)NCC(c1nc(C)cs1)C 58932,c1(C(=O)NCCOC2CCN(C(C3CC(C)N(C)C3)=O)C2)c(F)cc(F)cc1Cl 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58951,Cc1cccc(C(=O)N(C2CCCCC2NC(C2OCCCO2)=O)C)c1 58952,N1(C(C(C2CCC2)OC)C(=O)NC2CCOC2)C2CCC1CC(=O)NC2 58953,C1(CN(C)C(C2C3CC4C(C3)C24)=O)CCC(NC(c2ncccc2CO)=O)CC1 58954,N1(C(C(CC)NC(N)=O)=O)CC2(CCN(CC=CCCOC)CC2)CC1C 58955,N1(C(c2ccn(CC)c2C)=O)CCN(C(c2ccc(O)c(C)c2)=O)CC1C 58956,CN(NC(=O)C(N)CCC(=O)OC(C)(C)C)c1ncccn1 58957,c1(CNC(C(N2CC(C)C(F)(F)C2)c2nc(CC)[nH]n2)=O)ccc(F)c(F)c1 58958,c1(C(=O)NCCCN(C(CCOCC#C)=O)C)c(C)nc2sc(C)nn12 58959,c1(OC(C)=O)ccc(OCCC2CCCN(C(C)C)C2)cc1C 58960,C1(OC)CC2CCC(C1)N2C(=O)CC(CC(C)C)NC(=O)C(C)OCCC(C)C 58961,C1(C(=O)NC(CC=C)C(=O)NCC2CCCC(=O)N2)CC2(C1)CC21CC1 58962,c1(C(=O)NC(CNC(CSC)=O)(C)C2CC2)nc(O)[nH]c(=O)n1 58963,CCCCCC(O)C(=O)N1CCC2CCCC12C(=O)N(CC)OC 58964,c1(CCC(=O)NCCCOCCCNC(C(CC#C)C)=O)cccc(F)c1F 58965,n1(C(CC)C)ccc(=NC(=O)C(CC(N)=O)NC(c2cc(C(N)=O)c[nH]2)=O)[nH]1 58966,C1(NC(C2N(C)CC(O)C2)=O)C2CC3C(C2)C13C(N1CC(F)(C#N)C1)=O 58967,C1(CC(=O)NCCN(C(C=CCOC)=O)C2CC2)CC(C(F)F)(OC)C1 58968,c1(CC)ccc(F)c(C(=O)NC2CCC2NC(C2CCOC2C(C)C)=O)c1 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59006,C1(NC(c2cc(F)cc(F)c2)=O)CC2CN(C(=O)CC3CCSCC3)CC12 59007,N1(C(C(C2CCC2)OC)=O)CC2CCCC2(NC(c2cccc(SC)c2)=O)C1 59008,C1(CNC(C(=Cc2cccs2)C)=O)(Nc2ncn(C(C)(C)C)n2)CCCCC1C 59009,c1(C(N(C2CCC(NC(C(C)SCCCC)=O)CC2)C)=O)cc([N+](=O)[O-])ccn1 59010,CN=c1nc(N2CCC(C)(N(C)C)C2)[nH]c(=NCCc2ccccn2)[nH]1 59011,c1(C(N2CCCC(N(C(C(CC=CC)C)=O)CCF)C2)=O)cc(C)cc(C)c1O 59012,c1(C(=O)NCC(CC)NC(C2CCCC(F)C2)=O)c(OC)cccc1O 59013,c1(C(=O)NC(CNC(C(C2CCC2)OC)=O)C(C)(C)C)c(C)cc(C)nc1O 59014,C(=O)(C(O)CCCNC(=O)CC1(O)CCCOC1)N1CCC(C(C)OC)CC1 59015,c1(N(C)Cc2ccc(CO)cc2)ccc(S(=O)(=O)NC2CSC2)cc1Br 59016,C(c1ccc(F)c(F)c1)=C(C)C(=O)NCC(C)(O)CNC(C12CC(O)C1C2)=O 59017,C12(C(=O)NCC3(C)ON=C(C)C3)CC(CN(C(=O)CCC(C)C)C1)C2 59018,CCC(CC)C(C)C(=O)N1CCC(CCNC(C2CSCN2C(C)=O)=O)C1 59019,C(CC(C)C)(C(=O)NCC1CN(C(c2cccnc2O)=O)CCCO1)NC(C)=O 59020,C1(C(N(C(CCCC)C)C)=O)CC2CCC1N2C(c1n[nH]cc1Cl)=O 59021,C1(C(=O)NC(C2CCS(=O)(=O)C2)(C)C)CC2(CCC2=O)C1 59022,C(=O)(CCCC(=O)OC(C)(C)C)NC(CC1CCN(C(CCCCOC)=O)CC1)C 59023,Cc1ncc(C(N2C(C(=O)N(CCCCN(C)C)C)CCC23CC3)=O)c(C)n1 59024,C1(C(=O)NCCC2(C(=O)NCc3cc(C)ncn3)CC2)CC2CCC1CC2 59025,C(=O)(C1=CCN(C(C2CC2OC(C)=O)=O)C1)N1CCC(=C)CC1 59026,Cc1ncsc1C=CC(N1CCC(C(C)NC(C2C(C)(C)C2(F)F)=O)CC1)=O 59027,c1(C(N2CCOCC(NC(=O)CCCN3CCCC3)C2)=O)cn2ccncc2n1 59028,C(C)(CCC(=O)N(C1CCN(C(=O)C(F)(F)c2csc(C)c2)C1)C)SC 59029,C(=O)(C(O)CC(F)F)NCC(c1ccc(F)cc1)NC(CN(CC)CC)=O 59030,C1(CNC(C=C=C(C)C)=O)CCN(C(=O)Cc2ccoc2)CC1C 59031,N1(C(c2c(C)nc(C)s2)=O)CCCN(C(C2C(Cl)(Cl)C23CC3)=O)CC1C 59032,C1(CC=C)(NC(=O)CCN2CCCCC2)CCN(C(C2(C(=O)NC)CC2)=O)C1 59033,C1(C2CCCCC2)(NC(c2ccccc2SC)c2n(CC=C)nnn2)CC1 59034,C1(NC(C(C)Cc2ccccc2)=O)CC12CC(NC(=O)CCCC1CC1)C2 59035,CCC(C)C(C)C(=O)N1CC(N(C(=O)CCc2c(C)nn(C(C)C)c2C)C)C1 59036,c1(C(N2CCC(CCNC(c3ccc(COC)[nH]3)=O)C2)=O)cc(N)c(O)c(F)c1 59037,N1(C(C2CCN(C(C)=O)CC2)=O)CC2(CCC2NC(=O)CC2CCCCCC2)C1 59038,C1(CNC(N2C(C(C)O)CC2)=O)CCN(C2CCCCC2O)CC1 59039,C(c1cccc(F)c1F)=CC(N1CC(NC(c2nocc2Cl)=O)C(O)CC1)=O 59040,c1(C(=O)NC(C)CN(C)C(C2(C)CCCN2C)=O)ccc(=O)n(CCF)n1 59041,CCS(=O)CC(=O)NCC(C)(C1CC1)NC(=O)CC1CC(C)(C)C1 59042,c1(C(C(=O)N(CCCC(=O)NC)C)NC(C2CC(CF)C2)=O)c(C)cccc1Br 59043,C1(C)(NC(C(n2cc(Br)cn2)C)=O)CCCN(C(C2(O)COC2)=O)C1 59044,c1(N(S(=O)(=O)c2cc(Br)cc(Br)c2)CC)ccc2c(c1)CCC(=O)N2 59045,C(=O)(C(C)CS(=O)(=O)c1ccc(F)cc1)NCC1=CCN(C(CC=CC)=O)CC1 59046,C1(C)(C(N(C)CC2CCN(C(c3ccon3)=O)C2)=O)CCCN1C 59047,CC(C)CC(O)CNC(C1(CCNC(=O)CC=CC(C)(C)C)CCC1)=O 59048,n1(CC)cc(Br)c(C(=O)NCC(O)CCNC(c2[nH]c(O)nc2C)=O)n1 59049,CC(CC(F)(F)F)C(=O)NC(CCF)C(=O)NCC1CCC(=O)O1 59050,c1(C(CC)C(=O)NC(C)(C)CCNC(=O)CSc2nc[nH]n2)cccc(Cl)c1 59051,N1(C(c2ncn(C)n2)=O)CC2CC(NC(=O)C=Cc3cccs3)CC(C2)C1 59052,C1(N(C(CN(CC#C)C(C2CCSC2)=O)=O)C)CCCOC1 59053,C12(C(=O)NC(C)C(=O)NC(C)(C)C)CC(CCO1)N(C(=O)C(C)N(C)C)C2 59054,C1(C(N2CC(C)(NC(c3cncc(-n4ccnc4)n3)=O)C2)=O)CCC2CC1CO2 59055,C1(CNC(C(C)OCC#C)=O)(CO)CC12CCN(C(=O)CC1CC=CC1)CC2 59056,Cc1nc(C(N2CCSCC2C(=O)NCc2ccncc2)=O)ccc1Br 59057,N1(C(C2C(=C)CC2)=O)CCC2(CCC2CNC(=O)C2=CCOCC2)CC1 59058,C=CCC(C(=O)N(C1CCCCN(C(=O)Cc2cccnc2OC)C1)C)C(C)C 59059,c1(C(N2CC(NC(C3(CC)CCNC3=O)=O)C(F)C2)=O)ccc2ncn(C)c2n1 59060,CC1CCCc2cc(C(=O)NCCCNC(C3CCC4(CCC4)OC3)=O)nn21 59061,N1(C(CC(C)N(C)C)=O)Cc2nccn2CC(NC(=O)Cc2cnccc2Cl)C1 59062,N1(C(c2ccc(C)c(F)c2F)C(=O)NCCOC)CC(C)OC2CCCCC12 59063,Cc1n[nH]c(C)c1CC(=O)NCCC(C)NC(c1coc(-c2ccccn2)n1)=O 59064,C1(CCN(C)C(C23CC(F)C2C3)=O)CCN(C(C2CC3CC3C2)=O)CC1 59065,c1(C(N2CCC(F)(CNC(c3cn(C)nc3Cl)=O)C2)=O)coc2ccc(F)cc12 59066,c1(C(N2C(CNC(C3CC34CC4)=O)C=CC2)=O)cc([N+](=O)[O-])ncc1Br 59067,c1(OC)ccc(Cl)c(CNC(C2CN(Cc3ccc(C(F)(F)F)cc3Br)C2)=O)c1 59068,c1(C(=O)NC2CCN(C(C3(C#N)CC4CC4C3)=O)CC2)ccnc2ccccc12 59069,C1(C(=O)NC2(C3CCCN3C(c3ccoc3)=O)CC2)CC12CCOC2 59070,C1(C(N2CC(NC(C(CC=C)(C)C)=O)CC3(C2)CC3)=O)CCc2nnnn2CC1 59071,C(C(CO)(CO)NC(=O)C(C)Cc1cnc[nH]1)N(C(C(C)OC)=O)C 59072,CCCC(C)(CCC)C(=O)N1CCCCC1C(N1CCCC(C)(C)C1)=O 59073,N1(C(C(C(C)NC(C(=O)NCC)=O)C)=O)CC2CCC(C1)O2 59074,N1(C(c2ccc3cc[nH]c3n2)=O)CC(C2CCN(C(c3n[nH]cc3Cl)=O)CC2)C1 59075,N1(C(C2C(=C)C2COC)=O)CC=CC1(C(=O)NCC(C)(C)O)C(=O)NC 59076,N1(CC(=O)N(CC(c2ccccc2)C)C)C(=O)C=CC1=O 59077,N1(C(c2ccc(C)cc2F)C(=O)NCC(F)F)CCC2(CCCNC2=O)CC1 59078,C1(C)(C(N(CCCO)C)=O)CC12CCN(C(C1CC3CCC1O3)=O)CC2 59079,CC1CN(C(C2CCN(C)C2=O)=O)CC(C)CN1C(c1cc(O)cs1)=O 59080,CCCC(CCC)CC(=O)NCC(O)CNC(c1sccc1CC)=O 59081,c1(C(=O)NC(CNC(C2CC(OCC)C2)=O)(C)C)cc(Cl)c(Cl)cc1OC 59082,CN1CCC(C(=O)NCCC2(O)CCN(C(=O)CCC3CC3(C)C)C2)CC1 59083,c1(NC(C2(c3cc(F)cc(F)c3)CC2)=O)cc(F)c(CO)c(F)c1 59084,CC1(CNC(=O)C=CC(=O)NC2CC2)CCCN(C(=O)CC(F)(F)Cl)C1 59085,C(N=c1[nH]c(=NC2CC3CC4C(C3)C24)c2ncccc2[nH]1)c1cn(C)nc1Br 59086,O=C(C#CCNC(C1CCC(=O)O1)=O)NCCOCCF 59087,S(=O)(=O)(c1ccc(=NCCn2cccnc2=O)[nH]c1)NCC1C(C)CC1 59088,C(=O)(C1CCc2cccnc21)N1CCC(CNC(=O)C2=COCCO2)C1 59089,c1(NC(C(CC)N(C2CC(OC(C)C)C2)C)=O)cn(C)cc1C 59090,c1(CC)ccc(C(=O)Nc2ccc(NC(=O)CC3(O)CN(CC)C3)cc2)cc1 59091,C1(NC(c2cc3ccsc3[nH]2)=O)CC2CC(C1)N(C(C1Cc3nccn3C1)=O)C2 59092,C(c1ccc([N+](=O)[O-])s1)=CC(=O)NCC1CN(C(C(C)N(C)C)=O)CC1O 59093,c1(C(=O)NC2CC(NC(=O)COc3ccc(F)cc3)C2)ccc(Br)c(Cl)n1 59094,C(=O)(C(CC)C(C)(C)CC)NC1CCC(CNC(c2ccc(C#C)o2)=O)CC1 59095,C1(NC(CC(C)n2cccn2)=O)C2CCC1CN(C(=O)C(=O)NCC(F)F)C2 59096,C1(C(=O)NC(CCCNC(Cc2cc(C)ns2)=O)C)CCN(C)C(=O)C1 59097,Cc1c(C(=O)NCC#CCNC(=O)CC2CCCC2(F)F)sc2ccccc12 59098,c1(CNC(c2ccc(OC)cc2OC)CC(=C)C)ncc(Cl)cc1Cl 59099,C12(NC(c3cccc(Cl)c3)=O)CCCCC1N(C(c1ccncc1)=O)CC2 59100,O=[N+]([O-])c1cncc(-n2ccc(Nc3ncnc4ccsc34)n2)c1 59101,Cn1nc(Cl)c(C(=O)NC2CCN(C(=O)CCC(C)(C)C)C(C3CC3)C2)c1Cl 59102,C#Cc1cc(C(=O)NCC2(NC(=O)CC3OCCO3)CC2)cc(C(F)(F)F)c1 59103,c1(CNC(COCC(=C)C)=O)csc(CNC(=O)Cc2cncnc2)n1 59104,c1(N2CCC(NC(C(C3CC3)OCC)=O)(CF)C2)ncc(Cl)c(O)n1 59105,N1(C(C(N2CCCCC(CN)C2)=O)=O)CCC2(CC1)CC2(F)F 59106,C1(CCNC(Cn2ccc(C)n2)=O)C(C)CCCN1C(=O)COc1cnn(C)c1 59107,c1(C(=O)NC2CCCC(NC(c3c(C(C)C)nn(C)c3)=O)C2)nccc(Cl)c1O 59108,C1(NC(c2cc(C)nn2C2CCC2)=O)Cc2ccccc2N(C(=O)C=CI)C1 59109,c1(C(N(C)CCN(C)C(c2cncs2)=O)=O)ccc(F)c(S(=O)(=O)NCC#N)c1 59110,N#CC1CCN(C(C2(NC(c3ccoc3)=O)CCOCC2)=O)C1 59111,n1(C(C)(C)C)nnnc1C(C1CC1C1CC1)NCCc1noc(C(F)F)n1 59112,C1(C#N)(C(N(C(CNC(CCSCCCC)=O)C)C)=O)CC2CCC1C2 59113,C1(N(C(=O)C(N)=O)C)CN(C(=O)Cc2cnn(C(F)F)c2)CC12CC2 59114,C1(N(C(=O)C(=O)NC(c2cccc(OC)c2)C2CC2)CC)CCS(=O)(=O)C1 59115,c1(C2CCN(C(c3ccn(CCF)n3)C(=O)NCC(C)C)C2)cccc(Br)c1 59116,CC1(C)CCCC(CC(=O)NCCC2CCCN2C(=O)CN=S(C)(C)=O)O1 59117,N1(C(c2ccn(C(C)C)n2)=O)CC(C)CN(C(=O)CS(=O)(=O)C(C)(C)C)C(C)C1 59118,c1(CNC(C(COC)(C)C)=O)nnc2n1CCN(C(=O)CC(C)(C)C(C)(F)F)C2 59119,C1(NC(CNC(C)=O)=O)CC(NC(c2cnc(CC3CC3)s2)=O)C12CCC2 59120,N#CC1(C(=O)NCC2CC(O)CN2C(c2cnc[nH]2)=O)CCCO1 59121,C1(C(N(C2(C(F)(F)F)CCC2)C)=O)CS(=O)(=O)C12CCN(C(=O)OC(C)(C)C)CC2 59122,C#CC1(OCC(=O)NC(C)CC2CN(C(=O)CCOCC(=O)NC)C2)COC1 59123,c1(-c2cn(CCN(C(C3CC(CF)C3)=O)CC)nn2)cc(F)ncc1Cl 59124,C1(NC(c2c(C)[nH]cc2)=O)CCCCC1NC(=O)C(c1ccc(Cl)s1)C 59125,c1(NCC)ncc(C(=O)N(C)CCN(C(=O)C(C2(O)CCCC2)F)C)cc1Cl 59126,n1(CCC)cc(C(=O)NC2CCCN(C(=O)COCC(F)F)C2)c(C)n1 59127,C12(CNC(C3CCC3)=O)CCCCC1CN(C(c1ccc3c(c1)OCCO3)=O)C2 59128,S(=O)(=O)(c1ccc(NC2CCCC3(CCCCC3)C2)c(C#N)c1)NCC(CC)C 59129,c1(CNCC2C(C)CC2)oc(C(=O)O)cc1Br 59130,c1(C(C(=O)NC2CCC2)N(CCC2=CCCCC2)C)cc2cc(Cl)ncc2o1 59131,N1(C(c2c(OCC)nsc2)C(=O)Nc2ccccc2)CCN(CCC#N)CC1 59132,n1(C(C)C)cnc2c(NCC3CCC3(F)F)nc(N3CCN(C)C(C)C3)nc12 59133,c1(N2CC(C(c3ncccn3)CCC)C2)cc(Br)c(F)cc1C#N 59134,C(C(CC(C)C)C(=O)NCCc1ccn(C)n1)NC(C(CCOC)C)=O 59135,C(=O)(C(O)CN(C)C)N(CC(CC)NC(=O)C(n1cc(C)cn1)C)C 59136,N1(C(Cc2ccc(OC)nc2)=O)CCC(C)C(NC(C2(OC)CCSCC2)=O)C1 59137,CCCCCCC(C)C(=O)N1C2CCC1CC(N(C)C(c1nc(C)oc1C)=O)C2 59138,c1(Cc2nc(C(C)OC)nn2-c2ccn(C)n2)ccc(Cl)c(Br)c1 59139,N1(C(C(C)NC(C)=O)=O)CC(NC(c2cc(C(C)C)[nH]n2)=O)C2CC2C1 59140,C(C(CC1CCCC1)C(=O)NC1CCC(O)C1)NC(=O)CC1(CO)CC1 59141,c1(C(N2CCC(CNC(C3C(C)OCC3)=O)C2)=O)cnn2ccn(C)c12 59142,C12(NC(C(C=C)CC)=O)CCC(C(=O)NCCCn3cnnc3)(CC1)C2 59143,CCS(=O)CC(=O)N(CC(C)CNC(=O)CCCSC(C)(C)C)C 59144,CC1CN(C(=O)Cc2ccnn2C2CCOCC2)CC1NC(=O)Cn1ncnn1 59145,c1(N(C)C)cc(-c2ccc(C(=O)NCC3COCCO3)nn2)cc(C#N)c1 59146,C(CC(C(=O)NC(CC1CCC1)CO)NC(C1CC(OC2CC2)C1)=O)SC 59147,S(=O)(=O)(c1cccc(N(C)Cc2scnc2C)n1)N1CCC(OCC=C)C1 59148,c1(C(=O)NC2CC(CCNC(=O)CN3C(=O)CNC3=O)C2)nnn2c1CCCC2 59149,C(N=c1[nH]c(=N)[nH]c(=NCCS(=O)(=O)CCO)[nH]1)C1(C=C)CCOCC1 59150,S(=O)(=O)(CCC(F)(F)F)N1CCC(CNC(c2cnc(Cl)cc2I)=O)C1 59151,N1(Cc2cccc(OC)c2F)Cc2ccccc2C1C(=O)N1CCOC(CO)C1 59152,c1(C(=O)NC2CN(C(C3N(CC)CCCC3)=O)C2)cc(C)c(Cl)cn1 59153,c1(CCCC)cc(C(=O)NCC2(NC(=O)C=Cc3cocn3)CCOC2)c(C)o1 59154,c1(OC)ccc2occ(C(=O)NC3CCCCC3CNC(=O)C=CC(C)C)c2c1 59155,C1(C(=O)NCC(CCOC)NC(c2cc(C3CC3)on2)=O)(C(F)F)CCCCC1 59156,C(=O)(CCC(=O)NCC(C)(CO)NC(C1CCC12CCC2)=O)N(CC)CC 59157,c1(C(=O)NCCCN(C(=O)C(F)(F)CO)CC)ccc(=O)n2c1COCC2 59158,c1(C(=O)NCCC(C)N(C(Cc2cc(C)no2)=O)C)c(C(F)F)cnn1C 59159,C(C(C(=O)NCC(C)(O)CN(C)C)N(C)C)NC(C(C)NC(=O)CC)=O 59160,N1(C(CS(=O)(=O)NCC)=O)CCCC12CCN(C(=O)C(c1ccccc1Cl)O)C2 59161,C(=O)(CC(F)(F)CC(=O)N1CCN(C)CC1CNC(=O)CC(C)(C)OC)OC 59162,c1(C(N2CC(NC(C(C(C)C)(C)C)=O)C(C(F)(F)F)C2)=O)ccc2nccn2n1 59163,C1(CC)(CNC(c2nnnn2C(C)(C)CC)C2CCOC2)CCCCCC1 59164,C12(C(=O)NC3C(NC(c4cccc(OC)n4)=O)CCC3)CCCCC(OC)(C1)C2 59165,C1(CC)(CC)CCCN1C(C1CCN(C(=O)Cc2ccn(C)c2)C1)=O 59166,N1(C(C(C)OCCC#C)=O)CCCC(NC(C2(C(C)(F)F)CC2)=O)CC1 59167,C(=O)(CCC(F)(F)F)NC1C=CCN(C(C(CC#C)C2CC2)=O)C1 59168,C1(NC(C2C3(CC3)C23CC3)=O)CCN(C(=O)CN2CCOC2=O)CC(O)C1 59169,N1(C(CN(CCOC)C)=O)C2CCC(C2)C1CNC(=O)Cn1nc(C)oc1=O 59170,C12(CNCC3(N)CCC3)CC3CC(CC(C3)C1)C2 59171,C1(NC(c2nc(CCC)sc2)=O)CN(C(=O)COc2cccnc2)CC(C)(C)C1 59172,Cc1ccc(Br)c(C(N2CC3(CCNC(c4ccccc4)=O)CCC2C3)=O)n1 59173,C(=O)(C1=NOC2COCC12)NCCC1=CCOCC1.C12COCC1N2C(=O)CC1CC1 59174,Cn1nc(C(N2CCC(C(N3CC(c4ccccc4)C3)=O)C23CC3)=O)cc1C#N 59175,C(=O)(C(C)(C)CNC(C1CC(C)N1C(=O)CCc1cnco1)=O)OC 59176,N1(C(c2cc(CC)c(CC)o2)=O)CC(C2CN(C(=O)C(C)(O)CC)C2)C1 59177,c1(NC(COC(C(CC)Sc2ccccc2)=O)=O)c(C)nn(C(C)C#N)c1C 59178,C(=O)(C1=NOCC1)NC(c1ccccc1)C(C)NC(c1c(CCC)nns1)=O 59179,C(c1ccc(Cl)cc1F)=CC(N1CCCC(C)(CNC(c2ccc(F)s2)=O)C1)=O 59180,C(CCCCC(=O)NC(CC1CC1)CO)NC(c1cc(OC)ns1)=O 59181,Cc1cc(C(N2CCC3(CC2)CC3CNC(C2CCO2)=O)=O)c2c(C)noc2n1 59182,C1(NC(CCC=C)=O)CN(C(=O)C(C)CN(C)C)CC1OCC 59183,Cn1c(O)nc2cc(C(N3CCC(CCNC(=O)CCCC#N)C3)=O)ccc12 59184,Cc1ccc(C)n1CC(N1CCCC1CCC(N1CCCC(F)C1)=O)=O 59185,C1(C)(CC)CCC(C(=O)NNC(=O)c2cnsn2)O1 59186,c1(N2CC3CC(C)(C)C3C2)nc(=NCCc2cccc(F)c2)[nH]c2c1COCC2 59187,c1(C(=O)NC(CNC(C2CN(S(CC)(=O)=O)C2)=O)CCOC)cc2n(n1)CCO2 59188,C(=O)(C(c1ccccc1)=CC(C)(C)C)NC12C(CN(C(CCCOCC)=O)C1)C2 59189,c1(NC(CC2CCN(Cc3ccc(C)o3)C2)=O)ccc(F)cc1C#N 59190,C1(C(N(C2(C(=O)OC)CC2)C)=O)CC(C)N1C(c1ncn(C)n1)=O 59191,CC(CC(N)=O)C(=O)NC1CCCC1NC(c1cc(N(C)C)ccn1)=O 59192,Cc1ccc(Cl)cc1-c1cn(CCCNC(=O)CCNC(N)=O)nn1 59193,c1(OCCCC(=O)NC2C(NC(C3CC(CC)(CC)C3)=O)C2)c(C)cccc1C 59194,N1(C2CCN(C(CCCOCC=C)=O)C2)CCN(C(c2ccc(Br)o2)=O)CC1 59195,C(=O)(C(F)C(C)(C)O)NCC(=O)NCC(F)F.C(C1C(=O)N1)N(C)C 59196,C12(NC(c3nc(C(C)C)oc3)=O)CCCC1CN(C(=O)CN1CC3CC3C1)C2 59197,c1(CC)nccnc1C(=O)NCC(C)(CO)NC(c1c[nH]c(C#N)c1)=O 59198,S(=O)(=O)(c1cccc(F)c1Cl)Nc1ccc(C=C)cc1 59199,c1(C(N2C(CNC(C3(C=C)CCC3)=O)C(C)CCC2)=O)ccc2c(n1)CCCC2 59200,c1(CN2C(C(=O)Nc3c(C(C)=O)cccn3)CC3CC32)c(C)cc(Br)cc1C 59201,c1(C(=O)C(=O)NC2CC(CF)C2)ccc(Br)cc1F 59202,c1(C(N2CC(NC(c3ccco3)=O)C(F)C2)=O)ccc(Cl)c(F)c1F 59203,c1(COC(C)C(=O)N(C)CC2CCS2(=O)=O)cn(CCCC(=O)O)nn1 59204,C(=O)(CC1CCc2ccccc21)NCCC1CN(C(c2c(C)onc2)=O)CC1C 59205,c1(OC)ncc(C(=O)N(C(C)CN(C)C(C2(C)CC3(CCC3)C2)=O)C)cc1Cl 59206,C(C#Cc1ncccn1)N1CCC(OC(C)(C)C)C1 59207,C(CCC1CCC1)(C(=O)NC(c1nccn1C)CC)NC(CC=CCC)=O 59208,CCC(C)CC(C(=O)OC)NC(C12CC(C)(C1)OC2CN)=O 59209,C=C(C)CC(C(=O)N1CCC(CCCC)C1)NC(=O)C(C1CCOCC1)F 59210,c1(CC(=O)NC(C2(CNC(=O)C=CCN3CCCC3=O)CC2)C)nonc1C 59211,N1CCCC(C=O)C1.Cc1cc(C(C2CN(C3COC3)C2)=O)on1 59212,C1(C(N(CCNC(C(c2c(OC)cccc2)(C)C)=O)C)=O)CCCCNC1=O 59213,C1(C(N2C(CC(=O)NC(C=C)(C)C)CCCC2)=O)CCC(=O)N(C)C1 59214,C(=O)(C1=NN(C)C(=O)CC1)N1CCC(N(C(c2c(C)nns2)=O)C)C1 59215,N1(C(c2c(OC)c[nH]n2)=O)CCC(NC(=O)C=Cc2cccc(F)c2)C(CO)C1 59216,c1(C(N2CCC(C(=O)OC)CC2)=O)n[nH]c2c1CN(C(=O)C(C)(C)F)C2 59217,N1(C(c2coc(C3CC3)n2)C(=O)NC(C)C)CCCN(C(C)C(=O)N(C)C)CC1 59218,c1(C(=O)NC(CC)CN(C)C(C2CCOC(C)(C)C2)=O)ccc(=O)n2c1CCC2 59219,N1(Cc2c(OC)cccc2)CCC2(CC1)CC2C(N1CCCC1C(C)C)=O 59220,N1(C(CCC2N(C(CCN=[N+]=[N-])=O)CCCC2)=O)CC(C2CCCOC2)C1 59221,Cc1occc1CC(=O)N(CCNC(=O)C(C)n1cccc1)C(C)C 59222,C1(NC(c2c(C)sc(Br)c2)=O)CC2CCCC(C1)N2C(C12CC(C1)C2)=O 59223,C12(CNC(C3CCN(C4CCCCC4)C3)=O)CCC1CN(C(=O)CC1CCC1)C2 59224,Cc1ccc(CNC(C2CCCN(C(C3CC4CCC3C4)=O)C2)=O)c(O)c1 59225,Cc1nc(C(=O)NC2CCCC2(C)CN(C(=O)C(O)CC(C)C)C)cc(O)n1 59226,N1(C(Cc2c(C)nc[nH]2)=O)CCC2(CCCN(C(C3CN(C4CCC4)C3)=O)C2)C1 59227,N1(C(CCC=C)=O)CCSCC1C(=O)NCCOC1CCOC1 59228,N1(C(C2(CCC)CCC2)=O)CCN(C(C2CC3CCCC23)=O)C(C2CC2)C1 59229,C(CS(=O)(=O)c1ccc(C(=O)NC2CC2NC(=O)CCSC)cc1)OC 59230,C(C)(CCC(C)(C)C)NC(C1CCC(NC(c2c(CC)nn(C)c2)=O)C1)=O 59231,C1(C(=O)OC)CCC2(CC2)N(C(C2CCC3(CCC3)C2)=O)C1 59232,N1(C(C=C(CC)CC)=O)CC(C)C(NC(=O)CCc2cncnc2)C(C)C1 59233,CC1=C(C(=O)NCC2CCCN(C(c3coc(C(F)F)n3)=O)C2)COCC1 59234,C1(C(C)NC(c2cc(Cl)c[nH]2)=O)CCCN(C(=O)CC23CCC(CC2)C3)C1 59235,c1(OCC)cc(Br)c(NC(=O)C=Cc2ccc(C)nc2)c(Br)c1 59236,N1(C(C2C(CC)CCO2)=O)CCC(C(=O)NC(CN(C)C)C(C)(C)C)C12CCC2 59237,C(=O)(C1=CC2C=CC(C1)C2)N(C(CCC=C)C(=O)Nc1ccccc1)C 59238,Cc1nc(C(C)(C)C)c(C(=O)NCC2(NC(=O)CC3(O)CCCOC3)CCC2)s1 59239,N1(C(C2CC(C(=O)OC)C2)=O)CC(C(F)(F)F)OCC1CNC(=O)CCSC 59240,c1(CC)ncc(C(=O)NC(C2CCCN2C(c2cnn(CCOC)c2)=O)C)s1 59241,c1(C(=O)NCC2(F)CC(NC(C(C)NC(C)=O)=O)C2)ccc(C)c(S(C)(=O)=O)c1 59242,N1(C(CC(C)N(C)C)=O)CCCCC1CC(=O)NCC1COCCO1 59243,c1(OC)ccc2nccc(C(C)Sc3c(F)cccc3I)c2c1 59244,C1(C(N(c2cnn(C(F)F)c2)C)=O)CN(C(C2CC(CF)C2)=O)CCC1(C)C 59245,C1(NC(C=CC(C)(C)SC)=O)C2CCN(C(C3CC(=O)NC(=O)C3)=O)CCC12 59246,C1(C(N2CC(OC)C(O)C2)=O)CC(O)C(O)CC1CNC(=O)Cc1cncn1C 59247,c1(NC(C2CC(O)(CNC(c3cocn3)=O)C2)=O)ccc(Cl)cc1O 59248,N1(C(c2n(CC)nnc2)=O)CCC2(NC(=O)Cc3cc(Cl)sc3Cl)CC2C1 59249,N(C(=NCC1CCCO1)NC1CCN(c2cccs2)CC1)CC1(CCC)CCC1 59250,C1(NC(CC2CCC(=O)NC2)=O)CCN(C(=O)CC2C=CCCC2)C12CCC2 59251,C#CCCC(C(=O)NC(CCC)C(=O)NC)NC(=O)C(F)C(F)(F)F 59252,N1(C(C2(C)CC=CCC2)=O)CCC2(CC(C(=O)N3CCCC3C(N)=O)=NO2)C1 59253,C1(C(=O)NCC2CC(NC(c3cc(C4CC4)ccn3)=O)C2)CCc2ncsc2C1 59254,c1(C(N2CCC(O)C2)=O)cnc2c(-c3ccc4[nH]ccc4c3)cccc2c1 59255,C1(=CC(N2CC(C(C)C)N(C(=O)CCCC3CC3)CC2)=O)CCCCCC1(F)F 59256,C1(NC(C2CCN(C)C2)=O)CC2(C1)CC1(CC(NC(C3(C)CC3(F)F)=O)C1)C2 59257,C(=O)(C1=Cc2ccccc2C1)N1C(CC)C(NC(=O)C(F)(COC)C(C)C)CC1 59258,N1(C(C2CCCC3(CC3)C2)=O)CCC2(CC1)CN(C(=O)C(O)C1CCC1)C2 59259,c1(OC)cc(-c2ccc(F)cc2F)c(OC)cc1CN1CCCC(N(C)C)C1 59260,C1(NC(c2ccc(CN(CCC)C)o2)=O)(CF)CCN(C(C2CC(C)(F)C2)=O)C1 59261,C#Cc1ccc(OCC(N2CCC(NC(c3scc(C)c3Cl)=O)C(C)C2)=O)cc1 59262,C(=O)(C1=CCCOCC1)N1CC(CN(c2nc(C(=O)OC)c(Cl)cn2)C)OCC1 59263,CC1CCN(C(c2nonc2N)=O)CC1NC(c1cn(C)c(=O)cn1)=O 59264,N1(C(C(C)Sc2ncccn2)=O)CC2(CCN(C(=O)C=C(Cl)Cl)CC2)CC1C 59265,N1(CCSc2nc(NC(c3cnn(C(F)(F)F)c3)=O)sn2)CCS(=O)(=O)CC1 59266,C1(OC)(CNC(=O)Cc2ccc(C)s2)CCN(C(C2CCC(=O)NC2)=O)C1 59267,c1(C(=O)NCC2(OC)CN(c3cc(C(=O)OC)ncn3)C2)cc(F)ccc1F 59268,C1(C)(C(=O)NC(C#C)C)CCN(C(c2n[nH]cc2I)=O)C1 59269,C1(C(N2CC(C)(NC(C(C)N(C)C)=O)C2)=O)CCCCN1Cc1ccccc1 59270,c1(OC)ccc2cc1C(=O)OCCCOc1c(noc1)CNC2.C(N)(=O)OC 59271,C1(OC)C(NC(=O)NCc2cc(O)n(C)n2)CC1(C)C 59272,C1(Nc2ncc(C(=O)OC)cn2)COCCN(CC2(C#C)CCCC2)C1 59273,C1(NC(CCc2c(C)cccn2)=O)C(C)CCN(C(c2ccc(C#N)s2)=O)C1C 59274,C12(C(N3CC(CC)OCCC3)=O)CCC(CC1)N(C(c1ncncc1Cl)=O)C2 59275,c1(C(CC)NC(=O)NCC(C)(CO)c2ccccc2)cnc(C)cn1 59276,C1(C(C)OC(c2ccc(C(CCC)=O)cc2)=O)NC(=O)CNC1=O 59277,CC(C)CC(C(=O)NC1CC1(C)C(F)F)NC(c1cnn[nH]1)=O 59278,O=C1CCCC(CC(=O)NC2CC(NC(=O)CCc3cocn3)C(O)C2)N1 59279,C1(CC(=O)NCC2(CN(C(=O)C(F)CC3CCC3)C)CC2)CC(F)(F)C1 59280,N1(C2C(C)OCC2)CCN(C(c2ccc(CNc3cccnc3N)cc2)=O)CC1 59281,c1(CNC(C2(CNC(C3(C4CCCO4)CC3)=O)CCCC2)=O)ccncc1Br 59282,Cc1nc(CC(=O)NCC23CC2CN(C(C2C(F)(F)C24CCC4)=O)C3)cc(O)n1 59283,c1(C(=O)NC(C)C(C)(C)NC(=O)C=Cc2cc[nH]c2)ccc2nn[nH]c2c1 59284,c1(CCOC)cc2cnccc2[nH]1.c1(C(CC)C)nccc(N2CCNC2=O)n1 59285,Cc1cc(Cl)c(C(N2CCCC2CN(C(=O)C(C)CC(C)C)C)=O)cc1N 59286,c1(OCC(N2CC(NC(C(C)=C(C)C)=O)C3C2C3)=O)ccc2c(c1)CCC2=O 59287,N1(C(C(N2CCN(C)CC2)C)=O)CCN(C(c2ccc(N)c(N)n2)=O)C(C)C1 59288,c1(-c2cnc(NC(c3ccc(OC)cc3F)=O)nc2)cnc(C#N)c(F)c1 59289,C1(C(=O)NC2(c3cccs3)C(C)C2)CCC(c2ccccc2)O1 59290,C(CC(=O)N1CC2(CC(O)C2)C1)(C(F)(F)F)NC(CCC=C(C)C)=O 59291,C1(NC(C2N(C(c3n(CC)nc(C)c3)=O)CCCC2)=O)CCC(C2CC2)C1 59292,C12(C(=O)NCCC(=O)NC)CCC(C(=O)NCc3n(C=C)ccn3)(CC1)CC2 59293,N1(C(c2ccc(OC)nn2)=O)CC(C)C(C)(C(=O)NC2(C)CCCCCC2)C1 59294,C12(CNC(C=C(C)C)=O)CC(NC(=O)CSC(F)F)(C1)C(C)O2 59295,C(=O)(C=C1SCC(=O)N1C)N(C1CCCC(NC(COCC#C)=O)C1)C 59296,C1(C(=O)NCc2ncoc2CCNC(C2CS(=O)(=O)C2)=O)(COC)CCCCC1 59297,C12(C(N3CC(O)(CCC)C3)=O)CC1CCN2C(c1ccn(C2CC2)n1)=O 59298,CC1CCc2c(C(N3CC(C)(C)CC3CNC(=O)CC3CC34CC4)=O)csc2C1 59299,C1(CCC)CN(C(=O)CC(C)COC)CCN1C(c1cn(C)nn1)=O 59300,c1(OC)cc(C(N2CC(NC(=O)CCc3n[nH]c(=N)s3)CC(O)C2)=O)cc(C)c1 59301,C=CCC(CC(F)F)c1nc(CC)nn1-c1ccc(F)c(C)c1 59302,N1(C(c2n(CC)cc(Cl)c2)=O)CCCC(O)(CNC(C2CN(C)CCO2)=O)CC1 59303,c1(N(C(C2C3CCC2(c2ccc(Br)cc2)C3)=O)CC)cccc2c1OCCO2 59304,N1(CC)N=C(C(=O)NCC2C=CC(NC(c3ncc(Cl)cc3Cl)=O)C2)CCC1=O 59305,C(CCCCC(=O)N1CCN(C(C2CCOC2C)=O)C(C)C1)=CC 59306,N1(C(C(C)P(C)(C)=O)=O)CCOC2(C1)CN(C(C1CC13CC(O)C3)=O)C2 59307,C1(NC(C2Cc3nncn3C2)=O)CN(C(c2ccsc2Cl)=O)CC2(CC2)C1 59308,c1(C(c2n(CC)nnn2)NCC2CC(=C3CCC3)C2)ccc(F)c(C)c1Cl 59309,C1(NC(CCSCCCC)=O)CCN(C(=O)C=C2CC2)C1Cc1ccccc1 59310,C(=O)(C1CCCc2sc(=N)[nH]c21)NCC(CCCC)NC(=O)CC(C)C 59311,C(C(=O)NCC1(CNC(=O)CCNC(=O)C(C)(C)C)CC1(F)F)(C(C)C)SC 59312,Cc1cc(Cl)c(C(=O)NCCC2CCCN(C(=O)COCc3nc(C)no3)C2)s1 59313,c1(C(N2C3CCN(C(c4c(CC)nc[nH]4)=O)CC3C2)=O)cn2ccc(F)cc2n1 59314,c1(CN2C(C(N3CCN(C(C)=O)CC3)=O)CC2)cc(F)cc(Cl)c1 59315,c1(NC2CCN(C(c3cn(CCOC)nc3)=O)CC2C)nc[nH]c2ncnc1-2 59316,C(=O)(CCC(C)CC)N1CCC(CC=C)(C(N2CC(CS(C)=O)C2)=O)C1 59317,C1(CC(=O)N(C(C)CNC(c2c[nH]nc2C(C)(C)C)=O)C)CCCC(C2CC2)O1 59318,O(P(C)(=O)CNC(C1CC(F)CN1C(=O)CC1CCCOCC1)=O)CC 59319,CCCCCCCCOCC(=O)NCC1CCCN1C(c1cc(N)nc(Cl)c1)=O 59320,N12CCCN(CC1)C(=O)C(Sc1cccc(C)c1)CC2=O.C(=O)(C1CC1)OCC 59321,C12(CNC(c3c(C)nsc3)=O)CCCC1N(C(=O)C(C)C1CCOC1)CCC2 59322,C1(CN(C(C(C=CC)O)=O)C)CN(C(=O)CC(CC)c2ccccc2)CCO1 59323,N1(C(C(=O)NC2CC(C(=O)OC)C2)CCC2CC2C)CCCC2(CCCOC2)C1 59324,c1(C(N2CC(CCNC(C3CC(SC)C3)=O)(OC)C2)=O)cnc2cc[nH]c2c1 59325,C1(CNC(c2nc(COC)oc2)=O)CCN(C(C2CC3(CC3)C2)=O)CC1O 59326,C1(C(=O)Nc2cn(CC=C)nc2)CSCCN1C(=O)Cn1cccn1 59327,C(=O)(C(C(C)(C)C)NC(N)=O)NC1C(CNC(c2c(C)cno2)=O)C1 59328,CCC(C(=O)NCCCOC1CCN(C(C2CC3(C2)CC(O)C3)=O)CC1)C(C)O 59329,Cc1ccc(C(=O)NCC2CN(C(C3CCC3C(C)(C)C)=O)CCO2)c(F)c1Cl 59330,C(=O)(CCCCNC(C1C(NC(=O)CC2CC(C)(C)CO2)C1(C)C)=O)OCC 59331,c1(C(=O)NC(CCCNC(C(C)NC(C)=O)=O)C)ccn2ccnc2c1 59332,C1(CN(C(C2CC(C(F)F)(OC)C2)=O)C)CCN(C(C2CC(O)C2)=O)CC1 59333,C(N=c1cc(CC)nc[nH]1)C1CCCCC1C.CCC(C(=O)NC1CCCC1)OC 59334,C1(C(N2CC(NC(=O)C(C)(C)C)CC(OC)C2)=O)CS(=O)(=O)CC(=O)N1 59335,N1(C(C=CCOC)=O)CC(O)CC1C(N1CCCC1C1(C)CC1)=O 59336,c1(CNC(C2CC(c3ccon3)C2)=O)ccccc1CNC(C1CCCCO1)=O 59337,N1(C(c2cnc(CC)[nH]2)=O)CCC(CC)C1CNC(=O)C(CC)N(C)C 59338,C1(Br)(C(=O)NCCOCCN(C(C2(C)C(C)C2)=O)C)CC1(F)F 59339,N1(C(c2cn(C)nc2Cl)=O)CC2CC(C1)C(CO)C2NC(c1cccc[n+]1[O-])=O 59340,N1(C(C(CC#C)NC(c2sc(C)nc2C)=O)=O)CCn2ncc(C)c2C1 59341,c1(C(CC)CN(C2CC2)C(c2nc[nH]n2)C)ccccc1 59342,CCCC(C)CC(=O)NC1COCCN(C(c2c(C)cccc2N)=O)C1 59343,CC1(C(=O)NC2CCCC(C(=O)O)C2)CCCN(C(=O)C2=CCCCO2)C1 59344,N1(C(C(CC)F)=O)CCC(N(C)C(c2cc(-c3ccoc3)[nH]n2)=O)C2(CC2)C1 59345,CC(C)CC(O)C(=O)NC1CN(C(c2cccc(SC(F)(F)F)n2)=O)CC1C 59346,CC1CC(N=c2c(Br)c[nH]cc2[N+](=O)[O-])CCN1C(=O)C(C)(C)C 59347,C(CC(C)CCNC(c1cc(C(C)CC)no1)=O)NC(CCCOCC)=O 59348,c1(C(=O)NC2CN(C(c3c(O)ccc(F)c3F)=O)C2)cc(F)cc2nc[nH]c12 59349,C(=O)(C(CCOCC)NC(=O)C(C)C1CCCC1)N(CC=C)CCOC 59350,CC1(C)CCCC(CC(N2CCC(CO)(CO)C2)C(=O)NCc2ccc(F)cc2)O1 59351,c1(C(=O)NCC(C)(C2CC2)NC(CC(C)OC)=O)c(Cl)c2ccccc2n1C 59352,C1(N(C(C2C(SC)CCC2)=O)C)CCN(C(c2cnn(C3CC3)c2C)=O)CC1 59353,C(=O)(C(C)CC(F)F)NC1C(NC(CCc2cccc(C)c2)=O)CCCC1 59354,c1(C(=O)NCCCN(C(=O)Cc2cnsc2)C(C)C)cccc(=S)n1O 59355,C(=O)(C#CC(C)(C)C)NCC1(C(=O)NCC2(C)CCN(C)C2)CC(C)(C)C1 59356,C(=O)(C(C)(C)CC#N)N1C(C)CC(CNC(=O)COCCSc2cccnc2)C1 59357,N1(C(c2ccc(Br)c(F)c2)C(=O)NC)CCOC2(CCS(=N)(=O)CC2)C1 59358,C1(C2(O)CCOC2)(C(N2CCC(F)(CNC(c3ncc[nH]c3=O)=O)CC2)=O)CC1 59359,n1(CC(=O)NC2CC(CNC(=O)C(O)C3CC3)C2)cc(Br)cn1 59360,c1(OC)cc(OC)[nH]c(=NCc2ccc(CN3CCOC(C(N)=O)C3)cc2)n1 59361,Cc1nc(C2CCCO2)sc1C(=O)N(C)CC1CCN(C(=O)CC2(O)CCC2)C1 59362,C1(CC(NOC)=O)(NC(c2cccc(OCF)c2)=O)CCN(c2cnccn2)CC1 59363,n1(CC2(C)CC2)nc(SC(F)F)nc1CCC1CSC1 59364,C1(NC(=O)NCc2nc(C(C)C)on2)CCCC(O)CC1 59365,C1(NC(C=Cc2n(CC)ncc2)=O)C2CC3C(C2)C13C(=O)OCC 59366,C1(CNC(CC)=O)CCCN(C2CCc3ccc(Cl)cc32)C1 59367,CC1(CCCO)CCCN1C(c1ccoc1CNC(c1cnn(C2CC2)c1)=O)=O 59368,C1(C(=O)NCC2CN(C(C3CC=CCC3)=O)CCO2)CCOC2(CCCC2)C1 59369,C1(NC(c2sc(C(C)C)nc2C)c2n(CC)nnn2)CC(O)CC(C)(C)C1 59370,C(=O)(CC(C)(C)CN(C)C)N1CC(OC)C(NC(c2sccc2Br)=O)C1 59371,C1(c2ncc(C(=O)OC)s2)CCN(C(=O)N(C)C)CC1.C1CCS1 59372,C(=O)(C(C)C(C)COC)NCC#CC(=O)NC(CC#C)C 59373,N1(C(=O)CCc2cscn2)CC(NC(C23CC(c4ccccc4)C2C3)=O)C(O)C1 59374,c1(C(=O)NCC2CCC(CNC(CC(COC)O)=O)CC2)cc(C)cc(Cl)n1 59375,C(CCCCC(=O)N1CCCC(CC(=O)NC(C)(C)CCCO)CC1)=CC 59376,C1(NC(C(CC)(C)OC)=O)CC=C(C(=O)NCC(C)(C)CO)C1 59377,N1(C(CCC=CC)=O)CCN(CC2(NC(=O)C(C)CC=CCC)CC2)CC1 59378,C1(C(=O)NCC(C)N(C(c2sc(C)c(Br)n2)=O)C)CNC(=O)C(C)(C)C1 59379,c1(C(=O)NCC(CC)NC(=O)CCc2ccnn2C)cn(CCC(C)C)nn1 59380,N1(C(C(C)CC(C)(C)C)=O)CCC2CCN(C(c3cc[nH]c(=N)n3)=O)C2C1 59381,C1(C(N2C(C)CSCC2)=O)N(C(=O)CC2OCCO2)CC12CCCC2 59382,c1(-c2cn(C)nc2)cccc(C(=O)NCC2(O)CN(C(=O)CC3CC3)C2)c1 59383,C(C)(CNC(C1CCN1S(C)(=O)=O)=O)(C(C)C)NC(Cc1c(C)ocn1)=O 59384,c1(C(=O)NCC2CCN(C(=O)CSc3cccs3)C2)cc(F)cc2cnccc12 59385,c1(C(N2C3CC(NC(C(CC)(C)O)=O)CC2CC3)=O)cccc2oc(C)nc12 59386,CC1(C)CCN(C(C23CC2COC3(C)C)=O)CC1CNC(=O)C=CBr 59387,C1(C(C)C)(C(=O)NCCC2(O)CN(C(=O)Cn3cnnn3)C2)CCCO1 59388,c1(C(=O)OCC)ncc(NC2CN(C(=O)CC(C)(O)c3ccccc3)C2)nc1C 59389,C(=O)(C1=CCCN(C(=O)CC2CC2)C1)NCC(C)C1CCC1 59390,Cc1[nH]c(C#N)cc1C(=O)NC1CCCCN(C(=O)CC2CC3CCC2CC3)C1 59391,CCCCC(C)C(=O)NCCOC1CN(C(=O)C(c2ccn(C)c2)C)C1 59392,CCCCC(C(=O)NCCN1CC(CF)C1)NC(C1CCOC(C)(C)C1)=O 59393,C12(NC(c3cnc(C4CC4)o3)=O)CCCC1N(C(c1ncccn1)=O)CCC2 59394,C1(C(=O)NC(c2nccs2)CC)CCCCC1(C)NC(=O)C=CC=C(C)C 59395,N1(C(C=C)=O)CC2CC(NC(=O)C(=Cc3ccccc3)C)C2C1 59396,c1(CC(=O)NCCC(C)(C)NC(=O)CO)ccnc(-c2nn[nH]n2)c1 59397,c1(C(=O)NC2CC(C(=O)Nc3c(OC)nc(Br)cn3)C2)ccc(C#N)cc1Cl 59398,Cc1ccc2c(c1)N(C(=O)C(CNC(=O)Cc1ccc(O)cn1)C(C)C)CC2 59399,CC(C)CCCC(=O)N1CCC(C=CC(=O)NC(CO)CC(C)C)CC1 59400,C1(C(=O)NCc2nc(C(C)C)on2)CN(C(c2ccccn2)=O)CCN1 59401,c1(OC)cc(Cl)ncc1C(N1CCN(C(c2oncc2C)=O)CC1CC#N)=O 59402,Cc1ncn(C)c1C(=O)NC(C)CN(C)C(c1cnn(C(C)(C)C)c1)=O 59403,n1(CC#N)nccc1C(=O)NC(c1ccccc1)CNC(C12CSCC1C2)=O 59404,C1(NC(=O)CCc2ccccn2)CCN(C(c2coc(O)n2)=O)C12CCCC2 59405,c1(OC)cnc(C(N2CCC(NC(=O)Cc3ccc(F)cc3)C2)=O)c(F)c1 59406,c1(C(N2CCCCCC2CCO)=O)cnc2c(Br)cccn12 59407,N1(C(C=CC2N(C)CCC2)=O)CCC(NC(=O)Cc2ccoc2)C2(CCC2)C1 59408,C1(C(=O)NC2(C)C(C)OCC2)C2CC3C(C2NC(=O)CN2CCC(F)CC2)C13 59409,c1(OC)cc(NC(C2CCCC(NC(c3cnnc(O)c3)=O)CC2)=O)ccc1O 59410,C(=O)(C(CCC(C)C)NC(c1nonc1C)=O)NC1CN(C(C)=O)C1 59411,C(CNC(C(=O)NC)c1cncs1)(CO)(CO)N(C1CC1)CC 59412,Cc1cc(-c2cn(C3CC(C(=O)Nc4ncccc4F)C3)nn2)cc(F)c1 59413,Cc1nc(Cl)[nH]c(=NC2CN(C(c3ccc(N(C)C)cn3)=O)CC23CCC3)c1F 59414,C(=O)(C(=O)C(C)(C)C)NC1(CNC(c2n[nH]c(C)c2C)=O)CC1 59415,N1(C(c2c(C)noc2)=O)CCCN(CCCCNC(C2CC3CCC2O3)=O)CC1 59416,c1(C(=O)NC2CC(N(C(c3sc(C)c(Br)c3)=O)C)C2)cccc(F)c1N 59417,CN=c1[nH]c(=NC2C=CC(CO)C2)[nH]c(=NC2COc3ccc(Cl)cc32)[nH]1 59418,N1CCCC(CC(C(=O)C(F)=CC2CC2)=O)C1.C1(CCN(C)C)(NCCO)CC1 59419,C1(NC(C=CCCC)=O)CCC(C)(CNC(c2cnc(O)o2)=O)C1 59420,N1(C(C)CNC(C2CC(C)(O)C2)=O)CCN(C(=O)CC2(n3cncn3)CC2)CC1 59421,c1(SC(C)C(N2CC(F)(CNC(=O)NCC3CNC(=O)N3)C2)=O)ccccc1 59422,c1(N)[nH]c(=NCC2(C)CSC(C)=N2)nc2ncn(CC)c12.CCCCCCO 59423,c1(C(=O)NC(C)CCNC(=O)CCN2CCC2)ccc2c(c1)NC(=O)CO2 59424,Cc1cc(C(=O)NC(CNC(c2c(C3CCC3)cnn2C)=O)CO)cc(F)c1 59425,C1(C(=O)NCCOCCNC(Cc2c(C)ccnc2)=O)C2CCN(CC2)S1(=O)=O 59426,C1(S(N)(=O)=O)CCC1.N1(C(C2C(C)(N)CC2)=O)CCCC(c2c[nH]nn2)C1 59427,CCC(C(=O)NCCN(CC(C)O)C(=O)Cc1c(Cl)c(CC)nn1C)C(C)C 59428,C(C(F)(F)C(F)(F)F)OCCC(=O)NCC(CCOC)NC(C1CC(SC)C1)=O 59429,CC1(F)CC(C(=O)NCC(CNC(=O)CNC=O)CO)C1 59430,N1(C(c2nccc(CN(C)C)c2)=O)CC2(CCN(C(=O)C(CO)N(C)C)C2)C1 59431,C1(C(=O)NC2C(CCC)CN(C(=O)C(O)CCN(C)C)C2)CC(C)(C)CCO1 59432,c1(C(N2CCC(N(C(CN(C)CC)=O)CCO)C2)=O)ccc(C(C)(C)C)cc1C 59433,N1(C(CCCCC(C)(C)C)=O)CCC2C(CCCN2C(c2ccncc2O)=O)C1 59434,C(=O)(CCCOC1CC(NC(=O)CNC(C2CC2C)=O)C1)OC 59435,C(=O)(C(C)C(F)(F)C(F)F)N1C(CNC(c2cc(CC)cc(F)c2)=O)CCC1 59436,C1(C(N2C(CCNC(C(C)(C)CO)=O)CCC2)=O)Cc2ccc(Cl)cc2C(=O)O1 59437,c1(NCCC(c2nnnn2C2CCC2)C2(C(=O)OC)CC2)ccc(Br)c(Cl)c1 59438,CC1(C(=O)NCC2(O)CC(NC(=O)CSC3CC3)C2)CCC(O)CC1 59439,Cn1cnc2c1CCN(C(=O)C(F)C(F)(F)F)C21CCN(C(=O)CC2(C)CC2)C1 59440,c1(C(N2CC(CN(C)C(C3CC3C(C)(F)F)=O)C2)=O)cc(C(N)=O)c[nH]1 59441,C1(C(=O)NC2(CC)CCCCC3(C(C=C)C3)C(=O)NC2)CCOC2(CCCCC2)C1 59442,Cc1[nH]nc2cc(NC(=O)Cc3cccc4c3OCCC4)ccc12 59443,C12(CC(=O)NCC3CCCN(C(C(CC#C)C)=O)CC3)CCC(CC1)C2(C)C 59444,C1(C(=O)NCC2(C(F)F)CCN(C(Cc3c(C)ccs3)=O)C2)CCC2(CCC2)C1 59445,C1(N(C(c2ncc(CCC)s2)=O)CC2CC2)CCN(C(=O)CC(=O)NCC)CC1 59446,c1(CN)cn2ccc(C(=O)NCCc3ccc(C(F)F)cc3)cc2n1 59447,c1(C(N2CCC(CN(C(CCC=CC)=O)C)C2)=O)csc(Br)c1C 59448,c1(N2CCN(CCCNC(C(CC)(C)CC)=O)CC2)cccc(F)c1C#N 59449,C=CCCCC(C(=O)NCCCC(=C)Cl)NC(=O)C(C)OCC 59450,c1(COC)ccc(C(=O)NC2CCCC(C(N3CCSCC3)=O)C2)cc1 59451,C1(C)(C(=O)NC(CC)CC(=O)NCC2(CC)CCCO2)CC(=O)N(C)C1 59452,CN1CCC(C(=O)NCCC2(CNC(C3CC(N(C)C)C3)=O)CC2)C1=O 59453,C1(CC)CN(C(c2cc(Cl)ncc2F)C(=O)NC(C)(C)C)CC(=O)N1 59454,N1(C(CCC2CCC(C)O2)=O)CCC(C(=O)NCCN(C(C)C)C2CC2)C(O)C1 59455,CC1(C)CN(C(=O)CCCc2c[nH]c(C(=O)O)c2)C(C)(C)C1O 59456,C(=O)(C(CN(C)C)CC)NCC(C(N1CCC(CC=CC)C1)=O)O 59457,C=CC(C)(C)CC(=O)NC1CC(F)(F)CC1NC(=O)Cc1cccc(F)c1F 59458,C1(CC(N2CCC(c3cnco3)CC2)=O)CNCCS1(=O)=O 59459,C1(C(N2CC(N(C(c3cccc(NCC)c3)=O)C)C2)=O)CC12CC(C)(C)C2 59460,C(C(CNC(c1cncc(N)n1)=O)C(F)(F)F)NC(c1c(C)ccs1)=O 59461,c1(C(=O)NCCNC(c2ccc(C)cc2Cl)=O)cc(Br)cc2c1OCC2 59462,c1(CC(=O)NC(C2CCN(C(C3CCC3(C)C)=O)C2)C)coc2ccccc12 59463,Cc1nn(CCO)cc1C(=O)N(C)CC1CCCN1C(c1ccccn1)=O 59464,CCC(C)C(C)C(=O)N(C(C)CNC(=O)Cc1csc(C(=O)OC)c1)C 59465,CC1CN(C(C2CC2c2ccnn2C)=O)CC1NC(c1cnsn1)=O 59466,Cc1cc(CCC(=O)NCCC2CN(C(=O)CN3C(C)CCC3C)C2)cc(C)n1 59467,N1(C(C(CSC)(C)C)=O)CCC2(CNC(=O)CCCC3CCCC3)CCCC12 59468,CC1CN(C(=O)CCCCCN(C)C)CC(C)C1NC(=O)Cn1cccnc1=O 59469,O=C1NCC2(CCN(C(C3C=CCN(C(=O)C(O)CC(F)(F)F)C3)=O)C2)O1 59470,C1(C(=O)NC(COC(C)=O)CO)(COC)C=CCN1C(=O)C(n1ccnc1C)C 59471,CC1(C)CN(C(=O)CC(CNC(C2(C)CC3CC3C2)=O)C2CCC2)CCCO1 59472,C1(C(=O)NC2CC3CN(c4c(C)cncn4)CC32)CCc2ccc(F)cc2O1 59473,C1(CNC(C(C)O)=O)COCC1NC(=O)C(F)(F)Oc1ccccc1 59474,C(=O)(CCC(F)(F)F)N(C)CC1CCCN1C(C1CC(CC(F)F)C1)=O 59475,C12(C(N3CCCC(C)C3CNC(=O)Cn3cc[n+](C)c3)=O)CC=CCN1CCC2 59476,N1(CC(=O)NC(=O)NCC)CCCN(C(C2CCCC(OC)C2)=O)CC1 59477,Cn1nc([N+](=O)[O-])cc1C(=O)NC1(CCCNC(c2ccc(F)c(Cl)c2)=O)CC1 59478,c1(C(=O)NCCN(C(=O)CCc2ncc(C(C)(C)C)o2)CC)cc(SC)oc1C 59479,C(C)(CCC(=O)Nc1ccc(C(=O)NOCC=CCl)o1)OCC 59480,c1(OC)nccc(N(CC(C)NC(=O)Cc2ccns2)C)n1 59481,c1(C(=O)NC2CCCCCN(C(C(CC)(C)CO)=O)C2)cc(F)c(Cl)c(N)c1Cl 59482,N1(C(C23N(CC(OC)C2)CCC3)=O)CC2(CCN(C(c3cocc3C)=O)CC2)C1 59483,C1(NC(C(C(C)C)C#N)=O)CC2CCC1C(NC(C1(C(=O)N(C)C)CC1)=O)C2 59484,C12(C(N(CCCN(C(C3(C#C)CCCC3)=O)C)C)=O)CCC(C)(C(=O)O1)C2(C)C 59485,C1(C(N2CC3C(CC(=O)NCC(CC=C)(F)F)C3C2)=O)CC2(CCC2O)C1 59486,c1(C(N2CCCC(N(C(C(C)=C(CC)C)=O)C)C2)=O)ccc2cnnc(O)c2c1 59487,C=CC(C)(C)C(=O)NCC1CCC(CN(C)C(C2CC2C(=O)OC)=O)CC1 59488,N1(C(CCC=C(C)C)=O)Cc2nccn2CC(NC(C2CCSC2)=O)C1 59489,c1(CC)ccc(C(N2CCCC(NC(=O)CC3CCC(C)(C)O3)CC2)=O)cc1F 59490,C(=O)(CCCCC(F)(F)F)NCC(C(C)C)NC(CC(CC)C)=O 59491,c1(C(N2CCC(NC(CC(CC)O)=O)CC2C)=O)c(C)nn2cccnc12 59492,N1(C(c2ccc(-c3ccco3)s2)=O)CCC2CCC(C1)N2c1nnc(C(F)F)s1 59493,c1(COC)nc(C)c(C(=O)NC(C)(CNC(=O)CNC(=O)C(C)(C)C)C(C)C)s1 59494,C1(C)(c2cn(CC3(C)CCC3)nn2)COCCN1C(=O)CC1CC(F)(F)CO1 59495,N1(C(c2ccn(-c3cccnc3)n2)=O)CCC2(CCCN2C(C2CCO2)=O)CC1 59496,N1(C(c2cc(OC)cc(F)c2)C(=O)NCC(F)F)CC2CCCCCC2(C#N)C1 59497,c1(C(N(C(CNC(c2cnsn2)=O)C2CC2)C)=O)ccc(=O)n2c1COCC2 59498,C(=O)(CS(C)(=O)=O)NCCC(C)NC(=O)COc1ccsc1Cl 59499,Cc1c(C(=O)NC2CCC(CNC(c3n[nH]cc3C(C)C)=O)C2)sc2nccn12 59500,Cc1cn2cc(C(=O)NC3CCN(C(=O)C(C)S(C)(=O)=O)CC3O)sc2n1 59501,N1(C(C2CCN(C)C2)=O)Cc2ccc(C(N3CC4CC3CO4)=O)cc2C1 59502,N1(C(c2c(CCC)nns2)=O)CCCC(C)C1CCNC(c1ccnc(S)c1)=O 59503,N1(C(CCCC)=O)CC2COCC2(C(N2CCCC(C(C)O)C2)=O)C1 59504,C(CCN=C(NCC1(C)CCS(=O)(=O)N1C)NCC12CCC(CC1)C(C)O2)OC 59505,N1(C(C(CC2CCC2)NC(COC(CC)(C)C)=O)=O)CCCN(C2CC2)CC1 59506,c1(CC)cc(C(=O)N(C2CCN(C(C3(CF)CCOCC3)=O)C2)CCO)ncn1 59507,c1(C(N2CCCC(O)(CNC(C3C=CC=CC=C3)=O)C2)=O)ccc2nncn2c1 59508,C1(N(C)C(c2cn(C)nc2O)=O)CC2CCC(C1)N2C(=O)C(N)=O 59509,N1(CC(c2cccc(NC(=O)NC(C)=O)c2)=O)CC2CCC(CC2)C1 59510,C1(CNC(C2N(C(C(c3cnn(C)c3)C)=O)CC2)=O)CC2(CC2)CO1 59511,c1(C(C)OC(Cc2c(C)cco2)=O)cccc(Cl)n1 59512,C1(ONC(=O)OCC)(CNC2CCOCO2)CCCSC1 59513,c1(C(N(C)CCNC(=O)CNc2cc(F)ccc2F)=O)occ2c1CCCC2 59514,N1(C(C2CC(=O)NCC2)=O)CC2(NC(C3CCC3)=O)CCCC2(F)C1 59515,N1(C(COCCSC)=O)CCCN(C(c2cccc(F)c2N)=O)C(C)C1 59516,Cc1nc2ncnn2cc1C(=O)N(CC(C)(C)NC(=O)CO)C 59517,c1(OC)cc(OC)cc(N2CC(Nc3ccc(-c4ccnn4C)cc3C)CC2=O)c1 59518,c1(C(CC(=O)NCC2CCCN2C(C2(C3CC3)CC2)=O)O)ccc(Cl)cc1 59519,c1(C(N2CCCC(CNC(c3cccc(C)c3I)=O)C2)=O)cnc2snnc2c1 59520,c1(C(N2CC(F)CC(NC(C3CCCC(C)(C)O3)=O)C2)=O)ccc2nnnn2c1 59521,N1(C(C(C)(C)OC)=O)CCC(C)(CCNC(C2CC2C2CC2)=O)C1 59522,C(=O)(CCCCCc1ccccc1)NC1C(CNC(c2ccc(SC)s2)=O)C1 59523,CC1CC(=O)NC1C(N1CC(OCCNC(c2conc2C2CC2)=O)C1)=O 59524,c1(SCC(=O)NC2(CS(N)(=O)=O)CCC2)ccc(Br)cc1 59525,c1(N2CCC3(C(C(=O)Nc4cc(N(C)C)cc(F)c4)C3)C2)ncnc2occc12 59526,Cc1nc(C)n(CC(=O)NC(c2ccc(F)cc2)CNC(=O)C=CC(F)(F)F)n1 59527,c1(N(C(C2C(C(=O)OC)C2)=O)CC#N)ccccc1NC(c1cccc(Cl)c1)=O 59528,c1(C(N2CCCC2CN2CCC(C(=O)NC)C2)C(=O)NC)cc2ccccn2n1 59529,c1(CC)cc(C(=O)NCCCCC(C)NC(=O)CCCc2ccccn2)ccn1 59530,N1(C(C2CC(N(C)C)C2)=O)CCN(C(=O)C=Cc2ccn(C)c2)CC(C)(F)C1 59531,N1(C(Cn2nnc(C3(C)C(C)OCC3)n2)=O)CCC(CO)C(F)C1 59532,CCCCC(C(=O)N1CC(C)C1NC(=O)CCCOCCOC)N(C)C 59533,c1(C(N2CCC(NC(N)=O)CC2)C(=O)NCC(=C)C)cc(-c2ccco2)oc1C 59534,CC1=NOC(C)(CNc2cc(N3CCC(C(C)C)(CO)C3)ncn2)C1 59535,C(=O)(CCCN=[N+]=[N-])NC1CCC(C(=O)OC(C)(C)C)C1.C12CCC1CC(=O)N2 59536,Cc1ccc(C)c(C(N2CC(O)CCC2C(=O)NCCCSC(F)F)=O)n1 59537,c1(C(=O)NC2CC(CCNC(C(C(CC)C)O)=O)C2)ccc(OC)c([N+](=O)[O-])c1 59538,C(=O)(CCCCC1CC1)N(C1CCN(C(=O)CC2C(=O)NN=C2C)CC1)CC 59539,C1(C(=O)NCC(C)N(C)C(C2CCCN2c2cnccn2)=O)CCCC12CC2 59540,c1(C(N2CCC(NC(C=CC(C)(C)SC)=O)(CF)C2)=O)ccc(F)c(F)c1N 59541,C(=O)(C#CC1CCCO1)N(C(C)CN(C)C(c1coc(CO)c1)=O)C 59542,c1(OCC)ccc(CC(=O)NC2CC(F)(CNC(=O)CC3CS(=O)(=O)C3)C2)cc1 59543,CC1(C)CCCC(C(=O)NC2CCN(CCCNC(=O)Cc3ccon3)C2)C1 59544,c1(CC(=O)NC2C(NC(c3c(CC)con3)=O)CC2)ccc(C)cc1F 59545,C(=O)(C1OCCn2ccnc21)NCC(CNC(c1c(NC)ccc(F)c1)=O)CO 59546,C=C(Cl)CN=C(NCC1(C)CCCCCCC1)NC(C1CC1)C1CC1 59547,CC1ON=C(C(=O)N2CCN(C(=O)C(C)(C)CN(C)C)CC2C2CC2)C1C 59548,CCCCCC(C)CC(=O)NC(C)(C)C(C)NC(=O)CC(C)(C)CN(C)C 59549,CC1CN(C)CC1C(N1CC(C)(NC(C2CCN(C(=O)N(C)C)CC2)=O)C1)=O 59550,C1(NC(c2n(CCSC)nnn2)c2csc(SC)c2)CCOCC1(C)C 59551,N1(CC)N=C(C(=O)NCC2CC(O)(CNC(=O)Cn3nccc3C)C2)CCC1=O 59552,Cc1ccc(C(=O)N(CC(C)C(=O)N2CCC(CC(F)F)C2)C)n1C 59553,N1(C(c2cnc(CC)[nH]2)=O)CC(C2CCN(C(=O)CCCNC(C)=O)C2)C1 59554,c1(OC)c(F)ccc(NC(=O)C(C)N(S(C)(=O)=O)C)c1F 59555,Cc1ccc(O)cc1C(=O)NCc1nocc1C(=O)Nc1ccc(O)c(Cl)c1 59556,Cc1nc2cccc(C(=O)Nc3[nH]nnc3C3CCN(C(=O)OC(C)(C)C)C3)c2s1 59557,C1(NC(c2cccnc2)=O)CC=C(C(=O)Nn2cncn2)C1 59558,c1(CNC(COCC(=C)C)=O)occc1C(=O)NC1CC=CCC1 59559,C(=O)(C1OCCc2ccc(C)cc21)NCCCOCCN(C(C1C(C=C)C1)=O)C 59560,C1(CNC(c2c(NC)cccc2)=O)CN(C(c2ccc([N+](=O)[O-])o2)=O)CC1(C)C 59561,CCCC(C(=O)NCc1cccc(CNC(C2(C)C=CCC2)=O)c1)OCC 59562,c1(C(CC)C)ccc(C(=O)NC(C)(CNC(=O)C(O)C(C)C)C2CC2)cc1 59563,Cc1cc(Cl)c(C(N2CCCC2CCCNC(=O)C(c2cccc(Cl)c2)O)=O)s1 59564,C(C)(C(CC(=O)NCC12CC(CN1C)C2)NC(=O)C(C)SC(C)C)OC 59565,C1(C)(C(=O)NC2C(COC)CCC2)C=CCN1C(=O)CC1CCOCC1OC 59566,N1(C(CCCC(=O)N(C)C)=O)CCCC2(CCN(C(=O)Cc3ccns3)C2)C1 59567,c1(OC)ncc(NC(c2ccc(OC)c(C3CC3)c2)=O)c(C)n1 59568,c1(N2C(=O)CC(C(=O)NC3CCC(O)(CO)CC3)C2)cc2ccccc2o1 59569,C1(CNC(c2c(CC)con2)=O)(COC)CCN(C(C2CC(C)(C)O2)=O)CC1 59570,CCCC(F)(F)C(=O)NCC(COC)NC(=O)C(O)CN(C)C 59571,c1(CC)cnccc1C(=O)NC1CC(NC(=O)COc2ccc(C)cc2)C1 59572,C(CCC(=O)NCC(CO)NC(c1cnc(C2OCCO2)s1)=O)NC(N)=O 59573,CC1CC(C(=O)NCC2(C)CCOCC2)CN(C(=O)COCCCN(C)C)C1 59574,C(=O)(C1=CC2C=CC(C1)C2)NC(CC(C)NC(c1c(OC)c(C)sc1)=O)C 59575,N1(C(C(C)N2CCC2)=O)CCCC2(CNC(c3cccnc3Cl)=O)CCCC12 59576,CCCC(C)CC(=O)N(C(C)C(=O)NOCC1CCC1)C 59577,c1(N2C(C)CCC(NC(C(C#C)(C)C)=O)C2)cc(C(C)C)nc2ncnn12 59578,C=CC1CN(C(C2CN(C(c3cnn(C)c3Cl)=O)CC2OC)=O)CCO1 59579,C(C)(C(C)COCC)(c1n(CC=C)nnn1)Nc1ccccc1C 59580,c1(C(N2CCOCC2CC2CCCC2)C(=O)NCCC)ccc(N(C)C)nc1 59581,c1(C(=O)NC23CC(NC(c4ccc(Cl)cc4Cl)=O)(C2)C3)ccc(Cl)c2[nH]ccc12 59582,C=CC(C)CC(=O)NCC12CC1CN(C(c1ccn(CCN(C)C)n1)=O)C2 59583,N1(CC(=O)NCC2CCN(C(c3cn(CCC)nn3)=O)C2)CCN(C)CC1 59584,c1(C(N(CCC#C)C)=O)ccc(CNC(C2(C)CNC(=O)C2)=O)cn1 59585,C=CCC(C(=O)NCC1(O)CCN(C(=O)CN2CCOC2=O)C1)c1ccccc1 59586,c1(C(=O)NCCCCCNC(C2N(CC)CC2)=O)cc(C)c(C(=O)OC)o1 59587,c1(C(=O)NC2CCCC(NC(C(C)OCC=C)=O)C2)nc(C)ccc1O 59588,c1(C(=O)NC2CCCN(C(C3(CC(=O)OC)CC3)=O)C2)cccc2c1COC2 59589,Nc1ccc(C(=O)NC2CCCC2NC(c2ncoc2C(F)(F)F)=O)cc1Cl 59590,N1(C(c2cccc(CCC)c2)=O)CC2(CC(NC(C3(C)CCC(=O)N3)=O)CO2)C1 59591,c1(C(=O)NC2CC(CC)(CC)N(C(=O)C3=NOC(C)C3)C2)c(C)ccc(C)c1O 59592,N1(C(C2N(C(c3ccc(C(C)=O)[nH]3)=O)CC=CC2)=O)CCOC(C)(C)CC1 59593,c1(NC(CNC(C(F)=CCC)=O)C(C)C(C)C)ncnc2cc(F)c(F)cc12 59594,Cc1cnc(C(C)NC(=O)C(COC(C)C)NC(=O)CC(=O)NC2CC2)o1 59595,C1(NC(CCN(C)C(=O)OC(C)(C)C)=O)C2CC3CN(C(=O)C4CC4)C1C3C2 59596,N1(C(C=C(CCC)CCC)=O)CCC2(C1)CN(C(=O)C(c1ccnn1C)O)C2 59597,N1(C(CCC2(C)CN(C(C3(CC(C)=O)CC3)=O)C2)=O)CC2CC(O)CC1C2 59598,C1(C(N2CC(O)CC(OC)C2)=O)CN(C(c2cc(C)cc(F)c2)=O)CCC1(C)C 59599,O=C1NCc2c1ccnc2C(N1CC(CNC(C2CC(O)C2)=O)C(O)C1)=O 59600,C1(C(N2C(C)(C(=O)NCCC3CCN(C)C3)C=CC2)=O)CCCC(C#N)C1 59601,C(C(C)(C)CC(C)O)NC(C(C1(C)CC1)NC(Cc1c(C)ccnc1)=O)=O 59602,c1(CC(=O)N(C(C2CCCC2C)C)C(=O)OC2CCC2)cccc(Br)c1 59603,Cc1cccc(NC(C2CCN(C(=O)Cc3cc(F)ccc3Br)C2)=O)c1[N+](=O)[O-] 59604,C1(C)(CNC(=O)OC(C)(C)C)CCC(NC(=O)C(=O)NCCN2CCCC2=O)C1 59605,N1(C(c2cncc(C#C)c2)=O)CCC(NC(=O)C#CC2CC2)C12CCC2 59606,N1(C(Cc2cc(OC)no2)=O)CC2CCN(C(C3CS(=O)(=O)C3)=O)C2C1 59607,c1(C(=O)NC2C(NC(CCC=C)=O)CCC2)nc2ncccn2n1 59608,C1(C(=O)NCC(=O)OCC#C)(NC(C2CC2(Cl)Cl)=O)CSC1 59609,c1(N(C)C)cccc(C(N2CCC(CNC(C3CC(C#N)C3)=O)C2)=O)n1 59610,Cc1sc2ncc(C(=O)NC3CC3CNC(c3ncoc3C(C)(C)C)=O)n2c1C 59611,Cc1cc(C(=O)NC2CC(NC(=O)CC3CCC4(CCC4)O3)C2)cc2c[nH]nc12 59612,c1(COCC(=O)NCC(CNC(CCNS(CC)(=O)=O)=O)O)ncc(C)o1 59613,n1(C(C)C)cc(C(=O)NCC2CCN(C(C3(F)CCOC3)=O)C2)c(Br)n1 59614,C=CCC(C)(C)CC(=O)NCc1cncc(C(=O)NC2CN(C(N)=O)C2)c1 59615,C1(CC(=O)NC(CC(=O)NCCC(C)(C)O)C2CC2)CC2(CC2)CO1 59616,Cc1ccc(F)c(O)c1C(N1CCC2C(NC(c3c(Cl)cnn3C)=O)C2CC1)=O 59617,C1(C(N2CCOC(CC)C2)=O)(CNC(C(COCC)C)=O)CC12CCC2 59618,c1(C(N2CCN(CC(=O)NCC3N(CC)CCC3)CC2)=O)cc(F)cnc1O 59619,c1(C(C(=O)NCC(C)OC)NC(=O)OC(C)(C)C)cn(C)nn1 59620,CC(C)C(C(=O)NC(C)Cc1ccncc1)NC(=O)Cc1cccnc1 59621,c1(SCC(=O)NCC(CNC(CC2CC(SC)C2)=O)C)ccc(C)c(C)c1 59622,c1(OC)cccc2sc(C(=O)NCC(O)CNC(=O)C(C)n3cccn3)cc12 59623,c1(CC(=O)NC2C(NC(C(c3ccc(Cl)s3)C)=O)COC2)cnn(C)c1Cl 59624,C1(C(N(CCNC(CC(=C)I)=O)C)=O)CCC(C(F)(F)F)CC1 59625,C(=O)(N=c1nc2cccc(F)n2[nH]1)c1cccc(CCC2=CC(O)C(OC)C2)c1 59626,C1(COC)C=CCCN1C(=O)CC(O)CNC(c1ccncc1N)=O 59627,c1(N(CC(c2cccc(F)c2)N2CCCC2)CC)cc([N+](=O)[O-])c(C#N)s1 59628,C1(NC(COC(C)C)=O)(CF)CCN(C(=O)CCC2CCCCN2C)C1 59629,c1(C(=O)NC2C(CNC(=O)CC3CCOC3)C2)c[nH]c2cc(Cl)ccc12 59630,CC1CC(CNC(C2CC3CC3C2)=O)CCN1C(=O)CCOC1CCOCC1 59631,C1(C)(NC(c2c(C)cc(CNC(CC(=C=C)C)=O)o2)=O)CCCC1(F)F 59632,c1(C(=O)NC2C(OC(C)(C)C)CCC2)cnc2scc(Br)n12 59633,c1(OC)cc(C(=O)Nc2cc(C)cc(C)c2Br)c(N)cc1Cl 59634,c1(C(N(CC(C)CNC(=O)CN2CCCCC2=O)C)=O)cccc(F)c1N 59635,C(CC(=O)N1CC(C)(C)C12CCC2)(CC(C)C)NC(CC(COC)(C)O)=O 59636,C1(C(=O)NCCCN(C)C(c2ccc(Cl)c(O)c2)=O)COc2ccccc2C1 59637,N1(C(C(CO)NC(C2C3CC(=O)CC32)=O)=O)CC2(CCNC2=O)C1 59638,c1(C(N(CCNC(C2C=CCS2)=O)CC)=O)cnn(C(C)C)c1O 59639,C=CC(C)CC(=O)NC(C1CN(C(=O)CCc2cncnc2)C1)C 59640,C1(C(=O)NCC(C2(CCO)CN(C(=O)OC(C)(C)C)C2)=O)CCc2ccnn2C1 59641,c1(C(N(CCOCCN(C(=O)Cc2csnn2)C)C)=O)cccc2c1CCOC2 59642,N1(C(c2cc(SC)nn2C)=O)CCC(N)c2ccc(F)cc21 59643,c1(C(N2CC3C(N(C(=O)CC4(C)CC4(Cl)Cl)C)C3C2)=O)cncn(C)c1=O 59644,c1(C(=O)NCCCN(C(CSCC=C)=O)C(C)C)ccc(Cl)c(OC)c1 59645,Cc1ccc(C(=O)NC2CC2C(=O)N(CCO)C2CC2)cc1[N+](=O)[O-] 59646,c1(C(N2C(C(C)(C)NC(C(C3CC3)OCC)=O)CCC2)=O)nccc2n[nH]cc12 59647,C(CC(=O)NCC1CCCN1C(C)=O)(C(F)F)NC(c1cc(CC)ncc1)=O 59648,N1(C(C2(C)CCCN2C(c2ccn(C3CC3)n2)=O)=O)CCCCCCCC1 59649,Cc1nc2ccc(C(N3CC(Cc4cccc(Cl)c4)C3)=O)cc2o1 59650,Cc1n[nH]c(C)c1CC(C)C(=O)NC(C)CC(C)NC(=O)C(C)O 59651,C(=O)(C(CNC(=O)CC(C)(F)F)CC1CC1)NCc1ccc(CC)o1 59652,C1(CCNC(c2ccc(CC3CC3)s2)=O)CCCCN1C(C1(O)CCC1)=O 59653,c1(CC(N2CC(OCCNC(COCc3cc(C)no3)=O)C2)=O)c[nH]ccc1=O 59654,CCCC(F)C(=O)NC1(CCCNC(=O)CCCNC(=O)OC)CC1 59655,CC(C)(C)C(=O)C(=O)N1CCN(C(c2sccc2C(F)F)=O)CC1CF 59656,CON1CCC(CC(=O)NC2CC(F)(CNC(=O)CN(C3CCSC3)C)C2)CC1 59657,C1(NC(c2nccc(OC)c2)=O)CCCC12CN(c1ccncn1)C2 59658,C1(COC)(NC(C2CC2c2ccsc2)=O)CCN(C(=O)Cc2ccccc2F)C1 59659,C1(c2ccn(-c3c(Cl)cccc3)n2)CCCN1N1CCC(CCC#N)CC1 59660,C1(CCCC)CCC(N=c2[nH]c(N3CCOC(C)C3)nc3c(F)cccc23)CC1 59661,CC(C)(C)C#CC(=O)N1CCN(C(=O)CC2CCS(=O)(=O)CC2)C(CF)C1 59662,C1(OC)CN(C(c2nc(CC)oc2)=O)CC1NC(c1ccccc1NC)=O 59663,C(CCC(=O)NC(CSCC)C(=O)NC1CCN(C(N)=O)C1)OCC=C 59664,Nc1ccc(C=CC(=O)NCC2CCCN(C(C3CCCOCC3)=O)C2)cc1N 59665,CCC(C)C(O)C(=O)NC1CC(CNC(c2cc(-c3ccccc3)ccn2)=O)C1 59666,C(CC(C(C)(C)C)NC(=O)Cn1cnnc1)N(C(c1c(C)nccc1)=O)C 59667,CCC(CC)(CCNC(=O)C(C)Cn1ccnc1)NC(c1cc(F)n(C)n1)=O 59668,Cc1c(Cl)c(C(N2CCC(C)(NC(C3CC34CCCC4)=O)C2)=O)nn1C 59669,N1(C(C(=O)NC(C(=O)N(CC)CC)C)=O)CCCC2(C=CCO2)C1 59670,C12(CNC(C3C(C=C)C3)=O)CC1CN(C(=O)CSc1cnn(C)c1)C2 59671,C1(C(N2CC(O)(CNC(=O)Cn3cc(C(C)=O)nn3)C2)=O)(COC)CC1(F)F 59672,CC(C)(C)CC(N)CCN1CCC(C)(C)C1=O 59673,N1(C(COCCCCC)=O)CCCC1CN(C(C1CCC1CF)=O)C1CC1 59674,N1(C(Cc2n(C)nnc2)=O)CC2(C(=O)NC3CC(CO)C34CCC4)CCC1CC2 59675,c1(CNC(N(C2CCCOC2)CCC)=O)cnc(COC)s1 59676,c1(OC)nccc(C(=O)NCC(C)(C)CN(C(=O)CCc2cncc(C)c2)C)n1 59677,CC1(F)CCN(C(=O)C(C2CC2)NC(=O)CC2CC(F)(F)C2)C1 59678,CC(C)CC(C(=O)N1CC2CC(C(N3CCC(F)CC3)=O)CC2C1)C(N)=O 59679,c1(SC)c(C(=O)N(c2cccn(C)c2=O)C)cccc1Br 59680,N1(C(C(CC(C)C)O)=O)CCC2(CC(NC(c3cc(C4CC4)ccc3F)=O)C2)C1 59681,C1(C(=O)NCCOC2CCN(C(C3(C)CC3(F)Cl)=O)C2)CN2CCCN1CC2 59682,c1(C(N2CC(N(C(C=COCC)=O)C)C3(C2)CC3)=O)ccc2c(c1)C=CS2(=O)=O 59683,C1(CNC(c2n(C(CC)C)ncc2)=O)CCCN(C(=O)C(C)(C)CC)C1 59684,C1(C)(CNC(c2cccc(CC)n2)=O)CCCN(C(C2CC23CCCC3)=O)C1 59685,C(=O)(C(F)C(F)(F)C(F)(F)F)N1CCC(NC(C2CC(C)(C)C(=O)NC2)=O)CC1 59686,C(C(N=c1[nH]c(Cl)ncc1Br)C1CC1)NC(C1N(C(CCC)=O)CCC1)=O 59687,n1(C(C)C)cnc2c(NCCC(C)S(C)=O)nc(N(C)CC3CC(F)(F)C3)nc12 59688,C(C)(C)(C(=O)NCC(C1CC1)NC(C1(F)CCOC1)=O)NC(=O)NCCC 59689,C1(Cl)(C(=O)NCC2(NC(c3nc(CC(C)C)sc3)=O)CCOC2)CC12CCC2 59690,c1(NCC)cc(NC(CC)C(c2nnnn2C)NC(=O)OC(C)(C)C)ncn1 59691,c1(C(=O)NCCC2(CNC(C(C)=C3CC3)=O)CC2)ccc2nc(S)oc2c1 59692,C(CNC(=O)CC1(N(C)C)CC1)(C(C)(C)C)NC(C(C=C)C)=O 59693,c1(C(C(=O)NCC)N(CC(C)OC(C)(C)C)CC)cc(C)c(C)c([N+](=O)[O-])c1C 59694,[N-]=[N+]=Nc1ccc(C(=O)NC2CCC3CN(C(=O)Cc4cccnc4)CC23)cc1 59695,C1(C(=O)NC(C)CCCNC(=O)Cc2ccco2)CC2CS(=O)(=O)CC2C1 59696,C1(CNC(C(C=C)OC)=O)CN(C(c2cc(F)n(C)n2)=O)CCN1C 59697,C1(CC(=O)NC(CC#C)C)CN(C(C2(O)CC(CF)C2)=O)CCO1 59698,c1(CC(=O)O)cn(CC2CCN2C2CN(C(c3ccc(-c4cccs4)[nH]3)=O)C2)nn1 59699,N1(CCCCNC(CC(C)OC)=O)CCCN(C(=O)C=CC2(C)COC2)CC1 59700,C12(C(=O)NC(CNC(CCC=C(C)C)=O)CO)CCC(C)(C1)OC2 59701,n1(CC(N2CC(CC(C)NC(C)=O)C2)=O)nc(C(F)(F)F)c(Cl)c1C 59702,N1(C(c2c(CC)noc2)C(=O)Nc2ccccc2C)CCC(O)CC1(C)C 59703,O=C(CC(C(F)F)c1ccc(F)cc1)Oc1ccc(N2CCN(C3CC3)CC2)cc1 59704,C1(C(=O)NCc2cc[nH]c2C(=O)NC2COC(=O)C2)(OC)CCOC1 59705,c1(CC(=O)NC)ccc(C(=O)NCC2C=CCN2C(C2CC2(C)C)=O)cc1 59706,N1(C(c2c(CC)cns2)=O)CCN(C(=O)CCc2cncc(F)c2)CC1CCO 59707,C1(C)(C(N2CCC(F)(CNC(c3c(CC)nn[nH]3)=O)C2)=O)CC(C(C)(C)C)=NO1 59708,C1(NC(C2(C)C=CCN2)=O)CCCC12CCCC2 59709,N1(C(C(CSCC)NC(c2ccsc2)=O)=O)CCC2(CCC(OC)C2)C1 59710,C1(c2cnc(C)[nH]2)NC(=S)N(C2CC2)C2=C1C(=O)NCC(C)C2 59711,C1(C)(C(N(CCC)CCNC(=O)COCC2CCCOC2)=O)CCC(C)=C(C)C1 59712,C1(NC(c2cc(C)sc2C)=O)CC(NC(=O)CCCNC(N)=O)C12CCOCC2 59713,c1(C(=O)NCC2CC(NC(C3CC=CCC3)=O)C2)ccnc(-c2ccccc2)c1 59714,CCC(CC(=O)NC(CO)C(N1CC(C)(C)CCC1C)=O)C(F)F 59715,N1(C(CCOCCC)=O)C2CCC(C2)C1CNC(=O)Cc1cc[nH]n1 59716,C#CCC(C)(C)C(=O)N1CCCC(CC(N2CCOC3(CC3)C2)=O)CC1 59717,N1(C(Cc2c(OC)ccc(C)c2)=O)CC(C2CN(C(C3CC(C)CCO3)=O)C2)C1 59718,CC1(C)CCC(N=c2[nH]c(=NCC(C3CC3)C3CC3)[nH]c3c(F)cccc23)C1 59719,C1(C(N(C(CNC(C(C)O)=O)C2CC2)C)=O)CC(S(C)(=O)=O)C1 59720,Cc1ccc(OCC(=O)NC2CC3CCC2(NC(c2cncnc2)=O)C3)cc1C 59721,C=CC1CN(C(c2cccc(COC)n2)=O)CC1NC(C12CC(F)(C1)C2)=O 59722,N1(C(C(CCC)CNC(C2CC(=O)NC2(C)C)=O)=O)CCC(O)C12CCC2 59723,C1(C(C)(C)C)CCc2c(sc(NC(c3cc(CN)c4occc4c3)=O)c2C#N)C1 59724,C(=O)(CC(C)C(C)(C)CC)N1CC(CCC)N(C(=O)C(C2CC(F)(F)C2)O)CC1 59725,c1(SCC)nccnc1C(=O)NC1CCCC(NC(C2(OC)CCSCC2)=O)C1 59726,c1(-c2cc(C)cc(C)c2)cccc2c1CCN(C(c1ccc(CCO)cc1)=O)C2 59727,C(=O)(CS(C)(=O)=O)N(CC(=O)NCC(COC)(C)O)CC(C)C 59728,c1(C(N(C2CCN(C(CC(c3c(C)noc3C)C)=O)C2)C)=O)cn2c(n1)CCC2 59729,N1(C(CC)=O)CC2CC(C)N(C(c3cc(N)cc(Br)c3O)=O)C2C1 59730,CC(C)(CC(=O)N1CCN(C(c2ccc(S(C)(=O)=O)o2)=O)CC1CO)C(F)F 59731,c1(C(=O)NC2CN(C(c3c(C)n(C)cc3)=O)C(C)C2)c(F)cccc1Br 59732,C#CCCN=C(NCC(c1ccccc1)CO)NCC1(C)CCCCO1 59733,c1(C(=O)NCCC2CCN(C(c3c(CC)csc3)=O)C2)ncc(N(C)C)cn1 59734,c1(C(=O)NC2C(CNC(C(C)(C)N3CCCCC3)=O)CCC2)cnc2n1CCCC2 59735,CC(C)C(O)C(=O)NC1CCC(NC(C2(Cc3ccccc3)CCC2)=O)C1 59736,c1(C(N(C2CCN(C(C3(SC)CC3)=O)C2)CC)=O)ccc(Cl)c(C(=O)NC)c1 59737,C(CC(F)F)(C(=O)NCC1(C)CC(C)(C)C1)NC(c1cn(C)nn1)=O 59738,C1(NC(=O)CCn2cnnn2)CC(F)(CNC(C2CCOC2)=O)C1 59739,c1(C(=O)NCC(C)CNC(=O)CNC(N)=O)cc2c(C(F)(F)F)cc(O)nc2o1 59740,C1(CNC(C2(CC=C)CCCC2)=O)CC(F)CN1C(C1CC1OC)=O 59741,N1(C(C(COC)C)=O)CC2(C)CN(C(c3ccn(CC4CC4)c3C)=O)CC2(C)C1 59742,CCCCCC(O)C(=O)N1CCC(NC(=O)COc2ccc(C(C)C)c(C)c2)C1 59743,c1(C(=O)NCCc2cn(-c3ccc(Br)cc3Cl)nn2)ccc2ncsc2c1 59744,C12(C(=O)NCC3(NC(CCC=C=C)=O)CCCC3)CCCCC1C2(F)F 59745,Cn1cc2cccc(C(=O)NC(=O)CCC3(C)CN(C(=O)CNC4CC4)C3)c2n1 59746,N1(C(c2c(N)c(C(F)(F)F)ccc2)=O)CCCC2CN(C(c3cnc[nH]3)=O)CCC12 59747,n1(CC(=O)N(C(C)C2CC2)C2CC2)nc2ccccn2c1=O 59748,C=CCC(C)(C)CC(C(=O)NC1(C)CC1)N1CCC(C)(F)C1 59749,Cn1ncc2nc(O)c(C(N3CC(CNC(=O)Cc4cccs4)C3)=O)cc12 59750,C1(CC)CN(C(C2CC(C#N)(OC)C2)=O)CCN1C(=O)CCc1cccc(C)n1 59751,Cc1cc(CC(=O)NCCCN(C(=O)C(C2CC(C(F)F)C2)C)C2CC2)n(C)n1 59752,C(CNC(c1cc(OC)no1)=O)(CC(F)(F)F)NCC(N1C(CC)CCC1)=O 59753,c1(C(=O)NC2CCN(C(c3cc(=O)cc(Cl)[nH]3)=O)CC2F)cccc2sccc12 59754,N1(C(C(C)=C2CC2)=O)CCC(NC(=O)COC2CCOCC2)C2(CCC2)C1 59755,C(=O)(C(C)C(CC)CC)NCC(CC)NC(=O)CCCC1CCOCC1 59756,c1(CC)cc(C(=O)NC(C)(CSC)C(=O)NCC2CC2Cl)n(C)n1 59757,CC(O)C(C)C(=O)NCCOC1CN(C(c2nccnc2-n2ccnc2)=O)C1 59758,CCC(C)C(C(=O)NC1(CO)CC2CCCC12)NC(=O)C=CC(F)(F)F 59759,c1(C(C)=O)ccc(=NCCNC(c2ccc(-c3cccs3)cc2)=O)[nH]c1 59760,Cc1cnc2c(cnn2CC(=O)N(CC(C)NC(=O)CC2CCOC2)C)c1 59761,C12(NC(CCCOC)=O)CCC1CN(C(=O)CCN1CCCS1(=O)=O)C2 59762,N#CC1CN(Cc2ccccc2)CC1NC(=O)NCCc1ccccc1Br 59763,C(=O)(C1=C(Cl)CCCC1)N1CCCC(C)(C(=O)NC(c2nc(C)on2)C)C1 59764,C1(N(C(C(CC#C)C)=O)C)CCCCN(C(c2onc(CC)c2C)=O)C1 59765,C1(CC(=O)NC2CN(C(C(C=CC)O)=O)CC(C)C2)C2CC3CC(C2)CC1C3 59766,CN1CCC(O)C(NC(N2CCN(CC3CCCCC3)CC2)=O)C1 59767,N1(C(c2c(C)nc(COC)s2)=O)CC2CCN(C(=O)CCc3ccco3)C2C1 59768,CC1(C)CC(C)(CNC(=O)Cc2nc[nH]n2)CN1C(=O)CCn1cccc1 59769,c1(C(C(=O)NCC#CCNC(Cc2c(C)cco2)=O)=O)sc2ccccc2c1C 59770,Cc1ccc(C(=O)NCCSCC(=O)NCC(C2CCCO2)C)c(F)c1 59771,C(=O)(C1=NNC(=O)CC1)N1CCCC(NC(C2CCCC(C(=O)OC)C2)=O)CC1 59772,c1(C(N2C3C(N(C(C=C(C)C)=O)C)CC(C3)C2)=O)cc([N+](=O)[O-])cn1C 59773,c1(CCC(=O)NC(C)CNC(=O)C2CC2)ccc(Br)cc1 59774,Cc1ccc(-c2cccc(CNCc3cccn4ncnc34)n2)c2cn[nH]c12 59775,CCCCCCCC(F)C(=O)NCCC1CCCN(C(=O)C(O)C2CC2)C1 59776,N1(C(C(C)n2cccn2)=O)CCN(C(=O)CNC(C2CCCC23CC3)=O)CC1 59777,N1(C(C2CC3(CC(C)C3)C2)=O)CCN(C(C2CCCC3(CC3)C2)=O)C2COCC12 59778,C1(COC)CCN(C(=O)Cn2c([N+](=O)[O-])cnc2C)CC1(F)F 59779,N1(CCCC(CC)=O)CCN(Cc2ccccc2)C2CC12 59780,N1(C(C2N(C)CCC2)=O)CC2CC1C2NC(C1CCN(CC(F)(F)F)C1)=O 59781,c1(C(N2CC(OC)(CNC(C3(CCF)CC3)=O)C2)=O)ccnc(F)c1 59782,C1(NC(C2(CO)CCN(C(c3n(CCC)ncc3)=O)C2)=O)CCCC(O)C1O 59783,C1(CN(C)C(C2CC2F)=O)CN(C(=O)CCOC2CC2)CC12CC2 59784,c1(C(N(C(CNC(C2CC(C(F)F)C2)=O)C2CC2)C)=O)cccc2nccn12 59785,C1(NC(C(CC)N(CC)CC)=O)CCCC12CN(C(c1cc(C#N)[nH]c1C)=O)C2 59786,N1(C(C(C)NS(C)(=O)=O)=O)CCCC(C)(CNC(=O)CCSc2ccccc2)C1 59787,C1(CC(=O)NCCN(CCCN(C)C)C(=O)C=C(C2CC2)C2CC2)NC(=O)NC1=O 59788,N1(C(CSC(C)C)=O)CC(NC(C23CCC(F)(CC2)C3)=O)C2CCCCC12 59789,c1(C(=O)NCC(CC)(CC)NC(C2SCCC2C)=O)ccc(Cl)cc1O 59790,C(=O)(C#CC(C)(C)C)N(C(C)CNC(c1snnc1C1CC1)=O)CC 59791,Cc1ccc(Cl)cc1C(=O)NCCN(C)C(C1COCC(=O)N1C(C)C)=O 59792,N1(C(CC=C)=O)CC(F)CC1CN(C)C(c1cn(-c2ccccc2)cn1)=O 59793,S(=O)(=O)(c1cnc(NCCc2cc(Br)no2)c(Cl)c1)N1CCn2c(C)ncc2C1 59794,CCC(C)C(O)C(=O)N1C2CCC1(CNC(C1(C)CCC1)=O)CC2 59795,c1(C(=O)NC2C3CC2CN(C(C2CC(O)C2)=O)C3)cc2scc(Br)c2[nH]1 59796,C1(CNC(CC2C(C)C2)=O)(CO)CCN(C(c2ccc([N+](=O)[O-])o2)=O)CC1 59797,C(CNC(=O)Cc1cnnn1C)(CC(F)(F)F)NC(C(C)SC)=O 59798,C1(NC(C(C)(N(C(=O)C=CCN2CCCC2)C)C2CC2)=O)CNC(=O)OC1 59799,c1(NC(C2CC=CC(NC(C(C=C=C)C)=O)C2)=O)ccc(F)cc1O 59800,Cc1nc2cc(C(=O)NCC3COCC3NC(=O)CSCc3ncc[nH]3)[nH]c2s1 59801,c1(SC)nc(N2CC(Nc3ncc(C4CC4)cn3)C(F)C2)ncc1F 59802,N1(C(C(C)OCC#C)=O)CCN(C(c2c(C)noc2C)=O)CC1c1ccccc1 59803,N1(CC)CC(NC(=O)C(CC2CCCC2)NC(=O)C(C2CCOCC2)=O)C(C)C1 59804,N1(C(CC2(CC(=O)OC)CCCC2)=O)CCCC(C)(C(=O)NC2CC(CF)C2)C1 59805,CCC(C)C(O)CC(=O)NC1(CN(C(=O)Cc2n[nH]c3ccccc23)C)CC1 59806,N1(C(C=CC(=O)OCC)=O)CC2C(NC(C3CN(CC)CCO3)=O)C2C1 59807,N1(C(C2(C#C)CN(C(=O)CN3C(=O)CCCC3=O)C2)=O)CC2(CC2)CC1CO 59808,C(=O)(CS(=O)(=O)C1CC1)NCC(C(C)C)NC(C1(CC(=O)OC)CCCC1)=O 59809,C(=O)(C(CCC(C)(C)C)N(c1ccccc1C(C)C)C)NC1CC(C(=O)OC)C1 59810,C(c1ccccc1Cl)=CC(=O)NC1CCCN(C(=O)CC2COCCO2)CC1 59811,C(c1ccncn1)=CC(=O)NC(C(C)NC(c1cscc1F)=O)C 59812,C1(C(N2C(C)(C)CC(NC(C3CCCSC3)=O)C2)=O)COC2COCC2O1 59813,C1(CCC)CC1N=c1[nH]c(N(C)Cc2nn(C)c3ccccc23)nc2ccsc12 59814,c1(C2(C(=O)NC(CC)C(C)(C)O)CC2)ccc(C)c(Cl)c1 59815,c1(N2CCC(C)(C)CC2)ccncc1S(=O)(=O)N1CC(C)(C)OCC1CO 59816,c1(C(=O)NC2CC(C)(NC(C(C=C=C)C)=O)C2)cc(O)nc(C)n1 59817,c1(C(=O)NCC2C=CC(NC(C3(CC)C=CCC3)=O)C2)[nH]c(O)nc1C 59818,CCCC(C(=O)N1CCOC(CCNC(=O)C(F)=C(C)C)C1)N(C)C 59819,N1(C(CCNC(=O)OC)=O)CCC(NC(=O)CC2COCCN2C)C1C(C)(C)C 59820,C1(C(=O)NCCC(C)CCO)(OC)CCN(C(=O)OC(C)(C)C)C1 59821,c1(C(N(CC(C)O)CCNC(c2cncnc2)=O)=O)ccc(Cl)cn1 59822,N#Cc1cc(C(N2CCC(CC(=O)Nc3ccc(F)c(F)c3Cl)C2)=O)ccc1F 59823,C1(NC(C2(NC(CC=C)=O)CC(F)C2)=O)CCOC1C=C 59824,N1(C(=O)NC(c2ccncc2Br)C)CCC2CCC12c1cccs1 59825,N1(C(Cc2c(C)cco2)=O)CCCC(NC(c2ccc(C(C)(C)C)cc2)=O)CC1 59826,C1(C)(C(=O)NCC(C(=O)OC)(C)C)CCCN(Cc2cccc(O)n2)C1 59827,CC(C)CC(C)N(C(=O)CONC(c1coc(C(F)F)c1)=O)C 59828,C(=O)(C(F)C(C)CNC(c1cc(C)c(N)cn1)=O)N1CCC(C(=O)OCC)C1 59829,C(=O)(CC1C(=O)Nc2ccc(C)cc21)NC(CNC(C(CCCC)O)=O)(CO)CO 59830,C(CCN=c1[nH]c(C)cc(=NC(C)c2c(F)cccc2F)[nH]1)C1C(C)=NNC1=O 59831,C(=O)(C1CNc2ccccc21)NCC1CN(C(CC2C(C)(C)CCCO2)=O)C1 59832,C12(NC(C3CCCCN3C(C3CCC3)=O)=O)CC(C1)N(C(=O)CCCCO)C2 59833,c1(C(N2CC(CC(C)NC(C3(Cl)CC3(C)C)=O)C2)=O)cc(-c2cnn(C)c2)[nH]n1 59834,CC1CN(C(=O)C(=O)C2CCCC2)CC(C)CN1C(=O)Cc1cc(C(N)=O)co1 59835,c1(C(CC)NCC2=CCCCCC2)cc(Cl)cc(Cl)c1F 59836,Cn1cc(C(=O)NC(C)(CNC(c2csc(C(F)F)c2)=O)C2CCC2)nc1O 59837,c1(CNC(CN(C(=O)C(CC)OC)CCC)=O)ccnn1CCF 59838,C1(C(N2CCCCC2C2CC2)=O)C2CC(O)C(C2)N1C(=O)C(O)CC(F)(F)F 59839,CC1=NN(C)C(=O)C1CC(N1CCC(NC(c2ccnn2C(C)C)=O)C1)=O 59840,C1(O)(C(=O)NCC(N(C(c2ncn(CC)n2)=O)C)C2CC2)CCC(C)CC1 59841,c1(OCCCN(CC(O)CN(C)C(=O)C2CC2)C(C)C)ccc(F)cc1Cl 59842,c1(CC(=O)N(C(C)CNC(c2cscn2)=O)CC)conc1C 59843,N1(CC(=O)NC2CC(N(C(=O)CNS(=O)(=O)N(C)C)C)C2)CCCCCCC1=O 59844,C(=O)(CC(C(F)(F)F)NC(=O)COCC=C)NC1(CC#C)CC1 59845,N1(C(C2(CC#C)CCOC2)=O)CC=CC(C(=O)Nc2cc(OC)ncn2)C1 59846,c1(C(=O)NC2C(CNC(c3ccnnc3O)=O)CCC2)cccc2[nH]nc(O)c12 59847,C#Cc1cncc(C(N2CCCC2C2CCN(CCN3CCNC3=O)CC2)=O)c1 59848,C(=O)(CCC(C)(F)F)NCCCCC(C)NC(C(C)C)=O 59849,c1(Nc2ccc(SCC(N3C(CC)(CC)CCC3)=O)cn2)ccccc1[N+](=O)[O-] 59850,C(=O)(C(C(C)C)NC(C)=O)N(CC(CN(C(CCN(S(CC)(=O)=O)C)=O)C)O)C 59851,c1(NC)ccccc1C(N1CC(C)(NC(C2C3CC4C(C3)C24)=O)C1)=O 59852,c1(C(=O)NC2CCC(NC(c3cnc(OC)nc3)=O)C2)ccc(I)c([N+](=O)[O-])c1 59853,C1(NC(c2ccn(C(F)F)n2)=O)CC12CCN(C(C1CC1n1cccn1)=O)CC2 59854,c1(C(N2CCC(C(C)NC3CC3)CC2)=O)ccccc1F.c1(N)nccc(C(=O)O)n1 59855,C12(C(N(CC(c3nn[nH]n3)C)Cc3ccc(C)cc3)=O)CC=CCN1CCC2 59856,c1(N2CC(CC(C)NC(COCCCCCC)=O)C2)ncc([N+](=O)[O-])cc1C#N 59857,Cc1cccc(Cl)c1-n1cc(C(N2CCC(NC(=O)CCN(C)C)CC2)=O)nn1 59858,C(=O)(CC(C)CC(=O)OC)N1CCCC(CC(=O)N(CC(C)OC)C)C1 59859,c1(N2CCC(NC(C(=Cc3cccs3)C)=O)(CF)C2)cc(Cl)nc(C2CC2)n1 59860,CC(C)CC(C)(CO)NC(=O)C(CNC(=O)Cc1cccnc1)CC1CC1 59861,C1(CCNS(=O)(=O)c2ccoc2Cl)CCC2(CCOCC2)CO1 59862,c1(CN2C(COC(CN3CCC(C)CC3)=O)CCCC2)cc(F)c(Cl)cc1O 59863,Cn1cnc2c(NC3CCN(Cc4ccc(Br)c(Cl)n4)C3)ncnc12 59864,C1(NC(C)=O)CCC(C(=O)NCC2CCCN(C(C3(C(C)(F)F)CC3)=O)C2)CC1 59865,C12CCCN(C1)C2=O.C1(c2nnnn2C(C)C)(NCC=C(C)C)CCCC1 59866,C1(CN(C)C(C2CCC(=O)N2C2CC2)=O)CCCN(C(=O)C=Cc2cc[nH]n2)C1 59867,c1(C(=O)NCCN(CC(C)O)C(=O)Cc2ccco2)ccn(C2CCC2)n1 59868,S(=O)(=O)(CC(=O)NCC1CN(C(c2cnc(Cl)n2C)=O)CC1O)NCC 59869,C1(COC)(CNC(=O)CC(C)F)CCCN1C(c1cccc[n+]1[O-])=O 59870,CCCC(CCC)C(=O)N1CCCN(C(=O)Cn2cccc(N)c2=O)C(C)C1 59871,C1(C(=O)Nc2cc(O)ncn2)CN(C(c2ccc(O)nc2)=O)CCC1O 59872,S(=O)(=O)(C1CCCN(C(=O)OC(C)(C)C)C1)N1CC(c2c(SC)cccc2)C1 59873,N1(C(c2cn(CCNC(c3c(COC)noc3)=O)nc2)=O)CCC(CO)C(O)C1 59874,N1(C(C(C)CO)=O)CC2(C1)CN(C(c1cn(C)cc1C(F)(F)F)=O)C2 59875,C1(C(=O)NCCOC)CC12CCN(C(c1ccsn1)=O)C2 59876,C1(c2n(CC=C)nnn2)(NC(C)(C)C2CC2)CC2CC1CC21OCCO1 59877,c1(C(=O)NC2C(NC(CCC(c3ccc(C)cc3)=O)=O)C2)cc(F)ccc1Cl 59878,C(CNC(C1CC=CC1)=O)(C(C)C(C)C)NC(c1c(NCC)cccn1)=O 59879,N1(C(C(N2CCNC2=O)C)=O)CCCC(N(C(=O)Cc2n[nH]c(=N)s2)CC2CC2)C1 59880,N1(C(C2CC(Cl)(Cl)C2)=O)CC2CN(C(C3CC(CF)C3)=O)CC2C1 59881,c1(C(=O)NC2CCC(C(N3CCC(O)CC3)=O)C2)ccc2occc2c1 59882,C12(CC(=O)NC3CN(C(=O)CCc4nc[nH]n4)CC3O)CCC(CC1)C2 59883,c1(NC(C2CC3C(C2)C3(F)F)=O)nc(Cl)cc(Cl)n1 59884,CCC1=C(C(=O)N2CCCCC2CCNC(=O)CC(O)CN(C)C)CCCO1 59885,N1(C(C(c2ccn(C)c2)C)=O)CCCC1CC(N1CC(F)C1)=O 59886,C(=O)(C(C(C)(C)C)NC(c1ccccn1)=O)N1CCN(C(CC)=O)CC1 59887,C1(C(=O)NCCC2(CNC(Cc3c(C)ocn3)=O)CC2)CCn2ccnc2C1 59888,C1(C(N(CCC=C)CC)=O)CC2(CC2)CN1C(c1cn(CCO)nn1)=O 59889,C1(NC(c2nc(C(C)C)sc2)=O)CC2(CCCCN2C(C2(O)CCC2)=O)C1 59890,C(=O)(C(F)(F)c1cncs1)NCC(C)NC(=O)C(c1ccc(Cl)s1)C 59891,N1(CC(N2C(c3ccc(C)cc3)CCC2)=O)C(=O)CN(C)C1=O 59892,Cc1nc(N2CCC2(C)C(=O)Nc2cccc(S(=O)(=O)F)c2)nc2ccccc12 59893,C1(O)(C(=O)NCC2CC(NC(C(C)(C)NC(C)=O)=O)C2)CN2CCC1CC2 59894,C#CCCN=C(NCCc1ccccc1C#N)NCCc1ccn(C)c1 59895,CC1C(C)N(C(=O)Cc2ccc(C#N)cc2)CCN1C(=O)CN1CCOCC1 59896,N1(C(COC(C)=O)=O)CC(NC(C2(C)CC=CC2)=O)CC12CCC2 59897,C(CC(C(=O)N1CCCCC1CCNC(=O)CCCn1ccnc1C)OC)OC 59898,c1(C(=O)NC2CC3CCC(C2)N3c2cc(=O)n(C)cn2)nc2ccccn2c1F 59899,c1(C(C(=O)NC2CC(F)(CNC(c3cc(F)c[nH]3)=O)C2)=O)ccc(F)c(F)c1 59900,N1(C(CC2CC(OC)C2)=O)CC(C(=O)Nc2cc(C)cnc2O)CC(C)C1 59901,C(=O)(C1=CCCCO1)N1C(C(=O)NCC2CCCN(C)C2)CC1 59902,c1(C(=O)NC(CCN(C)C(C23CC4CC2C3C4)=O)(C)C)ccc2c(n1)CCCN2 59903,C(C1C(C(=O)NCC2(CN(C(=O)CC(C)O)C)CC2)C1(C)C)=C(C)C 59904,CC1(C)CN(C(=O)COC2CCOCC2)CC(CNCC2(C(N)=O)CC2)O1 59905,c1(C2(C(=O)NCC=CCNC(CCC(C)OC)=O)CC2)ccccc1C#N 59906,C1(NC(C=COCC)=O)C2CCCC1CC(NC(=O)C(O)CCSC)C2 59907,c1(C(N2CC(CNC(C(c3ccccc3)NC(N)=O)=O)C2)=O)cc[n+]([O-])cc1 59908,C1(O)(CNC(c2c(C)cno2)=O)CCCN(C(C2(N3CCOCC3=O)CC2)=O)CC1 59909,C1(NC(C(CNC(c2c(NC)scn2)=O)(C)C)=O)CN(C)C(C)(C)C1 59910,Cc1ccc(C)c(CCCC(=O)NC2(CN(C(=O)COCC(C)(C)C)C)CC2)c1 59911,C#CC1(NC(=O)CN(C(=O)CN(c2ncccn2)C)CCOC)CCC(C)(C)C1 59912,c1(COCC(=O)NCCC2CCC(CC3(NC(N)=O)CC3)C2)ccc(Cl)cc1 59913,C(C(=O)NC(CC)C(=O)N1CC(O)(CCO)C1)(C(C)C)SC 59914,C(=O)(C(C)(C)C)N.C(C)(C)(CCCNC(CN(C)CC=C(C)C)=O)N 59915,c1(C(=O)NCC2(O)CCN(C(C(C)SC)=O)C2)coc2ccc(OC)cc12 59916,C(=O)(C1=C(Cl)CCOC1)N1CCC(CC)CC1C(N1CCC1(C)C)=O 59917,C12(C(=O)NC(C)C(C)(C)C)CCCC1CCN2C(c1cn(C)c(=O)cn1)=O 59918,CC1(C)CCCN(C(=O)CSCCc2ccccc2)C1CNC(c1cscn1)=O 59919,C1(C(=O)NC2CC(CC=CC(=O)OCCCN(C)C)C2)CCCC(F)C1 59920,C=C(C)CCC(=O)NC(CN(C(=O)C(C)(c1cccnc1)OC)C)(CO)CO 59921,CC1(C)Cc2cc(C(=O)NC3CC(C)(NC(C4CCCC(C)(C)C4)=O)C3)sc2C1 59922,N1(C(=O)CC2COC(=O)C2)CCCN(C(=O)C(=O)NCC(F)(F)F)CC1 59923,C1(F)(C(=O)NCCCC(C)NC(C2(c3ccnn3C)CC2)=O)CCCN(C)C1 59924,C(C(O)CC(=O)NC1CC(=C2CC2)C1)NC(CC1C(=O)OCC1)=O 59925,c1(C(=O)NCC2N(C(c3cncc(C=C)c3)=O)CCC2C)ccc2c(c1)CCO2 59926,C1(OC)(CNC(=O)CSCC(F)F)CCN(C(=O)Cc2cnc(C)[nH]2)C1 59927,N1(C(c2[nH]cc(C)c2)=O)CC2OCC(NC(=O)CCc3ccc(O)nn3)C2C1 59928,c1(C(=O)NCCC(=C)CNC(=O)CCN(C(CC)CC)C)ccc(O)c(N)n1 59929,c1(OC)ccc(CN2CC3CC3(C(=O)Nc3cc(Cl)ncc3Cl)C2)cc1Br 59930,C1(CC(=O)NC2(C(N(C(C)C(N)=O)C)=O)CC2(C)C)C(C)(C)C1(C)C 59931,Cc1nc(C)c(CC(=O)N(CC(C)(C)CNC(C2(CCN(C)C)CC2)=O)C)s1 59932,C1(NC(C(CC)=CC)=O)CCN(C(c2ccnc(NC(C)=O)c2)=O)C(C)C1 59933,N1(C(CC=C(C)C)=O)CC2CC(NC(=O)C(C(C)C)n3ccnc3)C1C2 59934,N1(C(c2scc(C(C)=O)c2)=O)CCCC(C)(NC(=O)COCC2CCOC2)C1 59935,Cc1c(F)ccc(C(N2CCCN(CC#N)CC2)=O)c1C#N 59936,c1(C(N2CCCC(C)(NC(c3cc(CC)no3)=O)C2)=O)cc(F)c(F)c(Cl)c1F 59937,c1(C(N2CC(C(=O)Nc3nnc(C)o3)C(O)CC2)=O)cc2cccc(O)c2[nH]1 59938,Cc1cc(F)ccc1C1CCCN1CC1(C(=O)O)CCCOC1.n1(C)nnnc1OC 59939,CC1=C(C(=O)N2CCC(CNC(C3OCCC3(C)C)=O)C(C)C2)C(=O)OC1(C)C 59940,C1(NC(C2C(=C)C2)=O)CC(F)CN(C(c2ncc(C)cc2F)=O)C1 59941,CC1(C(=O)NCCC(N)=O)CCN(Cc2ccncc2Cl)C1 59942,C1(CC(N2CC(O)(CNC(c3cc(C(N)=O)oc3)=O)C2)=O)COCCOC1 59943,N1(C(c2ncc(N(C)C)nc2)=O)CC2=C(C1)CN(C(=O)C#CC1CC1)C2 59944,C(=O)(C(F)(F)C(F)F)NCC(CNC(CCC=CC)=O)(C)C 59945,C(C(CNC(C1(Cc2cnn[nH]2)CCCC1)=O)CO)NC(c1cscn1)=O 59946,C1(NC(C(C2CCCC2)OC)=O)CCC12CCN(C(c1cnn(C)n1)=O)CC2 59947,c1(N2CCC(C3N(C(CCCC(C)=O)=O)CCC3)C2)nc2cccnc2s1 59948,Cc1sc(Br)c(C(=O)NC2CC(F)CN(C(=O)C=CCO)C2)c1C 59949,CC1CN(C(C2(C#N)CC2)=O)CCN1C(=O)C(C)C(F)(F)F 59950,Cc1cccc2cc(C(=O)NCC(C3CCC3)NC(C3CCCN(C)C3)=O)nn12 59951,C1(C)(C(=O)NCCN(C(c2cn(CC)nc2)=O)C)CC(C(F)(F)F)=NO1 59952,N1(C(CC2ON=C(C)C2)=O)CCCC(NC(c2c(C)nc(C)n2O)=O)CC1 59953,Cc1ccc(C=CCC(=O)NC2(CCNC(C3CC3F)=O)CC2)cc1 59954,Cc1c(C(N2CC(NC(=O)C3=CCCCO3)C(C)C2)=O)sc2cncn12 59955,N1(C(c2c(C)coc2C)=O)CCC(NC(c2cnn(C)c2C(F)(F)F)=O)C(F)C1 59956,c1(CC(=O)NCC(CCOC)NC(C2(O)CC(CF)C2)=O)cccc(Cl)c1F 59957,c1(CC(=O)NC2C(CNC(CNC(C)=O)=O)CCC2)cc(O)ccc1Br 59958,C1(NC(C2C(OC)C2)=O)CN(C(=O)CC2CC2)CC1c1ccnn1C 59959,N1(C(C2C(C=C)C2)=O)C(CNC(c2c[nH]nc2C(F)F)=O)CC2CCCC12 59960,CCC(C(=O)NCC1(C2(O)CN(C(=O)CC3(O)CCCC3)C2)CC1)C(C)(F)F 59961,n1(CCN(C(C(=O)Nc2n(C(CC)CC)ncc2)=O)C)cccnc1=O 59962,c1(C(C(=O)NCC(CC=C)NC(=O)Cc2cccc(OC)c2)=O)ccc(O)cc1 59963,O=[N+]([O-])c1ccc(CNCC2CCN(c3ncnc4cc[nH]c34)CC2O)cn1 59964,C=C1CCCN(S(=O)(=O)CC)C1.C1C(C)C(=O)N1CCOC 59965,N1(C(C=C(CCC)C)=O)CC2(CC(NC(=O)CCCCC(C)C)c3nccn32)C1 59966,CCC(C)(COC)C(=O)N(CCCN(C(=O)C(C)c1ccon1)C)C 59967,C1(F)(CNC(c2ccn(C(F)F)n2)=O)CCCN(C(c2ccccc2Br)=O)C1 59968,N1(C(C(C)N(CC)CC)=O)CC(F)(C(=O)NCC2CC(SC)C2)C1 59969,Cc1cc(NC(=O)C(N2CCCC2CC(c2ccccc2)O)=O)c(C)s1 59970,N(C(=NCCc1ccc(F)cc1C)NC1CC1)CC1(OCC)CCSC1 59971,C(CCC(C)C(=O)N1CC(C)(OCC(=O)NC2CCC(=O)NC2C)C1)OC 59972,N1(C(c2cccc(OC)n2)=O)C2CCC1C(CNC(c1cc(C)cc(Cl)n1)=O)C2 59973,c1(C(=O)NC(C(C)(C)NC(CCSCCC)=O)C)cc(F)ccc1F 59974,O=C(C1CCc2c[nH]nc21)NC1CC(NC(c2ccn(C3CCCCC3)n2)=O)C1 59975,N1(C(C23CCC(N=[N+]=[N-])C2C3)=O)C2CCCC1CN(C(=O)C=C1CCC1)C2 59976,C1(CNC(c2csc3nnsc23)=O)CC2CCC(C1)N2C(c1cscn1)=O 59977,c1(NC2CC(CC#N)C2)cc(Br)ccc1S(=O)(=O)N1CCSC(C)(C)C1 59978,c1(C(N2CCC3C(C2)CN3C(c2n[nH]cc2Br)=O)=O)ncc2[nH]ncc2n1 59979,O=CN1CCCC1C(N1CCC(CNC(c2csc(O)n2)=O)C1)=O 59980,c1(N(C)Cc2ccc(-n3cncn3)cc2)nc2c(F)cccc2n1C 59981,Cc1ccc2ncnc(N(C3CNCC(C)C3)c3ncccn3)c2c1 59982,c1(C(N2CC(CC)(NC(=O)Cn3ccnc3C)C2)=O)cnc2[nH]cncc1-2 59983,C1(NC(C2(F)C(C)C2)=O)(CNC(=O)CCCOC(C)=O)CCCC1 59984,N1(C(C2C(C3(C)COC3)C2)=O)C2CCC(C(N3CCCC(F)(CO)C3)=O)C1CC2 59985,C(=O)(C(O)CC(F)(F)F)N1C(C(C)C)C(C(=O)NCC(C)Cc2cn[nH]c2)CC1 59986,c1(CNC(C)=O)cccc2c1CCN(C(c1ccc3c(=NC)[nH]cnc3c1)=O)C2 59987,Cc1nc(-c2ccc(CN(C(=O)C(c3cnn(C)c3)C)C)cc2)sc1C(=O)O 59988,c1(NC(=O)NC(P(C)(C)=O)CCc2ccccc2)ccc2c(c1)C=CCCC2 59989,C1(COC)(CNC(c2nnc(C)s2)=O)CN(C(=O)C(c2ccc(C)s2)C)C1 59990,C12(NC(c3ccc(OCC=C)cc3)=O)CCC(CC1NC(=O)CNC(N)=O)C2 59991,c1(CNC(CN(C(c2n(CC)ccn2)=O)C)=O)ccccc1CO 59992,c1(OCC)cc(C(=O)NCC(CNC(C2(CC)CC2(F)F)=O)CO)ccn1 59993,c1(C(N2CCC(N(C(=O)COCC(F)F)CC)C2)=O)c(C)ccc(C)c1O 59994,N1(C(C(C(C)SC)O)=O)CC(NC(C2CN3CCCN2CC3)=O)CC12CCCC2 59995,CC(C(=O)NCCC1(NC(c2ccc(C(C)(C)C)cn2)=O)CCC1)S(N)(=O)=O 59996,c1(C(=O)NC2CC(CNC(C3(COC)COC3)=O)C2)sc(C)c(C)c1C 59997,CCCC(CNC(=O)C(=O)N(C)C)C(=O)NCC12CC(CO)(CO1)C2 59998,C1(NCC(=O)N(c2ccc(C)cc2)C(C)C)COC2(COC2)C1 59999,C1(NC(=O)CCC2CCCO2)CC2CCC(C1)N2C(C1CCC2C(C1)C2(F)F)=O 60000,CC1CN(C(c2cnc(CC(C)(C)C)s2)=O)CC(C)C1N=c1nc[nH]s1 60001,N1(C(=O)COCC2(F)CC2)CC2CCC1(CO)C2 60002,N1(C(CN(C)CC)=O)CCC2CC1CN(C(=O)CCc1cnc3n1CCOC3)C2 60003,CC1(C)OC2CCN(C(=O)Nc3nccn4ccnc34)CC2O1 60004,Cc1cc(=NCc2nnc(C)n2C)[nH]c(N2CCC(C(N)=O)CC2)n1 60005,Cc1nc(C(=O)NCC(CNC(=O)C(C)C(F)(F)F)CO)ccc1[N+](=O)[O-] 60006,N1(C(c2ccc(CC)[nH]2)=O)CCOCCC1C(=O)NC(c1cc(C)on1)C 60007,c1(C(C(=O)NCC2N(CCc3nc(C)sc3)CCC2)(C)C)cc(F)cc(F)c1 60008,c1(CC)ccccc1CC(=O)NCC12CC1CN(C(C1CC(SC)C1)=O)C2 60009,C12(CNC(=O)C3=CCCCCC3)CCCC1N(C(c1cccc(O)n1)=O)CCC2 60010,c1(C(N2CCC(C(C)NC(C(C(CC)C)O)=O)C2)=O)cnc2c(c1)c(C)nn2C 60011,c1(C(N2CCC(CC(C)(C)C)C2)C(=O)NCC)cncn1C 60012,C1(Cc2cn(CC(CNC(c3sccc3C(C)=O)=O)OC)nn2)C(C)(C)C1(F)F 60013,CN1CC2CC1CN2C(=O)CC1CN(Cc2cnc(Cl)nc2)CCO1 60014,C1(C(N2CC(CC=C)(C(=O)NCC(C)C(C)(F)F)C2)=O)CC2(CCC2)CO1 60015,C1(C(N2CC(OCC3CC3)C2)=O)(SC)CN(C(=O)CC2C(CO)C2(F)F)C1 60016,C12(NC(c3nc(CC)sc3N)=O)CCC(CNC(=O)C(O)C(C)OC)(CC1)OC2 60017,C(=O)(C1(C)CCn2ccnc21)NC1C(C(N(CC(CN(C)C)O)C)=O)COC1 60018,C(=O)(CC(C)C(F)(F)F)NC1(C(N2CC(CC)C(O)C2)=O)CC1 60019,C(CC)(CC(=O)N(C)CP(C)(C)=O)NC(COCC)=O 60020,C1(F)(CNC(c2ccon2)=O)COCCN(C(c2ccc(Cl)s2)=O)C1 60021,N1(C(C(C)CC(F)F)=O)CC2(CCCC2NC(c2cc(-c3ccco3)c[nH]2)=O)C1 60022,c1(C(C)C)scnc1C(=O)NCC(O)CNC(c1ncc(C(F)F)s1)=O 60023,C=C(C)CC(C(=O)NC1C2CCC1CC2)NC(C1CCN1CC)=O 60024,c1(C(=O)NCC2(CNC(CC(C)(C)OC)=O)CC2)ccc(OC(F)(F)F)cc1F 60025,n1(CC(=O)NCC2C3CN(C(CC(=C)C)=O)CC32)cc(P(C)(C)=O)cn1 60026,Cc1ccc(C(N2CC(F)CC2C(N2CC3C(CN(C)C)C3C2)=O)=O)nc1C 60027,c1(CNC(CCOCCN(C(CC(C)CN(C)C)=O)C)=O)cccc2c1OCC2 60028,CC1CCCCC1(CO)NC(C1(CCNC(c2csc(O)n2)=O)CCC1)=O 60029,c1(C(CCC)N(C)C(=O)NCCc2nccn2CC)ccc(Br)cc1 60030,S(=O)(=O)(c1cnn(CC)c1)NCC(=O)N(CCCCC)CCC=C 60031,N1(Cc2cccc(C)c2)Cc2ccc(C(=O)Nc3cncc(Cl)n3)cc2C1 60032,C1(C(=O)NC2(CC=C)CN(C(C3CC4CCC3CC4)=O)C2)CC2CCC1CC2 60033,c1(C(=O)NCC2CC(C)N(C(=O)C3CC3)C2)nc(O)nc(O)c1F 60034,c1(NCC2(OC)CCCCCC2)nccc(=NCc2nc(C3CCCO3)cs2)[nH]1 60035,N1(CC2CCN(C(c3cncc(C(=O)O)c3)=O)C2)CCc2ccc(O)cc2C1 60036,C(=O)(C(CCF)NC(=O)CCOCC(F)F)N1C(C(=O)OC)CC1C 60037,N1(C(c2ccc(SC)cc2)=O)CC(NC(c2cc(Br)ncc2F)=O)C(F)(F)C1 60038,CC1(C)CCCC1(C)NC(c1cnc(CNC(=O)CC2COCCO2)nc1)=O 60039,c1(C(C)(C)C)nc[nH]c1S(=O)(=O)NC1CNCC12CCC2 60040,c1(CNC2CCCC(C)C2)cc(Cl)c(Br)cc1F 60041,c1(CC(C)C)nc(C)n(-c2ccc(Cl)cc2)n1.C1(C=O)CCCCO1 60042,C1(C(=O)NCCCCN(C)C)(CC)CCCSC1.C12(CC1)C(=O)N2 60043,c1(N2CCC(CC(C)O)CC2)nc(=NCC2CCCS2)[nH]c2c1CSC2 60044,N1(C(CCCn2cnc(C#N)n2)=O)CCC2CCN(C(=O)COC3CC3)C2C1 60045,C(=O)(C(F)C(F)(F)C(F)(F)F)NCC1(F)CCC(NC(C2(C)CCC2)=O)C1 60046,C(=O)(C(CCC(C)C)N=C1NS(=O)(=O)c2ccccc21)NCCNC(=O)NC 60047,c1(C(=O)NCC(CN(C)C(c2coc(Br)n2)=O)O)ccccc1S(C)=O 60048,c1(C(N2C(CNC(C(C3CCOCC3)OCC)=O)C=CC2)=O)cncc(Cl)c1C 60049,N1(C(CC(C)SC)=O)CC2(C1)OC1(C)CC2(NC(=O)C(C)Oc2ccccn2)C1 60050,C1(NC(C2(OCC)CCOCC2)=O)CCC(C)N(c2ncc(Br)c(C)n2)C1 60051,N1(C(CNC(CC)=O)=O)CCC(C)(C)CC1C(=O)N(CC(C)C(C)(C)C)C 60052,CC1(C)OC(=O)c2cc(C(N3CC(O)(CNC(C4CC4C(F)F)=O)C3)=O)ccc21 60053,C(=O)(C(CC)CC(F)F)N(C1(CC=C)CN(C(=O)CC(C)n2ccnc2)C1)CC 60054,C1(C(N2CCC(CNC(c3cnn(CC4CC4)c3)=O)C2)=O)CCS(=O)(=O)C1 60055,c1(OC)ccc2c(c1C(=O)C(C1CC3CCC1CC3)C#N)CNCC2 60056,Cc1cc(OCCC(=O)NCC2(F)CCCN(C(=O)CCC(F)F)C2)cc(C)c1 60057,C#CCC(C)(CNC(=O)CCCN(C)C(C1CC2CC2C1)=O)CO 60058,CC1SCCC1N=c1nc(N2CCC(=NO)CC2)c2c([nH]1)COC2 60059,Cc1ncc(C=CC(=O)NCC2COCC2NC(C2(C)CC2(Cl)Cl)=O)s1 60060,c1(C(=O)OCC)c(C)ccnc1SC1CCN(CC)C1=O 60061,C(=O)(CC(=O)NC1C=CC(CNC(=O)C(F)CC2CCC2)C1)OC 60062,N1(CC)CC(C(=O)N(C)CC2CCN(C(=O)Cc3ccc(Cl)cc3)C2)CC1=O 60063,c1(C(=O)NCC(C)F)cc(O)nc2c1CN(C(C1CC1(Cl)Cl)=O)CC2 60064,C1(C(N(CCCC)C)=O)CCCN(N2CCC(NS(C)(=O)=O)C2)C1 60065,C1(C(=O)NC(C(=O)NCCOCC(C)C)c2ccco2)CCS(=O)CC1 60066,C=CCC(C(=O)N(C)CC1(O)CCN(C(=O)C2=NNC(=O)C2)C1)C(C)(C)C 60067,C=CC1(O)CN(C(=O)C(C)N(C(=O)CC2CC3C=CC2C3)C2CC2)C1 60068,Cc1nc2cccnn2c1C(=O)NC1COCCN(C(C2CCN(C)C2=O)=O)C1 60069,C1(CNC(CC(COC)C)=O)CCN(C(c2ccc(C)c(C)n2)=O)C12CC2 60070,C(CCCOC)(C(=O)N(C)CCN(CC)CC)NC(C(COCC)C)=O 60071,C1(F)(CNC(C=CCCC)=O)CCCN(C(=O)CCn2c(C)c(C)sc2=O)C1 60072,Cc1cncc(F)c1C(=O)NCC(=O)NC1CCC(C(C)C)C1 60073,C1(C(=O)NCC(n2cc(C3(O)CCCC3)nn2)C)(COC)CCCO1 60074,C(=O)(CC(C)(C)C(F)(F)F)NCC1N(C(CCOC)=O)CCC1C1CC1 60075,c1(SC)ccc(C(=O)NC2CN(C(=O)CC3COC(C(F)(F)F)C3)C2)cc1 60076,CC(C)(C(=O)NCCC1CCCN1C(C1(F)CCOC1)=O)C(F)(F)F 60077,Cc1cc(C(=O)N(C)CCN(C(=O)C2=NOCC2)C)c2[nH]cnc2c1 60078,N1(C(C(C)=CC)=O)CC2(CNC(c3cn(-c4cnn(C)c4)cn3)=O)CCC1CC2 60079,CCC(CC)C(F)C(=O)NCC1(C)CN(C(c2cnc(C(C)C)o2)=O)CC1C 60080,Cc1cc(C)c(C)c(C(N2CC(F)(CNC(=O)Cn3nnnc3C)C2)=O)c1C 60081,C1(C(N2C3C(NC(C(CC)OC)=O)(CCC3)CC2)=O)CC2CC1C1C2C1(F)F 60082,C1(NC(C(c2cc(C)sc2)(C)C)=O)CC(O)CN(C(c2c(O)cccc2F)=O)C1 60083,c1(C(C(=O)NC2CCSC2)C2CCCC2)cccc(NCC2CCCO2)c1 60084,C1(C)(C(N(C)Cc2ccco2)=O)CCCN(C(=O)CCc2cncn2C)C1 60085,c1(OC)nc(OC)nc(N2CCC(C(N3CC4CCCC4C3)=O)C2)n1 60086,c1(NC(N2CCC(C(F)(F)F)(OC)C2)=O)ccc(Br)c2cccnc12 60087,C(CCSC)(C(N)=O)NC(C(C)N(CCC)C(c1ccc(Cl)cc1)=O)=O.C(C)=O 60088,C1(C(N2CCC(=C)CC2)=O)CN(C)CCN1C(=O)Cn1ccnn1 60089,c1(C(N)=O)cccc(C(N2CCOCC2CNC(=O)C=C2CCC2)=O)c1N 60090,C1(NC(C(=O)NC(C(=O)OCC=C)C2CC(=C)C2)=O)COc2c(OC)cccc2C1 60091,CCC(CC(=O)N(C)CCOCCOC)NC(=O)CC1CCOC1C 60092,c1(CN(S(=O)(=O)c2cccc(C(F)(F)F)c2)C)cc2c(O)cccc2s1 60093,C(CC(C)CCO)NC(c1cncc(C(C)(C)C)c1)c1n(CC(=C)C)nnn1 60094,N1(C(CC(OCC)OCC)=O)CCN(C(=O)CS(=O)CC)CC12CC2 60095,c1(C(C)OC)nc(C)c(C(=O)NC(CNC(=O)COCCF)C2CC2)s1 60096,C=C(C)CCC(=O)NC(C1CCN(C(=O)C(C)N(CC(F)(F)F)C)CC1)C 60097,N1(C(C(C)OC)=O)CCC2CN(C(C3(O)CCC3)=O)CC2C1 60098,c1(C2(C(N3CC(CCNC(CCOCC)=O)C3)=O)CCCC2)cccc(Cl)c1 60099,C1(CC)CCC(C)CN1C(=O)CCOC1CN(C(=O)C(C)CC2CC2)C1 60100,C1(C(=O)NC(c2nncn2C)C)CN(C(=O)CCc2cn(C)cn2)CC12CCC2 60101,C1(NC(CCc2c(OC)cc(C)cc2)=O)CCN(C2CC2)CC1C#N 60102,c1(CCC)cc(C(=O)NCC2COC(CNC(=O)CN3CCOCC3)C2)c(C)o1 60103,CC12CSCC1CN(c1ncncc1Br)C2 60104,c1(C(=O)NCC2CCCN(C(C=CC3(C)COC3)=O)C2)ccc2ccsc2c1 60105,c1(CC)nnc2n1CCN(C(C(C)=Cc1ccccc1)C(=O)NCCOC)C2 60106,C1(C)(CNC(c2ccc(Cl)c(Cl)c2)c2n(CC=C)nnn2)CCS(=O)(=O)CC1 60107,c1(CC)ncccc1C(=O)NC(C1CCCCC1)C(=O)NCc1ccns1 60108,c1(OCCC)cccc(C(=O)NCC(O)CNC(=O)CCc2ccc(C)nc2)c1 60109,C1(CC(=O)NC2C(CNC(=O)C=CCN3CC4CC4C3)COC2)CCCCCC1 60110,N1(C(CSC)=O)CC(NC(c2cc3sccc3s2)=O)CC12CCCOC2 60111,C1(CNC(c2cocn2)=O)C2CN(C(=O)CCc3nc[nH]n3)CC12 60112,C(C(C)(CO)NC(c1csc(CS(C)(=O)=O)n1)=O)NC(C(F)=C(C)C)=O 60113,C(=O)(C(C)(C)CN1CCCC1)N(C)CC1CCN(C(C2C(C)C2C)=O)C1 60114,C12(NC(C)=O)CC1CN(C(=O)CN(CC(C)C)C1CCC1)C2 60115,N1(C(C(COC)C)=O)CCN(C(=O)Cc2ccc(Br)s2)C(CO)C1 60116,C(=O)(C(F)C(C)CNC(=O)CCC(C)(C)OC)N1CCC(OC)C1C(C)C 60117,C1(C)(C(=O)NC(C)CCNC(=O)Cc2cnoc2)CC1(F)Cl 60118,c1(N2CC3CC(NC(CC4C(C)(C)CCO4)=O)C3C2)ncnc(Cl)c1C#N 60119,c1(C(=O)NC(CC)CNC(c2cc(Cl)n(C)n2)=O)c(O)nnc2c1CCC2 60120,c1(C(=O)NC2C(NC(c3ccc(C(N)=O)cc3)=O)C2)cccn2ccnc12 60121,Cc1cc(O)ccc1C(N1CCC(NC(=O)Cc2cnsc2)CC1C1CC1)=O 60122,C1(NC(C(C)OC)=O)CN(C(=O)CCS(=O)(=O)N(C)C)C(C)(C)C1 60123,C(=O)(CCCn1cc(CCC(N)=O)nn1)NCC(=O)NC(C)(C)C 60124,C(CC)(CCC(=O)NCC1(SC)CC1)NC(CCC=CCC=C)=O 60125,C1(NC(c2c(CC)c[nH]c2)=O)CCC2CN(c3ncc(C)c(CC)n3)CC2C1 60126,C(C(CC(C)C)C(=O)NC1CC(CNC(C23CCC(N=[N+]=[N-])C2C3)=O)C1)OC 60127,CC(C)C(S(=O)(=O)N1CCC2(CC2)C1)c1ccccc1 60128,N1(C(c2ncn(CC)c2)=O)CC2CN(C(c3cn(C(C)C)cc3C)=O)CC2C1 60129,c1(C(=O)NC(C(CO)NC(c2cc(C)cc(C)c2)=O)C)cc2n(n1)CCCC2O 60130,CCCCC(C(=O)NCCNS(C)(=O)=O)NC(c1cnn(C)c1)=O 60131,CCC(C)(COC)C(=O)N1CCN(CCNC(=O)C=CS(C)=O)CC1 60132,N1(C(CCC#C)=O)CC=C(C(C)(C)C(=O)NC(C)C(=O)NCCF)C1 60133,C(CNC(=O)C(CO)NC(N)=O)(CC(=O)N=c1ccn(CC(C)C)[nH]1)OC 60134,C1(CCNC(c2c(COC)ccs2)=O)COCCN1C(=O)CC1CCC(C)(C)C1 60135,c1(C(N(CC(C)NC(c2c(O)ccc(C)n2)=O)C)=O)cnc2c(c1)OCC(=O)N2 60136,C(CNC(C1CC2CC2C1)=O)(C(=O)N=c1cc2n([nH]1)CCCC2)N(C)C 60137,C(C(=O)NC1(CCCCNC(c2cncs2)=O)CC1)(C1CCC1)OCC 60138,CC(C)CC(C(=O)NCC1CCOC1(C)C)NC(=O)CCC(F)(F)F 60139,CC1(C)OCc2c1nc(Cl)[nH]c2=NCc1c(F)ccc2ccc(Br)cc12 60140,C1(C(C)C)CN(C(c2ccns2)=O)CCN1C(c1c[nH]c(=S)cn1)=O 60141,N1(C(c2cnn(CC)n2)=O)CCC(C2CC2NC(=O)C(C(C)C)OC)CC1 60142,C(C(C)(C)C(=O)NC1CCC(CNC(=O)CC2CC2(C)C)C1)N(C)C 60143,C1(C2CC2)(C(=O)NC2CCC(NC(c3c(C)nc(CCCC)s3)=O)C2)CC=CC1 60144,c1(CC(N2CCC(NC(C(COC)C)=O)C23CC3)=O)cnc2n1CCOC2 60145,CC1C(C(N2CCC(O)CC2)C2CC3CCCC23)CCN1Cc1ccccc1 60146,C(=O)(CCCC(C)(C)C#N)N1C(C(=O)NC(c2onc(C)n2)CC)C(CC)CC1 60147,c1(C2(C(=O)NCCN(C(CSC)=O)C(C3CC3)C3CC3)CC2)ccccc1Cl 60148,O=C(C1CCSc2ccccc21)NC1CCCN(C(=O)Cc2cnccn2)CC1 60149,c1(C(=O)NC2CC(NC(c3cncc4c[nH]nc34)=O)C2)n[nH]c2c1NCCC2 60150,N1(C(CCC(C)C#N)=O)CC2(C1)OC1(C)CC2(NC(c2c(Cl)cnn2C)=O)C1 60151,CC1(C(=O)NCCCN(C(=O)Cn2ccnn2)CCO)CCCS1(=O)=O 60152,Cc1cnc2nc(C(=O)N(CC(C)(C)CNC(=O)C=CC3CCCO3)C)nn2c1 60153,N1(C(c2scc(COC)c2)=O)CC2CC2(CNC(=O)CSc2ccc(C)cc2)C1 60154,C1(C)(CC)C=C(C(=O)NCC(C)CC(=O)NCC(C)CC(=O)OC)C1 60155,CC1NC(=O)OC12CN(C(=O)CCOCCCNC(=O)CCc1ccccn1)C2 60156,N1(C(CC2N(C)CCC2)=O)CCC2(CCCCN(C(=O)C(F)(F)CO)C2)C1 60157,c1(C(=O)Nc2c(C)c(F)ccc2)cc2cc(-c3ccc(OC(C)C)s3)cnc2[nH]1 60158,c1(OC)cc(C(=O)NC(CNC(=O)CCn2cnc(=N)[nH]2)CO)ccn1 60159,C1(C(=O)NCC(CNC(c2cc(Cl)ccc2O)=O)O)CC12CCOCC2 60160,c1(OC)ccnc(F)c1C(N1CCC(O)(C(=O)NCc2nccnc2Cl)C1)=O 60161,CCC(CC)(CO)C(=O)NC1CCN(C(C2CCCCC2C(N)=O)=O)C1 60162,CCCC(CC)C(=O)N(C1CCCN(C(=O)CSc2ccncc2)C1)C 60163,N1(C(CCc2c[nH]c(=N)[nH]2)=O)CCCC(NC(C2CCNC2=O)=O)CCC1 60164,O=C1CCC2(CCCN(C(=O)Nc3cccc(CCO)c3)C2)CN1 60165,c1(C(N(CC(CC)NC(=O)C(C)P(C)(C)=O)CC)=O)coc2c1CCCC2 60166,N1(C(C(C(C)C)C2CCC2)=O)CC(C(N2CC(N(C)C)C(C)C2)=O)C(F)(F)C1 60167,CC1CN(C(c2c(C(F)F)cnn2C)=O)CCCN1C(C1CNC(=O)N1C)=O 60168,C1(CC(=O)NC2CCCN(C(=O)C(c3ccc(Br)cc3)O)C2)CCC(O)CC1 60169,N1(C(c2c(O)nc(=N)[nH]c2)=O)CCCC(C2(NC(=O)COCCN(C)C)CC2)C1 60170,C(C(C)C(=O)N(CCCn1ccnc1)C)N(C(C(C)C)=O)C 60171,C1(CC)CCN(C(=O)C(=O)NOC)C1CNC(=O)CSc1ccccc1 60172,c1nc2ccccc2cc1C(=O)NCC1(CO)CC1.N1(OC)CCC2(C1)CN(C)C2 60173,c1(CC)cc(C(=O)N(C)CCN(C(C2CCOC(CC)C2)=O)C(C)C)ncn1 60174,CC1CN(C(c2cc(Cl)no2)=O)CCC1N(C(=O)CNC(S(=O)(=O)C1CC1)=O)C 60175,C1(C)(OC)CCC(NC(C2CN(C(c3ccccc3O)=O)CC2(F)F)=O)CC1 60176,c1(C(N2CCCC(NC(CC3CCC(C)(C)C3)=O)CC2)=O)ccn2nccc2n1 60177,c1(CC)c(C(N2CCCC2CNC(=O)CN2C(=O)CNC2=O)=O)cnn1C 60178,C1(F)(NC(=O)CNC(=O)C(F)F)CCOC1.C1CC(=O)OCC#CCN1 60179,N1(C(CC2(OC)CN(C(c3cn(C)c(C)n3)=O)C2)=O)CC2(CCC(=O)N2)C1 60180,c1(CC(C)C(=O)NC2CC2NC(=O)CC2(CO)CC2)cccc(Cl)c1 60181,C1(C(c2n(CCC)nnn2)NCC(CO)OC)CCC(C)(C)CC1 60182,C1(CNC(C2C(C)C2)=O)CC2(CC2)CN1C(c1cnccc1Br)=O 60183,C1(NC(C=Cc2ccc(C)o2)=O)CC2CCC(C1C)N2C(c1ccncc1Cl)=O 60184,C(=O)(C1=CS(=O)CCC1)N1CC(NC(c2cc(CC)nc(O)c2)=O)C(CO)CC1 60185,C1(CNC(c2cc(CF)on2)=O)CN(C(C2(O)CCSCC2)=O)CC12CCC2 60186,C1(CNC(=O)CCCF)CCCCN(C(c2cc(Cl)cc(C(F)(F)F)n2)=O)C1 60187,C1(CNC(CN(C2CC2)CC)=O)CN(C(=O)CCC#N)CC(C(F)(F)F)O1 60188,c1(C(=O)NC2CC(C(=O)NCCCCSC)C2)nocc1Cl 60189,c1(C(=O)NCC(C)N(C)C)n[nH]cc1-c1ccccc1 60190,c1(C(=O)NC(c2cccnn2)C)csc(CCN)n1 60191,c1(C(=O)NCC2(F)CC(CNC(C(C)N(C)C)=O)C2)ccc(SC(F)(F)F)nc1 60192,C1(NC(=O)COCCF)CN(C(=O)CCCn2cncn2)C2(CCC2)C1 60193,N1(C(Cc2ccc(C)s2)=O)CC=C(C(=O)NCC2COC(=O)N2)CC1 60194,C(=O)(C(C)CCCCCC)NCc1c(C(N2C(C)(CCC)CC2)=O)con1 60195,C1(CNC(c2c(SC)cccc2)=O)CCCN(C(=O)Cn2nc(C)cc2C)CC1 60196,c1(C(N(CC(C)O)CCNC(C2C(OC)CC2)=O)=O)cocc1C 60197,C1(CNC(C2CC(F)C(=O)N2)=O)CCCCC1C(N1CC=CC1)=O 60198,N#Cc1ccc(CN2CCC(C(=O)Nc3nc(C4CC4)c(Br)s3)C(O)C2)c(Cl)c1 60199,N1(CC(N2CC(N(C(CC(C=C)C)=O)C)C2)=O)CCCCC(O)C1=O 60200,C(=O)(CC(C)(C)CC(F)(F)F)NC1(CO)CN(C(Cc2ccc(C)s2)=O)C1 60201,c1(OC)ccc(C(=O)NC2CC(NC(c3cnc(O)s3)=O)C(O)C2)c(N)c1 60202,C#CC1CCC(C(N2CCCC(N(C)C(c3cccc(F)c3OC)=O)C2)=O)CC1 60203,c1(CCSc2c(C(C)NCc3c(C)cccc3)cnn2C)c[nH]c2cc(F)ccc12 60204,c1(C(N2C(CNC(c3cc(CC)[nH]n3)=O)COCC2)=O)cnn2ccnc(N)c12 60205,S(=O)(=O)(c1ccccc1Cl)N1CC(CN(C(C(N2C(C)CCC2C)C)=O)CCO)C1 60206,CC(C)C(C(=O)N1CCCC(CC(=O)NCc2ncccn2)C1)N(C)C 60207,n1(CC(N2CCC(n3cc(Cn4cccn4)nn3)CC2)=O)ncc2ccccc12 60208,c1(C(=O)OC)ccc(NC(C2(C)CS(=O)(=O)C2)=O)c(I)c1 60209,C(=O)(CC1=CCOCC1)NC1C(CNC(CCOc2cc(C)cc(C)c2)=O)CC1 60210,c1(OC)ccc2c(=NCC3CCCN3C)[nH]c(N(C)Cc3ccnn3C)nc2c1 60211,C1(C(N2CCC(N(C(=O)CC3CC=CC3)C)C2)=O)CCC(=O)N(C2CC2)C1 60212,Cc1cccc(C(N2CC(CC(=O)NOCC3CC4C=CC3C4)CC2C)=O)c1.C1CC1 60213,CC(C)(CC#N)C(=O)NC1COCCN(C(c2c[nH]nc2Br)=O)C1 60214,c1(C(=O)NCCC2(OC)CN(C(C(=O)OC)=O)C2)ccc(C2CCC2)nc1 60215,C1(C(=O)NCC(C)N(C)C(C2(CC3CC3)CCC2)=O)CC2(CC(=O)C2)C1 60216,CCCCCCC(F)C(=O)NCCCCC1CN(C(=O)CCC2CC2(F)F)C1 60217,CC(CO)C(C)N=c1nc(N2CCn3nncc3C2)c2c([nH]1)COC2 60218,CC1(F)CC2(CN(C(C3(NC(=O)C(CO)C(C)(C)C)CCCC3)=O)C2)C1 60219,C1(CNC(C(C)NC(N)=O)=O)(NC(=O)CC2CCCCC2)CCCCC1 60220,C1(CNC(C(=O)NCCNS(C)(=O)=O)=O)CC2(CCNC2)CO1 60221,C1(F)(CNC(CCNC(C2C(C)C2)=O)=O)CCCN(C(C2CC23CCC3)=O)C1 60222,Cc1cc(N(C2CCN(C(=O)C(O)CCc3ccccc3)C2)C)nc(C)c1C#N 60223,C12(NC(CN3CC(C)(C)C3)=O)CCC(CC1NC(c1cnn[nH]1)=O)C2 60224,C12CCCN(C1)C2=O.c1(SC)nnc(C(c2snnc2C)=O)o1 60225,c1(CN2CC3N(C(c4cc(Br)ccc4F)=O)C(C3)C2)c(F)ccc([N+](=O)[O-])c1F 60226,C(CCCOC)(C(=O)N(CC(C)(C)COC)C)NC(C=CC(=O)OCC)=O 60227,CCCC(C)(C)CNC(=O)CC1CC1CNC(=O)CCc1ccc[nH]1 60228,C(CCC(C)(C)NC(C1CCCCCC1)=O)NC(C1(CC)COC1)=O 60229,c1(C(N(C2CCCN(C(c3n[nH]cc3[N+](=O)[O-])=O)C2)C)=O)ccc(S(C)=O)cc1 60230,c1(-c2cncc(C(N3CCCC(CN(C)CC4CC4)C3)=O)n2)ccc(O)cc1 60231,c1(C(=O)NCC(N2C(C)C(C)(C)CC2)=O)n[nH]c2cc(Br)ccc12 60232,n1(C(COC)C)cc(C(=O)NC2CC2NC(=O)C=CCO)ccc1=O 60233,CC1(C)CC(C(=O)NCC(C)(O)CNC(C2CCS(=O)CC2)=O)CNC1=O 60234,S(=O)(=O)(c1cn(CC)nc1CC)NCC(=O)OCCNCCCC 60235,N#Cc1ccc2c(c1)CC(NCC1CNCCS1(=O)=O)C2 60236,C#CCC(CC#C)C(=O)NCC1COCCN(C(c2ccc(C)cc2O)=O)C1 60237,c1(C(N2CC3C(CNC(c4c(C)n[nH]c4)=O)(C3)C2)=O)cnc2snc(C)c2c1 60238,N1(C(CSCC(N)=O)=O)CCCCC1C1(NC(C2CCC(C(F)(F)F)O2)=O)CC1 60239,N1(C(C2C(C(C)C)OCC2)=O)CCCC2(C1)CN(C(c1ccnc(Cl)c1N)=O)C2 60240,C1(C(=O)NCC2CC(O)C(O)C2)CCCCCN1C(C1CC1Cl)=O 60241,c1(OC)ccnc(O)c1C(=O)OCC(=O)NCC1(c2ccc(F)cc2)CCC1 60242,N1(C(C2(COC(C)C)CC2)=O)CC2CCC(C1)N2C(C1Cc2nncn2C1)=O 60243,c1(CCC(=O)N(C(C)C(=O)N(CCCCOCC)C)CCC)nccn1C 60244,O=C1CC2OCCC2(C(=O)NCC2CN(C(c3cnc(S)nc3)=O)C2)CN1 60245,c1(CCC(=O)NC(C(CO)NC(CC(=C=C)C)=O)C)ccc(Br)c(C)c1 60246,CC1CCN(C(=O)Cn2ccc(=N)[nH]2)C1CNC(=O)CCN1CCCCCC1 60247,c1(OC)noc(C)c1NC(=O)C(c1ccccc1)NC(=O)CC1CCCC12CC2 60248,N1(C(COC(CC)(C)C)=O)CC2CC(NC(c3csc(C)c3C)=O)CC(C2)C1 60249,C(=O)(C1CCCn2cncc21)NCC1(CNC(C(CCCC)O)=O)CCCCC1 60250,C1(C)(C(=O)OC(C(=O)NC)C)CC(C(C)C)=NO1 60251,C(C)(CCCCNC(C1CCOC1(C)C)=O)NC(c1cc(CCCCCC)on1)=O 60252,N1(C(C)C(=O)OCCOc2ccc(Cl)cc2)Cc2ccccc2C1=O 60253,CN1CCC(C(=O)NCC2(F)CCN(C(c3ncncc3Cl)=O)CC2)S1(=O)=O 60254,CC1(C)COC(CC(N2CCCCC2C(=O)NCCNC(=O)CO)=O)C1 60255,N1(C(c2cn(CCNC(CC(CC=C)(C)C)=O)nn2)=O)CCC2(CNC(=O)C2)C1 60256,C1(NC(C2N(C(c3cccc(C)n3)=O)C3(CC2)CC3)=O)CCc2ncnn2C1 60257,C1(NC(c2cc(OC)n[nH]2)=O)C2CC1CN(C(=O)C(F)CC1CCCCC1)C2 60258,C12(CNC(C=CCCC)=O)CC(NC(=O)C(C)C(F)(F)F)(C1)C1(CCOCC1)O2 60259,c1(CNCC2(C(N3CC(C(=O)OC)C(F)C3)=O)CC2)cc(I)ccc1Cl 60260,c1(C(N2CC(C(C)NC(C3CN(C)C3)=O)OCC2)=O)cnc2cc[nH]c2c1 60261,CCC(CNC(=O)CCP(C)(C)=O)(CC)C(=O)N(C1CCC1O)C 60262,C1(N(C)C(c2ccc(CO)o2)=O)CN(C(=O)CCc2ccsc2Cl)CC12CC2 60263,N1(C(CCc2cc(OC)no2)=O)C(C)C2CC1C2NC(=O)C(CO)N(C)C 60264,N1(C2CCN(C(C(CC)O)=O)C2)CCN(C(=O)CC(=O)N(C)C)CC1=O 60265,N1(C(CC2OCCN(C(C3CCN(CC)C3)=O)C2)=O)CCOC(CC)(CC)C1 60266,C(=O)(C(CC)CCCCCC)N1CCC(CC=C)(NC(=O)CSS(C)(=O)=O)CC1 60267,c1(C(=O)NCCC2C(C)CN(C(C3CCCC3)=O)C2)c(F)ccc2cnn(C)c12 60268,N1(C(=O)OCc2cc(OC)c(Cl)cc2)CC2CC(C)N(C(=O)C3CC3)C2C1 60269,C(C(CNC(=O)CCn1ccnn1)C(F)(F)F)NC(C(N1CC(C)C1)C)=O 60270,C1(NC(c2cncc(Br)c2)=O)CC2(C1)CC(C(=O)NCc1cnco1)C2 60271,c1(C(=O)NC(CN(C(=O)CC2CCC(=O)NC2)CC)C)cc(C)cc(C)c1C 60272,N1(C(C2=CCC(NC(C(CCC)CCC)=O)C2)=O)CCc2nnnn2CC1 60273,C1(C(N2C(CNC(C(CC(C)C)(C)C)=O)C=CC2)=O)CCc2ccccc2CC1 60274,c1(NC(c2nnc(C)n2C)c2nnnn2-c2ccccc2Cl)cc(Cl)c(O)c(Cl)c1 60275,c1(CC)oc(C)cc1C(=O)NC1CCCC1C(=O)NC(CC)C1CC1 60276,C(C(O)C(=O)NC1CC(F)(CNC(=O)CCC#N)C1)N(C)C 60277,c1(N(CCOCCNC(C(C)(C)NC(=O)OC)=O)C)cc(C#N)ccc1[N+](=O)[O-] 60278,c1(NC(C2CC(F)CN(Cc3cc(Br)ccc3I)C2)=O)cnc2ccc(F)cn12 60279,CCC(C(=O)N1CCC(CNC(c2csc(CC(F)F)n2)=O)C12CC2)C(F)(F)F 60280,c1(C(C)(C)C)ccc(C(=O)NCCOC2CN(C(=O)CCC3CC3(C)C)C2)[nH]1 60281,c1(C(N(c2ccc(C)c(F)c2)C)=O)cc2c(nc1N)CCC2 60282,C1(C(N(C(C)CCNC(=O)CCSC(F)(F)F)C)=O)C2CC3C(C2=O)C13 60283,C1(CNC(COc2cc(C)on2)=O)CN(C)CCN1C(C1CCCN1C1CC1)=O 60284,N1(C(C2CCC(C(C)C)CC2)=O)CC2CC1CN2C(=O)CC1CCS(=O)(=O)CC1 60285,C(C)(C(=O)N(C)CCN(C(=O)CCC1CCCO1)C)NC(=O)NC 60286,C1(NC(C(N2CCCN(CCC)CC2)=O)=O)C2CC3CC1CC(O)(C3)C2 60287,c1(OCC)c(CC(N2CC(OC)C(NC(=O)C(C)CC(N)=O)C2)=O)cccc1Cl 60288,C#CC1(C(N2CCN(C(C)CNC(=O)CC(C)F)CC2)=O)CCCCC1 60289,C1(N(C(=O)C(O)CC2CCCO2)C)CCN(C(=O)C(C)(C)c2ccccn2)CC1 60290,c1(CCC)cnnc(C(=O)N(CCC)CCNC(c2scc(OC)c2OC)=O)c1 60291,c1(C(=O)NC(CCC)CNC(=O)C(N2CCCC2)C2CC2)cn(CC)nc1C 60292,C1(OC)NC(C(=O)NCCn2cc(CN3CCNC3=O)nn2)CCC1Br 60293,N1(Cc2c(OC)cc(Br)cc2)Cc2[nH][nH]c(=NC(=O)c3ccc(F)c(C#N)c3)c2C1 60294,N1(C(C(C=C)(C)CCOC)=O)CCC2(CC1)OCCC2NC(C1(CCF)CC1)=O 60295,N1(C(C=CCC)=O)CC2CC1CN(C(=O)Cc1cc(C)[nH]n1)C2 60296,N1(C(C(C)COc2ccccc2)=O)CCC2CCC(C1)N2C(=O)CCC(F)F 60297,N1(C(C2(COC)CN(C(C3(CCCC)CC3)=O)C2)=O)CCC(C)(C2CC2)C1 60298,CCC(C)CCC(=O)NC(CNC(=O)CC12CNC(=O)C(C1)C2)CC 60299,N1(C(C(CCCC)NC(N)=O)=O)CCN(C(=O)C=Cc2ccsc2)CCC1C 60300,Cc1cc(Cl)cc(C(=O)N(C)CCNC(c2ncc(Cl)cc2Cl)=O)c1N 60301,C(=O)(C(C)C(C)S(C)(=O)=O)NCC1(CNC(CCOCCC)=O)CCCC1 60302,Cc1nccnc1CCNC(C1CSCN1C(C1CC(C)(C)CO1)=O)=O 60303,C(C)(C(O)C(=O)NCCOC1CN(C(=O)C(N)=O)C1)SC 60304,c1(C(c2n(CC)nnn2)Nc2cccc(CO)c2)cc(Cl)c(Br)cc1F 60305,c1(OC)ncc(Br)cc1CN1CCCN(C(c2ccn(C(F)F)n2)=O)CC1 60306,N1(C(c2ncc(C)nc2)=O)CCC2(CC1)CC2(CO)CNC(c1cocn1)=O 60307,C1(C(=O)NCC(CNC(c2c(CC)scc2)=O)(C)C)CCC(N(C)C)CC1 60308,C1(NC(C(OC)OC)=O)CS(=O)(=O)N(C)C12CCN(C(=O)CC1(C)CCC1)CC2 60309,c1(OCCC)cccc(C(=O)NC(c2cnsn2)C)c1 60310,C1(NC(C2(N(C)C(c3ccccc3)=O)CC2)=O)CCCN1C(C(C)(CO)CO)=O 60311,c1(C(=O)NC(C(C)NC(c2csc(CO)n2)=O)C)ccccc1Br 60312,C(CCC(C)(C)NC(c1nc(C)n(C)n1)=O)NC(CN(C(COC)=O)C)=O 60313,C(=O)(CC(C)(C)CC(F)F)N(C1CC2N(C(C3C(C=C)C3)=O)C(CC2)C1)C 60314,N1(C(c2cn(CCOC)c3c2cccc3)=O)CC(C)(C)OC2(CCOC2)C1 60315,C1(CCCNC(c2c(C)occ2)=O)CN(C(=O)CN2CCOC2=O)CCO1 60316,c1(OC)cc(OC)cc(C(=O)NCCC2CC(NC(C3CCCC3(F)F)=O)C2)c1 60317,Cc1ncc(C(N2CCC(NC(C3C4CNC(=O)C34)=O)C2)=O)cc1C#N 60318,C1(C(N(C2CN(C(=O)C3CC3)CC2O)C)=O)CC2(CCCO2)C1 60319,N1(c2nccc(OCCC)n2)CC2(CCC(NC(c3ccc(O)cc3)=O)CC2)C1 60320,N1(C(CS(=O)(=O)NC)=O)CC2CCCC(NC(=O)C(O)C3CCCC3)C2C1 60321,N1(C(c2c(C)ccs2)=O)CC2CCN(C(=O)C(c3ccc(Cl)cc3)O)CCC2C1 60322,N1(C(c2cccc(OC)c2)=O)CCC(C(=O)NCc2cnccc2C)CC1(C)C 60323,C1(CNC(c2c(CC)ocn2)=O)C2CC2CN1C(c1cncc(O)c1)=O 60324,c1(C(=O)NCCCCC(C)NC(CC(C)O)=O)ccc(O)c(C(C)(C)C)c1 60325,C1(CC)C(C(=O)NCCc2cccnc2C)CCN1C(=O)C(=O)NC1CC1 60326,c1(OC)cc(F)c(Br)cc1C(=O)NCC(O)CNC(=O)C=Cc1cnc[nH]1 60327,Cc1c(C(N2CC(O)(CC(N3CC(N(CC(C)C)C)C3)=O)C2)=O)ccn1C 60328,N1(C(C(C)C(C)(C)C)=O)CC(NC(c2occc2Cl)=O)C(C2CC2)C1 60329,CC1CCN(CCC(=O)NCC2CCCN2C(=O)COCC(C)(C)C)CC1 60330,C1(C)(CCC(N2CCC(OCC=CC)C2)=O)CCCN1C(=O)C(C)C(C)C 60331,C=CCN=C(NCC(=C)Cl)NCC.c12csc(n1)COC2 60332,CC1CCN(C(c2c(C#N)ncn2C)=O)CC1CC(=O)NC1(C(F)(F)F)CC1 60333,C(=O)(C1=C(C2CC2)C1)N1C(C(=O)NCC(C(C)C)O)C=CC1 60334,c1(C(=O)NC(CN(C(C(C(CC)O)C)=O)CC)C)cc2ccc(Cl)cc2[nH]1 60335,c1(-n2ccc(C)n2)ccc(C(N2CCOC(C)C2)C(=O)NCC2CC2)cc1 60336,N1(C(c2c(CC)cno2)=O)CC2CCC(NC(=O)Cn3nccc3C)CC2C1 60337,C=CC1(CC(N2CC(=CC)C2)=O)CN(C(C2(C)CCOC2)=O)C1 60338,C(N=c1nc2sccc2c(N2CC3CCC2C3)[nH]1)c1cnc(-c2ccn(C)c(=O)c2)s1 60339,C1(NC(C2CCCN(C(C)C)C2)=O)CN(C(=O)C(c2cnn(C)c2)C)CC1(C)C 60340,C1(NC(C=CCN(C)CC)=O)CCC(C(=O)NC2(CO)CC(F)C2)CC1 60341,Cc1c(C=CC(N2CCC(C)C(NC(=O)C(C)(C)N3CCCC3)C2)=O)cnn1C 60342,c1(C(=O)NCCC(C(C)C)NC(C(C=CC)O)=O)ccc(Cl)c(F)c1 60343,c1(CC)[nH]nc(C(=O)NC2CCCCCC2NC(=O)CC(C)C)c1[N+](=O)[O-] 60344,C(CCN(C)OC)NC(C1(C)CN(C(C(CC2CC2)OC)=O)C1)=O 60345,CN1CCN(C(c2cnc[nH]c2=N)=O)CC1C(=O)NC1(C)CCCC1O 60346,c1(C(N2CCC(N(C(CNC(CC(C)C)=O)=O)C)C2)=O)ccc(CF)cc1 60347,c1(CNC(CCCC#CC)=O)ccc2c(c1)CN(C(c1cccc(Cl)c1C)=O)C2 60348,C1(C)(C(N(CC)Cc2ccoc2)=O)CC(O)CN1C(=O)CC1CCCC2CC12 60349,CCC(Cc1ccccc1)CC(=O)NC(CNC(=O)CC1(O)CCOCC1)CC 60350,C1(C(N(CCN(C(C)C)C(C2CC2c2cccs2)=O)C)=O)SCCCS1 60351,C(=O)(CC(C)(C)C#N)NC(C)CNC(=O)C(C)CO 60352,c1(C(=O)NCCOCCN(C(C2(CCOC(C)=O)CC2)=O)C)cc(Cl)ccc1C 60353,c1(C(=O)NCC2N(C(C3(CC)COC3)=O)CC2)coc(C(N)=O)c1 60354,N1(C(c2c(C)cccn2)=O)CCC2(CCN(C(C3OCCN(C)C3=O)=O)C2)C1 60355,C(=O)(C1CCCc2sccc21)NCC(C)NC(c1cn(C(C)C)nc1C1CC1)=O 60356,c1(C(=O)NCC2CCN(C(C(C)OCC#C)=O)C2)ccc(C(=O)CC)cc1 60357,Cc1c(C(N2CC=CC2CNC(c2c[nH]nc2C(F)(F)F)=O)=O)cccc1C#N 60358,C1(NC(COC)=O)CC2(CCN(c3ccc([N+](=O)[O-])c(C(N)=O)c3)CC2)C1 60359,C=CC(C)(O)CC(=O)NC1C=CCC(C(=O)N(C)CCC2CCCC2)C1 60360,CC(C(C)(C)C#N)NC(C1CCCCN1C(=O)COC1CCCCC1)=O 60361,N1(C(c2cc(C)sn2)=O)CC(C(=O)NCC2(C)CC=CCC2)C2(CC2)C1 60362,C12(NC(=O)Cc3ccc(Cl)s3)CCCC1CN(C(c1cccc3c[nH]nc13)=O)C2 60363,c1(CNC(C2COCCN(C(=O)COCCO)C2)=O)ccc(F)cc1Br 60364,N1(C(c2ccc(CC)[nH]2)=O)CC(NC(=O)Cn2nc(C)cc2C)CC(O)C1 60365,c1(C(N(C(CNC(CC2C(C)=NNC2=O)=O)C)C)=O)ccc2c(c1)CCC2(C)C 60366,N1(C(C=NOC)=O)CCC2(CC1)OCCC2NC(C1CC1c1ccccc1)=O 60367,c1(C(N2C3C(NC(C=Cc4scc(C)n4)=O)CC(C3)C2)=O)cccc2c1CCO2 60368,c1(C(=O)NCCCC(C)NC(CC2(C=C)CCCCC2)=O)coc(S(N)(=O)=O)c1 60369,C1(CC)CCCCCCN1C(C1CC(NC(C2OCCC2(C)C)=O)C1)=O 60370,c1(C(N(CC(CNC(C(C)C#N)=O)O)C)=O)nn(C)c2ccccc2c1=O 60371,c1(CNC(C2CC(F)CN(C(c3ccc(I)c(Cl)c3)=O)C2)=O)cccc(F)c1Cl 60372,C(C(=O)N1CCCC(CN(C(=O)CCOCCN(C)C)C)C1)(C(C)C)OC 60373,CC(C)CCC(=O)NCC(=O)NC1CCC(NC(c2nc(C3CC3)cs2)=O)C1 60374,C1(OC)(CNC(=O)Cc2nnc(O)s2)CCN(C(=O)CC(C)C2CCCO2)C1 60375,c1(C(N2CCCC(NC(C(C)OCCC=C)=O)C2CC)=O)cnc2n1CCCC2 60376,c1(NC(N2C3CN(S(CC(=O)OCC)(=O)=O)CC32)=O)ccc2nc[nH]c2c1 60377,N1(C(c2cnc(CCC)s2)=O)CC(C)(C)CCC1CNC(C1CCCN1N=O)=O 60378,C(=O)(CS(C)(=O)=O)NCC1CC(N(C(=O)CC2CC=CCC2)C)C1 60379,N1(C(C(C)(C2CCC2)NC(=O)Cc2ccsc2)=O)CC2CC(O)CC2C1 60380,CN1N=C(CC(=O)NC2(C)CCN(Cc3ccncc3Cl)C2)CC1=O 60381,c1(C(C)(C)C)ccc(C(=O)NC2(CNC(c3ccoc3)=O)CCOC2)s1 60382,C1(C(=O)NC2CCN(C(C(c3cn(CC)nc3)=O)=O)CC2)CC2(CCC2OC)C1 60383,C1(NC(c2[nH]cc(CC)n2)=O)CCCN(C(c2cc[nH]c2C2CC2)=O)C1C 60384,CCCC(C)C(C)NCC1CC1C(=O)OC(C)(C)C 60385,C1(NC(C(CCC)CNC(=O)CCCN(C)C(C)=O)=O)C2CCCCCCC12 60386,Nc1cnc(C(=O)NC2CCC2NC(c2cccn2C2CCCC2)=O)cn1 60387,c1(C(N2CC3CC2C3C(N2CCC2(CO)CO)=O)=O)ccc2[nH]nc(Cl)c2c1 60388,c1(C(=O)NCCOC(CNC(c2cnc(CCC)s2)=O)(C)C)cnc(N)c(Cl)c1 60389,C1(CNC(c2c(C)snn2)=O)(OCCNC(C2CCC3(CC3)C2)=O)CCOCC1 60390,c1(C(C(=O)NCCC(=C)CNC(c2ccnc(OC)c2)=O)O)ccc(Cl)c(Cl)c1 60391,C(=O)(CCN(C(=O)COCC1CC1)C(C)C)N(CCOC)C 60392,N1(C(C)=O)CC(NC(C2CC2c2cccc(C(C)C)c2)=O)CC1(C)C 60393,C(=O)(CC(C(F)(F)F)n1ccnc1)NCCC(C)NC(c1ncc(F)cc1F)=O 60394,C=CCC(CNC(c1ccncc1Cl)=O)C(=O)N1CCC(CC(C)O)CC1 60395,c1(CSC)ncc(CNC(=O)NCCN2CCNC2=O)c(C)n1 60396,Cc1cn2ccc(C(=O)NC(CNC(=O)C(C)(C)N(C)C)C(C)C)cc2n1 60397,c1(C(=O)NC2C(CC(=O)NC(CC#C)CC)C(O)C2)nccnc1C 60398,c1(NC(C)C(=O)NCCOCCN(S(C)(=O)=O)C)cnn2ccn(C)c12 60399,c1ccc2c(N3CCC(OCC4CCCC4)CC3)nsc2c1 60400,C(c1ccsc1)=CC(=O)NCC=CC(=O)NCC1CC(=C2CC2)C1 60401,CC=C=CCCN=c1nc(N2CCN(C)CC(C)C2)c2ncccc2[nH]1 60402,c1(C(=O)NC2C(CNC(C3CC(=C)C3)=O)C2)cc2c(N(C)C)cccc2s1 60403,c1(C(N2CCC(c3nc(C)c(C)s3)CC2)=O)nc2ccsc2s1 60404,N1(C(c2c(CC)[nH]cc2)=O)CCCC(O)(CNC(C2(CO)CCOCC2)=O)CC1 60405,c1(CCC(=O)N(c2ncc(SCCO)s2)C(C)=O)ccc2ccccc2c1O 60406,c1(CC)nc(N2CCCC(CNC(c3cc(Cl)nc(Cl)c3)=O)C2)c(CC)c(Cl)n1 60407,C1(NC(c2ccc(C(C)F)cc2)=O)CCCC12CN(C(c1ccnc(S)c1)=O)C2 60408,c1(C(=O)NC2CC(NC(Cn3c(C)c(Cl)cn3)=O)C2)cc(O)cc(Cl)c1Cl 60409,N#CC1(C(=O)NCC2CC(C(=O)NC3(c4ccoc4)CC3)C2)CCC1 60410,c1(NC(c2nnnn2CCC2CC2)(C2CC=CC2)C)ccc(S(N)(=O)=O)c(F)c1 60411,CS(=O)(=O)CCCNC12CC(C(=O)NCc3cccc(C4(C#N)CC4)c3)(C1)C2 60412,N1(C(c2cc(C)sc2C)=O)CC(F)(F)CC1C(=O)NC1(C)CCCC1(C)C 60413,C1(CC(=O)NC2C3CC2N(C(c2coc(C4CCC4)n2)=O)C3)CCC=CCC1 60414,c1(N2CCCC(C=C)C2)nc(=NC2COCC2C2CC2)[nH]c2ncn(C)c12 60415,c1(C(=O)NC2C(CNC(c3cccc(C)c3Cl)=O)CCC2)cn2ncccc2n1 60416,N1(C(CN(C(COC)=O)C)=O)CCC2(CC1)C(NC(=O)CCSC)CS2(=O)=O 60417,C1(NC(c2ccc(OC)cc2)=O)CC2CCC(C1)N2C(=O)CCc1ccccc1 60418,c1(C(=O)NC2CN(C(C(C(C)C)OC)=O)CC2C)cn2cc(Br)sc2n1 60419,N1(C(Cc2cc(C)on2)=O)CCC(NC(=O)Cc2c(C)n[nH]c2C)C(CO)CC1 60420,S(=O)(=O)(c1ccc(Br)cc1NCCCn1c(C)ncc1)NCC1(CCCO)CC1 60421,CC(C)C(=O)C(=O)NC1CCC(CC(=O)N(C(CO)CO)C(C)C)CC1 60422,C1(C(=O)O)(NC(=O)C(F)(F)Br)CC(O)C12CCC2.N12CC(C1)C2=O 60423,C1(CCNC(C2(C)CC(F)C2)=O)CCCN(CC(=O)N)C1.c1(CN)ccccc1 60424,c1(CCC(=O)NC2(C(=O)Nc3ccc(C)cc3O)CC2)ccc2ccn(C)c2c1 60425,C1(CC(N2C(Cc3ccc(OC)cc3)CCC2)=O)CNC2(CC2)CO1 60426,c1(CC)ncc(C(=O)NC(C)CCNC(c2sc(=N)[nH]c2C2CC2)=O)cn1 60427,N1(C(C(C)O)=O)CCc2[nH]nc(CNC(=O)CCC3CCOC3)c2C1 60428,S(=O)(=O)(c1csc2ccccc12)NC1CN(C(c2nc(Cl)ccc2F)=O)CC1O 60429,C(=O)(CCC(C)C)NCC(CCOC)NC(=O)CCC1CCCCO1 60430,CC(C)C(CCC(=O)N1CC2CC3CC2C1C3)NC(=O)CC1OCCO1 60431,C(CS(=O)(=O)CC(=O)NCC1CC(C)N(C(=O)CCCC(C)O)C1)OC 60432,CC1(Cc2ccccc2C(F)(F)F)CCCN1N1CCCC2(CC1)NC(=O)NC2=O 60433,N1(C(CCCC)=O)CC2CC(CNC(c3cc(C(F)(F)F)ccc3Cl)=O)C2C1 60434,C12(NC(C(=O)NC3CC3)=O)CCC(CC1)N(C(c1ccncc1)=O)C2 60435,C1CC(=O)N1C.C1(NCC2CC2)CC(NC(=O)OC(C)(C)C)C1 60436,CC(C(=O)NCCOCCNC(=O)COC1CC=CC1)c1ccsc1 60437,N1(C(C(C=C)OC)=O)CC(C2CCCN(C(=O)CC3CC4CC4C3)C2)C1 60438,C1(CC(c2nnnn2CCCC2CC2)NC(C)C(=O)NO)CCC(C)(C)CC1 60439,c1(CC)cc(N(C(C2(C)CCC(=O)N2)=O)C(C)C)ncn1.C1CCN1 60440,C1(CN(C)C(c2cccc(O)c2)=O)CCCN(C(=O)CN2CCCC2CO)C1 60441,N1(C(C2CC3(CCOCC3)C2)=O)CC2(C1)CN(C(C1(CF)CCC1)=O)CC2CO 60442,c1(C(N2C(CC(=O)NCCc3ccccc3Cl)COCC2)=O)cccc(F)c1Cl 60443,n1(CC(=O)Nc2cccc(NC(C3CCC(=O)NC3=O)=O)c2)ncc2ccccc12 60444,CC1(NC(C2C=CC(NC(c3cc(O)cs3)=O)C2)=O)CC(F)C1 60445,N1(C(C2C(C)(CC)C2)=O)CCOC(CNC(=O)CCCCN2CCOCC2)C1 60446,C(=O)(C(C(C)CC)C1CCC1)NC(CCOCC)C(=O)NCc1ccc(CO)o1 60447,N1(CC)CCC(NC(=O)CN(C(=O)CCc2ccc(C)[nH]2)CC)C(C)C1 60448,c1(OC)csc(C(=O)NC(C)CC(C)NC(=O)CC2(OC)CCC2)c1 60449,c1(C(N2CCC(C)C2CNC(=O)CC2(C)CC2(Cl)Cl)=O)cc[nH]c2nccc1-2 60450,C1(NC(C2CC(O)(CNC(c3c(C)nc[nH]3)=O)C2)=O)CCCC(=O)N1C 60451,c1(C(N(CCN(C(c2cccc(OC)c2)=O)C(C)C)C)=O)ccc2c[nH]nc2n1 60452,N1(C(c2cc(OC)n[nH]2)=O)CCOC2(CCN(C(C3CCCC(F)C3)=O)C2)C1 60453,Cc1c(CCC(=O)N(N(C(C)CCC(C)C)Cc2cccs2)C)cccc1F 60454,c1(C(N(C)CC2N(C(CC(C(C)C)O)=O)CCC2)=O)ccn2ccnc2c1 60455,C1(C(=O)NCCC2(CNC(C(CSC)O)=O)CC2)CC(=O)N(c2nccs2)C1 60456,c1(C(C(C)NC(=O)NCc2cn(C)nc2-c2cccnc2)OC)ccccc1F 60457,c1(C(N2CCC(NC(C(F)=CC)=O)C(C)C2)=O)c(C)oc2ncnc(O)c12 60458,C1(NC(C(SC)SC)=O)C2CC(NC(C3CCN(C)C3C)=O)CC12 60459,c1(C(=O)NC(CCC)CNC(=O)C(C)=C(C)C)cc(Cl)nn1C 60460,C(=O)(C1CC(=O)Nc2ncccc21)NC(C)(C)CCCNC(c1ncccn1)=O 60461,c1(NC(CC)C(=O)NCC(C)(C)NC(=O)Cc2cncn2CC)cccc(C)c1 60462,c1(C(=O)NCCN(CCCCCC)C(c2coc(CO)c2)=O)ncc(N)cc1Cl 60463,c1(CCN(C2CCN(C(C3CC(F)(F)C3)=O)C2)C)cc(F)ccc1F 60464,C1(CNC(C2CCC(C)(C)O2)=O)CC(F)(F)CN1C(c1ccc(Cl)nn1)=O 60465,C(=O)(C(CN(C)C)NC(=O)CCC1CCCN1C)NC(C)C(=O)NCCF 60466,C(=O)(C(CC(C)C)OC)NCC(CC)N(C)C(C1COCCN1C)=O 60467,C1(C(=O)Nc2cccc(C)c2C#N)C2CCCC1CN(C(c1c(C)cc[nH]1)=O)C2 60468,Cc1cc(C(=O)NC2(CN(C)C(C3CC(OC(F)(F)F)C3)=O)CC2)c(C)c(C)c1 60469,c1(C(C)(C)C)cccc(C#CCN(CCO)Cc2cc(Cl)c(Br)cc2F)c1 60470,C1(NC(C2(OCC)CCC2)=O)CCN(CCCNC(=O)CC2C=CCC2)C1 60471,C1(C(N(C)CC2(NC(C=CCCC=C(C)C)=O)CC2)=O)Cc2cccnc2C1 60472,CCC(CNC(c1coc(N(c2ccccc2)C)n1)=O)CCl 60473,C1(C(=O)NCCN(C(CC2(C=C)CC2)=O)CCc2ccccc2)CN(C)CCO1 60474,CCCC(C(=O)N1CCC(C(C)(C)C(=O)NCCOC2CCCC2)C1)NC(N)=O 60475,CC(=O)CCCC(=O)N1CCN(C(C23CCCCC2C3)=O)CC1C 60476,c12ccc(F)c(c1)-c1c[nH]nc1C(=O)N2.CC(C)CCSCCC(C)C 60477,N1(CCCC(=O)NC(c2ccccc2Cl)CC)CCCC(C(C)NC(=O)CC)C1 60478,c1(CNC(C(C)OCCOC)=O)nocc1C(=O)N(C)Cc1cnn(C)c1 60479,c1(CC)cccnc1C(=O)NC1CCCC1NC(C1COC(=O)O1)=O 60480,c1(NC(=O)Nc2nc(C(N(C(C)=O)C3CC3)=O)cs2)c[nH]c2cccc(F)c12 60481,c1(C(CN2C(CNC)CC2)=O)cc(Br)ccc1C 60482,C1(CCCC)CN(C(c2n[nH]c(C)c2Br)=O)CCN1C(=O)CC(C)F 60483,C1(NC(C2(CC)CCCC2)=O)CCOC12CCN(C(C1CC=C(C)CC1)=O)CC2 60484,S(=O)(=O)(c1ccc(F)cc1F)N(C1CC2CC1CN2)C(c1cc(C(C)C)no1)=O 60485,c1(C(C)OCC)noc(CN(C)C(C2(C)CCCS2)=O)n1 60486,c1(N2CCC(OCCNC(Cc3nc(C)c(C)s3)=O)C2)ncnc2sccc12 60487,C1(C(=O)NC2CCC(NC(c3nc(Br)c[nH]3)=O)C2)CCC2(CCC2)C1 60488,CCC(C)C(C)(O)CNC(C1CCCC1NC(c1cncc(O)c1)=O)=O 60489,CC(N=c1[nH]c(N(C)CC2CCN(C)CC2)nc2c1SCC2)c1cc(Br)no1 60490,N1(C(C(CC(C)(C)NC(c2cn(CCC)nn2)=O)F)=O)CCC2(CC=CCO2)C1 60491,c1(C(=O)NCC2(C)CCCN(C(C3=CCCCC3C)=O)C2)cnc2ncnn2n1 60492,C(CN=c1c(C#N)c[nH]c2ccc(C)cc12)N(C(C1CCC(C)C1)=O)CC 60493,O=S(=O)(c1cnc(N2CCCC(OCCO)C2)c(Cl)c1)NCC1(CCCO)CC1 60494,c1(C(=O)NC2CCC(NC(CC(CC)OC)=O)CC2)ccc2c(c1)CCN(C)C2 60495,c1(C(N2CC(CNC(Cc3ccc(OC)cc3)=O)C2)=O)ccc(P(C)(C)=O)s1 60496,C1(CC)CN(Cc2ccccc2N(C)C)CCN1C(=O)Cc1ccsc1 60497,C1(C(=O)NCC(C2CC2)SC)CC2CN(C(=O)Cn3nnc(C)n3)CC2C1 60498,c1(OC(C)C)ccc(C(=O)NCC(CO)NC(c2ccccc2)=O)cc1 60499,CCCC(C)(C)CC(=O)NC(CCC(=O)N1CCC1C(N)=O)C(C)C 60500,C1(CC)(CNC(C2(NC(c3ccn(C4CC4)n3)=O)CC(O)C2)=O)CCOC1 60501,c1(C(=O)NCC2(C)CCC(NC(C3(C=C)CCC3)=O)CC2)cc(C)nc(Cl)c1N 60502,Cc1ccc(C(=O)NC2(CS(N)(=O)=O)CC2)nc1C 60503,C(=O)(C(C)(CSC)NC(=O)C=Cc1ccoc1)NC(C#C)C 60504,C1(NC(C(=O)NCC2(CC)CC2)=O)CC(C)(C)C(C)(C)C1 60505,C(C(C)(C)CNC(c1ncoc1C1CCC1)=O)N(C)C(c1coc(Br)n1)=O 60506,CC1C2CCCCC2CN1C(=O)C(CC1CC1)NC(C1CCC(=O)O1)=O 60507,c1(CSCCC(=O)NCCC2CCN(C(CC(=O)OCC)=O)C2)ccc(F)cc1 60508,N1(C(c2ccc(C#C)cc2OC)=O)CCC2C(CCCN2C(=O)CC(C)(C)C)C1 60509,C=CC1(C(=O)N(C)Cc2ncn(C)n2)CCN(C(=O)CCc2cccs2)C1 60510,CC1(C#CC(=O)NC2CC3CCC2N3C(c2cc(Cl)c(Cl)s2)=O)CC1 60511,C1(C(=O)NC2CCN(C(C)=O)CC2)CCC2(CN(C(=O)C(O)C(C)C)C2)O1 60512,C1(OC)CN(C(c2cccc(Br)n2)=O)C2(CCC2)C1.C123COCC1CN(C2)C3=O 60513,c1(C(NOC(C(C(=O)N2C(C(=O)OCC)CCC2)(C)C)=O)=O)nccc(Cl)c1C 60514,CCC(C)CC(=O)NC1CCCC1NC(c1cccc(N2CCCC2=O)c1)=O 60515,CC(CC(=O)NCCCC1CCOCC1)NC(=O)COc1cnn(C)c1 60516,C=CCC(CC(=O)N1CCC(COC)CC1)NC(=O)C(CC=C)OC 60517,C1(F)(C(=O)NC(COC)C2CC2)CCCN(C(=O)CC2CC(C)(C)CO2)C1 60518,CC(CC(=O)NC(C1(O)CCCCC1)C(N1CC=CC(O)C1)=O)C(F)(F)F 60519,C(CCCCC(=O)NCc1nccn1C)N(C)C(C1(F)CCOCC1)=O 60520,c1(C(=O)NCC2CCN2S(=O)(=O)C2CC2)nc(C(F)(F)F)ccc1Cl 60521,C1(C(=O)NCCCC(C)NC(C2CCC3(CC3)C2)=O)C2CC3C(C2)C13 60522,CC1(C)CCCN(C(=O)CCCC2CCCO2)C1C(=O)NC1CC=CCC1 60523,C1(NC(C(C=C=C)C)=O)CCCCN(C(c2cnc(OC)s2)=O)C1 60524,CC1(NC(=O)CC2CCCC23CC3)CCN(C(=O)Cn2nnc(=N)[nH]2)CC1 60525,CC#CCCCC(C)N(c1ccc(C(C)C)cc1)CCC#N 60526,c1(OC)ccc(F)c(C(=O)N(CC(C)(C)CNC(C2CCCC2(C)C)=O)C)c1N 60527,C(C(C)C(C)C(=O)N1CCCC1CN(C(=O)CCNC(c1ccco1)=O)C)OC 60528,CC1CC(C(N2CCCC2CCc2ccccc2)=O)CCO1 60529,C12(CNC(c3ccoc3)=O)CCCC1N(C(c1ncnc3sccc13)=O)CCC2 60530,C1(NC(CC2CCC(=O)NC2)=O)CCCCN(C(=O)C(c2cccc(Cl)c2)C)C1 60531,C1(NC(CC2(OC)CCCCC2)=O)CC(C)CN(C(=O)CCc2csc(=N)[nH]2)C1 60532,C1(CCC)(NC(=O)CCc2cnoc2)CCN(C(c2ccc([N+](=O)[O-])s2)=O)CC1 60533,C1(C(=O)NC(CNC(CCc2n(C)ccn2)=O)(C)C)CCC(F)(F)CC1 60534,N1(C(c2cn(C(C)(C)C)nn2)=O)CCN(CCCNC(c2n[nH]cc2Cl)=O)CC1 60535,CCC(C)(CN(C(=O)CN1CC2CC2C1)CCOC)C(=O)N1OC2CCC1CC2 60536,C#CC1CCN(C(C2COCCN2C(=O)C(C)=C2CCCC2)=O)CC1 60537,CC1(C(=O)NC2CN(C(c3cccc[n+]3[O-])=O)CC2CO)CCC(O)CC1 60538,c1(C(=O)NCC2CCCCN2C(=O)C2=NOCC2)n[nH]c2cc(Br)ccc12 60539,c1(C(=O)NC2CC3CN(c4ncc(C#N)nc4)CC32)nnn2c1COCC2 60540,C12(NC(CC(COC)NC(=O)Cn3nc(C)nc3C)=O)CCC(C1)OC2C 60541,C1(NC(CNC(CC)=O)=O)(CC)CCN(C(C2CC2Cl)=O)CC1 60542,C=Cc1cccc(CN2CCCC(C(N3CCCC3c3ccccc3)=O)C2)c1 60543,C1(NC(C(C)(CO)OC)=O)CN(C(c2cc(C)cc(Br)c2)=O)CC1N=[N+]=[N-] 60544,c1(CNC(C(=O)OCC)CC2CCC2)ccc(OC)c(Br)c1 60545,CCCCC(O)C(=O)NCC(CC1CC1)C(=O)NCCN1CCC(C)(C)C1 60546,c1(C(=O)NCCN(C(C(c2cnn(C)c2)OC)=O)C)nc(C)n2ccccc12 60547,CC(CC(C)(C)C)C(=O)NCC(C)(CO)NC(=O)CCCn1cncn1 60548,c1(C(N2CC(F)(F)CC2CCNC(=O)C(F)(F)CC2CC2)=O)cccc(=S)n1O 60549,c1(OC)ccccc1C(N1CCCC(CCNC(=O)CC(O)CN(C)C)C1)=O 60550,Nc1cccnc1S(=O)(=O)NC1CC(=O)NC1=O 60551,c1(C(=O)NC2C3CN(C(C(C(C)(C)C)SC)=O)CC32)cccc2cc(F)ccc12 60552,c1(C(=O)NCC(C)N(C(c2c(C)c(F)ccc2)=O)C)cc(N)c(Br)c(F)c1 60553,N1(C(C2C(SC)CCC2)=O)CC2CCC(CNC(C3CCCN(C)C3)=O)(C2)C1 60554,C=C(C)C1OCCCC1C(N1CCC2(C1)CN(C(c1cc(O)ncn1)=O)C2)=O 60555,C1(NC(C=C(C)c2ccsc2)=O)CCC2(CC1)CN(C(=O)C(C)S(C)(=O)=O)C2 60556,CN1CCNC(=O)C12CCCN(Cc1cnc3ccc(Cl)cn13)C2 60557,C1(C(=O)NCC2(CO)CCCC2)CC2(CCC2)CN1C(c1ccnc(O)c1F)=O 60558,C(c1ccc(C)cc1)=CCC(N1CC2C(CNC(C(CCC)OC)=O)(C2)C1)=O 60559,C1(NC(=O)CC2CC3C=CC2C3)CC2CC1N(C(C1CCCCC1)=O)C2 60560,c1(C(N2C(C(N3CCCC(CCC)C3)=O)CNC(=O)C2)=O)ccc2[nH]ccc2n1 60561,C1(OC)CCC2(C(=O)N(CC(C)C(=O)NC(c3cnc[nH]3)C)C)CC12 60562,Cc1cc(Br)cnc1C(N1CCC(NC(=O)CN2CC=CC2)C1C1CC1)=O 60563,C(CN=c1nc2c(ncn2C)c(NC2CCN(C)C(C)C2)[nH]1)NCCOCCC 60564,c1(C(=O)NCC(CC(F)(F)F)NC(=O)C(O)C2CCC2)cc2ccc(F)cc2[nH]1 60565,C1(NC(c2c(CC)nc[nH]2)=O)CC2(CCN(C(=O)C(C)CCCOC)C2)C1 60566,C(CCC(O)C(=O)NC1CCOC(C)(C)C1)NC(C(CCC)NC(C)=O)=O 60567,N1(C(CCCc2onc(C)n2)=O)CCC2(NC(c3cnc(C(C)C)[nH]3)=O)CC2C1 60568,N1(C(CCCCN(C)C)=O)CC2CCN(C(c3snc(Cl)c3Cl)=O)CC2C1 60569,Cc1cnc(C)c(C(=O)NCC(C)CNC(=O)CSc2ccc(F)cc2F)c1 60570,c1(C(=O)NC2C(NC(C(CC)(C)C#N)=O)CC2)cc2c(cc1F)OCC(=O)N2 60571,N1(C(C)=O)CCCC(CC(=O)NC(C)(CNC(=O)C2=COCC2)C(C)C)C1 60572,c1(SC)cc(C)c(CNC(=O)CSC2(C(C)(C)C)CCN(C(C3(O)CC3)=O)C2)s1 60573,C(=O)(C(C)C(C)(C)C)NCc1cc(C(=O)NCC(C#C)C(C)C)sc1 60574,c1(C(N(C)CCOCC2(O)CCOC2)=O)ncc(C(C)(C)O)cn1 60575,c1(OC)cnc(Cl)nc1N1CCCC(C(C)NC(c2cnn(C)c2C2CC2)=O)C1 60576,C1(NC(C(F)=C(C)C)=O)COC2(CCCN(C(=O)CC3(CO)CCOCC3)C2)C1 60577,c1(-c2cc(COC)on2)nc(C2CCCCC2)nn1CCS(C)(=O)=O 60578,c1(OCC)ccc(-c2ncc(C(=O)NCCN(C)CCn3cncn3)s2)cc1 60579,Cc1ncnc(C)c1C(=O)N(CCCNC(=O)C1=NOC(C)C1)C 60580,C1(C(=O)NCC2OCCN(C(COCCCN(C)C)=O)C2)(OC)CCS(=O)(=O)C1 60581,c1(CC)cc(Nc2ccccc2CN2CCOC(CC(=O)OC)C2)nc(C#N)c1 60582,N1(C(COCC)=O)CCC(C(=O)NC2(CO)CC(F)(F)C2)C1CC 60583,N1(C(C2CC(OC)C2)=O)CC2OCCN(C(c3cc4c(cc3N)CCC4)=O)C2C1 60584,N1(C(c2csc(CO)n2)=O)CCCC2C1CCCN2C(c1cc(=O)cc(Cl)[nH]1)=O 60585,C1(NC(CCN(C)CC)=O)CCC2(CCN(C(C3(C)CC(F)(F)C3)=O)C2)C1 60586,C(C(C(=O)NC(c1cnn(CC)c1)C)NC(C1C=C(C)CS1)=O)OCC 60587,c1(C(=O)OCC)cncc(CC2CCCC2C(F)F)c1.c12csc(n1)NC2=O 60588,C1(CNC(CCCOC)=O)CC2CN(C(=O)C(C)(COC)CC)CC12 60589,c1(OC)ccc(C=CC(=O)NCCCCCNC(=O)C(C)(C)C2CC2)cc1 60590,C(CC)(CC)(CCNC(=O)CCCCC#N)NC(c1ncc(CC)nc1)=O 60591,c1(C(N(CCN(C(C)C)C(C2CCC(C)S2)=O)C)=O)c[nH]c2c(C#N)cccc12 60592,C12(NC(C(Cc3c(C)n[nH]c3C)C)=O)CCCC(CN(C(=O)C#CC3CC3)C1)C2 60593,CCC(C)(F)C(=O)NCCC1CCC(NC(c2ccccc2NC(N)=O)=O)C1 60594,C#CCC(CC(F)F)C(=O)NC1CC=C(C(=O)NC2(CO)CC(F)(F)C2)C1 60595,C1(CC(=O)NCC2CCC(=O)O2)C2CCCC2N1C(=O)CC1CCOC1=O 60596,c1(C(=O)NCCC(C)(C)NC(Cc2cccc(OC)c2)=O)ncc(F)c(OC)n1 60597,Cc1ccc2[nH]c(C)c(CC(N3CCC(NCC(C)C)CC3C)=O)c2c1 60598,N1(C(c2ccc(C(C)C)s2)=O)CCC(C)(CNC(=O)CC2C(C)C2(F)F)C1 60599,c1(C(=O)NC2CN(C(C(CC=C)C(C)C)=O)C2)[nH]c2c(F)cc(F)cc2c1C 60600,CCC(C)C(O)C(C)C(=O)N1CCCC(CC(N2CCC3(CCOC3)C2)=O)CC1 60601,C1(N(C(CCN(C)CC)=O)CC)CN(C(c2snc(C)c2N)=O)CC1O 60602,C1(C(=O)NCCNC(C2CC(C)(CC)C2)=O)CCC(=O)N(c2cnn(C)c2)C1 60603,C1(NC(C(C=C)CC)=O)CN(C(=O)CCC(C)OCC)CC1C1CC1 60604,Cc1c(C(=O)NCC2CCCCC2NC(=O)COc2cnn(C)c2)cccc1O 60605,c1(CC(=O)N(C2(CC(=O)NCCn3ccnc3)CC2)C)cncnc1 60606,N1(C(C2CCC(OC)CC2)=O)CCN(C(c2ncn3c2CCC3)=O)C2CCCC12 60607,N1(C(CC(c2ccc(C)cc2)C)=O)CC2CC(CNC(=O)CC(=O)N(C)C)C2C1 60608,N1(C(C(C)O)=O)CCC2CN(C(c3ccncc3N)=O)CC12 60609,c1(CNC(CC2CCC(C)C2)=O)ccc(-n2cc(-c3ccc(Cl)cc3)nn2)cc1 60610,C(C(O)CN=c1[nH]c(Cl)ncc1[N+](=O)[O-])NC(c1ccc(CC)nc1)=O 60611,C=CCC(C)(C)CSc1ccc(NC(C2(CO)CCCC2)=O)cc1 60612,N1(C(C2CC(C)C2)=O)CC(NC(=O)Cn2nnc3ccccc23)C2(CCCC2)C1 60613,C(c1ccc(Cl)cc1F)=CC(=O)NC1CC(F)(CNC(C23CC(C)C2C3)=O)C1 60614,N1(C(CC2CC(C)(O)C2)=O)CC(CNC(c2cccc(F)c2Cl)=O)CC12CCC2 60615,N1(C(C2(CC)CCC2)=O)CCCC1C=CC(=O)NCC1(O)CCN(C)C1 60616,c1(C(=O)NC2C(NC(CC3CCC(C)(C)C3)=O)CC2)ccc2nc(O)[nH]c2n1 60617,c1(C(N2CCC(O)(C(C)NC(c3ccncn3)=O)C2)=O)nccc2n[nH]cc12 60618,c1(CC(=O)NCC2CCC(NC(c3cnc(OC)s3)=O)C2)cc(C)ccc1OC 60619,N1(C(C(CCC)C)=O)CC2(C1)CN(C(C1(C)CCCCO1)=O)CC2CO 60620,C1(NC(CCNC(=O)NC)=O)CCC(O)CN(C(c2cn(C)c(O)n2)=O)C1 60621,N1(C(CC2CC(=C)C2)=O)CCN(C(c2ccc(N)cc2OCC)=O)CC(C)(C)C1 60622,Cc1nc(O)c2c(n1)CCN(C(c1ccsc1S(C)(=O)=O)=O)C2 60623,N1(C(C(N2CCCCC2)C)=O)CCOC(CCCNC(=O)CP(C)(C)=O)C1 60624,C(=O)(C(=O)N=S(C)(C)=O)NC1C(C)CN(C(c2ccc([N+](=O)[O-])s2)=O)CC1 60625,C1(O)(C(C)NC(C)=O)CCN(C(c2ccccc2-c2cc[nH]n2)=O)CC1 60626,c1(C(=O)NC(CN(C(=O)CC2CCC(=O)NC2=O)C)(C)C)ccc(F)cc1N 60627,CN1CC=C(CC(=O)NC(C)(CNC(C23CCCC2OCC3)=O)C2CCC2)CC1 60628,c1(C(N(CC2CCN(C(C=CC(=O)OCC)=O)C2)CC)=O)cn2c(n1)SCC2 60629,N1(C(C)C(N2CCCC2c2ccc(Cl)cc2)=O)CCCCC1C#N 60630,C1(CCC)CCCN(C(C2(C(C)C)CCN(C(c3cc(C)c[nH]3)=O)C2)=O)CC1 60631,C(N=c1nc(C)[nH]s1)C1C(NC(C(CC)N2CCCC2=O)=O)CCC1 60632,N1(C(CCC(=O)NCC)=O)CCC(CNC(c2ccc(Cl)cc2F)=O)C12CC2 60633,c1(C(=O)NC2C(CNC(CC(=C)Br)=O)C2)ccc(C)c(CO)c1 60634,c1(C(=O)NCC(CC)NC(c2n[nH]c(C)c2O)=O)cccc(N=S(C)(C)=O)c1 60635,N1(C(c2n[nH]c(CC)c2C)=O)CC(C)N(C(c2ccc(F)cn2)=O)CC1C 60636,C1(C(=O)NCCCNC(c2scc(OC)c2OC)=O)CC(S(C)(=O)=O)C1 60637,C1(CCNC(=O)C=CC2CCOC2)(OC)CN(C(=O)CCOCCOC)C1 60638,c1(CC)c(C(N2CCCC(N(C(=O)CN(C)C(C)=O)C)C2)=O)oc2ccccc12 60639,c1(C(=O)NCCC2(O)CCCN(C(C3C(C=C)C3)=O)C2)cc2ccccn2c1 60640,c1(CC)[nH]nc(C(N2CCCC2CCC2CCCCN2C(=O)CNC=O)=O)c1C 60641,C1(CCC)CN(C(c2cc(C)c(C)s2)=O)CC1C(N1CCCC1CN(C)C)=O 60642,CC(c1ccsc1)=CC(=O)NCC(CC(C)C)NC(=O)CC12CC(C1)C2 60643,N1(C(C2C(C=C)C2)=O)C(CNC(=O)Cc2ccc(OC)c(F)c2)CC2CCCC12 60644,CON1CCC(C(=O)NC(C(C)NC(c2ccc(N(C)C)cc2)=O)C(C)C)CC1 60645,Cc1ccnc(O)c1C(=O)N(CC(N1CCN(C(C2CCCOC2)=O)CC1)=O)C 60646,C1(NC(C2(C)CCN(C)C2)=O)CN(C(c2cn3c(n2)SCC3)=O)C(C)(C)C1 60647,n1(CC(C)C(=O)NC2CCSC23CN(C(=O)C(Cl)=CCl)C3)cnc2ccccc12 60648,C1(c2cn(CCC(=O)Nc3cccc(NCC4CC4)c3)nn2)CC2CCC1CC2 60649,C1(CNC(CCC=C=C)=O)CN(C(c2cnc(C)[nH]c2=N)=O)C2(CCC2)C1 60650,Cc1nn(CC(N2CCC(NC(C3C=CCC3)=O)C(C)C2)=O)c2ncccc12 60651,c1(C(=O)NCCNC(C2CCC(=O)NC2)=O)coc2c(F)c(Cl)ccc12 60652,c1(C(=O)NCC2(C)CCCN2C(C2C3CCC23)=O)ccc(F)c2cccnc12 60653,c1(CNC(C2(CC=C)CC2)=O)cnn2c1CN(c1nnc(C)c(C)c1C#N)CC2 60654,C1(NC(CSCCOC)=O)CCCC(NC(=O)Cc2n[nH]c(C)n2)C1 60655,n1(CC)ncc(C(=O)NC(CNC(c2csc(C)c2C)=O)CC)c1Br 60656,N1(C(C(C)NC(COC)=O)=O)CCN(C)CC1CNC(c1scnc1C)=O 60657,Cc1ccc(F)cc1C1(C(=O)NCC(C)CNC(C23CCCC(C2)OC3)=O)CC1 60658,C1(C(=O)NC2(CCC)CCC2)CCN(C(C2C3CCC(C3)C2C)=O)C12CC2 60659,C(=O)(C(C#N)C(C)(C)C)NCC=CC(=O)NCC(CC(C)(C)CO)=O 60660,CS(=O)CCC(O)C(=O)NCCCNC(c1cc(O)cc(Cl)c1Cl)=O 60661,N1(C(CCC(C)(C)OC)=O)CCC2CCCC12CNC(C1(C)CC=CC1)=O 60662,C1(C(N2CCN(C(CN(C(C3CC(OC)C3)=O)C)=O)CC2)=O)CC(F)C(=O)N1C 60663,Cc1cnc(C)c(C(=O)NC2(C)CCN(C(=O)CCC3CCCN(C)C3)C2)c1 60664,c1(C(N(C2CCN(C(C(CCC)(C)C)=O)C2)C)=O)cn2cc(C)sc2n1 60665,CC1=C(C(=O)NC2CC(C(F)F)(NC(C34CSCC3C4)=O)C2)CCO1 60666,N1(C(c2c(C)ccnc2O)=O)CC2OCC(NC(c3coc(Cl)n3)=O)C2C1 60667,CCC(COC)C(=O)N1CC(OCCC(=O)NCCC(C)SC)C1 60668,C(=O)(CC(CC1CC1)NC(=O)C(C1CCCC1)OC)NC(CCC)c1nn[nH]n1 60669,N12CC(Cc3cc(OC)ccc31)C2.c1(OCC)cc(C(C)(C)C)ccc1SCC 60670,c1(C(N2CCCC(CNC(C3CCC4CC34)=O)C2)=O)cc(Cl)cc2c1CCC2 60671,N1(C(c2cc(SC)oc2)=O)CCC(C)(CNc2cnc(F)cn2)C1 60672,c1(C(=O)NC2(C)CN(C(=O)Cn3[nH]cnc3=N)C2)cc(=NS(C)(=O)=O)cc[nH]1 60673,Cc1nc(-c2ccsc2)ccc1-c1nc(-c2ccco2)nn1C1CCC(C)(C)C1 60674,N1(C(COC(C)C)=O)CCCCC(C(=O)Nc2cncnc2O)C1 60675,N1(C(C2ON=C(C)C2)=O)CCC(C)C1CNC(c1ccnn1C(C)C)=O 60676,c1(C(=O)NCC(C)(C2CCC2)NC(C(CC#C)O)=O)cc([N+](=O)[O-])n[nH]1 60677,C1(NC(C2CCCN(CCC)C2)=O)CCN(C(C2(CCF)CC2)=O)C12CCCC2 60678,N1(C(CCC)=O)CC(NC(c2cc(F)cc3nccnc23)=O)C2CCCCC12 60679,C12(CNC(CN(C)CC)=O)CCCC1CN(C(C13CCC(CC1)CC3)=O)C2 60680,N1(C(C(c2cccc(C)c2)=O)=O)CCC(CNC(C2CN(C)C(=O)N2)=O)C12CC2 60681,Cc1nnc(COCC(=O)NC(C)C(CO)NC(C2CCCOC2)=O)s1 60682,C1(N(C)C)(CNC(=O)C(CC2CCCC2)NC(C2(O)CCOC2)=O)CCCC1 60683,C1(SC)CN(C(c2ccc(F)cn2)=O)CC1n1cc(CCCC(C)=O)nn1 60684,N1(C(C(C)N(C)C)=O)CCC(C(C)(C)C)CC1CNC(=O)CCc1ccc[nH]1 60685,c1(OC)c(Cl)ccc(Cl)c1SCc1cnc(C)o1 60686,CCC(CC(=O)NC1CCCCCC1C(=O)N(C1CCCC1O)C)C(C)C 60687,C1(S(C)(=O)=O)(C(=O)NC2CCN(C(c3cnc(CCC)s3)=O)C2C)CCOCC1 60688,c1(C(c2n(CC=C)nnn2)NC2(CO)CC2C(F)(F)F)ccc(F)c(Cl)c1F 60689,C12(C(=O)NC(CCC)CCCNC(=O)CP(C)(C)=O)CC1COC21CCC1 60690,C1(C)(C(N2C(CNC(CC3ON=C(C)C3)=O)CCC2)=O)CS(=O)(=O)C1 60691,N1(C(c2cncc(CC)c2)=O)CC(CO)C2(C1)CN(C(c1coc(Cl)n1)=O)C2 60692,O=C(C1=CCSC1)NCC(c1ccccc1)CNC(c1cccnc1C1CC1)=O 60693,C1(C(=O)NC(c2nnc(C)o2)C)(CC)CCN(C(=O)Cc2cccc(C)n2)CC1 60694,n1(C(C)C)cnc2c(NCC3CC4C=CC3O4)[nH]c(=NC3CC(C)(CO)C3)nc12 60695,C1(C2(O)CCCOC2)(C(=O)Nc2ccc(SCCN3CCCC3)cc2)CC1 60696,C(=O)(C(CC1CCCC1)NC(=O)COC1CCCOC1)NCCSCC(=O)OC 60697,CC1(C)CC(NC(c2cc(CO)ccn2)=O)CN1C(C1CC12CCSCC2)=O 60698,CC1CCS(=N)(=O)CCN1C(=O)C(C(C)(C)C)n1cc(C2CCC2)nn1 60699,C(C)(CNC(c1ncccc1Cl)=O)(CC(C)C)NC(C(CC)OC)=O 60700,C1(NC(c2n[nH]c3c2CCC3)=O)COC2C(NC(C3CCCOC3)=O)COC12 60701,N1(C(C2CC(CCC)C2)=O)CCC(C(=O)NC2(CC(C)(C)C)CC2)C1C 60702,N1(C(C(n2c(C)ccn2)C)=O)CC(F)(F)CC1C(=O)N(C)CC1COCCO1 60703,C1(N(CCOC)Cc2ccnc(Cl)c2)CCN(C(=O)C(C)C2CCOC2)CC1 60704,c1(SCC(=O)NC2C(CNC(C3(CCC)CC3)=O)C2)ccccc1F 60705,N1(CC2(C)CCC(=O)N2)CC(=O)N(CC(c2ccc(Cl)cc2)(F)F)C1=O 60706,C1(C(N2CCN(C(CC)=O)CC2C)=O)CN2CCCN1CC2 60707,N1(C(c2ccc(F)c(F)c2)=O)CC(C(N2CCC=C(Cl)C2)=O)C(C2CC2)C1 60708,N1(C(c2cn(CC)nc2)=O)CCCC(N(C)C(c2cc(CO)[nH]n2)=O)CC1 60709,n1(CC(F)F)nnnc1C(CCc1ccccn1)NCC1(CC2CCC2)CC1 60710,CC(CCCNC(=O)CCc1ccncn1)NC(=O)C(C)n1cnnn1 60711,C1(NC(c2cc(C)nnc2O)=O)CS(=O)(=O)C2CN(C(c3cn(C)cn3)=O)CC12 60712,c1(N(CCOCC=C)C)nc(=NC(C)c2ccc(F)c(Cl)c2)[nH]c2c1CSC2 60713,C1(C(=O)NC23C(CN(C(C(C)(C)OC(C)C)=O)C2)C3)CCOC(=O)CC1 60714,O=S1CCC(Nc2ccc(N3CCNCC3)c(F)c2)c2ccccc21 60715,c1(C(N(C)CC2CN(C(=O)CC(C)(O)C3CC3)CCO2)=O)cc(O)nc(O)n1 60716,C1(CCC2N(C(c3c(OC)ocn3)=O)CCC2)CCCCN1C(C)=O 60717,Cc1ccc(C=CC(N2CCC(NC(=O)C(C)Oc3cccc(Cl)c3)C2)=O)cn1 60718,N1(C(C2CC=C(C)CC2)=O)CCCC2(NC(c3ccc(Cl)nc3Cl)=O)CC2C1 60719,Cc1ccc(OCCCC(=O)N(C)CCNC(=O)C(C)N2CC(C)C2)cc1 60720,c1(C(=O)NCCN(C(=O)CCC(C)OCC)CCC)c[nH]c2c(CC)cccc12 60721,c1(C(N2CC(NC(C=NOC)=O)C2)=O)ccc(CC#N)cc1 60722,CC1(C)CC(CC(=O)NCC2(Nc3ncccn3)COC2)CO1 60723,N1(CC(=O)NCC(CCCC)NC(=O)Cc2occc2C)C(=O)CN(C)C1=O 60724,CCCCCCN(C(=O)Cn1cccn1)CCN(C(C1CCCC1C)=O)CC 60725,Cc1cc(NC(c2ccc(S(C)(=O)=O)s2)c2nnnn2C(C)(C)C)cc(C)c1F 60726,c1(C(C)C)sc(Cl)nc1C(=O)NCC(C)(O)CNC(C1(C(C)C)COC1)=O 60727,C1(C(=O)NC(CCNC(C(c2ccc(C)cc2)=O)=O)C)CC12CCSCC2 60728,c1(C(=O)NC2CC3CC(NC(C(F)=CC)=O)C3C2)c[nH]c2ccc(Cl)cc12 60729,c1(C(=O)NC(CNC(CCC2OCC(C)(C)C2)=O)C2CC2)cc(Cl)ccc1Cl 60730,c1(C(=O)NCC2CCN2C(c2cnco2)=O)cnn(CC2CCCCO2)c1 60731,C(CCC(=O)NC1(C(=O)NCC(c2cccs2)C)CCC1)NC(C)=O 60732,C(=O)(C#CC1(C)CC1)N(C)CC1CCCN1C(c1cn(C)c(C(F)F)n1)=O 60733,CCCCCC(C)CC(=O)N1CCC(C)C(CNC(c2sccc2C(C)C)=O)C1 60734,Cc1cc(C(N2CCCCC2CC(=O)NCc2noc(C3CC3)n2)=O)sc1C 60735,c1(C(C)(C(=O)NCC2CC(C(F)(F)F)CO2)N(C)C)ccc(Br)cn1 60736,c1(CCCC(=O)NC2C(OC)CN(C(c3cnoc3C)=O)C2)ccc(F)c(F)c1 60737,c1(C(N2CC(NC(=O)CCC3CC3)CC(C)C2)=O)ccc2nc3n(c2c1)CCC3 60738,c1(CNC(c2n(CC)nc(C)c2)=O)ccc(CNC(=O)C(C)NC(C)=O)cc1F 60739,CC1=C(C)CC(C(=O)N(C2(CC(N3CCCC(C)C3CO)=O)CC2)C)CC1 60740,C1(CNC(CN2CCC(CCNC)C2)=O)CCC(=O)N1C.C1(O)CCC1 60741,C1(C)(NC(C(c2cccnc2)NC(C(C)=CC(C)(C)C)=O)=O)CCSC1 60742,CCC(F)(F)CC(=O)N1CCCC(C2CCCCN2C(C23CSCC2C3)=O)C1 60743,C1(C(N(CCCC)CC(N)=O)=O)CC2CN(C(c3cc4occc4[nH]3)=O)CC2C1 60744,N1(C(C2(C)CC(C)C2)=O)CCC(NC(=O)C=CSc2nc[nH]n2)C(O)C1 60745,CC1(C)C(CC(N2CCOC3(CC3)C2)=O)CCN1C(=O)Cn1cnnc1 60746,C1(CC)CN(C(c2cnc(Cl)cc2I)=O)CCN1Cc1ccnc(OC)c1 60747,c1(C(N2C(CNC(c3ccnc(S)c3)=O)CCCC2)=O)cc2nc[nH]c2cc1F 60748,CC1(CNC(C2C=CCN(C(c3nc(Cl)cs3)=O)C2)=O)CC2CCC1C2 60749,N1(C(=O)Nc2nc(Br)cs2)CCc2ncncc2C1 60750,c1(C(C)(F)F)cccc(C(=O)NC2CC2NC(=O)CC2C=CS(=O)(=O)C2)c1 60751,N1(C(c2cc(C)c(C)[nH]2)=O)CC=C(CC(=O)NCc2cccc(F)c2)CC1 60752,N1(C(C2CC23CC3)=O)CCN(C(=O)C(F)CC2CC2)C2(CC2)C1 60753,c1(CC(=O)NC2CCN(C(C=C(C)C3CC3)=O)C2C)cc(C(F)(F)F)c(O)nn1 60754,C(CCCCC(=O)N1CC(CC(=O)NCC2(C)CC=CCC2)(OC)C1)=CC 60755,N1(c2nccc(OCC)n2)CCC(C)C(NC(c2cnn(C)c2C#N)=O)C1C 60756,N1(C(=O)C=CCO)CCOC2(C1)CN(Cc1ccc(Cl)cc1O)C2 60757,Cn1cc2c(n1)CCCC2C(=O)N1CCCCC1C1(NC(=O)CC#N)CC1 60758,C1(C(N(CCCN(C)C)CCNC(C2CC23CCC3)=O)=O)CC2(C1)CC(F)C2 60759,C1(CN(C)C(c2ccnc(C3CC3)c2)=O)CCCCN1C(c1cccn1C)=O 60760,C1(NC(C(C)Cc2ccccn2)=O)CC2CC1N(C(=O)Cc1csnn1)C2 60761,N1(C(CSCCCC)=O)CC2CCCCC2(NC(=O)CCCC(=O)N(C)C)C1 60762,CCCC(C(O)C(=O)NC1CCN(C2CC2)C1)NC(C1(n2cccc2)CC1)=O 60763,c1(C(c2noc(-c3cccc(F)n3)n2)(C)C)ccc(S(C)(=O)=O)cc1 60764,C(C1c2ccccc2CN1C(C1C2(CC2)C12CC2)=O)NC(C(C)OCCCC)=O 60765,N(C1CCCn2ncnc21)C(C(C)N(C(=O)CC(C)C(F)(F)F)CCC)=O 60766,Cc1nc(C(=O)NC2CC(NC(C3CCCN3C3CCCCC3)=O)C2)cc(O)n1 60767,C=CC(CC)CC(=O)NC1C2CC1N(C(c1cc(COC)oc1C)=O)C2 60768,C1(NC(c2cc[n+]([O-])cc2)=O)CCCC12CN(c1nc(Cl)ncc1Br)C2 60769,C1(C)(C(=O)NCC(C)(C)OCCNC(c2cc(Br)no2)=O)C=CCCC1 60770,N1(C(C(=O)NC(C)C)=O)CCC2(CCN(C(c3cccnc3NC(C)C)=O)C2)C1 60771,c1(C(=O)Nc2ncc(Br)cc2I)cc2c(s1)CCN(Cc1cc(Cl)cc(I)c1)C2 60772,CON1CCC(C(=O)NC2CC(C)N(C3CC3)C2)CC1.c12csc(c1)CNC2=O 60773,C1(N(C(C(C)=C2CC2)=O)C)CC2CCC(C1)N2C(=O)COc1ccsn1 60774,C1(CC(C)NC(c2ccc(N)cn2)=O)CCN(C(=O)Cc2cncs2)CC1 60775,CC(C)(C)C(=O)C(=O)N1CCCOC(CNC(=O)CC2CCNC(=O)C2)C1 60776,Cc1c(C(C)OC(=O)N(C)C)cnc2ccnn12 60777,c1(C(=O)NCC(C)N(C(=O)C(C)CF)CC)ccccc1NC(N)=O 60778,c1(OC)cccc(-c2nc(C(=O)Nc3c[nH]nc3C#N)cs2)c1OC 60779,c1(CC(N2CC3C(C(N4CCC(CC)C4)=O)(C3)C2)=O)cccc(C#N)c1 60780,N1(C(C2CCN2CC2CCC(F)C2)=O)CCCCC1CO 60781,N1(C(c2ncn(CC)c2)=O)CCCN(C(C2CCC(C(C)C)NC2=O)=O)CCC1 60782,CC(C)CCCC(=O)NCCNC(c1scnc1C(C)C)=O 60783,C1(CC(=O)NC2CC(CNC(C3CC4CCC3C4)=O)C2)CCC(F)(F)C1 60784,N(C(=NCCCF)N1CCC2C(C1)NC(=O)N2C)Cc1c(C)nn(C)c1C 60785,C1(C(N)=O)(OC)CN(C(=O)C(C2CCCC2)NC(c2csc(C3CC3)n2)=O)C1 60786,c1(C(N(C)CC2C3CC2N(C(=O)C(F)C2CCC2)C3)=O)ccc(C=O)cc1.CN 60787,CC1CN(C(C2CC(C)(F)C2)=O)CCC1NC(c1cc(C(=O)O)cs1)=O 60788,C=C(C)CC(C)C(=O)NCC(C)(C)NC(c1ccsc1C)=O 60789,c1(CC)ccc(C(=O)N(C2CN(C(=O)C#CC3(C)CC3)CC2(C)C)C)c(O)c1 60790,N1(CC(=O)N(C(C)CN(C)C(c2cc(O)ccc2F)=O)C)Cc2ccccc2C1 60791,N1(C(Cc2ccc(C)cc2)=O)CCC(O)C(NC(=O)C(O)C2CC2)C1 60792,N1(Cc2ccc(C(=O)NCCC(C)OC)o2)CC2CCC(NC(C)=O)CC2C1 60793,C1(NC(C2C(C)C2)=O)CCC(C)(NC(=O)Cc2c[nH]ccc2=O)CC1 60794,Cc1ccc(CCC(N2CC(O)(CCNC(C3CC3(C)C(F)F)=O)C2)=O)o1 60795,C1(CNC(C2(C3CCCO3)CC2)=O)CCCCN1C(c1cnsn1)=O 60796,c1(C(=O)NCC(C)(CO)NC(C(C)N(C(C)=O)C)=O)ncc(C)cc1F 60797,CC1C(NC(c2c[nH]cc(F)c2=O)=O)CCCN1C(c1ccccc1F)=O 60798,C1(CCC)(NC(=O)CS(=O)CC)CCCN(C(=O)C2=CCCCC2)C1 60799,c1(C(N2CC(SC)CCC2(C)C)C(=O)NCCC)cn2cc(F)ccc2n1 60800,C(=O)(CCC(C(=O)O)c1ccccc1)Nc1ccc(COC)cc1Br 60801,N1(C(C=C(C)c2ccccc2C)=O)CCC2C1CCCN2C(=O)C=C(C)C(F)F 60802,C(=O)(CC1OCCc2ccccc21)N1C2CC(NC(C3CC3F)=O)CC1CCC2 60803,C1(CC(=O)NC(C)CCCNC(=O)CNc2cnn(C)c2)SC(=N)NC1=O 60804,c1(C(=O)NCC(C)(CO)NC(C2CC(C)C2)=O)ccc2cccc([N+](=O)[O-])c2n1 60805,c1(OCC)ccc2ccccc2c1CN1CC2(CN(C(c3occc3C)=O)C2)C1 60806,CC(O)C(C)C(=O)N(CCNC(=O)C=CCCC(F)(F)F)CCOCCO 60807,c1(C(=O)NC(CN(C(=O)CCC(C)(C)OC)CC)C)cnn2c1NCCC2 60808,N1(C(c2cc(C)nnc2)=O)CC2CS(=O)(=O)CC2(CNC(=O)C#CC(C)(C)C)C1 60809,C1(NC(c2cc(C)[nH]n2)=O)CN(C(c2snc(O)c2Cl)=O)C2(CCCOC2)C1 60810,N1(C(CC2C(C)=NNC2=O)=O)CC(CNC(c2[nH]cnc2C#N)=O)C(C)(C)C1 60811,N1(C(CC2ON=C(CC)C2)=O)CCC(C(=O)N(CC(=O)OCC)C)C(C)C1 60812,c1(C(N2CC(O)(C(C)N(C(C3CCC(C)C3)=O)CC)C2)=O)cnccc1C(F)(F)F 60813,C(C(COC)CC(=O)NC(CNC(=O)C(C)n1ccnc1)C(C)(C)C)OC 60814,CC1CCCc2cc(C(=O)NC3(CNC(=O)COCCCF)CCOC3)nn21 60815,CC1(C2CCN(C(C3CCN(C(=O)COc4cccnc4)CC3)=O)C2)CC1 60816,c1(NC2C(OC)C(C)(C)C2)nc2cccnc2c(=NCc2ccncn2)[nH]1 60817,S(=O)(=O)(c1cc(Cl)c(Cl)cc1Cl)NC(C1C(C(C)C)(CC)C1)=O 60818,c1(C(=O)NC2CC(C)(NC(C3C(C)OC(=O)N3)=O)C2)cnc(S(C)(=O)=O)s1 60819,c1(C(=O)NC(C2CCCCN2C(c2cnnc(Cl)c2)=O)C)nc(=O)n(C)[nH]1 60820,C12(CC)CCC(CC1)N(c1nc(C(C)C)c(C(N)=O)s1)C2.C12CC1C(=O)NC2=O 60821,C1(C(N2CCC(O)(C(=O)Nc3c(C)[nH]nc3Cl)C2)=O)CCc2ccccc2O1 60822,C1(NC(CC(COC)C)=O)CC2CC1CC21CC1.C12(CCOC1)C(=O)N2 60823,c1(C(=O)NC2CCN(C(c3c(SC)csc3)=O)CC2C)cnn2ccc(C)cc12 60824,c1(C(N(CCC)CCNC(=O)C(C2CCOCC2)F)=O)ccc(C)cc1O 60825,C(CCCCC(=O)NC1CCN(C(=O)C(C)SC)CC1)n1cc(COCC)nn1 60826,C(=O)(CC(C)C(C)C)NCC1(CNC(C2N(CC)CCC2)=O)CCC1 60827,N1(C(CC2N(C(C(C)SCCCC)=O)CC(O)C2)=O)CCC(F)(C#N)C1 60828,c1(C(=O)NCC(N(C(=O)C(=O)Cc2ccccc2)C)C2CC2)cccc(=O)o1 60829,C(CC(C)(C)CC(=O)NC(C1(O)CN(C(=O)CC(C)c2ccccc2)C1)C)OC 60830,C1(CN(C(=O)NCc2nnc(CC)o2)C)(SC)CCCCCCC1 60831,N1(C(C2C(CNC(C(CCCC#C)C)=O)OCC2)=O)CCC2CCCC2CC1 60832,C1(SC)CN(C(=O)CC2CCC(=O)N2C)CC1NC(C1CC=CC(O)C1)=O 60833,C1(C(=O)NC(C=C)C(F)(F)F)C2CC3C(C2NC(=O)C(C)OC)C13 60834,c1(C(N2C(C(N3CCCC(C)(O)C3)=O)C3CCC2C3)=O)n[nH]c2ccc(F)cc12 60835,CCC(C)(C(=O)NCC(CNC(C1(Cc2cccc(Cl)c2)CC1)=O)CO)OC 60836,N1(C(c2ccn(CCNC(C3C(=C)C3)=O)c2)=O)CCN(C)C(=O)C1CC 60837,CC1CN(C(c2c[nH]cc2C(C)(C)C)=O)CC1NC(C1CCC(=O)N1)=O 60838,c1(CC)ccc([N+](=O)[O-])cc1C(=O)Nc1cccc(OCC2(CN)CC2(F)F)c1 60839,Cc1cc(C(C)NC(N2CC3CC(C)C3C2)=O)ccc1C#N 60840,C(Cc1cnc[nH]1)(C(=O)N(CCO)CCO)NC(C(c1cnn(C)c1)C)=O 60841,c1(C(N2CCC(NC(CNC(CNC(C)=O)=O)=O)(CF)C2)=O)cc(O)ccc1C 60842,c1(CC)nc2n(n1)CC(NC(=NCCCSC)NCC1(CC)CCNC1=O)CC2 60843,c1(CC)cc(C(=O)N(CC(C)NC(=O)C=Cc2nc(C)cs2)C)ccc1OC 60844,CC1CCN(C(=O)CCNC(=O)CO)CC1CNC(c1cc(F)cc(F)c1)=O 60845,CC(C)C(O)C(C)(C)C(=O)N1CCC(C(=O)NCC2(C)CCCCC2O)O1 60846,c1(CC)n[nH]c(=NC2CCN(C(c3cnn(-c4ccncc4)c3)=O)C(C)C2)s1 60847,N1(C(N(CC)CC)=O)CCN(c2ccnc(NCC3CNC(=O)C3)n2)CC1 60848,C=CCCCC(C(=O)OC)NCc1cc(Br)c(F)cc1OC 60849,c1(CCCC(=O)N(C)CC2(NC(c3cnn(CC)n3)=O)CC2)ccccc1OC 60850,C1(C(=O)NCCC2CC(C(=O)NCCC(O)C3CCC3)C2)CCCN1C=O 60851,Cn1nnc2cc(C(N3CC4CCC4(NC(c4csc([N+](=O)[O-])c4)=O)C3)=O)sc12 60852,C1(C(=O)NC(CN(C(c2cnc(O)n2CC)=O)CC)C)CCCCC1(C)C 60853,C(C1c2ccsc2CCN1C(C1CCCC1)=O)NC(C(C)NC(=O)C(C)(C)C)=O 60854,Cc1cc(C(N2CCCCC2CS(N)(=O)=O)=O)ccc1Br 60855,S(=O)(=O)(c1cc(C)cnc1Cl)N1CCC(CNc2cccc(C(C)=O)c2)C1 60856,C(=O)(C(=O)CCC(C)C)N1CCC(NC(CCC(C)SC)=O)CC1C 60857,C#Cc1ccnc(C(=O)NCCOC2CCN(C(=O)CC(C=C)CC)CC2)c1 60858,Cc1cc(-n2nc(CCN(C)C)nc2CN2CCC(OC(F)(F)F)CC2)ccc1Cl 60859,c1(OC)cccc(-c2cn(C3CCC(C(=O)NCC4CNC(=O)O4)C3)nn2)c1F 60860,c1(-n2c(C)nc(SC)n2)cc2ccccc2c(O)n1.C12(O)CCN(C1)C(C)(C)CNC2=O 60861,C=CC1(C(=O)NCCCN2CC=CC2)CCN(C(=O)C(C2CCCCC2)C)CC1 60862,c1(C(=O)NC(CCCNC(c2c(NCC)scn2)=O)C)cnc2c(c1)CCOC2 60863,c1(C(C)C)cnn(C)c1C(N1CC(NC(=O)CNS(N)(=O)=O)C(C)C1)=O 60864,c1(OC)c(C)csc1C(=O)N(C)CCN(C(=O)C(C)Sc1ccccc1)C(C)C 60865,c1(-c2cc(OC)cc(OC)c2C#N)cnc2[nH]cc(C(=O)N=c3nc[nH]s3)c2c1 60866,c1(C(=O)NC(C)Cc2ccc(CNC(C3(Br)CC3)=O)cc2)ccc(N)cc1F 60867,C1(CNC(C(n2cc(Cl)cn2)C)=O)CC2(CCC2)CN1C(C1CCCC12CC2)=O 60868,Cc1ccc(O)c(NC(c2nnn(C)c2C)=O)c1 60869,C1(NC(C2N(CC)CCOC2)=O)CC(O)CN(C(=O)C(F)(F)c2nccs2)C1 60870,CC(c1ccsc1)=CC(=O)NCCCC(C)NC(c1ccc(CO)s1)=O 60871,C(c1cccnc1)=CC(=O)NCC1CCC(NC(=O)CC2(O)CCCOC2)CC1 60872,c1(C(=O)NC2(CCNC(=O)CCn3cc(Cl)cn3)CC2)cc(O)nc(O)n1 60873,Cc1cc(C(=O)NC2CCC2NC(c2[nH]nnc2C2CC2)=O)cc(C)c1Cl 60874,C1(C(N2CC(NC(c3c(CC)ncs3)=O)(CO)C2)=O)CC(=O)N(C2CCCC2)C1 60875,C1(CNC(C(CC=C)NC(C)=O)=O)COCCN(C(=O)C(=O)NC(C)C)C1 60876,C1(CN(C)C(C2(C3CCCCO3)CC2)=O)CCCN1C(C1CCCN1C)=O 60877,C1(C(=O)NC(C2CCOC2)CC)(CNC(c2ccns2)=O)CCCC1 60878,c1(C(N2CCC(F)(CNC(C(C)CC3CCC3)=O)C2)=O)ccc2c(n1)COCC2 60879,c1(NC(C)=O)cnccc1C(=O)N(CCNC(C1CC1(C)C(C)C)=O)C1CC1 60880,C#Cc1ccc(CC(=O)N(CC(C)NC(=O)C=CC(C)CC)C)cc1 60881,c1(C(N(CCNC(=O)C(C2(O)CCCC2)F)CC)=O)ncnc2c(C)csc12 60882,Cc1ccc(C2CC2C(N2CCCC(N(C)C(c3cnccc3Cl)=O)C2)=O)cc1 60883,c1(C(=O)NCC2N(C(CSC)=O)CC=C2)cccc(-n2cccn2)n1 60884,C1(C(=O)NC(CC=C)CO)CC2(CCN1C(C1CCCC(C#N)C1)=O)CC2 60885,C(c1cccc(Cl)c1)=CC(=O)N(C1CCN(C(c2c(C)coc2)=O)C1)CCO 60886,C1(CC(=O)NCC(CO)NC(C(C)C2CC2)=O)CCN(CC(F)F)CC1 60887,C1(C(=O)NC2(C)CC(NC(c3ccn(CC(C)C)n3)=O)C2)CN2CCN1CC2C 60888,C(N=c1cccc(S(=O)(=O)NC2CCCC(C)C2)[nH]1)c1c(C)ccc(C2CC2)c1 60889,N12CCC3(CCCCC13)NC(=O)COCC2=O.Cc1cccc(NC(N)=O)c1F 60890,Cc1nc(Cl)[nH]c(=NCC2C3CN(C(c4cc(Cl)sc4Cl)=O)CC23)c1F 60891,C(=O)(C(O)C(CCC)NC(=O)C(C#N)C(C)C)NCC1(C=C)CCC1 60892,C12(CNC(C(CC=C)(F)F)=O)CCC(CNC(C3CCCC(F)C3)=O)(CC1)CO2 60893,c1(CN(CCOC)Cc2ccc(-c3nccc(C=C)c3)s2)cccn2ccnc12 60894,CC(C)CCCCC(=O)NCC(O)CC(=O)NC(CCO)C1CCCC1 60895,N1(C(C2C(=C)C2)=O)CC(n2cc(C3(OC)CCC3)nn2)C(O)C1 60896,C1(CNC(=NCCOC)NCC2=CCOCC2)CN2CCCCC2CO1 60897,C12(CNC(NCC3(COC)CCCCO3)=NCC(C)C)CC3CC(CC(C3)O1)C2 60898,N1(C(Cn2c(C)ccn2)=O)CC(C)CN(C(=O)C2=CSCCO2)C(C)C1 60899,[N-]=[N+]=NC1CC2(C(N3CC(O)(CCNC(C4(Cl)CC45CCC5)=O)C3)=O)CC12 60900,N1(C(C(C)OCC2CCCO2)=O)CCC(NC(C23CCC2C3)=O)CC1 60901,c1(C(C(=O)NCCCF)N(C)Cc2ccsc2)ccc(OCC#N)cc1 60902,C=Cc1ccc(C(N2CC3CN(C(=O)C(c4ccccn4)N)CC23)=O)cc1 60903,C(=O)(C1CCCn2ccnc21)NCC1C2CN(C(=O)OC(C)(C)C)CC21 60904,O=CN1CCCC1C(N1CC(O)CC1CNC(=O)C(O)c1ccco1)=O 60905,Cc1nc(CCC(N2CCC(CNC(=O)CC3CSCCS3)C2)=O)cs1 60906,c1(OCC)ccc(S(=O)(=O)NC2CC(S(C)(=O)=O)C2)cc1-c1cccc(C)c1 60907,Cc1cnc(C)c(NC(C2CC(F)CN(C(=O)Cc3cccs3)C2)=O)n1 60908,C1(NC(c2cnc(C)o2)=O)CCN(C(C2CC23CCSCC3)=O)C1(C)C 60909,S(=O)(=O)(c1ccc(Br)cc1NCCc1ncccn1)N(CC)CCO 60910,N1(C(C2C(C)C2C)=O)CC(NC(c2cc(N)nc(Cl)c2)=O)CC(C)(C)C1 60911,c1(OC)ccc(CN2CC(CNC(c3ncoc3C)=O)C2)nc1Br 60912,C1(C(N(CC(C)NC(CC(C)n2ccnc2)=O)C)=O)CC2(C1)CC2F 60913,C=CC(C)(O)C(=O)NC(C1CN(C(c2ccnc(CC)c2)=O)CCO1)C 60914,N1(C(CN(c2ccccn2)C(C)=O)=O)CC2CC1C2CNC(c1c(C)ccn1C)=O 60915,CN1CC2CCN(C(=O)CC3CCCCN3C(=O)CNC(N)=O)CC2C1 60916,CN1CCCC(CCC(N2CC=CC(NC(c3csnn3)=O)C2)=O)C1 60917,c1(C(=O)NCC(CN(C)C(C2(C(F)(F)F)CC(C)(C)C2)=O)O)cn2c(n1)CCC2 60918,c1(C(N(C)CCN(C(=O)C(O)CC(N)=O)C)=O)cc2cc(Cl)sc2[nH]1 60919,C1(NC(C2(CC)CCC2)=O)CCN(C(=O)CSCCOC)CCC1CO 60920,N1(C(CCOCC(C)C)=O)CC(NC(c2cccc[n+]2[O-])=O)C2(CCC2)C1 60921,CCCCS(=O)(=O)NC(C)C(=O)NCCCN(C(=O)CC1(CO)CC1)CCO 60922,c1(C(N(C)Cc2ccccc2CNC(=O)CSC(F)(F)F)=O)cnc(Cl)cc1Cl 60923,c1(CC(=O)NCC(C)N(C(c2ccnnc2)=O)CC)cc(Br)cnc1OC 60924,N1(C(CNC(C2CCCC2)=O)=O)CC2CS(=O)(=O)CC2(NC(C2CCC2)=O)C1 60925,C1(CNC(CCNC(C)=O)=O)CC(C(=O)NCCN2CCCCC2)CO1 60926,c1(OCC(N2CCC(C)N(Cc3ccccc3)CC2)=O)ncnc2ccccc12 60927,CCC(C(=O)NCCC1CC(F)(F)CN1C(c1nc(O)sc1C)=O)C(C)(C)CC 60928,C(CC(C(=O)NCCC=CCCC)NC(c1cc(C2CC2)on1)=O)=CC 60929,O=C(C1=CCCO1)NCCN(C(=O)C(F)n1cccn1)C1CC1 60930,CC1CCC(CNC(=O)Cc2cncnc2O)CN1C(c1cc(=O)n(C)cn1)=O 60931,CCC(C)C(O)C(C)C(=O)N1CC2CCC1CN2C(=O)CN1C(=O)CNC1=O 60932,Cc1nc2cccc(C(=O)NCC(CO)NC(C3(C)CCN(C)C3=O)=O)c2[nH]1 60933,N1(C(C(C)(Cl)CCl)=O)CC2CC1CC2NC(c1cccs1)=O 60934,C(=O)(C(=O)N=S(C)(C)=O)NCCC1CN(C(=O)C=Cc2ccsc2)CC(C)O1 60935,c1(CN2CC3N(C(C4CC4c4ccc(F)cc4)=O)C(C3)C2)cc(Br)cc(Cl)c1F 60936,C1(NC(c2n[nH]c(C3CC3)c2Br)=O)CCCCN(C(=O)CC2CCCC2)C1 60937,c12ccc(Br)c(c1C)NC(=O)N2.C1(C(=O)OC)(C(=O)OC)CCCO1 60938,N1(C(CCC)=O)CCCC2C1CCCN2C(=O)C=Cc1cccc(Cl)c1 60939,C1(NC(=O)Cc2ccccc2C2CC2)CCS(=O)(=O)C12CN(C(=O)CC1CC1)C2 60940,CCC(CC(=O)NC1COCC1NC(c1ccnc(C2CC2)c1)=O)C(F)F 60941,N1(C(C(=O)NC2CC2)=O)CCCC1C1CCN(C(C2CCCCS2)=O)C1 60942,c1(CC(C(=O)N(C)CC2(O)CN(C(C(COC)N(C)C)=O)C2)C)cccc(F)c1 60943,CCCCCC(O)CNC(c1ccc(OC(C)C)nc1)=O 60944,N1(C(CC(=C)C)=O)CC2CC(NC(c3c[nH]nc3-c3ccsc3)=O)CC(C2)C1 60945,C(C(=O)NNC(=O)C(F)(F)F)Cc1c(C)cc(C)c(C(C)=O)c1C 60946,Cc1nc(C)n(CC(=O)NC2COCCC2C(=O)NCC2(F)CCOC2)n1 60947,N#Cc1ccc(CCC(N2CCOCC2CC2CC2)=O)cc1 60948,C(=O)(C(C)(C)C(=O)NCC(C)NC(c1ccc(SC(F)(F)F)s1)=O)OCC 60949,c1(C(N2CC(CC)(NC(=O)CC3CC(=O)NC3=O)C2)=O)cncc(F)c1C 60950,N1(C(c2sccc2Br)=O)CC2(C1)CN(C(c1ccc(O)cc1F)=O)C2 60951,Cc1cc(CCC(=O)NCC(C)(C)CN(C)C(C2CCN(C)C2)=O)nn1C 60952,C(=O)(C(F)CC(C)(C)NC(c1ccccc1)=O)N1C(C)(CC)CC1 60953,C(CC(C)(C)NC(c1cnoc1-c1cnn(C)c1)=O)N(C(=O)C=CC(F)(F)F)C 60954,C1(NC(c2n(C)nc(Br)c2)=O)CCN(Cc2cccc(C(F)(F)F)c2O)CC1F 60955,C1(NC(=O)COCCCF)CN(C(c2cnc3ncccn23)=O)C2(CCCC2)C1 60956,C(=O)(C(C)(C)C)NC(C)C(=O)N(C)CCN(C)C(C1(CC2CC2)CCCO1)=O 60957,Cn1cnc2ccc(-c3cnc(F)c(F)c3)cc12 60958,c1(CNC(=O)C(N2CCC3(O)CCCC23)=O)ccc(Br)cc1Br 60959,n1(CC(CC)O)cc(C2(O)CN(C(=O)Cc3csc(Br)c3)C2)nn1 60960,C1(NC(CS(=O)(=O)NC)=O)CCN(C(=O)C(n2cc(Cl)cn2)C)CC1O 60961,c1(CC(=O)NCC(CNC(Cn2c(C)c(Cl)cn2)=O)C)cc(C(C)C)cc(F)c1 60962,C1(NC(COCc2ncc(C)o2)=O)CCC(C)(CNC(=O)C(C)(C)N(C)C)C1 60963,c1(C(=O)NC2C(CNC(c3cn(C(C)C)nc3)=O)CC2)cccc2c1CCCC2 60964,N1(CCO)CCN(CC(c2ccccc2)F)CC1.c1(NCCF)ccccc1 60965,c1(C(=O)NC2CCCC(NC(C3CCCS3(=O)=O)=O)C2)cnc2ncc(Cl)cn12 60966,C1(C2CCN(C(=O)Cc3cc(Cl)ccc3Cl)CC2)(NC(C2CNC(=O)N2)=O)CC1 60967,C1(C(=O)NCCC2CCCCN2C(=O)COCCCF)CC2CC1CC2(F)F 60968,c1(OCC(=C)C)ccccc1C(N1CC(NC(C2CC(SC)C2)=O)C1)=O 60969,O=C(CC1COc2ccccc21)NC1CC(NC(=O)C(F)(F)c2cncs2)C1 60970,C(=O)(CC(C(F)F)C(C)(C)C)N1CCC(CCNC(C2=C(C)CCC2)=O)CC1 60971,c1(C(N2CCC(N(C(C(C)OCC=C)=O)CCO)CC2)=O)ccc(F)cc1C 60972,N1(C(CCCC)=O)CC(OC)C(OC)C1CNC(=O)CCc1scnc1C 60973,C(=O)(C(O)C(F)(F)F)N(CCCNC(c1cnns1)=O)Cc1ccccc1 60974,CCC(CC(=O)N1CCCC(CN(C(=O)Cc2cnccc2OC)C)C1)C1CC1 60975,C1(NC(C2(C(=O)OC)CC2C)=O)CCN(C(=O)CNC2CC2)CC1 60976,N1(C(CNC(=O)NC)=O)CCC(CO)C(NC(=O)CN2CCC(C)(C)C2)C1 60977,Cc1cc(=NC(C)C(c2ccccc2)NC(=O)C(C)S(C)(=O)=O)[nH]c(C)c1C#N 60978,c1(OC)cc(C(=O)NCC2CCN(C(=O)C(C)N(CC(F)(F)F)C)C2)cc(C)c1 60979,c1(CC)c(C(=O)NC(C)CCCNC(c2conc2C2CCC2)=O)cccc1C 60980,C1(CNC(COCC)=O)CC(NC(=O)COCCSC(=O)N)C1(C)C.CC 60981,C(CC(C)C)(C(=O)N1CCC(CNC(c2nnn(C(C)(C)C)n2)=O)C1(C)C)OC 60982,CC(C)CCC(=O)C(=O)NC(C1CN(C(=O)CC2C=CCC2)C1)C 60983,CC1(C(=O)NCC(C2CCOC2)NC(c2cnc(N(C)C)cn2)=O)CCCCC1 60984,c1(C(N2CCCOC2C)C(c2ccn(CC)c2C)=O)csc(=Nc2ccccc2)[nH]1 60985,C1(CC)CN(C(=O)Cn2ncnn2)CCN1C(=O)Cc1cc(O)ccc1Br 60986,C1(CNC(C=C(C)C)=O)(CNC(=O)Cn2cnc([N+](=O)[O-])n2)CC2CCCC2C1 60987,c1(OC(C(=O)NCC(C(=O)NC)N(C)C)C)cccc(C)c1 60988,C1(CNC(C(C)OCC#C)=O)CC(C)N(C(c2cc(C(F)(F)F)no2)=O)C1 60989,c1(OCC)csc(C(=O)NCC=CCNC(C2CCC(C(F)(F)F)C2)=O)c1 60990,C12(C(N3CCC(C(C)(C)C(=O)OC(C)(C)C)C3)=O)CC1CS(=O)(=O)C2 60991,N#Cc1sc(=NCC2CCN(C(c3cc(Cl)no3)=O)C2)[nH]c1Cl 60992,C1(NC(C2OCCN(C)C2)=O)CC2(CCN(C(c3ccc(C#N)c(O)c3)=O)C2)C1 60993,c1(C(=O)NCC2C(CNC(=O)C(F)n3ccnc3)C2)cc(-n2ccnc2)ncn1 60994,N1(C(c2cnn(CCC)c2C)=O)CC(CNC(=O)C=CS(C)=O)OC2CCCC12 60995,c1(C(=O)NCC(N2CCCC(CN(C)C(N)=O)C2)=O)ccccc1[N+](=O)[O-] 60996,CC(C)C(O)C(=O)N(CCCNC(=O)CCN1CCCCCC1)C(C)C 60997,c1(C(N2CCC(CNC(C(CCC)O)=O)C2(C)C)=O)nccc2cccnc12 60998,Cc1noc(-c2cn(CC(=O)NCC(C3CC3)N(C)C(c3ccon3)=O)cn2)n1 60999,C1(N(C(C(C)(O)c2cccc(Cl)c2)=O)CC=CCCC=CC#N)CSCCN1c1ncncc1Cl 61000,CS(C)(=O)=Nc1ccc(C(N2CC3CCCC3(CNC(C3(F)CC3)=O)C2)=O)cc1 61001,Cn1cnc(NC(=O)NCC2(c3cccc(C(F)(F)F)c3)CCC2)cc1=O 61002,N1(C(c2ccc(C)o2)C(=O)OC(=O)NC(C)(C)C)CCn2c(C)nnc2C1C 61003,C=CCC(C(=O)OCC)NC(=O)CCN(C(C1CCC1C)=O)CC1CC1 61004,C(=O)(CCC(C)C#N)NCC1N(C(c2c(C)coc2C(C)C)=O)CCC1 61005,c1(C(=O)NCC2(OC)CCN(C(=O)C=CC3CCCO3)C2)cc(C)c(C)cn1 61006,[N-]=[N+]=NC1CN(C(=O)Cn2cnnn2)CC1NC(=O)COc1ccccc1 61007,Cc1[nH]nc2c(C(N3CCC(CO)(NC(C4CNC(=O)N4)=O)CC3)=O)cccc12 61008,N1(C(C2CN(C(CNC(=O)OC)=O)CC(F)(F)C2)=O)CCC2(CCOC2)CC1 61009,C(N=c1[nH]c(=NCC(C)(F)c2ccccc2)c2[nH]ccc2[nH]1)C1N(C)CC1 61010,C(C1CCCN1C(c1cnn(C)c1N)=O)=CC(N1CCC(CN(C)C)C1)=O 61011,c1(NC(C)=O)ccc(SCC(N2CCC(N(C(=O)C=CBr)C)C2)=O)cc1 61012,N1(C(C(CC(CC)C)C)=O)CC2CCCN(C(=O)COC3CC3(C)C)C2C1 61013,C1(C(C(=O)NCCC(CNC(C(CSC)(C)C)=O)O)O)CCCCCCC1 61014,C1(NC(C2CN(CCC)C(=O)C2)=O)CCC12CN(C(c1cn(CC)cn1)=O)C2 61015,CC1(C)C(CNC(=O)Cn2cnc([N+](=O)[O-])n2)CCN1C(=O)COC1CC=CC1 61016,C12(NC(CCc3cnc(C)o3)=O)CCN(C(c3ccn(C)c3)=O)CC1C2 61017,c1(OC)cc(Nc2ncc(Cc3ccc(C(C)(C)C)cc3)s2)ncn1 61018,c1(C(=O)NCC(C)NC(=O)C(F)CC2CC2)ccc(Br)cc1 61019,c1(CC)nn(C)c(Cl)c1C(=O)NC1C2CN(C(C3(c4cc[nH]n4)CC3)=O)CC12 61020,Cc1nn(C(C)(C)C)c(C)c1C(N1CCC(c2cc(N)ccn2)CC1)=O 61021,CC1CN(C(=O)CNC(=O)Cc2ccccc2)CCN1C(=O)C(CO)N(C)C 61022,c1(C(=O)NCC(C(=O)Nc2c(CC)cccc2)(C)CC)ccc2nccn2c1 61023,C1(NC(C(CC#C)(C)NC(c2c[nH]c(=NC)o2)=O)=O)CC2CC1CC21CC1 61024,C1(NC(CCC=C(C)C)=O)CN(Cc2ccnc(Cl)c2C)CC1C#N 61025,N1(C(CN(CC)CC)=O)CCCCC1C1(NC(=O)COCC(C)C)CC1 61026,N1(CCC#C)CCN(C(=O)NC2C3CCC(F)C23)CC1 61027,C(=O)(CS(=O)(=O)Cc1cncn1C)OC(c1ccc(Cl)cc1)C(C)C 61028,CC1CC(C)N(C(c2cn3c(Br)cccc3n2)=O)CCN1C(=O)CNC(N)=O 61029,N1(C(Cc2cccc(OCCC)c2)=O)CCN(C(=O)CCCF)CC1CCOC 61030,C1(NC(C2CCC(C)O2)=O)CCC2CN(C(=O)C(c3ccccc3)C)CCC2C1 61031,c1(CC(N2CC(C(N)=O)(CNC(C3C(C)C3C)=O)C2)=O)cccc(Br)c1 61032,N1(C2CCC(NC(COCCCCC)=O)C2)CCN(C(=O)C(Cl)=CCl)CC1 61033,CC(C)=C=CC(=O)N(CC(O)CN(C(=O)COCC1CC1)C)C 61034,C1(CNC(C(CC#C)C2CC2)=O)CC2(CCC2)CN1C(c1ccnc(CO)c1)=O 61035,N1(C(CCOCCC)=O)CC(NC(C2CC(Cl)(Cl)C2)=O)CC12CCC2 61036,C(=O)(C(C)S(C)(=O)=O)NC1C(CC)N(C(=O)CCn2ccnc2)CC1 61037,N(C1CCCc2cc(C#N)ccc21)c1cccc(N2CCN(C(C(C)C)C#N)CC2)n1 61038,C(C(C)C(F)C(=O)NC(C)C(C)n1cccn1)NC(CC1(CC(=O)OC)CC1)=O 61039,C(=O)(C1=CC2CCCC12)N1CCCC(C)(NC(C(c2c(C)noc2C)C)=O)C1 61040,Cc1onc(C(F)(F)F)c1C(=O)NC1CCN(C(=O)CN2C(C)CCC2C)CC1 61041,Cc1ccc(=O)n(CC(=O)NCCCCNC(=O)C(c2ccc(F)cc2)(C)F)n1 61042,CCC(=O)CCC(=O)N1CCC(CCC(=O)NC2CCC=CCCC2)C1 61043,C12C(CC)CCN1C(=O)C(C)OC(=O)NC2=O.c1(Sc2ccco2)ccccc1 61044,CC(CCN=c1[nH]c(=NCC2CC23CCC3)c2cc(Cl)ccc2[nH]1)CC(C)(C)C 61045,CCCC(C)(O)CC(=O)NC1CCC(CNC(=O)CCn2cnccc2=O)CC1 61046,C1(Cl)(C(=O)NCCNC(c2cnc(C(F)F)s2)=O)CC12CCOCC2 61047,C12(CNC(C3(CC)CC3)=O)CCCCC1CN(C(c1ccc(CSC)cc1)=O)C2 61048,Cc1nc(NC(CNC(c2cc(C(C)C)no2)=O)C(C)C(C)C)c2cc[nH]c2n1 61049,c1(C(=O)NCC(C)N(C)C(c2cnn(CC(F)F)c2)=O)cc(C(C)(C)C)c[nH]1 61050,c1(C(N2C(C)CN(C(c3ccc(SC)s3)=O)C(C)C2)=O)ccc2c(c1)N(C)CC2 61051,C1(C(=O)NCC(O)CNC(=O)Cc2n[nH]cc2Br)(OC)CCCCC1 61052,C(=O)(N=c1[nH][nH]c2c1CN(C(c1c(F)cc(Br)c(F)c1F)=O)C2)C1C(C)(C)C1 61053,CCC(C)C(C=O)N1CCC(C(=O)N(C)C)CC1.C1(NCCC#N)CCOCC1 61054,C1(C(=O)NCC2CCN(C(c3ccccc3O)=O)C2)CCC2C(CC1)C2(F)F 61055,C1(NC(Cc2c(C)ccs2)=O)CCCC(NC(=O)CC(=O)N(C)C)CC1 61056,C12(C(=O)NCC(C(CC)C)C)CC(CO1)N(C(C1CCC(C)(C)OC1)=O)C2 61057,c1(C(N(CCOC)CCNC(=O)C(O)C2CCC2)=O)cc(P(C)(C)=O)cs1 61058,c1(C(=O)NCC(C)N(C(c2c(NCC)scn2)=O)C)c[nH]c2ccc(F)cc12 61059,c1(C(N2CC(CNC(CC(CCC)O)=O)CC2(C)C)=O)ccc(N)cc1[N+](=O)[O-] 61060,C1(OC)CCC(C)(C(N2CC(CNC(c3cccc(F)c3Cl)=O)C(O)C2)=O)CC1 61061,CC(C)C(C)C(=O)NCc1cc(C(=O)NOCC2CCOC2)on1 61062,Cc1ccc(C(=O)NCC(c2ccccc2)CNC(=O)CC#N)c(F)c1 61063,n1(CCC)cc(Cl)c(C(=O)NC2CCC(CNC(c3[nH]ccc3C3CC3)=O)C2)n1 61064,C1(CC(C(=O)NCCC#N)N(C)CCn2cncn2)CCC(C)(C)O1 61065,Cc1ccccc1C=CC(N1CCC(C(N2CC3(CC3)CC2C)=O)C1C(C)C)=O 61066,c1(C(=O)NC2CC(NC(C3(C)CCCCO3)=O)C2)cc2sc(Cl)cc2s1 61067,N1(C(C(CC)NC(N)=O)=O)CC(NC(=O)C#CC(C)C)C(C)C1 61068,C(c1cc[nH]n1)=CC(=O)NC1C(C(=O)N(CC(=O)NC2CCCC2)CCO)CCC1 61069,Cc1cccc2c1OCCC2NC(=NCCN1CCCC1C)NCC1CC1 61070,CC(C)(CS(C)(=O)=O)C(=O)NCC1COCCN1C(=O)CC1CCCNC(=O)C1 61071,C#CCC(C(=O)N1CCCC(OC)C1)NC(=O)C(C)(C)NC(C)=O 61072,C1(CC)CCN(C(c2cscc2Cl)=O)C1C(=O)NC1(CC(C)C)CC1 61073,c1(CC)ncc(C(=O)NCC2(F)CC(NC(=O)CN3CC4CC4C3)C2)s1 61074,CC1(C)CC2(CC2C(N2CCC2CNC(c2ncc(N)cc2Cl)=O)=O)C1 61075,C(=O)(C(CCC)C(C)C)N1CC(NC(CCC=CC)=O)C2(C1)CC2 61076,N1(C(C(CSCc2ccccc2)NC(C)=O)=O)CC2(CC(NC(=O)C(C)C)CO2)C1 61077,C(C)(CNC(c1cn(C2CC2)cn1)=O)(CO)NC(C(C)c1cccs1)=O 61078,c1(OC)cccc(C(C)CC(=O)NCC2CC(NC(=O)Cc3ccnn3C)C2)c1 61079,CCCC(C)(CC)C(=O)N1CCC(CN(C(=O)CSCC(=O)NC)C)C1 61080,CC1(C)CN(C(c2scnc2C(F)F)=O)CC(CNC(C2(C)CC2Br)=O)O1 61081,Cc1c(C(=O)NCC2(NC(=O)C(C(C)C)NC(N)=O)CCOCC2)cnn1C 61082,C(CC(=O)N1CCC(CC(N)=O)C1)(C(C)(C)C)NC(Cc1ccc(C#C)cc1)=O 61083,N1(C(c2c(C)ncn2O)=O)CCN(C(c2cccc(N)n2)=O)CC(C)(F)C1 61084,Cc1cc2c(C(=O)N(C(C)CCNC(C3CCNC(=O)C3)=O)C)cccc2o1 61085,c1(NCC2CC(N(C)C)C2)cc2oc(-c3ccccc3)cc2[nH]1 61086,c1(C(=O)NC2CCN(C(C(C)(C)NC(=O)OC)=O)C2)cc(C)nc2cc(C)nn12 61087,C1(CNC(C2C(CNC(C(CC#C)O)=O)C2)=O)CCC2(CC2)CO1 61088,c1(C(=O)NCC2(C)CC(NC(C3CC3Cl)=O)C2)cnc2cc(C(F)(F)F)ccn12 61089,C(=O)(C1=NOC(C)C1C)NCCC(=C)CNC(c1cc(CC)on1)=O 61090,c1(C(N(C)CC2CCCN(C(CC(COC)C)=O)C2)=O)c(OC)cccc1F 61091,C#Cc1cncc(C(=O)NCC(O)CNC(c2cnc(C(F)(F)F)c(C)c2)=O)c1 61092,Cc1cc(C(=O)NCCCN(CCO)C(c2ccc(C(C)(C)C)s2)=O)[nH]c1C 61093,C1(CC(N2CC(O)(C(C(=O)NCC(C=C)O)F)C2)=O)CC2(CCC2)C1 61094,C1(NC(c2ccc(N(C)C)cc2)=O)CC2CC1CN(C(c1cc(Cl)no1)=O)C2 61095,c1(C(=O)NC2C(NC(CCc3n(C)cnc3)=O)CC2)ncsc1S(N)(=O)=O 61096,CCS(=O)CC(=O)NCC1CCCC(CNC(C2(n3cccc3)CC2)=O)C1 61097,C(=O)(C1CCc2cccnc21)NCC(CCNC(c1ncn(C)n1)=O)O 61098,C=C(Cl)CCC(=O)NC1CN(C(C2CCCCC2c2nc[nH]n2)=O)CC1C 61099,N1(C(C2C(C(=O)OC)C2)=O)CC2(CCN(C(c3ccc4occc4n3)=O)CC2)C1 61100,C#CCCCC(=O)N1CCN(c2ccccc2NC(C2CC=C(C)CC2)=O)CC1 61101,Cc1ccc([N+](=O)[O-])cc1CN1CC(O)CC1C(=O)Nc1c(O)cccc1C#N 61102,c1(CN2C(C(N3CC(F)C(F)C3)=O)CC3CC32)c(F)cc(F)cc1Br 61103,C(C)(CCC(=O)NC(CCC1CCC1)C(=O)NCCc1ncccc1F)OCC 61104,CC1(C)CC(NC(=O)CC2CC3(C2)CN(C(=O)CC2CCC(=O)NC2)C3)C(=O)O1 61105,c1(CC)ccc(C(N2CCCC(C)C2C(=O)OC)C(=O)NC(C)C)cc1CC 61106,c1(CS(C)(=O)=O)oc2ccccc2c1NC(c1csc2ccc(Cl)cc12)=O 61107,N1(C(CN2CCC(C)C2)=O)CCC2(CC2)CC1C(=O)Nc1cnc(Cl)nc1 61108,c1(C(=O)NC(CNC(C(CCCC#C)C)=O)C)cnc2[nH]c(C)nc2c1 61109,c1(-c2ccc3[nH]nc(C(=O)NCC(=O)NCC)c3c2)nc2cc(C)cc(C)c2[nH]1 61110,CCC(CC)C(C(=O)N1CC2(C)CC1(C(N1CCCCC1CC(C)C)=O)C2)OC 61111,C=CC(C)(CC)C(=O)N1CC(Cc2cn(CC3CCC3)nn2)C1 61112,CC(N=c1nc2c(ncn2C)c(NCCCCC(F)(F)F)[nH]1)c1cnsc1 61113,C1(NC(C(CCC)NC(N)=O)=O)CC2CC1CN(C(=O)CCCCC(C)C)C2 61114,CC1(C)C(c2cn(Cc3cccnc3)nn2)CCN1C(C1CCN1C(C)(C)C)=O 61115,C=C(C)C(C)(C)C(=O)NCCC(O)CNC(=O)C(F)(F)C1(O)CCC1 61116,CC(C)(CC1CCOCC1)C(=O)NCC1CC2CC2N1C(C1CC2CCC2C1)=O 61117,c1(C2C(=O)O2)ccccc1Br.C(=O)(CNC(=O)OC(C)(C)C)OCC 61118,C1(C(=O)NC2CN(C(CN3CCC(C)CC3)=O)C2)CN2CCC1(C)CC2 61119,CC1CN(C(=O)CC2(C)CCCCC2)CCC1CNC(C1(C)COC(=O)N1)=O 61120,C(=O)(C#CC(C)(C)CNC(=O)CCNC(=O)OC)NC(C=C)(C)CC 61121,C1(O)(C(C)NC(CCC(=O)c2ccc(C)s2)=O)CCN(C(C2CCCS2)=O)CC1 61122,N1(CCNC(=O)CC2CCCC23CC3)CCN(C(=O)CN2CCCNC2=O)CC1 61123,c1(C(N(C2CCCN(C(=O)CCc3ncc[nH]3)C2)C)=O)cnc2c(Cl)cccn12 61124,S(=O)(=O)(CCC(=O)NC1CCN(C(=O)Cc2c[nH]ccc2=O)C12CC2)NC 61125,c1(C(=O)NCC2N(C(COCC)=O)CCC2C)ccc2c(c1)N(C)CCO2 61126,N1(C(Cc2c(C)cc(C)s2)=O)CCCC2(CCN(C(C3C(C)C3(F)F)=O)CC2)C1 61127,c1(C(=O)NCCNC(C2(C)CCCNS2(=O)=O)=O)cccc2c1OCCCO2 61128,N1(C(=O)CSc2nc[nH]n2)CCCC2(C1)CN(C(c1cnc(O)s1)=O)CCO2 61129,Cc1nc2ccccc2c(C(=O)NCC2CCCN2C(c2ccc(Cl)s2)=O)c1O 61130,N1(C(=O)Nc2c(OC(F)(F)F)cccc2F)CCC2(CC1)CC(O)(C(F)(F)F)C2 61131,CCC(CC=O)N(C(=O)C(C)CC1CC1)C.C1(C(=O)O)CC(C(F)F)C1 61132,Cc1oc(C)c(S(N)(=O)=O)c1C(=O)NCCCN(C(=O)C(C)CF)C 61133,Cc1cc(NC(=O)CCc2ccc(C(=O)NCC3(C)CCC3)[nH]2)ccc1[N+](=O)[O-] 61134,C(C)(CCC(=O)C(CCC(=O)NCCCCC1CC1C)=O)N.CCCCO 61135,CCCCC(C)(F)C(=O)NCC1CC(F)CN1C(c1ccc(N2CCC2)nc1)=O 61136,C1(CCC(=O)NC(CNC(C2(COC)CCC2)=O)(C)C)C(=O)ON=C1C 61137,c1(C(=O)NCCCCCN(C(C2CN(CC(C)C)C2)=O)C)cc(F)ccc1O 61138,C(=O)(C1COc2ccccc21)NC(c1ccc(N(C)C)cc1)CNC(=O)CO 61139,C(=O)(C1=CCCC1C)N(C1CCN(C(c2cc(C(C)=O)oc2)=O)C1)C 61140,C1(COC)CN(C(c2ccc([N+](=O)[O-])[nH]2)=O)CCN1C(C12CCC(F)(CC1)C2)=O 61141,CC(C)CC(CNC=O)CC(=O)NCC(C)N(C)C(c1cccc2nonc12)=O 61142,N1(C(c2cccc(OC)c2)=O)CCCC2(NC(C3CN4CCC3CC4)=O)CC2C1 61143,Cc1nc(C2CC2)[nH]c1C(=O)NC1CCCC1NC(=O)CC1CCC(C)(C)C1 61144,C1(CNC(CCOCC#C)=O)CC2(CC2)CN1C(c1ccc(Cl)c(CC)c1)=O 61145,C1(CC(=O)NC(C2CCOC2)CNCC=Cc2cocn2)(OCC)CCCCC1 61146,C12(NC(c3nccc(C)n3)=O)CCCC1N(C(=O)Cc1cc(C3CC3)no1)CC2 61147,C1(NC(CCCOCC=C)=O)CCCCN(C(=O)Cn2cc(C)ccc2=O)CC1 61148,CC(C(=O)NC(C(=O)NCc1ncn(C)n1)c1cccs1)S(N)(=O)=O 61149,c1(OC)ccc(C(N2CC(NC(=O)C=CCN3CCCC3)CC2C)=O)nc1Cl 61150,Cc1ncc(Cl)cc1C(=O)NCCOCCN(C(=O)C(F)(F)c1cnn(C)c1)C 61151,N1(CCCC(=O)NC)CCCC(CO)(NC(=O)CN2CCCCCC2=O)C1 61152,N1(C(c2c(NC)cncc2)=O)CC(CNC(=O)CC(C)(C)SC)CC(C)(C)C1 61153,Cc1ccnnc1C(N1CCC(Cn2cc(-c3ccc(Cl)s3)nn2)C1)=O 61154,C(CCF)(C(=O)N1CCCC(Cc2cn(CCCCF)nn2)C1)SC 61155,C(=O)(CC(C(F)(F)F)NC(C1CCCN1C(N)=O)=O)NC1CC(C)OCC1 61156,CCC(C)CCC(=O)NCC1(OCC)CN(C(c2cc(=O)cc[nH]2)=O)C1 61157,N1(C(C(C2(C)CC2)NC(CC2CCN(C)CC2)=O)=O)CC2(CCC(=O)N2)C1 61158,c1(OC)cc(C(=O)C(N2CC(OC)C(NC(C3(O)CC3)=O)C2)=O)ccc1Cl 61159,c1(C(=O)NC2(CNC(C(C)NS(C)(=O)=O)=O)CC2)ccc(C2CCC2)nc1 61160,C12(NC(c3nn(C)c(Cl)c3)=O)CCCC(NC(=O)C(=O)NCC(F)(F)F)(C1)C2 61161,C1(NC(C(C)=CC2CC2)=O)C2COCC1CN(C(c1nnc(O)nc1O)=O)C2 61162,N1(C(c2c(C)nc(Cl)cc2)=O)CCOC2(CCN(C(c3ccon3)=O)C2)C1 61163,CC(C)C(CNC(C1CCC(C(N)=O)O1)=O)C(=O)N1CC(S(C)(=O)=O)C1 61164,CCCCC(=O)C(=O)N(C(C)CCNC(C1(c2cccc(Cl)c2)CCCC1)=O)C 61165,CC1=C(C(=O)N2CCCCC(CNC(C3CCC3)=O)C2)CCC1 61166,C(=O)(C(N)CCCCC#N)N(C1CCCN(N(C)C(C)c2ccc(CO)cc2)C1)C 61167,C1(C(=O)NCC23C(CN(C(c4ccc(SC)s4)=O)C2)C3)CCc2nnnn2C1 61168,n1(CCC)ccc(=NC(=O)N2CCN(C(=O)C(C)(C)C(=O)OC)CC2)[nH]1 61169,Cc1noc(C)c1CN(C(=O)C(C)SC(C)C)C.c12cn(C)nc1C2 61170,Cc1conc1C1CN(C(=O)CCCC2CN(C(=O)Cc3cnsc3)C2)C1 61171,C1(CC(=O)NCCN(C2CCCCC2)C(C2CCCO2)=O)CCCCCC1 61172,C1(NC(C2(C)CCN(Cc3c(C)ccs3)C2)=O)CCC2(CCC(=O)N2)CC1 61173,C1(C(N2CC3C(NC(C4N(C)C(=O)CC4)=O)(CC3)C2)=O)CC(C)(C)SC(C)(C)C1 61174,c1(OC)cc(C(=O)NONC2=NCCCS2)c(CO)cn1 61175,c1(NS(CCC)(=O)=O)cccc(C(=O)N(CCCNC(=O)CCN(C)CC)C)c1 61176,CC1(C)CCN(C(c2cc(C3CC3)no2)=O)C(C(=O)NCC2(C)CCCO2)C1 61177,c1(C(C(=O)NC2CC(NC(C3CN(S(C)(=O)=O)C3)=O)C2)OC)c(F)cccc1F 61178,c1(C(N2CCCC(CN(C(=O)C(O)COC)CC)C2)=O)cnc2cc(C)ccn12 61179,C(C(C(=O)NC(CC)C1CC1)NC(c1cc(CO)[nH]n1)=O)OCC 61180,C1(NC(C=CCN(CC)CC)=O)C=CCC(C(N2CC(N3CCOCC3)C2)=O)C1 61181,N12CCOC(C1)CCOCCNC(=O)C2=O.C(C(C)(C)O)NC(=O)OC(C)(C)C 61182,C=CC1(C(=O)NC(c2ccncc2)C)CCN(C(c2cnsc2C)=O)C1 61183,C(=O)(C(CCSC)OC)NCCN(C(=O)CCSc1ccccc1)CCC 61184,N1(C(c2n(CCC)ccc2)=O)CC(NC(=O)Cc2cnn(CC)c2)C(C)C1 61185,c1(C(N(CC(C)NC(c2nocc2Br)=O)C)=O)cccc(Cl)n1 61186,c1(CC)nc(C)n(C)c1C(=O)NC1C2CN(C(c3csnn3)=O)CC12 61187,C(=O)(CCC(=O)c1cccnc1)N1CC(CCCC(=O)O)(OC)C1 61188,c1(C(COC(C2C(c3cn(C)nc3)CCC2)=O)=O)c[nH]c2cccc(Br)c12 61189,C1(O)(CN(C)C(c2cc(Cl)cc(Cl)c2)=O)CCN(C(c2cn(C)c(O)n2)=O)CC1 61190,c1(CC)cc(Cl)ccc1C(=O)NC(CN(C)C(C1CCOC1CC)=O)(CO)CO 61191,Cc1cc(C(N2CCCC3(NC(=O)CCC4CCCC4)CC23)=O)cnc1C(F)F 61192,C1(C#N)(C(=O)NCC(CC=C)NC(=O)Cc2[nH]cnc2C)CCCC(=O)C1 61193,N1(C(Cc2c(C)nsc2)=O)CCN(C(=O)C(C)(C)C)CC(C)(C)C1 61194,C1(O)(CN(C(C2C(OC)CCC2)=O)C)CCCN(C(c2ccncc2Cl)=O)C1 61195,C#CC1(C(N2CC3CCC2C3)=O)CN(C(=O)CCc2ccc[nH]2)C1 61196,c1(NC(c2cnc(NC(C(CC)N(C)C)=O)s2)=O)cccc(CC(F)(F)F)c1 61197,c1(C2CN(n3cc(CCC4N(C(=O)CO)CCC4)nn3)C2)cccc(Cl)c1Cl 61198,C1(NC(C2SCCS2)=O)COC2(C1)CN(C(c1occc1Br)=O)C2 61199,C(=O)(CC(C)P(C)(C)=O)NCC12N(C(c3c(C)cns3)=O)C(CC1)CC2 61200,c1(C(=O)NC2CCC(CN(C(CC(C)(C)OC)=O)C)CC2)ccc2c[nH]nc2c1 61201,CC1CC2(CCO1)CCN(C(=O)Cc1ccc([N+](=O)[O-])cc1C(=O)O)C2 61202,C1(O)(C(C)CNC(=O)C=CC(F)(F)F)CCN(C(c2cnc(S)n2C2CC2)=O)C1 61203,N1(c2nc(C(C)C)nc(N3C4CCC3CC(O)C4)c2)CC(=O)N2CCCC2C1 61204,CCC(CC)CC(F)C(=O)NC1(C(N2CCC(NC(C)=O)C2)=O)CC(CO)C1 61205,C1(C2CCCCC2)(C(=O)NC(CNC(C(COCC)(C)C)=O)C2CCC2)CC1 61206,c1(C(=O)NCCCN(C(CC(C)C2CCCC2)=O)C2CC2)nccc(C(F)F)n1 61207,C1(CCCNC(c2c(C)scn2)=O)CCCCN1C(=O)CCc1ccncc1 61208,C1(SCC)CCc2nn[nH]c2C1.C12CCN(C1)CCN(CCC)C(=O)N2 61209,c1(C(N2CCC(N(C(CC=CCC)=O)C)C2)=O)cc(Cl)c(C)cn1 61210,c1(C(=O)NC(C2(O)CCN(C(CC=CC)=O)C2)C)cc(F)cc2cc[nH]c12 61211,N1(C(CSC(C)C)=O)CC2CC(NC(=O)C(c3ccnn3C)C)CC(C2)C1 61212,CC(C)C(C(=O)NC1CC2CCC1O2)SCc1ccccc1 61213,c1(C(N2CC(NC(C(CC)O)=O)CC2(C)C)=O)cc(S(=O)(=O)NC)c[nH]1 61214,C1(CN(C(=O)CCOC2CCC2)C)CN(C(c2c[nH]c(C#N)c2)=O)CCO1 61215,C(c1ccccc1)=C(C)C(N1CCCC1CC(=O)NCc1[nH]cnc1C)=O 61216,C(CN=c1nc(C2CC2)[nH]s1)C1CCC(NC(CCN2C(C)CCCC2)=O)CC1 61217,C1(C(=O)OC)CCCC(C(=O)NCC2(NC(=O)C(=C3CCCCC3)F)CC2)C1 61218,c1(C(N2CCC(NC(C(C)NC(COC)=O)=O)C2CO)=O)cc(O)cc(N)c1Cl 61219,C(=O)(C(C)(C)C(F)c1ccccc1)N1CCC(NC(c2c(Cl)cn(C)n2)=O)C1 61220,c1(C(N2CC(C)C(Cc3ccccc3)C2)=O)cnc(O)n(C2CC2)c1=O 61221,c1(C(N(CC(=O)OC)Cc2cn(CCCO)nn2)=O)cc(Br)cc2nc(O)[nH]c12 61222,CCC(O)CCc1cn(C(COCC)C(=O)N2CC(C(N)=O)(OCC)C2)nn1 61223,c1(C(=O)NC(C(C)NC(C(C)NC(COC)=O)=O)CO)ccc(CC2CC2)cc1 61224,CC(c1ccc(F)cc1)=CC(=O)NC1CN(C(c2ccc(C(C)C)s2)=O)C1 61225,N1(C(C(CCC)O)=O)CCN(C(C2CC(N(C)C)C2)=O)C(c2ccncc2)C1 61226,c1(C(=O)NC2C(CNC(C#CC3(CC)CC3)=O)CCC2)cc(OC)c(OC)cc1N 61227,C1(C(N(C)CCc2cccnc2)=O)CC(O)CN1C(=O)Cn1cc(Cl)cn1 61228,C1(NC(Cc2c(CC)con2)=O)CCC(NC(=O)COCC(F)(F)F)CC1 61229,c1(OC)nscc1CNC(c1ccoc1CNC(=O)CCCC1CCC1)=O 61230,Cc1ccc(C2CC2)c(C(N2CC(O)(C(C)NC(c3conc3C)=O)C2)=O)c1 61231,N1(C(C2(COC)CC2)=O)CCC2(CCN(C(=O)Cc3ccsc3)CC2)C(C)C1 61232,N1(C(C(C)N=[N+]=[N-])=O)Cc2[nH]nc(C(=O)Nc3cccc(N(C)C)c3)c2C1 61233,CCC(C#N)(CC)C(=O)N1CCC(OCC23CCC2C3)C1.C12CCN(CC1)C2=O 61234,CC(C)(CN=C(NC1CCOCC1)NCC1(C)CCCO1)Oc1ccccc1 61235,C(CC(C(=O)NCCC(C(C)C)N(C)C)NC(=O)CCNC(N)=O)SC 61236,C1(C(=O)NCc2ccc(C(C)NC(c3cnc(S)nc3)=O)cc2)NC(=O)OC1(C)C 61237,c1(C(C)(C)C)cc(C(=O)NC2CCC(CNC(=O)Cn3cnnc3O)C2)on1 61238,N1(C(Cc2cccc(C)c2Cl)=O)CC2CC1CCN2C(c1nncn1C1CC1)=O 61239,C(=O)(C(CC(C)C)N(C)C)N1CC(SC)C(NC(c2nc(C3CC3)cs2)=O)C1 61240,c1(C(N(CC(CN(C)C(c2c[nH]cc2C(F)(F)F)=O)O)C)=O)ccc(N)c(O)c1 61241,N1(C(CC(CCC)O)=O)CC2CCC1CN2C(=O)CCc1cn(C)cn1 61242,N1(C(C2CCC(CC)O2)=O)CCC(C(=O)NOCc2ccc(F)cc2)C(O)C1 61243,N1(C(c2cn(C)nn2)=O)CC(NC(=O)CNC(=O)CCF)C(O)C1 61244,N1(C(C2C3(CCN(C(c4cc(C)c(C)nc4)=O)C3)C2)=O)c2ccccc2CC1C 61245,c1(C(C)C(=O)NC2C(C(=O)OC)C2(F)F)ccc(CNC(C2(CC)CC2)=O)cc1 61246,c1(-n2cc(CNC(c3cc(-c4ccccc4I)no3)=O)nn2)c(F)cccc1Br 61247,CCCCCCC(CC)NC(C1CC=CCC1NC(c1cscn1)=O)=O 61248,CC1(NC(c2n[nH]c3c2COC3)=O)CCC(NC(C2(C)CCCCO2)=O)CC1 61249,C(C(C)(C)CCNC(=O)CCc1ccsc1)NC(C(C)OCC(C)C)=O 61250,CC12COCC1CN(Cc1nnc(CC3CC3)o1)C2 61251,CCC(=O)NNC(=O)C(C)SCC1CCC2(CC2)C(=O)O1 61252,C(=O)(C1=NN(C)C(=O)CC1)NC1CCC(N(C(c2c(C)c(N)cnc2)=O)C)C1 61253,n1(CC)cnc2c(N3CCCC(C#N)C3)[nH]c(=NCc3nn(C)cc3CO)nc12 61254,C1(C(=O)NC(CCOC)CNC(c2cnns2)=O)CC2(C1)NC(=O)NC2=O 61255,c1(C(N2C(C)CC2CO)=O)ccc2c(-c3ccc([N+](=O)[O-])cc3F)n[nH]c2c1 61256,C1(NC(C=CCNC(C2CN(C(C)C)C2)=O)=O)(CO)CC2CCCC12 61257,C1(F)(CNC(C(C2CCCO2)OC)=O)CC(CNC(=O)COCC(F)F)C1 61258,C(C)(CCN=c1[nH]c(=NCC(C)(C)N(C)C)[nH]c2ccc(Cl)cc12)OC 61259,N1(C(c2c(Cl)ccnc2Cl)=O)CCC2C(CCN2C(=O)Cc2cccc(Cl)c2)C1 61260,C1(C)(CNC(C(C)S(C)(=O)=O)=O)CN(C(c2ncc3ccccn23)=O)C(C)(C)C1 61261,N1(C(CC=C=C)=O)CCC(C)(C)C1C(=O)NC1CC2OCCCC12 61262,N1(C(C(C)OC)=O)CC=C(CNC(c2ncccc2Cl)=O)CC1 61263,c1(CNC(C2CCC(CNC(=O)C=CCO)C2)=O)cnccc1Cl 61264,N1(C(C2CC(C)SCC2)=O)C2CCC1CC(C(=O)NCCN(C)C)C2 61265,Cc1cccc(C(=O)N(CCCNC(=O)C(c2cnccn2)C)C2CC2)c1Cl 61266,c1(CC(=O)NC2CC(NC(Cc3c(C)n[nH]c3C)=O)C2)c(F)cccc1Br 61267,C(CC(C)C)(C(=O)N(C)CCOCCCN(C)C(c1ncc(C)cc1F)=O)OC 61268,N1(C(CNC(CC2C(C)CCC2)=O)O)CCN(C(=O)C(C)(C)NS(C)(=O)=O)CC1 61269,c1(C(=O)NCCCNC(N(C(C)C)C)=O)cccc(Br)c1 61270,C(=O)(CC(C(C)C)NC(c1cnncc1C)=O)N1CCC(CC)(CC)C1 61271,c1(CCCC)ccc(C(=O)OC)c(C#N)c1.C12(CC1(F)F)C(=O)NC2 61272,N(C1CCc2cc(CNC(c3csnc3C)=O)ccc21)C(c1cnc(C)[nH]1)=O 61273,c1(C(=O)NC(CNC(c2cnc(OC)s2)=O)C)sc(F)cc1Cl 61274,C1(CC)CC(OC)CN(c2nnc(COc3ccc(F)cc3)n2CC(C)(C)O)C1 61275,N1(C(C(C2CCN(C(c3c(CC)noc3)=O)C2)C)=O)CCC(CO)C(C)(C)C1 61276,N1(C(c2cnn(CC)c2Cl)=O)CCN(C(=O)CCc2ccoc2)CC1CO 61277,c1(C(N(CC(C)NC(C(C2CCOCC2)OCC)=O)C)=O)[nH]cnc1C#N 61278,N1(C(c2c(C)nsc2C)=O)C2CCC1C(C)C(NC(C1CC(C)(C)CN1C)=O)C2 61279,N1(C(=O)NCCc2n(C)c(=O)on2)CCN(CC(F)(F)F)C(=O)C1 61280,C1(N(C(c2nnc(C)n2C)COC)C(C2CCC(OC)C2)=O)CC2CCC1C2 61281,c1(NC(N2CCN(C3CCOC34CCOC4)CC2)=O)c[nH]c2cccnc12 61282,c1(C(N2CCC(CCNC(c3csc(S)n3)=O)CC2)=O)cccc([N+](=O)[O-])c1 61283,N1(C(C(CC#C)CC#C)=O)CC2CCCC(C1)N2C(=O)CC1(C(F)F)CC1 61284,Cc1cc(=NC(=O)N2CC(C)CC3(CC3)C2)[nH]n1Cc1ccc(Cl)c(Cl)c1 61285,C1(OC(C)C(N2CC(O)(C(C)(C)CNC(c3nccn3C)=O)C2)=O)CCOCC1 61286,CC(C)CC(C)C(=O)NCC1CCCN(C(C2CCCN2c2ncccn2)=O)C1 61287,C1(NC(c2nn(CC)nc2C)=O)CCN(C(=O)CCc2cscn2)C12CCC2 61288,n1(CC(=O)NCC(CNC(C2(Cl)CC2(C)C)=O)OC)cc(C)cn1 61289,c1(OCCCC(N2CC(NCCOC)OCC2)=O)cc(C)ccc1C 61290,c1(C(N2CC3CCN(C(CC(C)SC)=O)C3C2)=O)ccnc2ncccc12 61291,C1(NC(C2CC3CC3C2)=O)CCC2CN(C(c3ccc(C(F)F)cc3)=O)CC2C1 61292,c1(OC)cc(C(N2CCCC2C=CC(=O)NCC2CC2(C)C)=O)ncn1 61293,C(N=c1[nH]nc(CC)s1)C1C2CN(C(C3(CCCC)CC3)=O)CC21 61294,CCC(CCC(=O)Nc1ccc(CO)nc1)NC(=O)C(C)c1cccs1 61295,C1(C(=O)NC(C)CNC(C23CC2CCC3(F)F)=O)(OC)CCC(C)CC1 61296,c1(C(=O)NC23CC(NC(C4CCC(CC)O4)=O)(C2)C3)n[nH]c2c1CN(C)CC2 61297,CCCC(C)(O)C(=O)N1CCOCC(NC(=O)C(C(C)C)c2ccccc2)C1 61298,C1(NC(C=CC)=O)CC2CCC1N(C(c1cnn(CC(F)F)n1)=O)C2 61299,CC(C)C(CC(=O)NC1(C)CCN(C(c2cc(C#N)on2)=O)C1)c1ccon1 61300,c1(C(N2CC(C)C(NC(=O)C=CCN(C)C)CC2)=O)ccc2c(c1)C(=O)NCC2 61301,C1(C(N2CC(O)(CNC(C=C(c3ccn(C)n3)F)=O)C2)=O)CCc2ccnn2C1 61302,C1(C(=O)OCC2CC3(CC3)CO2)(CC)CCN(C(=O)NC(C)(C)C)C1 61303,C1(CCNC(C(CO)OC)=O)CCN(C(C2C3COCC23)=O)CC1(F)F 61304,CC1CC(C(=O)NCCN2CCN(CC(F)(F)F)CC2)CCS1 61305,C1(C(N(CC(=O)O)Cc2cn(C3C(C)(O)CCC3)nn2)=O)CC2(CC(=O)C2)C1 61306,C(C(C)(C)C(=O)NC1CCC(CNC(c2cc(Br)oc2C)=O)C1)OC 61307,N1(C(c2nc(C(C)OC)sc2)=O)CCC2CCN(C(c3cc(N)ccn3)=O)CC12 61308,Cc1cc(NC(C2(C)CN(C(=O)CCc3ccccn3)C2)=O)cnc1F 61309,c1(C(=O)NC2C(C(=O)NCC(c3cccc(O)c3)O)CCC2)cccc(F)c1F 61310,C(=O)(CCC(C)(C)[N+](=O)[O-])NC(CN(C(=O)C=Cc1ccccc1Cl)C)(C)C 61311,C(=O)(C1CNC(=O)c2ccccc21)NCC(C)(C)NC(c1c(C)ccc(N)c1)=O 61312,N(C(=NCC1CC1(F)F)NCC1CCCO1)C1CC(N(C(=O)COC)C(C)=O)C1 61313,N1(C(C(=O)NC(CCCCC(C)C(=O)OC)OCC)=O)CC2(C1)OC(=O)NC2C 61314,C1(NC(C2(C(N)=O)CC2)=O)CC(CNC(=O)C=CC2CCCO2)C(O)C1 61315,N1(C(c2nncc(OC)c2)=O)CC(O)CCC1C(=O)NCC1(Cl)CC1(F)F 61316,Cc1oc(C(N2CCCCC2CNC(c2ccc(C(F)(F)F)[nH]2)=O)=O)cc1Br 61317,Cc1cnc(C(N2CC3CC2C3NC(=O)Cc2cc(Cl)cs2)=O)nc1 61318,N1(C(C(F)=CCC)=O)CCN(C(C2CCCCC2(C)C)=O)CC1CS(C)(=O)=O 61319,c1(C2(C(=O)NCC(CC)(C)NC(c3conc3C)=O)CC2)ccnc(Cl)c1 61320,C(=O)(C1=C(Cl)CCC(C)C1)NCC(CCCC)NC(c1ccc(Cl)o1)=O 61321,c1(CNC(c2c(C)coc2C)=O)cc(O)nc(CNC(=O)CC(O)C(C)C)n1 61322,c1(OC)ccc(-c2ccc(N)cc2CNC)cc1COC1CC(C)C1 61323,C(C(F)(F)C(=O)NCC1(NC(=O)C(n2cc(C)cn2)C)CCCCC1)OC 61324,CC(C)CC(CNC(=O)C(C)C(F)(F)F)C(=O)Nc1ccc2nc[nH]c2c1 61325,CCC(C)(C(=O)NCC1(F)CCN(C(C2(C)COCCO2)=O)CC1)C(F)F 61326,c1(OC)cc[n+]([O-])c(C(=O)NCC(O)CCNC(=O)C2=NNC(=O)C2)c1 61327,N1(C(C(C(C)C)C)=O)CC(NC(=O)C(C)(C)C)CC1(C)C 61328,C(=O)(CC1=Cc2ccccc2C1)N1CC(CCC)N(C(C2CCNC2=O)=O)CC1 61329,C=C(C)CCCC(=O)N(C(CNC(c1ccc(OCCC)c(N)c1)=O)C1CC1)C 61330,C#Cc1ccc(C(N2CC(C3(NC(=O)C(CC4CCCC4)CC)CC3)C2)=O)cn1 61331,N1(C(C2=C(C)OCCS2)=O)CC(NC(=O)C2=CSCS2)CC2(CCC2)C1 61332,Cc1cn2cc(C(=O)NCC3(O)CCCN(C(=O)CC4CC=CC4)CC3)sc2n1 61333,N1(C(C2CCN(CC)C2)=O)CC2CCC(C1)N2C(=O)C=Cc1scnc1C 61334,N1(C(C(C=C)O)=O)CCC(CC)(NC(=O)CC(C(N)=O)NC(C)=O)CC1 61335,N1(C(C2C(C(C)C)C2)=O)CCC2CN(C(c3cn(CC4CCOC4)nn3)=O)C2C1 61336,C#Cc1nc(C(N2CCN(CCNC(C3SCCC3C)=O)CC2)=O)cs1 61337,C(=O)(C1=CCC(C)(C)CC1)NCC1CCN(C(COC(CC)C)=O)C1(C)C 61338,C1(NC(C(C(C)C)C#N)=O)CN(C(C2CC3(CSC3)C2)=O)CC2(CCC2)C1 61339,c1(NC(c2ccc(F)cc2)C(CC)C)ncc(OCC)cn1 61340,C(C)(C(O)C(=O)NCC1(CCNC(=O)CCn2nc(C)cc2C)CC1)SC 61341,C(CCCCCNC(=O)C(c1ccoc1C)C)NC(C(C)SCCOCCOC)=O 61342,C(=O)(C(Cc1ccccc1)NC(C)COc1ccccc1)NC 61343,C1(CNC(c2c(COC)cco2)=O)CC2CCC1N2C(c1cc(OC)ns1)=O 61344,N1(C(CC2(OC)CN(C(COC)=O)C2)=O)CCN(CC2CCOC2(C)C)CC1 61345,N1(C(C(C)SC(C)C)=O)CCC(C(O)CNC(=O)C(C)n2cncn2)CC1 61346,c1(C(=O)NCC2N(C(c3[nH]cc(C#N)c3)=O)CC2)cnc2ccc(F)cc2c1 61347,CC(C)CC(O)C(=O)NCC(Cc1ccccc1)NC(C1CC1(Cl)Cl)=O 61348,C1(C(=O)Nc2cncs2)CC2CC2N1C(c1cccc(Cl)c1)=O 61349,N1(C(C(CO)NC(=O)C2CC2)=O)CCCCC1C.O=CC=C1CCC1 61350,c1(OC)ccnc(F)c1C(=O)NCC12CC(CN1C(=O)C(C)OC)C2 61351,C1(n2cc(CCNC(C)=O)nn2)CCCN(C(c2csc(C(F)(F)F)c2)=O)C1 61352,c1(C(=O)NCC2CN(C(c3c(Cl)nc(OC)s3)=O)CC2C)cc2ncccn2n1 61353,Cc1ccc(C(N2CCCC(N(C)C(C3CC34CC4)=O)C2)=O)c(F)c1C 61354,c1(C(=O)NCC2CN(C(CCc3ccnc(C)n3)=O)CC2C)ccc(=N)[nH]c1Cl 61355,Cc1cc2c(C(=O)NCCCCCCN(C)C(C3CCCC3O)=O)cccc2[nH]1 61356,C(CN=c1[nH]c(=NCCN2CC3CCCCN3C2=O)[nH]c2c1COC2)OCCC 61357,CCC(C)(C)C(=O)N1CCC(C(=O)NCCN=[N+]=[N-])O1 61358,C#CCCC(O)C(=O)N(CC(C)CNC(=O)CCC(=O)N1CCOCC1)C 61359,CC(C)C(C(=O)NCC1CCCS1)n1cc(CCN(C(=O)C(C)O)C)nn1 61360,Cc1ccc(CCCCN2CCCC(n3cc(CCCC#N)nn3)C2)cc1C 61361,C1(C(N2CCC(CNC(c3cnccn3)=O)CC2)=O)CC2CCC1NC2 61362,Cc1nc(CC(N2CC(NC(c3cc(C(N(C)C)OC)[nH]n3)=O)C2)=O)co1 61363,CCC(C)(C(=O)NCCC1CC(NC(C2CC2c2cccnc2)=O)C1)C(F)F 61364,CC(C)CC(F)(F)C(=O)NC1CCCCC1CNC(=O)CCC1CCCCN1C 61365,n1(CCC)nnnc1C(c1nc(C)co1)NC(c1nnc(C)s1)C 61366,c1(C(=O)NC2CCCC(NC(C(COC)(F)F)=O)C2)cccc2c1NC(=O)CC2 61367,C1(NCCC2CC(OCC)C2)CCS(=O)C1 61368,c1(C(=O)NC(C(C)(C)NC(C(COCC)C)=O)C)cc(C)n(C(C)C)n1 61369,Cc1c(C(=O)NCC(C)CN(C(=O)C=C2CCC(C)C2)C)ncn1C 61370,C(=O)(CCC(=O)NC1CCCCC1CNC(=O)CCCN1C(=O)CCC1=O)NC 61371,C1(C(=O)NCCCCCCC)CC2(CCN1C(C1CN(C(C)=O)C1)=O)CC2 61372,C1(NC(c2c(CC)scc2)=O)CCC2(CCCN(C(=O)CCC(CF)CF)C2)C1 61373,Cc1nc(C)c(S(=O)(=O)NC(C(C)C)C2CCNC2)o1 61374,C1(C(N(c2ccc(C#C)nc2)C2CC2)=O)CCN(C(=O)CC(C=C)CC)C(C)(C)C1 61375,N1(C(c2cc3sccc3[nH]2)=O)CC2CCN(C(=O)CC34CCC(CC3)C4)C2C1 61376,c1(C(N(C2CCN(C(c3n[nH]c(C4CC4)c3Cl)=O)C2)C)=O)cc(Cl)c(Cl)cc1N 61377,C1(CC)CCCC(NC(=O)CC(C)NC(c2cn(C(C)C)nn2)=O)C1 61378,C(CCCCCNC(=O)C(F)n1ccnc1)NC(=O)CCCn1ccnc1 61379,C12(C(=O)NCCCN(C(=O)CCOC(C)CC(C)C)CC)CCCC(CO1)C2 61380,Cc1nc(C#N)ccc1NC(C1CC(F)CN1C(c1ccc(Br)cc1CO)=O)=O 61381,C1(CC(=O)NC2CC(OCC(=O)NC(CO)C3CC3)C2)CCC(=O)N1 61382,c1(C(N2C(CN(C(C3C(C)C3C)=O)CC)CCC2)=O)ccc2cccc(F)c2n1 61383,N1(C(CCC(=O)OC)=O)CC2(CCCC(CNC(c3n[nH]c4c3CCC4)=O)O2)C1 61384,CC(C(=O)N1CC=CC1CNC(c1ccc(Cn2ccnn2)o1)=O)C(C)(C)C 61385,c1(C(=O)NCCC(C)CCNC(C2CCCOCC2)=O)ccc2c(c1)C(=O)NC2 61386,Cc1ncc(C(=O)NC(C2(CNC(=O)CCN3CCCCC3C)CC2)C)c(=N)[nH]1 61387,CCC(CC)CCC(=O)N1CC2CC1CC2NC(c1sc(C)nc1C)=O 61388,N1(C(=O)C(=O)NC2CC2)CC=CC1Cn1cc(C2(O)CCC2)nn1.C1CO1 61389,c1(OC)nc(C(=O)NCC2CC3CCC2N3C(c2cc(C)c(C)[nH]2)=O)cc(O)n1 61390,C(=O)(C1=C(Cl)CCOC1)N1CCC(N(C(=O)CSCc2ccccc2)C)CC1 61391,C1(NC(C2C(C)C2)=O)CCN(C(c2ccccc2Sc2ccccc2)=O)CC1O 61392,N1(C(c2cnc(C)[nH]2)=O)CC(NC(c2cc(C(C)(C)C)nn2C)=O)C(C)C1 61393,C(=O)(N1CC(O)C(O)CO1)C1(NC(C(C)C2CCCO2)=O)CCCCC1 61394,N1(C(C2CCCN(C(N)=O)C2)=O)CCN(C(C23CC4CC2C3C4)=O)CC2(CC2)C1 61395,C1(C(=O)NCc2cscn2)CC12CCN(C(c1cnc(Cl)cc1Cl)=O)C2 61396,C1(NC(CC(C)OCc2ccccc2)=O)CN(C(=O)C(Cl)=CCl)CCC1(C)C 61397,N1(C(CC2(OC)CCC2)=O)CC2CC1CN2C(=O)CCC(C)c1nn[nH]n1 61398,C(CCC(CC)CC)NC(=NCC=C)NCC(C)(C)COC 61399,N(C(=NCC(F)(F)COCC)NC(C)C)C1CCCC(OCC)C1 61400,C1(N(C(C=CC)=O)C)CCCN(C(=O)NC2CC2c2ccncc2F)C1 61401,c1(C(N2CC(C)(CNC(C(C)OCC3CC3)=O)OCC2)=O)cnc2ccoc2c1 61402,N1(CC)CCC(CNC(C2C(C)CCN2C(C2CC(F)CN2C)=O)=O)CC1 61403,c1(C(=O)NC2(C)CN(C(C3COCCOC3)=O)C2)ccccc1OCC1CC1 61404,N1(C(=O)Cc2cc(C3CC3)on2)CC2CN(C(C3(F)CCC3)=O)CCC12 61405,c1(C(N2CCC(NC(CN(c3ccncc3)C)=O)C2)=O)ccnc(Cl)c1O 61406,c1(-c2n(-c3ccc(OC)cc3Cl)nc(C)n2)c[nH]c2c(C)c(Cl)ccc2c1=O 61407,c1(C(N(C(C)CNC(=O)CSCC(F)(F)F)C)=O)csc(C(F)(F)F)n1 61408,C1(C(N2CCC(NC(c3c(C(C)(C)C)con3)=O)C2)=O)CC2(C1)CC(F)C2 61409,C1(CC(N2CCC(CC)C2)=O)CCCN(C(c2ccc(C(C)C)o2)=O)C1 61410,n1(CC(=O)NCCC2=CCN(C(=O)C=C(Cl)Cl)CC2)nc2n(c1=O)CCCC2 61411,CC1CCCCCN1C(c1ccoc1CNC(C1COCC1(C)C)=O)=O 61412,C=CCC(C(=O)OCC)NC(=O)CC1C=CC(NC(=O)C(C)C=C)C1 61413,c1(C(=O)NC(C2CN(C(CCNC(C)=O)=O)C2)C)ccnc(S)c1 61414,C1(CCC)CN(C(c2sccc2F)=O)CC1NC(=O)CN(CC)CC 61415,CCC(C(=O)NC1(C)CCC(NC2(CC(=O)NC3CC3)CC2)CC1)C(C)(C)CC 61416,N1(C(CCCC(N)=O)=O)C2CCCC1CN(C(=O)CCN1CCCC1)CC2 61417,Cc1cc(CNC(N2CCC(C)CC2C(C)O)=O)cnc1C 61418,C(=O)(C(C)(O)CC=C)N1CCCC(C(CC(=O)NCC(=O)NCC#C)C)C1 61419,N1(C(C2CCC(NC(c3ccccc3)=O)C2)=O)CCCCCC1C(=O)O 61420,c1(C(N(CCN(C(=O)Cn2cnnc2O)C(C)C)C)=O)ccc(C(F)(F)F)cc1 61421,C1(C2CCOCC2)(C(N2CCN(C(CCC)=O)CC2CS(C)(=O)=O)=O)CC1(F)F 61422,n1(CC(=O)N(C(C)C(=O)NC(CC)C(C)O)CCC)ccc(C)n1 61423,Cc1nsc(C)c1NC(C1(NC(=O)CC(=O)N(C)C)CC(F)C1)=O 61424,N1(C(C2CC(C)(F)C2)=O)CCC2C(C1)NC(=O)CN2C(c1ccc(O)c(Cl)n1)=O 61425,c1(CN2C(CC(=O)Nc3nc(C)c(C)s3)COCC2)cnc(Br)c(F)c1 61426,C1(CC(N2CC(NC(C(C3CC3)OCC)=O)C(C)C2)=O)C(=O)N(C)N=C1C 61427,C1(C(=O)NC(CCNC(c2c(CC=C)cccc2)=O)(C)C)CS(=O)(=O)CCO1 61428,c1(C(=O)NCC(C)(C)NC(C(c2ccccc2)SC)=O)ncoc1C 61429,CC1(CNC(=O)C=Cc2ccccc2)CCC(NC(=O)COC2(C)CCC2)CC1 61430,N1(C(c2c(NCC)ccc(Cl)c2)=O)CCC(C)(C)C(NC(=O)CCC2CC2C)C1 61431,N1(C(CCC)=O)CC2CCC(NC(=O)CCC(C)c3ccccc3)CC2C1 61432,N1(C(c2nccc(C#C)c2)=O)CCN(C(=O)C(F)(F)C(C)O)C2(CC2)C1 61433,N1(C(c2cnc(CCC)s2)=O)CCC(NC(=O)C(C)Cc2cnc[nH]2)C(CO)C1 61434,c1(C(=O)NCc2c(C(=O)NC(C)C(C)(C)O)nco2)cc(C#N)n(C)n1 61435,C(=O)(C1CCCc2nc[nH]c21)CCn1c(C)c(C(=O)O)cn1 61436,N1(C(CCOCC)=O)CC2CC(NC(=O)CCOC3CCC3)CC1C2 61437,CC(C)(C)CCCCNC(C1C(CNC(=O)CCc2ccccn2)C1(C)C)=O 61438,C(=O)(C(O)P(C)(C)=O)N1CC(c2cn(C)nn2)C1.C1(COC)CCCC1 61439,Cc1c(C(N2CC(CNC(=O)C(F)C3CCC3)C(F)(F)C2)=O)[nH]ccc1=O 61440,c1(CS(=O)(=O)NC(C2CCC3(CCNCC3)O2)=O)ccc2ccccc2c1Br 61441,c1(CNCC2N(C(Cc3cn(CC)nc3)=O)CCC2)c(F)cc(Br)c(F)c1F 61442,NS(=O)(=O)C1(C(=O)NCCN(C2CCCCC2)C(C2CC(F)(F)CS2)=O)CC1 61443,C(=O)(C(F)C(C)(C)O)NCC(c1ccc(F)cc1)NC(CC1(C=C)CC1)=O 61444,CC(CCCCNC(C1CCC(=O)N1C)=O)NC(c1ccn(CCF)n1)=O 61445,c1(C(N2CCOC(c3ccco3)C2)C(=O)NCC=C)ccc2cc(Br)ccc2c1 61446,C1(=O)C(C2CCOC2)N1.C1(C(=O)NCC2(COC(C)C)CC2)(OC)CC1 61447,Cc1cccn(CC(=O)NC2CC(F)CN(C(=O)Cc3ccc(Cl)nc3)C2)c1=O 61448,N1(C(=O)C(C2CC2)NC(C23CSCC2C3)=O)CC2(CCOC2)C1 61449,C1(=O)CCCCC(=O)N(C)CC2(O)CCN1C2.C1(C=O)CCCO1.CN 61450,C12(C(N(CCOCCN(C(CC(C(C)C)O)=O)C)C)=O)CCCC(C)(C1)OC2 61451,Cc1cc(=NCCCCC#N)[nH]cc1S(=O)(=O)N1CCC(C)C1C 61452,c1(NC(c2n(CCCSCC)nnn2)(C)CC2CCC2)ccc2cnn(C)c2c1 61453,c1(C(N2CCC(CC)C2CNC(c2cncc(OC)n2)=O)=O)nc(C)ccc1C 61454,CC1(C)COC(CS(=O)(=O)Nc2ccc(C3(C)CC3(F)F)cc2)CO1 61455,c1(C(C)OC)nc(C(=O)NCC(C2CCCC2)NC(C2CC23CCC3)=O)cs1 61456,N1(C(CSCCOC)=O)CCC(C(C)(C)C(=O)NCCC(=O)NC(C)C)C1 61457,N1(C(CCC=C(C)C)=O)CCc2nc(CNC(C3(C)CC(C)=NO3)=O)sc2C1 61458,C(=O)(C(C)(C)CS(C)(=O)=O)N(CCNC(c1c(C)ncn1O)=O)C 61459,N1(C(C(CCC)OCC)=O)CCC(C2CC2)C1C(=O)NC1CCCC1CN(C)C 61460,C1(C(=O)NCC(C)Sc2cccc(-c3nn[nH]n3)c2)CC2CCC1O2 61461,C1(NC(CS(C)(=O)=O)=O)CC2CN(C(=O)Cn3cccnc3=O)CCN2C1=O 61462,C1(C(=O)NC(C(=O)OC)C2CC2)COC(CNC(=O)CCc2ccoc2)C1 61463,N1(C(=O)OCC)CCC(C)(CN2CCN(C3CCOCC3)CC2)CC1 61464,N1(C(Cc2c(C)scc2)=O)CCOCC1CCNC(C12CC(C(F)F)(CO1)C2)=O 61465,C1(CNC(c2cnn(CC)n2)=O)CC(C)N(C(=O)CCCN(C)C(C)=O)C1 61466,C1(C(=O)NCCC2(CNC(c3nsnc3O)=O)CC2)(CC)CCCC1 61467,c1(CNC(=O)C(c2ccccc2)Nc2ccccc2)ccc(S(F)(F)(F)(F)F)cc1 61468,N1(C(C(CC)(CC)CO)=O)CCC2(CCC2NC(c2cnc[nH]2)=O)CC1 61469,c1(CCN(C(=O)CCn2cc(-c3cccc(CO)c3)nn2)C)cccc([N+](=O)[O-])c1 61470,C12(C(NOCCCC)=O)CCC(CC1)N(C(c1cccc3[nH]ncc13)=O)C2 61471,C1(C(C)NC(COCC=C)=O)CCCN1C(c1csc(C(F)(F)F)n1)=O 61472,C(=O)(C(C)(C)S(C)(=O)=O)NC1C(c2n(C)ncc2)CN(C(C2CCOC2)=O)C1 61473,CC(C)(C)C(O)C(=O)NC1CC(F)CN(C(c2ccc(-n3cccc3)cc2)=O)C1 61474,C(=O)(C1=CCCC1C)NC(C1(C(N(C)Cc2cn(CC)nn2)=O)CC1)C 61475,c1(C(=O)NCc2cnc(CC)[nH]2)cc(Cl)cc(Cl)c1F 61476,C(=O)(CCCCN(C(=O)C(C1CC1)OC)C)NC(c1cccnc1)CC 61477,N1(C(c2cc(CC)ncn2)=O)CCCN(C(=O)C=CCF)C(C(C)C)C1 61478,Cc1cc(F)c(N)cc1C(=O)NCC(CC(C)C)NC(=O)CC=C(Cl)Cl 61479,N1(C(C(CC#C)NC(=O)CCC2CCC2)=O)CCC(C2CC2)C1 61480,c1(OC)cccc(F)c1CNC(C1CCN1C(c1ccc(C)s1)=O)=O 61481,c1(OC)ccccc1CNc1ncnc(NCCOC)n1 61482,N(C1c2ccccc2OCC1F)C(N(c1ccc(S(N)(=O)=O)cc1)C1CC1)=O 61483,C#CCCCC(=O)NCCCC(CO)NC(c1ccncn1)=O 61484,N1(C(c2ccc(CC)c(N)c2)=O)CC2CCN(C(c3ccc(CO)nc3)=O)CC12 61485,N1(C(C(CC)(COC)CC)=O)CC2(C=C(C(=O)NCCC(C)(C)OC)CO2)C1 61486,C(N=c1nc(N2CCC(CCO)C2)cc(C)[nH]1)C1(CCC=C)CCCC1 61487,C1(CNC(c2c(C)n[nH]c2)=O)CC2(CC2)CN1C(=O)C(C)CN1CCOCC1 61488,CCCCCC(F)C(=O)N1CCC=CC1C(=O)N(CC1CCCCC1)OC 61489,C1(N(C(C(C)=CC)=O)C)CS(=O)(=O)C12CCN(C(C1(CO)CCCO1)=O)CC2 61490,C12(CNC(c3c(C)nco3)=O)CCCC1N(C(=O)CCC1(C)CC1)CCC2 61491,c1(C(C)C)c(N2CCC(CNC(=O)C(=O)Nc3ccc(Cl)cc3)C2)ncnc1Cl 61492,c1(C(=O)NC(CN(C(=O)C(CC2CC2)OC)CC)C)cc2oc(C)cc2[nH]1 61493,C1(Nc2nc(C)nc(C#N)c2)CCC2(CC1)CN(C(C1CC1(C)Br)=O)CCO2 61494,c1(C(N(CC(O)CN(C)C(c2cc(O)ncn2)=O)C)=O)cc2c(=O)cc[nH]c2s1 61495,n1(CC(N2CCC(CN(C)C(C3C=CCC3)=O)C2)=O)cc(Br)c(O)nc1=O 61496,C1(c2n(CCSC)nnn2)(NCc2ccnn2Cc2ccccc2)CC2CCCC12 61497,C(=O)(C1=NOC2(CCC2)C1)NC(C1(CNC(C2(C)COC(C)(C)CO2)=O)CC1)C 61498,C(=O)(CCCCC(N)=O)NC(C1CCCN1C(c1cc(CN(C)C)c[nH]1)=O)C 61499,N1(C(C(C)(C)N(C)C)=O)CCC(NC(C2CN3CCN2CC3)=O)C(O)C1 61500,N1(C(C(C)O)=O)CCN(C(=O)CCc2n[nH]c(=N)s2)C(C(F)F)C1 61501,CC(C)CC(C)(O)C(=O)NC(CNC(c1ccccc1SC(F)(F)F)=O)C(C)C 61502,C1(C(C)NC(COC(C)C)=O)CCN(C(=O)Cc2cnn(C)c2)CC1 61503,C(C)(CNC(c1ccc(C)c(Cl)c1)=O)(CC(C)C)NC(C(C)OCCC=C)=O 61504,Cc1c(C(=O)NC2(C)CN(C(=O)CC3CC4CCC3C4)C2)cncc1Cl 61505,C12(OC)CCC(C(=O)NC3CCN(C(C4CC45CCCC5)=O)C3)(CC1)C2 61506,C(C(C)(C)CNC(c1ccc(F)s1)=O)N(C(=O)C(C)(C)n1cc(Cl)cn1)C 61507,C1(NC(CCc2c(OC)cccc2)=O)CCN(C(=O)Cc2ncoc2C)C12CC2 61508,C=CCC(CNC(=O)CCCF)C(=O)N(C)CCn1cccn1 61509,Cc1cc(C(=O)NC2CN(C(c3cccc4c3OCO4)=O)C2)c2c(C)noc2n1 61510,N1(C(C2C(C#N)C2)=O)CCCCC1C(=O)NC1CCCC1CF 61511,N1(C(C2(C)CCN(C)C2=O)=O)CC2CCC1C(CNC(=O)C=Cc1ccoc1)C2 61512,c1(C(N2CC3CN(C(C4CC4F)=O)C3C2)=O)cc(F)c(Cl)c(F)c1 61513,C1(CC)CN(C(=O)C(F)(F)C2(O)CCC2)CCC1NC(c1nc(C)ccc1C)=O 61514,c1(C(NOCC(=O)NCC2(CC3CC3)CC2)=O)ccncc1F 61515,C(c1nc(C)c(C)[nH]1)=CC(=O)NC(C(C(C)C)NC(C=CCCC)=O)C 61516,N1(C(CCC)=O)CCCN(C(c2cccc(N3CC=CC3)c2)=O)CC1CO 61517,n1(CCN(C(=O)CCOC2CCOC2)C)cc(-c2ncoc2Br)nn1 61518,c1(C(N2CC(CCNC(CCC(=C)Cl)=O)(OC)C2)=O)coc2ccc(Cl)cc12 61519,N1(C(c2nc(F)ccc2Br)C(=O)NC)CC2CN(C3CCC3)CC2C1 61520,C(=O)(C(O)CC(F)(F)F)NC(C(=O)OC(=O)N1CC1)C1CCCC1.C1CCS(=O)CC1 61521,C(C1=CCN(C)C1)NC(C(C1CCN(C(C2(F)CC2)=O)CC1)C)=O 61522,n1(CC)ncc(C)c1NC(N1CCSC(c2ccccc2)C1)=O 61523,n1(CC(=O)NCC(CNC(COc2ccc(C)cc2)=O)O)c([N+](=O)[O-])cnc1C 61524,C1(CNC(C(CO)N(C)C)=O)CC2(CC2)CN1C(=O)Cc1cccc(C(F)F)c1 61525,C1(C(=O)NC(C2CC(NC(c3cnn(CCO)c3)=O)C2)C)C2CC3C(C2)C13 61526,c1(C(N2CCC(C(N(N3C(CC)CCC3)C(C)C)=O)C2)=O)ccc([N+](=O)[O-])[nH]1 61527,c1(C(N2C(C(=O)NCc3cc(C)nn3C)COCC2)=O)ccc(Br)c2nsnc12 61528,c1(CCCC)ccc(C(=O)NC(C)C(C#N)CC)cc1[N+](=O)[O-] 61529,c1(C(=O)NCC(CNC(C2(CC#C)CCOC2)=O)O)cc(O)cc(F)c1F 61530,c1(C(N2CC(NC(c3ncc(C)cn3)=O)C(C)CC2)=O)cccc2scnc12 61531,C1(CC)CN(C(=O)CC2COCC2(C)C)CCC1NC(C1CCCC(=O)C1)=O 61532,Cc1nc2c(NCC3CC(CNC(=O)Cn4ccnn4)CO3)ncnc2s1 61533,Cc1c(C(N2CC(CNC(c3c(F)ccc(F)c3O)=O)C2)=O)nn2c1OCCC2 61534,C(=O)(CCCC(OC)OC)NC(C(=O)NCC(CCOC)(C)C)C1(C)CC1 61535,c1(OC)cc(F)c(CNC2CC2C(=O)Nc2cc(Br)c(F)cc2Br)cc1F 61536,N1(S(=O)(=O)CC2CCCOC2)CCC(O)C(F)(F)C1 61537,c1(C(N2CC(C(=O)NCCCc3ncc[nH]3)(SC)C2)=O)cc(C)nnc1C 61538,C1(CNC(c2n(C(C)C)ncc2)=O)CN(C(=O)C2=CCCC2)CCC1C 61539,n1(CC(=O)NCC(C2CCC2)NC(C(CC=C)(F)F)=O)cc([N+](=O)[O-])nc1C 61540,Cc1nnccc1C(N1CC2CC1(C(=O)N(CCC(C)C)C)C2)=O 61541,c1(CC)cc(C(=O)NC2CCCCC2NC(C2CCC(=O)N(C)C2)=O)ccc1O 61542,c1(C(N2CCC(O)(CNC(c3cncc(C)c3Cl)=O)C2)=O)noc2c1CCCC2 61543,N1(C(C2(C3CC3)CNC2)=O)CCCC12CCC2 61544,C1(C(N2CC(C#N)C2)=O)CC(F)(F)CN1C(c1cccc(O)n1)=O 61545,c1(CN(C)C(C2C=CCCC2)=O)cnn2c1CN(C(c1cc(CO)[nH]n1)=O)CC2 61546,c1(C(=O)NC2CCCN(C(c3c(C)cccc3O)=O)CC2)ccc2ccsc2c1 61547,CC(C)C(C)CC(=O)NC1CCCC(NC(c2ccoc2C2CC2)=O)C1 61548,c1(OC)cccc(C(N2CCN(C(=O)C3=C(C)OCC3)C3CC23)=O)c1C 61549,C1(NC(c2ccnc(-c3cccc(C(F)(F)F)c3)c2)=O)COC2(CCC2)C1 61550,c1(OC)ccc2[nH]cc(-c3ccc(C(=O)Nc4nc(SC)ncc4Cl)nc3)c2c1 61551,c1(N2C(C)CN(C(C3CCS3(=O)=O)=O)CC2)nc(Cl)nc2ccc(Cl)nc12 61552,CON=Cc1ccc(C(=O)N(CCC(C)NC(C2(C(F)F)CC2)=O)C)cc1 61553,C#CCC(CC#C)C(=O)N1CCC2(C1)CN(C(C1CC(O)(C#C)C1)=O)C2 61554,N1(C(C(C=C)(F)F)=O)CCC2(CC1)OC1(CO)CC2(NC(c2cncn2C)=O)C1 61555,c1(C(C(=O)N(CC(CNC(C2(n3ccc(C)n3)CC2)=O)O)C)C)ccccc1Cl 61556,C(=O)(C1CCSc2ccccc21)NC(C(C)C)CN(C)C 61557,c1(OC)cnnc(C(=O)NCCCCC2CN(C(C3(O)CCSC3)=O)C2)c1 61558,CC1CN(C(C2CCS(=O)(=O)CC2)=O)CCC1NC(=O)CC=CC(C)(C)C 61559,C(C)(C)(CCF)N(C(C(C)=CCC)=O)CCOCC 61560,N1(C(C(C)SCc2ccccc2)=O)CC(NC(=O)CC(C)(O)C2CC2)C(C)(C)C1 61561,c1(OC)ccccc1C(=O)NC(CN(C)C)C(=O)NCC(N1CCCC1)=O 61562,Cc1nnc2c(C(N3CC(NC(=O)Cc4cncs4)CC34CCC4)=O)cccn12 61563,C1(CC(=O)NC(CNC(CC(C)C)=O)C(C)C)CCCCCO1 61564,CCC(CCCC(=O)NCC1(F)CC(CO)C1)NC(c1cccc(CC#N)c1)=O 61565,c1(CC(=O)OCC(=O)N(C(C(C)=O)Cc2ccccc2)C2CC2)cc(Cl)sc1Br 61566,C1(CNC(C(=C(C)C2CC2)F)=O)CN(C)CCN1C(C1CC1(C)C(F)F)=O 61567,[N-]=[N+]=NCC(F)CCNC(C1CC=CC(NC(c2ncncc2Cl)=O)C1)=O 61568,Cc1oc(C(F)(F)F)nc1C(=O)NCC(C)CNC(C1CC1(Cl)Cl)=O 61569,c1(CNC2C(C(N(CC)Cc3cccc(Br)c3)=O)C2)c[nH]c2cc(Br)ccc12 61570,O(NC(=O)C(F)C1CCCN1C(=O)Cn1[nH]cnc1=N)CCC 61571,CC1CN(C(c2ncc(F)cc2F)=O)CCC1NC(c1nn[nH]c1Cl)=O 61572,C1(C(=O)NCC(CC)NC(c2cc(CCO)on2)=O)CCC(O)CN1C 61573,Cc1ccc(NC(N2CCCC(C(C)(C)C)CC2)=O)c(O)n1 61574,N1(C(C2N(C(C(N3CCSCC3)C)=O)CSC2)=O)C2CCC1CC(CO)C2 61575,C1(C(N2CC3(NC(C(CC)C)=O)CC2(COC)C3)=O)CCc2nc[nH]c2C1 61576,Cc1nccnc1C(C(=O)NC1CN(C(=O)OC(C)(C)C)C1)N(C)C1CC1 61577,C1(NC(c2c(C)non2)=O)CCC(N(C(=O)CC2CCCOC2)CC2CC2)CC1 61578,C1(C(=O)NCC2N(C(CC(=O)NC3CC3)=O)CCC2)CC12CCc1ccccc12 61579,C(=O)(C1=CCCOC1)NCC(C1CCN(C(c2c[nH]cc2C2CC2)=O)CC1)C 61580,CC1CC(NC(C2(C)CCOCC2)=O)CN1C(=O)Cc1ccn(C)n1 61581,C1(N(C(=O)CCc2cn[nH]c2)CC2CC2)CCCN(C(=O)CC2CCOC2=O)C1 61582,c1(C(=O)NC(C)CCCCNC(c2ccco2)=O)n[nH]cc1[N+](=O)[O-] 61583,CC(CSc1ccc(Cl)s1)C(=O)NC1CCCC1 61584,c1(N(CC(=O)NCC(C)NC(=O)C(C)(O)c2ccccc2)C)ccccc1 61585,C#Cc1cncc(C(=O)NC2CC(N(C(=O)CCSCc3ccccc3)C)C2)c1 61586,CCC(C)C(CC(=O)NC1CC(C2CC2)C1)NC(=O)COCC(=O)NC 61587,c1(C2CCCN(C(C(=O)NCCCSC)c3ccns3)C2)ccccc1C#N 61588,CC(Cc1ccccc1)C(=O)N(CC(O)CNC(C1CCCC1)=O)C 61589,N1(C(C(C)(C2CC2)NC(C)=O)=O)CCC(CN(C(=O)C(C)CC2CCC2)C)CC1 61590,c1(N(C)Cc2nccs2)nc(=N)nc(NCC(c2ccccc2)(C)F)[nH]1 61591,C(CC(C(=O)N1CCCC(OCC)C1)NC(=O)CCCSC)OCC 61592,N1(C(C(CCSC)O)=O)CC2CCCC(CNC(C3CC(C)(C)CCO3)=O)C2C1 61593,C1(C(=O)NCCCC(C)C)CC(NC(=O)CCC2(C)CC2)CCO1 61594,C1(C(N(CCCNC(C(C)(C)OCC)=O)C)=O)CC(N=[N+]=[N-])C1 61595,C1(NC(CC=CC)=O)CC(NC(C2CCC(CCCCC)CC2)=O)CC1O 61596,C#CCC(CC(=O)N1CC(C)(C(=O)OC)C1)NC(C1(OC)CCCOC1)=O 61597,C#Cc1ccc(C(=O)NC2CC(C)CN(C(c3cnc(O)o3)=O)C2)c(OC)c1 61598,c1(C(=O)NC2(C)CN(c3c(OC)c(C)ncn3)C2)noc2ccc(Cl)cc12 61599,Cc1ccc(F)c(C(=O)NCC(C(=O)N2CCC(C(F)F)CC2)C(C)C)c1 61600,N1(C(C2C(CCOC)C2)=O)CCC(F)C(NC(c2cscc2C)=O)C1 61601,C1(CC)(NC(C2CCCOC2)=O)CCN(C(c2ccc(F)c(CO)c2)=O)CC1 61602,C(=O)(CC(=O)NCCn1cc(CC(C)O)nn1)NC 61603,C1(C)(SCC2CCCN(C(=O)NCCn3c(C)csc3=O)C2)NC(=O)NC1=O 61604,Cc1cc2ncc1S(=O)(=O)N2.N1(CC(C)N(C2(C)CC=CC2)C)CCCCC1 61605,CC1(C)CCC(C)(C(=O)NCCOCCNC(=O)Cc2ccccc2O)CC1 61606,CCCCCC(O)C(=O)NCCN(C(=O)CC1CC(=O)NC1=O)C 61607,C(=O)(CCCC(=O)NCCC1CCCN(C(C2CC3C=CC2C3)=O)C1)N(C)C 61608,c1(C(=O)NC(CN(C(C(COC)(C)O)=O)C)C)coc2c(F)cccc12 61609,c1(C(N2CCCC(F)(CNC(C(C)=C3CC3)=O)C2)=O)cccn2nccc12 61610,N1(C(C(=O)NCc2cccc(OC)c2)c2ccns2)CCSC2COCCC12 61611,c1(CC(=O)N(C)C)ccc(C(=O)NCC2CCN2C(=O)CCn2cncn2)cc1 61612,C12(C(=O)NC(CN(C(C(C)NS(CC)(=O)=O)=O)C)C)CC=CC(C1)OC2 61613,c1(C(N2CCC(OCCNC(C(C)S(N)(=O)=O)=O)C2)=O)cc2cc[nH]c2cn1 61614,c1(C(=O)NC2CC(CNC(c3ncn(CC)c3)=O)C2)c[nH]c2ccccc2c1=N 61615,N1(C(c2ccc(N(C)C)nn2)=O)CCC2CN(C(=O)C=Cc3ccncn3)CC12 61616,c1(CC)nc(C)cc(=NCC2CN(C(c3cnn(CC(F)F)c3)=O)CC2C)[nH]1 61617,c1(C(C(=O)OC(CC=C)C)OC(=O)CC(C)n2ccnc2)cccc(F)c1 61618,CC1C(CO)CCCN1CC(=O)Nc1cccc(OC(F)(F)C(F)F)c1 61619,C(=O)(C1=CC(O)C(NC(c2ccc(C)c(F)c2)=O)C1)NCC1CC(OCC)C1 61620,C(=O)(C1=CCCCCC1)N1CCCN(CCNC(C(n2cc(Cl)cn2)C)=O)CC1 61621,C1(C(N2CC(C3N(C(C(OC)OC)=O)CCC3)(O)C2)=O)CC(C)CCO1 61622,C(C(O)C(=O)NC1CCC(CCC(=O)NCCN(CCCF)C)C1)=CC 61623,N1(C(C(C)O)=O)CCCC(NC(C2CC3C=CC2C3)=O)CC1 61624,c1(OC)ccc2c(ccn2CC(=O)NCC(CNC(=O)Cc2ccsn2)OC)c1 61625,Cc1cc(C(=O)NC(C2(O)CCCCC2)C(=O)NCC2(F)CC2)n(C)n1 61626,c1(OCC(=O)NC(C2(OC)CCOCC2)CC)ccc(C(F)(F)F)cc1Br 61627,c1(OCC)cnc(C(=O)N(C2CCCC(NC(c3cc(C)cs3)=O)C2)C)c(Cl)c1 61628,Cc1cc(C(C)NC(c2oc(C3CCCNC3)nc2C)=O)ccc1Br 61629,C1(NC(C2CC(SC)C2)=O)CCCCCCC1NC(=O)CC(C)C(F)F 61630,C1(CNC(C2(CC#C)CCCO2)=O)CN(C(c2ncc(CCC)s2)=O)CC1C 61631,N1(C(c2ccccc2)CC)C(=O)C2CSC(C)N2C1=O.C1(=O)CO1 61632,C1(C(=O)NCC2N(C(C(c3ccc(C)o3)C)=O)CC=C2)CC(S(C)(=O)=O)C1 61633,c1(N(CCNC(C)=O)C)cccc(S(=O)(=O)NC2CC2C)n1 61634,C(=O)(C(F)CC(C)(C)NC(=O)CCC(C)(C)N(C)C)N1CCN(CCCC)CC1 61635,c1(C(C)C(=O)N(C)CCNC(=O)CN(C2CCSC2)C)c(F)cccc1F 61636,N1(C(CC(C=C)CC)=O)CC2=C(C1)CN(C(C1CC(OC)C1)=O)C2 61637,C1(C)CC(N(CC(=O)NC2CCCCC2)C)C(=O)N1C.C1(CO)(O)CCC1.CS 61638,N(C(=NCCNC(c1cccs1)=O)NCC(F)F)C1CC(OC)C1 61639,c1(C(C(=O)NCCCSCC)N(CC(C)C)CC#N)cc(Cl)cc(Cl)c1 61640,C#Cc1cccc(CC(=O)Nc2nc(SC)ns2)c1 61641,CC(C)CC(C(=O)N1CC(NC(C2CCC=CO2)=O)CC(C)(C)C1)C(C)C 61642,CC(C)C(=O)C(=O)N(C)CC1CCN(C(c2ccnc(C3CC3)c2)=O)C1 61643,N1(C(C(CCCNC(c2c(F)ccc(C)n2)=O)(C)C)=O)CCC2CCC(O)C1C2 61644,C1(NC(COCCOC)=O)CC2(CCCN(C(=O)CC3CCC(F)(F)CO3)C2)C1 61645,CCC(O)C(C)C(=O)NCC1CC(NC(=O)C(=Cc2cccs2)C)C1 61646,c1(C(=O)NC(CC)(C)CNC(C2CCN(C)CC2)=O)nc(OC)cc(OC)n1 61647,C=CCCC(C(=O)NC(C)C(C)(C)CO)NC(=O)CCCCNC(N)=O 61648,n1(CCOC)nccc1C(=O)NCC1(F)CN(C(=O)C(O)CC2CCCCC2)C1 61649,C1(C(=O)OCC)CCC(C(=O)NCC2CCN(C(c3sccc3C(C)C)=O)C2)C1 61650,C1(CNC(c2csc(C(F)(F)F)n2)=O)CCN(C(C2CCS2(=O)=O)=O)C12CC2 61651,c1(-n2cc(C3CN(C(C(C)Sc4ccccc4)=O)C3)nn2)ccc(F)cn1 61652,N1(C(C23OCC(C(=O)OC)(C2)C3)=O)CCC2(C1)CN(C(=O)C(C)O)C2 61653,Cn1cnc([N+](=O)[O-])c1NC(=O)C(N1CCC(CCCN2CCOCC2)CC1)=O 61654,CC1CC(CO)CN(C(c2ccn(C3CC3(F)F)n2)C(=O)NCC(F)F)C1 61655,C1(NNC(C2N(CC)CC2)=O)C2CC3C(C2)C13C(N1CC(N2CC(O)C2)C1)=O 61656,Cc1noc(C)c1C(=O)NCC1(F)CCC(NC(C2(CO)CCC2)=O)C1 61657,c1(C(N2CCCC(C)(CNC(C(C(C)C)F)=O)C2)=O)cc2cc(Cl)c(Cl)cc2[nH]1 61658,N1(C(C2(OC)CCOC2)=O)CCC(F)(CNC(=O)CC2CCCC(=O)C2)CC1 61659,C1(CCNC(C=C(C)Cl)=O)CN(C(=O)CCCc2ccsc2)CCS1(=O)=O 61660,c1(C(=O)NC(CCNC(C2CC(C)C2)=O)C)cccc(S(C)=O)c1 61661,c1(C(C(=O)NC2(CC(=O)NC(CSC)C)CCC2)F)ccccc1 61662,N1(C2CCN(C(C3(NC(C)=O)CC3)=O)C2)CCN(CC2CC(C)(C)CO2)CC1 61663,c1(C(=O)OCC(c2cc(Cl)cc(Cl)c2)=O)cccc2snnc12 61664,CC1CCCC(C)N(C(=O)CC2CCN(C(C3CCC3C)=O)C2)C1 61665,c1(C(=O)NC(C(C)NC(C2CCCS(=O)(=O)C2)=O)CO)ccc2ncccc2c1 61666,CN1CCN(CC(=O)NCC2CCCCN2C(C2CC(C)(F)C2)=O)CC1 61667,CC(C)C(Cc1ccccc1)C(=O)N1CC(CCNC(C2CCNC2=O)=O)C1 61668,C1(NC(Cc2c(C)cccc2F)=O)CN(C(=O)Cc2cscn2)CCC1(C)C 61669,Cc1ccc(C(=O)N(CCCNC(=O)CC2(C)CC2(F)Cl)C(C)C)c(O)c1 61670,Cc1nn(C)cc1C(N1CC(C(C)NC(=O)C=C(Cl)Cl)C1)=O 61671,n1(C(C)C)nccc1-c1cn(CC2CCN(C(=O)CSc3nnnn3C)C2)nn1 61672,CC(=O)C(C)CC(C)C(=O)N1CCCCCC(NC(=O)CCSCC(N)=O)C1 61673,Cc1nn(C)c(C)c1CC(=O)NCC1CCC(C)CN1C(=O)CCc1cnc[nH]1 61674,CCC(C(=O)NC(CCCNC(=O)Cc1cnns1)c1ccccc1)SC 61675,c1(CC)ncc(C(=O)NC2CCC(CCNC(=O)CC3CC(F)(F)C3)C2)[nH]1 61676,Cc1ccc(C(N2CC(NC(c3cc(C)c(C)s3)=O)C3CC23)=O)cc1C 61677,c1(C(N2CCC(NC(C3(CC=C)CCCC3)=O)C(C)C2)=O)c(C)ncn(C)c1=O 61678,C(=O)(CCCC(=O)NCC1(C)CC(NC(c2cc(OC)ccc2N)=O)C1)NC 61679,C(=O)(C1Cc2ccccc21)NCC(CNC(c1cc(C2CC2)ccc1F)=O)O 61680,c1(-c2cn(CCN(C(C(C)Sc3ccc(C)cc3)=O)C)nn2)cc(Cl)ccc1O 61681,C(=O)(CN=c1cc[nH]cc1)N1C(C(C)(C)NC(C2C(C)SCCC2)=O)CCC1 61682,C1(NCCCC(c2ccccc2)NC(c2c(C)ccnc2)=O)CCC(C)(C)CO1 61683,C(CC(C)N=c1nc(COC)[nH]s1)NC(C(CC)CCOC)=O 61684,N1(C(C2(C)CCCN(C(=O)CC(F)(F)F)C2)=O)CC2CCNCC2C1 61685,C=CCC(CC)C(=O)NC1(c2ccccc2)CN(C(=O)CC(C)C(F)F)C1 61686,CC1CC(Nc2ncncc2Cl)CCN1C(=O)C(O)C1CC1 61687,N1(C(c2c(C)c[nH]n2)=O)CC(C2CCCCN(C(C3(F)CCOC3C)=O)C2)C1 61688,CC#CCCCC(=O)N1CCC(N(C(C2(OC)CC2)=O)CCC)C1 61689,C(CN=c1cc(C)nc(N2CCC(NS(C)(=O)=O)C2)[nH]1)(C1CCC1)OC 61690,C1(CNC(C2(N(C)C)CCCC2)=O)CN(C(=O)CCC2CC(C)(C)CO2)CCO1 61691,N1(C(c2c[nH]c(=NCC)s2)=O)CCCC1C1CCCCN1C(=O)CCCF 61692,S(=O)(=O)(c1cccc(F)c1)N1C(C(=O)Nc2cccc(C)n2)CC2CC21 61693,C(=O)(CP(C)(C)=O)NCC(C)CN(C(=O)C(C)(C)Oc1ccc(Cl)cc1)C 61694,CCCC(O)C(CO)NC(C1CCCCCC1NC(c1ccc(CO)cn1)=O)=O 61695,C(=O)(N=c1[nH]nc(CC(C)C)s1)C1(CC#C)CCCCN1C(=O)OC 61696,n1(CCC(=O)NC(c2c(OC)cccc2)c2cccs2)cnc(C)cc1=O 61697,c1(OC)ccc(F)c(OC)c1C(=O)NCC(C)NC(=O)CCCNC(C)=O 61698,c1(C(=O)NC2CCC(NC(c3ccc(CC)c(N)c3)=O)C2)cncc2c1CCC2 61699,C1(NC(C)=O)(CO)CCN(C(c2cccn(C3CCC3)c2=O)=O)CC1 61700,CC1(C)CCN(c2nc(Cl)ncc2C2CC2)CC1CNC(c1ccc(F)cn1)=O 61701,c1(CC(N2CCC(NC(c3scc(C)c3)=O)C2C2CC2)=O)ccc(O)c(Cl)c1 61702,c1(CC)ncnc(NC(CNC(=O)CCN2C(=O)CCC2=O)CC)c1F 61703,C1(F)(CNC(C2(C)CCC2)=O)CCCN(C(=O)CC2(C)CCOCC2)C1 61704,C1(NC(CCOC(C)C)=O)CC2CC1CN(C(c1ncccc1Br)=O)C2 61705,C1(C(N(C2CCN(Cc3nc(CC)on3)CC2)C)=O)CCCN(CP(C)(C)=O)C1 61706,c1(C(N2C(COC)CN(C(C3(C)CCCN3C)=O)CC2)=O)cc(C)c(C)nc1C 61707,C1(O)(CC(=O)OCC)CCN(S(=O)(=O)Cc2[nH]ccc2CC)C1 61708,c1(C(=O)NC(C(C)NC(c2ccc(CCF)cc2)=O)(C)C)cnn2ccncc12 61709,C(=O)(C(CCCC(=O)OC(C)(C)C)N1CCC2C(O)C(C)(C)C12)NCCCC 61710,C1(F)(C(=O)NC(c2c(C)nccc2)C)CCN(C(=O)C(C)CC(N)=O)CC1 61711,S(=O)(=O)(c1nc(Br)cs1)Nc1c(OCC)c(F)ccc1 61712,CC(C)(CC1CC(F)(F)C1)C(=O)N1CC(NC(C2CSCCS2)=O)C(CO)C1 61713,N1(C(c2cc(CCC)[nH]n2)=O)CCN(C)C(C(=O)NC2CCC3CC2CO3)C1 61714,c1(C(=O)NC2C(CNC(c3cnc(OCC)s3)=O)C2)ccccc1C(N)=O 61715,c1(OC)noc(C)c1C(=O)N(C)CC1(O)CCN(C(=O)C(c2nc(C)cs2)C)C1 61716,Cc1ccc(CCC(=O)N(C(C)CCNC(=O)C(C(C)C)NC=O)C)cn1 61717,C1(OC(C(C(CC)C)O)=O)CC(=O)OC12CCCCC2 61718,c1(CC)n[nH]c(COC(C)(C)C)n1.c1(C2C(C)NC(=O)N2)ccccc1 61719,C1(COC)CN(C(c2cnn(C)c2C)=O)CCN1C(c1ncccc1Br)=O 61720,c1(OC)cc(CNCc2ccncc2C(F)(F)F)cc2cc(C)oc12 61721,c1(C(C)(C)C)nc(C(=O)NC2CCCC2C(N2CCC(Br)C2)=O)co1 61722,N1(C(CCSCC=C)=O)CCCC(NC(=O)CCNC(=O)NC)C1 61723,C1(C(N2CC(O)(CC)C2)=O)COCCN(C(=O)C(CC2CCCC2)NC(C)=O)C1 61724,C(=O)(C(C)CC(C)C)N1CC(C(=O)N(C)Cc2cnccn2)(COC)C1 61725,C(C(=O)N1CC(O)(CNC(C2CC(n3cnnc3)C2)=O)C1)(C(C)(C)C)N(C)C 61726,C12(C(N3CC(C)(NC(c4ccn(C(C)(C)C)n4)=O)C3)=O)CCCC1CS(=O)(=O)C2 61727,C(=O)(CCC(C)(C)C(=O)OC)NCC(CC)NC(C1(C)CC2CC2C1)=O 61728,C(=O)(C(C)(CCc1ccccc1)CC)N(C)CC1(CNC(C(=O)N(C)C)=O)CC1 61729,N1(C(C(N2CCCS2(=O)=O)C)=O)CCCCC1CNC(c1ccncc1F)=O 61730,c1(CC(=O)NCC2(F)CC(NC(=O)CSc3ccccn3)C2)ccccc1O 61731,CN1CCN(C(=O)C(C(C)(C)C)NC(c2csc(C#N)c2)=O)CC1(C)C 61732,c1(OC)cc(C(N2CC(NC(C3CCOC3(C)C)=O)C(O)C2)=O)cc(N)c1O 61733,Cc1ccn(C)c1C(=O)NCC1(CNC(=O)CC(O)C2CCCC2)CC12CCC2 61734,c1(SCC(=O)NCCN(C(C2C(C)(COC)C2)=O)CCSC)cc(F)cc(Cl)c1 61735,N1(C(C(N2CC(C)(CO)C2)=O)=O)CCCOCC1 61736,c1(CN(c2ccc(OCCC(=O)OC(C)(C)C)cc2)C)cccc(F)c1F 61737,N1(C(=O)C=C2CCCC2)CCC2(CCCN(C(=O)Cc3ccc(O)nc3)C2)CC1 61738,c1(NC(CNc2cc(OC)c(Br)cc2)=O)cc2c(OC)c(F)ccc2[nH]1 61739,S(=O)(=O)(c1ccn(C2CC2(F)F)n1)NCC1(C)CNCCC1O 61740,C1(C(N(CC(COC)O)C)=O)CCCN(C(=O)C(C)N(C)C)C1 61741,N1(CCC)CCN(C(C2(OC)CCN(C(c3ccc(F)cn3)=O)C2)=O)CC1 61742,n1(CC)nnc(C)c1CNC(C1(CCCO)CCCC1)=O 61743,C12(C(=O)NCC(CN(C)C(C3(CCF)CCC3)=O)O)COCC1C2(F)F 61744,c1(C(=O)NC)cccc(C(=O)NCC2(O)CCN(C(=O)CCOCCOC)C2)c1 61745,c1(NC(C(C)C)=O)ccccc1C(=O)NC1CCC(NC(c2ncccn2)=O)C1 61746,C1(O)(C(CNC(C2(OC)CC2)=O)C)CCN(C(=O)C(C)(C)c2ccnn2C)C1 61747,N1(C(C2(CC)CCCN2C(C2CCC(C)(C)C2)=O)=O)CC2CC1CN2C 61748,c1(C(=O)NCC2C(C(=O)NCC(C)(C3CC3)OC)CCO2)nccc2cc[nH]c12 61749,C(=O)(C(F)C(CC)CC)NC(CN(C(C(C)OCC=C)=O)C)C 61750,N1(C(C(C2CCC(O)CC2)(C)C)=O)CCC(C)(NC(c2ncccc2N)=O)CC1 61751,C1(C(=O)NCC2CN(C(CC(C=C)C)=O)C(C)(C)C2)CC2CCC1C21CC1 61752,Cc1ncc(C(N2CCCCC(CNC(C3CC3C3CCCO3)=O)C2)=O)cc1N 61753,C1(COC)(CNC(=O)C(C)n2cccn2)CN(C(c2cn(C(C)(C)C)nn2)=O)C1 61754,C1(NC(COCC=CC)=O)CCC12CN(C(c1ccc(NC(=O)C(C)C)cc1)=O)C2 61755,c1(Cc2n(C)cnn2)cc(NC(=O)NC(CO)CC(F)F)ccn1 61756,C1(CNC(C2COCOC2)=O)CCCCN(C(=O)C(F)=CC2CC2)C1 61757,C1(C(=O)NC(CC)C2CC2)(CO)CCN(C(c2ccc[n+]([O-])c2)=O)C1 61758,C1(CCNC(C=COCC)=O)CN(C(=O)CCc2scnc2C)CCCO1 61759,c1(OC)cc(CN2CCCC2)ccc1C(C)NC(c1ccnc(O)c1)=O 61760,N1(C(C(C)(C)O)=O)CCC(c2ccccc2)C(NC(C2(S(C)(=O)=O)CC2)=O)C1 61761,CCC(F)(F)CC(=O)N1CC(CO)(NC(=O)C2=C(Cl)CC2)C1 61762,c1(C(=O)NCC(C2(O)CCN(C(CC3(C=C)CC3)=O)C2)C)cc(OC)cc(Cl)c1 61763,c1(C(=O)NC2CCCN(C(CN3CCC(C)CC3)=O)C2)cc2c(s1)CCC(C)C2 61764,C1(C(=O)NCC(CNC(C(CCC)(C)C)=O)(C)OC)CCc2cnnn2C1 61765,c1(C(=O)NC2CC(c3ccccc3)(NC(C3CCCO3)=O)C2)ccc(C(F)F)s1 61766,c1(OCC)ccc(C(=O)NCCCN(C(=O)CCn2ncn(C)c2=O)CC)cc1 61767,C1(N(C)C(C2CCCN2S(C)(=O)=O)=O)CC2CC1N(Cc1ccc(Cl)c(F)c1)C2 61768,CC1(C)CC1(Cl)C(=O)NCCC1CCCN1C(c1cnn(C2CCCCC2)c1)=O 61769,C(C(C)C(=O)NCC(C)N(C(=O)Cc1[nH]cnc1C)C)OCC 61770,c1(C(N2C3C(NC(c4cccc(C)n4)=O)CC(C3)C2)=O)coc2c1C(O)CCC2 61771,S(=O)(=O)(c1c[nH]c(C(N2CCN(C(=O)CN3CC=CC3)C(CO)C2)=O)c1)NC 61772,N1(C(c2nnn(CC)c2C)=O)CCN(C(=O)C=CSC)CC1CF 61773,c1(NCCNC(=O)NC2(C(C)C3CC3)N=N2)cccc(Br)n1 61774,N(C1CC2CCC(C)(C)c3cccc1c32)C(c1c(F)ccc(OC)c1N)=O 61775,C1(CN=[N+]=[N-])CCN(C(c2cn(CCNC(c3c[nH]c(=S)cn3)=O)nn2)=O)CC1 61776,C(C)(CNC(c1cnc(S)nc1)=O)(CC(C)C)NC(CC(=O)NCC)=O 61777,c1(COC)ccc(C(=O)NC2CN(C(=O)C(C)SCc3ccccc3)C2)[nH]1 61778,C(=O)(C(C)CCCC(C)=O)NC(C(=O)NCC1(OC)CCOC1)c1ccco1 61779,C1(N(C(C2C(CC)CC2)=O)CC)CCC(NC(=O)C(CC2CC2)OC)CC1 61780,c1(NC(C(C)C)=O)ccc(C(=O)OC2COCC2F)cc1 61781,Cc1cc(CCNC(=O)CCN(C)C)cc(Cl)c1 61782,C1(NC(CC(=C)Br)=O)CC2(C1)CN(C(=O)C=Cc1ccccc1F)C2 61783,CC1CCCn2ncc(C(N3CC4C(CNC(C5(C6CCC6)CC5)=O)C4C3)=O)c21 61784,c1(C(N(C)CC2(NC(C(c3ccc(Cl)cc3)C)=O)CC2)=O)csc2c1CCCC2 61785,C1(C(=O)NC(C)CC#N)CCCCN1C(=O)Nc1ccccc1Cl 61786,c1(CCC(=O)NCCC(N2CCN(C(C3C(=C)C3)=O)CC2)=O)nnc(S)nc1O 61787,C(=O)(C1=NOC(C)(C)C1)NC1N(C(C23CCCC2(C(N)=O)C3)=O)CCC(C)C1 61788,C1(C(N2CCC(NC(C=C(C)C)=O)C(O)C2)=O)CCc2nnc(C)n2C1 61789,C1(CC(=O)Nc2cn(CCC#C)nc2)CCCN(C(C2CCOCC2)=O)C1 61790,N1(C(CC(C(C)C)C)=O)C2CCC1C(C)C(NC(C13CC(CC(F)F)(C1)C3)=O)C2 61791,C1(CNC(C2(C#C)CC2)=O)C2CN(C(c3cc(COC)[nH]n3)=O)CC12 61792,c1(OC)cc(C(=O)NC(C)C(C)NC(c2cnc(C(C)C)n2C)=O)cc(F)c1F 61793,c1(OCC)cc[nH]c(=NCCC(C)NC(=O)C=Cc2cncs2)n1 61794,N1(C(=O)COc2ccc(Cl)cc2Cl)CCC2OCCN(C(C3CC=CC3)=O)C2C1 61795,c1(CNC(CN(S(C)(=O)=O)C)=O)ccc(CCNC(C2CCCC2F)=O)cc1 61796,C1(CCC(=O)NC(CC)CC2CC2)CCCCC1 61797,c1(OC)cc(N)c(F)cc1C(N1CC2CCC1CN2C(=O)CC1CCOC1C)=O 61798,c1(CC(N2C(Cn3cc(C(CC)OC)nn3)CCC2)=O)ccc(O)cc1C 61799,C1(C(=O)NC2CN(C(c3ncccc3Br)=O)CC2O)CC2(CCCC2)CO1 61800,C1(C)(C(=O)NCC(CNC(C=CC)=O)C)COCCO1 61801,C1(NC(N(CC(C)(C)O)CC)=O)CCC(C)C1 61802,C1(NC(=O)C=Cc2ccco2)CC2(CCN(C(=O)C#CC3CCCCO3)CC2)C1 61803,N1(C(c2cc(OCC)ns2)C(=O)NCCC#N)Cc2cccc(F)c2C1 61804,c1(C(=O)NCC(CNC(Cc2cncc(C)c2)=O)(C)O)cn2cccc(Cl)c2n1 61805,Cc1cnc(C(=O)NCC(C)(O)CNC(c2c[nH]c(=N)s2)=O)cc1Br 61806,Cc1ccc(Br)nc1NC(C1COCCN1C(C1CCN(C)CC1)=O)=O 61807,C(C(CC1CCCC1)C(=O)N1CCC(C(N)=O)C1)NC(C(OC)OC)=O 61808,c1(SC)ccc(C(N2CC(CO)CC(F)C2)C(=O)NC2CC2)cc1[N+](=O)[O-] 61809,CCN=c1cc(-c2nc(Cc3cc(C)c(F)c(F)c3)n(C(C)C)n2)cc[nH]1 61810,C(c1ccccc1C)=CC(N1CCC(C(C(=O)N(C2CCN(C)C2)CC)C)CC1)=O 61811,n1(CC(=O)NC(C(=O)NCc2ccc(Cl)o2)C2CCC2)cc(Cl)cn1 61812,c1(OCCCC(=O)NCCN(C(=O)CC2(C)CC2F)CC)ccc(Cl)cc1C 61813,c1(CNC(c2cc(C)no2)=O)ccc(CNC(=O)C(F)C(F)(F)F)cc1F 61814,c1(N2CC(C)CN(C)CC2)[nH]c(=NCCS(C)=O)nc2scnc12 61815,C1(SC)CCCC1C(=O)NCC1(C(N2CCC(N3CCOCC3)C2)=O)CCCC1.N=O.C1CC1 61816,C(=O)(CCC(F)(F)C(F)F)NCCCCC(C)NC(CC(C)OC)=O 61817,C(=O)(C1=CC2CCCC12)NCCOCCCN(C)C(c1n[nH]c2ccccc12)=O 61818,N12CCC(CC1)CC2=O.C(=O)(NOCC(=O)OC)C1(COC)CC1 61819,C1(NC(CCCC)=O)CN(C(C2CCn3c(cnc3C)C2)=O)C2(CCCCC2)C1 61820,c1(C(=O)NC(CC)(C)CNC(=O)Cc2cncs2)cnc(C)c(C#N)c1 61821,C12(CCNC(c3c(C)nn(C)c3)=O)CCC(C1)N(C(C1CCC3CC1CO3)=O)C2 61822,c1(C(=O)NCC(C)N(C)C(c2c[nH]c(=O)cn2)=O)cnc(C(F)F)cn1 61823,C1(NC(c2c(CC)csc2)=O)CC=C(C(=O)NCCc2ccon2)C1 61824,n1(CC)cnc2c(NCc3ncn(CC)n3)[nH]c(=NCC(C(C)(C)C)SC)nc12 61825,C12(CNC(CC(C=C)(C)C)=O)CCCC1N(c1ncc(F)cn1)CCC2 61826,CC12CCN(C1)C2=O.C1(C=O)CCCC2CC12.c1(-c2ccccc2)ccccc1F 61827,C12(C(N3CC(CNC(c4cccc(CC)n4)=O)OCC3)=O)CCCC1CCC2 61828,N1(C(c2noc(CC)c2C)=O)CCC2CCN(C(c3nc(C)nn3C)=O)CC12 61829,CC1(C)CC(NC(c2snnc2C2CC2)=O)CCN(C(=O)Cc2ccsc2)C1 61830,C#Cc1ccc(CC(N2CC(NC(=O)CCC3CCCOC3)C(CC)C2)=O)cc1 61831,n1(CCC(N2C(C(C)(F)F)CCC2)=O)nc(O)c2c1CCCC2 61832,c1(CNC(C(=O)NC(CCCCC)C)=O)cc(F)ccc1C 61833,c1(N2CCCC(CN(C)C3CC3)C2)nc2ccccc2c(=NCC2CCCS2)[nH]1 61834,C1(C(N2C(CC)CC2)=O)CCN(C(=O)Cc2nccn2C)C1(C)C 61835,c1(C(N2CC(=C(CNC(c3nccs3)=O)F)C2)=O)cccc2c1OCO2 61836,Cn1c(O)nc2cc(C(N3C4CCC3CC(CNC(C3CCC3)=O)C4)=O)ccc12 61837,CN(C)S(C)(=O)=Nc1nc(C(=O)NC2(CNC(c3ccncc3O)=O)CC2)cs1 61838,c1(NC(C)CCO)[nH]c(=NCc2nc(Br)n(C)n2)nc2c1cnn2C 61839,N1(C(CCCOCCC)=O)CCN(C(=O)C(C)c2ccco2)CC1C1CC1 61840,C(c1cccnc1)=CC(=O)N(C(CNC(COCc1onc(C)n1)=O)C1CC1)CC 61841,N1(C(C2CC3CCCC3C2)=O)CC2CCCN(C(=O)CSC(F)(F)F)C2C1 61842,C(CS(=O)(=O)CC(=O)N1CCC(C2CC2)C1CNC(c1c[nH]nc1C)=O)OC 61843,C1(N(C(C2(OC)CCCOC2)=O)C)CCCN(c2ccnc(C(F)(F)F)n2)CC1 61844,C1(CNC(C=C(CCC)C)=O)CCCCC1NC(c1cc(CC)c(C)s1)=O 61845,C(=O)(CC1CC(=O)c2ccccc21)NCC1CN(C(CCN(S(C)(=O)=O)C)=O)C1 61846,C(CC(O)CNC(=O)C(C)N(C(=O)CN1CCNC1=O)C1CC1)OC 61847,c1(CN2CCC(NC(C(c3ccccc3)OC)=O)C2)cc(Cl)c(O)c(Cl)c1 61848,N(C)(C1CCc2c(F)cccc21)C(C(C)C(C)c1ccccc1Cl)=O 61849,C1(C(=O)NCC(CNC(C2C(C(C)(C)O)C2)=O)(C)O)CCCCC(=O)N1 61850,CC1(C)C(NC(=O)CC2CCCCC2)CCN1C(=O)CC(F)(F)Cl 61851,N1(C(C)=O)CC(NCCC(=O)NC(C2CCCC2)CNS(=O)(=O)CC)C(C)(C)C1 61852,C1(CNC(=O)Nc2c(OC)c(C)ccc2)(CO)COCC2CCCCN12 61853,c1(C(=O)NCC(C2CC2)OC)n[nH]c2c1CN(C(=O)C(C)CC1CCCC1)C2 61854,C1(CCNC(C2CCN(C)C2)=O)CN(C(=O)CCCCCN(C)C)CCCO1 61855,c1(C(=O)NCC2C(C)CN(C(C3CCOCC3)=O)C2)cccc(Cl)c1N 61856,c1(NC(C)=O)ccc(C(N2CCN(C(c3nncn3CC3CC3)=O)CC2)=O)cc1F 61857,CC(CN=c1nc(C2CCCC2)[nH]s1)NC(N)=O 61858,C1(CNC(=O)CCc2ccc(Cl)s2)CCN(C(c2nnc(O)nc2O)=O)C12CC2 61859,c1(NC(C2(C)N(Cc3ccc(C)nc3)CC2)=O)cnc2c(C#N)cccc2c1 61860,c1(C(N(C2CCCC2)CC#CC)=O)cccs1.C(=O)(CC(C)n1ccnc1)NC 61861,c1(C(=O)NC2CC(C)N(C(=O)C(C)n3cccn3)C2)nc(F)ccc1Cl 61862,C1(CCC(=O)NCC(=C)CCNC(=O)C(O)c2ccsc2)CCCC(=O)N1 61863,c1(CC)nc2ccccc2c(C(=O)NCC2(SC)CCOC2)c1C 61864,C(=O)(C(C)(C)CN=c1[nH]c(=NCCS(=O)(=O)CCO)c2cccc(F)c2[nH]1)NC 61865,C1(C(N(CC(=O)NCC2CCOC2)Cc2ccncc2)=O)C2CN(CCO)CC12 61866,C1(C(=O)NCCC2CCC(CO)CC2)CC(C2CCC2)C1 61867,Cc1c(CC(=O)NCC2CC2NC(=O)C2=CC(C)(C)C2)c(O)nc2[nH]nc(O)c12 61868,CON(C)S(=O)(=O)c1cccc(C(N2CC3CC2C3NC(C2CC(F)C2)=O)=O)c1 61869,Cc1cc(C(=O)NCc2cccc(C(=O)NC(C)C(F)(F)CO)n2)c(C)s1 61870,CC1(C)CCN(C(C2CSCCS2)=O)CC1NC(c1coc(Cl)n1)=O 61871,CC(C)(O)C(C1CC1)NC(=O)C(O)C1CN(C(=O)COCC(F)(F)F)C1 61872,C(N=c1ccc(C#N)c[nH]1)C1OCC(CNC(c2c(Cl)cn(CC)n2)=O)C1 61873,Fc1ccc2c(c1)C(N=c1ccnc(NCC3CCCO3)[nH]1)CCO2 61874,Cc1ccc(-c2nc(C)c(C(=O)NC3CCC(CNC(=O)C(N)=O)C3)s2)c(F)c1 61875,c1(CC(=O)NCC(CCNC(CCC=CC)=O)(C)C)coc2c(F)c(F)ccc12 61876,C(C(C)C(F)(F)F)NC(C(CO)NC(C(C=C)OC)=O)=O 61877,c1(C(=O)NCC(C2CCOC2)NC(=O)C=CCO)cnsc1 61878,CCN=C(NCCS(=O)(=O)c1ccccc1C)N1CCC2(CCCC2)C1 61879,CCC(C)C(C(=O)NC1CN(C(=O)Cc2ccnc(OC)c2)CC1C)N(C)C 61880,CN1CCN(C(C2CNC(=O)N2)=O)CC1CNC(c1ccc(-c2ccco2)o1)=O 61881,Cc1oc(S(N)(=O)=O)cc1C(N1CCN(C(C2CCC3(CCC3)O2)=O)C(C)C1)=O 61882,CCS(=O)(=O)c1cnc(O)c(C(=O)NCCCN(C(C2CC2CF)=O)C2CC2)c1 61883,C(=O)(C(O)CC(C)(C)C)NCCN(CCC)C(C1CNC(=O)C1)=O 61884,C#CC1(NC(=O)CC2(CNC(=O)C(C)=CC(C)(C)C)CC2)CCC(C)(C)C1 61885,c1(C(=O)NC2CC3CC(NC(C(C(=C)Cl)(C)C)=O)CC32)cc(F)c(F)c(C#N)c1 61886,c1(C(=O)NC2C(NC(C3CC(=O)NCC3)=O)COCC2)cc2n(n1)CCOC2 61887,S(=O)(=O)(CC(C)(C)C)N(C1CCCC(O)C1)C 61888,c1(CCC(=O)NC(C2CN(c3cc(F)ncn3)CCO2)C)ccc(F)c(F)c1 61889,c1(OC)cccc(C2(C(=O)NCCN(C)C(C3CC=CCC3C)=O)CC2)n1 61890,c1(NC(C)=O)ncc(-c2nc(-c3ccc(N4CCN(C)CC4)cc3)no2)cn1 61891,C1(C(=O)NC2(C)CN(C(C(C)SC(F)(F)F)=O)C2)CCN(C(=O)C(N)=O)CC1 61892,c1(C(=O)NC(C(CO)NC(COCCC)=O)C)ccc2c(c1)COCC2 61893,CCC(CC(=O)NC1CCC(O)CN(C(=O)Cc2cccc(OC)c2)C1)C(C)C 61894,c1(C(=O)NCCC23C(CN(C(C(C)(C)C(F)F)=O)C2)CC3)cnc2occc2c1 61895,C1(C(C)C(=O)NCC(C2CC2)NC(C2CCC2CF)=O)CCCCC1 61896,CCCCC(C(=O)N(C1CC1)CC1CCCCN1C(=O)CSC(C)C)C(C)C 61897,c1(C(=O)NCC(C)CNC(=O)C(C)CC2CC2)nc(Br)n2ccccc12 61898,N1(C(CCN(CC)CC)=O)CC2CCC2(CNC(c2c(C)ccn2C)=O)C1 61899,C1(NC(C(C)SCC)=O)(CO)CCCN(C(c2cccc(OC)c2O)=O)C1 61900,C1(NCC)CCCCC1N=c1ccnc(NCc2cn[nH]c2)[nH]1 61901,n1(CCC(=O)NC(CC=C)CNC(=O)C(F)(F)C(C)O)nc(O)c2ccccc12 61902,N1(C(c2ccnc(C(=O)OC)c2)C(=O)NCCOC)CCCC(O)(C(C)C)C1 61903,N#Cc1cc(C(N2CC(NC(C3CCCOC3)=O)CC(F)C2)=O)ccc1F 61904,n1(CC(=O)NCC2CN(C(=O)C(O)CC3CCOCC3)CCO2)ncccc1=O 61905,CC1(C)CCOC1C(=O)NCC1(C(=O)Nc2cncc(Cl)c2)CC1 61906,C(CCCC(CO)NC(=O)C(O)Cc1cc(Cl)sc1Cl)NC(=O)COC1CC1 61907,N1(C(C23C(CN(C(c4ccc(OC)cc4Br)=O)C2)C3)=O)CCn2cncc2C1 61908,c1(SCC(=O)N(CCNC(c2cnsn2)=O)CC2CCCC2)ccc(F)cc1Cl 61909,N1(C(=O)NCc2cccc(CC)c2)CC(=O)Nc2ccc(C#N)cc21 61910,c1(C(=O)NC(C)CCN(C(=O)CCn2cc(Br)cn2)C)cccnc1O 61911,C(=O)(C(O)C1=CCCCC1)NC(C(=O)NCC(C#C)OC)CC(=C)Cl 61912,c1(CCC)ncoc1C(=O)N(C)CCNC(c1cnn(C(F)(F)F)c1)=O 61913,CC(CC(C)NC(C1CC2CC2C1)=O)N=c1ccnc(C(F)(F)F)[nH]1 61914,CC(C)C(C)CC(=O)NC1(C2CCCN2C(=O)CN2C(=O)CCCC2=O)CC1 61915,c1(NCC2CCCN(C)C2)ccc(S(=O)(=O)NCCOC2CC2(F)F)c(Cl)c1 61916,C1(C)(COC)CN(N2CCCC(n3cccn3)C2)CCO1 61917,C(C(C)(C)CNC(=O)CN1CCCC1CO)N(C(COCC=C)=O)C1CC1 61918,C1(NC(c2nc(C3N(C(C)=O)CCC3)sc2)=O)CCC(CSC2(C)CCC2)CC1 61919,c1(C(=O)NCC(C2CC(F)(F)C2)OCC)cc(OC)ncc1Cl 61920,C12(NC(c3c(SC)csc3)=O)CCCC1CN(C(=O)CC(C1CC1)C1CC1)C2 61921,N1(C(C(C(CC)C)N)=O)CCC2CN(C(=O)Cc3cccc([N+](=O)[O-])c3)CC12 61922,C1(CC)CN(C(=O)CNC(c2ccoc2)=O)CC1NC(C1CC(=O)N(C)C1)=O 61923,C=C(Br)CN=C(NCC(=O)NC1CCCCO1)NCC(=O)NCC(F)F 61924,N1(Cc2ccc(C)o2)CCCC(O)(CNC(=O)C(=O)C(C)C)C1 61925,c1(OC)ccc(CN(C(c2ccccc2OC)C(=O)NC2CCCC2)C)nn1 61926,CCC(C(=O)OC)C(=O)NC1CC1CNC(c1cn(C)nc1-c1ccccn1)=O 61927,c1(C2CN(C(C(C3CC(C#N)C3)NC(C=CC(C)(C)SC)=O)=O)C2)cc(O)n[nH]1 61928,O(NC(=O)CCCN(C)C(C1CC(C)(C)CN1C)=O)CC(=C)C 61929,N1(C(c2c(N)ccc(C)c2)=O)CCC2(CCN(C(C3(C(N)=O)CC3)=O)C2)C1 61930,C1(C2(NC(C3(C(=O)OC)C=CCC3)=O)CC2)CCCCN1C(c1ncncc1Cl)=O 61931,CC1(CNC(C23CCCC2CCC3)=O)CCCN(C(c2cc(N)c(F)cn2)=O)C1 61932,c1(CCOC(c2occ(C(=O)OC)c2)=O)c(C)nc(SC)nc1O 61933,C1(C)(NC(C2CC(=C)C2)=O)CCN(C(=O)CCn2c(-c3cccs3)nnc2S)CC1 61934,n1(CCCOC)nc(-c2ccncc2)nc1C(c1noc(C(C)(C)C)n1)C(C)C 61935,CC(C)CC(C(=O)N1CCC(CCN(C)C(C2(C)C=CCCC2)=O)CC1)N(C)C 61936,CC1N(C(=O)CC2N(C(C3CCN(C)C3)=O)CCC2(C)C)CCOC1(C)C 61937,C=C(C)C(CC(=O)N1CCC(NC(=O)CN2CCC(CC)C2C)CC1C)OCC 61938,c1(C(N2CCC(CCN(C)C(C3(C4CC4)CC3)=O)CC2)=O)cccc2sccc12 61939,C1(C)(OCC(=O)NC(CCSC)C)CN(C(c2scnc2C2CC2)=O)C1 61940,Cc1cc2ncnc(NC3CC4CN(C(=O)Cc5c(Cl)cnn5C)CC34)c2[nH]1 61941,C(C(CNC(C1C2(CC2)C12CC2)=O)S(C)(=O)=O)NC(C(c1c(C)cccc1)C)=O 61942,c1(C(=O)NCC2C(CNC(c3c(C)cc[nH]3)=O)C2)cc2ncn(C)c2cn1 61943,N1(C(c2cc3cccnc3o2)C(=O)NCCCC)CCNC(=O)C(F)(F)C1 61944,C1(CC)(CC)CC(NC(=O)Cc2nonc2C)CN1C(c1ccc(C)s1)=O 61945,c1(CN(CC(O)CN(C(=O)C=Cc2cn[nH]c2)C)C)cccc(F)c1[N+](=O)[O-] 61946,C1(CC(=O)N(C2CCCCC2)CCNC(C2CC2C2CCC2)=O)Cc2nncn2C1 61947,N1(C(c2c(C)n[nH]c2)=O)CC(C2CN(C(c3ccc(Cl)c(C(F)(F)F)c3)=O)C2)C1 61948,c1(C(=O)OC2CCC(CC)CC2)cc2cc3c(cc2[nH]1)OCCO3 61949,C1(O)(C(C)NC(c2cc(Cl)n[nH]2)=O)CCN(C(=O)CN2CCCC2)C1 61950,C1(C(N2CC(NC(C)=O)C2)=O)CN(C(C2(C)SCCCS2)=O)Cc2cccn2C1 61951,O=C(C(F)(F)C(F)c1ccccc1)NC(c1ccc(F)cc1)c1ccc(Cl)cc1 61952,c1(C(C)NC(N)=O)ccc(CNC(=O)CCc2cnc[nH]2)cc1.C1(C)CCCCO1 61953,CC(O)C(F)(F)C(=O)N1CC=CC(NC(=O)CCc2ccc(O)nn2)C1 61954,c1(CC(=O)NCC2CCC2NC(C2CC3CC3C2)=O)c[nH]c2cccc(F)c12 61955,c1(N2CCC(C=C)C2)nc(N2CCC3(CCC(O)C3)C2)nc2ccsc12 61956,c1(C(=O)NCCn2cc(CNC(COCCC)=O)nn2)cc(F)ncc1OC 61957,C1(N(c2ccc(SC)c(Cl)c2)C(c2cnc(CO)s2)=O)(CC)CCCC(C)(C)C1 61958,c1(NCC2(F)CC(CNC(C(=O)N(C)C)=O)C2)ncnn2cccc12 61959,c1(CC)c[nH]c(C(=O)NCC2C(CNC(=O)CC(=O)N3CCCCC3)C2(F)F)c1 61960,c1(C(=O)NC2CCCN(c3nc(O)n[nH]3)C2)c(Cl)cc(F)cc1Br 61961,Cc1nsc(N(C)CCOCCNC(C2CCC(C)O2)=O)c1C#N 61962,N1(C(C(CC)=O)=O)CCC(C(N2CCN(C(N)=O)CC2)=O)C(C(C)C)C1 61963,c1(SCC)ccc(C(N2CCC(F)(C(=O)N(C)C)C2)=O)cc1 61964,CC1CC(=O)NCC1C(N1CCC(C)(CNC(=O)CCc2ccn(C)n2)C1)=O 61965,C1(C(=O)NCCCC(=C)Cl)CCN(C(C2CCN(C)C(=O)C2)=O)CCO1 61966,N1(C(C(C)C2(O)CCC2)=O)CC2(NC(=O)CN3CCOC3=O)CCCC2(F)C1 61967,N1(C(C)=O)CCCC(CN2CCC(N3CCCC3)CC2)C1 61968,N1(C(C(C)SC)=O)CCCC(C)(C)C1C(=O)NCC1CCCN1C 61969,CN1C(=O)CCC(C(=O)NC2CC2c2cn[nH]c2)C1=O 61970,c1(C2C(CNC(=O)C(N3CC(F)(F)CC3CO)=O)C2)c(F)ccc(F)c1Cl 61971,CCCCCCC(=O)NC(C1CCCC1)CNC(c1ccncc1C(F)F)=O 61972,Cc1cc(C(N2CCC(NC(C3CC4(C3)CC(C)(C)C4)=O)C2)=O)c(N)cc1F 61973,C(=O)(C1=CCS(=O)(=O)C1)NCCOC1CCN(C(c2nn(C)c(=O)cc2)=O)C1 61974,C(=O)(C1=CCCC1P(C)(C)=O)NCCN(C)C(c1cc2occc2s1)=O 61975,c1(C(=O)NCC2C(NC(C(C(C)C)(C)O)=O)CCC2)cccc2cc[nH]c12 61976,C1(C(N2C(C3(NC(Cc4n(C)cnc4)=O)CC3)CCC2)=O)OCCOC12CCC2 61977,C1(CC(N2CCCC(CNC(=O)C3CC3)C2)=O)Oc2ccccc2NC1=O 61978,N1(CC2(C(=O)O)CC(=C)C2)CC2(C)CC1CCO2 61979,c1(OC)cc(C(=O)NCC(C(C)C)NC(C23CCC(F)(CO2)C3)=O)cnc1OC 61980,c1(CC)c(C(N2CCC(Cn3cc(Cc4ccc(Cl)cc4)nn3)CC2)=O)csc1C 61981,c1(CC(C)NC(c2c(F)cccc2F)CCOC)ccc(OC)c(F)c1 61982,C1(C)(C(C)C)CCN(C(CCc2cnn(C)c2)C(=O)NCCCOCC2CC2)C1 61983,N1(C(C2CCC(Nc3ncnc4ccccc34)CC2)=O)CCC2(CCCOC2)C1 61984,CN1CCN(C(C(=O)N(CC)CC2CCCO2)c2ccco2)C(c2ncc[nH]2)C1 61985,C(=O)(CCCCC(C)(C)C)N(C1C2CCCC1COC2)C 61986,C1(C)(C(=O)NCC(=C2CN(C(CC(C)C3CCCO3)=O)C2)F)CCOC(C)C1 61987,Cn1cnc2[nH]c(C(=O)NC3(CNC(=O)C(C)(C)F)CCC3)cc12 61988,c1(C(=O)NC(C(C)NC(c2ccn(CCF)n2)=O)C)cccc2cncn12 61989,N1(C(=O)CCN2C(=O)CCC2=O)CCC2CCN(C(c3cncc(Cl)c3)=O)C2C1 61990,C(=O)(C#CC1(C)CC1)N1CCC(C)(CCNC(C2CN(C)C2)=O)C1 61991,c1(CCC(=O)NCC2CC2NC(=O)CC2CNC(=O)C2)cccnc1Br 61992,CCCCCCCCC(=O)Nc1cccc(S(=O)(=O)N(CCO)C(C)C2CC2)c1 61993,C(=O)(CC(C(F)(F)F)NC(=O)Cc1cccnc1O)NCCSCC#C 61994,C#CC1(Nc2cc(N3CCC(C)(CN(C)C)CC3)nc(CC)n2)CCN(C)CC1 61995,C1(Cc2n(C)cnn2)CN(C(=O)CCS(C)(=N)=O)CCC1c1ccccc1 61996,c1(COC(c2ccoc2C(=O)OCC(CC)(C)CC)=O)ccc(C)c(F)c1F 61997,Cc1cccc2c(C(=O)NCC3(C)CCCN(C(=O)Cc4cnns4)C3)coc12 61998,C(C(C)(O)C(=O)N1CC(CC(F)C(=O)OC)C1)C(=O)NC 61999,C1(NC(=O)CCn2cc(-c3cccc(Cl)c3)nn2)CC(CO)C12CCC2 62000,N1(C(C(=C(C)C2CC2)F)=O)CC2(COC(CNC(=O)C(F)C(F)(F)F)C2)C1 62001,C1(CC)CCc2sc(C(=O)NCC3(O)CN(C(C4CSCCS4)=O)C3)cc2C1 62002,n1(C(C=C)C)nc(-c2ccsc2)nc1-c1nn(C)nc1Br 62003,C1(N(C)CCNC(=O)CN(C)C(=O)OC(C)(C)C)CC(N(C)CCO)C1.C=O 62004,C(c1ncc[nH]1)=CC(=O)NCC(CO)NC(=O)C=CC1CCOC1 62005,CC1CNC(=O)CN1C(=O)C=CC1CCN(C(C2CC2Cl)=O)CC1 62006,Cc1cc(C)c2[nH]cc(C(N3CCC(O)(C(F)(F)F)CC3)=O)c(=O)c2c1 62007,N1(c2nccc(-n3c(C)cc(C)n3)n2)CCC(NC(c2cccnc2)=O)C(O)C1 62008,C(CCC(CCC)NC(=O)CC1CC(OC)C1)NC(C(F)=CC)=O 62009,CC1(C)COC(CC(=O)NC2CC(NC(=O)C=C3CCC3)C2)CO1 62010,C(=O)(C1=CN=C2N=CNN2C1)N1C(C)CN(C(C2(F)CCCC2)=O)CC1 62011,CCC(C)(C)C(O)C(=O)N1CCC2CC1CN2C(c1cccc(F)c1Cl)=O 62012,N1(C(c2cc(C)cc(Cl)c2)=O)CCC2(CC1)CN(C(=O)C1=CCC1)CC(C)O2 62013,C1(CNCc2ccc(C)s2)COCCN1C(=O)C(c1ccc(NC(N)=O)cc1)O 62014,C1(C(N2CCC(O)(C(F)F)C2)=O)(NC(=O)C(O)CN2CCCC2)CC(F)(F)C1 62015,CC1(C)CC(NC(=O)Cc2cc(N)c(Br)cc2[N+](=O)[O-])CC(C)(C)S1(=O)=O 62016,c1(CC)ncc(C(=O)NC(C)CCN(C(=O)Cc2cccc(O)c2F)C)c(C)n1 62017,N1(C(c2cccc(I)c2)C(=O)NCC(=C)C)CCN(C2CCCC2C(N)=O)CC1 62018,CCCCC(C(=O)N1CCN(C)CC1C(=O)NC(CCC)c1nn[nH]n1)C(C)C 62019,c1(C(=O)OC)ccc(O)nc1N1CCC(CCNC(=O)C(=O)NCC2CC2)C1 62020,C1(CCNC(CC(=O)OC)=O)CN(C(c2cc(O)n(C)n2)=O)CCCO1 62021,N1(C(C2(COCC)CC2)=O)CCC(CCN(C)CC2SC3C=CC2C3)CC1 62022,C1(NC(CSCCC)=O)CN(C(=O)C=Cc2ccccc2C)C2CCCC12 62023,N1(C(C=COCC)=O)CCC2(CC1)CCN2C(c1cccc2[nH]ncc12)=O 62024,C1(C(=O)NCC(C2CCN(C(C(C)n3cccn3)=O)CC2)O)CC(=O)NC(=O)N1 62025,c1(C(=O)NC(C2CCN(C(=O)C=CCOc3ccccc3)C2)C)ncc(Cl)s1 62026,c1(C(=O)NCCCCNC(CC(=O)NCC#C)=O)c(C)cc(OC)cc1C 62027,C(CC(CNC(=O)CC1(C)CCC1)NC(c1cnnn1-c1ccccc1)=O)OC 62028,Cc1cnc2cc(C(=O)NC3CC4CCC3CC4NC(=O)C=CS(C)=O)nn2c1 62029,Cc1nn(-c2ccccc2)cc1C(=O)N(CC(O)CN(C(=O)C=CS(C)=O)C)C 62030,O=C1NCc2ccc(C(N3CC4CCC3CN4C(C3CC3C3CCC3)=O)=O)cc21 62031,CC(C(=O)NCC1(C(N)=O)CN(C(=O)CC2CCCC(F)(F)C2)C1)S(C)(=O)=O 62032,Cc1csc2cc(C(=O)NC34CC(NC(C5CC6(CCC6)CO5)=O)(C3)C4)[nH]c12 62033,c1(OC)cccc(OC)c1NC(=O)C(CC(C)C)n1ccnc1 62034,Cc1cc(C)c(OC(=O)C(O)CC[S+](C)C)c(Br)c1 62035,Cc1ccccc1C1(NC(N2CCC2C2(C(F)(F)F)CC2)=O)CC1 62036,C1(NC(c2cccc(C(F)(F)CF)c2)=O)(CF)CCN(C(=O)CN2CCCC2)C1 62037,Cc1cccc(C)c1CCN=C(NCCOc1ncccn1)NC(C)C(C)C 62038,c1(C(=O)NC23CC(NC(c4csc(C(F)F)c4)=O)(C2)C3)cc(Cl)c2n[nH]cc2c1 62039,C(=O)(CC(C)C(C)(C)C)NCCN(CCCCCC)C(=O)CC1CCOC1(C)C 62040,c1(C(=O)OCC)nc(=NC(C)CN(C(=O)CCC(C)OC)C)cc(C(C)(C)C)[nH]1 62041,c1(OC)cc(C(=O)NCCC(C)NC(C2CNC(=O)C2)=O)cc2c(C)c(C)[nH]c12 62042,N1(C(C(F)(F)C2(OC)CCC2)=O)CC(N(C)C(C2CC3(CC3)CO2)=O)C(F)C1 62043,c1(C(=O)OC)ccc(C(=O)NC2CC2NC(C23CCCC2C3(F)F)=O)c(C#N)c1 62044,CC1CN(C(=O)C(C)(F)F)CC(C)N(C(C2CCC3(CC2)N=N3)=O)C1 62045,c1(C(N2C(C)C(NC(=O)Cc3cncnc3O)CC2)=O)cn2c(n1)SCC2 62046,C#CCCCC(C)C(=O)NCC(CC=C)C(=O)N1CCC(CN=[N+]=[N-])C1 62047,C12(CNC(CC3N(C)CCC3)=O)CC1CN(C(=O)CCNC(=O)CO)C2 62048,N#Cc1cccc(NC(=O)CC2(NS(=O)(=O)c3cn[nH]c3)CCC2)c1[N+](=O)[O-] 62049,N1(C(C(c2ccc(F)cc2)NC(C#C)=O)=O)CCCCC1CNCCCO 62050,Cn1cc(C(N2CCC(C(F)CNC(=O)CCS(C)=O)CC2)=O)c(Cl)n1 62051,c1(C(N2CCC(CC(=O)NC(c3nncn3C)C)C2)=O)cccc2cnccc12 62052,C(=O)(CCCCCC#N)NC(C)C(=O)NC(CCO)C(C)(C)C 62053,CC(C)(C)C(CC(=O)N1CCC1CNC(=O)Cc1cccc(C(N)=O)c1)C(F)F 62054,Cc1ncc(Cl)cc1CC(=O)NC1CC(NC(=O)CCn2cnc([N+](=O)[O-])c2)C1 62055,C1(C(=O)N(CCCC2(NC(C(CCC)OC)=O)CC2)CC)CCCCC1(F)F 62056,Cc1cc(C(N2CCN(C(C3(c4ccc(O)cc4)CC3)=O)CC2C)=O)cnc1Cl 62057,Cc1cc(C)c(C(N2CC(CC(C)NC(=O)CC3SC(=N)NC3=O)C2)=O)[nH]1 62058,C1(C(=O)N)C2CC3C(C2)C13.C1(C(N)=O)(CO)CN(C(C2CC(C(F)F)C2)=O)C1 62059,c1(CC(=O)NC2CN(C(c3c(=N)[nH]cnc3)=O)C3C2C3)ccc(F)c(Cl)c1 62060,C(=O)(C(C)(C)CC(=O)NCC1CCC(C(=O)NCc2cc(C)no2)C1)OC 62061,C(=O)(CCCC(=O)NC(C1COCCO1)C1CC1)NC 62062,c1(C(=O)NC(C)(C)CCNC(=O)C2=CCC2)cc(C(F)F)cc(C(F)(F)F)c1 62063,c1(C(=O)NC(C(C)C)CNC(c2cccc(Cl)c2Cl)=O)nccc(C#N)c1F 62064,N1(C(COCCC=C)=O)CCC2CCN(C(=O)C(c3ncccc3C)(F)F)CC12 62065,CC(C)C(C)(C)C(=O)N(CCC(=O)NCCCCCN(C)C)C 62066,CCCCC(CNC(c1cncc(N)n1)=O)NC(=O)C(C(C)C)c1ccccc1 62067,C1(NC(C(C=C)O)=O)C2CC1N(C(C1(S(C)(=O)=O)CC1)=O)C2 62068,c1(C(=O)CC(F)F)cc(NC(C2CCCN(c3cnccn3)C2)=O)cc(F)c1 62069,N1(C(C=C(CCN(C)C)Cl)=O)CCOC(C)(CNC(c2ccncc2F)=O)C1 62070,c1(CNC(=O)CSC2CCOCO2)ccc(N2N=CCC2=O)cc1 62071,c1(C(=O)NC(CCN(C(c2c(C)[nH]nc2Cl)=O)C)C)ccc(S(C)=O)cc1 62072,C1(CNC(c2nn(C)c(Br)c2)=O)CC2(CCC2)CN1C(=O)C(F)=C1CCC1 62073,C1(CC#C)(C(=O)NCCC(C)CCNC(c2c[nH]cc2C)=O)CCOCC1 62074,c1(C(=O)NC(C2OCCN(C(C3CC(N(CC)CC)C3)=O)C2)C)cncc(Cl)c1C 62075,C(=O)(C(C)(O)C(F)(F)F)N(C1CCCN(C(=O)CC23CC(C2)C3)CC1)CC 62076,Cc1cc(C)c(C(=O)NCC2CCC(C)CN2C(c2coc(O)n2)=O)cc1N 62077,N1(C(CC(C)OC)=O)CCC(NC(=O)CSc2nnnn2C2CCCC2)C12CC2 62078,Cc1ccc(N)c(C(N2CC(O)(CCNC(C3CC(C)CC(=O)N3)=O)C2)=O)c1 62079,CCCC(C)(CCC)C(=O)NCCOC1CCN(C(=O)CC2CCC2(C)C)C1 62080,C#Cc1cc(C(=O)N(CCNC(=O)C(C)(C)CN(C)C)CC2CC2)cc(F)c1 62081,C#CC12CC(CN1C(C1CCC(CNC(=O)C(C)CC(C)C)CC1)=O)C2 62082,C(C(=O)Nn1nnc2c1CCCC2)C1N(C(Cc2c(C)n[nH]c2)=O)CC1 62083,C1(C(=O)NCC(C)N(C(=O)C=C2CCN(C)C2)CC)CCOC2(CCC2)C1 62084,c1(CNC(=O)CC2CCN(S(=O)(=O)CCCN3CCOCC3)C2)ccnc(F)c1 62085,c1(OC)cc(C=CC(N2CC(=CC(=O)O)C2)=O)sn1 62086,c1(OC2(CCCNC(CCC(=O)NC)=O)CC2)cc(CCC)cc(OC)c1OC 62087,c1(OC)cc(C(=O)NC(c2ccc3c(c2)CCC3)C)nc2ccccc12 62088,C1(c2n(CC=C)nnn2)(NCCCCO)CC2CCC(C1)N2C1CC1 62089,C1(NC(C=CCC(C)(C)NC(Cn2c(C)ncc2)=O)=O)CCSC(C)C1 62090,C1(NC(C2CN(C)C2)=O)CCN(C(c2cn(C)c(=O)cn2)=O)CC1O 62091,C1(C(=O)NCC(CC(C)C)NC(=O)C(C)n2cccn2)CC(S(C)(=O)=O)C1 62092,C1(F)(CC)CCN(Cc2nc(Cc3ccccc3)cs2)C1 62093,N1(C(CCNC(N)=O)=O)CCC(C2CCN(C(C34CCC(F)(CC3)C4)=O)C2)C1 62094,c1(CC(=O)OCC)ccc(NC(CNC(=O)COCCCC(C)C)CC)cc1 62095,C#CC1CCCN(Cc2ccc(C(N3CC(C(=O)OC)C(F)C3)=O)cc2)C1 62096,c1(CC(N2CC(C)C(NC(=O)CN(C)S(=O)(=O)N(C)C)C2)=O)cc(F)ccc1O 62097,N1(C(C(=Cc2cccs2)C)=O)CC(NC(=O)CCN2CCC(F)C2)C(C2CC2)C1 62098,c1(C(C(=O)NC)N(C(Cc2ccccc2F)CO)C)cc(Cl)c2c(c1)OCCO2 62099,c1(C(C)=O)ccc(C(=O)NCCCC(C)NC(c2cc(C3CC3)no2)=O)o1 62100,N1(C(c2ccn(CC)n2)=O)CC(CNC(c2c(C3CCC3)cnn2C)=O)C(C)C1 62101,c1(NC(=O)CNC(C2CC2C)=O)cccnc1C(N(CCC(F)(F)F)CC)=O 62102,C1(OCC)CN(C(C2(F)CCCOC2)=O)CC1CNC(c1occc1C)=O 62103,C(N=c1[nH]cnc(Cl)c1C)c1ccc(C(C)NC(c2c(Br)ncc(C)c2)=O)cc1 62104,c1(C(=O)NC2(CNC(C(CCS(C)=O)O)=O)CC2)cc(O)nc2c1CCCC2 62105,CCCC(CNC(=O)Cc1cn(C2CC2)cn1)NC(=O)C(F)(F)C1CC1 62106,c1(N(S(CCC(=O)OC)(=O)=O)C2CCNCC2F)ncc(C#N)c(OC)n1 62107,Cc1cc(=NC(=O)CN(C)C(c2nn(C)c(C)c2N)=O)[nH]o1 62108,N1(C(C2C(C)C2)=O)CC2CC1CN2C(c1cccc(-c2ccncc2)n1)=O 62109,C1(NC(C2CC(C)CN2C(c2ccc(C#N)o2)=O)=O)CC(C)N(C)CC1C 62110,CC(CCN=c1[nH]cnc2cccnc12)NC(=O)CCC1CCCOC1 62111,CC1CCN(C(=O)Cc2cnccn2)C(C)C1NC(=O)CCCC1CCCCC1 62112,N1(C(C(=O)NCC(F)F)C2C(C)C2)CCC(CC(N2CCCCCC2)=O)CC1 62113,C(CC(C(C)(C)C)NC(C1CCC(C)(C)C1)=O)N(C(C1(CCCC)CC1)=O)C 62114,c1(NC(=O)Nc2ccc(C(N(CC)CC)=O)cc2)cc(C)c2c[nH]nc2c1 62115,C(=O)(C(C)C(=O)N1CC2(NC(c3sc(C(F)(F)F)nc3C)=O)CC1C2)OC 62116,N1(C(C(C(C)C)C)=O)CCN(C(c2ccc([N+](=O)[O-])s2)=O)CC(CO)C1 62117,C#Cc1ccc(C)c(NC(C2CC(C)(NC(=O)CC3CCC(=O)N3C)C2)=O)c1 62118,CC1CN(C)C(C)CC1NC(C1C(NC(=O)CSCC(F)F)C1(C)C)=O 62119,c1(OC)cc(C(=O)NCc2cn(C3CCN(C(=O)C(C)=C(C)C)C3)nn2)sc1Cl 62120,Cc1[nH]nc(C(N2CCOCC2CN(C(=O)C(F)(F)c2nccn2C)C)=O)c1N 62121,C12(C(=O)NCC3(C(N4CCC(C(=O)OCC)C4)=O)CCCO3)CCN(CC1)CC2 62122,c1(C(=O)NCC(CNC(C2(C(=O)OCC)CCCC2)=O)C)ccc(S(N)(=O)=O)o1 62123,c1(CC2(C(N)=O)CN(C(=O)CC3CC3)C2)sc(Cl)cc1Cl 62124,c1(C(=O)NC2(C)CCN(c3ncc(C(=O)OC)cn3)C2)cc2n(c1)CCSC2 62125,c1(C(=O)NCC2(CN(C(c3ccc(C)s3)=O)C)CC2)ccc(Cl)nc1N 62126,c1(CCC(=O)NC2CN(C(=O)C(O)CC3CC3)CCC2O)nc2ccccc2o1 62127,C1(NC(CCc2nc(C)sc2)=O)CCC(NC(C2C3COCC23)=O)CC1 62128,C1(C(=O)NC(C#C)C)(NC(=O)C(COC)N(C)C)CC1(C)C 62129,C1(CNC(C(CC)NC(C)=O)=O)CC2CCC1N2C(=O)CCCCN(C)C 62130,C1(NC(=O)C(F)CC2CC2)CC(Nc2cc(O)ncn2)C12CCC2 62131,C1(C(=O)NC2(CCCNC(c3ccc(Cl)c(Cl)c3)=O)CC2)COC2(CCC2)C1 62132,C1(c2nnnn2Cc2ccccc2)(NCCc2nc(C)sc2)CCCCCC1F 62133,N1(CC#C)CC2(CCC1=O)C(c1nnnn1C1CC1)N2.c1(C)csc(C)n1 62134,C1(C(N(CCCNC(=O)C(N2CCCC2)C2CC2)CC)=O)CNC(=O)CC1(C)C 62135,C1(CNC(C(F)=CCC)=O)CCCC1NC(c1cc(C(=O)OC)[nH]n1)=O 62136,C1(CNC(C(CC)CC)=O)CCN(C(C2CC3CC(=O)C2O3)=O)C12CCC2 62137,C(=O)(C(O)C(C)(C)C)N1C(C2CCN(C(CCC(C)OCC)=O)C2)CCCC1 62138,C(=O)(CCCC(C)C)NCC1CN(C(NOCCC)=O)C(C)C1 62139,c1(SC)ccc(C(=O)NC2CC(NC(=O)CN(C)C(C)=O)C23CCC3)c(Cl)c1 62140,CC(C)(C)CC(=O)NC(C(N1CCC(OCCF)C1)=O)C1CC1 62141,C(=O)(NNC(=O)CC(N(c1ccccc1)C1CCC1)=O)c1ccc(CC)cc1 62142,N1(C(CCn2c(C)ncc2)=O)CCC2(CCCC2NC(=O)Cc2n[nH]c(=N)s2)C1 62143,CN1CCCC(NC(c2cn(CCNc3cncc(N4CCCC4)n3)nc2)=O)C1 62144,C(=O)(CCCC(C)(C)C#N)NCC(C)(C)NC(Cc1cc(OC)cc(OC)c1)=O 62145,N1(C(C(C2CC(F)(F)C2)OC)=O)CCC2(CC1)CC(NC(c1cnsn1)=O)CO2 62146,n1(CC(=O)NCC2C3N(C(C(COC)O)=O)C(CC3)C2)nc2ccccn2c1=O 62147,C1(C(=O)NC(C)(C)C=CC(=O)NC(C2CCOC2)(C)C)C2CCC(F)C12 62148,N1(C(c2c(OCC)cccc2)=O)CCC2(CCCN2C(=O)CC(O)C2CC2)CC1 62149,c1(C(=O)NCC2N(C(C(C)c3cccs3)=O)CC2)cc(NC2CC2)ncc1Cl 62150,c1(CC)cc(C(=O)NC2C3CC2N(C(c2oc(C)nc2C)=O)C3)ccc1C 62151,CCC(CN1CCOCC1)(CC)NC(=O)NNC(=O)c1cscn1 62152,c1(CCC)cc(C(N2CCC(C(C)NC(c3cnc(CC)n3C)=O)C2)=O)nn1C 62153,N1(C(C(C)CF)=O)CCCC(N2CCN(C(=O)CCc3n[nH]c(=N)s3)CC2)C1 62154,c1(C(=O)NC2CC(NC(c3c(CC(N)=O)occ3)=O)C2)nc2n(c1Cl)CCCC2 62155,c1(C(=O)NC(CNC(C(C)C2CCCC2)=O)(C)CO)cc2c(s1)CC(C)(C)C2 62156,n1(CC)nc(C(=O)NC(C2CCN(C(C3CCCCS3)=O)CC2)C(C)C)cc1C 62157,c1(N(C)C)nc(NCC2CC(C)(NC(=O)OC(C)(C)C)C2)ccn1 62158,C1(NC(C=CC=CC)=O)CCN(C(c2ccccc2-c2ccncc2)=O)CC1C 62159,N1(C(c2ccnn2CC(F)F)=O)CCC(Nc2cccc(C(F)(F)F)c2)CC1 62160,c1(C(N2CC(CCC)C(NC(=O)CC(C)OC)C2)=O)cc(C)nc(C)n1 62161,c1(NC)ccccc1OC.C1CC(OC)CNC(=O)C=C(CC)C=CC(=O)N1.CC=C 62162,C(=O)(CCCC(=O)NCCCCNC(c1ccccc1N1CCCC1)=O)OCC 62163,C1(NC(C(CC=C)(C)O)=O)CCCC2CN(C(=O)C(O)C(F)(F)F)CC12 62164,CCN=C(NCCC1(C)CC1(F)F)N1CCc2c(Br)cccc2C1 62165,C1(O)(C(C)NC(=O)CC(C)n2cccn2)CCN(C(c2ccco2)=O)CC1 62166,c1(C(N(CC(C)CO)C)=O)coc(CNC(C2(O)CCOC2)=O)n1 62167,c1(NC)c(C(=O)NCC2CN(C(C3CC4CCCC34)=O)C2)cccc1N 62168,C(=O)(C(C)CCCc1ccccc1)N1CCC(N(C(C2CC2(C)C)=O)CC)C1 62169,C1(C)(CNC(C2N(CC)CC2)=O)CC(OC)CN1C(=O)CC(C)n1cccn1 62170,C1(C(N2CCC(F)C(O)C2)=O)CC2CC1CN(C(C1CC3(C1)CC(O)C3)=O)C2 62171,C12(C(=O)NCCC(C)N(C(c3ccc(C(=O)OC)[nH]3)=O)C)CCCN(CCC1)C2 62172,N1(C(C=C2CCN(C)CC2)=O)CCCN(C(c2ccc(Cl)nc2N)=O)CC1 62173,CN1CC(C(NC(c2cc(Cl)cc(I)c2)=O)NC23COC(CF)(C2)C3)OCC1=O 62174,C1(NC(CCCCSC)=O)COC2(CCN(C(=O)Cn3ccc([N+](=O)[O-])n3)C2)C1 62175,c1(C(=O)NC(C)(C)C(=O)N2CCCC2)ccccc1C1CC1(F)F 62176,C1(CNC(CC)=O)CCN(CCC(=O)NCC(=O)Nc2ncc(Cl)s2)CC1C 62177,c1(C(N(CCNC(C(C)OCCCCCC)=O)CCC)=O)cccc2c1CCO2 62178,c1(CC(=O)NC2CCN(C(CCC(=O)NC)=O)C(C)C2)csc2nc(C)cn12 62179,Cc1cc(N)cnc1C(N1CC(CC(F)C(=O)NCC(CC)C(C)(F)F)C1)=O 62180,c1(C(=O)NC2CC(NS(=O)(=O)c3cccnc3)C2)cc(Cl)nc(Cl)c1F 62181,c1(SCC(=O)Nc2ccc(C#N)c(I)c2)c(Br)c(O)c(O)c(Br)c1Br 62182,n1(CC(=O)NCc2onc(-c3cccc(C)c3)n2)c(C(C)C)nc2ccccc12 62183,C1(CNC(COCC(=C)C)=O)CC(C)CN(C(=O)C(C)(O)CC)C1 62184,N1(C(c2c(OC)cnc(F)c2)=O)CCCCC(NC(c2ccncc2C)=O)CC1 62185,n1(CCC(=O)NCCCC2(NC(C(C)C#N)=O)CC2)cnc2sccc2c1=O 62186,c1(NC(=O)CC2CN(C(=O)CC3CN(C(F)(F)F)CCO3)C2)ncc(Cl)nc1Cl 62187,C1(NC(C(CC)(C)O)=O)COC2(C1)CN(C(=O)C1=CCCOCC1)C2 62188,N1(C(Cc2ccn(C)n2)=O)CC2CC(NC(C3CCCC(C)(C)C3)=O)CC1C2 62189,C1(NC(C=CC(C)NC(c2n(CCC)ncc2)=O)=O)CCN(C)CC1C 62190,N1(C(C2CCCN(CCC)C2)=O)CCN(C(=O)C(C)S(N)(=O)=O)CC(C)(F)C1 62191,c1(C(=O)NCCC2(NC(c3c(F)ccc(C)n3)=O)CC2)cccc2scnc12 62192,c1(C(=O)NC2(C)CCCN(C(Cc3c(C)cc(F)s3)=O)C2)n[nH]c2c1CSCC2 62193,CC1CCCC(C(N2CC3C(CNC(=O)C=Cc4cnn(C)c4)C3C2)=O)C1 62194,Cc1ccc([N+](=O)[O-])c(C(=O)NCC2CC3CC3N2C(C2CC3CCC2O3)=O)c1 62195,CC1CC(=O)NC(C(=O)NCc2cccc(NC(=O)C(F)(F)c3cncs3)c2)C1 62196,N1(C(CCC#CC)=O)CCCCC2(CCN(C(=O)C3=C(C)CCCC3)C2)C1 62197,CC(O)CCN=c1[nH]c(N2CCC(N3CCOC3=O)C2)nc2c1COC2 62198,C1(CNC(=O)CCn2cncn2)CC(F)CN1C(C1CCCCC1)=O 62199,c1(SC)cc(F)ccc1C(=O)NC(C)(C)CNC(c1c(C(F)F)nn(C)c1C)=O 62200,C12(CS(N3CCN(C(c4ccc(OC)cn4)=O)CC3)(=O)=O)CCC(CC1)C2(C)C 62201,c1(CCC(=O)N(CC(CC)NC(=O)C(C)Cc2cccnc2)C)c(C)noc1C 62202,C1(C(=O)NCC(CC=C)NC(=O)CC)C(C)(C)CCCC1(C)C 62203,Cc1nc(C(=O)NC2(C(N3CCC(CCF)CC3)=O)CCCC2C)c(C)o1 62204,C1(OC)CCC(CC(=O)NCC2(C)CCCN2C(c2occc2C)=O)CC1 62205,C(C(O)C(F)(F)F)NC(c1cncc(OCCN2CCCCC2)c1)=O 62206,N1(CC(C)NC(N)=O)CCN(C)C(=O)C1.N12CC(C1)C2=O 62207,C1(CC(=O)NC2CN(C(C(C)OCC3CCCO3)=O)C2)COCCOC1 62208,c1(C(c2nnnn2C)NC2(CO)CC(OC)C2)ccc(N2CCC2)cc1 62209,N1(C(C2(C)C(C)C2)=O)CC(NC(c2csc(-c3ccco3)n2)=O)C(O)C1 62210,C1(CNC(=O)COc2ccsn2)CN(C(=O)C(c2ccccn2)O)CCCO1 62211,CC1CC2(CCN(C(=O)CCC3CC3)CC2)CN1C(c1ccc(S(C)=O)cc1)=O 62212,c1(N2CC(C(C)NC(C3(OC)CCCC3)=O)C2)nc(Cl)ncc1Cl 62213,c1(C(N2CCCCC(NC(=O)C=C3CCOCC3)C2)=O)cc2n(n1)CCCN2 62214,CC1(CNC(=O)C(C#N)C2CC2)CCCN1C(c1cnc(S)[nH]1)=O 62215,c1(C(=O)OCC)sc2ccncc2c1NC(=O)COC(=O)CCc1ccc(CC)o1 62216,Cc1ccc(C(=O)NC(C)CCN(C(=O)CCc2cnn(C)c2)C)nc1 62217,N1(C(CCSC)=O)CCC2C(CCN2C(c2ccc(C(C)(C)C)[nH]2)=O)C1 62218,C1(NC(CC)=O)(CNC(=O)CNc2nc(C)cs2)CCCCC1C 62219,c1(NC(C2C(NC(CC(C=C)(C)C)=O)C2(C)C)=O)cccc([N+](=O)[O-])c1 62220,C1(SC)CN(C(=O)NCC2CC(C)(C)NC(=O)O2)C2(CCOCC2)C1 62221,OCC(F)(F)CCCCN=C(NCc1ccon1)NC1CCC1 62222,Cc1cc(Cl)ncc1NC(=O)C(C)C(C)NC(c1ccn(CO)c1C)=O 62223,C1(C(=O)NCC(C)(C)OCCNC(C=C(C)C(F)F)=O)CC(C2CC2)C1 62224,Cc1cc(NC(c2cncc(NC(=O)C(C)(C)Br)c2)=O)c(O)c(C)c1 62225,C=CC(CCC)CC(=O)N1CCN(C(=O)CCc2cccc(O)n2)CC1 62226,Cc1nc(N(C)C)sc1C(N1CCC(C)C1CNC(C12CC(C1)C2)=O)=O.C1=CC1 62227,CCCCN=C(NCCc1cccc(F)c1F)NC1CN(C2CC2)C1 62228,C1(CNC(C2(CC#C)CCOC2)=O)CC2CCC1N2C(=O)C(C)(CC)CC 62229,C1(CNC(C23CC(NC(CC(C)C)=O)(C2)C3)=O)CCNC(=O)C1 62230,CCCC(C(=O)OC)C(=O)N1CC(C2(NC(C3CCS(=O)(=O)C3)=O)CC2)C1 62231,c1(N(CCCCO)C)nnc(C(F)F)n1CC(=O)NCC1CC=CCC1 62232,Cc1nc(C=CC(=O)NCC(O)CNC(=O)CCOC2CCOCC2)cs1 62233,c1(CC)cc2c(N(C(C)CCNC(C34CCC(CC3)C4)=O)C)nc(C)nc2s1 62234,C#Cc1ccc(F)cc1C(=O)NC1CN(C(c2ccc(F)cc2C#N)=O)CC1C 62235,N1(C(C(Cc2cnc[nH]2)NC(c2n(C)ccn2)=O)=O)CCOCC2(CCC2)C1 62236,N1(C(c2c(-n3cc(C(C)(C)CO)nn3)cc(F)cc2)=O)CC(C)(C)C(O)C1(C)C 62237,C1(C)(C(=O)NCC(C)(C(C)C)NC(C(CCC)=CCC)=O)CCCCC1(F)F 62238,c1(C(=O)NC2CN(C(C(CC=CC)C)=O)CC23CC3)cc(C)c(C#N)cn1 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62291,C1(C2CCC2)(C(=O)NC2CC(NC(C3(COC)CCOCC3)=O)C2)CC1(F)F 62292,n1(CC(=O)NC2(COC)CN(C(=O)C(C)(C)F)C2)ccc(C)cc1=O 62293,c1(N2CCC(C3(NC(CC(C=C)(C)C)=O)CC3)CC2)cc2c(cn1)C(=O)CCC2 62294,c1(C(N(CCCCN(C(C(C)C2CCOC2)=O)C)C)=O)ncccc1N 62295,c1(-c2cn(CC(N3CCC(c4ccc(F)cc4)C3)=O)nn2)cc(F)c(F)c(F)c1 62296,Cc1cc(F)c(CC(=O)NCCCCCCNC(C2COCCC2C)=O)cc1F 62297,c1(CNC(C(C)N(C(=O)C(C)C2CCC2)CC)=O)sc(C)cc1C 62298,c1(C(=O)NC(COC)C)cc([N+](=O)[O-])ccc1Sc1ccccc1-c1nn[nH]n1 62299,C1(C(C)C)CN(C(c2cnco2)=O)CCN1C(C1CN(CC(F)(F)F)C1)=O 62300,c1(OC)ccnc(OC)c1C(N1CC(CNC(c2cn(CC)nn2)=O)C(C)C1)=O 62301,CCC(CC(=O)NCCn1cc(C(=O)Nc2ccc(C)c(O)c2)nn1)C(C)C 62302,N(C1CS(=O)(=O)N(C)c2ccccc21)C(=O)NC(c1cccnc1)CC 62303,Cc1[nH]c2ccccc2c1C(=O)C(N1CCC(N)(c2ccccc2)CC1)C 62304,CC1(C)CC(NC(C2CCC23CCC3)=O)CCN(C(C2CN(C3CCC3)C2)=O)C1 62305,N1(C(CN2C(C)CCCC2)=O)CC(NCN(C(=O)C(C)(C)C(N)=O)C)C2(CC2)C1 62306,Cc1c(Cl)ccc(C(=O)NCC2CCN(S(=O)(=O)C3CC3)CC2)c1F 62307,c1(C(=O)NC(C)CNC(=O)C(C)n2cncn2)cccc2c1OCCN2 62308,c1(C(=O)NC2(CF)CC2)ccc2nc(CCCNC(c3cc(Cl)cs3)=O)[nH]c2c1 62309,C1(C(CC)C(=O)Nc2ccccc2)CCC(C)CC1.c12cnoc1c2=O 62310,C1(C(N2CC(NC(c3c(C)cn(C)n3)=O)C(C)C2)=O)CC2CCC(C1)C2 62311,C(C1c2ccccc2CN1C(C1CC1C1(C)COC1)=O)NC(CN(C(C)C)C)=O 62312,N1(C(C(C)C2CCCC2)=O)CC(NC(=O)CCc2cn(C)nn2)C(F)C1 62313,N1(C(C(=O)NCCC(O)C2CCCC2)=O)CCc2nc(S)[nH]c2C1 62314,c1(SC)ncc(C(N2CCN(C(c3cnc(=N)[nH]c3)=O)C(CF)C2)=O)c(O)n1 62315,N1(C(C#CC(C)C)=O)CC2COCCC2(NC(c2nccnc2N)=O)C1 62316,C1(CNC(C(F)=CCC)=O)CC2CCC1N2C(c1cccc(Cl)c1CC)=O 62317,CC(C)C(O)C(=O)N1CC(NC(=O)CC2CC(F)(F)C2)C(c2ccccc2F)C1 62318,Cc1cc(C(=O)NCC(C)(C)CNC(=O)C(O)Cc2ccc(F)cc2)cc(C)c1 62319,C(=O)(C(C)(C)CCCF)NCC1(CC(=O)NCC(c2n(C)ncc2)O)CC1 62320,C1(CCNC(C(C)SC)=O)CCN(C(=O)CSCC(C)C)C1 62321,c1(C(N2CCN(C(C(CC#C)O)=O)C(CO)C2)=O)cnc2c(cnn2C)c1O 62322,C1(NC(CNS(CC)(=O)=O)=O)CN(C(=O)C(CC)SC(C)C)Cc2nccn2C1 62323,CC1(C(=O)NC2CCC(NC(=O)CCc3nc(=N)[nH][nH]3)C2)CCC(=O)NC1 62324,c1(NC(C)C)ccc(C(=O)NCC23CC2CN(C(=O)Cc2cscn2)C3)c(Cl)c1 62325,Cc1ccc(C(=O)NCCC(C)NC(c2cnc(C(N)=O)s2)=O)c(N)n1 62326,CC(CCCCNC(C1CCC(N(C)C)C1)=O)NC(C1CC1c1cnc[nH]1)=O 62327,CCCCS(=O)(=O)CC(=O)N1CCC(NC(c2n[nH]c(C(C)(C)C)n2)=O)C1(C)C 62328,C1(C)(CC(=O)NCCOCCOCCNC(COCC=C)=O)CCC(=O)NC1 62329,C(=O)(C(C)CCC(C)(C)C)NC(CC)(CNC(c1sccc1COC)=O)CC 62330,N1(C(C2CCCN(CCC)C2)=O)CC(CNC(=O)CCc2ccco2)C(C)(C)C1 62331,c1(O)ccccc1Br.n1(CCCOC)nnnc1C(C1CC1)NCCCOCP(C)(C)=O 62332,CN=c1nc(N2CCC3(CCCOC3)C2)[nH]c(=NCC2CCOC(C)(C)C2)[nH]1 62333,c1(OC)cc(C2CC2)ccc1C(=O)NC1(C)CC(NC(=O)Cc2ccon2)C1 62334,Cc1nn(C(C)C)cc1C(=O)NC1(CNC(C2(CF)CC(F)(F)C2)=O)CCC1 62335,C1(C(=O)NCCC2(OC)CC2)CC12CCN(C(=O)CN(C)C(C)=O)C2 62336,Cc1nc(=NC(=O)CC2CN(Cc3cccc(NS(C)(=O)=O)c3)CCO2)s[nH]1 62337,Cn1ccnc1C(F)(F)C(=O)NC(CNC(C1(C2CCCO2)CC1)=O)CO 62338,c1(C(=O)NC(CN(C(=O)C(C)=CC2CC2)CC)C)cc(C2CCCO2)n(C)n1 62339,C1(NC(=O)OC(C)(C)C)COCC1S(=O)CCC(=O)N=c1ncn(-c2nccs2)[nH]1 62340,N1(C(c2ccc(C)c(C)c2)=O)CC(C2CN(C(c3cscc3C(F)(F)F)=O)C2)C1 62341,C1(C2CCN(C(C3(CO)CC3(F)F)=O)C2)(NC(Cc2c(C)cc(Cl)nc2)=O)CC1 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62360,Cc1[nH]c2ccc(Cl)cc2c1C(N1CC(NC(C2CC=CC2)=O)CC(O)C1)=O 62361,N1(C(Cc2c(OC)nccc2)=O)CCC2CN(C(c3c(Cl)cnn3C)=O)CC2C1 62362,CCCCC(CC)C(C(=O)Nc1ccc(F)cc1)N1CCCC1C1CCOCC1 62363,Cc1nc(Br)sc1C(=O)NC1CC(CNC(C2CCOC2)=O)C1 62364,C1(O)(CN(C(=O)C(O)CC2CCCC2)C)CCN(C(C2(C)CSC2)=O)C1 62365,N1(C(C2C(C)(NC(CCC(=O)N(C)C)=O)CCCC2)=O)CCOC2(CCCC2)C1 62366,S(=O)(=O)(c1cc(C(N)=O)ccc1F)NC(c1cccc(-c2nc(C)c(N)s2)c1)=O 62367,C1(C(=O)NC(C(C)(C)C)CNC(=O)C=CSc2ccccc2)CCC2CC1CO2 62368,Cc1nsc2ncc(C(N3CC(CNC(c4ccncc4)=O)CC3C)=O)cc12 62369,N1(C(C=CC(C)C)=O)CCC2(CCC2CNC(=O)CCNC(=O)C=CCl)CC1 62370,C1(NC(=O)CCF)CCCN(C(C2(C(=O)NCC3CC3)CCC2)=O)CC1F 62371,C1(CNC(c2ccc(CC)nc2C)=O)CC2COCC2N1C(c1nccn1C)=O 62372,C1(N(C(C2CC(CCC)C2)=O)CCNC(=O)C(C)c2ncco2)CCCCC1 62373,C1(C(=O)Nc2c(C(N)=O)ncs2)CC(F)(F)CN1C(=O)CCc1ccco1 62374,c1(C(=O)NCC2(NC(c3ccn(C4CCC4)n3)=O)CCC2)ccc(CO)o1 62375,C(=O)(C1=CS(=O)CCC1)N(CCC(C(C)C)NC(=O)COc1ccc(F)cc1)C 62376,N1(C(=O)NCCCCl)CC2CC1CN2C(=O)Nc1ncccc1C(F)F 62377,c1(NCC(C)OCCO)cc(=O)oc2cc(Cl)c(Cl)cc12 62378,C1(C(N2CC(OCCNC(C3CC3(C)C)=O)C2)=O)(CC)CCOC1 62379,C=C(C)C(C)(O)C(=O)NCCN(C(c1ccc(N(C)C(C)=O)cc1)=O)C(C)C 62380,C1(C(N2CC(CCC)C(OC)C2)=O)NCCOC1(C)C 62381,c1(C(=O)NC(CCNC(C(C)CO)=O)Cc2ccccc2)ncn2cccnc12 62382,CC1(CCC(=O)NCCOc2ccncc2)CN(C(c2cnco2)=O)C1 62383,c1(OC)c(C(=O)NCC(C)(C2CCC2)NC(c2ccc(CO)s2)=O)csc1C 62384,C1(C(N(C(CC)CNC(=O)COCC(C)(C)C)C)=O)CC2(CC2)CO1 62385,N1(C(c2n[nH]c(C)c2Cl)=O)CC2CCC2(CNC(=O)C=CC2(C)COC2)C1 62386,Cn1nc(C(=O)NCC23CC2CN(C(C2CCCC24CC4)=O)C3)cc1C#N 62387,C1(c2cn(Cc3c(C)cn(C)n3)nn2)CCN(C(=O)CCC(N)=O)C12CC2 62388,C1(C(=O)NC(C)Cn2cccn2)C=CCN(C(C2CCCC(=O)C2)=O)C1 62389,Cc1[nH]nc(C(C)C)c1C(N1CCCC1CNC(=O)Cn1cc(C(N)=O)nn1)=O 62390,N1(C(C2(C)COC2)=O)CCN(C(C2CCCC2n2cccc2)=O)C(CCO)C1 62391,c1(CC(=O)N(C)CCN(C)C(c2cocn2)=O)cccc2nonc12 62392,C(=O)(C1CCCc2nn[nH]c21)N1CCC(F)(CNC(c2nc(C)nc(O)c2)=O)C1 62393,N1(CC(C)C)CCN(C(c2ccc(CC(C)C)cc2F)=O)CC1=O 62394,C1(CNC(C(C2CN(C(C3(C)C=CCCC3)=O)C2)OC)=O)CCCC(=O)C1 62395,N1(C(C(CC)O)=O)CC2(C1)CN(C(c1cnc(C(C)C)[nH]1)=O)CC(C)(C)O2 62396,CCCC(O)CC(=O)N1CCN(C(C2(c3ccccc3)CC2(F)F)=O)CC1 62397,CC(C(F)(F)C(F)(F)F)=CC(=O)NCC1C2CN(c3ccnc(Cl)n3)CC12 62398,C1(C(=O)NC(C2CCOC2)C#C)CN(C(=O)CCS(C)(=O)=O)CC(C)O1 62399,C1(C)(C(N2CC(CCCC)N(C(c3n[nH]cc3F)=O)CC2)=O)CCCNS1(=O)=O 62400,N1(C(c2n(CC#C)cnn2)=O)CC(C2(NC(C3CCCSC3C)=O)CC2)C1 62401,C1(C(N2CC(C)(C)C(c3cc[nH]n3)C2)=O)Cc2ccccc2C(=O)O1 62402,c1(C(=O)NCCN(C(CC2(C)OCCO2)=O)C2CC2)ccc(Br)cc1F 62403,c1(OC(C(=O)N(CCNC(C=NOC)=O)C(C)C)(F)F)cccc(C(F)(F)F)c1 62404,c1(C(N(CC(C)NC(Cc2c(CC)cccc2)=O)C)=O)cc2n(n1)CCC2 62405,N1(C(c2cc(COC)on2)=O)CCCC2(CCN(C(=O)C=CC(C)C)C2)C1 62406,Cc1cc(Cl)c(C(N2CC(NC(=O)CC3CCCN3C(C)C)CC2C)=O)cc1C 62407,C(c1ccccc1)=CC(C(N1CCC(NC(C2(OC(C)=O)CC2)=O)C1)=O)C 62408,C1(COC)(NC(c2sccc2F)=O)CCN(C(=O)CC2(O)CCOCC2)C1 62409,N1(C(CC(CC(C)C)C)=O)CCC2CC(NC(c3ccn(C)c3)=O)CCC2C1 62410,N1(C(COC(C)(C)C)=O)CCCN(C(=O)CS(=O)(=O)Cc2cccs2)CCC1 62411,C1(C(N2CC(C#C)(C(=O)NCc3ccc(C)c(O)c3)C2)=O)CCC(C)=C(C)C1 62412,CC1CCCC(n2cc(C(C(N)=O)N(C)C(=O)OC(C)(C)C)nn2)C1 62413,Cc1cc(C(=O)NCC(F)CNC(C2CC(C)(C)O2)=O)nc(C)n1 62414,c1(NC(=O)NCC(=O)OCC)cc2cc(-c3cc(C)cs3)cnc2[nH]1 62415,c1(C(=O)NC(C)CN(C(=O)C(C)(C)N(C)C)C)nn(C)c(Cl)c1Br 62416,c1(CC)cnc(C(N2CCC(CF)(NC(c3ncoc3CC)=O)C2)=O)nc1 62417,CC1(C)C(NC(c2cccc(OC3CC3)c2)=O)CCN1C(=O)C1CC1 62418,CC1C(NC(C2(C)CCNC2=O)=O)CCCN1C(=O)COc1cc(Cl)ccc1Cl 62419,CC1(CNC(=O)Cc2sc(S)nc2C)CCCN1C(=O)C=CC1CCOCC1 62420,C1(C(N(CC)OC)=O)CC2CCCC2N1C(c1ccc(Cl)s1)=O 62421,C1(C(=O)NC2C(C(=O)NCc3c(C)nccn3)OCC2)CCOCC1(C)C 62422,c1(CC)ccc(C(N2CCC(O)CC2C(=O)NCC(=O)N(C)C)=O)cc1Br 62423,CC(C)(F)CCC(=O)NCCCNC(c1cc(-c2ccc(Cl)cc2)ns1)=O 62424,C(=O)(C(O)C(CCC)NC(c1cc(O)n(C)n1)=O)NCCC(CCC)O 62425,c1(OC)ccc2[nH]c(CC(N3CC(C)C(C)(CNC(=O)C(C)O)C3)=O)cc2c1 62426,N1(C(CC2C=CC(NC(c3nc(C)c(C)s3)=O)C2)=O)CC2CC(CO)C(C2)C1 62427,C1(CNC(=O)COCC2(F)CC2)(CC(=O)CSC2CC2)CC1(F)F 62428,N1(C(C(CCC)C(C)C)=O)CC(NC(=O)C(C)(C)CS(C)(=O)=O)CC12CCCC2 62429,C1(NC(CNC(C(C)(C)C)=O)=O)CCN(C(=O)C=CCN2CCCC2)CC1(C)C 62430,C(=O)(CCC(F)(F)CN=[N+]=[N-])N1CCN(C(C2CC(C(C)C)C2)=O)CC(O)C1 62431,O=C(CCCC(F)(F)F)NC1CC2CC(NC(c3c[nH]c4cccnc34)=O)C2C1 62432,c1(N(CCCCN(C(c2c(CC)nc[nH]2)=O)C)C)nc2ccc([N+](=O)[O-])cc2s1 62433,C1(C(=O)NCC(C)(F)CNC(=O)CC2CCCCCCC2)CCc2nncn2C1 62434,c1(CNC(NN(CC)CCO)=O)nn(C)c2cccnc12 62435,CCCCC(C(=O)N1CCC(F)C(NC(c2cocc2C)=O)C1)ON=C(C)C 62436,C(=O)(CCCNC(c1cnn(CCF)c1)=O)N1C(CC(=O)NC)CC1 62437,N1(C(C(=O)NC(c2ccco2)C)=O)CC2C3CCC(C3)C12.C12CCCN1C2=O 62438,Nc1sc2c(c1C(=O)NC1CCCC1NC(=O)C(=C1CCCCC1)F)CCC2 62439,C(=O)(C(CCCC(=O)OC)N1CCCC(C2CC2)CC1)NC 62440,N1(C(C2CCCC=C2Br)=O)CCCCC1C1CCN(Cc2cc(=O)cc[nH]2)C1 62441,Cc1cccc(C)c1C(=O)NCc1ccoc1C(=O)NCCC12CC(CO1)C2 62442,C1(CC#C)(C(=O)NCC(c2ccccc2)NC(C2C3CCCC23)=O)CCCO1 62443,c1(C(=O)NC2CC(CNC(C3CCC4CC34)=O)C2)ccc(=NCC2CC2)[nH]c1 62444,Cc1cc(N)ccc1C(=O)NCC(C)(C)CNC(C1CC2CCC2C1)=O 62445,N1(C(c2c(SC)cn(C)n2)=O)CCC(C)(C)C(CNC(=O)C(C)=CC2CC2)C1 62446,c1(C(=O)Nc2ccc(OC(C)C)cc2)cccc2oc(N(C)C)nc12 62447,N1(C(C(CCF)NC(c2n(CC)ccn2)=O)=O)CCSC(C)(C)C1 62448,C1(C(=O)NCC(CC(C)C)NC(c2cncc(F)c2Cl)=O)CCC(C)(F)CC1 62449,c1(C(N2CC(NC(C(C)O)=O)CC2(C)C)=O)csc(N=S(C)(=O)CCO)n1 62450,c1(C(=O)NC(CNC(C(C)N(CC)CC)=O)CC)cc(-c2cccn2C)[nH]n1 62451,c1(C(N2CC(NC(CC(CC)OC)=O)C(SC)C2)=O)cc(C)c(N)cc1Cl 62452,c1(OC)cccc(I)c1C(=O)OCCS(=O)(=O)C(F)(F)F 62453,c1(Cc2scc(C)n2)nc(Cc2noc(C3CCCO3)n2)n(C)n1 62454,C(CCCCCC(=O)N1CC(CC(=O)OC)CC1C)NC(C1C(COC)OCC1)=O 62455,c1(SC(C)C(N2CCN(C(C3(CCO)CC3)=O)CC2C)=O)ccc([N+](=O)[O-])cc1 62456,C(CC(C)C)(C(=O)OC(C)=O)ONC(CC1(NC(C2N(CC)CCCC2)=O)CC1)=O 62457,C1(NC(C2CC(C)N(C)CC2)=O)CC2CCC1CN2C(c1sccc1CC#N)=O 62458,N1(Cc2cnc(CC)[nH]2)CC2COCC2(CO)C1.C12CC(CN1)NC2=O 62459,C1(c2c(C(=O)NCC(=O)NCC)c[nH]n2)CCCCN1C(=O)C(C)C1CCC1 62460,C1(C(N2CCC(Cc3cccc(OCC)c3)CC2)=O)CCC(N)C(O)C1 62461,C1(CNC(c2cn(CC3(CSC)CCCCC3)nn2)=O)CC(F)(F)CN1CN 62462,c1(C(=O)NCCOC(C)(C)CNC(=O)Cc2ccon2)ccc2nccn2n1 62463,CC(C)(C)C(O)C(=O)N1CC(OCCNC(=O)C(N)=O)C1 62464,C1(n2c(CC(C)C3CC3)nc(-c3ccnn3C)n2)CC2CCC1(C)C2(C)C 62465,C12CC(O)(C1(C)C)C1(CS(=O)(=O)N2C(C)(C)C)CC1.C(CO)O 62466,c1(NC2(C)CCN(C(C3C(C(=O)OC)C3(F)F)=O)C2)cc(C)nc2cc(C)nn12 62467,N1(C(c2c(C)nco2)=O)CCOC(C)(CNC(c2cccnc2S)=O)C1 62468,c1(C(c2nnnn2C)Nc2c(CC)cccc2)cn(C)nc1OC(F)F 62469,C(C(CC1CC1)C(=O)NCCCC1CCCCO1)NC(c1c(C)nns1)=O 62470,C1(C(=O)NCC(C#C)CC2CC2)(CC#C)CCN(C(C2COCCN2C)=O)CC1 62471,C1(C(N2CC(CC(=O)OC)C2)=O)C2CCC(C2)N1C(=O)Cn1ccnn1 62472,Cc1cc(CC(=O)NCCNC(c2c[nH]nc2C(F)(F)F)=O)no1 62473,N1(CCCNC(c2c[nH]c(=N)o2)=O)CCN(C(c2ccc(C(N)=O)o2)=O)CC1 62474,C1(CC(C)C)CN(C(=O)CC2(CNC(C3CCN3C(C)(C)C)=O)CC2)CCO1 62475,C(C)(C(C(=O)NCCCCCN=[N+]=[N-])C(C)C)NC(C(C)=NOCC#N)=O 62476,c1(C(N2CCC(C(C)NC(=O)CC3(C#N)CC3)C2)=O)ccc2c(c1)CC2 62477,C1(C(=O)NC(C2CCN(C(c3nonc3N)=O)C2)C)CCCCN(C)C1=O 62478,C12(NC(CC3CCC(C)C3)=O)CCC(C(=O)NCC(C)(O)C3CCC3)(CC1)C2 62479,N1(C(C2C(CC(C)C)C2)=O)C2CCC1CC(N(C)C(c1ncncc1Cl)=O)C2 62480,Cc1ccc(Br)c(CN2CC(NC(c3cnc(O)c(Br)c3)=O)C3(CC3)C2)c1F 62481,C1(OCC(=O)NCCN2CCN(C(C3CC3(F)Cl)=O)CC2)CCC(F)(F)CC1 62482,C1(NC(C2(C)COC2)=O)CCN(C(=O)CSc2ccncc2F)CC1(C)C 62483,Cc1cccc(C(=O)NC2CC(CNC(C34CCCCC3C4)=O)C2)c1 62484,CCC(C)CC(C)C(=O)NCC1(C(N)=O)CN(C(c2ccc(OC)c(Cl)n2)=O)C1 62485,N(C1c2ccccc2CC12CCCC2)C(=O)NC(CSC)Cc1cccc(Br)c1 62486,C1(NC(c2cc(CCC)oc2C)=O)CCCN(C(c2nc(CC)no2)=O)C1C 62487,c1(C(N(C2CCCC2)CCSc2c(Br)ccc(C)c2)=O)ccc2c(c1)OCCO2 62488,N1(CC(=O)NCC(CNC(=O)CCc2n[nH]c(=N)s2)OC)CCS(=O)(=O)CC1 62489,Cc1ccc(-c2cnc(NCN3CCC(c4ncccc4F)C3)c(F)c2)cc1Cl 62490,c1(C(=O)NCC(CC=C)NC(c2ccc(NC)cn2)=O)ncccc1OC 62491,C1(CNC(C2CC(C)SCC2)=O)CN(C)CCN1C(c1cccnc1N)=O 62492,C1(C)(C(N(C2CSC2)C)=O)CCCN(C(=O)CC2NC(=O)NC2=O)C1 62493,c1(C(=O)NC(C(=O)NCC=C=C)Cn2cncn2)cc(O)ncn1 62494,C=CCC(CNC(C1CCC(CC)O1)=O)C(=O)NC1CC1CCOC 62495,C(=O)(C(C)C(F)(F)F)N1CCC(CC=C)(NC(c2cn(CC3CCCO3)nn2)=O)C1 62496,C(=O)(C1=CCC(C)CC1)N1CCC(CCNC(C2CCCC(OC)C2)=O)CC1 62497,c1(CC)nc(C(=O)NC(C2CN(C(c3cnn[nH]3)=O)C2)C)n[nH]1 62498,C1(OC)CCC12CC(C(=O)NCC(O)CCNC(C1CC3CCC1CC3)=O)C2 62499,c1(NC(C(c2ccc(OC)cc2)N2CCCC2CCO)=O)cccc([N+](=O)[O-])c1 62500,n1(CCCOC)cc(CCC2CN(C(=O)CC(C)C3CCCO3)C2)nn1 62501,c1(CC(=O)NCC2(NC(C(C)n3cccn3)=O)CCCC2)cccc(C(F)F)c1 62502,Cc1[nH]c(C(=O)NCC2CC(NC(C3CCCCC3(C)C)=O)C2)c(C)c1C 62503,Cc1csc(=NCC(=O)NCC2CC(C)N(C(c3cscc3F)=O)C2)[nH]1 62504,C1(NC(C(C)(C(C)C)OC)=O)CCC2(CCCN2C(=O)CS(=O)(=O)C2CC2)CC1 62505,CC1CCC(C(=O)NC(c2ncccn2)C)N1C(C12CC(C(=O)O)(C1)C2)=O 62506,C#CCC(C)(CNC(=O)C(CNC(=O)C(C)NC(=O)OC)CC=C)CO 62507,C1(CCC)CCCC1C(=O)N(C(C)CCNC(=O)C(C)OCc1ccccc1)C 62508,C1(NC(c2csc(CC(F)(F)F)n2)=O)CCN(C(c2cc(Cl)cnn2)=O)C12CC2 62509,c1(OC)ccc(C(=O)NCC2CCCCC2NC(c2n[nH]cc2F)=O)cc1F 62510,Cc1[nH]nc(C(=O)N(C(C)CNC(=O)C(C)CC2CCCC2)C)c1O 62511,N1(C(CC2(N(C)C)CCC2)=O)CC(C)(C)CC1CC(N1CCCC(C(F)F)C1)=O 62512,Cc1noc(Cl)c1CC(=O)NC1CCN(C(=O)CC2C=CS(=O)(=O)C2)C1C 62513,N#Cc1ccc(CN2CCC(CNC(=O)C=Cc3ccccc3F)C2)c(Cl)c1 62514,N1(C(CC(CC)CC)=O)CC=C(CC(=O)Nc2c(C)nn(C)c2C(N)=O)CC1 62515,O=C1CC2(C1)CC(C(=O)NCC(CC1CC1)C(=O)NCC(O)C1CC1)C2 62516,CC1CC2(CO1)CN(C(C1(C)C=CCN1C(=O)CCN1CCCCC1)=O)C2 62517,C1(CNC(=O)C(=O)NCC23CC(F)(C2)C3)CCCCS1.C1(C)CC1 62518,c1(C(=O)NC(CC=C)CNC(C2CCCC23CCC3)=O)ccnc2c1cnn2C 62519,N1(C(c2c(OCC)oc(C)n2)=O)CCC(N(C)C(c2cn(C)cc2C)=O)C(C)C1 62520,C12(NC(c3csc(C)c3C)=O)CC(C)(C1)OC21CN(C(C2CCC(=O)N2C)=O)C1 62521,c1(C(N2C(CNC(c3cc(OC)c(Cl)cc3)=O)CC2)=O)cc2sc(F)cc2[nH]1 62522,N1(CCc2cn(CCNC(c3c(C)nn[nH]3)=O)nn2)CC(C)OCC1C 62523,N1(C(C2(C)CCCS2)=O)CCC2(CCC2NC(c2cnc[nH]2)=O)CC1 62524,C(=O)(CC1=CCCC1)NCCC1(NC(CCc2c(C)noc2C)=O)CCOCC1 62525,C1(NC(c2cn(C)c(=O)cn2)=O)CCCC12CN(C(=O)CC1CC(C)(C)CO1)C2 62526,Cc1cc(=O)oc(C)c1C(=O)NC1CCC(F)(CNC(=O)C2=CC3CCC2C3)C1 62527,c1(C(=O)NCC23CC2CN(C(=O)CCCc2nccs2)C3)ncc2ccccn12 62528,N1(C(C(COC)C)=O)CC(NC(c2[nH]nc(C(F)(F)F)c2C)=O)C(O)C1 62529,c1(-c2n(-c3cccc(C)c3)nc(CC3CCC3)n2)nn(C)cc1S(C)(=N)=O 62530,c1(C(=O)NCC(C2CC2)NC(c2cccc3oncc23)=O)coc2c1COC2 62531,CCC(C)(CC(=O)N(CCCNC(c1ccc(O)nc1C)=O)C)C(=O)OC 62532,N1(C(C(OCC)Nc2cc3c(s2)CC(C)(C)C3)=O)CCCC(C2(OC)CC2)C1 62533,Cc1[nH]nc2ncnc(N3CCC(NC(=O)CCC(N)=O)C3C)c12 62534,c1(C(=O)NCC=CCNC(C2(Cl)C(C(C)=O)C2)=O)ccc2c(c1)NCCC2=O 62535,C(CC(N)=O)(C(=O)NCc1cc(C(C)C)on1)NC(C(CN(C)C)O)=O 62536,N1(C(c2n[nH]c(C)c2Br)C(=O)NCC=C)CCN(CC)CC1.C1CCC(=O)N1.OCC 62537,C1(CN(C)C(C2CCCCC2)=O)CCCN1C(=O)CCCc1nccs1 62538,c1(C(=O)NC2CCCC(NC(C3CCC(F)(F)C3)=O)C2)cc(F)ccc1C1CC1 62539,N1(C(CCOC)=O)CCC2(CC1)CCN(C(=O)C(C)CCC(C)(C)C)C2 62540,C1(=O)C(F)CC(C)(C)N1.CC(C)C(C)(O)CN1CC(N2CCNC2=O)C1 62541,Cc1ccc(C(=O)NCCOCCCNC(=O)CC2CC(=O)NC2=O)cc1F 62542,C1(NC(C(CC=CC)CC)=O)CCS(=O)(=O)C12CN(C(C1(CO)CC1)=O)C2 62543,n1(C(C)C)ncc2c(N3CCC(C)C3)[nH]c(=NC(C)c3cccnc3O)nc12 62544,C1(C(=O)NCC(COC)NC(C2CC=CCC2C)=O)CCCCC12CCC2 62545,CCCCC(CNC(c1ccc(=N)[nH]c1)=O)NC(=O)C(C)(C)n1cc(Cl)cn1 62546,c1(C(=O)NCc2cc(C(=O)NCC3C(C)OCC3)sc2)ccc(O)nn1 62547,O=[N+]([O-])c1ccc(OCCCCNC2CC3CCC2CC3c2ccccc2)cc1 62548,c1(C(N2CCC(CN(C(C(CC#C)O)=O)C)CC2)=O)cccn2nnnc12 62549,c1(C(=O)NCC(CNC(C2CCCS2)=O)OC)c(C)noc1C(F)(F)Cl 62550,c1(COC)nc2cccc(C(=O)N(CC(c3ccccc3)O)C)c2[nH]1 62551,c1(C(=O)NCC(=C)CCNC(=O)C(F)C2CCOC2)nn(CC)cc1[N+](=O)[O-] 62552,Cc1cc(F)ccc1NC(=O)C(=O)NC(c1ccccc1F)C 62553,c1(C(=O)Nc2ccc(OC(C)C(=O)N(C)C)cc2)cc(Br)c2occc2c1 62554,N1(C(c2n(CCC)ncc2)=O)CC2CC2(CNC(c2nn(C)cc2C)=O)C1 62555,c12cc(ncn1)NC2.c1(COC(C)CN2CCCC2=O)cnn(C)c1 62556,c1(C(N(CCC(=O)NC(CC)C(=O)NC)CC2CC2)=O)cnc(O)c(F)c1 62557,CC1CN(C(C23CC4CC2C3C4)=O)CC1NC(c1cc(N)ccn1)=O 62558,c1(-c2occ(C(=O)NCC3CC(NC(CC=C=C)=O)C3)n2)ccc(C(C)C)cc1 62559,C1(NC(C2(CC)CC2)=O)CCC2(CC1)CN(C(=O)C(c1ccc(Br)cc1)=O)C2 62560,Cn1cc(C(=O)NCC2CCCC2NC(=O)Cc2cn(C)nn2)n(C)c1=O 62561,c1(C(N2C(CNC(C3N(CC)CC3)=O)(CC)CCC2)=O)n[nH]c2c1COCC2 62562,N1(C(C(C)OCC)=O)CCn2cccc2C12CCCCC2 62563,C1(CNC(C=CC=CCC)=O)CC(O)CN1C(c1scc(C(F)(F)F)c1C)=O 62564,Cc1ccccc1-c1cc(C(=O)NC(C)COC(F)F)no1 62565,Cc1c(NC(C2CCC(C(C)C)N2C(c2c[nH]ccc2=O)=O)=O)cccc1CO 62566,c1(OC)cc(C)ccc1CNC(=O)CN(C(=O)C1=CCCC1)C(=O)C(C)C 62567,Cc1ccc([N+](=O)[O-])c(OCCCC(=O)NCCNC(=O)C(C)C2CCOC2)c1 62568,C1(CNC(C2(SCC)CC2)=O)CCN(C(C2C=CCC2)=O)CC1C 62569,c1(CC(=O)NCC2C(NC(c3cc(C)oc3)=O)CC2)ccc(C(F)(F)F)nc1 62570,N1(C(C2C(C)C2C)=O)CCN(C)C(CNC(=O)CC=Cc2ccccc2F)C1 62571,C1(NC(=O)CC2(CNC(c3scnc3Cl)=O)CC2)CCCCC1O 62572,C1(NC(C2CCN(C(c3c(CNC)cccc3)=O)C2)=O)CN(C)CC12CC2 62573,O=S(=O)(c1ccccc1)C1CC(NC(=NCC2CC2)NCC2C3CCCCC23)C1 62574,c1(C(=O)NC2C(NC(c3nc(C(=O)OC)sc3)=O)CC2)ccc2cncn2c1C 62575,N1(C(c2cccc(C)c2)C(=O)NCC)CC(O)CC2(CCCC2)C1 62576,C1(NC(C=CC(C)(C)NC(C(CSC)O)=O)=O)CCCCC12CC2 62577,c1(OC)cc(OC)nc(C(N2C3CCC2C(CNC(=O)CC2=CCCC2)C3)=O)n1 62578,c1(CNC(C(C)NC(C2CC2c2ccc(OC)cc2)=O)=O)cccc2nncn12 62579,c1(C(=O)NCC2C(CNC(c3c(C(C)(C)C)[nH]cn3)=O)C2)cc2occc2[nH]1 62580,C1(C(=O)NCc2c(C)cccc2)CCC(C)(C)N(C(C2CCCCCCC2)=O)C1 62581,C1(NC(c2c(N)nccn2)=O)CC12CCN(C(c1ncccc1Cl)=O)CC2 62582,CCC(CC(F)F)C(=O)NC(C1CCN(C(=O)Cn2cc(C)cn2)CC1)(C)C 62583,CCCC(C)CC(=O)N1CCN(C(C2CC3CC(=O)C2C3)=O)CC1 62584,C1(OCC(=O)NCC2(F)CCN(C(CNC=O)=O)C2)CCC(F)(F)CC1 62585,c1(CC)cc(C)c(C(N2CCC(CN(C(=O)Cc3csc(Cl)n3)C)C2)=O)o1 62586,Cn1nc(C(=O)NCCC2CSCCN2C(=O)CN2CCC(C)(O)C2)cc1Cl 62587,c1(C(CC(=O)N(CCN(C)C)C)NC(c2nccn2C)=O)ccc(C#N)cc1 62588,CC1CN(CC(=O)NCc2cnn(CC(F)(F)F)n2)CC2(CCC2)O1 62589,c1(C(=O)Nc2c(C)nc(-c3cnc(N(C)C)nc3)s2)ccc(O)c(Cl)c1 62590,C(N=c1nc(N2CCC(COC)CC2)c2[nH]ccc2[nH]1)C1(CC)CC1 62591,C1(C(C)CO)CCN(C(C2(C(C)C)CCCN2C(=O)CC2CCC(=O)N2)=O)CC1 62592,C1(=O)CCC(=O)NC(CCOC)CN1.C1(C(=O)NC)C(c2nc(C)cs2)C1(C)C 62593,C12(O)CCCN(CC1)C2=O.Cn1nncc1C(N1CC(n2cc(CN)nn2)C1)=O 62594,c1(C(C(=O)NCCC)N(CC(C)S(C)(=O)=O)C)snc(OC)c1Cl 62595,C1(C(N(CCCCCCNC(c2c(C)noc2C)=O)C)=O)CCN(C)S1(=O)=O 62596,C1(OC)CC(CNC(C2(C(F)F)CC(O)C2)=O)N(C(c2cc[nH]c2)=O)C1 62597,c1(C(=O)NC(CC(C)C)CNC(C2(C#N)CCC2)=O)cc(Cl)cc2ccncc12 62598,N1(C(C2=C(C)CCC2)=O)CCC2CC2(C(N(C)C[Si](C)(C)C)=O)CC1 62599,C=C1CC2CCC(C1)N2C(C1CCC(CNC(C2CCCCO2)=O)C1)=O 62600,N1(C(c2c(C)nc3ccccn32)=O)CCC(C2CCN(CC(C)O)C2)CC1 62601,C1(C(C)C)CCC(C(=O)OC2(c3cccc(Cl)c3)CC2)C(=O)N1 62602,n1(CC)c(C(=O)NCC2(C)CN(C(=O)OC)C2)cnc1O.C12CC1NC2=O 62603,C=CCS(=O)(=O)CCNC(c1ccccc1OCC(N)=O)c1nnnn1C(C)C 62604,CC(CC(N)=O)C(=O)NCC(=C1CN(C(C2(CF)CC2)=O)C1)F 62605,C1(C(N2CCC(OC)CC2)=O)C(C)OCCN1C(C1CCC1C)=O 62606,C1(CCC)CN(C(=O)CCCOC(C)=O)CC1NC(C1CCS(=O)CC1)=O 62607,CC(C)(C)C(C(=O)O)NS(=O)(=O)CC1CCCN(Cc2ccc(Cl)s2)C1 62608,c1(C(=O)NCC(C)(CO)NC(COC(C)=O)=O)cnn2cccc2c1 62609,N1(C(C23C(CN(C(CC)=O)C2)COC3)=O)CC(C)NC(=O)C2(CCN(C)CC2)C1 62610,c1(C(=O)NC(CCCC)CNC(=O)CC2CCC2)nc(OC)ccc1C 62611,C1(C(=O)NCC2(NC(C(C)O)=O)CC3CCC2CC3)COc2ccc(F)cc2C1 62612,c1(CNC(=O)NCCCCCl)cc(O)nc(O)n1 62613,c1(C(N2CCC(N(C)C(c3ccc[nH]3)=O)C2)=O)cnc(C2CC2)nc1O 62614,c1(C(=O)NCCOC2CCN(C(c3c(C)nn[nH]3)=O)C2)cnc(O)n(C)c1=O 62615,C1(CC(N2CCC(C)(CNC(C3C(=C)C3)=O)CC2)=O)CCC2(CCC2)CO1 62616,Cc1cc(NC(C)C)cc(-c2cncc(C(=O)Nc3ncc(C)cc3I)n2)c1 62617,Cc1nc[nH]c1C(=O)NC(Cc1nccs1)CO 62618,N1(C(c2c(C(C)(C)C)ocn2)=O)CCC2CCCC12C(=O)NC1CCNC1=O 62619,c1(OC)ccc(C(=O)NC2CN(C(=O)CC3COCCN3C)CC2(C)C)cc1O 62620,CN1CCC(O)(C2(C(=O)NCC(C3CC3)N(C(=O)CS(C)(=O)=O)C)CC2)CC1 62621,Cc1nc(CNC(c2ccc(CNC(c3csc(F)c3)=O)nc2)=O)sc1C 62622,CC1CN(c2nnc(-c3ccccc3)s2)CCC1NC(=O)C(C)(O)C1CCC1 62623,N1(C(c2c(C)con2)=O)CCCC2C1CCCCN2C(C1CC(C(F)F)C1)=O 62624,C1(N(C(CSCC#C)=O)C)CCCCN(C(=O)CSCCC)C1 62625,C(=O)(C(F)CC1CN(C(=O)Cc2c[nH]nc2C)C1)N(CCC)C1CC1 62626,N1(C(CCC2N(C(CC(=O)OCC)=O)CCC2)=O)CCOCC1Cl 62627,N1(C(c2c(CC)non2)=O)CCC12CN(C(c1c(C(F)F)cccc1N)=O)C2 62628,c1(OCC)ccc(C(=O)NC2(COC)CCN(C(=O)C(C(C)C)OC)C2)cn1 62629,N1(C(C2CCCC(=O)O2)=O)CCOC2CCN(C(c3cc(Cl)ccc3Cl)=O)CC12 62630,C1(O)(CNC(C(CC)OCC)=O)CCN(C(C2(c3ccnc(Cl)c3)CCC2)=O)C1 62631,C1(CCC)CN(C(=O)CNC(S(=O)(=O)CCCC)=O)CCN1Cc1n[nH]cc1F 62632,c1(C(=O)NC(C)(C)CCNC(C2CCS2(=O)=O)=O)ccc(C(O)CF)cc1 62633,N1(C(c2nc(CNC(C(C(=O)OCC)F)=O)oc2)=O)CCN(CC)C(C)C1 62634,S(=O)(=O)(c1cc(Br)cnc1N)N1CCN(C(C)C2CC2)CC1 62635,Cc1cc(F)cnc1C(N1CCCC(CNC(c2cn(C)ccc2=O)=O)CC1)=O 62636,CC1CC(CNC(=O)C(C)(C)c2ccccc2)CN1C(=O)CCOCC(F)(F)F 62637,c1(C(=O)NC2C(OC)CN(C(=O)C(C)c3ccco3)C2)cc(F)c(SC)cc1N 62638,C(CCCC(=O)N1C(CNC(C2CC2C)=O)CC2CC12)OCCC=C 62639,C1(NC(c2ccccc2)=O)CCCCC12CCCN(C(=O)COCC(F)F)C2 62640,c1(SC)ccc(C)c(C(=O)NCC2=CCN(C(c3c(F)cccc3F)=O)CC2)c1 62641,C#Cc1ccccc1NC(C1CC(O)CN1C(=O)C(c1ccc(Cl)cc1)=O)=O 62642,N1(C(COC2(C)CCC2)=O)CC2C(NC(c3cc(C#N)cs3)=O)C2C1 62643,O=C1CCc2c(C(N3CCC(CCNC(C4CCCO4)=O)C3)=O)cccc2N1 62644,C(=O)(C(C)(O)CC(C)C)NC(CCC)C(N1CCCC(C#N)C1)=O 62645,Cc1cc(C(=O)NC(C(C)NC(=O)Cc2c[nH]nc2O)C(C)C)c(O)nc1C 62646,C1(CC=C)(NC(C2CC2CC)=O)CCN(C(=O)COCCc2cccs2)C1 62647,Cc1ccoc1CC(=O)N(CC)CC1CCN1C(c1ccnn1CCN(C)C)=O 62648,C(=O)(C(C)(C)CCF)NCC1OCCN(C(COc2ccc(C)cc2)=O)C1 62649,c1(C(=O)NCC2(C(C)NC(c3n(CC)ncc3)=O)CC2)ccc(Cl)cn1 62650,c1(OC)ccc(CC(C)C(=O)NCC(C)(C)CNC(C2(C)CC2(C)C)=O)cc1 62651,C(=O)(CCCS(C)(=O)=O)NC1CC(NC(c2nc(C(CC)CC(C)C)sc2)=O)C1 62652,N1(C(C2=NNC(=O)CC2)=O)CCC2C(CCN2C(=O)C(CC(F)F)C2CCC2)C1 62653,C1(C(=O)NC2C(NC(c3c(CC)c(F)ccc3)=O)CCC2)CC12CCCCCC2 62654,C1(C(=O)NCCCOCCCNC(C(n2ccc(C)n2)C)=O)CCCCCCC1 62655,c1(C2CCN(CC(=O)N(C(C3CCCCC3C)C)CC)C2)ccc(O)cc1 62656,c1(NC(C2CC(=C)CN2C(=O)CCc2ccc[nH]2)=O)ccc(OC)nc1Br 62657,n1(CCC)cc(C(=O)N(CCCCCNC(=O)C(C2CCC2)OC)C)nn1 62658,c1(CC)c(NC(C2CCN(C(c3ccn(C4CCCC4)n3)=O)C2)C)ncnc1Cl 62659,N1(C(CC(CCC)O)=O)CC2CC1CCC2NC(=O)CCc1nnc(C)n1C 62660,c1(CC)cccc(C(=O)NCCOCCCN(C)C(c2cccc(C)n2)=O)c1F 62661,C(=O)(C1=CCCN(C(C2(CF)CC2)=O)C1)NCC1OCC(C)(C)C1 62662,C=CCC(CNC(=O)CCn1cnnn1)C(=O)NCC1CCCCCCC1 62663,C1(C(=O)NC2C(CC)N(C(=O)Cc3cncs3)CC2)CCc2nnn(C)c2C1 62664,c1(C(N(C2C3CCCCCC23)CCC(C(C)C)NC(C)=O)=O)ccnc2ccsc12 62665,N1(C(c2cccc(SCC#N)c2)=O)CC(NC(C2CSC2)=O)C2(CCC2)C1 62666,N1(CCC2CCC(C)C2=O)C(=O)CSC1(C)c1ccccc1 62667,N1(C(=O)NCC2(C#C)CCC2)CCCC(CC)C1 62668,c1(OC)nc(NC2CCCC2C)ns1 62669,N1(C(c2n(CC)nnc2)=O)CC2CCC(C(=O)N(c3csnc3C)C)(C2)C1 62670,CCC(O)C(F)(F)C(=O)NCC1C2CN(C(C3(C(=O)N(C)C(C)C)CC3)=O)CC12 62671,c1(C(=O)NC2(CNC(c3c(CC)nns3)=O)CCCC2)cc2c(cc1N)CCC2 62672,C1(C(=O)NC(CNC(C2(SC)CCC2)=O)CC(F)(F)F)CN2CCN1CC2C 62673,N1(C(C2C(C)(CC)C2)=O)CC=C(C(=O)N2CCCOCC2C)CC1 62674,N1(C(CCC(=O)OC)=O)CCC2C(CCCN2C(=O)CCCNC(C)=O)C1 62675,C=CCCCCCCC(=O)N1CCC(NC(=O)CC2(CSC)CC2)CC1C 62676,C1(C(=O)NC2CCC(NC(CC3(C)CC3F)=O)CC2)CCCCCCC1 62677,C(=O)(CC1NC(=O)c2ccccc21)NCCCC(C)NC(c1c[nH]nc1Br)=O 62678,CC1CN(C(c2cc(Br)co2)=O)CCC1NCC(=O)N(C)CCN(C)C 62679,c1(CC(=O)NCC(C)NC(c2cc(O)cc(F)c2F)=O)csc(S(N)(=O)=O)c1 62680,S(=O)(=O)(c1c[nH]c(C(=O)NC2CCN(C(c3cc(Cl)cnc3O)=O)C2)c1)N(C)C 62681,C1(CNC(c2c(C)n(C)nc2)=O)N(C(C2CCOCC2(C)C)=O)CCCC1(C)C 62682,N1(C(=O)Cc2cscn2)CCCC2(C1)CN(C(=O)CC1CC(O)C13CCC3)CCO2 62683,S(=O)(=O)(c1ccc(N2CC(CO)C3(CCC3)C2)cc1Cl)NC1CC(CC)(CC)C1 62684,CC1CC(C#N)(C(N2CCC(CNC(=O)CC3CCN(C)C3=O)CC2)=O)C1 62685,c1(C(=O)OC)cc(=NCC2CCCCC2NC(c2cc(Br)ccc2Cl)=O)[nH]cn1 62686,Cc1ccc(Cl)c(C(N2CCC(CCNC(C3CCCCO3)=O)C2)=O)c1N 62687,C1(C2CCN(C(c3ccc4cncn4c3)=O)C2)(NC(C=CCC)=O)CC1 62688,C1(O)(C(C2CC2)NC(c2cncs2)=O)CCN(C(=O)CN2CCn3nccc32)CC1 62689,c1(N2CC(CO)OCC2)[nH]c(=NCCC(O)C2CC2)nc2sccc12 62690,C1(CNC(c2nccc(CC)c2)=O)COC(C)(C)CN1C(C1CC(F)C1)=O 62691,Cc1cc(C(=O)NCC(O)CCNC(=O)C(C)C2CCC2)c2c(n1)CCCC2=O 62692,C1(C(=O)NC(CC=C)C2CC2)CN(C(=O)CCCC(=O)N(C)C)CC(C)O1 62693,C1(C(=O)NCCC(C)(C)NC(c2cc(CC)nn2C)=O)CC2(CCC2)CO1 62694,c1(C(=O)NCC(C2CCC2)NC(C2CC(OC)C2)=O)cc2cc(Cl)ccc2o1 62695,C(=O)(C(F)C(C)C)NC(C1N(C(c2nc(C(=O)NCC(=C)C)sc2)=O)CCC1)C 62696,CC1CCc2onc(C(=O)NCC(C)(C(=O)O)c3ccccc3)c2C1 62697,c1(CC(=O)N(CC(C)NC(c2cnc(O)c(F)c2)=O)CC)cnn2c1OCCC2 62698,CCC(CC)(CCNC(C1CC2(CCO1)CC2)=O)NC(C1C(C)(C)C1(F)F)=O 62699,S(=O)(=O)(c1ccncc1)NC1CCC(NC(c2ccccc2Cl)=O)C1 62700,C1(C#N)(N)CCNC1.c1(SC)ccccc1CC(c1ccnn1C)=O 62701,c1(C(N2CC(C)N(C(C3CCC4CC34)=O)CC2)=O)cnc2[nH]cnc2c1 62702,N1(C(C(=O)N(CC(F)F)C(C)C)=O)CCCCC1C1(NC(=O)CO)CC1 62703,c1(OCC(=O)NC2CC(CNC(C=Cc3c(C)ccs3)=O)C2)c(C)occc1=O 62704,N1(C(c2ccn(CC)n2)=O)CCC(C(F)CNC(c2nn(C)cc2Cl)=O)CC1 62705,C1(NC(c2cccc(C(N)=O)n2)=O)CC(F)CN(C(c2scnc2C(F)F)=O)C1 62706,c1(C(=O)NCCSCC(=O)N(C(CC)C2CC2)C)ccncc1Cl 62707,C(CCN(C)C)(C(=O)NC(C)CCCCO)NC(Cc1ccc(C)s1)=O 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62726,CC(C)C(O)C(=O)NCC(CC(=O)N1CCCC1(C)C)C1CCC1 62727,C1(CC(=O)NC2C(C(=O)Nc3cncc(OC)c3)CCC2)Cc2ccccc2C1 62728,CC(C)(C)CC(CO)NC(CC(N1CCCS1(=O)=O)c1cscc1C(F)(F)F)=O 62729,N1(C(Cc2cccc(C)c2)=O)CCN(C(=O)C(C)C2CC2)C(CCO)C1 62730,N1(C(c2ccc[nH]2)=O)CCCC(C2CCN(C(C3CCC(F)(F)C3)=O)C2)C1 62731,c1(C(=O)NC2CCCC(CC(N3C(C)CC3)=O)C2)cn2c(n1)CCC2 62732,C1(CC)(NC(=O)Cc2cnn(C)c2)CN(C(=O)C=CC(=O)N(C)C)C1 62733,CCC(CC)C(C)C(=O)NC1CCC(F)(CNC(c2n[nH]c(C)c2Cl)=O)C1 62734,C1(NCC(C)(C)C)CCCCN1C(=O)COCCN(C(=O)CN(CC(F)F)C)C 62735,c1(C(N2CCOCC(C)(CNC(C(CC)C)=O)C2)=O)cc(C)c2nc(C)nn2c1 62736,NS(=O)(=O)c1ccccc1NC(=O)CC1(O)CCN(C(C2CC2F)=O)CC1 62737,C1(CNC(C(Br)=C(C)C)=O)CC(O)CN1C(C1CCCN1C(C)C)=O 62738,C#CC1(O)CCCN(C(C2CCCC(NC(=O)C3=CCCC3)CC2)=O)C1 62739,C1(CNC(CCC(C)O)=O)CCCC12CCN(C(=O)C(=O)C(C)(C)C)CC2 62740,Cc1cnn(C)c1CC(=O)NC1(CNC(C2CC2C#N)=O)CCCC1 62741,C1(NC(c2cc(C)sn2)=O)C2CC1N(C(c1cccc(N)c1Br)=O)C2C 62742,C1(=CC(N2C(C)CCC(NC(CCN(CC)CC)=O)C2)=O)CCCCCC1(F)F 62743,C=CCCCC(N)C(=O)N1CC(N2CC(c3ccccc3)C2)C1 62744,N1(C(Cn2c(C)cc(C)n2)=O)CCN(C(c2cc(C)n(C(F)F)n2)=O)C2CCC12 62745,Cc1cc(C(=O)NCC2CC(C)N(C(=O)C=C3CCC3)C2)cc(S(C)(=O)=O)c1F 62746,N1(C(=O)CCC2CCOC2)CCN(C(=O)CSC(F)F)C(c2ccco2)C1 62747,N1(C(C2(CCCC)CCC2)=O)CCC(O)C(NC(c2ccc(C)c(OC)c2)=O)C1 62748,c1(C(N2CC(C)C(NC(c3c[nH]nc3C(F)(F)F)=O)C2)=O)ccc(Cl)c(F)c1 62749,C(CN=C(NCc1cnco1)NCC1CCCCC1(C)C)OCC 62750,C#CCC(C(=O)NCc1nc(C)cs1)NC(c1sncc1C)=O 62751,C(=O)(C(O)CC(C)C)N1C2CC(NC(c3n[nH]c(C)c3Cl)=O)(C2)C1 62752,c1(NC(c2ccccc2C(F)F)c2n(CCC)nnn2)cc(C)cc(Br)c1C 62753,C(=O)(C1CCc2c[nH]nc21)NC1(C2CCN(C(CN(S(C)(=O)=O)C)=O)C2)CC1 62754,CCCCC(=O)C(=O)N1CC(CNC(C2(CO)CCOCC2)=O)C(C)(C)C1 62755,N1(C(C(C2CCCN(C(c3c(C)scn3)=O)C2)(C)C)=O)CC2C(C1)C2(C)C 62756,C1(NC(c2cnccc2Br)=O)C(CNC(=O)C(F)F)CCC12CCC2 62757,N1(C(C2(C)CCC(C)C2)=O)CC2CCC1CN2C(C1C=CCC1)=O 62758,N1(C(C2CCn3nccc3C2)=O)C2CCC1CC(NC(C1(c3ccsc3)CC1)=O)C2 62759,C1(NC(c2c(CCC)occ2)=O)CN(C(=O)C=CC2CCC2)CCC1C(F)(F)F 62760,C(C(=O)N1CCC(C(N2C3CCC2CC3)=O)O1)C1C(=C)C1 62761,c1(C(N2CC(C)(NC(C(C)=C(CC)C)=O)C2)=O)ccnc(C(F)F)c1 62762,c1(C(=O)NCC2(C)CCN(C(=O)C(O)P(C)(C)=O)C2)nccc2ccsc12 62763,c1(C(N2CC(C)CC(C(N(CCC)CC)=O)C2)=O)c[nH]c2ccccc12 62764,c1(-c2nc(C(C3CCCO3)N)on2)cccc(-c2cscn2)c1 62765,N1(C(C(C)CN2CCOCC2)=O)C(C)C2CC1C2NC(=O)COC(F)F 62766,CC(CC(=O)N1CCC(C2CCCN2C(c2ccc(CO)cn2)=O)C1)C(F)F 62767,C1(C(=O)NCCN(C(=O)C2=NOCC2)CC)(Cc2ccccc2F)CCCCC1 62768,CCC(CCCC(=O)N(CCCn1ccnc1)C)NC(=O)C(C)N1CCCC1 62769,n1(CCNC(C(n2ccc(C3CC3)n2)C)=O)cc(-c2n[nH]cc2C)nn1 62770,c1(CCC)nc(C(=O)N(CCC)C(C)C)cs1 62771,n1(CC)ncc(C(=O)NCC2(C(C)NC(C3CCCN3C)=O)CC2)c1C 62772,C(C(C)(C)CNC(=O)C(C)(C)n1cnnn1)N(C(=O)COc1ccsn1)C 62773,CC(CNC(=O)CCc1ccsc1)(C1CC1)NC(=O)CCc1csnn1 62774,Cc1ccc(CCNCOc2c(NC(=O)NC)cccc2)c(F)c1.C1CC1.O 62775,S(=O)(=O)(c1cccs1)NC(C)C(=O)N1CCC1CNC(c1ccc(O)nn1)=O 62776,C1(CC=C)(NC(=O)C(C)CF)CC2CCC(C1)N2C(c1c(C)nc(C)nc1C)=O 62777,C(C(=O)N1CCC(C(=O)NCC(CC)CO)O1)N(CCC)C 62778,c1(N(C(C2C(NC(C=C(C)C3CC3)=O)C2)=O)C2CC2)nc(Cl)ccc1F 62779,Cn1ccc2ccc(CNC(=O)NC3CCOC4(CCC4)C3)cc12 62780,C1(NC(C(CNC(c2c(CC)cns2)=O)N(C)C)=O)CC(C)N(C2CC2)C1 62781,c1(NC(c2cccc(Cl)c2)CC)ncnc2c1CCO2 62782,c1(CCC)nnsc1C(=O)NCCC(C)(C)NC(=O)CN(C)CCOC 62783,CS(=O)(=O)c1ccc(CN2CC3C(C(N4CCCCC4CCO)=O)C3C2)c(F)c1 62784,N1(C(CCNC(NC)=S)=O)CC2CCCC2(N=c2cncc(Cl)[nH]2)C1 62785,c1(C(N2CC(CC(=O)Nc3cccc(CO)c3)OCC2)=O)ccc2cccnn12 62786,Cc1oc(-c2ccccc2)nc1C(=O)NC1CCN(C(=O)CSC(C)(C)C)CC1 62787,N1(CC)N=C(C(=O)NC2CCC(NC(=O)C=CC(C)(C)C)C2)CCC1=O 62788,c1(OC)cccnc1C(F)(F)C(=O)NCC1CCCN(C(=O)C(CO)N(C)C)C1 62789,N#Cc1cccc(C(=O)NCC(CNC(=O)CC2CCC(=O)N2)C(F)(F)F)c1 62790,N1(C(c2c(C)ccc(C)n2)=O)CC2CCCN(C(=O)C#CC3CCCCC3)C2C1 62791,C1(C(=O)NCCN(CCC)C(c2nocc2C(C)(C)C)=O)CC=CCO1 62792,Cc1cc(CNCC2CN(c3nccc(-c4cccnc4)n3)CCO2)cc(C)n1 62793,c1(C(=O)NC(CC)CN(C(=O)CN(C)CC)C)c(C)c(Cl)cc(C)c1N 62794,C1(NC(c2cc(OC)no2)=O)CC2CC1CC2C(=O)N(c1cnn(C(C)C)c1)C 62795,N1(C(C2(CCOC)CCC2)=O)CCCC(NC(=O)C(C#N)C2CC2)CC1 62796,N1(C(C=CC(CC)C)=O)CC(NC(=O)C=Cc2ccc(C(N)=O)cc2)C2(CC2)C1 62797,CCC(C)C(=O)NCC(=O)NCCC(C)(C)NC(=O)CC(C)n1cccc1 62798,C(=O)(C1CCOc2ccccc21)NC(C)C(C)(C)NC(c1scnc1Cl)=O 62799,C12(C(=O)NC(C#CCC)(C)C)CC(C)(CN1C(=O)Cc1cncc(C)c1)C2 62800,C1(C(=O)NC2C(CNC(CCN(CC(F)(F)F)C)=O)CC2)CC2CCC1O2 62801,N1(C(C(C)OCC)=O)CCC(CNC(=O)Cc2cccc(F)c2F)C(F)(F)CC1 62802,N1(C(C(C=C)(C)C)=O)CCN(C(c2cc(F)c(OC)c(Cl)c2)=O)CC12CC2 62803,C1(C(C)NC(=O)CNc2cc(CCO)on2)CN(C(=O)CN(C)C)CCCO1 62804,C12CN(CCO1)C(=O)CC2.c1(C(C)NC(CN2CCC2)=O)ccn(C)n1 62805,c1(CCC(=O)NC23CC(NC(c4c(COC)cc[nH]4)=O)(C2)C3)cccc(Cl)c1 62806,c1(C(=O)NC2COCCN(C(C3(CC(C)C)CCC3)=O)C2)cc(Cl)c(F)cc1Cl 62807,c1(C(N(C(C(=O)NCCC)C)CC2CCCO2)=O)ccc(CN(C)CCC)o1 62808,C1(N(C(CNC(C(CC)C)=O)=O)C)CCCN(C(c2ccnc(S)c2)=O)C1 62809,N1(C(CSS(C)(=O)=O)=O)CCCC(NC(c2ncc(Cl)cc2F)=O)C(F)C1 62810,c1(C(=O)NC2CC(NC(c3ccc(Cl)nc3O)=O)C2)cc2nn[nH]c2cc1F 62811,C1(O)(CNC(C2CC2(F)F)=O)CCCN(Cc2cc(F)cc(Br)c2)C1 62812,C=CCC(C)C(=O)N(CC(CC)NC(=O)CC=CCc1ccccc1)C 62813,C=CCC(C(=O)N1CCCCC1CCC(C)(C)NC(=O)CCSCCC)OC 62814,N1(C(C(CCC)CC)=O)C(C)CC2CN(C(c3cc(Br)c(N)cc3C)=O)CC12 62815,N1(C(COCCNC(CSCCC)=O)=O)CC(O)C2(CCCC2)C1 62816,c1(CNC(C2CCC(NC(=O)Cc3ccc(Cl)nc3)CC2)=O)cnc(F)c(Cl)c1 62817,C1(N(C)C(c2ccc(C3CCOC3)s2)=O)CCN(C(C2CCOCC2)=O)C1 62818,C(=O)(C(CNC(=O)C=C(C)C(C)C)CC(C)C)NCCC(CC)(C)O 62819,c1(C(=O)NCC(C)N(C(=O)C(O)Cc2ccc(F)cc2)C)coc2c1COC2 62820,c1(C(N2CC(COC)(NC(=O)CO)C2)=O)nc(C(C)C)oc1C.c1(CO)nc[nH]n1 62821,Cc1nc(C(F)(F)F)sc1C(C)N(C)CC1CC(CC2CC2)CO1 62822,Cc1cc(C(N2CC(CC(C)NC(=O)CC3CC4CC3C4)C2)=O)cc(C)c1C 62823,C1(NC(c2c(OC)nsc2)=O)CCN(C(=O)C=CCN(C)C)C1C 62824,N1(C(c2c(NC)nccc2)=O)C2CCC1CC(C(=O)NC1CC(C)(C)C13CC3)C2 62825,Cc1c(NC(c2csnn2)=O)cccc1C(=O)N(C)C 62826,Cc1cnc(C(=O)NCc2ccc(C(C)NC(C3C4COCC34)=O)cc2)c(C)c1 62827,O=C(C(O)C(F)F)NCCC1CCCCN1C(=O)CCN(C1CCCCCC1)C 62828,Cc1[nH]nc2c(C(N3CC(NC(c4cn(C)cn4)=O)CC3C)=O)cccc12 62829,c1(C(N(CC(C)NC(C2CC3CCC2C3)=O)C)=O)cnc2c(c1)N(C)CCO2 62830,C(=O)(C(C)C(=O)N1CCC=CC1C(=O)N(CC(O)CO)C)OC 62831,C1(NC(Cc2c(C)non2)=O)CCCCC1CNC(c1coc(Cl)c1)=O 62832,C(=O)(C(O)CSC1CC1)NCCC1(C(N(CC(COC)C)C)=O)CCC1 62833,c1(C(=O)NC2CC(NC(c3cc(C)c(C)s3)=O)C(O)C2)cnn2c1CC(C)CC2 62834,C(C)(C(=O)N1CC(O)(NC(=O)CC2CCOCC2)C1)(C(C)C)NC(C)=O.C1CN1 62835,c1(C(=O)NCc2cccc(Br)c2F)c(F)cccc1[N+](=O)[O-] 62836,Cc1ccc(CCC(=O)NC(CNC(=O)Cc2ccn(C)n2)CO)c(Br)c1 62837,O=C1CN(C(C2C3CCCC23)=O)C(C(=O)NC2CC3CCC2O3)CN1 62838,N1(C(C(CC=CC)C)=O)CCN(C(c2n[nH]cc2F)=O)CC1CCOC 62839,C1(NC(C(C(=C)Cl)(C)C)=O)COC2CN(C(=O)CCN(c3ncccn3)C)CC12 62840,C1(C(=O)Nc2cccc(CNC(C(C=C)(F)F)=O)c2)CCC2CCC(=O)N12 62841,c1(C(=O)NCC2OCCN(C(C=CC)=O)C2)cc(C(C)C)cc(Br)c1 62842,c1(C(=O)NC2CC(C)(NC(CC(CC)(C)C)=O)C2)cc2cccc(OC)c2o1 62843,C(=O)(C(C)(C)C(C)(F)F)NCC1N(C(CNC(=O)OCC=C)=O)CCOC1 62844,c1(CNC(NC(CC)CC)=NCc2ccc(C)c(Cl)c2)nc2ccccc2o1 62845,c1(OCC)cc(NC(=O)C(=O)NCC2CCN(c3cccc(C)c3)C2)cc(Cl)c1 62846,CCC(CC(=O)NCc1ccoc1C(N1CCC(OC2CC2)CC1)=O)OC 62847,c1(C(N2CC(C(=O)NC(CCCC)CO)C(O)CC2)=O)cc(F)c(F)c(F)c1 62848,c1(CN)ccccc1.C1(OCC)CN(C(=O)C2CC2)C1.C1(O)C(=O)N1C(C1CCC1)=O 62849,C1(NC(=O)C2=CCCS2)CCC2(CC1)CN(C(C1CC3(CCC3)C1)=O)C2 62850,N1(C(COCC)=O)CCCC1CCCNC(=O)C(CC1(C)CC1)c1ccccc1 62851,c1(CC)ccc(F)cc1C(N1CC(C)(NC(=O)CN(C2CCSC2)C)C1)=O 62852,C(=O)(C(C)CC(C)(F)F)N1CCC(C(C)NC(c2ccc(-c3cccs3)[nH]2)=O)CC1 62853,CCC(C)CC(C)C(=O)NCc1cn(CC(N2CCN(C)CC2C)=O)nn1 62854,c1(OC2CCN(Cc3ncc(C)nc3)CC2)c(F)cc(F)cc1Br 62855,N1(C(C2C(c3ccc(C)cc3F)C2)=O)CCCN(C(c2cscn2)=O)C(CO)C1 62856,CC1(NC(=O)C(F)C2CCOC2)CCCN(C(=O)C=CBr)C1 62857,N1(C(C(CC=C)NC(=O)Cc2ccoc2C)=O)CCS(=N)(=O)CC1 62858,N1(C(C2CN(C(C(C)NC(=O)OC)=O)CC2F)=O)CC2C3CCC(C3)C12 62859,C1(C(N(C(CC(=O)N(C)Cc2ccc(C)cn2)(C)C)C)=O)CC2(CCCO2)C1 62860,CC(O)CCCCCC(=O)N1CCCC1C(C)(C)NC(c1ncccc1Br)=O 62861,N1(C(CN2CCC(C)C2)=O)CCCCC2(CCN(C(=O)COc3ccsn3)C2)C1 62862,CC(C)CCC(=O)NCCN(CCOCCO)C(c1ccc(=O)oc1)=O 62863,c1(C(=O)NCC2CC(C)N(C(=O)C=Cc3cncs3)C2)cccc2sccc12 62864,c1(C(N2CC(OCCNC(c3c(OCC)nccc3)=O)C2)=O)ncc(N)nc1C 62865,C1(CNC(C=CCCC(C)C)=O)CN(C(=O)C(C)C(C)(C)C)C2(CCC2)C1 62866,C1(NC(C(C)Cn2ccnc2)=O)CCS(=O)(=O)C12CN(c1nnc(O)s1)C2 62867,C(=O)(CCCC(=O)N(C)C)NCC(C)(CO)NC(C(CNC(C)=O)C)=O 62868,N1(C(C(C)SCC)=O)CCC(NC(c2ccc3c(c2)CCC=C3)=O)C(F)(F)CC1 62869,C1(CN(C(=O)C(F)C2CCCC2)CC)CCCN(C(C2CC2C(C)(C)C)=O)C1 62870,C(CCC(C)(C)C(=O)NCC1CC1(C)C)NC(C(CC(=O)OC)C)=O 62871,Cc1cc(C(N2CCC(CNC(=O)CCc3nnc(C)o3)C23CC3)=O)cc(N)c1 62872,c1(CNC(=NCCCSC)NCc2cc(C(C)C)no2)cc2c(s1)CCCC2 62873,N1(C(C(C2N(C(C(CN(C)C)O)=O)CCC2)(C)C)=O)CC(O)C(O)C1 62874,c1(CC(=O)OC)ccc(NC(c2ccc(F)cn2)c2nnnn2C(C)C)cn1 62875,C1(CC(=O)OC)CN(C(=O)CCCc2c[nH]c3ccccc23)C2(CCC2)C1 62876,Cc1ccc(C(C)C)cc1NCC(=O)N(C1CN(C(=O)C(O)CN(C)C)C1)C 62877,C1(NC(CN2C(C)CCC2)=O)CCCC12CN(C(=O)Cc1cnoc1)C2 62878,C1(C(=O)NC(C2OCCN(C(C(C)NS(C)(=O)=O)=O)C2)C)CCC(N=[N+]=[N-])CC1 62879,c1(C(N2C(C)(CNC(CS(CC)(=O)=O)=O)CCC2)=O)cc2ccc(Cl)cc2s1 62880,c1(CN2C(C(=O)Nc3c(C(C)C)n(C)nc3)CC(O)C2)cc2ccccc2[nH]1 62881,C1(NC(C2(C)CCN(C(c3cnn(C)n3)=O)C2)=O)CCOC12CCCC2 62882,c1(CNC(C2CN(C(=O)NCCCl)CCO2)=O)ccc(Cl)c(Cl)c1 62883,CCCCC#CC(C)(C)NC(C1CN(C(C2(C)CCCC2O)=O)CC1C)=O 62884,C1(C(N(CCCNC(=O)C#CC2CCCC2)CC)=O)CCCN1S(=N)(=O)N(C)C 62885,c1(C(=O)NC2CC3(CN(C(CCSCCC)=O)C3)C2)nccc(C#N)c1F 62886,C(=O)(C(CC)CCOC)NC1(CC=C)CCN(C(=O)C=CCOC)C1 62887,C(CC(C(C)(C)C)NC(C1(C)CSC1)=O)N(C(c1c(OC)scc1)=O)C 62888,C1(NC(C(CSC)c2ccccc2)=O)CN(C(c2ccc(=N)[nH]c2)=O)CC1(C)C 62889,C(=O)(C(C(C)C)NC(=O)CC1(N(C)C)CCC1)NCC(CCC)OCC 62890,c1(CCC(=O)NC2CC2NC(C2CN(S(C)(=O)=O)C2)=O)ccc(F)cc1Cl.C1CC1 62891,C1(CNC(=O)NC2CCN(Cc3cccnc3)CC2)CC2C=CC1O2 62892,C(=O)(C(O)C(C)(C)C)NC(C)CC1CN(C(=O)C(F)=C2CCCC2)C1 62893,C1(C(=O)NCC(C2(O)CN(C(C=C(C)Cl)=O)C2)(C)C)CC2(CCCCC2)C1 62894,C1(CC)CN(C(C23CC4CC2C3C4)=O)CCC1NC(C1(C(F)F)CCOCC1)=O 62895,C(=O)(CCC(C)CN(C)C)NCC(c1cccc(C)c1)NC(CN(CCC)C)=O 62896,Cc1cccc(C(C(C)C)NC(=O)C(C2CCCC(=O)N2)F)c1 62897,C=CC(CC)C(=O)N1CCC(C(=O)NC2(CO)CC2)C1C 62898,C1(N(C)C(C2CCCS2)=O)CN(C(c2c[nH]c(C#N)c2)=O)CC12CC2 62899,N1(C(C2(OC)CCCC2)=O)CC(CNC(c2scnc2C(C)C)=O)OC(C)(C)C1 62900,C1(CNC(CC)=O)CC2CC1CN2C(=O)COCc1cccc(C)c1 62901,N1(C(Cc2c(C)noc2)=O)CC(C)N(C(=O)CC2(CO)CC2)CC1C 62902,C1(c2nnnn2C(C)(C)C)(NCCC2(OCC)CCC2)CC2CCOC12 62903,c1(CN2C(CNC(C3CCOCC3)=O)CCC2)cc(=O)n2ncsc2n1 62904,c1(C(N(CC(C)N(C(CCC)=O)C)C)=O)cc2cccc(C(F)(F)F)c2nc1O 62905,N1(C(C(C#C)(C)C)=O)CCC(C)(C)C(CNC(=O)COc2ccc(OC)cc2)C1 62906,C1(C(N2CCC(CCN(C)C)C2)=O)CC2(CCN1C(=O)C(Cl)Cl)CC2 62907,c1(CC(=O)N(C(C)CCNC(=O)CO)C)cc(F)c(N)cc1F 62908,C1(NC(C(C)SCC)=O)CCCCC12CCN(C(c1n[nH]cc1C1CC1)=O)CC2 62909,CC(C)(C)CC(O)C(=O)NC12CCCCC(NC(C3CSC3)=O)(C1)C2 62910,O=C1NCCc2occ(C(N3CCCC(CNC(=O)C(F)(F)CF)C3)=O)c21 62911,Cc1nc2cccc(C(=O)OCC3=CCOCO3)n2n1 62912,c1(C(N2CCN(C(C(C)N(C(C)=O)C)=O)C(C(F)F)C2)=O)c(F)cc(F)cc1F 62913,C(=O)(C(CC)C(F)(F)F)N1CC2C(CNC(C(C=C)CC)=O)(C2)C1 62914,CC(CC(F)F)C(=O)NC1(CNC(=O)CC2CN3CCN2CC3)CCCC1 62915,C1(CNC(c2ccc(SC)o2)=O)CCCCC1NC(C1CCN(CC(C)C)C1)=O 62916,C(CCSC)(C(=O)N(CC(O)CNC(C1(c2cc[nH]n2)CC1)=O)C)OC 62917,Nc1cc(F)cc(Cl)c1C(=O)NC1COCC1NC(C1CC1C(F)F)=O 62918,C1(C(N(CCn2cc(C(c3ccccc3)C)nn2)CC)=O)CCn2ncnc2C1 62919,O=C(C#CC1CCOCC1)NCCN(C(c1ccc(CO)o1)=O)CC1CCCC1 62920,N1(C(C2(C#C)CC2)=O)CC2(CO)CC1(C(=O)NC(c1ccc(C)cn1)C)C2 62921,N1(C(c2c(O)ccc(C)c2)=O)CCCN(C(=O)C(O)Cc2cnc[nH]2)C(C)C1 62922,N1(C(C2(C#N)C(C)(C)C2)=O)CC2(CC(C(N3CCOC(C#N)C3)=O)CO2)C1 62923,c1(C(=O)NCC(C2CCC2)NC(C(C=C=C)C)=O)cnc(C)c(C)c1 62924,N1(C(c2cn3ccsc3n2)=O)CC2CN(C(C3CC34CCCCCC4)=O)CC2C1 62925,C(=O)(C1=C(F)CN(C(=O)CCS(N)(=O)=O)CC1)NC1CCCN(CC)C1 62926,c1(C(=O)NC(=O)CCCc2ncco2)cc(C(F)(F)F)c(Br)cc1F 62927,C1(NC(CCOCC(C)C)=O)C2CC(O)C1N(C(C1(C)CC(=O)N(C)C1)=O)C2 62928,Cc1cc(CNC(=O)CCCOCCC(C)C)ccc1C1CC1 62929,c1(N(CCCCN2CCOCC2)C)nc(=N)[nH]c(=NCC2CC3CCC2C3)[nH]1 62930,CC(C)CC(C)CC(=O)N1C(C(=O)NCCCC(O)CO)CC1C 62931,N1(C(C2(NC(c3c(C)nc(O)cc3)=O)CC2(C)C)=O)CCCN(C)CCC1 62932,c1(C(=O)NC(CN(C(c2cc(CO)c(C)o2)=O)CC)C)c(C)noc1C(C)C 62933,CC(C)CC(C(=O)N(C)CCN1CCCCC1)N(C(=O)C(C)n1cccc1)C 62934,C1(CN2CCC(CNC(c3c(C)snn3)=O)C2)CCS(=O)(=O)CC1 62935,C(=O)(C1COc2ccccc21)NCC(CCNC(c1nc(Cl)cs1)=O)O 62936,S(=O)(=O)(CCC(=O)N(C(C(=O)NCC1(C)CNC(=O)O1)C1CC1)C)NC 62937,Cc1cc(C(C)C(=O)NC2C=CC(CNC(=O)CC(C)(C)F)C2)cc(F)c1 62938,C=C(C)CCCC(=O)NCC1CCC(CNC(C2(C#N)CC23CCC3)=O)CC1 62939,c1(C(=O)NCCC2(NC(c3ccnc(O)c3)=O)CCC2)ncnc(O)c1F 62940,C1(CNC(C2N(CC)CC2)=O)CCC2(CN(C(c3oc(Br)cc3C)=O)C2)O1 62941,CC1(CNC(C2CCCN2C(=O)C2CC2)=O)CCN(C(c2cnc(O)s2)=O)CC1 62942,c1(CC)cnc(O)c(C(N2CC(C(C)NC(C3CN(C(C)=O)C3)=O)C2)=O)c1 62943,C1(CNC(C(CC)C#N)=O)CN(C(c2cc(Br)no2)=O)C2(CCC2)C1 62944,C1(C(=O)NC2(C)CCN(C(Cc3cc(C)no3)=O)C2)CC(=O)NC1(C)C 62945,N1(C(CN(C2CC2)CC)=O)CC(C)C(C)(C(=O)NCC2(C)CC(O)C2)C1 62946,c1(C(N2C(C(=O)NC(CC(=O)OC)C)CC3CC32)=O)cc(F)c(F)cc1I 62947,C(=O)(CC(O)CC(C)(C)C)NC1C(NC(C=Cc2c(C)cccc2)=O)C1 62948,C1(NC23CC(C(=O)OCC)(C2)C3)CS(=O)(=O)CC1C(c1nc(CC)oc1C)=O 62949,c1(C(=O)NCC(C(C(C)C)C)NC(c2cccnn2)=O)cc2ccc(Cl)cc2o1 62950,N1(C(CCCOCC)=O)C2CCC(C2)C1C(=O)NCc1ccc(O)nn1 62951,N1(C(CCCCN(C(=O)Cc2cc[nH]c2)C)=O)Cc2cccc(F)c2C1 62952,c1(NC(c2cc(CNC(=O)C(C3CCCCC3)O)ncc2)=O)cccc(F)c1F 62953,c1(C(N(C(CC2(OC)CCCC2)=O)C)C)nc2cccc(C)c2[nH]1 62954,C1(NC(c2n(C3CC(F)(F)C3)nnn2)c2ncc(C(F)(F)F)s2)CCC(F)(F)C1 62955,N1(C(COC2(C)CCC2)=O)C(CNC(=O)CCn2cc(Cl)cn2)CC2COCC12 62956,N1(C(C2CCN(C(C(C)(O)C3CC3)=O)C2)=O)CCc2cnccc2C1 62957,c1(C(N2CC(NC(c3c(C)scn3)=O)C(C)(C)C2)=O)cnc2c(c1)CCC2 62958,N1(C(c2ccc(C(C)(C)C)s2)=O)CC2CC1CN(C(=O)CC#N)C2 62959,C1(NC(CS(N)(=O)=O)=O)CCN(C(c2ccoc2Br)=O)CC12CCC2 62960,N1(C(=O)C=Cc2ccncn2)CC2CC(C1)CN(C(=O)Cc1ccno1)C2 62961,c1(C(=O)NC(CCNC(C(C)C#N)=O)(C)C)cc2c(ncn2C)[nH]1 62962,c1(SCC(=O)NC2C(NC(C3C(CC)C3)=O)C2)n[nH]c(=N)s1 62963,CCCC(C(=O)N1CC2CC2(CNC(=O)CCF)C1)c1ccccc1 62964,C1(C(=O)NC2(C(=O)Nc3c(CC)n(C)nc3)CCCCC2)CC(C)CC(C)C1 62965,C1(CCC)CCC(C(=O)NC2CCN(C(c3cc(Br)nn3C)=O)C2C)CC1 62966,C1(CC(=O)NC2C(OC)CN(C=O)C2)CC2(CCC2O)C1.c1ccc(Cl)cc1 62967,c1(OC)cc(CC(=O)NCCC2CSCCN2C(c2cc(Cl)c(Cl)[nH]2)=O)ccn1 62968,c1(CN2CC3C(NC(c4cccc(N5CCCC5)c4)=O)C3C2)ccc(Cl)cc1I 62969,C1(C(N2CCSCC2)=O)(NC(C2CC(C(F)F)C2)=O)CCOCC1 62970,Cc1csc(C(=O)NC2CN(C(c3cnoc3C3CCC3)=O)C2)c1Br 62971,c1(-n2ncc(C(=O)NCC3(F)CC(CNC(C4C(C)C4)=O)C3)c2)ccccc1F 62972,C1(NCC(COC2COCC2)(C)C)CCC(=O)N1C 62973,c1(C(=O)NCc2ccc(OC)nc2C)c(F)ccc2c1OCO2 62974,C1(C)(N2CCC(N(C)CCn3nc(Cl)ccc3=O)CC2)CCS(=O)(=O)C1 62975,C#CCCCC(CC)N1C2CCCC2OC(=O)CC1.c1(OC)ccccc1 62976,C1(C(N2CC(CC=C)(NC(=O)Cn3cc(C)cn3)C2)=O)CC12CCC(F)(F)CC2 62977,c1(CC(=O)OCc2ccc(C(=O)OC)cc2)cccc2ncccc12 62978,N#Cc1cnc(C(N2CC3CC(NC(C4CCC(=O)NC4)=O)CC3C2)=O)c(Cl)c1 62979,c1(CN2CCCC(CC(=O)NCc3cc(Cl)cnc3Br)C2)cc(Br)cc(F)c1O 62980,CCC(C)CCC(=O)N1CCCCC1CCNC(c1cc(C)on1)=O 62981,c1(C(C)C)nc(N(C)C)cc(N(CC(O)CN(C)C(C2(C3CC3)CCC2)=O)C)n1 62982,c1(C(=O)NC2CCCN(C(Cc3onc(C)n3)=O)C2C)ccc2c(c1)CCOC2 62983,c1(CC(=O)NC2CC(CCNC(C(CSC)C)=O)C2)ccccc1N1CCCC1 62984,C1(C(=O)NCc2c(C(=O)NC(C)(C)CCCF)n(C)nc2)CN2CCC1CC2 62985,c1(CC(=O)N(CCCNC(C(C)=C2CCC2)=O)C)csc2c(F)cccc12 62986,c1(OC)cc(NC(N2CCC(N3CC(F)(F)C3)CC2)=O)cnc1Cl 62987,c1(C(N2CCC(C)(C(=O)NCC(N3CCCCC3)=O)C2)=O)cc(F)cc(I)c1 62988,C1(C2CN(C(c3ccncc3)=O)C2)(NC(c2nc(C(C)OC)oc2)=O)CC1 62989,C=CC1OCCC1C(=O)NCC1(NC(=O)CC2CC2(C)C)CCC1 62990,c1(NC(C)=O)ccc(C(=O)NC23CC2CN(C(c2cc(=O)n(C)o2)=O)C3)cc1F 62991,C12CCCC3(CCN(CC3)C1=O)O2.C(CC(=O)NC(C1CC1)C1CC1)OC(C)C 62992,C1(C(N(CCN(C)C(c2ccc(CC(C)(C)O)s2)=O)C)=O)C(F)(F)C12CC2 62993,c1(C(C)(C)C(=O)NCC2(CNC(C3CCCOC3)=O)CC2(F)F)cccc(F)c1 62994,c1(C(=O)NC2(C)CCN(C(=O)CNC=O)C2)ccc2ncccc2n1 62995,Cc1ccc(CC(N2CCC(F)C(NC(c3cc(Cl)c(Cl)cn3)=O)C2)=O)cc1C 62996,N1(c2c(C#N)ccnn2)CC2CCC(NC(c3ccc4nc(O)[nH]c4c3)=O)CC2C1 62997,C12(NC(Cc3ncc(CC)[nH]3)=O)CCCN(C(c3cncc(Cl)c3Cl)=O)CC1C2 62998,c1(C(=O)NC2CC(N(C(CCC(C)N(C)C)=O)C)C2)nn(C)c2ccc(F)cc12 62999,n1(CC(=O)NCC(C)NC(CCNC(=O)NC)=O)ccc(=O)c2ccccc12 63000,CCC(C(=O)OC)C(=O)NC1COCCC1NC(C1(Cc2cccnc2)CC1)=O 63001,c1(NC(c2cnn(C)c2)CC)ccc(S(=O)(=O)NCCc2n[nH]c(=N)s2)c(Cl)c1 63002,Cc1nn(C)cc1CC(=O)N(C1CCN(C(C2CC2c2ccn(C)n2)=O)CC1)C 63003,N1(C(c2c(Cl)cn(CC)n2)=O)CCC2C(CCN2C(=O)C(O)C2CCCC2)C1 63004,Cc1cnccc1C=CC(N1CC=CC(NC(C2CCNC(=O)C2)=O)C1)=O 63005,C(CC1CNC(=O)Cn2cc(nn2)O1)OC.C12CC(C1)NC(=O)C2.C(C)(=O)OC 63006,N1(C(c2ccn(CC)n2)=O)CC(OC)CC1CNC(=O)C1=CCCS1 63007,N1(C(c2c(Cl)nc(N(C)C)s2)=O)CC(CNC(=O)C(C)(O)C(C)C)CC1(C)C 63008,C12(C(=O)NCCC(C)NC(=O)C=CCOC3CCOCC3)CCOC(C)(C1)C2 63009,c1(C(N2CCOCC2Cc2cccc(Br)c2)=O)cccc(-c2nn[nH]n2)c1 63010,CC1Cc2cc(C(=O)NC3CCCCN(C(C4CC5CCC4O5)=O)C3)ccc2O1 63011,C1(C)(N(C)C)C2CC1CN(C)N1CCC3(CCC3)C(O)C1C2 63012,C1(NC(c2cncc(OC)c2)=O)CN(Cc2ccc(O)c(F)c2)CC(F)(F)C1 63013,CC(CN(C)C)CCC(=O)NCC1CC(C)(C)CN1C(C12CSCC1C2)=O 63014,c1(C(N2CCC(NC(CCOCCC)=O)C23CCC3)=O)ccc(S(C)(=O)=O)cc1 63015,C(=O)(C(C)(COC)OC)NC(CNC(C=NOC)=O)Cc1ccccc1 63016,c1(C(=O)NCC(CN(C(COCC#C)=O)C)O)ccc2c(c1)nc(C)c(=O)n2C 63017,N1(C(C(CNC(C2(C)CC2)=O)O)=O)CCC2(CCCO2)C1 63018,C1(CC(=O)NC(C(C)C)(C)CNC(=O)CCc2nncs2)CCCCC1(C)C 63019,CC(CC(=O)N1CC(C)(C)CC1C(N1CC2CCCC2C1)=O)C(C)(C)C 63020,C1(C(C(=O)NC(CC)(C)C)N(C(C)CC(N)=O)C)CCCC1O 63021,c1(C(=O)NCCC2(C)CC2)csc(CNC(=O)CN2CCOCC2)c1 63022,C1(C(N(CC(COC)O)C)=O)(CO)CCCN(C(c2cc(C)co2)=O)C1 63023,Cc1nc(C(N2CCCC(C(C)C)C2)C(=O)NCc2nnn(C)n2)c(Br)[nH]1 63024,C(C(O)C(=O)NC1CC(CNC(C2CCCN2Cc2ccccc2)=O)C1)SC 63025,c1(C(=O)NCC2C3N(C(c4ccn(C)n4)=O)C(CC3)C2)ccc(N)c([N+](=O)[O-])c1 63026,N1(C(c2cc(CNC(C3CN4CCN3CC4)=O)ncc2)=O)CCCCCC1CO 63027,c1(OCCCC)ccc(C(=O)NCCC(C)CCNC(C2CCS2(=O)=O)=O)cc1 63028,C1(CCC(=O)N(C2CCN(C(=O)Cc3nncn3C)C2)CCC)CCCCO1 63029,c1(NC(C(CNC(C(C)c2ccsc2)=O)N(C)C)=O)cn(C)nc1Cl 63030,N1(C(C(C)=CC(C)(C)C)=O)CCC(CC(N2CC(F)C2)=O)C1 63031,N1(C(CC(C)(C)OC)=O)CCCC1C1CCCN1C(c1cc(Cl)cc(F)c1N)=O 63032,c1(OC)ccc(C(=O)N(CC(O)CNC(c2ocnc2C2CCC2)=O)C)cc1F 63033,C1(F)(CNC(=O)Cc2cccc3sccc23)CC2CCC(C1)N2C(=O)CCF 63034,Fc1cc(F)c2nc(Cl)nc(N3CCC4(CC3)CC(N3CCCOCC3)C4)c2c1 63035,c1(CO)cccc(C2(CO)CC2)c1.c1(C(c2ccsc2)N)nnnn1CCC1CC1 63036,C1(COC)(NC(C2OCCN(C)C2=O)=O)CCCN(C(C2(F)CCOC2)=O)C1 63037,N1(C(C(CCC2CC2)NC(c2c(C)snn2)=O)=O)CCc2nncn2CC1 63038,CC(C)C(CC(=O)NCC1(CO)CCCO1)NC(C1CC2(C1)CC2(F)F)=O 63039,Cc1ccc(C=CC(=O)NCCCCNC(c2nocc2C(C)C)=O)cc1Cl 63040,C1(C(N2CC(O)(CC=C)C2)=O)CC(F)CN1C(C1CC(C)=NO1)=O 63041,C(CC1=CCN(C(c2ncn3cccnc23)=O)CC1)NC(C1C(C)C1)=O 63042,C#CCCCC(=O)N(C)CCOCCCN(C)C(C1CCC(CCO)CC1)=O 63043,C12(C(N(CCC(C)NC(=O)CCc3nc[nH]n3)C)=O)CCCCN1CCC2 63044,CC1(C)CCC(C(N2CCC23CCCSC3)=O)CN1C(=O)Cn1cnnn1 63045,Cc1cc(CNC(C2COCCN(C(C3CCC=CCCC3)=O)C2)=O)nnc1C 63046,COn1cnc(C)c1C(=O)NCC(CC(F)(F)F)NC(C1CC(CN(C)C)C1)=O 63047,C(CCCC(C)(c1nnnn1C1CCOC1)NCc1ncc(Br)s1)OC 63048,N1(C(C2N(N=O)CCCC2)=O)CC2C3CCC(C2C1)N(C(C1(Cl)CC1)=O)C3 63049,c1(CNC(c2csc(CNC(c3[nH]ccc3C3CC3)=O)n2)=O)cccc(CO)n1 63050,c1(CN(c2ccnc(NC(C3CCOC3)CC)n2)C)c(C)cccc1C 63051,C1(CNC(C2(OC)CC2)=O)CC(NC(c2sccc2C)=O)C12CCC2 63052,c1(C(=O)NC2C(NC(C(C)(Cl)Cl)=O)CCCC2)cc2n(n1)CCCO2 63053,N1(C(CN(C)CC)=O)CCCCC(CNC(C23CCCC2CCC3)=O)CC1 63054,c1(CCC(=O)NCC2(C(=O)NC3CC(CN(C)C)C3)CC2)ccc(F)c(Cl)c1 63055,C1(NC(C=C(C)C)=O)CN(C(=O)Cc2cccc3ncccc23)CCC12CCC2 63056,CC1(C)NC(=O)CC1C(=O)NC1CCCN(C(c2cnn(CCO)c2)=O)CC1 63057,C1(C(N(C2CCNC2=O)CC)=O)CN(C(C2CC3CC(=O)C2C3)=O)CC1(F)F 63058,C1(CC)CN(C(C23CCC(CC2)C3)=O)CCN1C(c1ccc(CC#N)cc1)=O 63059,c1(CC)occc1C(=O)NCCN(C(c1cc(C(C)=O)cs1)=O)CC1CC1.C=O 63060,N1(C(C(CC2CCC2)OC)=O)Cc2occ(C(N3CCC(CCO)C3)=O)c2C1 63061,c1(NC(C2(C)N(C(c3c(C)cc[nH]3)=O)CC2)=O)cc(N(C)C)cc(C#N)c1 63062,CC(C)S(=O)(=O)C(C)C(=O)N(C)CC1(O)CN(C(C2C(F)(F)C23CC3)=O)C1 63063,c1(C(N2CC(NC(CCCC(C)C)=O)C(C#N)C2)=O)ccc2nc(Cl)sc2c1 63064,C=C(C)C(C)(C)C(=O)N1CCC(C2CCCN2C(=O)CN(C2CCCC2)C)C1 63065,n1(CC(=O)N(C(C(C)C)C)C)cc(CNC(C2CCC(=O)O2)=O)nn1 63066,c1(C(=O)NCC(CNC(C2(C)CC(F)(F)C2)=O)F)ccn2ccccc12 63067,N1(C(CCC=C(C)C)=O)CCCC(C2CCN(C(C3(C)CC(O)CN3C)=O)C2)C1 63068,c1(SC)ccccc1CC(=O)N(C1CN(C(=O)Cc2ccc(Cl)nc2)CC1O)C 63069,N=S1(=O)CCC2(CC1)CN(C(=O)C(N)Cc1ccco1)CCO2 63070,N1(C(CSCC(C)=O)=O)CCC(N(C(=O)CN2CC=CC2)CC2CC2)C1 63071,CCCC(CCC)C(=O)NCC(C)NC(=O)CN(C)C(c1cc2c(s1)CCC2)=O 63072,C=CCC(CN=c1[nH]c(=NC)[nH]c(=NCC(C(C)C)SC)[nH]1)c1ccccc1 63073,C1(CNC(c2c(C)con2)=O)CC2(CN1C(=O)CNC(=O)C(F)(F)F)CC2(F)F 63074,c1(CC(C)C)cc(C(=O)NC2CCCC2NC(c2ccc(Cl)o2)=O)n(C)n1 63075,C#CC1(N(C)C)CCN(C(C(=O)NC2CCOC2)c2ccoc2)CC1 63076,c1(C(N2CC3C(N(C(c4cn(CC)nc4C)=O)C)C3C2)=O)c(F)cc(N)cc1F 63077,c1(C(N2C(COC)C(C)(C)C2)C(=O)NCCC#N)cc2ccc(Cl)cc2o1 63078,c1(C(=O)NCC23N(C(c4c(C)nccn4)=O)CCC2CC3)cc(F)c(Cl)cc1F 63079,C1(C(N2CCC(C(C)(C)NC(c3c(C)noc3C)=O)C2)=O)CC2(COCCO2)C1 63080,C1(CNC(=NCC=C)NC(C)CC)CS(=O)(=O)c2ccccc2O1 63081,c1(C(=O)NC(CCCNC(c2c(CC)con2)=O)C)cc(O)c2ccccc2c1 63082,N1(C(CCCCOC)=O)CCCCC2(C1)CN(C(c1[nH]c(C)nc1C)=O)C2 63083,c1(C(=O)NCC2(F)CC(NC(CC3N(CC)CCC3)=O)C2)ccc(OC)cc1 63084,c1(C(N2CCc3nc[nH]c3C2)=O)cn2cc(-c3cccc4cc[nH]c34)ccc2n1 63085,c1(CC)nn(C)c(-c2scc3c2OCCO3)c1N=S(C)(C)=O 63086,CCCCCCC(C)CC(=O)N1CCC(NC(=O)C#CC(C)(C)O)C1 63087,c1(C(=O)NCC(CC)NC(C2(F)CCS(=O)(=O)C2)=O)cc2c(C)sc(C)c2s1 63088,C1(CC=C)(NC(=O)C(C(C)O)c2ccccc2)CCN(C(=O)CN(C)CC)CC1 63089,C(=O)(C(CC(C)(C)C#N)N1CCCC(C)(C)C1C#N)Nc1ccc(OC)cc1 63090,C1(CNC(c2c(C)sc(Cl)n2)=O)CN(C(c2n[nH]cc2C2CCC2)=O)CCN1C 63091,N12CCC(C(F)(F)CC1)CNC(=O)OCc1c(OC)ccnc1C2=O.C(C)(C)(C)OC.C 63092,c1(CC)cc(C(=O)N(CC(C)CNC(=O)CC2CCCN2C(C)C)C)cc(Cl)c1 63093,C1(C(=O)Nc2cn(CCC#C)nc2)CCCN(C(=O)C(C)=C2CCCC2)C1 63094,C(CNC(=O)CNS(=O)(=O)NC)(CCCC)NC(C1(C#C)CCC1)=O 63095,N=c1nc(N2CCCC(n3nccn3)C2)[nH]c(=NCc2cccc(CO)n2)[nH]1 63096,N1(C(C#CC(C)(C)O)=O)CC(CNC(C2CCCC2)=O)N2CCC1C2 63097,c1(N2CC(CNC(C3(C)CS(=O)(=O)C3)=O)OCC2)ncccc1[N+](=O)[O-] 63098,c1(CC(N2CCN(C(=O)C(O)C(F)(F)F)C(CO)C2)=O)c(F)cccc1F 63099,C1(CCC)CCCC1C(=O)NC1(CC(=O)NCC2(N(C)C)CC2)COC1 63100,c1(C(=O)NC2C(NC(COc3ccc(C)cc3)=O)COC2)cc(F)ccc1F 63101,c1(C(=O)NCC2CC(NC(C(C3CCCC3)OCC)=O)C2)ccn2nncc2c1 63102,c1(C(=O)NC2(C)CN(C(=O)C(C)(C)c3ccno3)C2)scc(Cl)c1Cl 63103,c1(C(=O)NC2C(C)CN(C(=O)CCC(F)F)C2)n[nH]c2c1CC(C(C)(C)C)CC2 63104,C(=O)(C(C)C(C)(C)c1ccccc1)NCC(CC(C)C)NC(CC(COC)C)=O 63105,C1(C(=O)NCC(CCC)O)CC(NC(=O)CCC2(C)N=N2)C(O)C1 63106,C1(NC(C(CNC(CSC)=O)O)=O)COCC1(C)C 63107,Cn1cc2cc(C(=O)NCCC(C)(C)CNC(c3c[nH]c(=N)o3)=O)ccc2n1 63108,C1(CNC(CC2(C=C)CC2)=O)C2CCC(C2)N1C(=O)Nc1cccc(OCC)c1 63109,c1(C(=O)NCCOC2CCN(C(C(COC)(C)O)=O)C2)cc(Cl)c(C)cn1 63110,C(=O)(CC1C(=O)Nc2cc(Cl)ccc21)NC(C)CNC(=O)Cc1ccc(O)nc1 63111,c1(C(N2CC(NC(C(CC)OCC)=O)C2)=O)cc2sccc2s1 63112,C1(C(=O)NC(C(=O)NCC(C#C)OC)CC2CC2)CCCC(O)C1 63113,c1(Cn2cc(CC3N(C(Cn4c(C)ccn4)=O)CCC3)nn2)c(Cl)cccc1Cl 63114,C#CCCCCCC(=O)NC1CCC(NC(=O)CC2CCN(C)C2=O)CC1 63115,c1(NCCCN2C(C)CCC2)nc(N2CCC(CN(C)C)C2)nc2c1ncn2C 63116,N1(C(CC(CC)OC)=O)CC(NC(=O)C(c2ccccn2)C)CC12CCOCC2 63117,N1(C(c2c[nH]c(=N)o2)=O)CCC2(C1)CN(C(c1cscc1Br)=O)CCO2 63118,N#Cc1c[nH]c(C(=O)NC2CN(C(C3CC34CC4)=O)CC2n2cccn2)c1 63119,Cc1ccc(C=CC(=O)NCCN(C)C(C2CN(c3nnnn3C)C2)=O)o1 63120,N1(C(C(C(C)C)OC)=O)CC(C(=O)NCCc2ncccc2F)C(C2CC2)C1 63121,N1(C(CC(CC)(F)F)=O)CC2CCCCC2(CNC(=O)CCc2cnc[nH]2)C1 63122,CON(CCC(=O)N1CC(O)C(O)CO1)C(C)(C)C1CCOC1 63123,C1(C(=O)NC)C2CCC(C2)N1C(=O)Cn1c(C)ccc1C 63124,Cc1ccc(C=CC(N2CCC(C(O)CNC(c3cnc[nH]3)=O)CC2)=O)o1 63125,C(CCCCC(=O)NCC1=CCCC1)N(C(=O)C(F)CC1CCOC1)C 63126,CCCC(C)(C)CC(=O)NC1CC=C(C(=O)NC(c2ccnn2C)CC)C1 63127,CCCCC(C)(F)C(=O)NCc1nc(C(=O)NCc2cccnc2C)co1 63128,C(C)(C(=O)N(O)Cc1cn(C2CCCC2O)nn1)Oc1ccc(C)cc1 63129,c1(C(=O)NCCC2CC(NC(CCOCC)=O)C2)nc(C)sc1C 63130,N1(C(c2c(C)nc(Br)o2)=O)CC2(CCN(C(c3cccc4[nH]ccc34)=O)CC2)C1 63131,c1(OCC)cccc2c1C(C(=O)N1CC(NC(C3(F)CC4(CCC4)C3)=O)C1)CC2 63132,N1(C(C(C)Sc2nccn2C)=O)CCCC(O)(CNC(c2cnn(C)n2)=O)C1 63133,C(=O)(CCCCO)NCC(=O)NCCCCC1CN(C(COC(CC)C)=O)C1 63134,Cc1ccc(F)c(C(=O)NC2CC(C(F)F)(NC(c3n[nH]cc3C)=O)C2)c1 63135,c1(OC)cnc(C(=O)NCC2CCN2C(C2CC(O)C2)=O)cn1 63136,CCC(C)(C)C(O)C(=O)NCC1CCN(C(=O)Cn2ncc(C#N)c2N)C1(C)C 63137,c1(-c2cn(C3C(NC(C(C=C=C)C)=O)COC3)nn2)cc(F)c(F)cc1F 63138,N1(C(C2(COC)CC=CCC2)=O)CCCC(N(C(=O)COC(F)F)C)CC1 63139,c1(OC)ccc2cc(C(C)NC(=O)NC(C)CCC(C)C)oc2c1 63140,C12(C(=O)Nc3sc(C(=O)OCC)c(C)c3C(N)=O)CCC(F)(CC1)CC2 63141,c1(OCC)ncccc1C(=O)NCCOCCN(C(=O)CC1CCC1(C)C)C 63142,c1(OC)ccc(CCC(N2CC(F)(CNC(=O)C=C(C)C(C)C)C2)=O)cn1 63143,C1(CC(C)C)CN(C)CCN1C(=O)NC1CCC(O)C(C)C1 63144,c1(OC)ccccc1CC(C)CC(=O)N(C)Cc1ccc(Br)cc1 63145,c1(NCC(C)(C2CC2)NC(C2CC3CCCC23)=O)ncccc1C#N 63146,N1(C(CCCC)=O)CC2ON=C(CNC(c3cn(-c4cncc(F)c4)nn3)=O)C2C1 63147,C1(NC(c2coc3c2COC3)=O)CC2(CCN(C(C3(CO)CC3(F)F)=O)CC2)C1 63148,O=C(C(F)C(F)(F)F)NC1CC2(C1)CN(C(=O)CCc1ccc(F)cc1)C2 63149,N1(C(CCc2ccc(C)nc2C)=O)CC2CCCC2(c2cn(CC(N)=O)nn2)C1 63150,N1(C(C(C)(C2(C)CC2)OC)=O)CC2C(CNC(C3CCC=CCC3)=O)C2C1 63151,CC1N(C(=O)C(C2CCNCC2)F)CCCC1(C)C 63152,c1(SC)ncc(Br)c(=NC2CC2C(=O)NCCn2nc(C)nc2C)[nH]1 63153,N1(C(C(C=C)O)=O)CCC2(CC2NC(=O)CC(C)C(F)F)C1 63154,Cc1cnc(C(=O)NC2(C)CCCN(C(=O)CC3CCOC3)C2)c(Br)c1 63155,C1(OCC)CC(N(C(c2cc(C)sc2C)C(=O)NCc2cccs2)C)C12CCC2 63156,C1(CCCCC)(NCCn2cc(C)nn2)CCCC1.N12CCCC1C2=O.S(C)(=O)(=O)NC 63157,N#Cc1cccc(C(O)C(=O)NCc2ccnc(OC3CCCCC3)c2)c1 63158,O=C(C1=CC2C=CC(C1)C2)NCCCC(O)C(=O)NCCCC(F)F 63159,Cc1cncc(C)c1C(=O)NCC(O)CNC(=O)C(c1ccccc1)F 63160,C12(CNC(C3C(C)CC3)=O)CCC(CC1)N(C(c1cnn3c1CCCC3)=O)C2 63161,C(CNC(c1cnc(Br)s1)=O)(CC(C)C)NC(CN(CC)CC)=O 63162,C1(C)(C(=O)NCC(=O)N(C)CC)CCC2CC2C1.C12CCN(CC1)C(=O)C2 63163,C(CCC)(C(=O)NC(C)(CNC(c1c(C)n[nH]c1C)=O)C1CC1)=CCC 63164,c1(C(=O)NC2(CNC(C(C)(C)OC)=O)CCCCC2C)nnc2ccccn12 63165,c1(CNC(N2CCC(CSC)C2)=O)c(N2CCN(C)CC2)cccc1Br 63166,c1(C(N(CCCNC(COCCOCC#C)=O)C)=O)ccncc1Br 63167,N1(C(C(C)(C)NC(=O)NCC)=O)CCN(CCNC(C2COCC(C)O2)=O)CC1 63168,N1(C(C(C(CC)C)O)=O)CC2CCC(N(C)C(c3ccc(C(C)=O)cc3)=O)C2C1 63169,CCN1C(=O)C(N)C(c2ccccc2F)c2cccc(OCC3CC3)c21 63170,N1(C(c2nc(CC)sc2)C(=O)NCCCSC)CCc2nnnn2CC1 63171,C1(C(N(C)Cc2ncc[nH]2)=O)CN(C(C2CC(F)(CF)C2)=O)CC1F 63172,C1(OC)CC2(C1)CC2NC1CCN(C(=O)OC(C)(C)C)C1 63173,C(=O)(C(F)C(C)CC(C)(C)C)NCC1CC(CNC(CC(C)SC)=O)C1 63174,Cc1ccc(-c2nc(CCN3CCCCC3)cs2)cc1.N12CCN(CC1)NC2=O 63175,C(CC1CCCCC1)(CCNC(=O)C(F)(F)c1cccnc1)OC.C(=O)C1CC1 63176,c1(C(N2CC(O)(C(C(=O)NCCOCCCC#C)F)C2)=O)cnc(S)nc1 63177,CC1CS(=O)CCN1C(=O)C(Cc1cnc[nH]1)NC(C1CCC(C)(O)CC1)=O 63178,N1(C(C=CCCC(C)C)=O)CCCC1(C)C(=O)NC(c1cnsc1)C 63179,C1(C(=O)NC(CN(C(c2sc(CO)nc2C)=O)CC)C)CCC2(CCOCC2)O1 63180,C1(NC(C2(CF)CC2)=O)CC2CC(NC(C3CC(O)C3)=O)CC12 63181,Cc1nccc(C(=O)NC2CC(CNC(c3cc(C(C)C)on3)=O)C2)c1C 63182,c1(CCNC(CCC=C(C)C)c2nnnn2C)c[nH]c2cccc(OC(C)C)c12 63183,Cc1nc2ccccc2cc1C(=O)NCC(CO)NC(=O)C(O)CC[S+](C)C 63184,CC1(C(=O)O)CC(F)(F)CN1C(c1nc(C2CC2)n(-c2ccccc2)n1)=O 63185,N1(C(C2(COC)CC2)=O)CCCC(NC(C2CC23CC(O)C3)=O)CC1 63186,C(=O)(C1CCCn2cc(C(C)(C)C)nc21)OC(=O)NCC(n1c(C)cc(C)n1)C 63187,Cc1cc(-c2cn(CCOc3sc(C)cc3Br)nn2)n(C)n1 63188,C1(OC)CC(C(N2CC3CCCC(C2)N3C(=O)C(F)=C(C)C)=O)C12CCOCC2 63189,CC1CCC(C)N1C(C)C(N1CC(O)(CCNC(=O)Cc2cnnn2C)C1)=O 63190,c1(CN(C(c2ccc(I)s2)C(=O)NCCOC)C)ccc2nc(O)oc2c1 63191,C1(C(=O)NC2C=C(C)CCC2)C(C)OCCN1C(=O)Cc1cccnc1C 63192,c1(C(N2CCC(C(CNC(CCCC#C)=O)(C)O)CC2)=O)ccc2c(c1)CC2 63193,c1(C(=O)NC2C(CNC(C(C)C#N)=O)COC2)cc(Cl)cc2c1CCC2 63194,N1(C(C2CCC(CNC(COC)=O)C2)=O)CC2OC(=O)N(C)C2C1 63195,C1(C(=O)NCCC=C=C)CCN(C(C2CC2(F)Cl)=O)C12CC2 63196,C1(NC(C(CC)O)=O)CC(F)CN(C(c2ccccc2C2CCCC2)=O)C1 63197,CC(C)CC(O)C(=O)N(C(C)C(=O)NCc1ncn(C(C)C)n1)C 63198,c1(CC)n[nH]c(CC)c1CC(=O)NC1CN(C(=O)COC2CCC2)CC1C(F)F 63199,C1(CNC(c2cnn(C(F)(F)F)c2)=O)CN(c2cnc(F)cn2)CCO1 63200,N1(C(c2c(C)nc(COCC)s2)=O)CCC(NC(C2CC3(CCC3)C2)=O)C(F)C1 63201,C1(C(=O)NC(C)CNC(C2(CF)CC2)=O)CCC2(CCC2)CC1 63202,c1cccc(OCC)c1.C(CN=C(NCC1CC1)NC1CC1)c1scc(C(=O)OC)n1 63203,N1(C(CC(C)(C)OC)=O)Cc2nccn2CC(NC(C2(F)CCCOC2)=O)C1 63204,O=C1CC(C(=O)N2CCCC2CCNC(C2CSC2)=O)=NN1 63205,c1(C(=O)NCC2CCC(C(=O)NC3(CC)CCOC3)C2)ccnc(C)n1 63206,N1(C(C(CC)C)=O)CCCOC(CNC(c2ccccc2COC)=O)C1 63207,CC1(C)C(C(=O)NC(CNC(C2CCOC2)=O)C2CCC2)C1C#N 63208,Cn1c(-n2cc(C3CCCN3CC(F)(F)C(C)(C)O)nn2)nc2ccccc12 63209,c1(CC(=O)NCC2(OC)CN(C(c3sc(N(C)C)nc3C)=O)C2)ccc(Cl)nc1 63210,C(=O)(CCCCC(F)F)N1C(CNC(c2cc[n+]([O-])cc2)=O)C(C2CC2)CC1 63211,C1(NC(c2ccc(C)s2)=O)C=CCN(C(c2cnnn2C)=O)C1 63212,C(C)(CNC(=O)C=C(Cl)Cl)(C(C)C)NC(CCc1cc(C)[nH]n1)=O 63213,CC1(C)C(NC(=O)CC2CCC=CCC2)CCN1C(=O)C(c1cc(F)ccc1F)=O 63214,c1(CCC(=O)N(C2CCCN(C(=O)CCC#N)C2)CC)cncnc1O 63215,c1(C(N2CCC(C(C)NC(=O)CC3(O)CCC3)C2)=O)ncc(F)cc1N 63216,c1(C(N2CCC(COC)(NC(C3CC(=O)N(C)C3)=O)C2)=O)c(Cl)ccnc1C 63217,C1(C(=O)NCCC2OCCN(C(c3c(OC)cncn3)=O)C2)CC2(CCOC2)C1 63218,c1(C(N(C2CCC(NC(c3c(C)cc[nH]3)=O)C2)C)=O)nc(C2CC2)ncc1Cl 63219,N1(C(c2c(C(=O)OCC)c[nH]c2)=O)CCC(C)C(CNC(=O)CSC(F)F)C1 63220,c1(OC)cc(C(=O)NCC(CO)NC(=O)CC2CC=CCC2)cc([N+](=O)[O-])c1Cl 63221,Cc1c(N)ccc(C(=O)NCC(C)CNC(=O)CN2OC(C)(C)CC2=O)c1C 63222,c1(C(C)C)nc(NCCC2CC2c2ccccc2C)cc(=NC(C)C2CCC2)[nH]1 63223,N1(C(C)=O)CC(CC(=O)NCC2(CO)CCC2)CC1C 63224,c1(C(N2CCC(CCNC(c3c(CCC)occ3)=O)C2)=O)cccc(F)c1Br 63225,CCC(C)(C(=O)N1CCC(OC)CC1)OCC1CCN(C(=O)C(C)(F)F)C1 63226,C1(NC(C=CCOC)=O)CC2CC1N(C(=O)C(F)C(C)(C)O)C2 63227,N(C1CN(C(=O)C=Cc2ccc(Cl)cc2)CCc2ccccc21)C(C)=O 63228,C#CC(C)(C)C(=O)NC(CO)CCCNC(=O)CCCc1cnn[nH]1 63229,c1(OCC)cc2cc(C(=O)Oc3ncnc(C)c3F)[nH]c2cc1OC 63230,C(CC(F)F)(C(=O)NC1CCCN(C(C)C)C1)NC(c1cn(CC)nn1)=O 63231,N1(C(C(C)CO)=O)CCCCC(C2CN(C(C3CC4(CC4)C3)=O)C2)C1 63232,Cn1ccc2ccc(C(=O)NCC3CCC(NC(C4CCCCO4)=O)CC3)cc12 63233,N1(C(CC2C(C)(C)OCC2)=O)CC2(CCCC2)C1C(N1CCOC(CCO)C1)=O 63234,n1(CC)ncnc1C(=O)NC(CC(N)=O)c1ccccc1 63235,c1(C(=O)OC)ncccc1CN1CCC(F)(C(=O)Nc2ccc(SC)nc2)C1 63236,c1(C2CN(C(C3OCCCO3)=O)C2)ccc(Br)nc1 63237,CCCC(C)(CC)C(=O)N1CC(CO)C(CCO)C1 63238,C1(NC(C=C(C)Cl)=O)CC2CCC1N2C(c1c(C)nn(C)c1-n1cc(C)cn1)=O 63239,C(CC(C(=O)N1CCCCC1CCNC(c1cc(SC)oc1C)=O)NC=O)SC 63240,N1(C(c2cc(OC)ncc2Cl)=O)CC2CN(C(c3ccc(C#N)n3C)=O)CC2C1 63241,N1(C(c2c(C)scn2)=O)CCC2(C1)CN(C(c1nc(C3CC3)cs1)=O)CC(C)O2 63242,C#Cc1ccc(C(=O)N(C(C)C(N2CCCC(F)CC2)=O)CCC)cc1C 63243,CN(C)NC(=O)CCC(=O)N1CCC2(NC(c3c[nH]c(=N)o3)=O)CC2C1 63244,CN1CCC(C(=O)NCC2CC2NC(c2cc(C#N)c[nH]2)=O)CC1 63245,N1(C(c2cc(C3CC3)on2)=O)CC2CCN(C(C3CC3C3CCOCC3)=O)C2C1 63246,N1(C(CC(=O)NCC)=O)CCC(NC(=O)COCC)CC1 63247,Cc1cccc2cc(C(=O)NCCCN(C)C(C3(O)CCOCC3)=O)nnc12 63248,CCCCCC(CC)C(=O)N1CC(C)(C)CC1CC(=O)Nc1cc(C)cc(C)c1 63249,C1(C(=O)NCC2CC(OC)C2(C)C)(CC)CCCN(C(=O)C(F)C(C)C)C1 63250,C1(C(N(CCCCNC(C2CC(OC)C2)=O)C)=O)CC2(C1)CC21CC1 63251,C1(NC(C(C)OCC=C)=O)C2CC1N(C(C1CCCCC1c1nc[nH]n1)=O)C2 63252,c1(C(N2CC(C(=O)NC3CC34CCC4)C3(C2)CC3)=O)cc2ncccc2[nH]1 63253,CN1CC(C)(C)CC1C(N1CCC1CC(N1CCCC(CCF)C1)=O)=O 63254,c1(CNC(C2CC3CCC2N3C(C2(O)CC2)=O)=O)cc(F)ccc1O 63255,CCCCCS(=O)(=O)CC(=O)NCC(CNC(=O)CC(F)F)C(F)(F)F 63256,c1(NC(C(CC#C)NC(c2cc(Cl)n[nH]2)=O)=O)ccc2c(c1)CCO2 63257,N1(C(COCCSC)=O)CCC(F)CC1C(=O)NCC1CC(F)(F)CO1 63258,N1(C(=O)CCCOc2ccccc2)CC2CC(C1)N(C(=O)Cn1ncnn1)C2 63259,c1(CNC(CC2CCC(NC(CN3C(C)CCC3)=O)C2)=O)nc2ccccc2o1 63260,Cn1c(C(N2CC(NC(c3ccc(C(C)(F)F)cn3)=O)C2)=O)cnc1S 63261,N1(C(C(CN(C)C)(C)C)=O)C2CCCC1CC(NC(c1cc(N)c(F)cn1)=O)C2 63262,C(=O)(C(=O)NOCCOC(c1ccc(F)cc1)Sc1cccc(Br)c1)OC(C)(C)C 63263,C(=O)(CCCCCCn1cc(CC2(CO)CCC2)nn1)NC(CC)CC(C)O 63264,CC(C)CC(CC(=O)NCCCCNC(=O)CC(C)C1CC1)CC(N)=O 63265,c1(C(N(CCCNC(C23CCC2C3)=O)C)=O)cc2c(s1)CCCCC2 63266,C(C)(C(=O)N(C)OC)S.C1(OC)(OC)CCC1C(=O)NC1(CF)CCC1 63267,N1(C(c2ccc(C(=O)NC)nc2)=O)CCC2CN(C(C3CC3(C)C)=O)CC2C1 63268,O(NC(=O)C(c1ccoc1)NC(=O)CC1CC2CC2C1)CCCOC 63269,N1(CCn2nc(C)c(C)c2C)CCCC2(CN(C(c3ccnn3C)=O)CCO2)C1 63270,c1(C(=O)NC2(C(=O)NCC(C)C(C)(F)F)CC2(C)C)n[nH]c2c1CCC2 63271,N1(C(C2CCC3N(C(c4c(C)ccnn4)=O)C2CC3)=O)CCc2ccncc2C1 63272,c1(C(=O)OCC)nn(C)c(C)c1CNCC1NC(=O)CC1(C)C 63273,C1(C(=O)NCC(=O)NC(C=C)C2CCC2)CC(C)CC(=O)N1 63274,N1(C(c2c(C(C)=O)cn(C)n2)=O)CC(CNC(=O)C(O)C(F)F)OC2(CCC2)C1 63275,C1(NC(C(C)Cc2ccccn2)=O)COCCN(C(=O)Cc2cnnn2C)C1 63276,C1(NC(C2CC(OC)C2)=O)(CO)CCN(C(c2cn(C(C)C)nc2Br)=O)C1 63277,Cc1[nH]nc(C(F)F)c1C(=O)N(CC(O)CN(C)C(C1CCS1(=O)=O)=O)C 63278,Cc1ccc(F)cc1C(N1CC(CNC(=O)Cc2cn(C)nc2C)CCC1C)=O 63279,N1(C(C(C)=CC)=O)CCN2CCOCC2(CNC(c2ccc(C)c(Cl)c2)=O)C1 63280,Cn1ncc([N+](=O)[O-])c1C(=O)NC1C2CN(C(=O)COC(C)(C)C)CC12 63281,N1(C(C2OCC(=O)C2)=O)CC2CCCC(NC(=O)C(=O)C(F)(F)F)C2C1 63282,N1(C(C2CCN(C(C)=O)CC2)=O)CCCC2(NC(=O)CCNC(=O)N(C)C)CC2C1 63283,C1(NC(c2cccc(F)c2)=O)CCCC(O)C1 63284,N1(C(C2C(C)(COC)C2)=O)CCC2(CCC(CNC(=O)CN(C)C(C)C)O2)CC1 63285,C12(C(=O)NC3CCN(C(=O)CCC=CBr)CC3)CCCC1CCC2 63286,CCCCCCCc1cn(CC(C)NC(c2cc(C)co2)=O)nn1 63287,N1(C(=O)CC2CC23CC3)CC(C2CCCN(C(C3(F)CC4(CCC4)C3)=O)C2)C1 63288,C1(CNC(CCCSC)=O)CN(C(c2cc3cc[nH]c3cn2)=O)CC(C)(C)O1 63289,c1(C2(C(N3C4CC(NC(CN(C)C(N)=O)=O)(C4)C3)=O)CC2)c(F)cccc1Br 63290,Cc1ccc2c(c1)CC(C(=O)NCC(O)CNC(C1(C(F)F)CCC1)=O)O2 63291,C1(OCCOC)CC2CN(C(=O)C(c3ccco3)NC(=O)Cc3ccns3)CC12 63292,c1(OC)ccc(O)c(C(N2CCOC(CNC(=O)C(O)CC(N)=O)C2)=O)c1 63293,C(CN=c1cc(C)nc(-c2cccc(F)c2)[nH]1)OCCN(C(CCCOC)=O)C 63294,c1(CC(=O)NCC2CCN2C(C2CN3CCN2CC3)=O)c[nH]c2ncccc12 63295,C1(C(N(C2CCCC(O)C2)C)=O)(NC(c2ccncc2N)=O)CCOCC1 63296,c1(CN2C(C(=O)NCCCCCCN(C)C)CC2)cc(Cl)cc(Cl)c1 63297,N(C1CCOc2ccc(C(=O)O)cc21)C(N1Cc2c(C(N)=O)coc2C1)=O 63298,N1(C(C2N(C(CCC(=O)NCCC)=O)CCC2)=O)CCC(CO)C(C)(C)C1 63299,C1(C)(NC(C=CC(C)NC(=O)Cn2cnnc2O)=O)CC2(CCC2)C1 63300,C(C(CC)(CC)C(=O)N1CC2CC(C)(C)C2C1)NC(C(CCC)OC)=O 63301,c1(C(=O)NC2C(C)CN(C(c3scnc3C3CC3)=O)CC2)ccc(S(N)(=O)=O)[nH]1 63302,Cc1oc(Cl)nc1C(=O)NC1(C(=O)N(C)Cc2cnn(C)c2)CCSC1 63303,c1(C(=O)NCC(C)CNC(C2CCOC2C)=O)ccc2c(c1)CNC2=O 63304,N1(C(Cn2c(C)ccn2)=O)CCC(C(N2CC(N3CCCC3)C2)=O)C1C(C)C 63305,N1(C(COC2(C)CCOCC2)=O)CC2COCC2(C(=O)NCC2CCCS2)C1 63306,N1(C(c2c(CC)[nH]nc2Cl)=O)CCCC2C1CCCN2C(=O)CSc1nc[nH]n1 63307,N1(C(c2ccc(NC)c(F)c2)=O)CC2CCC1CN2C(=O)CC(C)CN(C)C 63308,c1(CC(=O)NC2CCC(NC(CN(C)CC)=O)C2)ccccc1[N+](=O)[O-] 63309,c1(C(=O)NC(C2CN(C(C3(C#N)CCCO3)=O)C2)C)cc2nccnc2cc1F 63310,c1(CCC(N2C(CNC(C3C(CC)C3)=O)CC2)=O)ccc2c(c1)OCO2 63311,C12(c3ccccc3)CCN(C1)C(=O)C(O)NC(=O)CN2C.c1(NC)ccccc1 63312,c1(CC(N2CC(CNC(C3COCCO3)=O)C(F)(F)C2)=O)nc2ncccn2n1 63313,c1(C(N2C(C)(C(=O)Nc3c(Cl)ccc(C(C)=O)c3)CC2)=O)cccc2c1CCC2 63314,C(=O)(C1=C(Cl)CCOC1)NCC1CN(C(CN(CCOC)C)=O)C(C)C1 63315,c1(NCC2N(CC)CCC2)nc(=NC2CC2CC)[nH]c2c(C)nn(C)c12 63316,c1(C(=O)NCCNC(C(c2ccccc2F)OC)=O)cc2ccc(Cl)c(F)c2o1 63317,c1(C(N(CC2C(C)CCC2)CC2CC2)=O)ccc(N2CCOCC2)cc1Cl 63318,C(C(CC(C)C)C(=O)N1CCC(CF)(NC(c2nc3ncccn3n2)=O)C1)OC 63319,N1(C(C2C(COC)C2)=O)CC2CC1C2NC(c1cnc(C(F)F)nc1)=O 63320,C1(CNC(C=CCCC)=O)CC(OC)CN1C(c1cnc(O)o1)=O 63321,c1(OC)cnc(F)c(C(=O)NCC(C)NC(C2CC2c2nc[nH]n2)=O)c1 63322,N1(CC(C)C)CCC(C(N2CCC(NC(=O)CC3CN(C)CC3O)C2)=O)CC1 63323,Cc1cnc(NCc2cc(C)no2)c(S(=O)(=O)NCC2(CO)CC(C)C2)c1 63324,CCCC(C)(O)C(=O)N1CC(CCNC(=O)C(c2ccccc2F)C)(OC)C1 63325,C#Cc1cc(C(=O)NC2CCC(NC(=O)C(C)O)CC2)cc(N)c1 63326,c1(C(=O)NC2CN(C(C3N(C)CCOC3)=O)CC2(C)C)c(Cl)nc2ccccn12 63327,C1(NC(c2c(CC)c[nH]c2)=O)CCC(CNC(C2(CF)CC2C(F)(F)F)=O)CC1 63328,c1(CN2CCC(C#N)(NC(c3cc(=O)cco3)=O)C2)c[nH]c2nc(Cl)ccc12 63329,C(C(C(=O)NCc1cc(OC)ns1)C(C)(C)C)NC(C(C)OCC)=O 63330,Cc1cccc2[nH]c(=NCCN(C(=O)CC3CC3C)C)oc12 63331,N1(C(CN(C)C(N)=O)=O)CCC(NC(=O)C(C)(C)C(=O)NC)C(CO)CC1 63332,Cc1ccc(SC(C)C)cc1.N1(C(=O)OCC2(Br)CC2)CC=CC1C=O 63333,c1(CC(=O)N(C)CC2N(C(C(C=C)O)=O)CCOC2)cc(F)c(Cl)cc1Cl 63334,N1(C(CC(c2c(C)noc2C)C)=O)CCN(C(=O)C(C)C(C)O)CC1CO 63335,C1(C(=O)NC(c2nc(CC)on2)C)CCCCCCN1C(=O)CC(C)O 63336,C(=O)(C(F)CCC(C)C)N1CC(NC(c2[nH]cc(C)c2)=O)C(O)C1 63337,c1(C(=O)OC)ccc(N2CC(CN(C(C)C(=O)NC3CC3)C)C2)nc1 63338,N1(C(c2c(C)n[nH]c2)=O)CCCC(C(C)NC(=O)Cc2cc(Cl)cs2)C1 63339,C(=O)(C1CCOc2ccccc21)NC(C)CN(C)C(c1c(Br)cnn1C)=O 63340,N1(C(C(CC)SC)=O)CCOCC(CNC(=O)CC2(N(C)C)CC2)C1 63341,CCC(C)C(O)C(C)C(=O)NCc1cc(C)c(C(=O)NC2CCOC2(C)C)o1 63342,N1(C(CC(C(F)F)NC(C2CCCC23CCC3)=O)=O)CCCC2CNC(=O)C12 63343,C1(O)(CCNC(C2(CC#C)CCCC2)=O)CCN(C(c2ccnn2C(C)C)=O)C1 63344,C1(C#N)(C(N(CCC(C)NC(C(C)N2CCC2)=O)C)=O)CCSCC1 63345,N1(C(C2N(C(c3c(C)c[nH]n3)=O)CCCC2)=O)CCOCC2(CC2)C1 63346,Cc1cn2nc(C(=O)NCC(C)(C)CN(C)C(c3ccccc3)=O)cc(C)c2n1 63347,C1(C(=O)NCC(CCOC)NC(c2cnccn2)=O)CCN(C(C)C)CC1 63348,Cn1cnc(NC2CCC(NC(=O)CCc3ccncc3)CC2)cc1=O 63349,C1(CNC(C(CCC)OC)=O)CCN(Cc2nnc(Cn3cccn3)o2)CC1C 63350,N1(C(C)=O)CCCCC1C(N1CCC(CNC(=O)CCCc2csc(=N)[nH]2)C1)=O 63351,C(C1CCOC1)=CC(=O)NCCC(O)CNC(=O)C(F)(F)C1CCCC1 63352,CC(C)(CCCC(=O)NCC1CCCC1O)NC(=O)C(N)=O 63353,C(=O)(C(CC)CC=CC)N1CCCC(CCC(=O)NCC(=C)CC)C1 63354,C(CN=C(NCc1ccnc(-n2ccnc2)c1)N(C)CC1CC=CCC1)OC 63355,C1(CN(C(=O)CCC(=O)N)CCOCC)NC(=O)CC1C(F)(F)F.C(=O)(C1CC1)N 63356,c1(C(c2nnnn2C2CC2)NCc2cn(C)nc2Cl)cc(S(C)(=O)=O)cs1 63357,CC1OC2(C)CC1(C(=O)N(C1CCC(NC(c3c(Br)cnn3C)=O)C1)C)C2 63358,CCC1=C(C(=O)N2CCC(C)C(NC(C3CSC(C)=N3)=O)C2C)CCCO1 63359,C1(C2CCC2)(C(=O)NC(CC)CNC(=O)CC(C)(C)SC)CC1(F)F 63360,C1(C(=O)NCCNC(CC)=O)C2Cc3c(Br)cccc3C12 63361,c1(SCC(=O)NCC(CC)NC(c2cccs2)=O)ccccc1N=NN(C)C 63362,n1(CC(=O)O)c(CCNS(=O)(=O)c2cnn(C3CC3(F)F)c2)nc2ccccc12 63363,C1(CNC(C2CC3C=CC2C3)=O)CN(C(c2cocn2)=O)CCC12CCOCC2 63364,C12(C(=O)NC3CN(C(Cn4c(C)ccn4)=O)CC3C(F)F)CC1COC2(C)C 63365,c1(C(N2C(C3CCN(C(=O)C(F)C4CCOC4)C3)CCC2)=O)cccc(F)c1O 63366,c1(C(=O)NC2CC(NC(c3ccccc3-n3ccnc3)=O)C2)cc(F)ccc1Cl 63367,c1(CCC(=O)N(CCC(C)NC(=O)C#CC2CCC2)CC)cc(F)c(F)c(F)c1 63368,Cc1cccc(C(N2CC3(NC(c4ccsn4)=O)CCC2C3)=O)c1Cl 63369,c1(CC(=O)NCC(C)NC(C2C(C(=O)OC)CC2)=O)coc2c(C)c(Cl)ccc12 63370,c1(C(=O)NCC2(NC(=O)CN3CCCC3=O)CCC2)cccc2cccc(O)c12 63371,N1(C(CN(C(COC)=O)C)=O)CC(NC(=O)C(C)(C)C2CCC2)C(O)C1 63372,N1(C(C(C)NC(CC)(C)C)=O)CCCC1(C(=O)NC(CO)C(C)C)CC 63373,N(C(=NCc1cccnc1-n1cncn1)NCC1CCOC1)CC(C1CC1)OC 63374,C(CC(C)(C)C)(C(=O)N1CC(C2CC2C(N2CCCC23CC3)=O)C1)OC 63375,c1(C(C)(C)N(CC(=O)N(C)CCc2ccccc2)C)nc(=O)n(C)[nH]1 63376,C(=O)(C1=CCC(F)(F)CC1)N1CCC(CNC(C(CC(C)C)OC)=O)C(F)(F)C1 63377,N1(C(CC(CC)C)=O)C(CC(=O)NC2CCCCCC2C)C2CCCC12 63378,C1(CC)CCN(C(=O)CCc2cn(C)cn2)C1C(=O)NCC#CCOC 63379,C(=O)(CCC(C)CN(C)C)NCC1(F)CN(C(C(C)NC(C)=O)=O)C1 63380,C1(C(CNC(CCC)=O)Cc2ccccc2)CCN(C(c2ccoc2Cl)=O)CC1 63381,c1(CC)cccc(C)c1NC(c1cccc(C(F)(F)F)c1)=O.C12CCOC1C2 63382,C=CC(CC)C(=O)N1C(C(=O)NOCC2CCCCC2)CCC1C 63383,N1(C(c2n(C(C)C)ncn2)=O)CC2(CC(NC(=O)CN3CCC3)CO2)C1 63384,CC1=C(C)CC(C(=O)NCC(C(=O)N(CC(C)C#N)C2CC2)C(C)C)CC1 63385,N1(C(C=CC2N(C)CCC2)=O)CCN(C)CC1CNC(C12CSCC1C2)=O 63386,Cc1cc(CNC(C2COC(CNC(c3sccc3C)=O)C2)=O)cc(C)c1 63387,c1(-c2cc(C(=O)NCC(C)N(C(C(COCC)C)=O)C)on2)ccccc1F 63388,Cc1cccc(C2(C(=O)NCCCC(C)NC(=O)C(O)C(F)F)CC2)c1 63389,N1(C(C(CCC2CC2)NC(c2c(OC)ccs2)=O)=O)CC2COC(=O)C2C1 63390,C1(CCNC(C2(OC)CC2)=O)CC(F)(F)CN1C(=O)CCC1CNC(=O)N1 63391,C1(NC(C2(c3cc(C)no3)CC2)=O)CCC(C)N(C(C2CC3(C2)CC(F)C3)=O)C1 63392,c1(-c2cn(CC3C(C)CN3C(=O)CN3CCCC3)nn2)ccc2ccn(C)c2c1 63393,c1(CC)ccc(C)c(C(N2CCC(NC(=O)C(c3cccnc3)O)C2)=O)c1 63394,CC(CCCC(=O)NC(C)(C)CC1CCOC1)NC(c1cc(Cl)no1)=O 63395,c1(C(=O)NCC2CN(C(=O)CC3(CO)CCC3)C2)ccc[n+]([O-])c1 63396,C1(C(=O)NCC(=C)Cl)CC2CC1CC2NC(=O)CC1CNC(=O)O1 63397,Cc1nc(C(=O)NC2CN(C(C3CCC3c3nc[nH]n3)=O)C2)cn(C)c1=O 63398,c1(C(=O)OCC)cc(C(=O)OC)c(OCc2cncc(Br)c2)c(Cl)c1 63399,c1(CC(=O)NCC(CNC(C2CC(C(F)F)C2)=O)OC)ccc2c(c1)OCCO2 63400,c1(CNC(c2ccc(CC)o2)=O)c(C)nn2c1CN(C(C1(C)CC1F)=O)CC2 63401,N1(C(=O)NCCC(=O)Nc2c(C)cccc2)CCc2ncc(Br)cc21 63402,c1(C(=O)NC(CNC(C(C(C)C)N(CC)CC)=O)CC(C)C)ccc(N)c(Cl)n1 63403,C=CCC(F)(F)C(=O)NCC1CC(C)N(C(=O)C#CC2CC2)C1 63404,O=S(=O)(CCO)CCNC(=S)NC1CCCCCCC1 63405,c1(C(N(C)CC2N(C(CCOCC)=O)CC(F)C2)=O)cc2n(n1)CCC2 63406,c1(C(=O)NCCN(C(=O)COC(F)F)C)ccnc2ncccc12 63407,c1(OCC(N2C(CNC(=O)CCCF)CCC(C)C2)=O)cccc(S(C)(=O)=O)c1 63408,c1(C(=O)NC(C(C)NC(c2c(OC)ccc(F)c2)=O)C)cccn2ccnc12 63409,C1(NC(COCCCCC)=O)CCCCC1NC(=O)C(c1cccc(C)c1)C 63410,N1(CC(C)NC(c2cc(C(C)=O)on2)=O)CCN(C(=O)Cn2nnc(C)n2)CC1 63411,C12(C(=O)NCC3N(C(C4CCC(F)(F)C4)=O)CCN(C)C3)C3CC(CC13)C2(F)F 63412,C(=O)(C(C)CC)NCC(CN(C(CN(C(COC)=O)C)=O)CCCF)O 63413,c1(N2C(CNC(C3(C)CCC(=O)N3)=O)CC(F)(F)C2)ccc(S(C)(=O)=O)cn1 63414,C1(C(=O)NCCOCC(=O)N(C)Cc2cncc(O)c2)CC2(CCC2O)C1 63415,CN=c1cc(C(N2CCCC(CO)(NC(c3cc(Br)oc3C)=O)C2)=O)cc[nH]1 63416,c1(C(=O)NC2C(NC(c3cn(CCO)nn3)=O)CC2)cccc2cnsc12 63417,CC(CC(=O)N1CCC(NC(c2cc3n(n2)CCOC3)=O)C1)CC(F)(F)F 63418,c1(NCCc2nc(CC)sc2)ncccc1S(=O)(=O)NC1CN2CCC1CC2 63419,C(C(C)(C)C(=O)NCC[Si](C)(C)C)N(C)C(c1ccc(C2CC2)o1)=O 63420,c1(C(N2CC(NC(C(CC#C)O)=O)CC(F)(F)C2)=O)c(F)cc(OC)c(F)c1F 63421,C1(C(=O)NC2CN(C(c3c(CCC)nsc3N)=O)C2)CC2(CCCC2)CO1 63422,C1(NC(=O)CCc2ccccc2)CN(Cc2cccnc2F)CC(F)(F)C1 63423,C12(C(=O)NC(COCCOC)C)CC(NC(=O)CCc3cccnc3)(C1)C2 63424,N#Cc1ccnc(C(N2C(CNC(C3CCCC(F)(F)C3)=O)CC3CC23)=O)c1F 63425,C(=O)(CCCCC(F)(F)F)NCCCCn1cc(CN(C(C)=O)C)nn1 63426,C=CC(C)(O)C(=O)N1CCC(CCOC)(NC(=O)C(C)(C)C)C1 63427,C12(NC(C3CC4(C3)CC(F)C4)=O)CCN(C(c3cc4sccc4s3)=O)CC1C2 63428,N1(C(Cn2cnc(=N)[nH]2)=O)CCN(C(=O)Cn2cc(C3CC3)nn2)CC1CCO 63429,Cc1cc(C)c2[nH]c(C(=O)NC3CCC3NC(=O)CNS(=O)(=O)C3CC3)cc2c1 63430,c1(OCC)cc(NC(C)CCNC(=O)C(O)C2CC2)ccc1[N+](=O)[O-] 63431,Cc1cc(O)ncc1C(=O)NC1CC(O)CN(C(c2ccnc(C(C)C)n2)=O)C1 63432,N1(C(C(CNC(C2CC3(CC(C)C3)C2)=O)(C)C)=O)CCN(C)C(C)C1C 63433,Cc1csc(C(=O)NC2CCN(C(c3c(C4CC4)noc3C(F)(F)F)=O)C2)c1C 63434,C1(CCN(C23CC(C2)C3)C(C2CCC(C(=O)OC)C2)=O)C2CCCC12 63435,C1(CC(N2CCC(C)(N(C)CC)C2)=O)C2CCCC2N1C(C1CC12CC2)=O 63436,c1(N2CC3C(NC(C(CC)C4CCOCC4)=O)C3C2)cc(S(C)(=O)=O)ncn1 63437,Cc1cc(C(=O)N(C(C)CCNC(=O)C(F)(F)c2cnn(C)c2)C)c(C)cn1 63438,O=C(CCCCCNC(c1cc[nH]c1)=O)NOC1CCCN(CCO)C1 63439,C1(C)(NC(C=C(CCC)C)=O)CCC(NC(c2ccc(C(N)=O)c(Cl)c2)=O)CC1 63440,CC(C)(F)CCC(=O)N1CC(F)CC1CNC(c1c(N)cccc1Cl)=O 63441,NS(=O)(=O)c1ccc(C(=O)NCC(O)COc2ccc(Cl)cc2)nc1 63442,N1(C(Cc2cc(C)sc2)=O)CC(CNC(=O)CCOC2CCC2)C2(CC2)C1 63443,N1(C(C(C)SCCCC)=O)CCC(NC(c2cc(C(C)=O)cs2)=O)C(C)C1 63444,C1(CN(C(C(CC=C)N(C)C)=O)C)CCCN(C(C2CCCCCC2)=O)CC1 63445,c1(C(C(=O)NCC(O)CC2CCC2)NC(c2ccccn2)=O)ccccc1 63446,C(=O)(C(C(C)C)C(C)C)N1CCOCC(C(=O)NCC(COCC)O)C1 63447,C(=O)(C1CCc2nccn21)N1CCCC(O)(CNC(C2N(C)CC3(CC3)C2)=O)C1 63448,CCC(CC(C)C)C(=O)N(C(C)C(=O)N(CC(C)O)CCOC)C1CC1 63449,c1(C(=O)NCC2N(C(C(CCC)(C)C)=O)CCCC2)cc2n(n1)CC(C)NC2=O 63450,c1(C(N2CC(NC(c3c(C)nco3)=O)C(C)CC2)=O)cc(N)cc2ccccc12 63451,c1(C(=O)OC)ccc(C)nc1N1CCCCC(NC(=O)CCCCN(C)C)C1 63452,CC(CC(=O)NCCN(C)C(C1CC1c1ccccc1)=O)n1ccnc1 63453,C12(C(N(CC(C)CNC(C3(CO)CC3)=O)C)=O)CC(c3ccccc3)C1C2 63454,Cc1nc(C#N)ccc1C(N1CCCC(CCNC(C23CC(CO2)C3)=O)C1)=O 63455,C1(C)(CN(CC(=O)Nc2ncc(S(C)(=O)=O)s2)C)CCCCNC1=O 63456,C1(C(=O)NC2CC(CCNC(c3c(CC)ocn3)=O)C2)CCCC(C)(C)O1 63457,CCC(F)(F)CC(=O)NCc1ncoc1CCNC(=O)C(C)(O)CCC 63458,C1(C)(OC)CC2CC1CC2NC(=NCCNC(=O)COC)NCc1ccccc1 63459,c1(OC)cc2nc(O)n(CN3CCCCC(CO)C3)c(=O)c2cc1OC 63460,Cc1ccc(C(=O)NCC(C)NC(=O)C(c2c(C)n[nH]c2C)C)c(N)c1Br 63461,C1(NC(C2(CC)CCCN2C(=O)C(F)C2CCCC2)=O)CCC2CC1CO2 63462,Cc1cc(C(=O)N(CC(O)CNC(=O)CC(C)F)C)nn1-c1ccc(Br)cc1 63463,C1(C)(C(=O)NCC2(NC(CCC(=O)OCC)=O)CCC2)CCCCC1C 63464,c1(C(N2CC3CC(C2)N(C(C2COCCOC2)=O)C3)=O)c(F)ccc2c1OCC2 63465,C(CC)(CC(F)(F)F)NC(C1(CCC=C)CN(C(=O)C(CC)SC)C1)=O 63466,C1(NC(c2c(CC)cno2)=O)CC2CC1CN(C(c1ccsc1C)=O)C2 63467,CC(CC(=O)NC1CCC1NC(=O)CC(=O)N(C)C)P(C)(C)=O 63468,Cc1ccc(OCCCN2CC3C(CNC(=O)C(C)CCC4CC4)C3C2)cc1 63469,C1(CNC(C(C2CCCO2)NC(C2CC=CC2)=O)=O)CC(C2CC2)=NO1 63470,c1(CC(N2C(CNC(C(CC#C)C)=O)CC3(CC3)C2)=O)cccc2c1CCC2 63471,C1(NC(=O)OC(C)(C)C)COC2(CCC2)CN1N1C2CCCC1C2 63472,CCCCCC(O)C(C)C(=O)N1CCCC(CCNC(C2CCN2CC)=O)CC1 63473,C(C1CCC(C)CC1)=CC(=O)OC(C)C(=O)Nc1ccc(C(N)=O)cc1 63474,CC1(C(=O)NC(CNC(C2(n3cc(C#N)cn3)CC2)=O)C2CC2)CCCCO1 63475,C1(CC(=O)NCC(C)CNC(=O)C(F)(F)c2csc(=N)[nH]2)CC(=O)NC1=O 63476,N1(C(CCSCCCC)=O)CCN(C(=O)CN(S(C)(=O)=O)C)CC1C1CC1 63477,C1(C(=O)NCC2(F)CC(NC(CCNC(C)=O)=O)C2)CCCC(O)C1 63478,CC1CN(C(=O)CN2CC(C)(C)C2)CC1NC(c1cccn1Cc1cccs1)=O 63479,C1(C)(C(=O)NC(CNC(C(CCCC)O)=O)CCOC)CCCCCCC1 63480,c1(CN2CC(C(=O)Nc3ncc(F)cc3Br)OCC2)ccc2ncnn2c1 63481,C(=O)(C(F)C(F)(F)F)NC1CC(CNC(c2c(C)cc(C)o2)=O)C1 63482,CC1CCCC1(C(=O)NCc1nncn1C1CC1)NC(=O)CSC(F)F 63483,c1(NC(NS(C)(=O)=O)=S)ccc(OC2CCOC2)c(F)c1.c12cnn(c1)C2 63484,C1(NC(CCc2cn(C)nn2)=O)CN(C(C2(O)CCOC2)=O)CC(C)(C)C1 63485,N1(C(CN(C(COC)=O)C)=O)CCN(C(=O)CCc2cncn2C)CC1C1CC1 63486,C1(CNC(C2C(C)CCCC2)=O)CC(C)CN(C(c2ccnn2CC2CC2)=O)C1 63487,N1(C(C=CC(CC)=CC)=O)CCC(C)(C)C(CNC(C2CCCC3(CC3)C2)=O)C1 63488,N1(C(CCOCCOC)=O)CC(NC(c2cncc(F)c2)=O)CC1C 63489,CN1CCc2cc(C(=O)NC3COCC3NC(=O)C(O)CC(C)(C)C)ccc2C1 63490,C#CCCC(C(=O)NOC)NC(=O)CC1CCCO1 63491,C(CN=C(NCC1CCCCO1)N1CC2CC1CS2(=O)=O)C1(COC)CCC1 63492,N1(C(C(C)OCC)=O)CC(C)(CNC(c2ccnc(C)n2)=O)CC1(C)C 63493,c1(C(=O)NCC(CC)(C)NC(=O)CC(C)n2cccn2)cc2c(ccn2C)s1 63494,C(=O)(CC1=CCOCC1)NCC1N(C(Cn2cnc(=N)[nH]2)=O)CCOC1 63495,C(N=c1[nH]c(Cl)nc2cccc([N+](=O)[O-])c12)C1CCN(C(C(C)C(C)(F)F)=O)C1 63496,Cc1cc(C(N2CC(NC(C3(CO)CCCO3)=O)C(O)C2)=O)cc(Cl)c1 63497,c1(CC)nc(NN(C)C(=O)OC)cc(=NCC(c2cccs2)N(C)C)[nH]1 63498,N1(C(CSCCC)=O)CCC2(CCN(C(C3CCOC(C)C3)=O)C2)C1 63499,Cc1cc(=NCC2(C)CCC(C)(C)CC2)[nH]c(=NCCCC(C)O)[nH]1 63500,N1(C(=O)CN2CCN(CCO)CC2)CCN(C(C2(F)CC=CC2)=O)CC1C1CC1 63501,C1(C)(CCC(=O)NCCN(C(c2csc(-c3ccsc3)n2)=O)CC)CCC(=O)N1 63502,C12(C(=O)NC(CC)CNC(C3(CC)COC3)=O)CCCN(C1)S(=O)(=O)C2 63503,N1(C(CSCC(N)=O)=O)CC(C2(NC(=O)Cn3ccc(O)nc3=O)CC2)C1 63504,O=C1NC(=O)N2CCN(C(=O)NC3CCC(C4CC4)CC3)CC12 63505,N1(C(CC)=O)CCN(C(=O)CC2CCCC(C)C2)CC1.C(=O)OCC 63506,C12(C(=O)N(C(C)C)CC)CC(C(N3CCCC3C(N3CCOCC3)=O)=O)(C1)C2 63507,N1(C(C2(OC)CCC2)=O)CC(NC(=O)Cc2cc(Br)cs2)CC(F)(F)C1 63508,C1(O)(C(=O)NC2CN(C(c3c(CC)noc3)=O)C(C)CC2)CCC(C)(C)CC1 63509,C1(C2(O)CN(C(C3CCc4nn[nH]c4C3)=O)C2)(CNC(CCNC(N)=O)=O)CC1 63510,c1(-c2cn(C(C(=O)N(C(COCC)C)C)C)nn2)[nH]nc(C(=O)OC)c1Br 63511,C#CCCCCCC(=O)N1CC(NC(=O)C(F)CC2CCOC2)C(CO)C1 63512,N1(C(COC(C)C)=O)CCCC(C)(C)C1C(=O)NC(CC1CCCC1)CO 63513,N1(C(CNC(C(C)(C)C2CCCCC2)=O)C(F)F)CCCS1(=O)=O 63514,c1(C(=O)OC)cnn2c1CC(NC(N1CCC(C)(C)CC(C)(C)C1)=O)CC2 63515,C1(N(CCC)C(C2CC2CF)=O)CCN(C(=O)C(F)(F)C2(OC)CCC2)C1 63516,C12(C(=O)NCC3CCN(C(=O)Cc4cnc[nH]4)C34CC4)CC3CC(CC1C3)C2 63517,c1(C(=O)O)nnc(CNC(=O)C(O)CC2CCOCC2)s1 63518,C1(CC=C)(C(=O)O)CCCCN1C(=O)C(F)CC 63519,CC(CC(F)(F)F)C(=O)N(C1CN(C(C2CC(n3cnnc3)C2)=O)CCC1O)C 63520,Cc1csc(C(=O)N(C)CC2CN(C(=O)CC#N)CCO2)c1Br 63521,c1(-n2cc(C(=O)OC)nn2)cccc(NC(c2ccoc2)C)c1 63522,CCC(CC#N)N=c1ccc(Br)c(S(=O)(=O)NCCS(=O)(=O)NC(C)C)[nH]1 63523,C(C(=O)NCC(C)CN(C)C(c1c(NC(C)=O)c[nH]c1C)=O)(C(C)C)OC 63524,N1(C(Cc2ccc(OC)c(Cl)c2)=O)CCN(C(=O)C(C#N)C2CC2)CC(C)(F)C1 63525,N1(C(=O)C=Cc2ccco2)CCC2CCN(c3c(Cl)cncc3[N+](=O)[O-])CC2C1 63526,c1(C(=O)NC(CN(C(C2(CCC=C)CCCC2)=O)C)C)nccc(Cl)c1O 63527,c1(C(=O)OC)cc(Cl)c(F)cc1S(=O)(=O)Nc1cc(Cl)cnc1OCC(F)F 63528,CCCCC(CC)C(=O)NCC1CCCN(C(=O)CC2CCOC(C)(C)C2)C1 63529,N1(CC(=O)NC2CCOCC2NC(C2CC(=C3CCC3)C2)=O)C(=O)CCC1=O 63530,Cc1cc(N2CC(C(N(C(C3CCC3)C)CC3CC3)=O)C2)nc(=N)[nH]1 63531,c1(CCC(=O)NC2C3CN(C(Cc4c(C)nn(C)c4)=O)C2C3)ccc(F)cc1F 63532,C(=O)(CC(C)(C)C(=O)NC1COCC1NC(C1CCC(C)(C)O1)=O)OC 63533,C1(NC(CCC(=C)Cl)=O)CN(C(=O)COc2cc(Cl)ccc2C)CC12CCC2 63534,CC1CC(C2CN(C(=O)C(C)N(C(c3cncn3C3CC3)=O)C3CC3)C2)=NO1 63535,C1(CC)CN(C(=NCCSc2ccccc2)NCCC2CCCOC2)CCO1 63536,N1(C(CCC(C)OC)=O)CCCC2(NC(=O)C(N3C(C)CCC3C)C)CCCC12 63537,c1(C(=O)Nc2ccc(NC(C(CCC)CC)=O)cc2C)cnc2c(c1)NCC(=O)N2 63538,N1(C(CNS(NC)(=O)=O)=O)CCCN(C(C2CC(O)C2)=O)C(C(C)C)C1 63539,C1(N(C(=O)CCOC2CN(C(C3COCCN3C=O)=O)C2)C)CCCCN(C)C1=O 63540,c1(C(N(CCC(C)NC(C2CC2C(c2ccccc2)C)=O)C)=O)ncsc1Br 63541,C12(NC(c3ccn(C4CC4)n3)=O)COCCC1CN(C(c1nc(Cl)sc1Cl)=O)C2 63542,C1(C(=O)NC(C)CNC(=O)C(C)(C)n2cc(Cl)cn2)CCC(=O)NC1 63543,C1(C(=O)NCCCCC(=O)NC)CCC2(CC2)N1C(=O)C(c1cncn1C)O 63544,Cn1c(C(=O)NCC23CC(CN2C(=O)C=CC=C(Cl)Cl)C3)ccc1C(F)(F)F 63545,c1(C(N2CC(c3ccccc3)(NC(c3cc[n+]([O-])cc3)=O)C2)=O)ccc(F)cc1 63546,c1(C(N2C(C(=O)Nc3cc(C)c(F)nc3)CC3CC32)=O)ccc2c(c1)C(=O)CC2 63547,N12CCC(CC1)N(C)C(=O)c1csc(n1)C2.c1(C(C)C)nnnn1CC(=O)OC 63548,N1(Cc2c(C)nc(Cl)cc2)CCC2(CC1)CC2NC(c1ccc(C#N)cn1)=O 63549,N1(C(C=C=C(C)C)=O)CCN(C(=O)CC(C)n2cccc2)C(CC(F)F)C1 63550,C(=O)(C(CC(C)C)NC(c1cnsc1C)=O)NCc1nc(CSC)sc1 63551,CC1CCN(C(C2(CO)CC(F)(F)C2)=O)CCN1C(=O)Cc1cnns1 63552,Cc1nccn1CCCC(=O)NC1CCC(CC(N2CCC(O)C2)=O)C1 63553,C(=O)(CC(C)(O)C(F)(F)F)N1CCCC(CNC(C2(SC)CC2)=O)CC1 63554,c1(C(C(=O)NCC)N2CCC2c2cccnc2Br)cccc(OCCCOC)c1 63555,C1(NC(C=Cc2n(C)ncc2)=O)CN(C(=O)Cc2n[nH]c(=N)s2)CC1S(C)(=O)=O 63556,c1(C(=O)NCCC2(OC)CN(C(CCCC#C)=O)C2)cc(C)nc(N(C)C)n1 63557,CC1(C)CN(C(C2C=CCS2)=O)CCC1C(=O)NC1CN(CC(F)F)C1 63558,C(=O)(CCC(C)(C)C#N)NC1C(C(C)C)N(C(=O)C(O)Cn2cncn2)CC1 63559,c1(C(=O)NC2CC(C(=O)NCC3C(C)OCC3)CC2O)cnn2cccc2c1 63560,C1(C(=O)NC(CCNC(=O)C(F)=CC2CC2)Cc2ccccc2)CC2CCC1O2 63561,C(=O)(C(F)CC(C)(C)N)NCCc1nnc(C(=O)OC)s1 63562,N1(C(C(C)(C)OC)=O)CCN(C(c2ccc(C#N)c(F)c2)=O)CC(C)C1 63563,C(=O)(C(C)(O)C(C)(C)C)NC1CCN(C(c2ccc(SC(C)C)cc2)=O)C1 63564,C12(NC(c3ccc(Cl)cc3F)=O)COCCC1CN(C(c1ccns1)=O)C2 63565,c1(C(N(C2CCN(C(C34CCC3C4)=O)C2)CC)=O)cc(-c2ccccc2)nn1C 63566,c1ccc(CN(C2CCNC2)CC2CCCCC2)cc1 63567,Cc1cncc(CCNC(=O)C(C2CCN(C(c3cnncc3O)=O)CC2)C)n1 63568,N1(C(C)C2CC2)CCN(C(F)(F)F)C(=O)C1.c12cnc(nc1)NC(=O)C(=O)N2 63569,c1(OCC(=O)NC2CC3CC2N(C(C2(C4CCC4)CC2)=O)C3)c(Cl)cccc1Cl 63570,c1(OC)ccc(CNC2CCS(=O)(=O)C2C)cc1S(=O)(=O)N1CCCCC1C 63571,C12(OC)CCC(CN(C)CC3CCO3)(CC1)C2 63572,c1(OC)ccc(CC(N2CCCC(CCCCOC(=O)C(C)=C(C)C)C2)=O)nc1 63573,c1(C(=O)NC2C(CNC(C3CCC(C)CC3)=O)CCC2)cccc2cncn12 63574,N1(C(Cc2c(C)scc2)=O)CCC(NC(=O)C=Cc2ccoc2)C(C)C1 63575,c1(C(N2C(CCNC(C=CC=CC)=O)CSCC2)=O)cc(C)cc([N+](=O)[O-])c1 63576,C(=O)(C(F)C(C)(F)F)NC(C(=O)N1CC(C(=O)NCC)C1)(C)CO 63577,c1(C(=O)NCC2C3CN(C(C4CC(C(=O)OC)C4)=O)CC32)c(Cl)cc(Cl)nc1N 63578,C(=O)(C(C)(C)CCCO)N(C)CC1CCCN1C(c1ccc(C(F)F)cc1)=O 63579,N1(CC(=O)NCC2CC2CC(N2CCC3CCC23)=O)C(=O)CCC1=O 63580,c1(C(N(CCC(C(C)C)NC(C(CC(=O)OC)C)=O)C)=O)cc2cn[nH]c2cn1 63581,O=C(C1CCCc2scnc21)NC1CCN(C(=O)CCOCC(F)(F)F)C12CC2 63582,C1(CC(=O)N(Cc2scc(C(=O)NCCc3c(C)ocn3)c2)CC)CCCNC1=O 63583,C1(N(C(=O)COCP(C)(C)=O)C)CN(C(C2CCN(CC(F)(F)F)C2)=O)CC12CC2 63584,C12(C(N3CCOCC(NC(C4CNC(=O)N4)=O)C3)=O)C3C4C1C1C2C3C41C(N)=O 63585,C1(NC(C2N(CC)CCOC2)=O)CCN(C(=O)Cc2cccs2)CC1(C)C 63586,N1(C(CC(CC)(C)C)=O)CCCCC(NC(c2ccsc2Br)=O)CC1 63587,Cc1c(C(N2CCCN(C(C3CCC(=O)N3)=O)C(C)C2)=O)[nH]c2cc(F)ccc12 63588,C(=O)(CCC(=O)N(C(C)(C)CNC(C1CCCC(F)C1)=O)CC)NCC 63589,C1(CNC(COCCCC#C)=O)CC(C)CN(C(c2occc2CC)=O)C1 63590,C1(NC(c2n(C)ccn2)=O)CN(C(C2CC2CF)=O)C(C)(C)C1 63591,c1(C(N(CCCNC(c2c(C)nc(CC)o2)=O)C2CC2)=O)ccc2c(n1)NCC2 63592,N1(C(c2n(CC)ccc2)=O)CCC(N(C(=O)Cc2c(C)noc2Cl)C)C2(CC2)C1 63593,C1(C2CC2)(NCC(=O)NCC2CC=CC2)CCCC1 63594,C1(NC(C2(C(C)C)COC2)=O)CCC(NC(=O)CCc2cccn2C)C1 63595,c1(SC)c(C(=O)NCC(C)NC(=O)CCCc2nc(C)no2)cccc1Br 63596,c1(C(N2C(CNC(c3c(C)coc3)=O)CC2)=O)c(C)nn(CC(F)(F)F)c1Cl 63597,Cc1nsc(C(=O)NC(C)Cc2csc(-c3cccs3)n2)c1NC(=O)OC(C)(C)C 63598,N1(C(C=CCNC(c2c(CC)n(C)nn2)=O)=O)CC(N(C)OC)C1 63599,C1(NC(c2nc(C)c(C)s2)=O)CCCN(C(=O)CN2CCCC2)CC1 63600,S(=O)(=O)(c1ccc(=NCCC2CCSC2)[nH]c1)NC1CC(C)(C)SCC1 63601,Cc1cc(C(C)C(=O)NCC2CCN(C(c3cnccc3C)=O)C2)c(C)o1 63602,CC1N(C(=O)N(c2ccc(F)cc2F)C2CCCO2)CCC1(C)C 63603,C=C(Cl)CCC(=O)NC(C1CC=CCC1)C(=O)NCC(C)(C)C1CCCC1 63604,N1(C(COCCC(C)C)=O)CCC(F)(C(=O)NCCN2CCCCC2)C1 63605,c1(CNC(=O)NC(CC)CCOC)cc(Br)c(C)s1 63606,N1(C(C2(CC)CCC2)=O)CC(CNC(c2cc(OC)nc(OC)c2)=O)C(C)(C)C1 63607,c1(NC(C)=O)cccc(F)c1NC(=O)CNc1ccc(F)c(F)c1 63608,CC1(C)CCC(CCNC(=O)C(CCF)NC(c2ccc(CO)nc2)=O)O1 63609,CC(C)C(O)C(=O)NC(C)(CNC(c1ccc(C(C)(C)C)s1)=O)C(C)C 63610,Cc1conc1C(=O)NC(C)C(c1ccccc1)NC(C1CSC1)=O 63611,CC(=O)CCCCC(=O)N1CC=CC1(C)C(=O)NCC(C)CC(F)(F)F 63612,C1(C)(C(N2CCC(O)(C(C)CNC(c3ccc(CO)o3)=O)C2)=O)CCC2CC2C1 63613,c1(CC(=O)NCC2(C)CCN(C(C3(CO)COC3)=O)C2)ccc(S(N)(=O)=O)cc1 63614,C1(NC(C2COCCO2)=O)CC(C(N2CCC(CCO)CC2)=O)C12CCC2 63615,C12(CC(=O)NCC(C)(C)CNC(=O)CCC3(C)CCOC3)CCC(CC1)C2(C)C 63616,CC1CCC(O)CN1Cc1nc(Cc2cccc(Cl)c2)no1 63617,N1(C(C(CCSC)O)=O)CC(C(=O)NC2CCCC2N=[N+]=[N-])CC(C)(C)C1 63618,c1(C(N2C(C(=O)Nc3cc(OC)n[nH]3)CC3CC32)=O)cnc(Cl)cc1OC 63619,c1(C(N(C2CCCC(NC(CCC=CC(C)C)=O)C2)C)=O)cc(Cl)cc(F)c1F 63620,c1(CCN(C)C(=O)NCc2nc(C3CCSC3)no2)cccc(F)c1 63621,N1(C(C2(CC)C(Cc3ccc(Cl)cc3)CCCN2)=O)CCC2(CC1)CN(C)C2 63622,C(C(C)(C)CC(=O)N1CCN(C(C2CCCN2C(=O)CNC(N)=O)=O)CC1)OC 63623,N1(c2ccc(-c3ccc(CC)cc3)c(C)n2)CCC(CO)C(C)(C)C1 63624,CCCCCCCCC(C)CC(=O)N1CC(NC(=O)CCNC(=O)OC)C(C)C1 63625,CN1CCN(CC(=O)NCCOCC(F)(F)C(F)F)CCC1=O 63626,C1(=CC(=O)NC2(CNC(C(C=C)C)=O)CC2)CCC(C)CC1 63627,C(CCCCCC(=O)N1CCCC1c1ccccc1C(F)F)n1cc(C(=O)O)nn1 63628,N1(CC)CCCC(C(=O)NCC2CN(C(=O)COCP(C)(C)=O)CC2O)C1 63629,Cc1noc(C(F)F)c1C(=O)NCC(C)(C)CCNC(C1(C(N)=O)CCC1)=O 63630,c1(C(N)=O)ccc(I)cc1OC(c1sccc1N1CCCC1)=O 63631,c1(SC)ccc(Cl)c(C(=O)NC2CN(C(=O)CN(C3CCC3)C)CCC2CO)c1 63632,C1(NC(CC2(CNC(C(CC)C)=O)CC2)=O)CC2CCCCCC12 63633,N1(C(c2c(C)snc2)=O)C(C(=O)NCC2CCOC2(C)C)CC2CCCC12 63634,C1(CC)CN(C(c2coc(CO)c2)=O)CCC1NC(=O)C(=O)NCC(F)F 63635,Cc1cc(CC(=O)N(C(C)CNC(=O)CC2CCC(=O)CC2)C)n(C)n1 63636,N1(C(c2c(SC)snn2)=O)CC2CC(CNC(C3CC4(CC4)CO3)=O)C2C1 63637,C1(CNC(N2C(C(=O)NC)CCC2c2ccccc2)=O)CCC(OC)CC1 63638,Cc1nc(=N)[nH]c(=NCCCCNC(=O)C=Cc2scnc2C)[nH]1 63639,c1(COC)nc(NC2CCCCC2NC(=O)C(C)NC(C)=O)cc(Cl)n1 63640,c12cc(ccc1F)Cc1csc-2n1.c1(C(N2CCOCC2)=O)ccc(O)cc1 63641,N1(C(C(C=C)(C)CC)=O)CC(C2CCCN(C(c3ncn4ccccc34)=O)C2)C1 63642,c1(C(N(CC(C)(C)NC(c2csc(C(N)=O)n2)=O)C)=O)cnc2[nH]cncc1-2 63643,C(=O)(C1=NOC2(CCC2)C1)N1C(CNC(Cn2c(C)ccn2)=O)CC2COCC21 63644,CCCCCC(O)CNC(C1CCN1C(c1coc(C(C)C)n1)=O)=O 63645,c1(C(=O)NC2(COC)CN(C(C3COCC3(C)C)=O)C2)cnc(C(=O)O)nc1 63646,c1(C(N2C(CC(=O)NC(CC)CSC)C(C)(C)CC2)=O)cccc2nccn12 63647,C1(CNC(c2cncs2)=O)CN(C(=O)CN2C(=O)CCC2=O)CCC12CCOC2 63648,CCC1CCNC1=O.n1(CCOC)ccc(C(=O)NCC(F)(F)CO)c1 63649,c1(N2CCCC(CC)C2)nc(N2CC=CC(C(=O)O)C2)nc2c1COCC2 63650,C(=O)(C(F)(F)C(C)O)NCCC1(OC)CN(C(=O)C(C2CCOCC2)C)C1 63651,c1(OCC(N2CCC(C(C)NC(=O)COCC3CCC3)CC2)=O)ccc(F)c(C)c1 63652,c1(OC)cccc2c1OC(C(=O)NC1C3CCC1N(C(C1(CF)CCC1)=O)C3)C2 63653,CCCC(CNC(C1CCCSC1)=O)NC(c1cnc(SC)[nH]1)=O 63654,C(=O)(C(C)C(C)(C)C)N1CC(CC)C1.n1(C(C(=O)N)C)ccnc1-c1ccccc1 63655,Cc1noc(C2(NC(C3(NC(=O)COCCC(C)C)CC3C)=O)CC2)n1 63656,c1(C(C2CC2)NC(c2n(CC)nnn2)CC2CC2)ccc(C(F)(F)F)cc1 63657,C1(NC(C(CC2CCCC2)NC(=O)CCc2ccc[nH]2)=O)C2C3CCC(C3)C12 63658,S(=O)(=O)(c1cccc(N2CC3CC2CS3(=O)=O)n1)N(C)CC1CN(C)CC1(C)C 63659,C1(NC(C2(C)C(C)C2)=O)CC(F)(F)CC1NC(=O)CCc1ccc(F)cc1F 63660,CC(C)C(CN(C)C)C(=O)N1CCCCC1CCNC(=O)CN(S(C)(=O)=O)C 63661,c1(NC(C2N(C(C#C)=O)CC(O)C2)=O)scc(Cl)c1C#N 63662,C1(C(=O)NCC2(OC)CN(C(C(CC=C)(C)C)=O)C2)CC2COCC(C1)C2 63663,c1(OC)ccc(C(=O)NCC2(CNC(C3CCC(C(C)C)CC3)=O)CCC2)cc1 63664,C(=O)(C1=CCC(NC(=O)C(CO)NC(N)=O)C1)NCCCCC1C(C)C1 63665,N1(C(CCC#C)=O)CCC2(CC1)C(NC(=O)CN1CCC(C)C1)CS2(=O)=O 63666,C1(CSC)(CN2CCC(c3nnc(C)n3Cc3ccccc3)CC2)CC(F)(F)C1 63667,C1(CCOC)(NC(=O)CC2CCC(C)(C)C2)CCN(C(=O)Cc2cscn2)C1 63668,C1(C)(NC(C(C)c2cccs2)=O)CCCN(C(=O)C=CC(=O)N(C)C)C1 63669,C(c1cccc(F)c1)=CCC(=O)NCC(C(C)C)NC(C1CC(NC)C1)=O 63670,C1(NC(c2ncn(C(C)C)n2)=O)COCCN(C(=O)CN2CCCCCC2)C1 63671,Cc1cc(=O)c2cc(C(N3CCC(NC(=O)C4=CCOCC4)C3C)=O)ccc2[nH]1 63672,CC1(C#CC(=O)N2CC3CN(C(c4cncc(Cl)c4)=O)CCC23)CCCO1 63673,C1(C)(C(N(CC(C)(C)NC(C(Cn2ccc(C)n2)C)=O)C)=O)CCC(C)(C)CC1 63674,C1(CC)CCN(C(=O)CCCC2CCCO2)C1CNC(C1C2CCCCC12)=O 63675,C1(C(N(C(C)CN(C)C(c2ccc(Br)o2)=O)C)=O)CS(=O)(=O)CC12CC2 63676,C1(CNC(CC2N(C)CCC2)=O)(CO)CCN(C(C23CCCC(CO2)C3)=O)CC1 63677,O=C(N=c1cc(Cl)nc(C(F)(F)F)[nH]1)C1CNCCN1Cc1c(Br)ccc(F)c1F 63678,Cc1cc(N)c(C(=O)NC2CCC2NC(=O)C(C)C(F)F)c(F)c1 63679,C1(CNC(C2OCCC2NC(COC)=O)=O)CC(=O)NC1=O 63680,N1(C(C(c2ccccc2)C)=O)CC2(CCCCN2C(c2cnc(S)n2C)=O)C1 63681,C(CC(C)C(=O)NCC1(NC(c2ccc(CS(C)(=O)=O)o2)=O)CC1)=CC 63682,c1(C(N2CCC(CCNC(CC(=C)Br)=O)C2)=O)nc2ncccn2n1 63683,C1(C(N2C(C(=O)OC)CC2C)=O)CCN(C(=O)COC(C)C)C12CC2 63684,C1(NC(C2CCN(C3CC3)C2=O)=O)CC2CCC1N2C(=O)CNc1ncccn1 63685,C(=O)(CC(C)C(=O)N1CC=C(CNC(=O)C(C)NS(C)(=O)=O)CC1)OC 63686,CC1(C)CN(C(=O)CCN(C(=O)C(C2CCCCC2)O)C2CC2)CCC1O 63687,C(C(CC)(CC)C(N)=O)NC(CN(CC#C)C(c1cccnc1S)=O)=O 63688,C1(NC(C2CCCCC2)=O)CC2CCC1N(C(c1ccn(C3CC3)n1)=O)C2 63689,C(=O)(C(F)C(C)C(F)(F)F)NCC1(C)CCN(C(CCSCCCC)=O)C1 63690,N#Cc1ccc(F)cc1NC(C1CC(F)CN1C(c1c[nH]c2cnccc12)=O)=O 63691,c12cc(ccc1O)C(=O)NC2.c1(CSC)cn(CCCOC(C)C)nn1 63692,CONC(=O)C(C)CN(C)C(C1CC1C(F)(F)F)=O 63693,C1(COCC)CCCCN1C(=O)C(C)C(C)O.c1(N)cc(Cl)c(Br)[nH]1 63694,C1(NC(c2scnc2C(F)F)=O)CN(C(=O)CC2OCCCO2)Cc2nccn2C1 63695,C(=O)(C(C)CNC(=O)C(CC1CCC1)NC(=O)CC1CC1C(F)(F)F)OC 63696,CC1C(C(=O)NCC2CC(F)(F)C2)CCN1C(=O)CCC1CCCC1 63697,C1(NC(C2CC(N3CCN(C)CC3)C2)=O)CCN(C(C2(C)CC2)=O)CC1F 63698,c1(NC(C2CN(C(c3cncnc3)=O)CCO2)=O)nc(C(F)(F)F)c(Cl)s1 63699,C1(NC(c2c(C)cc(CO)o2)=O)CN(C(=O)C=Cc2cccs2)CC2CC12 63700,C1(Sc2ccc(CNC(C(C)C)=O)o2)CCN(C(=O)C(=O)N2CCCC2)CC1 63701,C1(N(C(CS(=O)(=O)NC)=O)C)CCCCN(C(c2nnc(S)n2C)=O)C1 63702,CCC(CCCC(=O)NCC1CCOC1)NC(c1ncncc1C)=O 63703,C(CCCCC(=O)N1CC(NC(C2CC3COCC3C2)=O)C2(CC2)C1)OC 63704,c1(C(=O)OCC)cc(C)sc1NC(C1CCN1C(=O)C(C)Cc1c(C)noc1C)=O 63705,C1(NC(C2CC23CCC3)=O)CCN(C(c2cc3c(s2)CCCC3)=O)C12CCC2 63706,N1(C(c2ncn(C)n2)=O)CCN(C(=O)Cn2ncc(C#N)c2N)C(CC(F)F)C1 63707,N1(C(CCNC(CN(C2(N3CCCC3)CCOC2)C)=O)=O)CC2(CNC(=O)N2C)C1 63708,CC(CC(=O)NC(CNC(=O)C(N)=O)CO)S(=O)(=O)c1ccc(F)cc1 63709,CCCCC(CNC(c1cncc(F)c1)=O)NC(=O)Cn1ccnn1 63710,CC(Cc1ccccc1Br)N=c1[nH]c(N2CCC3CCC(C2)N3C)nc(=N)[nH]1 63711,C12(CNC(=O)OC(C)(C)C)CN(CC3(O)CCC(C(F)(F)F)CC3)CC1CCO2 63712,c1(CC(=O)N(CCN(C(=O)C(C)c2ccsn2)CC)CC)ccc2c(c1)CC2 63713,N#CC1CN(C(C2(C3CCCN3C(c3cnn(C4CC4)c3)=O)CC2)=O)CC12CCC2 63714,C(=O)(CC(C)CCC=C(C)C)NC1CC(N(C(c2c(O)ccc(OC)c2)=O)C)C1 63715,c1(C(=O)NCC(C)N(C)C(c2cc(C(F)(F)F)n[nH]2)=O)ccc(F)cc1C1CC1 63716,C1(C(=O)NCC2N(CC)CC2)CC(O)CCN1C(=O)C(C)CC#N 63717,CC1(C)CN(C(c2cc[nH]n2)=O)CC1NC(=O)CCc1cccc(Cl)n1 63718,CCCS(=O)(=O)CC(=O)NCCC(O)CNC(c1cc(OC)cs1)=O 63719,c1(C(CC(=O)O)NC(=O)Nc2ccccc2)cccc(Oc2ccccc2F)c1 63720,N1(C(C(CCC)NC(N)=O)=O)CCC(NC(c2ccc(C)cc2F)=O)C12CC2 63721,N1(C(CC(C(C)C)C)=O)CCCCC(C2CN(C(C3(C(F)(F)F)CC3)=O)C2)C1 63722,c1(C(N2C(C)CC(CNC(=O)C3=CCCS3)CC2)=O)cc2c(F)ccc(F)c2[nH]1 63723,c1(C(C(=O)NC2CC(CF)C2)N(C2C(OC)COC2)C)cc(C)c(C)cc1C 63724,CC(C(=O)N(C1(CC(=O)N(C)CC2CC2C)CC1)C)C1CCC1 63725,C(C(C)(O)C(=O)N1CCC(F)(C(=O)N(C)CC2(C)CCCO2)C1)OC 63726,c1(CC(=O)NC(C2CCN(C(c3c(C)n[nH]c3)=O)C2)C)ccn2cncc2c1 63727,c1(C(=O)NC(C)C(CO)NC(c2cccc3sncc23)=O)cccc([N+](=O)[O-])c1 63728,N1(CC(=O)N(CC=C)CC)CCCCCCC1CC.N12CCN(CC1)CC2=O 63729,c1(C(C(N2CCC(NC(CN3CC(C)C3)=O)CC2)=O)(C)C)c(F)cccc1Cl 63730,c1(C(=O)NCC2CN(C(C(C)O)=O)C(C)(C)C2)cccc2c1OCCCO2 63731,O=C(CCN(C1(C(=O)N)CC1)C1CC1)N.C1(CCOCCO)(C2CC2)COC1 63732,c12cc(cc(C(=O)O)n1)NC2=O.C1(CCO)(COC)CN(C(=O)Cn2cnnc2)C1 63733,C1(N(CCOCCN(C(CCOCCN(C)C)=O)C)C)CCN(C)CC1 63734,N1(C(c2nc(CC)sc2)=O)CC(C)C(NC(c2ccon2)=O)C(C)C1 63735,C(=O)(C(CCC(N)=O)OC)Nc1cccc(NC(c2ccc(OC)nc2F)=O)c1 63736,CC(C(=O)NC1CCCCC1CNC(c1cncc(O)c1)=O)C(F)(F)F 63737,c1(C(N(CCOCC=C)C)=O)coc(C(C)OC)n1.C12(CC1)C(=O)NC2 63738,CCCCC(O)C(=O)NCC1(O)CCCN(C(=O)CCCNS(C)(=O)=O)C1 63739,N1(C(CC2(OC)CC2)=O)CC(NC(=O)Cn2nc(C)c(C)c2C)CC(F)C1 63740,C(=O)(C(=O)N=c1ncn(Cc2ccc(Cl)cc2)[nH]1)NC(C)CN1CCOCC1 63741,N1(C(C(CC)CC)=O)CC(CNC(c2ccnc(C)c2C)=O)OC2(CCC2)C1 63742,N(C1c2ccccc2OCC1CO)CCC(=O)NC(c1cc(OC)cc(Br)c1)C 63743,CCC(C(=O)N1CC2CCC(CNC(C34CCCC3CCC4)=O)C2C1)C(F)(F)F 63744,C1(NC(C(C)OCC#C)=O)CC2CCC(C1)N2C(c1cccnc1OCCO)=O 63745,n1(CC)cncc1C(=O)N(CCNC(C1(CN(C)C)CCC1)=O)C(C)C 63746,c1(C(N(C2CCCCC2)C(C)C)=O)csc(=NC(CCO)c2ccccn2)[nH]1 63747,N1(C(c2ccc(OC)c(I)c2)=O)CC(NC(c2cnsn2)=O)CC(F)(F)C1 63748,CC(CC(=O)NC1(C)CCN(C(c2cnn(CCF)c2)=O)C1)C(F)F 63749,c1(OC)ncc(C(N2CC3CCC3(CCNC(=O)C(C)(C)CO)C2)=O)cc1C 63750,Cc1ccc2c(=NCCC3CC=CC3)[nH]c(=NC(C)c3ccccc3)[nH]c2c1 63751,C1(OC)CN(C(=O)C(C)=C(C)C)CCC1NC(=O)CN1CCCCC1C 63752,c1(CNC(C=CSC)=O)ccccc1CNC(c1coc(O)n1)=O 63753,Cc1cc(C(N2CC(C(N3CC=CCC3)=O)CC(C)C2)=O)nnc1C 63754,c1(CC)nnc(=NCC(C)N(C)C(C2Cc3nccnc3C2)=O)[nH]c1CC 63755,N1(C(c2c(OC)oc(C)n2)=O)CC(NC(c2ccc(C#N)s2)=O)C2(CC2)C1 63756,N1(C(c2n(C)cnc2)=O)CCCC(C2CN(C(=O)CCCC3CCCO3)C2)C1 63757,CC(C)(O)C(F)(F)C(=O)NC1CC(C(F)C(=O)NCCCSC(F)F)C1 63758,c1(CC(N2CCC(CCNC(C(c3ccc(C)s3)C)=O)C2)=O)c(C)nn(C)c1C 63759,c1(C(C)C)nc(-c2cccc(N)n2)nn1C(C1(C)CC1)C 63760,N1(C(CCC2N(C(C3N(C(C)(C)C)CC3)=O)CCC2)=O)CCC2(COC(=O)N2)C1 63761,C1(NC(CC2N(C(C)=O)CCC2)=O)CCC(CNC(c2cnnn2C)=O)CC1 63762,C1(CC)(NC(c2ccc(F)c(C(C)(C)F)c2)=O)CCCN(C(=O)C(C)(C)OC)C1 63763,c1(C(=O)NC2CCN(C(c3ccnc(OC)n3)=O)C2)cccn2ccnc12 63764,c1(NC(C2CCN(Cc3ccncc3O)CC2O)=O)cnc(Cl)cc1[N+](=O)[O-] 63765,C(CNC(c1n[nH]c2c1COC2)=O)(CC(F)(F)F)NC(CC(C)N(C)C)=O 63766,c1(C(=O)NCC2N(C(C(C)SC)=O)CC2)ccc(S(=O)(=O)N2CCCCC2)cc1 63767,c1(CN(C(=O)C(c2ccccc2)O)Cc2ccccc2)csc(C(F)F)n1 63768,Cc1cc(C)n(NC(=O)C2CNCc3nc(N(C)C)ncc32)c1C 63769,CCC(C(=O)NCC(C)(C)CNC(=O)Cc1ccsc1)NC(C)=O 63770,C(=O)(CCCCCC#N)N1CC(CNC(C(C)(C)SC)=O)OCCC1 63771,C1(F)(C(=O)NC2CC(C)N(C(C3CN(C)C(=O)N3)=O)CC2)CCC(F)(F)CC1 63772,C(=O)(CC1CCOc2ccccc21)N1CC(C)C(NC(=O)C=CBr)C1 63773,Cc1cccc(CC(N2CCC(C)(CCNC(=O)CC(C)(C)O)C2)=O)c1F 63774,N1(C(C(C)OCC=C)=O)CCCC2CN(C(c3ccc(CC(C)(C)O)s3)=O)CC12 63775,Cc1ccc(C(F)C(N2CCCC2C(C)(C)CNC(=O)C2CC2)=O)cc1 63776,c1(C(N2CCC(c3nc(-c4ncc(Br)cn4)no3)C2)=O)cccc2oc(O)nc12 63777,c1(CNC(c2c(C)nsc2)=O)ccc(C(=O)NC(c2ccccc2)C(N)=O)cn1 63778,N1(C(c2c(C(C)C)scn2)=O)CC(CNC(C2CCCN(C)C2)=O)C2(CCC2)C1 63779,S(=O)(=O)(CCC(=O)NC1CC(C)N(C(c2ccnnc2)=O)C1)NCCNC(C)=O 63780,c1(C2(C(=O)NC(CC)CN(C(=O)CC3CC(C)=NO3)CC)CCC2)cccc(Cl)c1 63781,C1(C(N(C2(CCO)CC2)C)=O)OCCC1NC(c1cnn(C(F)F)c1)=O 63782,C1(CC(=O)NCC(O)CNC(c2c(Cl)n[nH]c2C2CC2)=O)CCCCC(=O)N1 63783,C1(C(N)=O)CN(C(=O)C(CCF)NC(=O)CC2CC(=O)NC2=O)CC12CC2 63784,C(CC(C)C(=O)NC1CCC(NC(c2cscc2Cl)=O)C1)=CCC 63785,CCCCCC(F)C(=O)N1CC(CNC(=O)CCN2CCOC2=O)CC(C)C1 63786,C1(NC(=O)C=Cc2nccs2)CCOC(C(=O)NCCC2CC=CC2)C1 63787,c1(CNC(C(c2ccc(Cl)c(Cl)c2)N)=O)cc(C(F)(F)F)ccc1Cl 63788,C1(NC(C(=O)NCc2c(C)cc(C#N)cc2)=O)CCC2(CC1)OCCO2 63789,C12(NC(c3c(C)con3)=O)CCC(CC1)N(C(=O)CN1C(=O)CN(C)C1=O)C2 63790,Cc1nn(C)cc1C(=O)NC1CCCC1C(=O)NCC(O)C1(Cl)CC1 63791,C1(C(N(C2CCCN(C(=O)Cc3cscn3)C2)C)=O)CCCCCCC1 63792,C1(OC)CCC(C(N2CCCC(NC(c3cnn(C)c3Cl)=O)C2)=O)CC1 63793,CC1CCC(O)(C(N2CC3C(C(=O)NC(CC4CC4)CO)C3C2)=O)CC1 63794,C(C)(C(=O)N(C)Cc1cccnc1)(C1CCOCC1)OC 63795,Cc1cccn2cc(C(=O)NC(C)CCN(C(=O)CN(C3CCC3)C)C)nc12 63796,Cc1nc(NC(C)(C)CN(C(=O)CSC(F)F)C)cc(Cl)n1 63797,c1(C(=O)NC(CNC(COCC=C)=O)C(C)C(C)C)cc(Cl)cc(Cl)c1Cl 63798,Cc1cnc(C)c(NC(C2(F)CC=CCC2)=O)c1 63799,C1(C(=O)NC(CC)C)CC2CCC1N2C(=O)C=C=C(C)C 63800,N1(C(CCC#C)=O)CC2CCCC(CNC(C3CCC(OC)CC3)=O)C2C1 63801,CCCCCCC(C)C(=O)NCC(C(C)C)NC(c1c(C)cnnc1O)=O 63802,c1(C(N2C(CCNC(C=CC)=O)CCC2)=O)ccc(Br)c(COC)c1 63803,Cc1scc(C(=O)NC2CN(C(c3cc(O)ncn3)=O)CC2C(N)=O)c1C 63804,CC(C)C(C(=O)NC1(C)CC2(CCC2)C1)C(C)NC(c1cc(C#N)ccc1N)=O 63805,N1(C(C(COC(C)C)NC(C)=O)=O)CC(N(C(=O)CCn2cnnn2)C)C(O)C1 63806,C(=O)(C1=Cc2cc(Cl)ccc2OC1)N(CCN(C(C1C(C)C1C)=O)CC)CC 63807,c1(OC)cccc(CC(=O)NCC(C)NC(c2ccnc(OCCSC)c2)=O)c1 63808,N1(C(CSCC(N)=O)=O)CC2CCCCC2(CNC(=O)C=C2CCCCC2)C1 63809,c1(OC)cc(Cl)ccc1C(N1CCC(O)C(F)C1)C(=O)NCc1cccc(Cl)c1 63810,Cc1nccnc1C(N1CCC(CC(=O)N(C(C)C)CC2CCC2)C1)=O 63811,C1(CC(NOCC#C)=O)CC(NC(C2CCN2CC)=O)C1(C)C 63812,C1(C(C(=O)NCCCOC=C)NC(=O)CCn2cccc2)CC=CCC1 63813,c1(CC(=O)NCC(CNC(COCC=C)=O)(C)C)cc(Cl)cc(Cl)c1 63814,C1(C(=O)NC2C(CCC)CN(C(c3cc[nH]c3C)=O)C2)CSc2ccccc2O1 63815,N1(C(=O)Nc2c(C)cc(N3CCOCC3)cc2)CCN2CCOCC2C1 63816,Cc1ccsc1CC(=O)NCCC1CC(NC(c2nocc2C(C)C)=O)C1 63817,C1(C(NOCC(CC)C)=O)CCC(O)CN1C(C1CCCC(C#N)C1)=O 63818,N1(C(c2n(CCC)ncc2)=O)CC(C(=O)N(CC(=O)NC)CCC)CC12CCC2 63819,C1(C(=O)NCC(CC=C)NC(C2(n3cccn3)CC2)=O)(CC)CC(C)(C)C1 63820,c1(C(N2CCC3(CN(C(c4cc(C)ns4)=O)C3)C2)=O)cn2cccc(F)c2n1 63821,O=C(C1=CC2(CCOC2)C1)NC1CN(C(c2cc(C(F)F)no2)=O)CC12CCC2 63822,C(=O)(CC1CCOc2ccccc21)N1CC(NC(CSSC)=O)C(C)C1 63823,C1(CC(=O)OC)(NC(c2ccc(-n3ccc(O)n3)cc2)=O)CS(=O)(=O)C1 63824,C(c1ccc(F)c(Cl)c1)=CC(N1CC(C)C(NC(=O)CN2CSCC2=O)C1)=O 63825,C(CCCC(=O)NC1CCC1NC(=O)CSC(C)(C)C)N(C(C)C)C 63826,CC1CC(C(=O)NC(C2CCN(C(=O)CN3CCCNC3=O)C2)C)CCS1 63827,CN1CC(NC(c2ccc(-c3cscn3)nc2)=O)Cc2ccccc21 63828,CCC(Cc1cccc(C)c1)C(=O)NC(C)CN(C(=O)C(=Cc1cccs1)C)C 63829,c1(C(=O)OC)cc(=NCCC2CCCCN2C(C2CCCC(=O)N2C)=O)[nH]c(Cl)n1 63830,c1(OCC)cc(CNc2ccc(C(=O)NC(C)(C)C)o2)ccc1O 63831,c1(C(C)C)ccc(CNC(c2nnnn2C)C2CC2)cc1.C1(C)CC1 63832,S(=O)(=O)(C1CCNC(C)(C)C1)Nc1cc(C)cc(C(F)F)c1 63833,N1(C(C=C(CC)CC)=O)CCC2CCCC12C(N1CCCC1CSC)=O 63834,C1(C(C)C)CN(C(c2c(Cl)cccc2Cl)=O)CCN1Cc1cccc(I)c1O 63835,C(=O)(CCCCCN(C)C(C1CC(C)(F)C1)=O)NCCCOCCCC 63836,c1(C(=O)O)ncccc1S(C)(=O)=NC(=O)C1(Cl)CC12CCC2 63837,C1(C)(C(=O)NC2C(OC)COC2)CC12CCN(C(=O)C(N)C(C)C)CC2 63838,Cc1c(C(N2CCC(N(C)C(c3cc(Cl)ccc3O)=O)C2)=O)ccc2c1CCC2 63839,c1(C(N2CC(NC(CCCNC)=O)C(O)C2)=O)ccc(N(C)C)nc1Cl 63840,CC1CN(C(=O)CC2CCSC2)CC(C)N(C(c2nn(C)c3c2CCC3)=O)C1 63841,c1(CC)cccc(C(=O)N(CCC(C)NC(C2(CF)CCOCC2)=O)C)c1N 63842,C1(C(N2CCC2Cc2ccn(C)n2)=O)CCN(C(C2N(CCC)CC2)=O)CC1 63843,N1(C(C2C(C(=O)OC)C2)=O)CC(CNc2cc(C#N)nc(C)n2)C2(CCC2)C1 63844,C=CCCC(CC(C)C)C(=O)N(CCNC(=O)C(C(C)C)NC(=O)OC)CC 63845,C1(NC(C(=O)N(CCCC)CC)F)CCN(C(C2(C(C)C)CC2)=O)CC1 63846,C1(CC=C)(C(N2CCC2C(C)C)=O)CCCN1C(=O)CCCn1cccc1 63847,Cc1n[nH]cc1CC(=O)N(C1(NC(C2CC2C(F)(F)F)=O)CCC1)C1CC1 63848,C1(CC)CN(C(c2cc(C3CC3)cnc2Cl)=O)CCN1C(=O)C(C)OC 63849,C(=O)(C1=C(Cl)CCC1)N(CCOCCCN(C)C(C1COCC(C)(C)O1)=O)C 63850,c1(NC(CC)CSC)cc(=NCC(Cc2ccccc2F)CO)[nH]c(C)n1 63851,CC1CC(C)CN(CCCN(C(=O)CCc2nc[nH]n2)C(C)C)C1 63852,C1(CNC(c2ccc(C)o2)=O)CCCC2(CCN(C(=O)CC(C)C(C)C)CC2)O1 63853,n1(CC(=O)NC2C(C)CN(C(=O)CN3CC=CC3)C2)ccc([N+](=O)[O-])n1 63854,Cc1ccc(C(=O)N(CCC(C)NC(c2cnn(CCO)c2)=O)C)cc1F 63855,CN1CCC2(CCN2C(c2ccc(-c3cc[nH]n3)o2)C(=O)NC2CCOC2)C1 63856,N1(Cc2cc(Br)cc(OC)c2O)Cc2ccccc2CC1CCO 63857,Cc1cnc(C(=O)N(C2CCN(C(c3cc(Cl)ccc3Cl)=O)CC2C)C)c(C)c1 63858,CN1CCC(NC(=O)CC(C)(C)C)C12CCCN(C(C1(O)CCCCCC1)=O)C2 63859,C1(NC(CCNC(=O)CO)=O)CCOC12CCN(C(=O)CC1CCC(=O)C1)CC2 63860,c1(N2CC3(C(NC(C4C(C)(C)CCC4)=O)CCS3)C2)nc2cc(F)c(F)cc2s1 63861,N1(C(C2CCC(=C)CC2)=O)CC2(CCC2NC(c2cc(C(C)C)cnc2O)=O)C1 63862,c1(OC)ccc(F)cc1C(=O)NC1CCCN(C(=O)CC2OCCO2)C1C 63863,c1(C(N2CC(COC)(CNC(=O)CCCF)C2)=O)cnn2ccncc12 63864,CCC(C)(C)C(=O)NCC(C)(CO)NC(c1cnc(-n2cccn2)cn1)=O 63865,N1(C(CC2(OC)CCCC2)=O)CC(CN(C)C(c2cscc2SC)=O)C2(CC2)C1 63866,c1(OC)ccc2c(CC(N3CCC(CNC(=O)C(C)CN(C)C)C3)=O)coc2c1 63867,N1(C(C(=O)NCC2CCCCC2)=O)CC2CC1(CNC(c1cncnc1)=O)C2 63868,c1(NCC2C(NC(c3cnn(C)c3C3CC3)=O)CCC2)ncc(Br)cc1[N+](=O)[O-] 63869,c1(CC(=O)NC2CN(C(C3CCCC4CC34)=O)C2)ccc2c(c1)OCCO2 63870,C1(CNC(c2cc(C3C(C)C3)on2)=O)CCN(C(=O)Cc2ccn(C)c2)C12CC2 63871,C=Cc1ccc(C(N2CCC(NC(=O)Cc3ccccc3Br)CC2)=O)cc1 63872,c1(NC(C2(NC)CN(C(C3(C(=O)OC)CC3C)=O)C2)=O)ccc(Cl)cc1 63873,N1(C(c2c(CNC(c3cc(C)ncn3)=O)ocn2)=O)CC2CCC(O)C2C1 63874,C1(C)(CNC(CCOCC#C)=O)CCCN1C(=O)Cc1cn(C)nn1 63875,c1(C(=O)NCC2N(C(c3c(OC)c[nH]n3)=O)CC2)[nH]c(-c2cccc(C)c2)nc1C 63876,C(c1ccc(F)c(F)c1)=C(C(N1C2CN(C(C3(COC)CC3)=O)C(C2)C1)=O)C 63877,N1(c2n(CCCOC)c(-c3cc4c(s3)CCC4)nn2)CC2CCCC2C1C(C)C 63878,N1(C(C(C)NS(CC)(=O)=O)=O)CCC2(CC1)CCN(C(=O)C(C)C1CC1)CC2 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63896,n1(CC(=O)NCCCC2N(C(C3CC(=O)C3)=O)CCC2)cnc([N+](=O)[O-])c1 63897,C=C1CCC(C(=O)NCCN(CCCN(C)C)C(=O)CC2(OC)CCCC2)CC1 63898,c1(C(C(=O)NCC)N(C(c2ccccn2)C(=O)NC)C)cnc(C(=O)OC)[nH]1 63899,CCCCC(C(=O)N(C(C)CC(C)C)C)NC(C1CC(C)C1)=O 63900,c1(C(N2CCC(N(C(C(CC)O)=O)C)C3(C2)CC3)=O)cc2cccnc2cc1F 63901,N1(C(c2c(OC)cc(F)cc2)=O)CCCC12CN(Cc1cc(Cl)cnc1C)C2 63902,c1(C(=O)NC2CC(C)N(C(=O)CCCCO)CC2)ccc2c(c1)CCC=C2 63903,Cc1ncc(C(N2CC3CC(NC(c4nccc(Cl)c4F)=O)C3C2)=O)c(O)n1 63904,c1(C(=O)NCCCN(C(=O)C(O)c2ccco2)C)c[nH]nc1S(N)(=O)=O 63905,N1(C(c2cnc(C(C)C)o2)=O)CCC2CN(C(=O)C(O)CCN(C)C)C2C1 63906,c1(CN2C(C(=O)NCc3cccc(C)c3)CC(F)C2)cc(C)ccc1O 63907,CC1(C)CN(C(=O)CC2(C#N)CC2)C(CNC(=O)Cc2c(Cl)cccc2Cl)CO1 63908,C1(CNC(c2ccc(SC)s2)=O)CC(NC(c2nncn2CC2CC2)=O)C1(C)C 63909,N1(CCNC(C2CCN(C(C)C(=O)N(C3CCCC3)C)C2)=O)CCS(=O)(=O)CC1 63910,c1(C(N2C(CNC(c3nc(C)sc3C)=O)C3CCC2C3)=O)ccc2snnc2c1 63911,C1(C(=O)NC(C)(C)CCCNC(=O)C=Cc2ccccc2)CCC2(CCOC2)O1 63912,C12(C(=O)NC3C(CCC)C3)CC(CO1)N(C(c1cc(Cl)cs1)=O)C2 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64035,C1(NC(CC(CCC)O)=O)CN(C(c2cccc(Br)c2F)=O)CC2(CC2)C1 64036,N1(C(Cc2nc(C)c(C)[nH]2)=O)CCC(C)C(CNC(c2c(C)nsc2N)=O)C1 64037,c1(OC)c(C)cc(NC(N2Cc3[nH]nc(C(=O)OC)c3C2)=O)cc1C 64038,Cc1nn(C)cc1C(C)C(=O)NC(c1cn(Cc2ccc(Br)s2)nn1)C 64039,N1(C(C(C)SCCOC)=O)CC2CC(C1)C2NC(=O)C(C)(C)NS(C)(=O)=O 64040,C(=O)(CCC(=O)C(C)(C)C)N1CCC(C)CC1C(=O)NC1CN(C2CCC2)C1 64041,C#CCC(O)C(=O)NCC(F)CNC(c1cccc(C)n1)=O 64042,CC(N=c1nc(-c2ccccc2)nc(N2CCOCC(C)(F)C2)[nH]1)c1cc[nH]n1 64043,CCC(CN(C)C)N=c1[nH]c(N(C)Cc2cc(Cl)cs2)nc(=N)[nH]1 64044,N1(C(CCC(CC)NC(c2cnc(C(C)C)o2)=O)=O)CC(C)(C)C2CCCC12 64045,C1(CC(=O)N(CCOCC=C)C)CCN(C(C2CCCCC2O)=O)CC1 64046,C(=O)(C(C)(C)CN(C)C(C1CCOC(CC)C1)=O)NC(CCC)c1ccco1 64047,N1(C(C2N(CC)CC2)=O)CC2CC(C)N(C(=O)CN3CCCNC3=O)C2C1 64048,C(=O)(CC(=O)N1CCCC1C(C)(C)NC(C1CC1C1CC1)=O)NC 64049,C1(C(N(CC(C)NC(C23CCCC2(C(N)=O)C3)=O)CC)=O)CCC2(CCC2)CC1 64050,N1(C(c2c(C(N)=O)csc2)=O)CC2C(CNC(c3cc(Cl)c[nH]3)=O)C2C1 64051,CCC(CC(F)F)C(=O)NC(C)CN(c1cc(OC)nc(C2CCOCC2)n1)C 64052,N1(C(c2cc(C)ns2)=O)CCCC(F)(C(=O)NCc2cc(C)sc2C)C1 64053,Cn1nnc(CNC(=O)C(C2CCC2)NC(=O)C(F)n2ccnc2)n1 64054,c1(SC)cccc(F)c1C(=O)NC1CC(CO)N(C(=O)C(C)CF)C1 64055,C12(CC(=O)N(C3CCN(C(C4(C)CCNC4=O)=O)C3)CCC)CCC(CC1)OC2 64056,C(=O)(C(C)(O)CC(C)C)N1CCC(O)(c2cn(CCCOC)nn2)CC1 64057,C12(OC)CCCCC(C(=O)N(C3CCCCN(C(=O)CNS(N)(=O)=O)C3)C)(C1)C2 64058,C(=O)(CCCCCCN=[N+]=[N-])NCC(CC)NC(c1ccc(Cl)c(Cl)c1O)=O 64059,C12(NC(c3c(CC)c[nH]n3)=O)CC3CCC(C1C2)N3C(=O)CC1CCCO1 64060,N1(C(C2C(CCOC)C2)=O)CC(C)(C)CC1CC(=O)NC1CSC1 64061,N1(C(C=C(C)C)=O)C(C(=O)NC(c2ccc(Cl)cc2)C)CC2CCCCC12 64062,C=CC1OCCC1C(=O)NC1CC(CNC(=O)CCC#CC)C1 64063,C1(=CC(=O)Nc2c(C(N(C3CCCO3)CC)=O)n[nH]c2)CCC(C)CC1 64064,N1(C(c2cc(C)[nH]n2)=O)CCC2CN(Cc3ccnn3C)CC12 64065,c1(CCC(=O)NCCN(C(=O)C(C)CC2CCCCC2)CC)cc(C)[nH]n1 64066,CC(C)(C)C(CNC(C12CC(C1)C2)=O)NC(C1CC12CC(O)C2)=O 64067,c1(C(N2CCC([N+](=O)[O-])CC2)=O)c(O)ncc2c1CCC2 64068,N1(C(C(CC#C)NC(=O)CN2CCC(=O)CC2)=O)CC2CCC=CC12 64069,N1(CCC(=O)NC2C3CN(C(CC(C)(C)C)=O)C2C3)CCP(C)(=O)CC1 64070,N1(C(c2cc(SC)oc2)=O)C(C(=O)NCC(C)(C)C(N)=O)CCC1C(C)C 64071,c1(C(N2CC(C(C)NC(C3CCCC3C)=O)OCC2)=O)csc([N+](=O)[O-])c1 64072,N1(C(CC2CN(C)C2)=O)CC2CCC1C(NC(c1c[nH]cc(Cl)c1=O)=O)C2 64073,CCCCCC(F)C(=O)N1CC(CC(C)NC(C2(C)CC2(C)C)=O)C1 64074,C=CC(CCC)CC(=O)N1CC(CF)(NC(C2CC2CCOC)=O)C1 64075,N1(C(CCN(C(=O)C(C)SC)CC#C)=O)CCC(CN(CC)CC)C1 64076,N1(C(C2CCCC(C)C2)=O)CCCC2(CCCN2C(=O)CC2CCS(=O)(=O)C2)C1 64077,C1(OC)CCCC(C(N2CC(O)(CNC(=O)COc3ccsc3Cl)C2)=O)C1 64078,C1(NCC(=O)Nc2sccc2S(=O)(=O)N2CCSCC2)CC[Si]2(CCCC2)CC1 64079,Cc1cc(CC(N2CC(NC(=O)CP(C)(C)=O)CCC2C)=O)cc(Br)c1 64080,C(N1CC(C)C1c1ccccc1)c1cn(C(C)(C)COC)nn1.O[Si](C)(C)C(C)C 64081,c1(-n2ncc(CNC3C=CC(C(N(CC(O)CO)C(C)C)=O)C3)c2)ccc(Cl)cc1 64082,Cc1nnc(NC2CC(NC(c3snc(Cl)c3Cl)=O)C23CCC3)c(C#N)c1C 64083,c1(OC)ccc(C(CNC(=O)C(N2CCC(C3OCC3(F)F)CC2)=O)SC)cc1 64084,N1(C(C2CCC(CCCCC)O2)=O)CC=C(CNC(=O)CC2CC2(C)C)CC1 64085,C1(C(N(CCC)CCC)=O)CC2CN(C(C3(C)CCC(=O)CC3)=O)CC2C1 64086,c1(C(C)=O)ccc(F)c(C(=O)NC2CCN(C(c3cnc(O)s3)=O)C2)c1 64087,C1(NC(c2c(C)nc(C)[nH]2)=O)CCN(C(=O)CC2(O)CCCCCC2)CC1(C)C 64088,C1(c2nccc(C)c2)CCN(N2CC(CS(C)=O)C2)C1 64089,CCN=c1[nH]cc(C(=O)NCCOc2ccc(CC#N)cc2)s1 64090,C1(C)(CC)CC(C(=O)OC2(c3ccc(Cl)cc3)CC(OC(C)(C)C)C2)CCO1 64091,C(=O)(C#CC1CCCO1)NCC1(COC)CCN(C(C(CC)SC)=O)CC1 64092,CCCCCC(=O)N1CC(CC)NC(=O)C1.C1(=O)CN1C.C(=O)(CSC)NCC 64093,C=CCC(CC(F)F)NC(C1CC=CC(NC(=O)C(C)CCCC)C1)=O 64094,C(N=c1cc[nH]cc1C#N)C1C(C)CN(C(=O)Cn2cc(C3CC3)nn2)C1 64095,N1(C(C(c2c(C)ccc(F)c2)(F)F)=O)CC2CCCC(CNC(=O)C(C)O)(C2)C1 64096,C1(C(=O)NC(CC)C)CCOC12CCN(C(C)=O)CC2 64097,c1(CC(=O)NC2(CC)CN(C(=O)CC3COCCO3)C2)cc(F)ccc1O 64098,N1(C(CC2CC(OC)C2)=O)CC2CC(NC(=O)C(c3cccc(F)c3)O)CC1C2 64099,c1(C(N2CC(OC)C(NC(c3[nH]nnc3C)=O)C2)=O)cnc(C)c(C)c1 64100,CCCCC(F)C(=O)NCC1CCC1C(N1CC2CC1CN2C(C)C)=O 64101,C1(O)(C(=O)NCC(C(=O)NCCN(C(C)C)C)N(C)C)CCSCC1 64102,c1(C(=O)NC(CNC(CCN(C)CC)=O)CCOC)cc2sccc2s1 64103,c1(CC(=O)NC2CCN(Cc3cnc(F)c(F)c3)C2)cccc(Cl)c1F 64104,C(=O)(C1COc2ccccc21)NCC1N(C(C(C(CC)C)O)=O)CC(C)(C)C1 64105,c1(C(=O)NC2CC3CN(C(c4nncc(OC)c4)=O)C2C3)ccc2nccn2c1 64106,c1(C(=O)NC(CC)CN(C(=O)Cc2cnoc2)C)ncc(C)cn1 64107,c1(SC)ncc(C(N2CC(O)(CNC(C3C(F)(F)C34CC4)=O)C2)=O)c(O)n1 64108,C(CO)(C(=O)N1CCC(C(N2CC(c3ccon3)C2)=O)C1)OC 64109,n1(CC(=O)N(C2CCN(C(c3cc(C(N)=O)c[nH]3)=O)C2)C)cc(Br)ccc1=O 64110,N1(C(c2nn(C)c(F)c2)=O)CCN(C(=O)CC2CCOC2)CC1CO 64111,N1(C(C(C)(N(C(CC2CC(SC)C2)=O)C)C2CC2)=O)CC(C)(C#N)C1 64112,S(=O)(=O)(c1ccc(C2CNCCOCO2)s1)N(CCNC(c1cc(N)cnc1C)=O)CC 64113,CC1(C)CN(C(=O)C(C)(O)C(F)(F)F)CCC1C(=O)NC1CCCCCC1 64114,N1(C(C2(CCOCC)CCC2)=O)CCC(CNC(=O)C(C)O)(COC)CC1 64115,N1(C(C)=O)CCCCC1C(=O)NCC(C)NC(c1cccnc1Br)=O 64116,c1(C(N(C)CCN2CCN(C(=O)CC3CC(F)C3)CC2)=O)cc(N)cc(O)c1 64117,C1(C(N2CC(C)N(C(=O)CCCN3CCCC3)CC2)=O)CC2(C1)C(F)(F)C21CC1 64118,CC(C)CC(O)C(C)C(=O)NC(C(=O)N1CC(n2cnnn2)C1)C1CC1 64119,c1(C(N2C(CCNC(c3c(C)ncs3)=O)C(C)CCC2)=O)ccc2ncnn2c1 64120,C1(CCNC(c2nnnn2-c2ccccc2)CCSC)CCCN(C)C1 64121,CC1CC=CCC1NC(c1cc(CNC(c2coc(C3CC3)n2)=O)[nH]n1)=O 64122,N1(C(c2ccn(CC)c2C)=O)CC(C)(C)CC1C(=O)NC(CCO)C1CCCC1 64123,Cc1cccc(C=CC(=O)NCC(C)(C)OCC(=O)NCCC(O)C(F)(F)F)c1 64124,Cn1nc(C(N2CCCC2(C)CNC(C2CCC2CC2CC2)=O)=O)cc1CO 64125,c1(C(N2C3CCC(NC(c4cc(OC)n(C)n4)=O)(C3)C2)=O)cccc2c1NCC2 64126,n1(C(C)C)ncc2c(NC(CCO)c3ccco3)[nH]c(=NCCCC#N)nc12 64127,N1(C(CCCC(C)C)=O)Cc2nccn2CC(NC(C2(CN(C)C)CC2)=O)C1 64128,c1(C(N2CC3(C(C(=O)Nc4n(C)nc(C)c4Cl)C3)C2)=O)cc(C#N)ccc1F 64129,c1(C(N2CCC(C)(CCNC(C3CCCCS3)=O)C2)=O)cc([N+](=O)[O-])n[nH]1 64130,C1(C(=O)NCCCCN(C(CCC2CC(C)C2)=O)C)CCC2(CC1)CC(O)C2 64131,c1(C(N2CCC(C(C(=O)NCCC(=O)NCC)F)C2)=O)cc(C)ccc1O 64132,N1(C(CC2C(C)C2)=O)CC(O)(CCNC(c2csc(N3CCCCC3)n2)=O)C1 64133,Cc1cc(=NC(=O)C(=O)C(C)(C)C)[nH]n1-c1ccccc1 64134,C1(C(=O)NCC(C2CCCOC2)=O)(NC(=O)Cc2cccs2)CC(O)C1 64135,c1(C(=O)NC(C(=O)NC(c2nn(C)cc2O)C)C2CC2)ncccc1F 64136,Cc1oc(C(C)(C)C)cc1C(c1nnnn1C(C)C)NCCC1C=CCC1 64137,c1(C(N2C(C)CCC(c3ccccc3)C2)=O)cc2ccccc2oc1=O 64138,c1(OC)ccc(O)cc1C(N1CCCCC(NC(=O)C2=CCCC2C)C1)=O 64139,c1(CCC(=O)N(C)CC2CN(C(=O)CC3CCCC3)C2)ccn(C)n1 64140,CC(O)CCCC(=O)NCC1CCN(C(C2CN3CCC2CC3)=O)C1 64141,C1(CCNC(c2ccc(CC)o2)=O)CN(C(=O)C(c2ccc(C)o2)C)CCCO1 64142,c1(CS(C)=O)cccc(C(=O)NC2CN(C(=O)CC3C=CCC3)C2)c1 64143,C1(C(=O)NCC2(O)CCCN(C(C(C(CC)C)=O)=O)C2)CC(=O)N(C)C(=O)N1 64144,C1(O)(CCNC(CNC(=O)OCC)=O)CCN(C(=O)C(C)c2ccco2)C1 64145,C1(CC)CN(C(c2c(C)nsc2C)=O)CC1C(=O)NC(C)(CO)CCF 64146,Cc1cc(CN2CC(F)(C(=O)NCc3ccc(O)cc3F)C2)ccc1F 64147,N1(C(C(=O)NCCOCCOC)=O)CCCCC(C(=O)Nc2nn(C)cc2Cl)C1 64148,N1(C(C(CC)NC(C)=O)=O)CCC12CN(C(C1CCC(C(F)(F)F)O1)=O)C2 64149,C1(CC(=O)OC)Cc2ccccc2CN1C(c1cnc2c(Cl)cccn12)=O 64150,C1(CC(=O)N(CCC)Cc2ncc(C3CC3)o2)Cc2cc(C(F)(F)F)ccc2O1 64151,c1(C(=O)NCC2(NC(C(CC)=CC)=O)CCCCC2)cccc(S(N)(=O)=O)c1 64152,c1(C(N2C(CN(C(c3c(CC)n(C)cc3)=O)C)CCC2)=O)cnc2cc[nH]c2c1 64153,c1(C(N2CCC(NC(C3CCCC3(F)F)=O)(CO)C2)=O)ccn2c(O)nnc2c1 64154,C1(N(C(c2csc(C(=O)OC)n2)=O)CC)CCN(C(=O)COC)CC1 64155,C(CNC(c1cc(C(N)=O)co1)=O)(CC(F)(F)F)NC(c1ccc(OC)nc1)=O 64156,C1(CNC(=O)CCF)CN2CCCCC2CN1C(c1onc2ccccc12)=O 64157,Cc1cccc(C(=O)NC2(C)CCN(C(C3CC(C)(C)C3)=O)C2)c1N 64158,C=C(Cl)CC(C(=O)N1CCC2(CC1)N=N2)NC(c1cccnc1O)=O 64159,c1(NC)scnc1C(=O)NC(COC)C(=O)NCCCc1cccnc1 64160,C1(CCNC(c2c(C)snn2)=O)CCCCN1C(=O)COc1ccccc1Cl 64161,C(=O)(C(CC(C)C)NC(=O)C(C)CCOC)N(CC(CCC=C)O)C 64162,C1(NC(=O)CCc2cc(Cl)cs2)CC2(C1)CC2NC(c1cc(C2CC2)[nH]n1)=O 64163,C12(CNC(C=C(CCC)C)=O)CN(C(=O)C=Cc3ccc(C)cc3)CC(F)(C1)C2 64164,C1(S(N)(=O)=O)(C(=O)NC2CCC(NC(c3cnn(C)c3C(F)F)=O)C2)CCCC1 64165,N1(C(C(CCC)C)=O)CC(C2CCCCN(C(=O)CC3CSCCS3)C2)C1 64166,c1(C(=O)NC(CC)CNC(c2ccc(C)cc2F)=O)cccc2cccc(Cl)c12 64167,c1(N(CC(=O)NC)C)nc2cc[nH]c2c(=NC(C)c2ncccc2Cl)[nH]1 64168,c1(CC)cc(Br)ccc1C(=O)NC1CC(NC(c2csc(COC)n2)=O)C1 64169,N1(C(CC(CC(C)C)O)=O)CC2CCC1CN(C(=O)CN1CCSCC1)C2 64170,C1(NC(CC(C)c2cccnc2)=O)CC12CCN(C(=O)C(C)(C)CCC#N)CC2 64171,C(=O)(CC1C(=O)Nc2ccccc21)NCC1(OC)CCN(C(C(CC)C)=O)C1 64172,C1(CC)CN(C(C2CCC(C)CC2)=O)CCN1CC(c1cccc(C2CC2)c1)=O 64173,C(=O)(CCCCCS(N)(=O)=O)N1CCC(C)C1CNC(c1cc([N+](=O)[O-])c[nH]1)=O 64174,C(=O)(C(C)CN(C(=O)C(Cc1cc[nH]n1)NC(C1CC1C#N)=O)C)OC 64175,N1(C(C2C(C)CC(=O)CC2)=O)CC(NC(C2CCCCC2)=O)C2CCCCC12 64176,N1(C(C(C=C)O)=O)CC2CCCC1(CNC(c1cccc(OC)c1F)=O)C2 64177,c1(C(N2C(C)CN(C(C3CC(C#N)C3)=O)CCC2)=O)cc(S(C)(=O)=O)ccc1Cl 64178,CC(CC1CC1)C(=O)NC1CC(NC(=O)CCC2CC2(C)C)C1 64179,CC(CCC(C)(C)C)C(=O)N1CCN(CC(=O)NCc2cc(Cl)ccn2)CC1 64180,N1(C(CCC=C)=O)CC2(CCN(C(c3ccccc3-c3ncc[nH]3)=O)C2)C1 64181,CC1CCCC(CNC(c2cc(CNC(c3cc(Cl)n[nH]3)=O)nn2C)=O)CC1 64182,C1(C(=O)NCc2cccnc2O)CSCCN1C(c1ccnc(Br)c1)=O 64183,N1(C(Cc2cc(C)sc2)=O)CC=C(C(C)(C)C(=O)N2CCCCC2CCCO)C1 64184,c1(C(n2cc(C3(F)COC3)nn2)C)ccc(C(=O)NCCOC(C)(C)C)c(Br)c1 64185,N1(C(c2ccc(OC)o2)=O)CCCC(C2CCCCN2C(C2CCCOC2)=O)C1 64186,CC1(C)C(NC(=O)CCN2CCCC2)CC1C(=O)Nc1cccc(C(F)F)c1 64187,c1(C(N2CC(C)(OCC(=O)N(C)Cc3cc(C)no3)C2)=O)ccc(F)c(F)c1 64188,C(=O)(C(CC(C)(C)C)NC(c1ccc(F)cn1)=O)N(CCCCCC=C)C 64189,N1(CCC(=O)N(C2(O)CCCCC2)CC(C)CCO)CCOCC(C(=O)OC)C1 64190,Cc1nn(C)cc1S(=O)(=O)NC(c1cc(N(C)C)nc(Cl)c1)=O 64191,C12(NC(c3cc(O)ncn3)=O)COC(C1)C(NC(c1scnc1Cl)=O)C2 64192,N1(C(CCOCC)=O)CC2CC(NC(c3ccc(C4(C)CCO4)cc3)=O)CC1C2 64193,C1(C)(C(=O)NCC(CC)OC)CCCN1C(=O)C(C)N(CC)CC 64194,C(=O)(C(C(F)(F)F)C(F)(F)F)NC1CCN(C(CC2CCN(C)C2=O)=O)C1 64195,C1(CNC(=O)CCCC2CCCC2)CC2CCC1N(C(c1cccnn1)=O)C2 64196,C#CCCCCCNC(c1ccc(CNC(=O)CC2CCCCC2)nc1)=O 64197,c1(C(=O)NC(C(C)C)CNC(c2cnn(C3CC3(F)F)c2)=O)cnc(N)cn1 64198,c1(C(=O)NCC(C)N(C(c2n(CCC)ncc2)=O)C)ccc2c(c1)C(=O)CCN2 64199,N1(C(C)C)CC(C(N2CC(C(N)=O)(CNC(c3ccnnc3O)=O)C2)=O)CC1=O 64200,C(CCCCCO)(c1n(CC=C)nnn1)NCCCC(O)CC 64201,c1(C(=O)NCC2C(NC(C(CC)NC(C)=O)=O)CCCC2)ncc2[nH]ncc2n1 64202,N1(C(C(C2CCCO2)NC(Cc2cc(CC)no2)=O)=O)CCC(CCOC)CC1 64203,C12(C(N3CCC(C(C)NC(C=C(C)Cl)=O)C3)=O)CC3CCC(CC(C3)C1)C2 64204,Cc1cccc2c(CN3CCC(NC(=O)CCc4cnn(C)n4)C(O)C3)c[nH]c12 64205,C(c1nc(C)c(C)[nH]1)=CC(=O)NCC(CC)NC(c1ncc(C)cc1O)=O 64206,C1(CNC(c2ncncc2Cl)=O)C2CCC(C2)N1C(C12CC3CC1C2C3O)=O 64207,Cc1cc(=NCCC2CCC(=O)N2)[nH]c(N2CCN(CC(C)C)CC2)n1 64208,CCCC(CCC)C(=O)NC1CCCC(NC(c2cc(C(F)(F)F)on2)=O)C1 64209,CC1CCCCC1(C)C(=O)NCCOCCN(C(=O)COc1cncc(Cl)n1)C 64210,c1(C(=O)NCC2OCCCN(C(C3(C)COC3)=O)C2)ncnc2c1CCCC2 64211,C1(CNC(C(CC)CC)=O)CN(C(c2ccnc(C3CC3)n2)=O)CC1(C)C 64212,N#Cc1cc(C(N2CCN(C(C3CC4OC3C3CC43)=O)CC2CF)=O)ccc1F 64213,c1(N2CC3CN(Cc4cc(C)nc(C)c4)C3C2)ncnc2n[nH]cc12 64214,c1(CC)cccc(C(=O)NCC2(NCc3ccc(CSC)o3)CCOCC2)c1C 64215,Nc1cc(C(N2CCN(C(=O)CCCN3CCCC3)CC2C2CC2)=O)cc(O)c1 64216,c1(NC(NNC(=O)C23CC(n4cc(CCC)nn4)C2C3)=O)ncc(Cl)nc1OC 64217,C1(NC(c2n[nH]c(C)n2)=O)CCN(C(c2ccc(C(F)(F)F)c(F)c2)=O)C(C)C1 64218,c1(C(N2C(CNC(C3C(C(N)=O)C3)=O)CC2)=O)c(F)cc(F)cc1Cl 64219,c1(C(N2CC(C)C2)=O)c[nH]c2cc(-c3ccc(F)cc3F)cnc12 64220,c1(C(=O)NC(CC=C)CNC(C2(OC)CCSC2)=O)cn2ccsc2n1 64221,c1(C(N2CCC(N(C(CSCC)=O)CC)C2)=O)nnc(O)c(Br)c1O 64222,C(=O)(C1=CCC(C)(C)CC1)NC1C(C)N(C(=O)CCNC(=O)CO)CCC1 64223,C1(C(=O)NC2(C)CN(C(C(c3cscn3)N(C)C)=O)C2)CC2CCC(C1)C2O 64224,c1(C(=O)NCC(CC=C)NC(=O)CC)cnc2cccc(C)n12 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64242,C1(NC(COCCCC)=O)CC2CCC(C1C)N2C(c1cnn(CCF)c1)=O 64243,C(N=c1ccc(NC(c2cnnc(Cl)c2)=O)c[nH]1)c1c(SC)cccc1 64244,CCC(CC(=O)NCC1C=CCN1C(c1cc(OC)cs1)=O)C(C)C 64245,Cc1nc(C(=O)NCCC2CCCCN2C(=O)Cn2nnc(=O)[nH]2)c(C)s1 64246,C1(C(N2CCC(NC(C3CCOCC3)=O)C2)=O)(OCC)CCOCC1 64247,CCC(F)(F)C(C)(C)NC(=O)C(O)CNC(c1cc(OC)cs1)=O 64248,c1(C(=O)NCC(CNC(C2NC(=O)OC2)=O)O)ccc2nc(O)cc(O)c2c1 64249,Cc1cccc(Br)c1C(C(=O)NCC1(O)CCCOC1)NC(=O)CCC1(C)N=N1 64250,c1(C(=O)NCCC(C)(C)NC(C2C(C)OCC2)=O)ccc(C(F)(F)F)cn1 64251,CC1(C)CCCN(C(c2scnc2Cl)=O)C1CNC(=O)Cc1ccnc(Cl)c1F 64252,CCC(CNC(C)=O)CC(=O)NC1(CO)CN(C(C2CC(OC)(OC)C2)=O)C1 64253,c1(CC(=O)NC2CCCC(NCC3(C)CC3)C2)ccc2ccccc2c1 64254,C1(NC(C2(CC=C)CC2)=O)CCC2CCN(C(c3csc(=NC4CC4)[nH]3)=O)C1C2 64255,N1(C(C(C)CNC(C2CCCN2C2CC2)=O)=O)CCCCC(CO)C1 64256,N1(C(C(N2CCNC2=O)C)=O)CC2(CCCC2)C1C(=O)NC1CCC2CCC12 64257,C(C1CN(C(C2(C)CCCC2O)=O)CC1C(=O)NCC(C1CCCC1)OC)=CC 64258,C(=O)(C(C)(C)COCC)N(CC(=O)NC(C=C)CO)CCOC 64259,C1(N(C(CCOCCOC)=O)C)CCN(C(c2cnn(C)c2N)=O)CC1C 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64277,c1(C(=O)NC(=O)NCC(C)N(C(C(=O)N(CC)CC)C)C)cc(Cl)ccn1 64278,c1(CNC(C(=O)Nc2ccc(-c3n(C)ccn3)cc2)=O)cc(N)cc(F)c1 64279,C(=O)(CC(CC)C(C)C)N1CCN(C(c2c(OC)nccc2)=O)C(C2CC2)C1 64280,N(C1CCc2c1cc(F)c(F)c2F)C(c1c(C)c2ccc(C)cc2cc1)=O 64281,C(CCCC(=O)NC1CCCC1NC(=O)Cc1ccc(C)o1)OC 64282,c1(SC)nc(N(C(C)CCNC(=O)C(CO)NC(N)=O)C)cc(Cl)n1 64283,CN1C(=O)OCC1C(=O)NCC12CC1CN(C(=O)CC1(O)CC1)C2 64284,C(C(C(=O)NC1CC(N(C(=O)CCF)C)C1)C(F)(F)F)OC 64285,C(c1cocn1)=CC(=O)NCC1(C(=O)NCC2(C(C)(C)C)CCC2)CC1 64286,c1(CC)cc(C(=O)N(C2CN(C(=O)COc3cnn(C)c3)C2)C)c2c(c1)CCO2 64287,c1(CC(C)NCC2CC(CC(=O)O)C2)ccccc1 64288,c1(C(=O)NC2C(C(C)(C)C)N(C(=O)C(=O)N(C)C)CC2)nnn2c1CCCC2 64289,C(N=c1ccnc(C2CCCC2)[nH]1)C1(NC(c2c(C(C)C)ocn2)=O)CC1 64290,c1(OC)cc(C)c(C(=O)NC2(CCNC(C34CCCC3C4(F)F)=O)CC2)cn1 64291,c1(OC)c(Br)cc(CN2C(C(=O)NC(c3ccc(I)cc3)C)CC3CC23)cc1Br 64292,C(C(C(C)C)NC(=O)C(C#N)=C1CCCC1)NC(C(C)OCCOC)=O 64293,CC(C)(C(=O)NCC1CCC(NC(=O)CN2CCCC2=O)C1)c1cc[nH]n1 64294,c1(N2CCN(Cc3c(C)c(F)ccc3F)C3C2C3)ncnc2c(F)cccc12 64295,c1(C(N2CCCC(C(C)NC(c3cc(C)sn3)=O)C2)=O)n[nH]c2cc(Cl)ccc12 64296,Cc1cnn(CCC(N2C(C(N3CC(OCCF)C3)=O)CC2C)=O)c1 64297,C1(OCC)CC(NC(=NCCC(=O)N2CCCC2)NC2CCC2)C12CCOCC2 64298,C1(C(=O)NCC(CC2CC2)OC)CN(C(c2ccc(Cl)cn2)=O)CC12CC2 64299,CC1(C)CCCN(C(c2nccc(Cl)c2O)=O)C1CNC(=O)Cc1c[nH]nc1O 64300,c1(C(N)=O)cccc(CC(=O)NCCOCCCNC(=O)C(O)C(F)F)c1 64301,C1(NC(c2nc(C)oc2C)=O)CCN(C(=O)C(C)Cc2cnn(C)c2)CC1F 64302,CCC(CC(=O)NCC1CN(C(c2oncc2C)=O)C2COCC2O1)C(C)(C)C 64303,C(CO)(C(=O)N1CCCC1C(C)(C)NC(=O)C(C)OCC1CC1)OC 64304,c1(C(N2C(C)C(C)N(C(c3ccns3)=O)CC2)=O)cn2c(n1)C(=O)N(C)CC2 64305,Cn1cnc2c(C(=O)NCCC(O)CNC(C34CC(F)(C3)C4)=O)ccnc12 64306,C1(CNC(C(CC)n2cncn2)=O)CN(C(=O)Cc2csc(Cl)c2)CC1C 64307,C12(NC(c3csnn3)=O)CCOC(CNC(C3C=CC=CC=C3)=O)(C1)C2 64308,c1(C(N(CC(O)CNC(=O)COc2ccc(Cl)nc2)C)=O)cc(F)c(F)cc1F 64309,C1(CCNC(C2CCNC2=O)=O)(C(=O)Nc2ccccc2)CCCC1 64310,C1(NC(C2C(=C)C2)=O)CCCCC1CNC(c1cn(-c2ccccc2)cn1)=O 64311,C(=O)(CCC(C(=O)OC)NC(=O)C(N1CCC(F)C(O)C1)C1CCCSC1)OC 64312,N1(C(C2(NC(c3c(CC)c[nH]c3)=O)CCOCC2)=O)CC(OC)C2(CC2)C1 64313,O=C1NCC2(CCCN(Cc3nc4c(s3)CCCC4)C2)CO1 64314,C1(NC(CC2C(C)(C)C2)=O)CCN(C(c2cccc(O)c2)=O)CC1C(N)=O 64315,c1(C(=O)NCC2N(C(C(C(=O)OC)C)=O)CCC2)ccc(O)c(O)c1Cl 64316,C1(C(=O)NCC2CCCCN(C(Cc3c(C)noc3)=O)C2)Cc2ccncc2C1 64317,C1(C(=O)NCCC2(O)CN(C(C3(C#C)CC3)=O)C2)CC2CCC1CC21OCCO1 64318,Cc1[nH]c(C(=O)NCC(F)(F)F)c(C)c1C(=O)NCC1CN(C(C)C)CCO1 64319,CC#CCCCC(=O)NC(COC)CC(=O)NC(c1nncn1C)CO 64320,C12(C(=O)NCC3(OC)CN(C(=O)C(F)C(C)C)C3)CC(C)(C1)OC21CCOCC1 64321,c1(C(C)C)nc(NCC2CC(N3CCCC3)C2)cc(N(CCCC(F)F)C)n1 64322,C(N=c1[nH]c(=NC(CCO)C(F)F)[nH]c2c(F)cccc12)C1(OC)CCCC1 64323,N1(C(c2sc(CC)c(C)c2)=O)CCN(C(=O)C(C)OC2CCCCC2)C(C)C1C 64324,N1(C(C(CC)O)=O)CCN(C(CNC(c2cc(C(F)F)[nH]n2)=O)C(F)(F)F)CC1 64325,C1(CNC(c2ccc(CC)c(F)c2)=O)CC2(CCC2)CN1C(=O)C(C)C(C)(C)C 64326,c1(CCC(=O)NCCOCCNC(C(C)CO)=O)nc(=O)c2ccccc2n1C 64327,C(C(C)(CNC(c1nonc1CC)=O)OC)NC(C(C)OCC#C)=O 64328,C1(CNC(C2(CC#C)CCCC2)=O)COCCN(C(C2CC3(CC(=O)N3)C2)=O)C1 64329,C(=O)(C(F)CCC(C)(C)C)NC(C)CCCNC(c1cccnc1O)=O 64330,c1(C(N2CCC(OCCNC(CS(=O)(=O)NCC)=O)C2)=O)ccc(C)cc1F 64331,CCC(CC(C)C)C(=O)N1CC2C(CC(=O)NCC3CC3C(C)C)C2C1 64332,C12(N(c3cccs3)C(=O)NCCC3CCC4CC34)CCN(CC1)CC2 64333,N1(C(CC(C)(C)CC(F)F)=O)CC2CCN(C(c3ncccc3Cl)=O)CCC2C1 64334,N1(C2CC(C(=O)OC)C23CCC3)CC(NC(=O)OC(C)(C)C)CC(C)(C)C1 64335,C(=O)(C1=NOC2(CCC2)C1)Nc1c(C(=O)OCC)ncc(Cl)n1 64336,C1(n2cc(CCC(C)O)nn2)CN(C(c2cc(C3(O)COC3)on2)=O)CC1C 64337,c1(N(C2CCCN(C(C(CCC)(C)O)=O)C2)CCO)ncccc1[N+](=O)[O-] 64338,c1(CC)onc(C)c1C(N1CCC(OCCNC(=O)C(C)=CCO)C1)=O 64339,C(=O)(CC(F)(F)CC(=O)OC)NC(CNC(c1c(CC)n(CC)nn1)=O)C1CC1 64340,Cc1ccc(C)n1CC(=O)NC1(c2ccccc2)CC(NC(C2CC(F)C2)=O)C1 64341,CN=S(C)(=O)c1ccc(C(N2CCCCC2C(N2CCCC2)=O)=O)cc1 64342,c1(CN(C(Cl)C(F)(F)F)C)ccc([N+](=O)[O-])cc1OCCO 64343,c1(NCC(C)O)cc(S(=O)(=O)N2CCCC2CC(C)(C)C)ccc1C#N 64344,c1(CC(=O)N(C(CN(C(C(CCSC)O)=O)C)C)C)cc(F)cc(F)c1 64345,C(C)(c1cccnc1)=CC(=O)N(CC(CNC(CCC#C)=O)O)C 64346,c1(CNC(COC(C)=O)=O)ccnc(C(=O)NCC2CC(C)(O)C2)c1 64347,CN=c1nc(N(C)CCOCC(F)(F)F)[nH]c(=NCc2ccc(Cl)c(F)c2Cl)[nH]1 64348,c1(-c2cc(C(N(CCC3CC(C(=O)OC)C3)CC3CC3)=O)no2)cccc(O)c1 64349,c1(OC)ccc2c(c1)CCCC2NC(N1CCC2(CCCOC2)C1)=O 64350,C1(NC(CC)=O)CN(C(c2ccc(NC)cc2)=O)Cc2nccn2C1 64351,N1(C(c2cc(CC)nn2C)=O)CC2CCCC2C1C(N1CC(CO)CC(C)C1)=O 64352,C1(CN(C2CCC(c3ccccc3)C2)C(COC)C2(C)CC2)CCCC(O)C1 64353,c1(C(=O)NCC2(OC)CN(C(C(COC)OC)=O)C2)cnc(O)cc1OC 64354,c1(C(=O)NC(COC)CNC(=O)C(COC)N(C)C)cc(O)ccc1C 64355,c1(C(=O)NCCC2N(C(C=CC(=O)N(C)C)=O)CCC2)ccc(C)c(C)c1Cl 64356,C1(NC(CCCC#C)=O)CN(C(C2(C3CCCCC3)CC2)=O)C2CCCC12 64357,N1(C(C2C(C(=O)OC)C2)=O)CCOCC(C)(CNC(c2ccc(C)c(F)c2)=O)C1 64358,c1(NC(C2(C)CN(C(C(CC)=CCCC)=O)C2)=O)ccc(O)c(CO)c1 64359,N12CCOCC(C1)N2CCO.c1(NC=O)nc(C)n(C)n1.c1(OC)cccnc1 64360,N1(C(COCC=C)=O)CC(NC(=O)C=Cc2ccc(C)s2)CC12CCOC2 64361,C1(C)(C(=O)NC2CN(C(c3c(SC)cn(C)n3)=O)CC(F)C2)CCS(=O)(=O)CC1 64362,c1(C2(C(=O)NCC3(F)CN(C(C4CCCO4)=O)C3)CCCC2)ccc(F)cc1 64363,N1(C(C2N(C(C3=CCCC3C)=O)CC(C)(C)C2)=O)CC2CCC(O)C(O)C12 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64695,CC1(C)CCCC(C(=O)NCC2CC(NC(=O)C(c3ccccc3)O)C2)O1 64696,CC(CCC(C)(C)C)C(=O)NC1CN(C(=O)CN2CSCC2=O)CC1O 64697,c1(CN(C)C)ccc(-c2nc(C3CCCO3)n(-c3ccc(Br)cc3)n2)cc1 64698,c1(C(=O)OC)ccc(CNC(=O)N(C2CC2)Cc2ccco2)c([N+](=O)[O-])c1 64699,N1(C(C(=Cc2ccccc2)C)=O)CCC2(CCCN(C(C3CNC(=O)N3)=O)C2)C1 64700,c1(CC)nc(C)c(C(=O)NCCOCc2ccc(OC(C)=O)cc2)s1 64701,N1(C(C2(CN(C)C)CC2)=O)CCOC2(C1)CN(C(c1ccnnc1O)=O)C2 64702,CC1CC(F)(F)CN1C(=O)Nc1ccc(F)cc1-c1ccnn1C1(C)CC1 64703,Cc1cnc2c(cnn2CC(=O)NC2CCCN(C(c3cccs3)=O)CC2)c1 64704,c1(CC(=O)N(CC(CNC(C2C(COC)C2)=O)O)C)cc(C)cc(F)c1 64705,c1(CNC(c2n(CC)nnn2)CCCC2CC2)ccccc1OCC 64706,c1(CCNC(N2CCC(CNC(CC)=O)C2)=O)ccc2c(c1)COC2 64707,C(c1cc(C)cc(C)c1)=CC(=O)NCCN(C(C(C(C=C)C)C)=O)CC 64708,C1(NC(c2oc(C)c(CO)c2)=O)C2CC3C1C3C2C(N1CCC(C)(CCO)C1)=O 64709,CCC(C)(CO)C(=O)N1CC(CNC(=O)CN(C)C(=O)OC)C(F)C1 64710,C(CN=c1ccnc(NCc2cccc3ccccc23)[nH]1)C1C(C)(C)NC(=O)C1 64711,c1(C(=O)NCC2C(NC(c3ncc(OC)nc3)=O)COC2)cc(C)ccc1Cl 64712,CC1(C)CC(n2nc(C(F)F)nc2-c2nc(C3CC3)sc2Br)CCO1 64713,Cc1ccc(CCC(=O)NCC2CCC2NC(=O)CCC(=O)N(C)C)cn1 64714,c1(C(N2CCOC(C)(C3CC3)C2)C(=O)NCCOC)ccc(C)c(I)c1 64715,C(=O)(C1=NOCC1)N(C(CCNC(C1CC(CC)C1)=O)C)C 64716,N1(C(C2CC=CCC2)=O)CC2=C(C1)CN(C(C1(O)CC(F)(F)C1)=O)C2 64717,Cc1cc(C2CCC2)ncc1C(N1CCC(NC(C2CCC(C)(C)O2)=O)C1C)=O 64718,N1(C(C=CCCC)=O)CC(OC)C(NC(=O)C(C)(C)OCC)C1 64719,c1(C(=O)NCC2C(C)CN(C(=O)CS)C2)nc2ccccc2s1.c1cc(F)c[nH]1 64720,C#CC(C)(C)C(=O)NC1CNCCC1c1ccc(OCC)cc1 64721,c1(C(N(CC(CC)NC(C2CC(C)(C)C2)=O)CC)=O)cc2c(nc1O)CCCC2 64722,c1(CC)[nH]c(C(=O)NC(C)(CNC(C2CCOC2)=O)c2cccs2)nc1Cl 64723,O=C1CC(C(=O)NC2CCC=CCC2)N(C(=O)CCC2CC2)C1 64724,CCCCCCCN(C(=O)C(C1CCCO1)NC(=O)C=CC1CCC1)C 64725,C1(NC(C2CCC(C(C)C)CC2)=O)CN(C(C2CC2(C)Br)=O)Cc2nccn2C1 64726,Cc1ccccc1C=CC(N1CC(C(C)NC(c2cccc(F)n2)=O)C1)=O 64727,C(CN=C(NCc1ccc(C2CC2)c(F)c1)N1CCC(C)C1C)OC 64728,C1(C(=O)NC2CCN(C(CCC(C)C#N)=O)CC2)CCc2cn(C)nc2C1 64729,C(=O)(CCCCC(N)=O)N1CCC(c2cn(-c3c(F)ccc(OC)c3)nn2)C1 64730,N1(C(C(C)C)=O)CCC(C2CCN(C(=O)C(F)C3CCC3)CC2)C1 64731,c1(C(N2CCNC(C(N3CCC(O)C(O)C3)=O)C2)=O)cc(I)ccc1F 64732,Cc1[nH]nc2c(C(N3CCCC3CNC(c3ccc4cncn4c3)=O)=O)cccc12 64733,c1(C(N2CC(OC)C(NC(=O)CC3(C)CCCO3)C2)=O)cn2ccccc2n1 64734,C(CCCC(c1cn(C2(C(N)=O)CC2)nn1)NC(=O)CCn1cc(CO)nn1)OC 64735,C(=O)(CCCCCC(C)O)NCCCN(C(C=Cc1c(C)noc1C)=O)C1CC1 64736,C(=O)(C1c2ccccc2C2CC1C2)NC1CNCC(C)(C)C1 64737,C1(NC(C2N(C(C(C)Cn3ccnc3)=O)CC2)=O)CCN(C)C1=O 64738,CC1(C)CN(C(C2CCN(CCO)C(=O)C2)=O)CC1NC(=O)CCc1nc[nH]n1 64739,N1(C(C(CSC)O)=O)CC(CNC(C2(C)CCC3CC3C2)=O)CC1(C)C 64740,c1(C(N2C(C)(C(N3CCN(C)CC3)=O)CC2)=O)cc(Cl)cc([N+](=O)[O-])c1 64741,Cc1cc(CN2CC3CC3(C(=O)Nc3cc(C(F)(F)F)c(Br)cn3)C2)ccc1Br 64742,c1(C(N(CCCCNC(CC2CCC(C)C2)=O)C)=O)cccc(F)c1Cl 64743,C1(NC(=O)C2=CCN(C(c3ccc(CO)s3)=O)C2)CC2CCCC(C1)C2 64744,CC1CC2CC(C(=O)N(C3CN(C(=O)CCn4cccn4)C3)C)(C2)O1 64745,c1(OC)cncc(C(=O)NCCC(C)NC(=O)C(O)CCc2ccccc2)c1 64746,c1(C(=O)NCC2C3CN(CC(COC(COC)C)O)CC32)c(OC)cccc1F 64747,Cc1cccc(C(=O)NCCCCCNC(=O)C(c2cnn(C)c2)O)c1O 64748,c1(-c2ccc(C(=O)Nc3cc(OC)c(Br)nc3)nn2)ccc(S(C)(=O)=O)cc1Cl 64749,Cc1ccc(C)n1CC(N1CC(O)(C(C)NC(c2cnn(C3CC3C)c2)=O)C1)=O 64750,Cc1cc(=NC(CF)c2ccccc2Cl)[nH]c(-c2cccc(Cl)c2)n1.C1CO1.CCO 64751,C1(CNC(C2C(C)(COC)C2)=O)(OC)CCN(C(=O)CCNC(=O)CO)C1 64752,c1(C(=O)NC(CC#C)(C)C(=O)NCCCN=[N+]=[N-])ccc2cc[nH]c2n1 64753,N1(C(C(CCC#C)O)=O)C2CCC1CC(F)(CNC(c1cccc(CC)n1)=O)C2 64754,Cc1cc(C)[nH]c(=NCc2cn3ccc(-c4cnc(OC(C)C)nc4)cc3n2)n1 64755,N1(C(C(C(=C)C)(C)O)=O)CC(NC(c2ccc(CC3CC3)s2)=O)C(C2CC2)C1 64756,Cc1cc(=O)n(C)nc1C(N1CCCCC1CN(C(=O)CC1OCCO1)C)=O 64757,c1(C(N(CCCCN(C)C(C2CC(F)C2)=O)C)=O)n[nH]c2c1CCCCC2 64758,Cc1nn(C2CC2)c(C)c1CN1CC(C)CCC1c1ccccc1 64759,Cc1ccc(O)c(C(N2CC3CC2CN3C(=O)Cc2ccc(Cl)s2)=O)c1 64760,C1(CC=C)(C(=O)NC(Cc2cnc[nH]2)CO)CCN(C(c2csnn2)=O)C1 64761,N1(C(=O)OC(C)(C)C)CCC(CN2CCC23CCCC3)CC1NC(=O)C(F)(F)F 64762,C1(CNC(C23CC(C(=O)OC)(C2)C3)=O)(NC(=O)CC2CSCCS2)CCOCC1 64763,N1(C(c2cnc(CC)o2)=O)CCOCC1CN(C(=O)CCOCC(F)F)C 64764,C(CCCCC(=O)NC1CC(CNC(=O)CC2OCCOC2(C)C)C1)NC(C)=O 64765,C1(OCC)CC(N(C(NC(=NCCF)NCC2CC2)COC)C)C12CCCCC2 64766,CCCC(C)CC(=O)NC1CC(F)(CNC(c2cc(C)nn2C(F)F)=O)C1 64767,N1(C(c2cc(C(C)C)[nH]n2)=O)CC(NC(c2c(Br)cnn2C)=O)CC(C)C1 64768,Cc1cc(O)nc(C)c1C(=O)NCC(c1ccccc1)CNC(N)=O 64769,c1(CNc2c(CC(=O)NCc3ccc(F)cc3)cccc2)cnc(Cl)cc1F 64770,CC#CCC(C(=O)NC(c1cn(C)nc1C)C)NC(c1cn(C(C)C)nn1)=O 64771,C1(NC(=O)CC2CC3(CC3)C2)CCN(C(=O)CS(=O)(=O)Cc2cccs2)CC1F 64772,C(CC(C(=O)NC1C2CN(Cc3ccc(Br)[nH]3)CC12)NC=O)SC 64773,C1(CCNC(C2CC2C2CCCC2)=O)CCCN(C(=O)CCc2cn[nH]c2)CC1 64774,Cc1ccc(CCN=C(NCC(C)(C)C2CC2)NCC2CC2)c(O)c1.C(C)C 64775,c1(C(=O)NCC(Cn2cc(CCSCC)nn2)(C)C)nc2sccn2c1C 64776,c1(C(=O)NC2COCCN(C(C(C)(Cl)Cl)=O)C2)cccc2cnsc12 64777,N1(C(CCSCc2nc(C)sc2)=O)CC(O)CC1CNC(=O)Cn1cnnc1O 64778,Cc1ccc(CN(C(=O)CNC(=O)C(C(C)C)NC(c2ccco2)=O)C)c(C)c1 64779,Cn1ncc2c1CN(C(C1CC3CC3N1Cc1cc(F)cnc1Cl)=O)C2 64780,C1(C(=O)NC(C2CCCO2)C)CC(N(C(=O)CNC(C2CC(N(C)C)C2)=O)C)C1 64781,C1(C(=O)NC(c2ccc(F)cc2)CC)CC(O)CCN1C(c1sc(C)cc1C)=O 64782,C1(C(=O)NC(CCC(C)C)C)CC1C1CN(C(C2(O)CCCC2)=O)C1 64783,CCC(C(=O)N(C1CCN(C(c2ccsn2)=O)C1)CCO)SC 64784,c1(C(=O)NC2C(C)CN(C(c3cccnc3Cl)=O)C2)cn2cccc(Br)c2n1 64785,c1(C(N2C(C(C)(C)C(=O)NCc3ccccc3)CCC2)=O)cc2ncccc2[nH]1 64786,C1(CN=[N+]=[N-])CCCN(N2CCC(n3ccccc3=O)CC2)C1 64787,CC1=C(C(=O)N(C2CCN(C(=O)CCC3CC(F)(F)C3)C2)C)CCO1 64788,N1(C(C=C(CC)CC)=O)CCC2CN(C(c3c(N)sc(C)c3C)=O)CCC2C1 64789,N1(C(C(C)=CC=C)=O)CCC2(CCNC2=O)C1 64790,c1(CC(N2CCC(N(C)C(c3ccnc(C(F)F)c3)=O)C2)=O)cc(F)ccc1F 64791,N1(C(C(=Cc2ccccc2)C)=O)CCC2(CC2NC(=O)CC23CCCC2C3)C1 64792,c1(C(=O)Nc2cc(Cl)cc(F)c2F)noc2c1CCc1sccc1-2 64793,c1(C(=O)NCCCOCCNC(CCc2ccc(C)s2)=O)nccc(F)c1Cl 64794,C=C(F)C1(CC(N2CCCCC2CC(=O)NCC#CC2CC2)=O)CCC1 64795,Cc1ncsc1COC(CC1(C(C)(C)O)CN(C(=O)OC(C)(C)C)C1)OC.O 64796,N1(CC(CC)C)CCCC(NC(c2cc(C(F)(F)F)nn2CC)=O)C1C 64797,C(=O)(C(C)(C)C(=O)NCc1cc[nH]c1C(N1CCSC2CCC12)=O)N(C)C 64798,c1(CC)sc(C(=O)NC(C)C(C)NC(c2ccc(CF)cc2)=O)cc1Br 64799,c1(NC(C)=O)ccc([N+](=O)[O-])c(C(=O)NC2CCCC2NC(=O)CC2(C)CC2)c1 64800,C1(C(=O)NCC2(C(N)=O)CN(C(c3cc(C(C)C)on3)=O)C2)CCCC(F)C1 64801,CC(CC(=O)N1CC(F)(CO)C1)C(C)(C)NC(=O)C(c1ccccc1)F 64802,C1(CN(C(C=C(C)C(C)(C)C)=O)C)CC(F)CN1C(=O)COCC(F)F 64803,C1(C(N2CC(n3cc(CNC(c4ccccc4O)=O)nn3)C2)=O)CC1C1CCC1 64804,c1(C(C(=O)Nc2c(CC)cccc2)N(C2(C)CC2)C)ccc(C)cc1CC 64805,C1(CNC(C=Cc2ccc(CC)o2)=O)CC(F)(F)CN1C(=O)CC1C=CCCC1 64806,N1(C(CCCC(OC)OC)=O)CCCC12CCN(C(=O)C(CO)N(C)C)C2 64807,C(CC(=O)NC(C)(C)CCNC(=O)COc1ccc(Cl)c(F)c1)(C(F)(F)F)OC 64808,CCC(C)C(C)(c1nnnn1C1CC1)NCc1nc(C(F)(F)F)n[nH]1 64809,C(c1ccccc1Cl)=CC(=O)NC(CNC(C1C=CCC1)=O)CC(F)(F)F 64810,C1(C(N(CCN(C(=O)Cc2cn(C)nn2)CC)CC)=O)(OC)CCC(C)C1 64811,N1(C(c2c(C(=O)OC)n(C)nc2)=O)CC(NC(C2CNC(=O)C2)=O)CC2(CC2)C1 64812,c1(OC)n[nH]cc1C(=O)NCC(CNC(=O)Cc1ccsn1)CO 64813,c1(C(=O)NCCNC(C(C)C)=O)csc(C(C)NC(=O)C(=O)NC2CC2)c1 64814,c1(COCC)cccc(OC)n1.N12CC(C(CO)C1)CNC(=O)C1(CC1)C2=O 64815,N1(C(C2C(NC(CCOC(C)=O)=O)CCOC2)=O)CC2(CNC(=O)N2)C1 64816,N1(C(C2C3CC(NC(C4(C5(C)CC5)CC4)=O)C(C3)C2)=O)CC2CCC(C1)C(=O)N2 64817,C1(C)(c2cn(Cc3cc(C)on3)nn2)CCCN1C(=O)C(c1ccc(Cl)s1)C 64818,C1(C(N2CCC(OC(C)=O)C2)=O)CCN(C(=O)C(F)C2CCC2)C(C)C1 64819,N1(C(Cc2ccc(C)nc2)=O)CCN(C(c2ccc(C(N)=O)[nH]2)=O)CC1CF 64820,C(=O)(C(O)CC[S+](C)C)NCC1CC(NC(C(C)Cc2cccc(Cl)c2)=O)C1 64821,N1(C(C2C(C=C)C2)=O)CCc2c(CNC(=O)CCCc3nccs3)cccc2C1 64822,CON(C(=O)C1(C#N)CC1C)C(C)c1ccccc1C 64823,C1(CNC(C(=O)NC(c2cscn2)C)=O)(CO)CC2CC2C1 64824,C(=O)(C(C)(F)C(C)(C)F)NC1CC(CCNC(C(C(=C)C)(C)C)=O)C1 64825,C1(NC(CCN(C)CCO)=O)CCCCCC1C(=O)NCC1CCSC1 64826,Cc1ccc(-c2ccc(CN(CC(O)CO)C)cc2)cc1F 64827,C1(CCNC(C2(SC)CC2)=O)CCCCN1C(=O)CC1CCCC(=O)N1 64828,c1(C(=O)NCCCCN(C(CC2C(OC)CC2)=O)C)cnn(CC(C)(C)O)c1C 64829,c1(CC)ccc(C(N2CCC(OCCNC(=O)C(C)O)C2)=O)cc1CC 64830,C1(N(C(C(C)SC)=O)C)CCC(CNC(=O)Cc2sccc2Cl)CC1 64831,n1(-c2scc(C)n2)c(C(N2CCN(C(=O)C(C)O)CC2C)=O)nc2ccccc12 64832,c1(CCNC(=O)NC2C(CN(C)C)CCC2)nccc(=O)n1C 64833,CC1CC=C(C(=O)N2CCC(F)(F)C(CNC(C3CCCO3)=O)C2)CC1 64834,N1(CCCN2C(C(=O)O)CCC(F)C2)C(=O)C(=O)N(Cc2ccccc2)C1=O 64835,CC1(C)CC(C)(CO)CN1C(C1CC(=O)CN1C(C1CCCC(=O)C1)=O)=O 64836,Cc1cn(C)c(C(c2nnnn2C2CCCC2)NCCCCCCN(C)C)n1 64837,C1CCN(C(C=CSC)=O)CC1.c1ccnn1C 64838,N1(c2snc(C(C)(C)OCC)n2)CCC2CC(CNC(=O)C(C)CO)CCC2C1 64839,N1(C(CCOCC)=O)CC(NC(c2[nH]c(C)c(C(C)=O)c2C)=O)CC1(C)COC 64840,N1(C(=O)NC2CC(C#N)C2)CCC12CCCOCC2 64841,c1(CC(C)NC(=O)C(=O)N(CC(F)F)C(C2(O)CCC2)C)ccc(Cl)cc1 64842,Cc1ccc(N(CC(CO)NC(C2CCCN(C(=O)OC(C)C)C2)=O)C(C)=O)cc1 64843,C1(NC(Cc2nc(C)[nH]n2)=O)CCCCC1CNC(C1(C)CCN(C)C1)=O 64844,C1(C(=O)NCC(CC=C)(C)C)CCCN(C(C2CCC2(OC)OC)=O)CC1 64845,C(C)(c1cnn(C)c1)=CC(=O)NC(c1ccc(OCC#N)cc1)C(=O)OC 64846,c1(CNC(=O)NNC(=O)c2cc(I)n[nH]2)c(Br)cc(Br)c(O)c1Br 64847,CC(C(C)C(=O)N1CCOC(CNC(C2CC23CC(C)(C)C3)=O)C1)S(C)(=O)=O 64848,CC1CN(C(c2conc2C2(C)COC2)=O)CC1NC(=O)CC1(O)CCOC1 64849,c1(C(C(=O)NC(C2N(C(c3c(OC)n[nH]c3)=O)CCC2)C)O)ccc(Cl)cc1F 64850,C1(C(=O)NCC(C2CC2)OC)CN(C(C2(O)CCOCC2)=O)CC(C)O1 64851,C1(C(N(CCCC#C)C)=O)CN(C(=O)CC2(N(C)C)CCC2)CCO1 64852,C(=O)(CC(C)CC(C)C)N1CCN(CC(C)NC(C=Cc2ccc(C)o2)=O)CC1 64853,Cc1c(C(N2CCCC(C)C2CNC(=O)C2CC2)=O)cc([N+](=O)[O-])cc1Br 64854,c1(N(C)Cc2onc(CC)n2)cc(N2CCN(C(C)CNCC)CC2)ncn1 64855,c1(CC)nocc1CN(C(=O)C(=O)NCCn1cc(I)cn1)C 64856,n1(CC)cnc2nc(=NCc3ncc(Br)s3)[nH]cc12.C1(NC)CCCC1CO 64857,N1(C(CCC(C)OCC)=O)CCCC12CCN(C(c1cc(F)cnc1O)=O)C2 64858,Cc1nc(C(C)C)ncc1C(N1CCCC(CCNC(C2CCCS2)=O)CC1)=O 64859,CC(=O)CC(C)(C)CC(=O)NCCC1CCCN(C(=O)C(F)(F)CC(C)C)CC1 64860,Cc1cn2c(n1)CCC(NC(=O)NCc1ccnn1Cc1ccccc1)C2 64861,c1(C(=O)NC2CC(CNC(C(C#C)(C)C)=O)C23CCC3)cccc2sccc12 64862,c1(C(=O)NCc2ccc(-c3c(OCC)c(F)ccc3)cc2)c(Cl)ccc(Br)c1Cl 64863,c1(NC2CC(C)CC(C)C2)nccc(=NCCCCC2CCCC2)[nH]1 64864,C1(NC(C(C(C)C)F)=O)CCC2(CC1)CCN(C(=O)CCC1CCOCC1)CC2 64865,N1(C(CN(CCC)C)=O)CC(NC(c2ncoc2C)=O)C2CCCCC12 64866,CC1CCC(CNC(=O)CCN(C(=O)CN2CCNC2=O)C2CC2)C1 64867,c1(CC)conc1CC(=O)N(C)CCOCCNC(C1(OCC)CC(=O)C1)=O 64868,N1(C(c2c(C)n(-c3ccccn3)nc2)=O)CCCC(NC(=O)C2=CCSC2)CC1 64869,S(=O)(=O)(c1ccc(Br)cc1)NCCC(=O)NCCNC(c1ccccn1)=O 64870,C1(N(CC(=O)NC2CCSCC2)CCN2CCCC2)CC2CCC1C2 64871,O=CN1CCN(C(C2CC23CN(C(=O)CCc2ccc(Br)cc2F)C3)=O)CC1 64872,N1(C(C2C3(CCN(C(C4N(C)CC(F)C4)=O)C3)C2)=O)Cc2ccc(O)cc2C1 64873,CC(F)(F)C(C)(C)CS(=O)(=O)NCCc1ccnn1-c1ccccc1 64874,c1(C(=O)NC2C(CNC(c3cnn(CC)n3)=O)CCC2)cccc(OC)c1OC 64875,c1(C(C)=O)cc(C(=O)NC(CNC(c2cc(OC)nn2C)=O)C2CC2)oc1C 64876,c1(OCC)n[nH]c(C(N2CC(C)(C)C2c2cnn(C)c2)=O)c1Br 64877,Cc1nc(C)n(CCC(N2CCC(C(F)F)(CNC(c3c[nH]nc3C)=O)C2)=O)n1 64878,N1(C(Cn2cnc(=N)[nH]2)=O)CCCC(CNC(=O)CCc2ccc(O)nc2)CC1 64879,CC1CN(C(=O)CC2(CNC(C3(Cl)CCC3)=O)CC2)Cc2nncn21 64880,CC1OC(C)CC1C(=O)NC(C)CC1CN(C(C2CCCS2)=O)C1 64881,c1(CC(=O)NC(CC)CC(=O)NC(C(C)C)C2CCC2)cc(C)nc(O)c1 64882,Cc1ccc(C(=O)NC(C)CNC(c2cncc(C3CC3)c2)=O)c(C(C)C)n1 64883,C=CC(C)(O)CC(=O)NC(C)(C)CNC(=O)C(C(C)(C)O)Oc1ccccc1 64884,N1(C(c2cnc(C)s2)=O)C(CC(=O)N(CC(N)=O)CC(N)=O)C2CCCC12 64885,N1(C(C(C)NC(CC)=O)=O)CCC2(CC1)CC2(C)C(N1CCNC(=O)CC1C)=O 64886,C1(CNC(C(CCC)OCC)=O)CC2(CCN(C(=O)CC3CCC(C)C3)C2)CO1 64887,c1(C(C)(CO)NC(=O)NCC(c2ccccc2Cl)(C)C)cccc(Cl)c1 64888,N1(C(C2(OC)CCOC2)=O)C(C(=O)NCC2(O)CC3CCC2C3)C2CC(O)C1C2 64889,C1(C)(C(=O)NC2CC(CC(N3CC(c4nc(C)[nH]n4)C3)=O)C2)CCC(C)C1 64890,Cc1cnc(C(=O)NC(CNC(c2cnc(=N)[nH]c2)=O)CO)c(F)c1 64891,c1(CNC(C(=O)N(CC(N)=O)C)=O)nc2ccc([N+](=O)[O-])cc2[nH]1 64892,N1(C(CN(C)CCO)=O)CCC(CNC(=O)COc2ccc(Br)cc2)C1(C)C 64893,c1(CNC2CCC(C(=O)NC(C3CCCCO3)C)C2)cc(C#N)ccn1 64894,c1(C(=O)OC)ccc2c(n1)CCCN2C(c1ccc(-c2cnnn2C)cc1)=O 64895,c1(C(=O)NCC2COC(CNC(=O)C(F)n3ccnc3)C2)ccnc2[nH]ncc12 64896,N1(C(c2cn(CC)nc2)=O)CCCOC(CCNC(C2CCCSC2)=O)C1 64897,N1(C(C(C)S(N)(=O)=O)=O)CC2(CCC(CNC(c3ccncc3C3CC3)=O)O2)C1 64898,c1(OC)c(Br)ccc(F)c1C(=O)NCC(CNC(=O)C(C)(C)C)CO 64899,N1(C(c2ccc(C(C)=O)cn2)=O)CCC2(NC(=O)CC3CC3(C)C)CCCC12 64900,C(=O)(C(CO)C(C)(C)C)N1CCN(CCN(C(CNS(CC)(=O)=O)=O)C)CC1 64901,O=C(C#CC1CCOC1)NCC1CC2CCC1N(C(=O)CC1CCOC1)C2 64902,c1(NC(c2n(C(CC)(C)C)nnn2)(C)C(C)OC)ccc2nncn2c1 64903,C(=O)(C#CC1CCCOC1)NC1CC(CNC(C2(SC)CC2)=O)OCC1 64904,c1(COC)cc(C(N2CC3C(NC(C4CCCSC4)=O)C3C2)=O)c(C)o1 64905,CC(CC(=O)NCC1(C(N2CCOC(C#N)C2)=O)CCCO1)C(F)F 64906,C(C)(CO)(CC(C)C)NC(c1c(CCNC(c2c(C)cccc2)=O)n[nH]c1)=O 64907,c1(NC2CC(OCC)C2)nccc(=NC(CC)CC#N)[nH]1 64908,C#CC1CN(C(=O)C(C)C(CC)CC)CCN1C(=O)CCCOC(C)=O 64909,c1(C(N2CC(O)(CNC(C(C)SCc3ccccc3)=O)C2)=O)nc(=O)n(C)[nH]1 64910,c1(C(=O)NC2C(NC(C3(C)CCN(C(C)=O)C3)=O)C2)ccc2cc(C#N)ccc2c1 64911,CC(C(=O)N1CC(NC(=O)CC2CCCCCC2)C2(CC2)C1)C(C)(F)F 64912,c1(C(C(=O)NC)N(C)CC2(CC)CCC2)cccc(N2CCOC2=O)c1 64913,S(=O)(=O)(c1cccnc1NC(CCO)CC(C)C)NCC1(OC)CC=CCC1 64914,N1(C(CC2CNC(=O)O2)=O)CC2(CCC2)CC1CNC(=O)Cc1cc[nH]n1 64915,CC(C)CCCC(=O)N1CCC(O)(CCNC(C2(O)CC2)=O)CC1 64916,c1(C(=O)NCC2(O)CN(C(C3C4C5CCC(C5)C34)=O)C2)cccc2c1CCCN2 64917,C#CCCCC(C)C(=O)NC1CN(C(c2ccc(F)o2)=O)C1 64918,c1(C(N(CCCNC(=O)CC(O)C2CCCC2)CC)=O)ncccc1OC(F)F 64919,c1(N(C)C)ccnc(C(C2CCN(C3CCC3)C2=O)c2nnnn2C2CCC2)c1 64920,CC1(C)CC(CNC(=O)CN2C(=O)CNC2=O)CN1C(C1CC2(CCC2)C1)=O 64921,N1(C(C(CC)CC(F)F)=O)CC2(CCN(C(c3cccc(OC)c3)C)CC2)C1 64922,c1(OC)cc(OC)c(CNC(=O)NCC(c2ccccc2OC)(C)C)cc1Cl 64923,c1(C(=O)NC2CCN(C(CC(C)F)=O)C23CC3)nccc2ccsc12 64924,C#CCC(CC(=O)N1CCC(C)=C(C)C1)NC(C1(F)CC=CCC1)=O 64925,C1(CCNC(CCN(CC)CC)=O)CCCN1C(=O)CSC 64926,C=CCCC(C(=O)NCC(O)CC(C)C)NC(c1cccnc1O)=O 64927,C1(F)(C(=O)NCC(C)(C)CNC(C2(c3ccccc3F)CCC2)=O)CCCOC1 64928,c1(C(=O)NC(CC=C)CNC(=O)Cc2cncn2C)cccnc1C(F)F 64929,N=c1[nH]c2cc(C(=O)NCC3C4CN(C(=O)CCc5cc[nH]n5)CC34)ccc2o1 64930,c1(OCCC(=O)NCC(C)NC(c2sc(F)cc2Cl)=O)c(F)cccc1Cl 64931,c1(C(=O)NC(CC)CNC(c2nncn2C2CC2)=O)csc2c1CCC(C)C2 64932,C(C1=CCCCC1)(c1nnnn1C1CCC1)NC(c1n(C)cnc1)CO 64933,c1(OCC(=O)NC2CC(C)(NC(c3ccn(C(C)(C)C)n3)=O)C2)cccc(F)c1 64934,CC1(NC(c2ccc(C3CC3)s2)=O)CCN(C(C2(C)CCOC2)=O)C1 64935,C1(C(N(CC(F)(F)F)CC)=O)CC(F)CN(Cc2c(OC)cccc2O)C1 64936,Cc1n[nH]c(C)c1CCCNC(=O)NC(c1ccc(F)cc1)C1CCOC1 64937,c1(N(C2CN(C(=O)CCc3ccc(F)cc3)C2)C)ccc(Br)cc1[N+](=O)[O-] 64938,C1(C(=O)NC2C(C3C(C)C3)C2)CCN(C(=O)C2(O)CCCCCC2)O1 64939,c1(C(=O)NC2(C)CCN(C(C3CCN(CCC)CC3)=O)C2)cc(Cl)c(F)cc1Cl 64940,CC1CCN(C(c2cc(C(C)(C)C)on2)=O)CC1N(C(=O)CCC1OCCO1)C 64941,C(CNC(c1cc(OC)cc(C)n1)=O)(CC(F)(F)F)NC(C(COC)O)=O 64942,c1(CC(=O)NC2C(CNC(Cn3c(C)ncc3)=O)CC2)nc2c([nH]1)CCCC2 64943,C1(CC)C(CC(=O)NCCC(Cc2ccccc2)NC(=O)CNS(N)(=O)=O)C1(F)F 64944,C1(C2CCCN(C(=O)C(C)C#N)C2)(NC(c2ccn(C(C)C)c(=O)c2)=O)CC1 64945,C(CN1C(=O)Cc2ccccc21)NC(c1cn(C)nn1)c1nnnn1C(C)(C)C 64946,C1(NC(C2CC(=O)N2)=O)CN(C(c2cnn(-c3ccc(F)cc3)c2)=O)CC1F 64947,Cc1oc(C)c(C(=O)NC(C)CC2CCN(C(=O)Cc3nnc(O)s3)CC2)c1C 64948,c1(N2CCC(N(C(c3scc(C)c3C)=O)C)C2)ncnc2c1cnn2C 64949,C1(CNC(c2c(CC)nc(C)[nH]2)=O)CC2(C1)CN(C(=O)Cn1nc(C)cc1C)C2 64950,C=CCN=C(NCC1(CO)COCCN1C)N1CCC(C)(C)C2(CCOC2)C1 64951,N1(C(C=CCOC)=O)CCC(C2OCCC2NC(=O)Cn2ccnc2C)CC1 64952,CCC(C(O)C(C)C)NC(=O)NCC(c1ccc(Br)cc1)(C)C 64953,C1(O)(CN(C(CSCCCC)=O)C)CCN(C(=O)Cc2ccc(C(=O)OC)cc2)C1 64954,C#CCC(CC(=O)NC1CCCC(CO)C1)NC(=O)C(F)(F)CC 64955,C=CCCCC(=O)N1CC2C(NC(c3c[nH]cc3C(C)(C)C)=O)C2C1 64956,N1(C(C(CC)n2cncn2)=O)CCCCC1CCCNC(c1c[nH]c(C#N)c1)=O 64957,C1(OC)CCC12CC(C(N1CCC(C(C)NC(=O)C3=COCCC3)CC1)=O)C2 64958,CN1CC(C(=O)NCC2(C(=O)NCC3CCC(CN(C)C)O3)CCC2)CC1=O 64959,c1(C(N2CCN(C(C(CC)=CC)=O)C(CCOC)C2)=O)nn(C)cc1S(C)(=O)=O 64960,CCC(C)C(C(=O)NCC1=CCN(C(c2ccc(NC)cc2Cl)=O)CC1)OC 64961,C1(NC(C2(OC)CCN(C(C3CN4CCC3CC4)=O)C2)=O)CN(C)CC1(F)F 64962,c1(C(=O)NCC)cccc(C(N2CC(NC(=O)CC3COCCO3)C(F)C2)=O)c1 64963,c1(OC)ccc(NCc2ccc(CSc3ccccc3)o2)cc1C 64964,N1(C(C2(OC)CCCC2)=O)CCOC(CCNC(C23CCCC2(C(N)=O)C3)=O)C1 64965,c1(CCC(=O)OC(C(=O)Nc2c(C)ncc(C)n2)(C)C)cc(C)ccc1[N+](=O)[O-] 64966,c1(C(=O)NCCCN(C(c2c(C)nn(C)c2C)=O)CC)sccc1S(N)(=O)=O 64967,N1(C(CCSC)=O)CCCC(C)(CNC(=O)COc2ccccc2C(C)(C)C)C1 64968,n1(CC(=O)NCC(COC)NC(=O)Cc2cn(C)nc2C)cccc(C)c1=O 64969,C=CCC(CC)C(=O)NCCC1CC(NC(=O)Cc2cccc(NC(N)=O)c2)C1 64970,C(=O)(CCC(C)NC(C1(C#N)CC=CC1)=O)NCC(CSC)OC 64971,C1(c2ccc(F)cc2)(C(=O)NC(CC)CNC(=O)C(C2CC2)SC)CCOCC1 64972,CCC1c2cc(Cl)cc(Cl)c2CCN1Cc1cnc(-c2ccccc2)o1 64973,C(CNC(=O)CCc1nc[nH]n1)(C(=O)N(C)C(C1(C)CC1)C)OC 64974,CC1(CNC(c2cc(CC3CC3)on2)=O)CCN(C(=O)CNC2CCCC2)C1 64975,C(C(C(=O)N(C1CC1C1CC1)C)NC(=O)Cn1cc(C)cn1)OCC 64976,c1(CCC(=O)NC2C(C)(CC)C2)nc(C(C)OC)no1 64977,C1(CC)(CO)CCN(C(C2(C)CCCN2C(c2nccnc2N)=O)=O)CC1 64978,CC1Cc2ccccc2N1CCNC(=O)NC1(C(=O)O)CC(C2CCC2)C1 64979,CC(C)C(O)CC(=O)N1CCN(C(=O)CC2OCCC2(C)C)C(C)C1 64980,c1(CNC(CN(C(C)=O)C)=O)cnn(C)c1C(=O)NCCC1CCCC(C)C1 64981,N1(C(c2c(C)nc(O)cc2)=O)CCCCCCC1C(=O)NC1C2CCCC1CC2 64982,C1(NC(c2cc(C(C)C)no2)=O)CCCCCN(C(=O)C(=Cc2c[nH]cn2)F)C1 64983,c1(C(N2C(CC)C(C(=O)NCc3ncnn3C)CC2)=O)ccc(C#N)cc1 64984,c1(CN2CCC(F)(C(=O)Nc3cc(C)c(I)cn3)C2)cccc2cccc(C)c12 64985,C1(NC(COCC#C)=O)CC2(C1)CN(C(c1csc(C3CC3)n1)=O)C2 64986,S(=O)(=O)(c1c(F)cccc1F)NC1C(C(=O)Nc2cncc([N+](=O)[O-])c2)C1 64987,CS(=O)(=O)c1ccc(S(=O)(=O)NCCNC(=O)Nc2ccc(Cl)c(Cl)c2)cc1 64988,c1(C(=O)NCC2CCCCC2)ccc(NC2=NCCC2)cc1 64989,c1(CC)cnc(C(c2nnnn2C(C)(C)CC)NCc2nc(CC)cs2)[nH]1 64990,C=CCC(CC(=O)Nc1cnc(C2CC2)nc1)NC(C1CC(CC)=NO1)=O 64991,c1(C(=O)NC(C(CO)NC(C(CCCOC)C)=O)C)nnc(O)c2ccccc12 64992,C(=O)(CC(C)P(C)(C)=O)N1CCCC(CCNC(c2cc(C)cc(N)c2)=O)C1 64993,Cn1c(C(=O)NCC2CC(NC(=O)CC3CCCC(=O)C3)C2)cnc1O 64994,C1(CN(C)C)CC(O)CN1C(c1n[nH]cc1CNC(=O)CC1CC(=O)C1)=O 64995,n1(CCC)ncc(C(N2CCCCC2CCNC(C2CCS(=O)CC2)=O)=O)c1Cl 64996,C1(CNC(CC(C=C)CC)=O)CC2(CCN(C(=O)C(C)C(C)CC)CC2)CO1 64997,COn1cnc(C)c1C(=O)NCC1CCC1NC(c1cc(F)ccc1C1CC1)=O 64998,c1(C(=O)NC2C(NC(CCN(C3CC3)CC)=O)C2)cc(S(C)(=O)=O)oc1C 64999,C#Cc1cccc(C(=O)NC(CNC(=O)C(CC)N(C)C)C(C)C)c1 65000,N1(C(Cc2c(CC)con2)=O)CC(NC(C2CCO2)=O)C(O)C1 65001,c1(CN2CC3C(C(N4CCC(=C)CC4)=O)(C3)C2)c(C)cccc1C 65002,c1(CCOC(N2CCCC(ON(C3(CCO)CCC3)C)C2)=O)cc(Cl)ncc1O 65003,c1(C(N2C(CNC(C(c3cc(C)sc3)(F)F)=O)CC2)=O)cc(Cl)c2n[nH]cc2c1 65004,CCC(C)CC(=O)N(C1CC(NC(=O)Cc2sc(C)nc2C)C1)C 65005,C(=O)(CC1CCc2ccc(O)cc21)NCC(C)NC(c1cccc2cncn12)=O 65006,n1(CC)nc(C)cc1C(=O)NCC1CN(C(=O)C(C(C)C)NC=O)CC1O 65007,N1(C(Cc2c(C)cnn2C)=O)CCC2CC2(C(=O)NCC2(O)CC=CC2)CC1 65008,Cc1[nH][nH]c(=N)c1C(N1CCC(CNC(c2cnc(Cl)[nH]2)=O)C1)=O 65009,N1(C(C2(C#C)CN(C(C3CCC(F)(F)C3)=O)C2)=O)CCN(C)CC1C 65010,C1(C(=O)NCC2(O)CCCN(C(=O)C(C)CF)C2)(CC)CCC(O)CC1 65011,C1(CN(C(=O)CC(O)c2ccccc2)CC)CCCCN1C(c1cnc[nH]1)=O 65012,c1(C(N2C(CN(C(c3ccc(C(C)C)s3)=O)C)CCC2)=O)occ2c1CCOC2 65013,CCC(C(=O)NC(CC1CCCC1)C(=O)NCCCCCSC)N(CC)CC 65014,c1(OC)cc(N(CCNC(c2nn(C)c(Cl)c2Cl)=O)C2CC2)c(Cl)cc1[N+](=O)[O-] 65015,C(=O)(CC(C)NC(c1cn(C)nn1)=O)NC(CC#C)C 65016,Cc1cc(C(N2CCCC(NC(=O)Cc3ccsn3)C2C)=O)c(C)n1CC1CC1 65017,n1(CC)nc(C(=O)NC2CN(C(=O)COC(C)=O)CC2C)cc1C(F)(F)F 65018,c1(C(N(CCCN(C(C(C)OCC(C)C)=O)C)C)=O)ccc(CNC(N)=O)cc1 65019,C(=O)(C#CC(=O)N(C)C)N1CCC(C(C)NC(=O)C(C)n2ccnn2)C1 65020,C(=O)(C(C)C(F)(F)C(F)F)N1CCN(C(CC2CCC(C)CO2)=O)CC1CO 65021,C1(C(=O)NCC2CC(NC(C3CCS3(=O)=O)=O)C2)CCC([N+](=O)[O-])CC1 65022,c1(NC(C2CCC(C)(C(C)=O)C2(C)C)=O)cccc2c1COC(=O)N2 65023,c1(C(=O)NCC2N(C(C(CC=C)C)=O)C3CCC2C3)cccn2c(C)nnc12 65024,N1(C(C(CC)CN(C)C)=O)CC2(C)CC1(C(=O)NOCc1cncs1)C2 65025,N1(C(C(CCC)C)=O)CCN(C(=O)CSCC(C)C)CC1C 65026,N1(C(C(COC)OC)=O)CCN(C2CN(C(C3COCCN3C)=O)C2)CC1 65027,C1(C(C)(C)O)(CNC(=O)C=CC2CCC2)CN(C(=O)CC2C=CCC2)C1 65028,N1(C(=O)C=CC2CCOC2)CCN(C(C2CC(n3cnnc3)C2)=O)C(CO)C1 65029,c1(N(C)C)ccc(C(=O)NC2(C(F)F)CC(NC(=O)COC3CC=CC3)C2)cc1 65030,c1(COCC(N2C(CNC(COCCN(C)C)=O)CCC2)=O)ncccc1F 65031,N1(C(CCCN(CCC)CCC)=O)CCC2(CCCN2C(=O)C(C)SCC)C1 65032,Cc1cc(C(c2nnnn2-c2ccc(F)cc2)NC2(CCF)CC2)c(C)cc1Br 65033,Cn1cncc(C(=O)NC2CC(C)(CNC(=O)C(c3ccc(Cl)cc3)O)C2)c1=O 65034,CC1(C(=O)NCC2(F)CCN(C(c3ccc(CO)nc3)=O)C2)CCCCCC1 65035,C1(C)(C(=O)NCC2(OCC)CCC2)CC(OC)CN1C(=O)CCC(C)C 65036,Cc1cc(C(=O)NC2CCC2NC(=O)CCCCCN(C)C)c(C)n1CC1CC1 65037,C1(C(C(=O)N(c2cccs2)CC2(O)CCCOC2)F)CCN(c2ncccn2)CC1 65038,C1COC(C)(C)C1.CCC(C(=O)NC(CC(N)=O)c1cn(CC2CC2)nn1)N(C)C 65039,c1(C(=O)NCCC2CCC(NC(=O)Cc3cccs3)C2)cc(F)c2[nH]nnc2c1 65040,c1(C(C(=O)NCCSC)N(CC(F)F)C(C)C)ccc(C)c(F)c1F 65041,C1(C(N(CC(C)NC(C2(CC)CCC2)=O)C)=O)CCCN(c2ccnc(Cl)n2)C1 65042,C(C(F)(F)C(=O)NCCN(C(c1cc(-c2cccnc2)on1)=O)C1CC1)OC 65043,C(CN=c1[nH]c2ccc(F)cc2o1)NC(C1CCN(C(C(C(C)O)C)=O)CC1)=O 65044,C1(NC(C2C3CN(C(C(C)=C4CCCC4)=O)CC32)=O)CCCOC12CCC2 65045,c1(C(N2C(C)CCC(CNC(=O)Cc3cccs3)C2)=O)cncc2c1CCC2 65046,N1(C(C(C)=CC2CC2)=O)CCCC(CO)(NC(c2cncc(Cl)c2)=O)C1 65047,C#CC1CN(C(=O)CC2(N(C(=O)CC34CCC(CC3)C4)C)CC2)CCO1 65048,c1(C(=O)NC2(CF)CCN(C(C(C=C)O)=O)C2)cccc2c1COC2 65049,C1(NC(C2C(c3ccc(C)c(Br)c3)C2)=O)CC2(CCC(NC(C)C)CC2)C1 65050,C(CCC(C)(C)C(=O)N1CC(O)C(O)CO1)NC(c1c(NC)cnnc1)=O 65051,Cn1[nH]nnc1=NCC1(CNC(=O)CCn2cnnn2)CCC1 65052,N1(C(c2cnc3ncccn23)C(=O)NCCCC)CCC2(COC(C)C2)C1 65053,c1(CN2CCN(CCOC)CC2)ccc(-c2ccc(Cl)s2)cc1F 65054,c1(OC)cc(C(N2CC(O)(C3(CNC(=O)CCOC)CC3)C2)=O)c2c(c1)CCO2 65055,C1(C(=O)NCC(CCC)OC)CC=CCN1C(=O)CCc1nncs1 65056,N1(C(c2c(OC)cc(C)cc2)=O)CC2CC1CN(C(=O)CCC1(C)CC1)C2 65057,CCC(C(=O)NCC1CCN(C(C2CCN(CC)C2)=O)C1)n1cncn1 65058,c1(C(=O)NC(CSCC=C)=O)ccc(C2COCCN2C(c2ccsc2Cl)=O)n1C 65059,C1(C(N2CC(CC=C)(NC(=O)C(C)OCC3CC3)C2)=O)CCOC(C)C1 65060,CN1CCOC(C(=O)NC2CN(C(c3cc(-c4ccccc4)ns3)=O)CC2O)C1 65061,N1(C(c2cccc(SC)c2Cl)=O)CCN(C(=O)C(=O)C(C)(C)C)CC(O)C1 65062,C1(CN(C)C)CN(C(=O)C(=O)NC2CCN(CCS(N)(=O)=O)CC2)CC1O 65063,c1(CC)occc1C(=O)NC(CNC(c1cnc(C)s1)=O)CCOC 65064,C1(CNC(C=CCN(C)CC)=O)CCC2CN(C(c3ccc(CO)s3)=O)CC12 65065,N1(C(C2C(C)C2C)=O)CCC(N(C)C(C2C3CCC2CC3)=O)CC1 65066,C(=O)(CC(O)Cc1ccccc1)N1CC(NC(C2CSC2)=O)C1 65067,n1(CC(=O)NC2C(C)NCC2)nc2n(c1=O)CCCCC2 65068,c1(C(=O)NC(CN(C(=O)C(C(C)C)OC)CC)C)cc2cc(Cl)ccc2n1C 65069,c1(NC(C2CCCN(C(C3COC(C)(C)C3)=O)C2)C)ncc(I)cn1 65070,c1(CC)cccc(C(N2CC(F)CC2CN(C)C(c2ccc(F)s2)=O)=O)c1O 65071,c1(C(=O)NC2C(NC(C3(SC)CC3)=O)CCOC2)cc2cccc(Cl)c2nc1C 65072,c1(OC(C)C(N2CCCCC2CCNC(=O)CP(C)(C)=O)=O)cccc(F)c1 65073,C1(CNC(CC2N(C)C(=O)CC2)=O)CN(C(c2cc[nH]n2)=O)CCC1(F)F 65074,c1(-c2nc(C3C(C)(C)CN3)on2)cc(Cl)cn2ccnc12 65075,c1(C(=O)OCC)cc(C)sc1NCc1cn(-c2ccccc2OC)cn1 65076,C1(CNC(c2c(C)cn(C)c2)=O)CN(C(c2ocnc2C2CC2)=O)CC(C)(C)C1 65077,C(CCC(C)C(=O)N1CC=CC(NC(c2cc(Cl)n[nH]2)=O)C1)OC 65078,C1(C(N(CCCN(C(=O)CCn2cnnn2)C)C)=O)CCCNC1=O 65079,C1(NC(C(C)OC)=O)C2CN(C(=O)CCC(=O)N(C)C)CC12 65080,c1(C(=O)NCC2CN(C(C(CC(C)C)OC)=O)CC2(F)F)scc2c1OCCO2 65081,c1(C(N2CC(C)N(C(=O)C=CC3CCOC3)CC2)=O)cc(Cl)c(F)c(Cl)c1 65082,CC1N(N2CCOC(c3noc(-c4ccccc4)n3)C2)C2CCCC12 65083,C12(NC(C(C)=CC)=O)CN(C(=O)C(C3CCCCC3)O)C(COC)(C1)C2 65084,C1(N(C(C2CCN(C(Cc3c(CC)con3)=O)C2)=O)C)CCCC1C#N 65085,N1(C(c2[nH]cc(C#N)c2)=O)CC2CCC1C(Nc1ncnc(Cl)c1Br)C2 65086,N1(C(C2C(NC(C(C)(C)n3cnnn3)=O)CCCC2)=O)CCC(C2CCC2)C1 65087,c1(C(=O)NC(C(=O)NCCc2cnc(C)[nH]2)Cc2ccoc2)cnc(Cl)n1C 65088,Cc1nnc(C(=O)N(C(C)CCNC(C2CC2(F)F)=O)C)s1 65089,C1(CNC(CC2(N(C)C)CCCC2)=O)CCCCCN1C(=O)CCc1ccoc1 65090,Cc1ccc(C(N2CCC3CC23)=O)c(-n2cc(CN3C(=O)CCC3=O)nn2)c1 65091,N1(C(c2c(OC)ncc(F)c2)=O)CC2CCC1CN2C(C1COC(C)C1)=O 65092,N1(C(CCC)=O)CC2(NC(c3ccc(F)cc3CC)=O)CCC1C2 65093,Cc1ccc2c(=NCC(C)Cc3cn[nH]c3)[nH]c(=NCC3CCC3)[nH]c2c1 65094,c1(OCCC(=O)N(C)CC2CCCN2C(C2CNC(=O)C2)=O)ccc(F)cc1F 65095,C=CC1(NC(=O)C(CC2OCCO2)NC(=O)OC(C)(C)C)CCC1 65096,c1(C(N2CC(F)CC(NC(C(CC)C(C)C)=O)C2)=O)cccc2c(C)c(C)[nH]c12 65097,c1(C(=O)NCC2(COC)CCCN2C(=O)C(C)C(C)(C)C)cn2c(n1)CCC2 65098,N1(C(C(C2CC2)OCC)=O)CC(C)C(C)(CNC(c2ccc(N)c(O)c2)=O)C1 65099,c1(-c2cn(CC3N(CC(=O)Nc4ccc(Cl)nn4)CCC3)nn2)sc(O)nc1O 65100,C(=O)(C1CCc2nccn21)NCC1(C)CCN(C(c2cc(OC)c(Cl)cc2)=O)C1 65101,C1(NC(c2cc(C)nn2C(C)(C)C)=O)CC2CN(C(c3cnc(Cl)n3C)=O)CC12 65102,C1(CN(C)C)CC(C(=O)NC2CC(CNC(C3CN(S(C)(=O)=O)C3)=O)C2)C1 65103,c1(C(=O)OC)cccc(C(C(=O)NCCC#N)N(C)Cc2ncccc2Br)n1 65104,c1(CNc2c(CCC(=O)OC(C)(C)C)cccc2)c(Cl)cc(Br)cc1Cl 65105,C1(CCOC)CCCCN1C(C1CCN(C(c2cc(C)no2)=O)C1)=O 65106,c1(C(=O)NC2CC(CNC(C(C)SC(C)C)=O)CC2O)cc(F)c(N)cc1F 65107,N1(CC(=O)NC2(CO)CN(C(CC3CCC(C)C3)=O)C2)CCCNS1(=O)=O 65108,C(CC(C)(C)CO)NC(C1CC(C)N1C(C1CCCC(=O)N1)=O)=O 65109,CN(C[Si](C)(C)C)C(=O)CC1CCCCN1C(=O)CCc1cnco1 65110,C(=O)(C1Cc2c(Cl)cccc21)N(CCCCNC(CCC(=O)NC)=O)C 65111,c1(OC)ccc(C)nc1C(=O)NC1CCCC(NC(C2CC3(C2)CC(O)C3)=O)C1 65112,CC1CCCCC1OCC(=O)NCC1CC(NC(C2CC2(Cl)Cl)=O)C1 65113,Cc1cc([N+](=O)[O-])cnc1N1CC(CNC(C2(Cl)CC2)=O)OC2(CCC2)C1 65114,C1(NC(C2C(C)CC(C)O2)=O)CN(C(=O)OC(C)(C)C)CC12CCOCC2 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65150,Cn1nc(C(F)(F)F)cc1NC(C1CCC(NC(c2cnc(Cl)cn2)=O)C1)=O 65151,N1(C(c2c(OC)scc2)=O)CCN(C(=O)C(F)CC(C)C)CC(C)(C)C1 65152,c1(C(=O)NC2C3C(C)N(C(C4CCCCN4C)=O)C2C3)ccc2nc[nH]c2c1 65153,C1(C(=O)NC2CCN(CC(=O)NC(COC)C(C)C)CC2)CC2(C1)CC2(F)F 65154,c1(OC)cc(C(C(=O)NCc2cccc(Cl)c2)N(CCCN(C)C)C)c(Cl)cn1 65155,C12(NC(Cc3cnc(C)s3)=O)CCCC1N(C(=O)CCCOC(C)(C)C)CCC2 65156,N1(C(=O)CCCC(F)(F)F)CC2C3CCC(C2C1)N(C(C1CCCO1)=O)C3 65157,c1(C(N(C2CCC(NC(CCNC(CC(C)C)=O)=O)C2)C)=O)nnc(O)nc1O 65158,c1(OCCC)ccc(Cl)cc1C(=O)NC1CN(C(=O)C(C)(O)CC)CC1O 65159,C1(C(=O)NCCC2N(C(c3c(N)nccn3)=O)CCC2)CC12CCS(=O)(=O)CC2 65160,C(C)(c1ccco1)=CC(=O)NCC1N(C(C2C(COC)CC2)=O)CC1 65161,c1(C(N2CCN(C(CC=CC)=O)C(CF)C2)=O)nnc2ccccc2n1 65162,N1(C(C2C(C=C)OCC2)=O)CC2(CC2)CC1C(=O)NCC1CC2CCC2C1 65163,N1(C(CSS(C)(=O)=O)=O)CC2(CCCC(CNC(C3CCS3(=O)=O)=O)O2)C1 65164,C1(=O)C(C)(CO)N1.C(C(=O)N(C(COC)C)CC)=CCC 65165,C(=O)(CCC(=O)NCc1nc(C)c(C(=O)N(CCC(O)CO)C)o1)NCCC 65166,C1(C(=O)NCCC2(C)CCCO2)CCC(CNC(c2ccc[nH]2)=O)CC1 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65290,C(=O)(C(F)(F)CCNC(C)=O)Nc1c(-n2cc(CC(CC)(C)O)nn2)cccc1 65291,C12(CNC(c3ccnnc3O)=O)CCCC(CN1C(C1Cc3nncn3C1)=O)C2 65292,c1(C(=O)NC2CC(C(C)(C)C)C2)csc([N+](=O)[O-])c1.C123COC(C1)(C2)C(=O)NC3 65293,C(=O)(C(CC(C)C)C(C)C)NC12CN(C(c3cc(C)ncc3C)=O)C(CC1)C2 65294,Cc1c(C(=O)NC2CN(C(C3CC3F)=O)CCC2O)oc(=O)c2ccccc12 65295,c1(N(C)C)cccc(NC(C2CN(C(=O)CSCc3cccs3)CCO2)=O)c1 65296,C1(CC(=O)N(CCCCCC)CCNC(=O)CCC)CC(OC(C)=O)C1(C)C 65297,c1(C(=O)NC2CN(C(C(CCSC)O)=O)CC2O)cc2c(cc1F)OCC(=O)N2 65298,C12CCCCC1OC2.c1(CCc2ccon2)cn(C2CCSCC2)nn1 65299,c1(N2CCC(c3cccc(C)c3)C2)nc2ccccc2nc1NCCC(C)C(F)F 65300,C(=O)(C1=CCC(C)(C)CC1)NCCC(C(=O)NC1CCOCC1C)OC 65301,C12(C(N(C(C)CNC(C3COC(C)(C)C3)=O)C)=O)CCC(C(F)(F)F)(CC1)CC2 65302,C=CC(C)(CC)C(=O)NCc1cc(C)c(C(=O)N(CC(O)CO)C(C)C)o1 65303,CCC(CNC(=O)CC1CCCC1O)(CC)C(=O)N1CC(N2CC(O)C2)C1 65304,CCC(CC(=O)NC1(CO)CCCN(C(C)=O)C1)CC(F)(F)F 65305,N1(C(CSCC(N)=O)=O)CC2CC2(CNC(c2csnc2Br)=O)C1 65306,c1(NC(C2(CNc3cc(CC)ncn3)CC2)=O)ccc(Br)c2ncccc12 65307,N(C(=NCCC(C)=O)NCC1CCCC1CCC)Cc1n(CC)ncn1 65308,C(=O)(C1=C(C#N)CCC1)NC1C(N(C(CC(C=C)CC)=O)C)CCCC1 65309,C(C(C)(C)CCNC(=O)CC1COCCO1)NC(C(C1CC1)OCC)=O 65310,N1(C(C(C(=C)C)(C)C)=O)CC(CO)C2(C1)CN(C(c1cc(C)c(N)cc1F)=O)C2 65311,c1(C(N2CC(CNC(c3oc(C)c(CO)c3)=O)C2)=O)cc(O)ccc1Br 65312,CCCCCCCCCC(O)C(=O)N(CC(C)CNC(c1nccnc1C)=O)C 65313,C12(C(=O)NCc3nc(C)c(C(=O)NCC4CC(F)C4)o3)CCCC1C2(F)F 65314,C1(NC(c2cn(CCC)nc2)=O)CCN(C(=O)CCCCC(N)=O)CCC1(F)F 65315,CC(C)CC(C)CNC(=O)C(O)CNC(=O)CSC(F)(F)F 65316,N1(C(CCCC#C)=O)CC(CCNC(c2cnc(OCC)c(Cl)c2)=O)OC(C)C1 65317,N1(C(CCCSC)=O)CCC2(C1)CN(C(C1(F)CCCOC1)=O)CCO2 65318,c1(CC)cccc(CC)c1C(N1CC(F)(F)CC1C(=O)Nc1cnc[nH]1)=O 65319,C1(NC(CCC=C(C)C)=O)CC(C)N(C(=O)CSc2nncs2)C1 65320,CS(=O)c1ccccc1C(N1CC2(C1)CN(C(c1cnc(F)c(Cl)c1)=O)C2)=O 65321,C1(C(=O)NCCC2CCCN(c3ccnc(C)n3)C2)CCCC(C)(C)C1 65322,Cn1cnc(C(O)CNC(c2occc2CNC(=O)Cn2cnnn2)=O)c1 65323,c1(C(=O)NC(C)CN(C)C(C2CCCN2c2cnccn2)=O)ccc(Cl)cc1O 65324,CCCS(=O)(=O)C(C)C(=O)NC1CCCC1NC(c1cnc2n1CCCC2)=O 65325,C1(C(=O)NC(CNC(=O)Cc2sccc2Cl)C2CC2)CC=CC(O)C1 65326,C1(NC(=O)CCCNc2cccc(C(=O)O)c2)CCC2(CCCC2)C1 65327,C(C1=CCN(C(=O)C(C)S(C)(=O)=O)CC1)NC(CCCc1scc(C)n1)=O 65328,N1(C(Cc2n(C)ncc2)=O)CC(=O)NCC1C(=O)NCCOCCN=[N+]=[N-] 65329,C1(OC)CCOCC1NC(=O)CN(C(=O)CCC1CC1C)CC1CCC1 65330,C1(CNC(CCC)=O)C2CC1N(C(=O)CCc1ccccn1)C2 65331,C1(CC)C(C)CCN1C(=O)CN(C(c1ccnn1COC)=O)CCF 65332,C1(CNC(C2CC(OC)C2)=O)N(C(c2ccc(Cl)cc2Cl)=O)CCCC1(C)C 65333,c1(C(N(CC(C)O)CCNC(CN2C(C)CCC2)=O)=O)cc(C(F)F)ncn1 65334,C1(NC(C(C)NC(COC)=O)=O)CN(C(C2CC(C)(C)C2)=O)CCC1C(F)(F)F 65335,CC(O)C(C(=O)NCC12CC(NC(=O)COCC3CC3)(CO1)C2)N(C)C 65336,C#CCC(C)(CC)C(=O)NCC(C(=O)N(C)Cc1nc(C)ns1)C(C)C 65337,N1(C(C(C)Oc2cc(C)c(C(C)C)cc2)=O)CC(C)C(O)(C(F)(F)F)C1C 65338,CCC(F)(F)C(C)(C)C(=O)N(C(=O)Cc1ccc2ncccc2c1)CCN(C)C 65339,C(C)(C(=O)N1CCC1CNC(=O)C(C)=CC1CC1)NC(=O)NC 65340,C1(CNC(C(C2CCOC2)OC)=O)CCCC2(CN(C(C)C)C2)O1 65341,c1(C(=O)NC2CN(C(C3CCC3(F)F)=O)CC2CC2CC2)ccc(F)cc1F 65342,C1(NC(C2C(C=C)OCC2)=O)CCN(C(=O)CCC2CC(C)C2)CC1O 65343,C1(C(=O)OC)CN(C(=O)Cc2cnc(Cl)cc2C)CCC1CN 65344,CC(C)(CC(=O)N1CC=CC(NC(c2cccc(-n3cccn3)n2)=O)C1)C1CC1 65345,c1(C(=O)NCC2CCN(C(C(C(C)C)OCC)=O)C2)cccc2nc[nH]c12 65346,C(C)C(C)CC(C)C.C=CCCC(CC)N(C)C 65347,c1(NC(c2cnn(C)c2Br)c2n(C(CC)C)nnn2)cc(Br)c(O)nc1C 65348,N1(C(c2cc(CNC(CCC(C)C)=O)[nH]n2)=O)CCC(O)C12CCC2 65349,c1(CC(C(C)C)NC(=O)NCC2CC(F)CN2)ccccc1C(F)(F)F 65350,C(=O)(C1=COCCO1)NCCOC1(CNC(C(CC)F)=O)CCOCC1 65351,C1(Nc2nccc(N3CC(SC)OCC3)n2)Cc2ccccc2C1OC 65352,c1(OCC(C)C)cc(C(=O)NC2CCC2CNC(=O)C(C2CC2)N(C)C)ccn1 65353,C1(C)(CNC(C(C)N2CCC2)=O)CC(F)(F)CN1C(=O)C=Cc1ccc(F)nc1 65354,C1(O)(C(=O)NCCC2CCC(NC(C=CCCC)=O)C2)CCOCC1 65355,Cc1cc(NC(=O)CN(C)C2CC2)ccc1NC(=O)CCN1CCCC(C)C1 65356,C(=O)(CC(O)CNC(C1CS(=O)C1)=O)NC(c1scc(C)n1)C 65357,c1(C(C)(C)NC(C)=O)ccccc1OC(=O)Cc1ccc(F)cc1 65358,C=C(Cl)CC(C(=O)NCC(=C)C)NC(C1C=CCS1)=O 65359,C=CC(C)CC(=O)NCC1CC1CNC(=O)C(c1ccn(C)c1)C 65360,N1(C(C(c2ccccc2)SCC)=O)CC2C(CNC(C3CCOC(C)C3)=O)C2C1 65361,c1(C(=O)NCC(C)NC(=O)C(C)Cc2ccncc2)cnc2ccccc2c1 65362,C1(C(=O)NC2C(CNC(c3c(C)nco3)=O)CC2)CN(C)CCO1 65363,C#CC1(C(=O)NCCCc2ccccn2)CCN(C(c2ccc(Cl)cn2)=O)C1 65364,C=CCC(F)(F)C(=O)NCC(C)(C)CC1CN(C(C2C(F)(F)C23CC3)=O)C1 65365,CC(CC(=O)N1CCCCC1c1n[nH]cc1N)C(C)(C)C.C(=O)N(C)CCF 65366,C1(C(=O)NCCC2CCC2)CCCCN1C(c1cc(CO)ccn1)=O 65367,C1(CCOC)(NC(=O)CC(n2cnccc2=O)C)CCN(C(=O)CCC2CC2)C1 65368,N1(C(c2c(Cl)nn(C)c2Cl)=O)CCC2CN(C(=O)C3=CCCOC3)CCC2C1 65369,C(=O)(C(CC)(CC)CO)N1CC(CC)C(NC(c2snnc2C)=O)C1 65370,CN1CCN(C(C2C=CCCN2C(=O)C(C2(O)CCCC2)F)=O)CCC1=O 65371,C1(C(N(CCCNC(C(C)OC(C)(C)C)=O)C)=O)CCC(O)C1 65372,N(C1CCSc2ccc(Cl)cc21)C(c1nnnn1C1CC1)CCn1c(C)nnc1 65373,C(CCCCC(=O)NC1CCN(C(=O)COCc2cc(C)on2)C(C)C1)=CC 65374,c1(C(=O)NCCCN(C(C(N2CCNC2=O)C)=O)C2CC2)ccc2nonc2c1 65375,c1(CNC(=O)NC(Cn2c(CC)ncc2)C)cccc(N)c1C 65376,C1(NC(=O)NCc2ccc(C)cc2)CC(NC(C2(C3CC3)CC2)=O)C12CCC2 65377,c1(C(=O)NCC2C(CNC(c3ccc(C)cc3C)=O)C2)ccccc1P(C)(C)=O 65378,c1(C(N2C(CNC(CC(=O)NC)=O)CC(F)(F)C2)=O)c(C)nc2ncnn2c1C 65379,c1(OC)ccc(CN2CCC3(CCC3)C2)c(Cl)c1O.N12CC(C(O)C1)C2 65380,C(C(C)(C)C(=O)N(CC(O)CN(C(=O)CN1CCS(=O)CC1)C)C)OC 65381,N1(C(CC2C(C)=NNC2=O)=O)CC2(C=C(C(=O)NCc3cccnc3F)CO2)C1 65382,c1(C(=O)NC(Cc2cnc[nH]2)CO)cnc(CNC(C2CC3(CC3)C2)=O)nc1 65383,c1(C(=O)NC(C2(O)CCN(C(=O)C3=C(Cl)CC3)CC2)C)ccc(Cl)c(Cl)c1 65384,c1(CC)cccc(C(N2CCC(O)(CCNC(c3ccc(CO)o3)=O)C2)=O)c1F 65385,C(=O)(C(C#N)C(C)(C)C)N1CC(C(N2CC(SCC)C2)=O)C(F)C1 65386,N1(C(c2c(CC)ocn2)=O)CCCC(N(C(=O)CC2(O)CCCCC2)CCO)C1 65387,Cc1cc(CN2CCC2(C)C(=O)Nc2cc(F)c(F)cc2I)c(O)c(C)c1 65388,CC(C)(C)S(=O)(=O)CC(=O)N1CCN(C(=O)CC2CCOC2=O)CC2(CC2)C1 65389,C1(NC(C2CC3C=CC2N(C(c2cnc(Cl)s2)=O)C3)=O)CN2CCC1(F)CC2 65390,C(=O)(C(C(C)NC(c1ccc2[nH]ccc2c1)=O)C(C)C)N(CC(C(C)C)OC)C 65391,Cc1cnc(C(=O)NC2CC3CC2N(C(c2nc(Cl)ccc2N)=O)C3)cc1C 65392,N1(C(C2C(C)(C)NC(=O)C2)=O)Cc2[nH]nc(C(=O)NC3(C)CC=CCC3)c2C1 65393,CC(C)(C)C(CNC(=O)C(C)(C)c1ccc(Cl)s1)NC(c1cn(C2CC2)nn1)=O 65394,c1(C(C)OC)nc(Cl)cc(=NCC2CC(NC(c3c(OC)ncnc3C)=O)C2)[nH]1 65395,CCCCC(C(=O)NC(C(N1CC2(CCC(=O)NC2)C1)=O)C(C)OC)C(C)C 65396,CCC(CC(=O)NOCC(=O)NCC1CCC(=O)O1)CC(C)C 65397,c1(OC)cc(CSCC(=O)N(C)O)cc(Cl)c1OC 65398,c1(SCC(N2CCC(C)(C)C2)=O)ccc(F)c(S(=O)(=O)N(C)C)c1 65399,CCC1=NOC(CNC(C2CCC(NC(=O)Nc3cn(C(C)C)nn3)CC2)=O)C1 65400,N1(C(COC(C)C)=O)CC2CCN(C(=O)CCCF)CC12 65401,C#CC(CNC(=O)CC1CCN1C(=O)CCc1cscn1)CC 65402,c1(C2(C(=O)NC3CN(C(c4c(C)[nH]cc4)=O)CC3F)CC2)ccc(Cl)c(F)c1 65403,N1(C(Cn2nc(C)oc2=O)=O)CCC(C2CC2)C1C(=O)NOCc1ccccn1 65404,c1(C(N(CC(CC)NC(c2occc2C)=O)C)=O)sccc1Cl 65405,c1(NCCC(CCC)O)ncc(C)cc1S(=O)(=O)NCC#CC1CC1 65406,c1(CC)cccc(-c2nc(C(C)Sc3nnnn3C3CC3OCC)n(C)n2)c1 65407,c1(COCCC(C)C)ccc(S(=O)(=O)NC(C2(C)CCC2)=O)s1 65408,Cc1nc(C(N2CC(NC(=O)CN3CCSCC3)C(O)C2)=O)cn1C(F)F 65409,N1(C(C2N(CC)CCC2)=O)C2CCC(C(=O)Nc3ccc4occc4c3)C1CC2 65410,N1(C(C(C2CC2)OC)=O)CCN(C(c2cc3n(n2)CCN(C)C3)=O)CC(C)(F)C1 65411,c1(-n2cc(C3(O)CN(C(C4N(C(C)C)CCCC4)=O)C3)nn2)cccc2ccnn12 65412,C1(CN(C(c2nnc(-c3ccccc3)s2)C(=O)NCC(F)F)C)CCCSC1 65413,c1(C(=O)NCCCNC(C2(C)CCCNC2=O)=O)cc(F)c(Br)c(F)c1 65414,CC(C(C)C(=O)NCC(F)F)NC(C1COC(=O)N1C)=O 65415,c1(C(=O)NCC(C(=O)NCC(CC)(C)O)CC2CCCC2)n[nH]cc1[N+](=O)[O-] 65416,C1(C(=O)NC23C(CN(C(Cc4ccn(CC)n4)=O)C2)C3)CN2CCN1CC2C 65417,C12(C(N(CCOC)CCN(C)C)=O)C3CC(CC13)C2(F)F 65418,c1(CC(C)C)ccnc(C(=O)NC(c2ncccc2Br)C)c1 65419,N1(C(C2=CCN(C(c3ccc(CC#N)cc3)=O)CC2)=O)CC(C)C12CCOCC2 65420,Cc1cc(C(=O)NC2CN(C(=O)C#CC3CCCOC3)C2)cc(S(C)(=O)=O)c1F 65421,C(c1ccccc1OC)=CC(=O)NCC(=C)CCNC(c1cnsn1)=O 65422,c1(CC(N2CCC(O)(CNC(CCS(C)=O)=O)C2)=O)ccc2c(c1)OCO2 65423,CCN=c1ccc(C(N2CC3CC2C3CNC(C2OCCN(C)C2=O)=O)=O)c[nH]1 65424,CC1CN2CCN1CC2C(=O)NCC1CCCCN1C(c1cnco1)=O 65425,C(C)(C(C(=O)C(=O)C1CC1)C(C)C)NC(c1ccc(C)n1C)=O.N 65426,c1(CC)ccsc1C(C(=O)NCc1ccco1)N(CCF)C1CC1 65427,C(=O)(C(C(C)NC(=O)C(C)=CC1CC1)C(C)C)N1CC(OCC)(CO)C1 65428,c1(C(C)=O)cn(C)nc1C(N1CCC(NC(=O)CC23CC(C2)C3)C1)=O 65429,c1(CC(N2CCCC(NC(C(CCC)NC(C)=O)=O)C2)=O)cc(Cl)cc(Cl)c1 65430,C(N=c1[nH]c2cc(F)cc(F)c2o1)C1CC(NC(C2C(S(C)(=O)=O)CCC2)=O)C1 65431,Cc1cnc(C(N2CCC3(CC3NC(=O)CCC(=O)N(C)C(C)C)C2)=O)c(C)c1 65432,c1(CC(C(N)=O)NC(C)(C)C(=O)NCc2nnc(-c3ccco3)o2)ccc(Cl)cc1 65433,c1(NCC(C)N(C)C(c2cc(F)c(CO)c(F)c2)=O)ncccc1S(C)(=O)=O 65434,C(C)(CS(C)(=O)=O)N(C(C(=O)N(C(C=C)C)C)=O)C 65435,C1(CC(=O)NC(C(=O)N(CCCOC)C)Cc2cn[nH]c2)CC(=O)NC1=O 65436,n1(CCC(=O)NCCC(C)NC(CC(=C)C)=O)c(=O)n(CC)c2ccccc12 65437,c1(OC)c(C(=O)NC(C)(CNC(c2cnc(C3CC3)s2)=O)CO)csc1Cl 65438,CC1C(NC(C2CCCCC2O)=O)CCCN1C(C1CC(=O)N1)=O 65439,CNS(=O)(=O)N1CCN(CCNCCOC2CCOC2)CC1 65440,N1(C(C(CC)OC)=O)Cc2occ(C(=O)NC3CC4C=CC3CC4)c2C1 65441,c1(CC)cccc2c(C(=O)NCC(C)NC(=O)C(C)(C)C3CCOCC3)c[nH]c12 65442,c1(C(=O)NC2C3(CC(OCC)C3)C2)c(OC)c(O)nc2ccccc12 65443,CC(C)C(CO)C(=O)NC1CCCC1NC(=O)CN1CCC(C(N)=O)CC1 65444,C1(NC(CCN2CCN(C)CC2)=O)COCCN(C(C2CCCCN2C)=O)C1 65445,N1(C(CC2(C#N)CCC2)=O)CCCC(N(C(=O)COC(F)F)CCF)C1 65446,CN1CC=C(CC(=O)N2C3CCCC2CC(NC(=O)CC2(C)CCCO2)C3)CC1 65447,CCC(C(=O)N(CCN1CCC1C)C)N(C(C)=O)CCN(C)Cc1ccc(Cl)s1 65448,C1(C(C)C)(C(=O)NCCN2CCC(CO)C2)CCCN1C(=O)CN1CC(C)(C)C1 65449,c1(C(N2C(CNC(c3cccc(F)n3)=O)CC2)=O)ccc2cc[nH]c2c1 65450,C1(C(=O)NC(CNC(c2cc(CC)on2)=O)C2CC2)(COC)CCCNS1(=O)=O 65451,c1(C(N(CCNC(C(CC#C)O)=O)CC)=O)n[nH]c2ccc(F)cc12 65452,N1(C(C2N(C)CC(F)C2)=O)C(C(N2CC3CC2CS3)=O)CCC12CC2 65453,N1(C(=O)C=Cc2ccoc2)CCC2C(CCN2CC(O)CCl)C1 65454,C1(C(=O)NCC(CO)NC(C2CCCN(CC(F)(F)F)C2)=O)CN2CCN1CC2 65455,C1(C(N2CCCC(NC(C3C(c4n(C)ncc4)C3)=O)C2)=O)CCS(=O)(=O)CC1 65456,Cc1cc(C(=O)NC(C2CCOC2)CNC(c2cc(CO)n(C)n2)=O)ccn1 65457,C(C)(CO)(C(=O)NCC=CCNC(C1CCCOC1c1cn[nH]c1)=O)OC 65458,Cc1cc(C)c(C#N)c(NCCc2csc(C)n2)n1 65459,C1(CNC(c2cn3c(n2)CCC3)=O)CC(C(=O)N2CCC(F)(CF)CC2)=NO1 65460,CCC(C(=O)N(C(C)CN(C)C(c1cnn(CC)c1)=O)C)N(C)C 65461,Cc1sncc1C(=O)NCCCN(C)C(C1CC1(C)C)=O 65462,N1(C(c2c(C)scc2)=O)CC(NC(=O)C#CC2CCCCC2)C2CCCCC12 65463,C1(C(N(CC(C)OC)C)=O)(OC)CCN(C(c2ccc(Br)cc2F)=O)CC1 65464,c1(C(C)C(=O)NC2(C(=O)O)CC3(CNC3)C2)cnc2n1CCCC2 65465,CC1C(NC(c2nn(C(F)F)cc2Cl)=O)CCCN1C(=O)C(C)CC1CC1 65466,S(=O)(=O)(CC(=O)N1CCC(C)C1CNC(c1cccc(NS(N)(=O)=O)n1)=O)NC 65467,c1(C(=O)NCC(CC(C)C)NC(=O)C2=C(Cl)CCC2)ccc2c(c1)CCCC2=O 65468,c1(C(=O)NC2CC(C)(CNC(C3CCN(CC)C3)=O)C2)cc2cncn2c(O)n1 65469,N1(C(C(N2CCOCC2)C)=O)CCCC(O)(CNC(=O)C2=CSCCO2)C1 65470,CC1CC(CNC(=O)CCOC2CCC2)CN(C(C2CCCS2)=O)C1 65471,CC(C)C(CCN(C(=O)CC1COC(=O)C1)C)N=c1nc(-c2ccccc2)[nH]s1 65472,N1(C(CCC(C)c2ccc(Br)cc2)=O)CC2(CCCN2S(C)(=O)=O)C1 65473,c1(CCC)nsc(N(C)CC2CCCN2C(=O)CCc2nccn2C)n1 65474,c1(CC)nc(C)c(C(N2CCCCC2CNC(c2cnn(C)c2Cl)=O)=O)c(C)n1 65475,N1(C(c2scc(C(C)(C)C)n2)C(=O)Nc2ccco2)CCCCC1CC(=O)N(C)C 65476,C(=O)(C(O)(C(F)(F)F)c1ccccc1)N1C(COC)CN(c2ccccc2)CC1 65477,N1(CC(=O)NC(C2CCOC2)CNC(C(C)(C)C2CC2)=O)Cc2ccccc2C1 65478,N1(C(C(C2(O)CN(C(C(C)(CO)OC)=O)C2)F)=O)CCN(C)CC1C 65479,n1(CC)cc(NC(C2(CNC(C3C4CC5C(C4)C35)=O)CC3(CC3)C2)=O)c(C)n1 65480,N1(CC)CC(C(=O)NC(CCC2CC2)C(=O)NCC2(CC3CC3)CCC2)CC1=O 65481,N1(C(c2c(C)nn(CC)c2C)=O)CC(NC(c2n[nH]c(C)c2C)=O)C2(CCC2)C1 65482,Cn1cc(-c2cn(CC(C3CN(C(=O)CNC(=O)ON)C3)F)nn2)cn1 65483,N1(C(C(C=C=C)C)=O)CCC(C2CCN(C(=O)COC3CC=CC3)CC2)CC1 65484,C1(CC)CN(C(=O)Cc2cnc[nH]2)CCN1C(=O)CN1CCC(C)(C)C1 65485,CCC(CC)C(CNC(=O)C1CC1)N1CCC(c2cccc(F)c2F)C1 65486,N1(C(C=C(C)c2ccccc2F)=O)CCCCC2(CCN(C(C3CCO3)=O)C2)C1 65487,c1(C(=O)NC2(CNC(C3(C)CCN(C)CC3)=O)CCC2)n[nH]c2c1COCC2 65488,CC1=NOC2(CCN(c3cc(C(F)F)nc(Cl)n3)CC2)C1 65489,C1(NC(CC=C)=O)(CNC(c2ccc(C(=O)OC)nc2)=O)CCCCC1C 65490,c1(Cn2cc(N)cn2)cc(Cl)ccc1Cl.c1(C(C)NC(=O)C=CC2CC2)ccccc1 65491,c1(NC(c2c(C)nc(C(=O)Nc3c(C)nsc3)s2)=O)ncc2[nH]ncc2n1 65492,C(=O)(CCC(=O)N1CCC(C(C)(C)NC(C23CC(F)(C2)C3)=O)C1)OCC 65493,C=CCCN=C(NCC1(F)CCC(CO)CC1)NCC1CCC(C(=O)OC)O1 65494,C1(NC(c2cnc(C3CC3)nc2)=O)CCCCC12CCN(C(=O)C=CI)C2 65495,c1(CC(=O)N(CCCNC(C2C(CC)OCC2)=O)C)ccc(O)cn1 65496,C=CCC(C)(C)CC(C(=O)Nc1ccccc1Cl)N1CCC2(CC1)CNC(=O)N2 65497,C(=O)(CCCCC1CC1)NC1(CC)CN(C(C(C)OCC#C)=O)C1 65498,C1(NC(CS(C)(=O)=O)=O)CN(C(=O)C2=CCSC2)CC12CCC2 65499,c1(NC(C2(C)CCCC2)=O)ccnc(C(F)(F)F)c1.n1(CCN)cc(C(C)O)nn1 65500,N1(C(C(CCC)OCC)=O)C2CCC1CN(Cc1nc(Cl)sc1Cl)CC2 65501,N1(C(c2cc(C)sc2)=O)C2CCC(C(=O)NCc3cncc(Cl)c3)C1CC2 65502,c1(C(N2CCCC(NC(C(CC)(C)O)=O)C2)=O)ccc(OC(C)C)c(Cl)c1 65503,CC1CC(NC(=O)CCP(C)(C)=O)CN(C(=O)COc2ccc(Cl)nc2)C1 65504,N1(C(C(C)CS(C)(=O)=O)=O)CCN2CCOCC2(CNC(=O)C(C)(C)C2CC2)C1 65505,c1(C(=O)NCC(C)NC(c2nnc(CN(C)C)s2)=O)ccccc1C1CC1(F)F 65506,N1(C(c2c(C)ccnc2O)=O)CC2(CCCC2NC(=O)CSC2CC2)C1 65507,CC(C)C(C)(C)C(=O)NC1CC(CNC(C2(C)CC3CCC2C3)=O)C1 65508,Cc1nccc(Cl)c1C(=O)NCC1(O)CCCN(C(=O)Cc2cn(C)nc2Cl)C1 65509,CON1CC(C(=O)N(CC(=O)N(CCC(=O)OC)C)C)CC1=O 65510,CON(CCC(=O)N1CCC2(CCCN2C)C1)C(=O)Cc1ccn(C)c1 65511,C1(NC(COCCOCC)=O)CC2CN(C(c3nc(O)c(C)s3)=O)CC2C1 65512,C1(NC(C=CC=CC)=O)CCCC1NC(CC(=O)NCC(F)(F)F)=O 65513,O=C1NCc2c(C(=O)NC3CC3NC(c3onc4ccccc34)=O)cccc21 65514,c1(OC)cccc(C(C(=O)NC2CC(NC(c3sc(C)cc3Cl)=O)C2)OC)c1 65515,N1(C(C(C(C)NC(CC2(NC(C)=O)CC2)=O)C)=O)CC(S(C)(=N)=O)C1 65516,c1(C(=O)NCC(C)(CO)NC(c2cc(C)c(C)[nH]2)=O)cc2ccccc2oc1=O 65517,c1(-c2ccc(F)c(F)c2)ccc(NCc2cnc(Cl)s2)c(F)c1F 65518,C(=O)(C1=NN2CCCN=C2N1)N1CCC(C2CC2)(CC)C1 65519,c1(OC)ccc(C=CC(=O)NC2(C3CN(C(=O)C(C)O)C3)CC2)c(OC)c1 65520,C(CC(=O)NCC1CC(SC)C1)N(C(=O)CC1CC1(C)C)CC 65521,c1(C(N2CC(CC)N(C(c3csc(C)n3)=O)CC2)=O)cncc(S(C)(=O)=O)c1 65522,CC(C)C(C(C)NC(=O)CCC(F)F)NC(=O)C=C1CCCCC1 65523,Cc1cc(O)ncc1C(N1CC(C2CC2)(C(=O)NCC2CC(C#N)C2)C1)=O 65524,Cc1ccc(-c2nc(CC3CCCCC3)nn2CCCO)c([N+](=O)[O-])c1 65525,C1(NC(C2(OC)CCOCC2)=O)CCC2(CC1)CN(C(=O)C(C(C)C)N(C)C)C2 65526,c1(CC)nc(N2CCCC(N(C(=O)C(c3ccccc3)O)C)CC2)cc(C#N)n1 65527,N#Cc1ccc(C(O)C(=O)NC2CC(NC(=O)C(F)=CCCF)C2)cc1 65528,N1(C(C2(C(N)=O)CC2)=O)CC2CC2(CNC(=O)Cc2nccs2)C1 65529,C1(C(=O)Nc2cccc(NC(C(CC)(C)CC)=O)c2)CC2CCCCN2C1 65530,C1(CNC(c2cc(C)n(C)n2)=O)CN(C(c2c[nH]cc2Br)=O)C2CCN1C2 65531,C1(NC(c2c(C)coc2)=O)CCCC1(C)CNC(=O)CCc1n[nH]c(=N)s1 65532,c1(CC(=O)NC2CC(N(C(c3c[nH]c(=NC)o3)=O)C)C2)c(OC)cccc1Cl 65533,C1(NC(C(C)c2ccsc2)=O)CC2CCC1N2C(=O)COc1ccc(F)cn1 65534,C1(C(N(C(CNC(COCCOC)=O)C2CC2)C)=O)CNC(=O)CC12CCC2 65535,N1(C(Cc2ncc(C)o2)=O)CCN(C(c2n[nH]c(C)c2C)=O)CC(O)C1 65536,C#CC1(O)CCCN(C(=O)CSCCNC(c2ccsc2C(F)F)=O)C1 65537,C(=O)(C#CC1CCCCO1)NCCCC1OCCN(C(c2c(C)nc(O)[nH]2)=O)C1 65538,CC1(C)C(C(=O)NCC(O)CNC(C2(C)CCC(=O)N2)=O)CCS1(=O)=O 65539,[N-]=[N+]=NCCC(=O)N1CCCC1CCC(N1CC(F)C(F)C1)=O 65540,Cc1cnn(CC(N2CCC(C)(CNC(=O)COCC3CC3)C2)=O)c(=O)c1 65541,Cc1ccc(C(N2CC(N(C)C(c3ncn4c3CCCC4)=O)C2)=O)c2c1CCC2 65542,c1(NC(C2CCN(C(c3ccc(OC)nn3)=O)C2C)=O)cccc(F)c1O 65543,C(CC(=O)NOCC1CC1)(c1ccccc1)NC(C1(CC)CCCO1)=O 65544,N1(C(c2cncc(C)n2)=O)CCCC2C(CCCN2C(=O)COC2(C)CCC2)C1 65545,C12CCN(C13CCC3)C(=O)CO2.C(C)(C)(C)OC(N(C(C)C)C1CC1)=O 65546,N1(C(C2(C)CC2)=O)CC2(CC2)CC1CNC(C1CC2(CCC2O)C1)=O 65547,Cc1cc(C(=O)NC(CO)C(C)NC(=O)C(O)Cc2ccccn2)c(Cl)cn1 65548,C(c1ccccc1[N+](=O)[O-])=CC(N1CC2(N(C(C3C(CC)C3)=O)CC2)C1)=O 65549,C(=O)(C1CCCc2nncn21)NC1CC(NC(C2(C)CCSCC2)=O)C1 65550,N1(C(c2c(C)coc2)=O)CCN2C(=O)C(NC(=O)CCc3ncnn3C)CC2C1 65551,O=C1CC(CC(=O)N2CC3CC3(NC(=O)CN3CCC(C(F)(F)F)CC3)C2)=NN1 65552,c1(CCC(=O)NC(CNC(CNS(CC)(=O)=O)=O)(C)C)ccccc1 65553,C(=O)(CC1=CCOCC1)NC1CN(C(CCOCCCOC)=O)C1 65554,c1(C(=O)NCC(CN(C(c2c(C)nco2)=O)C)C)ccc2c(c1)OCCCO2 65555,C(c1cnc2ccccc2n1)=CC(=O)NC(C)(CNC(c1ccnnc1)=O)CO 65556,c1(CN2CCC(CC(=O)NCCC(=O)OCC)CC2)cc(C(F)(F)F)cc(Cl)c1F 65557,CCC(=O)CCC(=O)N1CCOCC1CCNC(=O)CCc1cccc(C)c1 65558,C1(C(N2CCC(CN=[N+]=[N-])C2)=O)(CC)CN(C(=O)CCC2CC(C)C2)C1 65559,Cc1ccc(C(N2CCC3CCCC23CNC(c2csnn2)=O)=O)c(=O)n1C 65560,CC1CN(C)CC(C(=O)NCC(C2CC2)N(C)C(c2nccnc2N)=O)O1 65561,c1(CCC)n[nH]c(=NCC(C)(C)NC(c2cnc(O)nc2O)=O)s1 65562,Cc1ncsc1C=CC(N1CCC(N(C(=O)C(C)CF)C)C1)=O 65563,N1(C(N2C(CNC(=O)Cc3ncncc3Cl)CCC2)=O)CCc2ccccc2C1 65564,N1(C(CC(C)OC)=O)CC(C2(NC(c3ccc(Cl)cc3C(F)F)=O)CC2)C1 65565,S(=O)(=O)(c1cc(F)cc(Br)c1)NC1CC(C(=O)NCC2CCCCC2)C1 65566,Cc1ccc2nc(C(=O)NCC3CCCC3NC(=O)COCCO)ccc2c1 65567,N1(S(C(C)C)(=O)=O)CCN(C(C2C(C(=O)NCCC(F)(F)F)C2)=O)CC1 65568,N1(C(c2c(C)cccc2)=O)CC2(CCN(C(=O)C(C)NC=O)CC2N)C1.C(C)(C)SC 65569,C1(NC(C(=O)NCCOC)=O)C2CCC1N(C(=O)C(c1ccc(OC)cc1)C)C2 65570,C(=O)(C(C)(F)C(=O)N1CCCC(CNC(c2nc(OC)ccc2C)=O)C1)OC 65571,CS(=O)(=O)C1(C(=O)NCC2(CCNC(C3CC(N=[N+]=[N-])C3)=O)CC2)CC1 65572,c1(C(c2ccccc2)NC(CN2C(C)CCOC2)=O)cccc(Cl)c1F 65573,C(=O)(C(C)(C)C)NCC(=O)NCCOCCNC(C1C(CC)C1)=O 65574,N1(C(C2C=CC(NC(CCC(CC)OC)=O)C2)=O)CCN(C)C2(CC2)C1 65575,N1(C(C(=CC2CCCC2)C)=O)CCOCC(NC(=O)C=CCF)C1 65576,C(C1=CCCN(C(c2scnc2C2CC2)=O)C1)NC(=O)COc1cccnc1 65577,C1(NC(c2c(C)n[nH]c2)=O)CCCCCN(C(=O)C(O)C(C)(C)C)C1 65578,c1(C(N2C(CNC(=O)Cc3cncnc3)CC2)=O)ccc2c(c1)NCCC2 65579,C1(C(=O)NC(CC)C(C)O)CC(C)CN1C(C1CCCC(C)C1)=O 65580,Cc1n[nH]c(C)c1CC(N1CCC(NC(C2(n3cncn3)CC2)=O)CC1)=O 65581,N1(C(c2c(C)n(C3CC3)cc2)=O)CCCN(C(C23CCCC2(C(N)=O)C3)=O)CC1 65582,CCCC(C(O)C(=O)N1CCOCC1C(C)C)NC(c1c(F)cncc1F)=O 65583,N1(C(C)=O)CCCC(C(=O)NCCN(C(=O)CSc2nnnn2C)C(C)C)C1 65584,N1(C(CCC2CC(NC(c3scc(C)c3C)=O)C2)=O)CCCC(C)(O)C1 65585,N1(C(=O)NC2CCCC2(F)F)CCC2CCC(C1)O2 65586,C(=O)(C1=CC2(CCOCC2)C1)NCC1(C(N)=O)CN(C(CCCC(CC)C)=O)C1 65587,c1(C(=O)NC2C(C#N)CN(C(c3ccc(Br)c(Cl)n3)=O)C2)c(Cl)ccc(Cl)c1F 65588,c1(C(c2n(C(C(=O)OCC)C)nnn2)NCC2CCC2)cccc(OC)c1F 65589,N1(CCOC)CC(C(=O)NCCc2cccnc2OC)CC1=O 65590,Cn1ccnc1C(O)CNC(=O)C(N)Cc1ccoc1 65591,C(=O)(C(C)CC(F)(F)F)NC(CC(C)C)CNC(=O)C1=CCSC1 65592,N#Cc1c(F)cc(C(=O)NC2CC3(C2)CN(C(=O)CCCC(F)(F)F)C3)cc1F 65593,CC1C(C(=O)NCCCCCCF)CCCN1C(C1CCCC(=O)N1C)=O 65594,CC1CC(NC(=O)Nc2ccccc2SCC(N)=O)CCN1CC(N)=O 65595,C1(C(N(CC#C)CCF)=O)(CC=C)CN(C(=O)CC2CCC(C)C2)C1.C 65596,CON1CC(C(=O)NC(C(N2CCC(C)(CCO)C2)=O)c2ccco2)CC1=O 65597,C(=O)(C(CC(C)C)N(C)C)NC1(CNC(C(CCC)N(C)C)=O)CCOCC1 65598,c1(C2C(C(=O)NC3CN(C(C4(OC)CC4)=O)C3)C2)ccccc1Br 65599,N1(C(c2c(C)sc(-c3cccc(C(C)O)c3)n2)=O)CCn2c(O)nnc2C1 65600,c1(C(N(C2CCN(C(C3(C)ON=C(C)C3)=O)CC2)C)=O)c(Cl)ccc(F)c1N 65601,C1(NC(C2C(C#C)C2)=O)CC12CCN(C(c1ccc(Br)cn1)=O)CC2 65602,C#Cc1ccc(CC(=O)N(C2CN(C(=O)CC(C)OC)CCC2O)C)cc1 65603,n1(Cc2nc(C)on2)nnc(NC)c1C.C1(N=[N+]=[N-])(C=O)CC1 65604,Cc1ccc(C=CC(N2CC(O)(C(C)NC(=O)CNc3ccc(Cl)cc3)C2)=O)o1 65605,C1(CNC(c2c(C#C)c[nH]n2)=O)CC2CN(C(=O)C(O)C(C)C)CC12 65606,c1(C(N(C(C)CNC(c2cc(O)nc(O)c2)=O)C)=O)ccc(F)c2ccncc12 65607,Cc1cc(Cl)c(Br)cc1S(=O)(=O)NC1Cc2ccccc2N(C)C1=O 65608,c1(-n2cc(C3CN(C(C4C=CCC4)=O)C3)nn2)ccccc1-c1ncc[nH]1 65609,c1(C(N2C(CCNC(C3N(C)CC(F)C3)=O)CCC2)=O)cccc2c1COCC2 65610,CC1CCCC1CC(=O)NCC(C)(F)CNC(=O)Cc1cccs1 65611,C(CS(=O)(=O)CC(=O)NCC(C)(CNC(c1c(C)ncn1O)=O)OC)OC 65612,C(=O)(CCCCSCC)NC(C(=O)OCC)C1CN(C(C2(C(N)=O)CC2)=O)C1 65613,c1(NC(C(=O)NCCC(OCC)OCC)=O)cc(C)n(-c2ccc(Cl)cc2)c1C 65614,c1(OC)ccc(C(C)C(=O)NCCCCCNC(=O)CSC2CC2)c(C)c1 65615,c1(C(N2CCN(CC3CN(C(=O)CCC4CC4)C3)CC2)=O)ccc2nc[nH]c2n1 65616,C(=O)(C(C)(C)CCC#N)NCC(C(N1CC(CC=C)OCC1)=O)CC1CC1 65617,c1(C(N(C(C)CNC(=O)C=Cc2ccnn2C)CC)=O)ccc(C(C)C)cn1 65618,C1(C(C)NC(C(C)(C)NC(=O)NCC=C)=O)CCCN(C(c2cc(Cl)c[nH]2)=O)C1 65619,CCC(CC(=O)NC1CC2CCC1CC2NC(c1cn(C)[nH]c1=N)=O)C(C)C 65620,Fc1c(I)c(N(CC2COCc3ccccc32)CCO)nc2ccc(Cl)nc12 65621,c1(-c2cn(C3N(C(=O)C(N4CCCCC4)C4CC4)CC3)nn2)cnn2c1NCC2 65622,CN1CCC(F)(CNC(=O)C(C)(CO)NC(=O)CC2CNC(=O)O2)C1 65623,CC1OCCCC1C(=O)NCc1nnn(C)c1C(N1CCC(C)(C(N)=O)C1)=O 65624,C1(O)(CCNC(C2CCS2(=O)=O)=O)CCN(C(=O)Cc2ccsc2)C1 65625,Nc1ccc(-c2nc(C(N3CCCC3)=O)n(-c3ccnc(Br)c3)n2)nc1 65626,CCCC(CNC(=O)CC(C)n1cccn1)C(=O)NC1(C2(OC)CCC2)CC1 65627,c1(CC(=O)NC23CC(CNC(C(CCC)OC)=O)(OC2)C3)ccc(CO)c(C)c1 65628,C=CCCCCCCCC(=O)NC(C1CCN(C(=O)CCC(=C)C)C1)(C)C 65629,c1(C(N2CCC(C(=O)NCCNC(CCC#C)=O)CC2)=O)cccc2nncn12 65630,C1(C(N2CCOCC2)=O)(NC(C=C(C)C)=O)CCCCC1.c12cccc(c1)N2 65631,N1(Cc2ccc(OCC=C)cc2)CCC(=O)N(CC2(F)CCC(CO)CC2)C1=O 65632,C1(C(N2CCC(=O)NCC=CC2)=O)CCS1(=O)=O.C1(SC)CCCO1 65633,CN1CCc2[nH]nc(C(=O)NCC3CC3CNC(=O)C3=C(Cl)CCC3)c2C1 65634,c1(N2CCC(CNC(C3C(C(C)C)(C(=O)O)C3)=O)C2)ccc(Br)cc1 65635,N1(C(=O)CC2CC3(CCC3)CO2)CC2CN(C(C34CCC(CC3)CO4)=O)CC2C1 65636,N1(C(C(C(C)C)C#N)=O)CCc2nc(CNC(=O)CCn3ccnn3)sc2C1 65637,c1(C(=O)NCC2CCCC2O)cnn(-c2cccc(F)c2)c1C(F)(F)F 65638,Cn1cnc2[nH]c(C(N3CC(NC(C4CCC(=O)N4)=O)CC(F)C3)=O)cc12 65639,C1(NC(C)=O)CCN(C(C2COCC2NC(=O)C(=CC2CCCC2)C)=O)C1 65640,c1(C(=O)NCC2N(C(CCC=CC)=O)CC2)cccn(C2CCOCC2)c1=O 65641,C1(C(=O)NCCC2CCOC2)CC2(CC2)CN1C(=O)C=CC(F)F 65642,C=CCC(C)(C)CC(=O)NC(C)(C)C(C)NC(c1cn(C)c(C(F)F)n1)=O 65643,Cc1nnc(NC(CCc2ccc(C(C)(C)NCC(C)C#N)cc2)=O)n1C 65644,N1(C(CS(CCC)(=O)=O)=O)CCC2CCN(C(C3CCCSC3)=O)C2C1 65645,c1(C(=O)NCCCOCCNC(C=CC(CC)C)=O)cn(C)nc1Cl 65646,C1(Cc2cn(CCC=C)nn2)CCCCN1C(c1scnc1C(F)F)=O 65647,c1(C(=O)NCC2CCCC(NC(CCN(C)CC)=O)C2)ccc2ncccn12 65648,N1(C(C(C2CCCC2)NC(CCCCC)=O)=O)CC2(CCC(=O)NC2)C1 65649,c1(C(N2C3CN(C(C(C)C4CCC4)=O)CC2CC3)=O)c(Cl)c([N+](=O)[O-])nn1C 65650,CC1=NOC(C(=O)NC(CNC(C2CC(NS(C)(=O)=O)C2)=O)CC(C)C)C1C 65651,N1(C(c2c(C)nc(COC)s2)=O)CCC(C2CC2)C1CNC(C1CC1C(C)O)=O 65652,c1(COCC(=O)N(CCC(C)NC(C2CC(Cl)(Cl)C2)=O)C)nnc(S)n1C 65653,n1(CC(=O)NC2CC(CCNC(C(C(COC)C)C)=O)C2)nnc2ccccc12 65654,N1(C(c2cnc(OC)s2)=O)CCCCC1C(=O)NCc1cc(Cl)no1 65655,c1(C(=O)NC2CC3(CN(C(C(C(C)C)C)=O)C3)C2)ccc2c(c1F)CCC2 65656,CCC(C)(C#N)C(=O)N1CCC(NC(c2cc(Cl)ccc2OC2CCC2)=O)CC1 65657,c1(-c2ccc(C)c(C)c2)ccccc1S(=O)(=O)NCC(O)CN1CCCC1 65658,N1(C(C(N2CCN(C)CC2)C)=O)CC(NC(C23CCCN2CCC3)=O)CCC1C 65659,N1(C(=O)CC(C2CC2)C2CC2)C(C(=O)NCc2nccs2)CCC1C1CC1 65660,C1(C(N2CC(OC)(CNC(c3ccc(-c4ccco4)s3)=O)C2)=O)CC(C)OC1C 65661,c1(COC)cc(C(=O)NCC(c2cccc(C)c2)NC(C2CC2(F)F)=O)c(C)o1 65662,C1(NC(c2ccc(C3CCCCC3)cc2)=O)CC(NC(C2CC2(Cl)Cl)=O)CC1O 65663,c1(C(N2CCOCC(C)C2)C(=O)NCCC2(C)CC2)ccc(F)c(Br)c1F 65664,C1(C)(C(N2CC(N(C(=O)CCCF)C)C(O)C2)=O)CCC2(CC1)OCCO2 65665,c1(OC)nn(C)c(Br)c1C(=O)NC1CC1NC(C1(C)CC1(F)F)=O 65666,C(CC(=O)N1CC2(CSC2)C1)(C(F)(F)F)NC(c1n(CCC)ncc1)=O 65667,Nc1ccnn1CC(N1CCCC1CNC(C1(CC2CC2)CC1)=O)=O 65668,c1(C(N(CCCN(C(=O)Cc2ccc(F)c(Cl)c2)C)C)=O)nc2cnccc2s1 65669,CN=c1[nH]c(C(=O)NCCC2CCCCN2C(c2cn(C)cn2)=O)cs1 65670,N1(C(CC2C(=O)OCC2)=O)CC2(CC(C(=O)NCC34CCC(CC3)CC4)CO2)C1 65671,Cc1cc(Br)c(F)cc1C(=O)NC1CC(NC(=O)CCOC(C)C)C1 65672,C1(OCC)CC2(C1)CC2C(N1CC(OCCNC(=O)CN2CCC2C)C1)=O 65673,C#CC1(C(N2CCOCCC2C)=O)CCN(C(=O)CCC(C)(F)F)C1 65674,CC1CCCC(CC(=O)NC(C2CCN(C(c3ccn(CCF)n3)=O)CC2)C)O1 65675,c1(C(N(CC(C)(C)OC)C)=O)cc(CCNC(c2ccn(C)n2)=O)on1 65676,C(C(CNC(c1cc2n(n1)CCC2)=O)C(F)(F)F)NC(CSCCOC)=O 65677,C1(F)(CNC(C(C)(C)OC(C)=O)=O)CCN(C(=O)C(C)C(C)(C)C)CC1 65678,C1(C(=O)NC(CC(C)C)CO)CC12CCN(C1CCC(=O)N(C3CC3)C1=O)CC2 65679,CN=c1cc(C(N2CCC(CNC(C3CC3CC(C)(C)C)=O)(OC)C2)=O)cc[nH]1 65680,N1(C(=O)CCc2cccnc2)CC2(C1)CN(C(C1(CCO)CC1)=O)CCO2 65681,c1(C(c2nnnn2C2CC2)NC(C=C)C2CCC2)cn(C)nc1C(F)F 65682,CCC(C(=O)Nc1cccc(C(C)(C)C)n1)C(C)C 65683,C1(C(N2CCN(C(=O)Nc3ccc(F)cc3F)CC2)=O)CCc2cncn2C1 65684,Cc1ccc(N(CCN(c2ccncc2)C)C(C2(Cc3nn[nH]n3)CC2)=O)cc1 65685,C1(NC(C2C(C)OCCC2)=O)CN(C(c2cscc2C(F)(F)F)=O)CCC1CO 65686,c1(C(=O)NC2(CCOC)CCN(C(=O)C3=CCCO3)C2)cc(Cl)ccc1C 65687,C1(C(C)C)CCN(C(c2cnc(C3CC3)o2)=O)CC1.C12(CCCO1)C(=O)NC2 65688,C1(CNC(C2CCCSC2)=O)CCC2(CN(C(c3c(O)ccc(Cl)c3O)=O)C2)O1 65689,CC1CCCC1C(N1CC(C)(CNCc2ccc(Cl)s2)C1)=O 65690,C1(CC23CN(C2)C3=O)CCCS(=O)(=O)C1.C1(C(=O)OCC)CCCC(C(N)=O)C1 65691,Cc1ncncc1C(=O)NC(C1CC=CCC1)C(=O)N(C1CCN(C2CC2)C1)C 65692,C1(N(CC#C)C(C2CC=CCC2)=O)CCN(C(c2ccnc(C(C)C)n2)=O)CC1 65693,C(=O)(C(C)=NOCC#N)NCC(CC=C)NC(=O)CNC(=O)NC 65694,N1(Cc2cn(C)nc2C2CCC2)CC(=O)N(CC2CC3CCC2O3)C1=O 65695,N1(C(CC(=O)NCC)=O)CCCC1(C)C(=O)NCCC1(OC)CCC1 65696,Cc1cc(=O)oc(C)c1C(=O)NCCc1ocnc1CNC(=O)C=CC1CCC1 65697,C1(F)(C(N2CCC(C)(CCNC(C3(C#C)CCC3)=O)C2)=O)CCCN(C)C1 65698,c1(C(=O)NC(CN(C(=O)CC2C=CCCC2)CC)C)scnc1Cl 65699,CCCC(CCC)C(=O)N(c1ccnc(N(CCO)CCO)n1)C1CCOCC1 65700,C1(CNC(C2CC(=O)NC2)=O)CCCCN1C(=O)CCNc1cncnc1 65701,c1(OC(C)C(=O)N(C2CC2)CC2CC(F)CN2C(=O)C2=CCC2)cccc(Cl)c1 65702,c1(OCC(=O)NC2C(NC(=O)OC(C)(C)C)C2)ccc(F)c(C=O)c1 65703,N1(C(C(N2CCN(C)CC2)C)=O)CCC(C2CCCN(C(C3(CF)CC3)=O)C2)C1 65704,C(CC(F)F)(C(=O)NCCN1CCCCC1C)NC(CC=C)=O 65705,c1(C(=O)NCC(CNC(c2oc(C)nc2C)=O)OC)ccc(C(F)F)nc1O 65706,N1(C(c2nnc(C)o2)C)CCC(NC(c2cccc(F)c2Cl)=O)C(C)C1 65707,C(CNC(c1cncnc1)=O)(CC(F)(F)F)NC(c1cnc(SC)s1)=O 65708,C=CC(C)(CC)C(=O)NCc1ccc(CNC(=O)C(C)NC(=O)CC)cc1 65709,n1(C(C)C)cc(Br)c(C(=O)Nc2ccccc2CC2NC(=O)NC2=O)n1 65710,c1(C(=O)NCC(CCCC)NC(C2C3CCCCCC23)=O)cccc2c1COC2 65711,c1(C(=O)NCC2(NC(C3CC(C)OC3)=O)CCCCC2)cc2n(c1)CCOC2 65712,C1(NC(c2cccc(C)c2)=O)CC2(C1)CN(Cc1cc(O)ncc1Br)C2 65713,C(=O)(C(CC)C(C)(C)CC)NCC(CNC(C(C)OCC#C)=O)OC 65714,C1(CC)CN(C(=O)Cc2occc2C)CC1NC(c1ccc(SC)cc1)=O 65715,C12CCN(C1)C(=O)CO2.c1(SCCNC(C2CC(=C3CCC3)C2)=O)cccnc1 65716,Cc1c(C(=O)NCCC2(C(=O)NC3COCCN(C)C3)CCC2)cncc1F 65717,CCC(C)CC(C)C(=O)NCC(C(C)C)NC(c1n[nH]c(C)c1Cl)=O 65718,c1(C(=O)NC2CCC(N(C(C(CC)n3ccnc3)=O)C)C2)ccc(F)c(C)c1O 65719,Cc1cnc2n1CC(C(=O)NCC(F)CNC(c1csc(Br)c1)=O)CC2 65720,C(=O)(CCP(C)(C)=O)NC(C(=O)NCC#CCOC)CCOC 65721,c1(NC(C)=O)ccc(Cl)c(C(N2CC(CN(C(=O)CC3CCCO3)C)C2)=O)c1 65722,c1(N(C(c2ccc(Br)cn2)C(=O)NC2COC2)C)cccc(Br)c1F 65723,C(=O)(CCC(O)C(C)(C)C)N1CCC(C)CC1 65724,Cc1cc(C(=O)N(CCC(C(C)(C)C)NC(=O)CCC2CC2(F)F)C)cc(C)n1 65725,N1(C(c2c(C)con2)=O)CCC2(CCCN2C(=O)C=CBr)C1 65726,N1(C(c2cc(CC)nnc2C)=O)CCCC12CCN(C(c1cc(Cl)ccn1)=O)C2 65727,Cc1nnnn1CC(=O)NC1(C)CC(NC2(C)CN(C(=O)OC(C)(C)C)C2)C1 65728,c1(C(=O)NC2COCC2CNC(C2CCC(=O)N2C2CC2)=O)nnc(O)nc1O 65729,CC1CCCC1NC(=O)C#CCNC(=O)COCc1nc[nH]n1 65730,Cc1cc(C(N2CCC(C)C(N(C)Cc3ccccc3)C2)=O)cc(C#N)c1 65731,c1(C(N(C(CNC(C2(C(=O)OC)CC2C)=O)C2CC2)C)=O)ccc(F)cn1 65732,C(c1ccc(C)c(Cl)c1)=CC(=O)NCC1CN(C(CC(=O)NCC)=O)CC1(F)F 65733,Cc1cccc(CC(=O)NCCCNC(=O)CN2CCNC2=O)c1Cl 65734,C(=O)(C(CCC)CC(C)C)N1CC2(CCN(C(CCC=CC)=O)C2)C1 65735,C(=O)(C1CCCc2n[nH]cc21)N1CCC(COC)(NC(c2c(C)ncn2O)=O)C1 65736,C1(C(=O)NC(CCNC(C=CC)=O)C)C(C=C(C)C)C1(C)C 65737,c1(C(=O)NCC(c2ccccc2)N(C(C(C)=C2CC2)=O)C)ccc(Cl)c(C)c1Cl 65738,CC(N=c1ccnc(N2CCC3(CNC(=O)O3)C2)[nH]1)c1cn(C)cn1 65739,N1(C(C(C)N(C(C)=O)C)=O)CCC(NC(=O)C2=C(Cl)CC2)C2(CCC2)C1 65740,CCC(CC(F)(F)F)N=c1nc(N2CCC(P(C)(C)=O)C2)c2c([nH]1)CCC(C)C2 65741,c1(OC)cc(C(N2CC(CNC(c3ccc(C#N)o3)=O)C2)=O)ccc1OC(F)F 65742,N1(C(C(C(C)C)(C)O)=O)CCC2(CCCN(C(=O)CCn3cc(Cl)cn3)C2)CC1 65743,C1(C(N2CC(OCC(=O)NC)C2)=O)CC(F)CCN1C(=O)CCCN=[N+]=[N-] 65744,CC1(C)C2CCC1(CCNC(c1ccccc1F)C(F)(F)F)C2 65745,c1(OCC)c(C(=O)NCCCCCNC(C2(C)CC3CCC2C3)=O)cccc1F 65746,Cc1cc(N)ccc1C(N1CCCC(N(C)C(C2CN(C3CCC3)C2)=O)CC1)=O 65747,C(C1CCOc2ccccc21)NC(c1cc(-c2ccccc2)c[nH]1)=O 65748,n1(CC(=O)NCC2(OC)CN(C(=O)CC3NC(=O)NC3=O)C2)c(C)c(C)sc1=O 65749,c1(C(N2CCC(NC(c3c(CC)ocn3)=O)C(C)C2)=O)nccn2cc(C)nc12 65750,c1(C(=O)NCC2CCCN(C(C(C=C)(C)O)=O)C2)cnc(OC)cc1C(F)F 65751,c1(OC)ncc(C(N2CCC(NC(=O)C(C)N(C)C)C3CC23)=O)cc1Br 65752,N1(C(C2C(C(C)O)C2)=O)CCCC1CN(C(=O)CCn1cc(Cl)cn1)C 65753,c1(C([N+]2([O-])C(C)CN(C(C3(O)CC3(C)C)=O)CCC2)=O)ccc2nnn(O)c2c1 65754,c1(C(N2C(C(N(CCCC)CCO)=O)CC3CC32)=O)ccc([N+](=O)[O-])cc1O 65755,c1(C(=O)OCC)cc(N2CCC(NC(c3cnn(C)c3Cl)=O)C(C)C2)nc(C)n1 65756,N1(C(C2N(C(C)=O)CSC2)=O)CCCCC1CNC(c1cc(OC(C)C)n(C)n1)=O 65757,C(C)(CC(=O)N1CC=CC1C(=O)NCCCc1nc(C)no1)SC 65758,C1(CNC(C(c2cccs2)NC(C(C)NC(=O)NC)=O)=O)CNC(=O)C1 65759,Cc1cc(CN(C(C)CCCCCl)C2CCC2)cnc1Cl 65760,c1(C(N2CCC(C)(NC(CCC=C)=O)C2)=O)[nH]c2ccc(F)cc2c1C 65761,CCCC(C(=O)NCC1(C)CCCN1C(c1nc(=O)n(C)[nH]1)=O)OCC 65762,N1(C(C(C2CC2)NC(=O)CC=C(Cl)Cl)=O)C2C=CCC1CC2 65763,c1(CN(C2CCCC(O)C2)C)cc(Cl)cnc1O 65764,C1(CCNC(C2(F)CCCCC2)c2n(CCC3(C)CC3)nnn2)CCC(C)CC1 65765,N1(C(C(C)(C)O)=O)CCCC2CN(C(c3cnc4sccn4c3=O)=O)CCC12 65766,C12(N(C)C)CCC(C(=O)NCCC(C)(C)NC(=O)Cc3cnnn3C)(CC1)CC2 65767,C1(CCC)CN(C(=O)CCC2CCC(=O)C2)CCN1C(c1c[nH]nc1C)=O 65768,c1(C(=O)NCC2N(C(c3nn(CC)c(O)c3)=O)CC2)cc[nH]c2nccc1-2 65769,C1(F)(CNC(c2cc(Cl)c[nH]2)=O)CN(C(C2CCCSC2)=O)C1 65770,c1(CC(=O)NC2C(C(N(CCC(C)C)C)=O)OCC2)ccnc(O)c1 65771,CCC(CC(=O)NCC1CN(C(=O)C(c2cnn(C)c2)=O)C(C)(C)C1)C(C)(C)C 65772,c1(C(=O)OC)cnc(C(N2CC3(CCN3C(C3(C)CNC(=O)C3)=O)C2)=O)c(N)c1 65773,C1(CC)CC(CC(=O)NCCCc2ccccc2I)CCO1 65774,c1(C(=O)NC(C2CCCN2C(c2cn(C)nn2)=O)C)nc(Br)c[nH]1 65775,C(C(C)CC(=O)N1CCC(OCCn2cc(C=CC3CCCCC3)nn2)C1)OC 65776,C(=O)(CS(=O)(=O)C1CC1)N(C(CNC(c1cc(N(C)C)ccn1)=O)C1CC1)C 65777,C1(C(=O)NC2(C)CCOC2)C2CN(C(=O)CCc3nc[nH]n3)CC12 65778,c1(C(N(CC(C)NC(C2(Cl)C3CCC(=O)C23)=O)C)=O)cc[n+]([O-])cc1 65779,C1(CNC(CC(C)SC)=O)CC(F)(F)CN1C(=O)C=C(C)C1CC1 65780,CC(c1ccc(F)cc1F)=CC(=O)NC(C)C(CO)NC(=O)C(C)(C)C(C)O 65781,C1(NC(C2(C)C(C)C2)=O)CCC12CCN(C(c1ccc3nn(C)cc3c1)=O)CC2 65782,N1(C(CCCCCCC)=O)CCC2(CCCN(C(C34CCC3CC4)=O)C2)CC1 65783,N1(C(c2cc(OC)n(C)n2)=O)CC(NC(c2sccc2Cl)=O)C2CCCC2C1 65784,c1(OC)cc(=O)n(C)cc1C(N1CC(N(C(=O)C#CC2CCCC2)C)C(O)C1)=O 65785,N1(C(C2(C)CC(C)C2)=O)CCCCC12CC(NC(c1cccc(CF)c1)=O)C2 65786,CCC(C)CCCCC(=O)NCC1(CNC(=O)C(C)CC(F)F)CCCCC1 65787,C1(C(=O)Nc2ccccc2Nc2ccccn2)CCC2(CC1)CS(=O)(=O)C2 65788,c1(C(N2CC(Cn3cc(-c4ccc(Cl)c(F)c4)nn3)C2)=O)cc2n(n1)CCCC2 65789,c1(OC)c(C(=O)NCC2CC2NC(C2(C)CC3CC3C2)=O)ccc(Cl)c1Cl 65790,C1(CNC(CN(CC)CC)=O)CC2CCC1N2C(c1cc(F)ccc1OC)=O 65791,C1(CNC(c2c(C(C)C)onc2)=O)CCN(c2ncnc(Cl)c2F)CCC1(F)F 65792,N1(C(C=CC(C)NC(c2c(OC)n[nH]c2)=O)=O)CC2(CC2)CC1C#N 65793,C12(NC(C=Cc3c(C)cccn3)=O)CCCN(C(=O)C=Cc3cn[nH]c3)CC1C2 65794,C(=O)(CCCCC(C)=O)N1CCCC(C)(C(=O)NC(CCC)(C)CC)C1 65795,CC(C)(CNC(=O)CCN(C(=O)CCc1nc(=N)[nH][nH]1)CC1CC1)C(N)=O 65796,C1(N)CCOC1C(N)=O.C(=O)(C(C)CO)N(CC(O)C(C)C)CC=C(C)C 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66077,N1(C(c2c(CC)noc2)=O)CCN(C(=O)Cn2c(C)csc2=O)C(CC(F)F)C1 66078,c1(SC)nccc(=NC(CNC(c2n[nH]cc2C(F)(F)F)=O)C(C)C(C)C)[nH]1 66079,CC(=O)CCN=C(NCCc1ccc(Cl)o1)NC1CN(C(=O)OC(C)(C)C)C1 66080,c1(NC(COC)CO)nc(N2CCOC(C3CC3)C2)nc2sccc12 66081,C#CCC(CC#C)C(=O)NCC1=CCN(C(=O)C(c2cccs2)SC)CC1 66082,O=C(C1c2c[nH]nc2CN1C(c1cnc(O)o1)=O)NC1C2COCC12 66083,c1(C(=O)NC2C(NC(c3coc(C(F)F)c3)=O)CCC2)ccc2c(c1)COC2=O 66084,C(=O)(C1=CCCSC1)NC1C(NC(CCc2ccc(OC(C)C)cc2)=O)CCC1 66085,C1(NC(C2(NC(c3ccnc(O)c3)=O)CCC2)=O)CCOCC1F 66086,CCC(C)CC(=O)NCC1CCC(NC(=O)C(C)(Cl)Cl)C1 66087,N1(C(C=COCC)=O)C(CNC(c2cn(C)nc2SC)=O)CC2CC12 66088,C#Cc1ccc(C(=O)NCCOC2CN(C(=O)Cc3n[nH]c(=NC)s3)C2)cc1 66089,C12(CNC(C(CCC)O)=O)CCC(CC1)N2C(=O)Cc1ccc(OC)cc1C 66090,C1(CNC(c2ncn(C)n2)=O)CN(C(=O)C(C)(F)F)CCO1 66091,C1(C(N(C(=O)CSC2CC(n3ccnn3)C2)C)=O)CCC(C#N)C1.C12(CC1)CC2 66092,CCCCC(C)CCC(=O)NCC1(CO)CCN(C(=O)CC2CC=CCC2)C1 66093,C(=O)(C(F)CCC(C)(C)C)N(C1(C(N2CCC(C(=O)NC)C2C)=O)CC1)C 66094,C1(C(=O)NCCC2(C(NOCCOC)=O)CCC2)CCCC1C 66095,Cc1nnc(O)c(C(=O)NC2CN(Cc3cccs3)C2)c1C 66096,C1(CC(=O)N(C2CCCC2)CCCNC(CC(CC)C)=O)CCCCCC1(F)F 66097,c1(C(N2CCN(C3CN(C(CSCCC(C)C)=O)C3)CC2)=O)ncc(F)cc1N 66098,C1(C(=O)OC)(C(=O)NC(C)CCNC(C2(CC(F)F)CCC2)=O)CCO1 66099,N1(C(C(C=C)(C)CC)=O)CCOC2(CCN(C(c3cccnc3)=O)C2)C1 66100,N1(C(C(CC)C)=O)CC2CC1CN(C(=O)C(N1CSCSC1)C)C2 66101,N1(C(CN(C(C)=O)C)=O)CCC(F)(C(=O)NC(CC2CCC2)CO)CC1 66102,N1(C(C2N(C)CCC2)=O)CCN(C(=O)C(F)=CC2CC2)CC1c1ccccc1Cl 66103,C1(NC(Cc2scc(C)c2)=O)CCN(C(c2cc(C)cnc2Cl)=O)CC1(C)C 66104,C1(C2(O)CCN(C(c3cscc3Cl)=O)CC2)(NC(=O)COCC2CCOC2)CC1 66105,C1(N(C(C2CCCCC2O)=O)CC)CCCN(C(C2CCC(C)CC2)=O)C1 66106,N1(C(c2c(C)nc[nH]2)=O)C2CCC1CN(C(=O)CCc1ccc(O)c(O)c1)C2 66107,c1(CC)ccnc(N(C)C(=S)NCC(c2ccc(F)cc2)O)c1 66108,N1(C(CC2C=NN(C)C2=O)=O)CC(NC(=O)CCn2ccccc2=O)CC(F)C1 66109,c1(N(C)C)c(F)cc(C(=O)NC2CC2C(=O)NCc2nc(Br)cs2)cc1F 66110,CCCCC(O)CC(=O)N1CCCC1C(C)(C)NC(=O)CSCCN(C)C 66111,N1(CC=CCNC(C=CCN(C)CC)=O)CCC(NC(c2sccc2Cl)=O)CC1 66112,c1(C(N2C(CNC(C(CC)=O)=O)CCC2)=O)cc(C(C)(C)C)cc(C(C)(C)C)c1 66113,C(CCC(O)C(=O)NCC1CCC1C(=O)OC)NC(=O)C(F)F 66114,S(=O)(=O)(c1cccnc1NC(CO)C1CC1)NC(C(C)(C)C)c1ncccn1 66115,C1(NC(C2(C=C)CCC2)=O)CCCN(C(c2ocnc2-c2ccccc2)=O)C1 66116,C(C(C)(C)C#CC(=O)NC1(C(N)=O)CC1)NC(Cc1scc(C)c1)=O 66117,c1(C(N2CCC(CNC(C3(N(C)C)CC3)=O)C2)=O)cccc2c1CCCC2 66118,C(=O)(C(F)C1=CCCCC1)N(CC(CNC(Cc1c(C)cccc1)=O)O)C 66119,N1(C(c2ccccc2OCc2ccccn2)=O)CC2(CO)CC1(CO)CC2 66120,N1(C(C(C)(C)c2cscn2)=O)CC(NC(c2cnc(C(C)(C)C)o2)=O)C2(CC2)C1 66121,c1(SC)cc(C)ccc1C(N1CCN(C(C2CSC2)=O)CC1CS(C)(=O)=O)=O 66122,c1(CN2C(CC)CCC2)cccc(C(F)(F)F)n1.C(C)(CC1CCC1)N1C(=O)N1 66123,N1(C(c2ccc(NC)cn2)=O)CC=C(C(=O)NC2CC2C2CC2C)C1 66124,c1(CNC(C2C(c3cc(=N)[nH]cc3)C2)=O)nc2ncccc2o1 66125,c1(C(=O)NCc2c(C3CN(C(C(C=C)O)=O)C3)ocn2)ccc(C2CC2)cc1C 66126,Cc1n[nH]cc1C(=O)NC1CCC(N(C)C)C1.C12(CCCC1)CCCNC2=O 66127,CC(C)C(CC(=O)NCC12CCCCC1C2)NC(CCCC(=O)OC(C)(C)C)=O 66128,c1(CC)nc(C#N)cc(=NCC2CN(C3CCN(C4CCN(C)CC4)CC3)C2)[nH]1 66129,Cc1nc(C)c(C(=O)NC2CCCC(NC(c3cnc[nH]c3=N)=O)C2)o1 66130,Cc1n[nH]c2nc(O)c(C(N3CC(O)(CNC(=O)C(F)n4ccnc4)C3)=O)cc12 66131,N1(C(C2CCC(OC)CC2)=O)CC(F)(F)CCC1C.C(=O)(N)N 66132,N1(C(CSC)=O)CC(O)C(O)C1CNC(C1CC(=C(F)F)C1)=O 66133,N1(C(C2(CNC(N)=O)CC2)=O)CCCC1.NC 66134,CC1(C)CN(C(=O)COc2ccc(F)c(F)c2)CC1NC(=O)CC1CC12CC2 66135,C1(NC(C2N(CCC)CCCC2)=O)CC2CCC(C1)N2C(c1c[nH]c(=NC)s1)=O 66136,c1(OC)cncc(C(=O)NC(C2CCN(C(=O)CC3CCC(=O)N3)C2)(C)C)n1 66137,c1(OCCCC)ccc(C(=O)NC(C)(C)CNC(c2cnc(CC)s2)=O)c(Cl)c1 66138,c1(C(=O)NCC(=O)NC(CCNC(c2c(C)ocn2)=O)C)sc2ccccc2c1Cl 66139,CC1C(NC(=O)CC(C)(C)C(F)F)C(C)CCN1C(=O)CCOCC(F)F 66140,CC1CC(NC(c2cnn(CC(F)F)n2)=O)CN1C(=O)Cc1cc[nH]c(=N)c1 66141,c1(C(N(C2CCCN(C(=O)C(O)C(F)F)CC2)CC)=O)nc(C)c(C)nc1C 66142,N1(CC(=O)N(C)Cc2cc(Br)cs2)CC(C)(C)OC2COCC12 66143,N1(CC(=O)N(CCC(=O)N2CC(N3CCCC3)C2)C(C)C)CCCC1C 66144,C1(NC(c2cccc(COC)c2)=O)CCN(C(c2cccc(CO)n2)=O)CC1O 66145,C1(CC)CN(C(C2(F)CC=CC2)=O)CCC1NC(C1CCC(CC#N)CC1)=O 66146,c1(NC(=O)C(N2CCCC(Cc3ccccc3)C2)=O)cc(Cl)cnc1Br 66147,C1(CN=[N+]=[N-])CCCN(C(c2cncc(CNC(=O)C=CC3CCC3)c2)=O)C1 66148,C(N=c1[nH]cnc2c1SCCC2)C1C(C)(C)CN(C(c2cnc(C3CC3)[nH]2)=O)C1 66149,C(C(O)CCNC(c1csc(-c2nc[nH]n2)n1)=O)NC(=O)CCc1cnn[nH]1 66150,c1(C(N2C(C(N3CCC(=C)C3)=O)CCC2C)=O)ccc(C#N)n1C 66151,C1(C(C)NC(=O)Cc2nnc(O)s2)CN(C(c2ccc(C(F)F)o2)=O)CCO1 66152,c1(C(=O)NC2C(NC(CCN(CC)CC)=O)CC2)cnc(O)cc1O 66153,c1(CC(=O)NC2CCC(CNC(Cc3ccn(C)n3)=O)C2)c(F)cccc1C#N 66154,Cc1ccnc(C(N2CC(NC(C3CC(F)C(=O)N3)=O)CC2CO)=O)c1 66155,C12(C(C)NC(C3CC(C)N3C(=O)C=Cc3ccnn3C)=O)CCC(CO1)C2 66156,N1(C(C(CCSC)(C)C)=O)CCC=C(C(=O)N(C)CC2C(C)(C)C2(C)C)C1 66157,c1(NC(C(CC(=C)Cl)NC(c2cc[nH]n2)=O)=O)cccc2c1CCO2 66158,C1(C(CNC(C(C2CC2)OCC)=O)F)CCN(C(c2csc(CO)n2)=O)CC1 66159,C12(C(=O)NC(C3CN(c4snc(CCOC)n4)C3)C)CCC(CO)(CC1)CC2 66160,c1(C(=O)NCC(CNC(C(C)n2cccn2)=O)CO)ccc(C#N)cn1 66161,c1(C(=O)NC2(CNC(C3CCNC(=O)C3)=O)CC(OC)C2)n[nH]c2c1CSCC2 66162,c1(OCC(=O)OCC(=O)N(C(C)C)CCN(C)CC2(C)CCC2)cccc(Br)c1 66163,c1(C(=O)NC2CCCN(C(=O)CSCC(F)(F)F)C2)ccc2c(c1)B(O)OC2 66164,N1(C(c2c(CC)noc2)=O)CCC(c2cn(C(C)C)nn2)CC1 66165,CC1CN(C(c2cc(CNC(c3ccon3)=O)[nH]n2)=O)CCC1O 66166,C1(C(N2C(CN(C(=O)C(CC(C)C)OC)CC)CCCC2)=O)CCCCCCC1 66167,C1(C(=O)NCC2(CCNC(c3cc(OC)n[nH]3)=O)CC2)CCCC1S(C)(=O)=O 66168,N1(C(CCOC)=O)CC(NC(c2ccc(F)c(C(F)(F)F)c2)=O)CC2(CC2)C1 66169,C(C(F)C(=O)NCC(O)CCNC(C1(C#N)CCC1)=O)N(CC)CC 66170,C1(NC(c2cc(CC)nnc2C)=O)CC2CCC1C(NC(=O)CN1CC=CC1)C2 66171,C(=O)(C(C)(C)COC)N1CC(C)(C(N(CCCCC=C)C)=O)C1 66172,C1(C(=O)NC(C)CNC(c2cncc(Cl)c2)=O)CCC2(CC1)CC2(F)F 66173,N1(C(C(c2cccc(C)c2)O)=O)CC2CC(C1)C2NC(C1CC1C)=O 66174,c1(C(=O)NC2CC(O)(CNC(=O)CC3CCC=CCC3)C2)ncnc2ccsc12 66175,C1(C(N2CC=CC(NC(=O)C=Cc3ccncn3)C2)=O)CCC2(CCC2)O1 66176,c1(NC(c2ncccc2NC(c2ccnc(Cl)c2F)=O)=O)cc(Cl)cc(Cl)c1Cl 66177,C1(NC(=O)C=Cc2ccsc2)(CF)CCN(C(C2CCC(=O)N2)=O)C1 66178,N1(C(c2ccc(C#N)cc2)=O)C2CCC1CC(CNC(=O)C(F)n1cccn1)C2 66179,C1(C(=O)NC2C=CC(CC(=O)N(CCCC)C3CC3)C2)C2CC3C(C2)C13 66180,N1(C(CC2CCN(C)C2=O)=O)C2CCC1C(F)C(NC(c1ccc(Cl)cn1)=O)C2 66181,CCC(CC(=O)NC1(CC2CCC2)CC1)NC(C1(Cl)CCCCC1)=O 66182,N1(C(CCOC(C)C)=O)CC(CNC(=O)CNC(=O)C(F)(F)F)CC1C 66183,c1(C(=O)NC2C(NC(CCc3nc(C)sc3)=O)CC2)ccccc1OCCF 66184,C1(C(=O)NC2CC(CCC(=O)N(C(CC)C(=O)OC)C)C2)OCCCC1(C)C 66185,C1(CC(=O)NCCCN(C(c2coc(C3CCCCC3)n2)=O)CC)COC(=O)N1 66186,C1(CNC(=O)CC2CCC2)CN(C(c2cn(CCF)nn2)=O)CC(C(F)(F)F)O1 66187,Cc1noc(N)c1C(N1CCC1CNC(=O)Cc1ccc(F)nc1)=O 66188,C(CC(C)C(=O)N1CCC(NC(=O)CC2CC(SC)C2)C1CC)=CC 66189,N1(C(C2(OC)CCCCC2)=O)CCCC2(C1)CN(C(=O)CC1=CCCC1)C2 66190,Cn1nc(C(=O)NCC2CCC2C(=O)NC(CC(N)=O)C2CC2)cc1F 66191,N1(CC(=O)NC2C(CNC(CCC(C)(F)F)=O)C2)C(=O)NC2(CCOCC2)C1=O 66192,N1(C(CCC(=C)C)=O)CCCC12CCN(C(=O)Cn1cc3ccccc3n1)CC2 66193,CC(C)(C)C(C#N)C(=O)NC1COCCC1NC(c1cnc(S)n1C1CC1)=O 66194,C1(CCC(=O)OC)CC(CO)N(C(=O)Cc2ccc(C(=O)O)cc2)C1 66195,C(=O)(C1=NOC(C)C1)NCCC1(C(N(C)Cc2nc(C)sc2)=O)CCC1 66196,n1(CC(N2CCC(O)(C(C)NC(c3cocn3)=O)C2)=O)cnc2sccc2c1=O 66197,N1(C(CCc2scc(C)n2)=O)CC(NC(=O)C(c2ccccc2Cl)O)C(C)(C)C1 66198,N1(C(C(COC)O)=O)CC2CCC(C1)N2C(c1cc(-c2ccc(O)nc2)on1)=O 66199,N1(C(Cc2c(C)ocn2)=O)CC2(CCN(C(=O)C(c3ccc(O)cc3)(C)C)C2)C1 66200,N1(C(=O)CCC2CCC2)CCCC2(CCN(C(c3ccc(O)nc3Cl)=O)CC2)C1 66201,CC1COc2c(C(=O)N(CCCCN(C)C(C3C=CCCC3)=O)C)cccc21 66202,C1(C(=O)NCC(CO)NC(c2c(COC)nn[nH]2)=O)CC2C(C1)C2(F)F 66203,c1(OC(C(=O)NCCC2(O)CN(C(CC#C)=O)C2)C)ccccc1Br 66204,C(N=c1[nH]c(C(F)F)nc(=N)[nH]1)C1C(C)CCN(C(c2cc(Cl)ncc2Cl)=O)C1 66205,CC#CCCCC(=O)N1CCC1CC(=O)NCC1(OC)CCC1 66206,N1(C(CSC)=O)CC(C(=O)N(C)Cc2ccsc2)C(C)C1 66207,C1(OCC)CC2(C1)CC2C(=O)NCC(C)CN(C)C(c1sc(C2CC2)nc1C)=O 66208,c1(OC)ccc(CNCC2OCC2(C)C)c([N+](=O)[O-])c1OC(C)=O 66209,c1(NC(=O)NC2CCCC(Cc3cn(CC)nc3)C2)cncc(C#N)c1 66210,c1(CC2(C(N(CCNC(=O)CC3CCC3C)CC)=O)CC2)cnn(CCO)c1 66211,c1(NC(C2C3CN(C(Cc4c(C)noc4C)=O)C2C3)=O)cnc(C#N)nc1 66212,c1(C(CC)C)nc(C)cc(=NC2CC(NC(=O)CC3CC4CCC3C4)C2)[nH]1 66213,C1(N(C(=O)CCNC(=O)CO)C)CCCN(C(=O)Cc2cnn(C)c2)CC1 66214,N1(C(=O)NCc2cc(OC)cc(F)c2)c2cccc(O)c2CCC1C 66215,N1(C(C2(CC#C)CCOC2)=O)CC2CC(NC(c3c[nH]cc3C3CC3)=O)CC1C2 66216,Cc1[nH]nc2c1CC(C(N1CCC(CO)(NC(=O)Cn3cccn3)CC1)=O)CC2 66217,n1(CC=C)nnnc1C(CC(C)C)NC(C)CC(=O)Nc1ccccc1 66218,C12(CCNC(COc3c(C(C)C)cccc3)=O)CCC(C1)N(C(C1CCC1)=O)C2 66219,c1(CC(C(=O)N(CCCNC(C2C(OCC)C2)=O)CC)O)ccccc1Cl 66220,c1(CN2CCN(CC(CC)NC(c3ccc(F)cc3)=O)CC2)ncc(Cl)cc1Cl 66221,C1(CN(CCO)CC2(OCC)CCCC(C)(C)C2)Cc2ccccc2C1C 66222,CCCC(CC)CCC(=O)N1CCC(N(C)C(c2cc(N)ccc2O)=O)C1 66223,c1(C(=O)NC2C(C)N(C(c3cnc4sccn34)=O)CC2)ccc([N+](=O)[O-])s1 66224,CC1CC2CCC(C(=O)NCC3(Nc4ncc(Cl)c(O)n4)CC3)CN2C1 66225,c1(C(N2C(C)CCC(NC(=O)CC=C(Cl)Cl)C2)=O)ccn2nccc2n1 66226,c1(C(=O)OCc2cc(F)ccc2F)cnc2c(cnn2Cc2ccccn2)c1 66227,c1(C(N2C3(CNC(C(C)=CC)=O)CCC(CC3)C2)=O)cnc2c(c1)N(C)CCO2 66228,c1(CC(=O)NCC2C(NC(c3cncc(C)c3Cl)=O)C2)cccc2nsnc12 66229,N1(C(C(C2CCOC2)OCC)=O)C2CCC1CC(CNC(C1CC(F)(F)C1)=O)C2 66230,CC1CN(C(c2ncncc2Cl)=O)CCC1CNC(C1CC2(CC2)C1)=O 66231,CC1CCCC(OCC(=O)NC2CCC2Cn2cc(-c3ccccc3Cl)nn2)C1 66232,N1(C(C(F)=C(C)C)=O)CCC(C(F)(F)F)C(NC(=O)C=C2CCN(C)C2)C1 66233,Cc1cnccc1C=CC(=O)NCC1(CN(C)C(c2cc(O)n(C)n2)=O)CC1 66234,Cc1cc(C(=O)NC2(C)CC(C(=O)NCc3ccc(C)s3)C2)nc(O)n1 66235,C(=O)(C1=C(C)CCC1)N(C(C(N1CC(CCC#C)C1)=O)C1CC1)C 66236,C1(NC(CCCOC)=O)CCC(NC(C23CC(CN2C2CC2)C3)=O)CC1 66237,C12(CNC(C(C)(C)OC)=O)CCCN(C(=O)C=Cc3cccc(F)c3)C1C2 66238,C1(C(N(CCC(=O)OCC)C)=O)CC2CCN(C(C34CC(CO)(C3)C4)=O)CC12 66239,C1(C#N)(C(=O)NCC(CC)(CC)NC(=O)Cc2cc[nH]n2)CC2C=CC1C2 66240,C1(CNC(=O)NCC23CCC(CC2)O3)CC12CCCOC2 66241,C1(C)(C(=O)NC(CN(C(c2ccccc2SC)=O)CC)C)CC(OC)CN1C 66242,C1(NC(=O)OC(C)(C)C)CN(Cc2cc(Br)cc(Br)c2O)CC2(CCOCC2)C1 66243,CN1CCCCN(C(c2cnc(C(C)(F)F)s2)C(=O)NCCC2(C)CC2)CC1 66244,C1(NC(c2nc(CCCCC)sc2)=O)CCCC(N(C)C(c2ccnn2C)=O)C1 66245,N1(C(c2nc(C(C)C)sc2)=O)CCC2CCN(C(C3(C)CC3C)=O)CC12 66246,C#Cc1cccc(C(=O)NCC2CN(C(c3cccc(Cl)c3)C)CCO2)c1 66247,c1(CN(C(COC)C)CC(C2CC=CCC2)O)ccc(Cl)s1 66248,c1(C(=O)NC2CC(F)(CNC(CCC)=O)C2)cnc(C(F)(F)F)c(F)c1 66249,C1(NC(C=C(CC)C)=O)CN(C(=O)CC2(C)CCCC2)CC1(C)C 66250,c12cc(F)c(F)c(c1F)NC2c1nnnn1CCCF.C1(C)(CSC)CCOC1 66251,CC#CCCC(=O)NC(C)(CNC(=O)CSCC1CCCO1)C(C)C 66252,C(=O)(CC(O)CC(C)(C)C)N1CC(C#C)N(C(c2ccnc3ncnn23)=O)CC1 66253,CCC(O)C(F)(F)C(=O)NCC(CCNC(C1(n2cc(C)cn2)CC1)=O)OC 66254,C1(NC(c2cc(C(=O)OCC)no2)=O)CCCC(NC(c2cc(C(C)C)no2)=O)C1 66255,N(C(=NCCCN(c1sccc1C)C)N1CCCC(Nc2ccccc2)C1)CC 66256,CCCC(C)CCCC(=O)N(CC(C)NC(C1(c2cccs2)CCCC1)=O)CC 66257,CN(C#N)C(=O)CNC(C1CCC1CNC(C1CC1(C)C)=O)=O 66258,C1(CNC(CC(CC)NC(c2cnc(=N)[nH]c2)=O)=O)OC(=O)CC1(C)C 66259,C1(NC(=O)NCC(C(C)C)c2ccccc2)CC2(C1)CC21CCC1 66260,C(C(O)C(F)F)NC(CCNC(c1cncnc1)=O)=O 66261,c1(C(=O)NC2CCN(C(c3c(C)[nH]cc3)=O)C2(C)C)ccc(Br)c(F)c1F 66262,c1(C(=O)NCC2(C)C(NC(c3c(OC)csc3)=O)CCC2)cc2c(Cl)cncc2o1 66263,c1(C(=O)NCC=CCNC(C(C=C)O)=O)ccccc1C1CC1(F)F 66264,C1(O)(C(N(C2CCN(C(=O)C(CNC(C)=O)N(C)C)C2)CC)=O)CC(C)(C)C1 66265,CC1CC(C)(C(=O)NC(C)CN(C(=O)CCCn2ccccc2=O)C)CC(C)O1 66266,c1(C(N(C2CCN(C(C(CCC)C)=O)CC2)C)=O)ccc2nc(C)n(C)c2c1 66267,C(=O)(CCCCC(=O)NC1CN(C(c2ccc(C(C)=O)c(F)c2)=O)CC1O)NC 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66581,C1(O)(CCNC(CC#N)=O)CCCN(C(c2cccc(C(F)(F)F)n2)=O)C1 66582,C(=O)(C(CCC(C)C)NC(C1CC2(CCC2=O)C1)=O)NCCN1CC=C(C)CC1 66583,N1(C(C(CC)n2cccn2)=O)CCC(O)(CN(C)C(C2CCC=CCC2)=O)C1 66584,N1(C(Cc2nc(C)sc2)=O)CC(NC(=O)CCC(=O)c2ccc(O)cc2)C(C)C1 66585,c1(C(N2CCOC(C3CCCO3)C2)C(=O)NCCOCC)cnc(CC)nc1 66586,Cc1cnn(CCCNC(=O)C(CNC(=O)C=CC(=O)OC(C)(C)C)N(C)C)c1 66587,c1(-c2c(C)c(F)ncc2)cccc2c(C(=O)NC(CO)C(C)C)n[nH]c12 66588,C12(C(=O)NCC(C(C)C)(C)NC(c3cscn3)=O)CCCC1CC(=O)C2 66589,CC1CC(C(=O)OC)CN1C=O.c1(NC(N)=O)ccccc1OC(C)(C)C 66590,C#CCC(CC(=O)OC)NC(=O)C(CNC(=O)C1=C(Cl)CCC1)CCC 66591,c1(SCCNc2n(CC=C)c(O)nc(=O)c2)c(OC)ccc2ccccc12 66592,c1(C(N(C)CC2(NC(Cc3c(C)nc(C)s3)=O)CC2)=O)ccc2oc(O)nc2n1 66593,c1(NC(c2ccc(OC)s2)=O)cn(C)c(C(=O)NCC2CC(F)(F)C2)n1 66594,c1(C(=O)NCC(CCNC(C2(COC)C=CCC2)=O)O)cnc2cccnn12 66595,CC1CC(NC(=O)C(C)NS(C)(=O)=O)CN(C(=O)CC=Cc2ccc(F)cc2)C1 66596,C(=O)(C(C)(CO)NC(c1cc(Cl)cs1)=O)NCCN(CC(F)F)C 66597,CC(C(=O)NC1CN(C(=O)CCCOCc2ccccc2)C1)S(N)(=O)=O 66598,CCC(CC(=O)N1CC(CNC(=O)CN2CC3C=CC2C3)CC1C)C1CC1 66599,c1(NC(C2C(C)C2c2cccs2)=O)ccccc1SC(F)F 66600,c1(C(c2n(CCOC)nnn2)NC2CCOCC2(C)C)cnn(C)c1S(C)(=O)=O 66601,C1(NCn2c(C)cc(C)n2)CN(C(=O)Nc2ccc(C(N)=O)cc2)CC1(C)C 66602,CCC(C)CC(=O)NCC(N1CCN(C(c2cc(C)n(CC3CC3)n2)=O)CC1)=O 66603,Cc1ccc(C(N2CC(C(C)NC(c3nc(F)ccc3Cl)=O)C2)=O)c([N+](=O)[O-])c1 66604,c1(C(N2CCCC(N(C(=O)C(O)P(C)(C)=O)CC)C2)=O)ccc2oc(=N)[nH]c2c1 66605,c1(C(=O)NC2COCC2NC(=O)C(O)CC2CCOCC2)cccc(C2CC2)c1 66606,C(CCC(=O)NCC1CC1CNC(=O)C(C)Cn1cccn1)NC(C)=O 66607,C1(N(C(C(C)OCCOC)=O)C)CCCC2CN(C(=O)CCc3cccs3)CC12 66608,C12C(CCN1C(=O)CCCn1cncn1)NC(=O)C2.C1(C(C)(C)C)CCC1(C)C 66609,N1(C(CC23CC(C)(OC2)C3)=O)CCCCCC(NC(c2scnc2C2CC2)=O)C1 66610,C1(OC)CCCN(C(C2CCN(C(c3c[nH]c(=N)o3)=O)C(C)C2)=O)CC1 66611,C(CC(CC)C(=O)NC12CCC1CN(C(=O)Cc1ccc(OC)nc1Cl)C2)=CC 66612,N1(C(C2(C)C(C(=O)OC)CC2)=O)CCN(C(c2cnns2)=O)C(CCO)C1 66613,Cc1cccc(C(=O)NCC(C2CCN(C(=O)C(O)C(C)C)CC2)(C)C)n1 66614,N1(C(C23C(CN(c4c(C)cncn4)C2)C3)=O)CCC(O)(CF)CC1 66615,C1(CNC(C(C)NC(N)=O)=O)CN(C(=O)CC2(C#N)CC2)CCC12CCOCC2 66616,C12(CNC(CCOCCOC)=O)CSC(C1)C2 66617,c1(C(=O)NC(CCNC(COCCC#C)=O)C)cc(Cl)cc2ccccc12 66618,C(C)(C(=O)NC1(C(=O)NC2C(CCOCC)CC2)CSC1)OCCOC 66619,Cc1nc[nH]c1CC(O)C(=O)N(CC(C)N(C)C(c1cn(C(C)C)nn1)=O)C 66620,C1(NC(C(CCSC)O)=O)CC2CCC(C1C)N2c1ncnc2onc(C)c12 66621,c1(NC(C2(C)CCN(C(=O)C(=O)Cc3ccc(O)cc3)C2)=O)ccc(Br)nc1Br 66622,N1(CCN2CCCC(C(=O)OC)C2)CC(=O)CCC1=O 66623,c1(CN(C)C)ccoc1C(=O)NCC(CNC(=O)Cn1cccc1)CO 66624,C1(C)(CC)CCN(C(C2CCCCC2(C)NC(=O)CN=[N+]=[N-])=O)CC1 66625,C1(C(N(CCNC(c2c(C)occ2)=O)C)=O)CN(C)CC1c1ccccc1 66626,C1(CNC(CC2CCCC(C)C2)=O)CC(C)(C)CN1C(=O)CC1C=CCC1 66627,N1(C(c2c(C)n[nH]c2)=O)CCN(CCN(C)C(C2CCC(=O)C2)=O)CC1 66628,c1(C(N2Cc3cnn(CCO)c3C2)=O)cc(Br)cc(F)c1F 66629,C(=O)(CC(C(F)(F)F)c1ccon1)NCCCNC(C1=NOC(C)C1)=O 66630,c1(CC)[nH]nc(C(N2CC(OC)C(NC(c3ccc(CC)[nH]3)=O)C2)=O)c1[N+](=O)[O-] 66631,c1(C(=O)NCc2c(C(N3CC(C)C(F)C3)=O)c[nH]n2)ccc2c(c1)CC2 66632,CC1CCOC(C(=O)N(CC(=O)NC(C(N)=O)C2CCCC2)C)C1 66633,C1(CNC(C(C)NS(CC)(=O)=O)=O)CCC(F)(CNC(=O)CCCSC)CC1 66634,C1(C(N2CCC(C)(O)C2)=O)CC2(CCN(Cc3cc(F)c(F)cc3Cl)CC2)CO1 66635,c1(N(C(CN(CCC(N)=O)CC)=O)Cc2ccccc2)cc2scc(C)c2[nH]1 66636,c1(OCC)ncc(C(=O)NC2CCCC2CNC(c2coc(N(C)C)n2)=O)s1 66637,C(=O)(C(C)CCCC(C)C)N(CC(CC)NC(=O)CC1CC(=O)NC(=O)C1)C 66638,CC(C)CS(=O)(=O)N1CCSC(C(N2C(C)CCC2C)=O)C1 66639,N1(C(c2cccc(C(=O)NC)c2)=O)C2CCC1CN(C(=O)C1=CC(C)(C)C1)CC2 66640,OCCCCN=c1[nH]c(=NCC2C3COCC23)c2c(F)cccc2[nH]1 66641,C12(CNC(C3N(C)C(=O)NC3)=O)CCC(CC1)N2C(=O)C=C1CCCCC1(C)C 66642,C1(NC(C(CCC)O)=O)CCCCCN(C(=O)C(=Cc2ccccc2)OC)C1 66643,N1(C(CNC(=O)OC)=O)CCC2(CC1)CC(C)N(C(c1cnc(O)cc1O)=O)C2 66644,C1(CNC(CC(C(C)C)C)=O)COC(C)(C)CN1C(c1cc(O)cc(O)n1)=O 66645,C1(C(N(CCCC)C2CC2)=O)CCC(C)(C)N(C(=O)CCOC(C)=O)C1 66646,Cc1ccn(CC(C)(O)C(=O)N(CC(C)NC(c2ccco2)=O)C)c(=O)c1 66647,c1(CC)cc(C(N2CCCC2CC)C(=O)Nc2ccc(F)cc2)cc(F)c1 66648,S(=O)(=O)(c1cc(C)c(Br)cc1C)N(CC1CC2(CC(OCC)(OC)C2)C1)C1CC1 66649,C#Cc1cnn(C)c1C(N1CCCC(C(=O)NCCC(C)CCO)CC1)=O 66650,C1(C)(CC)CC(NC(C23CC2CN(C(C2CCCC2F)=O)C3)=O)CCO1 66651,c1(C(=O)NC2C(CNC(c3cc(C4(C)CC4)on3)=O)C2)sccc1S(C)(=O)=O 66652,N1(C(=O)CSC(F)(F)F)CCN(C(C2(CCF)CC2)=O)CC(O)C1 66653,C1(NC(c2c(OC)csc2)=O)CN(C(c2cnc(C)[nH]2)=O)CC1O 66654,C1(C(=O)NCC2(C)CCCCC2)CCc2nc(-c3ccc4ccoc4c3)sc2C1 66655,C1(NC(C2C(CC(C)C)C2)=O)CC(C(F)C(=O)NCCCCN2CCCC2)C1 66656,N1(C(c2n(CC)ncc2)=O)CCCC(CC(=O)NC(c2ccc(C)cc2)C)C1 66657,C1(NC(C2CN(C)C(=O)CC2)=O)CCN(C(=O)CCC2CCCO2)CC12CCC2 66658,C1(NC(c2ccnc(Cl)c2)=O)CN(Cc2cccnc2O)CC1(F)F 66659,c1(OC)ccc(CN)cc1-c1ccc(C(=O)NCC2(N(C)C)CC2)o1 66660,CCCCC(C)N(C(=O)C(C)CN(C(=O)Cc1ccn(C)c1)C)C 66661,c1(C(=O)NC2(CO)CCN(C(=O)C(O)C3CCCC3)C2)ccc2ncsc2c1 66662,N1(C(COC(CC)C)=O)CCC(F)(CNC(C2CCC(C(F)(F)F)CC2)=O)C1 66663,Cc1cc(Cl)ccc1CC(=O)NCCC1COCCN1C(=O)Cc1cn(C)nn1 66664,C1(NC(CN(C(=O)Cn2c(O)nnc2O)CCOC)=O)CN(C)NC1=O 66665,Cc1c(C(=O)NC2CCC(c3cn(C4CCOCC4)nn3)CC2)cccc1C1CC1 66666,Cn1cc(C(N2CCC(C)(CNC(c3nsnc3O)=O)C2)=O)ncc1=O 66667,N1(C(CN2CCC(C)(C)C2)=O)CC2(NC(=O)COC3(C)CCCC3)CCC1CC2 66668,C(=O)(C(=O)N=c1ccn(C2CCCCO2)[nH]1)Nc1c(OC(C)(C)C)cccc1 66669,CC1(C)CCCCC(C(=O)NC2CCCN(C(c3cncc(O)c3)=O)C2)C1 66670,C1(C(N2CCCC2c2cc(C3CC3)on2)=O)CCCC2CC12 66671,Cc1cc(C(N2CCOC(CNC(C3CCN(C)C3C)=O)C2)=O)c(C)n1C(C)C 66672,c1(C(C)C)cccc(CC(=O)NC(CNC=O)C2CCC2)c1.C(=O)(C(C)N(C)C)N 66673,N1(C(C2(C)CCC(C)C2)=O)CC(C(=O)NC(C)(C)C)C2(CCC2)C1 66674,C1(S(C)(=O)=O)(C(=O)NC(C2CCN(C(C=CCC)=O)C2)C)CCOCC1 66675,Cc1cnc(O)c(CNC(c2cn(CCNC(C3(C)COC(=O)N3)=O)cn2)=O)c1 66676,c1(NC2CCCN(C(C3CC4(C3)CC4(F)F)=O)C2)ncc([N+](=O)[O-])cc1Br 66677,C1(NC(C2(COC(C)C)CC2)=O)C=CCN(C(=O)C(c2cccc(Cl)c2)C)C1 66678,N1(CCC)CC(C(=O)N(CCCCNC(c2ccc(C(=O)OC)[nH]2)=O)C)CC1=O 66679,c1(C(=O)NCc2cccnc2I)ccc(C(F)C(F)(F)F)cc1 66680,N1(C(C(CC)OCC)=O)CC2CCC1C(CNC(c1cc(C3CC3)[nH]n1)=O)C2 66681,CCC(CC)CC(=O)N1CCN(C(c2csc(-c3ccccc3)n2)=O)C2CC12 66682,c1(C(N2CCC(O)(CN(C(=O)CSC(C)(C)C)C)CC2)=O)cc2ccncc2s1 66683,N1(C(CC2(SC)CCC2)=O)CCCC(C(C)C(=O)NC(C2CC(SC)C2)=O)C1 66684,C1(S(N)(=O)=O)(C(=O)NCC(CNC(CC(C)c2ccncc2)=O)O)CC1 66685,N1(c2cc(NCCN3CCCCC3CO)nc(C)n2)CCCc2sccc2C1 66686,C1(NC(C2C(C)CCS2)=O)CCC(n2cc(-c3ccnc(C(=O)O)c3)nn2)CC1 66687,c1(N2CC3CN(CC)CC3C2)nc2c(c(=NC3C=C(C)CCC3)[nH]1)COC2 66688,c1(SCC)ccc(Cl)cc1C(N1CC2C(CNC(C3CC3C(=O)OC)=O)C2C1)=O 66689,n1(CC(=O)NCC(CCNC(C2(CC)CC(C)(C)C2)=O)O)nnc2c1CCCC2 66690,N1(C(c2c(C)ccc(C(F)(F)F)c2)C(=O)NC2CC2)CCCNC(=O)C(F)(F)C1 66691,c1(C(N2CCN(C(C(CC)C)=O)CC2COC)=O)cnc2ncnc(O)c2c1 66692,c1(C(N2CCC(CNC(c3nnn(C)c3N)=O)C2(C)C)=O)ccc2ncsc2c1 66693,Cc1cc(N)cnc1C(=O)NCCNC(=O)CCC1CC(C)(C)CO1 66694,CC1SCCCC1C(=O)N(CCNC(c1cnc(O)s1)=O)CC1CC1 66695,C=CCC(C)(C)C(=O)NC1CC(CC(N2CCC3CC23C)=O)C1 66696,c1(C(C)(C)C)c[nH]cc1C(N1CCC(Cn2cc(C3(O)CSC3)nn2)C1)=O 66697,C1(NC(C2(CSCC)CC2)=O)CN(C(=O)C(CC)OCC)CC(C)(C)C1 66698,c1(OCC)cc(-c2cccc(NC(c3cnn(C(C)(C)C)c3)=O)n2)ccn1 66699,CCCC(C(=O)OC)C(=O)NC(C)CN(C(=O)C(c1cccc(C)c1)C)C 66700,N1(C(C(CNC(COC(CC)CC)=O)CC2CC2)=O)CCC(N(C)OC)CC1 66701,N1(C(C(COCC)(C)C)=O)CC(CNC(C23CC(C)(CO2)C3)=O)CC(C)(C)C1 66702,C1(O)(C(C)C)CCCN(C(C2CCCCN2C(C2(F)CCCCC2)=O)=O)C1 66703,CC1(C)C(NC(=O)Cn2cnnc2)CC1C(=O)NCC(Cl)C(C)(F)F 66704,Cc1cc(C(=O)NCC2CCC(C(=O)N(C(C)CCC(C)C)C)C2)c(C)s1 66705,C(C(C)C)(C(O)C(=O)NC1CCCC(C(N2CCC(O)C2(C)C)=O)C1)OC 66706,c1(OC(C)C)ccc(Cl)nc1C(=O)N(CCC(C)NC(=O)C1=NOCC1)C 66707,C1(NC(C(C)NC(=O)NC)=O)CN(C(=O)C(F)OC(F)(F)F)CC2(CCC2)C1 66708,N1(CC(=O)NC(C=CC(=O)NC(c2ccnc(O)c2)C)(C)C)C(=O)CNC1=O 66709,C1(NC(CCCc2n(C)cnn2)=O)CCN(C(C2CC3(CCC3)C2)=O)CC1F 66710,c1(C(N2CC(CNC(CCCCCOC)=O)C(F)(F)C2)=O)c[nH]c2ccncc12 66711,C1(NC(c2ccc(C=C)cc2)=O)CCN(c2ncc(C(N)=O)cc2Cl)C12CCC2 66712,N1(C(c2n(C)c(C#N)cc2)=O)CCC2(CC(NC(=O)C(C)(C)c3cnsc3)C2)C1 66713,N1(C(C(C)(C)C2CCCN2C(=O)C(Cl)Cl)=O)CCCC(CCO)CC1 66714,c1(C(N2CC(OCC)(CNC(C3CN(C4CCC4)C3)=O)C2)=O)ccc(C)cc1 66715,c1(-n2cc(C(C)(C)NC(C3CCCC3O)=O)nn2)ccc(I)c(Cl)c1 66716,C(C(C)(C)C(=O)N(C)CC1CCCN1C(C1CN(C(C)C)CCO1)=O)NC(C)=O 66717,N1(C(C(C=CC)O)=O)CCN(C(C2(CC(=O)NC)CCCC2)=O)CC1CCO 66718,c1(N2CCC(NC(C34CCCN(CC3)C4)=O)C2)nc2ccccc2o1 66719,CCC(CC(=O)NCC(c1ccc(CO)cc1)NC(C1CSCCS1)=O)C(C)(C)C 66720,c1(C(=O)NCC(CO)NC(C(C)OCC)=O)ccc2ccc(Br)cc2c1 66721,c1(C(c2nnnn2CC=C)NCCCOC=C)ccc(OC)c(C)c1 66722,CON=Cc1ccc(C(N2CCC3CN(C(=O)Cc4cc[nH]c4)C3C2)=O)cc1 66723,C(=O)(N=c1[nH]c(Cl)ncc1O)c1c(CNc2c(C)cc(F)c(C#N)c2)cccc1 66724,N#Cc1ccc(CCC(=O)NC2(C(F)(F)F)CCCNC2)cc1 66725,c1(CC(=O)N(C(=O)C(C)(C)CF)C)ccccc1CNC(=O)C(C1CC1)C1CC1 66726,Cc1cc(C)c(C(N2CC(C(C)NC(=O)C(C)S(C)(=O)=O)C2)=O)c(=O)o1 66727,c1(C(=O)NC2(C)CC(NC(c3c(OC)c[nH]n3)=O)C2)ccc(C)c(Cl)c1 66728,c1(C(N(C(CNC(c2cnn(CC)c2C)=O)C)C)=O)cnc2ccc(Br)cn12 66729,CC(C)CC(C(=O)NCCOCCCN(C(=O)C(O)C(C)C)C)N(C)C 66730,C1(C)(CNC(C(C)NC(=O)NC)=O)CCN(C(C23CC(CO)(C2)C3)=O)CC1 66731,N1(C(c2cc(OC)cc(C)n2)=O)CCC(C)N(C(=O)CC2CCCCN2C)CC1 66732,C12(CCNC(C(C)OC)=O)CCC(C1)N(C(=O)CCC(=O)c1ccc(C)cc1)C2 66733,C(C(C(=O)NC(C(N1CC=C(C)C1)=O)c1ccoc1)N(C)C)OC 66734,C(=O)(C1=CCCN(C(c2ccc(C#N)cc2)=O)C1)NCC=CCOC 66735,c1(N(CCNC(c2ccsc2CO)=O)C2CC2)nccc(Cn2cc(Cl)cn2)n1 66736,Cc1nc(C2CCC2)oc1C(=O)NC(C)(C)CNC(C1(C#N)CC1C)=O 66737,CC1(C)C(NC(=O)C(C)(C2CCC2)NC(=O)COC2CCCOC2)C1(C)C 66738,N1(C(C2CCCC2C)C(=O)NC2CC(C3(C)CC3)C2)CCCC(C2(C)CC2)C1 66739,C1(O)(C(N2CCCC(CNC(=O)CCc3ccsc3)C2)=O)CN2CCC1CC2 66740,CCC(C)CC(=O)C(=O)N(CC(C)NC(=O)Cc1cccnc1O)C 66741,Cc1nnc(=NCC2CCCN2C(=O)C(C)C(C)C)[nH]c1C 66742,c1(COC)cc(CSc2ccccc2OCC2CCOC2)ccc1F 66743,N1(C(C(C)=C(C)C)=O)CCC(F)(F)C(CNC(c2cnoc2-c2ccco2)=O)C1 66744,CCC(CCCO)NC(c1conc1C(C)NC(=O)Cc1ccoc1C)=O 66745,C1(C(N2CC(N(C)C3CC3)C2)=O)CN(C(C2(F)C(C)(C)C2(C)C)=O)CC1C1CC1 66746,n1(CC)nc(C(=O)NCc2nc(C(N3CCN(C(C)CO)CC3)=O)co2)cc1C 66747,N1(C(Cc2c(C)ncnc2C)=O)CC2(CC(NC(=O)C(C)O)c3nccn32)C1 66748,N(C(=NCCF)N1CCC2(O)CCOCC2C1)CC1(C)CCCCC1 66749,CC1CCCCN1S(=O)(=O)N1CC(C(=O)OC)(CO)C1 66750,c1(C(N2CC(C(=O)OC)C2)=O)ccc(CN(C)Cc2cnn(C)c2C)cc1 66751,c1(C(=O)NC2CCCN(C(C(=C(C)C3CC3)F)=O)C2C)c(Cl)cccc1[N+](=O)[O-] 66752,C1(NC(c2nc(CC)oc2)=O)CCC2CCN(C(c3cnoc3C3CC3)=O)C1C2 66753,CC1CCC(NC(c2cnn(C)c2)=O)CN1C(=O)C=Cc1ccc(C(N)=O)cc1 66754,c1(C(N2C(C)CC(NC(c3cnc(O)o3)=O)C2)=O)cc(Br)c(C#N)s1 66755,C1(CNC(c2cc(C(F)(F)F)no2)=O)CC2C(O)CC2O1 66756,CC12CCCC1N(C(c1cnc(C(F)F)nc1)=O)CCN(C(c1ccsc1)=O)C2 66757,Cc1cc(C(=O)NC2CCN(C(C3CS(=O)(=O)C3)=O)CC2C)nc2[nH]nc(O)c12 66758,C1(C)(C(=O)NCC2C(C(=O)NCC(C3CCCCC3)C)CC2)CC(F)C1 66759,C#Cc1cccc(C(=O)C(C)=O)c1.C12(CC(c3cn(CC(O)C)nn3)C1)C(=O)N2.OC 66760,C1(C(=O)NC2(C)CN(C(c3cc(F)cc(Cl)c3O)=O)C2)Cc2ccc(F)cc2O1 66761,c1(C(=O)NC(CC(C)NC(=O)CSc2nccn2C)C)ccc(CCF)cc1 66762,Cc1c(C(=O)NC2CC(NC(C3CCCC34CC4)=O)C2)oc2ccc(Br)cc12 66763,N1(C(c2c(C)[nH]cc2-c2ccccc2)=O)CCCC(NC(c2csnn2)=O)C1C 66764,c1(C(N2CC(CNC(C(Br)=C(C)C)=O)C3(C2)CC3)=O)cc2cccn2cn1 66765,N1(Cc2nc(-c3ccc(OC)cc3)on2)CC(CO)OC2(CCC2)C1 66766,c1(C(=O)NCC2C(C)CN(C(C3CCOC3)=O)C2)nc2ccccc2cc1Cl 66767,C1(C(CNCC(C(CCC)=O)=O)(C)O)CCN(C(=O)C#CC2CC2)CC1.C(=O)(C(C)C)O 66768,c1(CNC(C2(C)CCN2C(c2cc(Br)co2)=O)=O)cccc(F)c1Br 66769,c1(C(CNC(C2(C)CC=CCC2)=O)NC(C(CO)OC)=O)ccccc1F 66770,c1(CC)nc(=N)[nH]cc1C(=O)NC1CCN(C(=O)C(F)C(C)(F)F)C1 66771,CC(CC(F)F)C(=O)NC1CC2C1CCN2C(c1ncccc1Br)=O 66772,Cc1cc(C(N2CCC(Cn3cc(CN)nn3)C2)=O)c2c(c1)CCC2 66773,C1(NC(C2C(C)(CC)C2)=O)(COC)CCN(C(=O)C=Cc2ccc(C)nc2)CC1 66774,C(=O)(CCCC(C)NC(=O)CC1CCC(=O)C1)Nc1cc(C)sc1C 66775,C1(C(=O)NCCCCNC(C2SCCS2)=O)C2(CCC2)C12CCC2 66776,N1(C(CCC(C)SC)=O)CC2(C(=O)Nc3ccc4c(c3)OCC4)CCC1CC2 66777,c1(C(=O)NCC2CC(OC)CN2C(C2CC(SC)C2)=O)ccc2nc(C)nn2c1 66778,CC(O)CC(C)(C)CNC(C1(CF)CCN(C(=O)CC(=O)NC2CC2)C1)=O 66779,c1(C(=O)NCC2C(CNC(Cc3cnc(C)o3)=O)C2)cc2nn[nH]c2cc1F 66780,N1(C(=O)NC(c2nc(C3CC3)n[nH]2)C)CCC(C#CBr)CC1 66781,C1(NC(c2cc(C(F)(F)F)on2)=O)CC2CCC(C1)N2C(c1cccc[n+]1[O-])=O 66782,Cc1cc(C(N2CCC2C(=O)NCc2cc(Cl)ccc2O)=O)cc(O)n1 66783,C1(OC)CC(C(N2CCC(NC(c3c(C4CC4)cnn3C)=O)CC2)=O)C12CCC2 66784,C1(NC(C=Cc2n(CC)ncc2)=O)C(C)CCN(C(c2n[nH]c(=N)[nH]2)=O)C1C 66785,C1(OC)(CNC(c2cc(C(C)(C)O)ccn2)=O)CCN(C(C2(C)C=CCC2)=O)C1 66786,N1(C(c2c(-n3cc(CC(=O)O)nn3)cccc2)=O)CC2CC3CCCN3C2C1 66787,C(=O)(C1=CN=C2N=CNN2C1)NC1CCCN(C(CSC(C)C)=O)C1C 66788,N1(C(CCCC(C)NC(C2N(CC)CCCC2)=O)=O)CCC2CN(C)CC2C1 66789,c1(OC)cccc(C)c1C(=O)NCC1CN(C(=O)C(O)C(C)(C)C)CCO1 66790,Cc1ncc(C=CC(N2CC=CC2CNC(c2c(C)ccnc2O)=O)=O)c(O)n1 66791,CC1(C)C(NC(=O)NCc2nc[nH]n2)CC1CC(N1CCC(OC2CC2)CC1)=O 66792,n1(CC)c(S)nc2c(Br)cc(C(N3CCSCC3)=O)cc12 66793,C#CCCCC(C)C(=O)NC(C(=O)NC(CC1CC1)CO)C(C)O 66794,c1(C(=O)NCC2(O)CCN(C(C3C(CC(C)C)C3)=O)C2)ccc2c(c1)N(C)C(=O)C2 66795,C(=O)(CC(C(F)(F)F)OC)NC(CCNC(C1CN(CC)C(=O)CC1)=O)(C)C 66796,Cc1cc(NC2CC(NC(c3ccc(O)nc3)=O)C23CCC3)c([N+](=O)[O-])c(C)n1 66797,C(=O)(CC(O)CC1CC1)NC(CNC(C=CCC)=O)(C)Cn1cccn1 66798,C12(C(N3CCCC(CNC(Cc4ccc(CC)cc4)=O)C3)=O)CCCC1CCC2 66799,Cc1noc(C)c1CC(N1CSCC1C(=O)NC1CC(C(C)(C)O)C1)=O 66800,CC1(C)CCC(C(=O)NCC2(O)CCN(C(c3cccc(F)c3)=O)C2)CO1 66801,c1(Cn2cc(C(C)O)nc2)cc([N+](=O)[O-])ccc1Br 66802,CC(C)(C)C(=O)C(=O)N1CCC(C)(NC(=O)C(CCc2ccccc2)C2CC2)C1 66803,C1(CC(C(C)(C)C)=O)CN(N2CCC(NC(c3ccccc3O)=O)C2)C1 66804,c1(C(N2CC3C(NC(c4cc(C)c(N)cc4)=O)C3C2)=O)ccc2cccnc2n1 66805,Cc1nc2ccccc2n1CC(=O)NC(c1ccc(Br)cc1)C(F)(F)F 66806,C1(C(=O)NC(CC2CCCC2)C(=O)NC2C3COCC23)CC2(CCC2)CO1 66807,N1(C(C(C)O)=O)CC2(C1)OC1(C)CC2(NC(C2CCN3CCCC3C2)=O)C1 66808,N1(C(c2cnc(C)s2)=O)CC2CC(NC(C3CCCC(F)(F)C3)=O)CC1C2 66809,CC1(C)CC(C(=O)NC2(C(=O)NCC34CCCC3C4)CC(O)C2)=NO1 66810,N1(Cc2nn(C)c(=O)o2)CCCC(C)(CN(C(C2CCCCC2)=O)CC2CC2)C1 66811,C(=O)(CC(C(C)(C)C)NC(c1cnnn1C)=O)NC(c1ccco1)C 66812,C1(C(=O)NC(C)C(C)NC(=O)C=C(C)CN2CCOCC2)(OCC)CCCC1 66813,C1(C(N(C(C)CCNC(=O)C(N)=O)C)=O)C(c2ccncc2)C1(C)C.C1CC1 66814,c1(NC(C2CN(C(=O)CCc3ccnc(Cl)c3)C2)=O)ccc2scnc2c1 66815,c1(NC(C2CC(F)CN2S(=O)(=O)Cc2cc(Cl)cc(Cl)c2)=O)ncc(F)cc1Br 66816,C12(C(N3CCC(CN(C(c4ccc(CC)o4)=O)CC)CC3)=O)CCCC(C1)OC2 66817,C1(NC(c2c(CC)scc2)=O)CCN(C(c2ccccn2)=O)C(C)C1 66818,c1(CN(C(C)(CC(=O)O)C(C)C)CC)cc(Cl)c(Br)cc1F 66819,c1(C(N2CCC(NC(CC3CCCCC(=O)N3)=O)C2)=O)ccc(F)c2ccsc12 66820,S(=O)(=O)(c1ccc(C2OCCO2)cc1)NCC1(NC(=O)OC(C)(C)C)CC1 66821,C12(C(N3CCN(C(COC(CC)(C)C)=O)C(CF)C3)=O)CCCC(=O)N1CCC2 66822,C(=O)(C(C(C)Cc1ccc(CC#N)cc1)N1CCCC(C(F)F)C1)NCCOC 66823,CCCCCS(=O)(=O)CC(=O)N1CCCC(O)(Cn2cc(CO)nn2)CC1 66824,c1(C(N2CC(CNC(C(CC)OCC)=O)C(C)C2)=O)cc(F)ccc1C1CC1 66825,N1(C(C2CC(OC)(OC)C2)=O)CC2CC(NC(c3cncc(C4CC4)c3)=O)C1C2 66826,C(C(C)(COC)C(=O)N(CC(=O)NCCN=[N+]=[N-])C)OC 66827,C=C(C)C(C)(C)C(=O)N1CCN(C(c2c[nH]cc(Br)c2=O)=O)CC1 66828,CC1(C(=O)NCC(C)(CO)NC(c2ccc(F)cc2)=O)CC2CCC(C1)S2 66829,c1(NC(c2noc(C)n2)CC)ccnc2c(Cl)cnn12 66830,CC(C)(CNC(c1cc([N+](=O)[O-])c[nH]1)=O)CC(=O)NCCCOCC1CCC1 66831,C1(CC(=O)NCC(C)N(C(C)=O)C)CC2(CCC2)CN1C(=O)C=Cc1cocn1 66832,c1(Nc2ccc(NC(=O)NC(c3c(C)cccc3)=O)cn2)cc(F)cc(C)c1O 66833,C12(NC(C(C)OCC#C)=O)CCC(C1)N(C(=O)CCCC(=O)N(C)C)C2 66834,Cc1ccc2c(C(=O)NC3(C)CN(C(=O)CCn4c(C)csc4=O)C3)coc2c1 66835,C1(OC)CCC(CC(=O)NC(C)C(C)(C)NC(C2CC(=C3CCC3)C2)=O)CC1 66836,CC1CC(C(=O)N2CCC(O)(CNC(C3(F)CCCC3)=O)CC2)=NO1 66837,c1(CCC(=O)NCCC2CCCN(C(C(CC)F)=O)C2)nc2cnccc2[nH]1 66838,c1(OC)ccc(CN2CCOC(CC(=O)Nc3nccnc3Br)C2)cc1[N+](=O)[O-] 66839,C1(NC(C2(C(=O)OCC)CC2)=O)CCN(C(c2ccc(N(C)C)nc2)=O)C1C 66840,N1(C(c2ccc(C(CC)C)cc2)=O)CC(NC(c2nc(C)no2)=O)C(C)(C)C1 66841,c1(C(N(CC(O)CNC(C2CC(Cl)(Cl)C2)=O)C)=O)cc2ccccc2c(O)n1 66842,c1(OC)cc(NC(=O)C(=O)NC2C(C)CCCC2C)ccc1Cl 66843,c1(C(N2CC(O)(CCNC(C3(C)N(C)CC(O)C3)=O)C2)=O)ccc(N=[N+]=[N-])cc1 66844,c1(C(=O)NCCC2CC(NC(CCNC(=O)NC)=O)C2)ccc(Br)c(F)c1 66845,Cn1ncc(Cl)c1CC(=O)NC12CC1CN(C(C1CC1CF)=O)C2 66846,C(C)(CC(C)(C)O)NC(C(C)N(C(=O)C(c1ccnn1C)C)CCC)=O 66847,N1(C(CSCCC)=O)CCCC(CCC(=O)N)C1.N1(CCO)CCC(C)CC1 66848,N1(C(CNC(C(CC)CC)=O)=O)CC2CCCCN2CC1CNC(=O)C(C)=CC 66849,C(C(O)CC(=O)N(C1CC1C)C)NC(c1c(C)ocn1)=O 66850,c1(NC(COCCCCNC(C(C(C)C)OCC)=O)=O)ccc(C2CC2)nc1C 66851,CC(C)C(C(=O)N(CCCCNC(=O)CC1(C(F)F)CC1)C)N(C)C 66852,C(CC(C)C(=O)NCCCC1CCCN1C(=O)C(=O)NCC(F)F)=CC 66853,N1(C(C2C=CCS2)=O)CCC2CN(C(=O)C(N3CCCC3)C3CCC3)C2C1 66854,C1(CNC(Cc2nnc(C)o2)=O)CCCC2CN(C(=O)CN(C)C(C)C)CC12 66855,Cn1cc(CCNC(c2c[nH]nc2CNC(C2(n3cnnn3)CC2)=O)=O)cn1 66856,c1(OC)ccccc1-c1noc(C(C)SC2CCCC(c3ccc(Cl)cc3)C2)n1 66857,C1(C)(CNC(CN(CC)CC)=O)CCCN1c1nnc(CO)s1 66858,c1(OC)cc(C(N2CCC(NC(c3ccc(N)cc3Cl)=O)C2)=O)cc([N+](=O)[O-])c1 66859,Cc1cccc(O)c1C(N1CCCC(C)(NC(=O)CCC(F)F)C1)=O 66860,CC1CN(C(=O)C(Cl)=CCl)CC(C)N(C(c2ccnc3c2ccn3C)=O)C1 66861,C1(C(=O)NOC2CCOCC2)CCOCC1NCC(=O)OCC1CC2(CSC2)C1 66862,c1(C(N2C(C(=O)NCCCOC)C3C(C2)C3(C)C)=O)cccc([N+](=O)[O-])c1C 66863,CC1CN(C(C2CCCN2C(C23CCCN2CCC3)=O)=O)CCCO1 66864,N1(C(C(C)(OC)OC)=O)CCCC(F)(C(N2CCC2C2CCC2)=O)C1 66865,C(=O)(C1=CCCCC1C)N1CC2C(NC(c3c(C)nc(CC(C)C)o3)=O)C2C1 66866,c1(CNS(C)(=O)=O)ccccc1NC(=O)C(=O)NCCC1CCOC1 66867,N1(C(c2c(C)nc(CCC)o2)=O)CC2(CCCC2NC(C2CCCN2CC)=O)C1 66868,Cc1cc(C(=O)NC23CCC2CN(C(c2c(C(C)C)cnn2C)=O)C3)cc(F)c1 66869,C(=O)(CC(C(C)C)NC(=O)Cn1c(C)ccc1C)N(CC(=O)NCCC)C 66870,C1(NC(c2ccc(CN(C)C)[nH]2)=O)CC2C1CCN2C(=O)OC(C)(C)C 66871,Cc1nc(C(=O)NCC2CC(CNC(c3c(C)cnn3C)=O)CO2)n(C)n1 66872,CCCC(CC(C)C)C(=O)N1CCC(C(=O)NC(C)C(C)(C)COC)(CC)CC1 66873,Cc1cc(=NCCNS(C)(=O)=O)[nH]c(=NCCc2c(OC(F)F)cccc2F)[nH]1 66874,c1(OC)ncc(C(=O)NCCOCCOCCNC(=O)CCC(C)(F)F)nc1C 66875,CC(C)CC(O)CC(=O)NC1(Cc2ncc(F)cn2)CC1 66876,C12(OC)CCC1CN(C(=O)CC1CCN(C(=O)CCCC3CCCC3)C1(C)C)C2 66877,Cc1c(C(N2CCSCC2CCNC(C2CN(C)C2)=O)=O)sc2nccn12 66878,N1(C(CC2N(C(CCC(C)OC)=O)CCC2)=O)CCc2nc(C)[nH]c2C1 66879,c1(C(N(C2CCN(C(c3cnco3)=O)C2)CC#C)=O)nocc1C 66880,c1(C(=O)NCC2N(C(c3c(C)cc[nH]3)=O)C3CCC2C3)cc(Br)cc(C)c1F 66881,O=C(CCCCCO)Nc1nc(-c2ccc(O)nc2)cs1.C12CC(F)CN(C1)C2=O 66882,N1(C(CCCC#C)=O)CCC(C2CCCN(C(=O)CCC(=O)C(C)(C)C)C2)CC1 66883,N1(C(CC2CCC(=O)NC2)=O)CCN(C(c2cccc(Cl)c2F)=O)CC(CO)C1 66884,Cc1cccn(CC(=O)NCCCCCc2ccccc2Br)c1=O 66885,CN=c1ccc(C(N2CC(O)CC2CC(=O)NCC(=O)N2CCCO2)=O)c[nH]1 66886,O=C(CS(=O)(=O)C12CC(C1)C2)NCCCNC(c1sccc1-n1cnnn1)=O 66887,c1(NC(C2CC23CCN(Cc2c(F)ccc(Cl)c2Cl)C3)=O)nccc2[nH]ccc12 66888,CCCCCC(O)C(=O)NC(C1(O)CN(C(C2CN(C(C)=O)CCO2)=O)C1)C 66889,C1(C(=O)OC)CCC(C)(C(=O)NCCN(C(=O)CSCCC#N)C)C1(C)C 66890,C1(C(=O)NC(C)CC(=O)NCC(C)(C)NC(C2C=CCC2)=O)CCC(=O)N1C 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67015,N1(C(C(CCN(C)C)N(C)C)=O)CC2(CCN(C(=O)CC3CCOC(C)(C)C3)C2)C1 67016,C1(CC(=O)NC2CCCC(N(C(C3(CC)CC3)=O)C)C2)CN2CCN1CC2 67017,N1(C(c2cc(-c3ccccc3)co2)C(=O)NC)CCC(N(C)C)(CO)C1 67018,N=c1[nH]c2ccccc2cc1C(N1CCCC1C(c1ccccc1)O)=O 67019,C1(NC(C23N(C(c4cccc(C)c4)=O)CC(C2)C3)=O)CC1C1CCCCC1 67020,CC1(CNC(C2(C3CC3)CN(C(c3ccnc(O)c3F)=O)C2)=O)CCCCC1O 67021,N1(c2nnc(CC)s2)CC2CC(NC(c3ccn(CC(F)F)n3)=O)CC1C2 67022,c1(C(=O)Nc2nc(-c3ccccc3C(F)(F)F)cs2)ccncc1Cl 67023,C(C(F)(F)C(F)F)N(c1ccccc1F)C(C(C1CCC1)NC(=O)C1CC1)=O 67024,C12(NC(=O)CC(O)C3CC3)CCCC1(F)CN(C(=O)C(F)(F)C1CCCC1)C2 67025,N1(C(C2(F)CCC(C)CC2)=O)CCOC2(C1)CN(C(=O)CC1(C)CCOCC1)C2 67026,C(=O)(C1=NOC(C)C1)NCC1CC(NC(c2cccc(SCC#C)c2)=O)C1 67027,N1(C(CN(c2ccccc2)CC(=O)OCC)=O)CCCC(C)(C)C1CNC 67028,C1(CC)CC(C(=O)N(CC(CC)NC(=O)C=C(C)c2ccco2)C)CC(=O)N1 67029,N1(C(c2cc(SC)c(N)cc2)=O)CC2CCN(C(c3snnc3C(C)C)=O)C2C1 67030,c1(CNC(CNC(=O)CC2CN(Cc3cccs3)C2)=O)cccc(Cl)c1 67031,c1(C(=O)OC)cc(C(=O)NC2CCCCC2NC(=O)CCS(C)=O)n(C)n1 67032,N1(C(C2CC=CC(NC(C3=CC(C)(C)C3)=O)C2)=O)CCCC(C2(C)CC2)C1 67033,C(C)(CSC)(C(=O)N(CC(O)C1CC1)C)NC(CC1CC(CC)C1)=O 67034,N1(C(Cc2c(C)nsc2)=O)CCN(C(c2nocc2Br)=O)C2CC12 67035,C(=O)(C(CC1CCCC1)NC1(C)CC(C(=O)NCC(F)(F)F)C1)OC 67036,CCC(C)CC(C)C(=O)N1CC(CCNC(=O)CCOc2ccccc2Cl)C1 67037,C1(C(=O)Nc2ccc(C)cc2F)CN(C(c2cc(C#N)oc2C)=O)CC12CCC2 67038,c1(C(N2CCN(C(C3(F)CC4C=CC3C4)=O)CC2)=O)cc(F)c(F)c(F)c1F 67039,N1(C(CCc2cccc(C)c2)=O)CCCCC(NC(c2nn(C)cc2Br)=O)C1 67040,C1(C(N(CC(=O)N(CC(=O)NC)C)C(C)C)=O)COCCN1C 67041,NS(=O)(=O)CCC(=O)NC1(CO)CN(C(C2(F)CCCOC2)=O)C1 67042,C1(NC(c2cnc(CCCC)s2)=O)CCN(C(c2cc(COC)on2)=O)CC1 67043,c1(NC(C2COC(C)(C)O2)=O)ccc2nccnc2c1 67044,c1(CNC(C(C)NC(CC)=O)=O)n[nH]c2c1CN(C(C1CN(C)C(=O)N1)=O)CC2 67045,C1(CNC(N2CCC(S(=O)(=O)N(C)C)C2)=O)CCc2cc(N)ccc2O1 67046,CC1(C)CCCC(CC(=O)NC2(C)CCN(C(C3(O)CC3)=O)CC2)O1 67047,C1(C#N)(C(=O)NC2CC(F)(CNC(C(C)OCCC=C)=O)C2)CCCOC1 67048,C1(NC(c2cn(CCNC(C(C=C)O)=O)nn2)=O)CCNC(=O)CC1 67049,N1(C(=O)CCc2cc[nH]n2)CCN(C(C23CCCC(C2)OC3)=O)CC1CCO 67050,c1(NC(C(CCNC(=O)CCCn2ccnn2)O)=O)ccc(O)c(F)c1 67051,Nc1cc(Cl)cc(F)c1C(N1CC(CNC(=O)C=Cc2ccc(C(N)=O)o2)C1)=O 67052,c1(C(=O)NC(CNC(C2(CC#N)COC2)=O)CO)cc(Cl)cc(F)c1Br 67053,S(=O)(=O)(c1cncn1C)NC(C)Cc1nccn1C 67054,C1(NC(C2C(=O)NCCC2)=O)CCC(O)CN(C(=O)C=Cc2cncs2)C1 67055,C1(NC(CC(=O)NCC#C)=O)CS(=O)(=O)CC1NC(c1nccc(N)c1Cl)=O 67056,c1(C(=O)NCC2C(NC(CCCNC(N)=O)=O)C2)c(Cl)nsc1Cl 67057,C(=O)(C(O)CCC(C)C)N1CC2C(NC(c3ccc(OC)c(C4CC4)c3)=O)(C2)C1 67058,c1(N(CCC)CCNC(=O)C=Cc2cccnc2)ncn(C)c(=O)c1Br 67059,c1(NC(CCCNCCC)=O)ncc2c(n1)CCN(C(=O)OC(C)(C)C)C2 67060,C=C(CC)CN=C(NCc1cccs1)NCc1ccc(OC)c(OC)c1C 67061,C1(NC(C2(C)CSC2)=O)CCC(O)CN(C(=O)Cn2ccc([N+](=O)[O-])n2)C1 67062,C(C(CC(=O)Nc1cnn(C(F)F)c1)NC(C1C=CCCC1)=O)OC 67063,O=C1CN(c2ccc(NC(=O)CN(C3CC3)Cc3ccccn3)cc2)CCCN1 67064,c1(C(=O)NCC(CC(C)C)NC(=O)C=C2CCC2)csc2ccc(F)cc12 67065,C(=O)(C#CC(C)(C)C(F)F)NC(C)CN(C)C(C1CCCN1c1ncccn1)=O 67066,C1(CNC(=O)CCF)CN(C(=O)Cc2sccc2Cl)CCO1 67067,Cc1ncc(Cl)c(C(=O)NCC2CCN2C(=O)Cc2nnn(C(C)(C)C)n2)n1 67068,N1(CC(=O)NCCC2CCN(C(c3cnn[nH]3)=O)C2)CCC(n2cccc2)CC1 67069,C1(CC)CCN(C(=O)Cc2ccsc2C)C(C(=O)N(CC(O)C2CC2)C)C1 67070,C1(N(C(CCOCC)=O)CC)CCN(CCC(C)C)CC1.c12nccc(n1)NC2 67071,C(=O)(C(CCCCCC)N1CCC(CC(C)(C)C)C1)NCC=C 67072,C=C(C)c1cncc(C(=O)NCCSCOC(C)=O)c1 67073,N1(C(C(C)c2ccco2)=O)CCCC(NC(c2ncc(Cl)nc2Cl)=O)C1C 67074,Cc1ncnc(C)c1C(N1CCCC(C(=O)NCC(C)(O)C2(C)CC2)C1)=O 67075,c1(-n2cc(C3OCCN(C(CCC4CCC(C)O4)=O)C3)nn2)cc(F)cnc1Br 67076,N1(C(C(CC)(C)OC)=O)CCCC2(C1)CN(C(C1CCO1)=O)C2 67077,c1(CC)noc(C)c1CNC(C1C2CN(C(c3ncc[nH]3)=O)CC12)=O 67078,c12ccc(cc1)SC(C)C(=O)C2=O.N1(C(C(=O)N)C)CCSCC1.CCN 67079,Cc1cccc(Cl)c1CC(N1CC2C(N(C(=O)COC3CCCC3)C)C2C1)=O 67080,C1(CC)CNC(=O)CN1C(=O)C(C1CCCC1)NC(=O)CC1(N(C)C)CCCC1 67081,CCC(CC(=O)NCC1(OC)CCN(C(c2nn(C)nc2Br)=O)C1)SC 67082,C1(NC(C(C)OCC(C)C)=O)CCCC(CNC(c2cnc[nH]c2=N)=O)C1 67083,c1(C(N2CC(C)C(NC(C3CCCC(CF)C3)=O)C2)=O)nn(C)c(Cl)c1Cl 67084,N#Cc1ccc(CCS(=O)(=O)NC2CC(c3ccncc3)C2)cc1 67085,Cn1c(NC(=O)CC(O)c2ccccc2)nc2cc(Br)c(Cl)cc12 67086,Cc1ccc(F)c(C(=O)N(C)CCN(C(=O)COC2CCCCC2)C(C)C)c1Cl 67087,CCC(CCOC)C(=O)NC(C)CCCC(=O)N1CCCC2(CC2)C1 67088,N1(C(C(C)NC(=O)NC)=O)CCN(C(=O)CCOC2CCCCC2)C2COCC12 67089,c1(CCC(=O)NCC(CNC(=O)CC2CC=CCC2)CO)ccccc1O 67090,C#Cc1ccc(C(=O)NC2CC(F)(CNC(=O)CCc3cncs3)C2)cc1F 67091,C(c1ccc(=N)[nH]c1C)=CC(=O)NC1(CC=C)CN(C(=O)CC2(OC)CCC2)C1 67092,CC1(C(=O)NCc2cc(C(=O)NCCCC3(O)CCC3)on2)CCOC1 67093,C1(C(=O)NC(CC)CNC(=O)CCc2scnc2C)CCCNS1(=O)=O 67094,N1(C(CC(C=C)(C)O)=O)CC2CC(NC(c3cncc(C)c3Cl)=O)C(C2)C1 67095,N1(C(COC(C)C)=O)CC2CCCC1(CNC(c1coc3ccccc13)=O)C2 67096,C(=O)(C#CC1CCOC1)NC1(C)CN(C(=O)CSCc2ccccc2F)C1 67097,C1(NC(CCCC)=O)CC2CCC1(CNC(c1cncc(C)n1)=O)C2 67098,C1(CNC(c2c(C)oc(CO)c2)=O)CC2(CCN(C(C3(C)CC3(F)F)=O)C2)CO1 67099,c1(C(=O)NCC2N(C(C3C(C)C3C)=O)CC(C)(C)OC2)c(F)cc(F)c(F)c1F 67100,Cc1ncc(C(=O)NCCCNC(=O)CN(CC(=O)OC(C)(C)C)C2CC2)cn1 67101,c1(C(N2CCC(C)(CNC(C3(CF)CC3)=O)C2)=O)cc2cc(F)ccc2[nH]c1=O 67102,C1(NC(c2cc(Br)n3c2CCC3)=O)CN(C(=O)CCC2CCC2)CC2(CC2)C1 67103,c1(C(=O)NCC23CCCC2CN(C(c2cnns2)=O)C3)cnn2c1C(=O)NCC2 67104,N1(C(C#CC(C)(C)C)=O)CC23CCCCC2(C1)CN(C(c1ccon1)=O)C3 67105,O(N1CCC(NC(C2(C)CC(NC(=O)C(C)N=[N+]=[N-])C2)=O)CC1)CC 67106,CC1CCC(NC(=O)CC2COCCO2)CN1C(C1CC1C(N)=O)=O 67107,c1(CCC(=O)N(C2CN(C(=O)CC3(CO)CCCC3)C2)C)ccc(F)cc1 67108,N1(C(c2cc(C(C)=O)[nH]n2)=O)CCOC2CN(Cc3c(C)cc(Br)cc3C)CC12 67109,CC1(C)C(=O)NC2CCC(C(=O)Nc3ccc(C4(c5nn[nH]n5)CC4)cc3)CC12 67110,C1(CCNC(c2cn(C)cc2C(F)(F)F)=O)CCN(C(C2CC23CC3)=O)C12CC2 67111,c1(CS(C)(=O)=O)ccc(CN(C)CC2CCN(C(CC(C)O)=O)C2)cc1 67112,C1(C(N(CC(CC)C)C)=O)(NC(=O)Cc2n[nH]c(C)n2)CC(CC2CCC2)C1 67113,CC(C)(CC(=O)NCC1CCC=CO1)n1cc(CCN2CCOCC2)nn1 67114,c1(CCC(=O)N(CC(C)NC(CCC2CC(OC)C2)=O)C)ccc(C)cc1 67115,N1(C(C2C(CC)C2)=O)CC2(COC(CNC(c3nnc(C)s3)=O)C2)C1 67116,S(=O)(=O)(c1ccc(C#N)c(N(C)CCF)c1)N(C1C(C)CCC1)C 67117,C1(CNC(CC(C)OC)=O)CN(C(=O)CC2CCCOCC2)CCC12CCOC2 67118,C1(NC(CCC(C)OC)=O)CN(C(=O)CCn2nc(C)cc2C)CC2CC12 67119,C1(NC(Cc2c(C)n(C)nc2)=O)CCCN(C(c2cc[n+]([O-])cc2)=O)C1C 67120,c1(CN(C(CN2CCCC(C)C2CCN=[N+]=[N-])=O)C)cc(N)cc(O)c1Br 67121,N1(C(C(C2(C)CC2)NC(=O)COCc2nnc(O)o2)=O)CCCC(C(N)=O)C1 67122,N1(C(c2c(CC)csc2)=O)CC(NC(c2cnc(C)s2)=O)C2CC12 67123,c1(C(=O)NCC2(F)CN(C(=O)CCC3CC(F)(F)C3)C2)cncc([N+](=O)[O-])c1 67124,CN1C(=O)CN(C(=O)CC2C3CN(C(C4CC(C)(C)CN4C)=O)CC23)CC1=O 67125,c1(C(N(CCNC(=O)C=CC2(C)CCOCC2)CC)=O)ccc2ncncc2c1 67126,C(=O)(CC(C)C(=O)N1CCC(F)C(NC(c2ccc(O)nc2)=O)C1)OC 67127,C1(O)(CNC(C2(CC=C)CCC2)=O)CN(C(=O)C(C)OCC2CCCO2)C1 67128,C(=O)(C(C(C)(C)SC)c1ccccc1)NC1C(CC)CN(C(=O)OC(C)(C)C)C1 67129,c1(CC)[nH]c(=N)sc1C(=O)NCC(O)CN(C)C(c1ccns1)=O 67130,c1(C(C)C(=O)NC2CCCN(C(=O)C=CCO)C2)ccc(S(=O)(=O)N(C)C)cc1 67131,N1(C(Cc2ccc(C)o2)=O)CC(C(N2CCC(C(F)F)CC2)=O)CC(C)C1 67132,c1(C(C(=O)NC(CC)CN(C(=O)CCSC(F)(F)F)CC)=O)ccc(C)cc1 67133,Cc1c(Br)ccc(NC(=O)C(=O)N(CC(C)C)C(C)C)c1I 67134,Cc1cc2cc(C(=O)N(C)CCNC(C3(C(F)F)CC3)=O)c(Cl)cc2[nH]1 67135,C1(C(=O)NC2CCC(C(=O)NCC(C)CC3CCC3)C2)(OC)CCOC1 67136,C(=O)(CC1CC(C)(OC)C(=O)N1)N1C(CCC#C)CCC1.OC 67137,N1(C(COCCCCC)=O)CC2(C1)C(NC(c1cc(C)oc1C)=O)CCS2(=O)=O 67138,C1(C)(NC(C23CC(COC)(OC2)C3)=O)CCN(C(C2CCCCC2OC)=O)CC1 67139,Cc1nc2sc1C(=O)NC2.C1(C(=O)Nc2nccs2)CCOC(C)C1 67140,N1(C(C2Cc3cc(F)ccc3O2)=O)CCCCC2(C1)CN(C(c1cc[nH]c1)=O)C2 67141,C1(COC)C=CCCN1C(C1(CO)CCC1)=O.C12CCN(C1)C(=O)CO2 67142,c1(C(CNC(C)=O)NC(c2c[nH]nc2[N+](=O)[O-])=O)ccc2ccccc2c1 67143,N1(C(C(C)SC)=O)CC(NC(=O)C=CCCC(C)C)CCC1C 67144,c1(OC(C(CC2CCC2)OC)=O)ccccc1C.C12(CCOC1)C(=O)NCC2 67145,Cc1nc2cccc(C(=O)NC3COCC3CNC(C34CCC(C3)C4)=O)c2[nH]1 67146,c1(CN(C)C(C2(F)CCN(C(c3cnc(Cl)nc3)=O)C2)=O)ccc(F)cc1 67147,c1(NCCCC(=O)Nc2nc(COC)nc(O)c2)ccc2c(c1)CCO2 67148,C1(F)(CNC(CCN(C2CC2)CC)=O)CCN(C(=O)Cc2nocc2C)C1 67149,C1(CC(=O)NCC2N(C(C(F)=CCC)=O)CCC2)COC2CC1C2 67150,c1(OC)c(NC(C2CCCN(C(C3CC3C)=O)C2)C)ncnc1Cl 67151,N1(C(C=NOC)=O)CCC2(CC1)CC(NC(=O)C(CO)NC(N)=O)C2 67152,S(=O)(=O)(CCCCCl)N1CC(C(=O)NC(C2CCCCC2)CO)C1 67153,C12(C(=O)NCC3C(C)CCN(C(C4(O)CCSC4)=O)C3)CCC(CC1)C2(C)C 67154,C=C1Cn2c(C(=O)NCC3CC4CN(C(=O)C=CSC)CC34)nnc2S1 67155,C1(NC(=O)CNC(=O)C2CC2)COC2(CCN(C(c3ocnc3C3CC3)=O)CC2)C1 67156,N1(C(Cn2c(C)c(Cl)cn2)=O)CC(C)N(C(=O)CC(F)(F)C(C)C)CC1C 67157,CC1C(NC(=O)CNC(C2CCCC2)=O)CCCN1c1ccc(C#N)nc1 67158,N1(C(CC(=O)OCC)=O)CC2(CC(CC(=O)NCC3(C#N)CC3)C2)C1 67159,C1(C(NC(c2ccccc2)(CC)CC)(C)C2CC2)CC(C2CC2)=NO1 67160,Cc1cc(C(N2CC(C)(C)C2C2CCN(C(=O)C(C)O)CC2)=O)ccc1O 67161,c1(OCC)ccc(Cl)c(NC(C2CCN2CC2CCCC2)=O)n1 67162,N(C1CN(C(=O)C2=CCCOC2)Cc2ccccc21)C(Cn1c(C)nnn1)=O 67163,CC1CCCC(CNC(=O)CN(C2CC(C#N)C2)C(=O)CC2CCCCC2)C1 67164,CC(C(=O)N1CC2CC2(NC(=O)Cc2ccc(F)c(C(F)(F)F)c2)C1)C(F)(F)F 67165,c1(N2CCC(CNC(C(CN(C)C)(C)C)=O)C2(C)C)cc(C#N)nc(C2CC2)n1 67166,c1(C(N2CCN(C(C(CC)OC)=O)C(C3CC3)C2)=O)cc2ccc(F)c(F)c2o1 67167,C1(c2cn(C(C)(C)C)nc2)CN(C(=O)C(c2cnn(C3CC3)c2Cl)=O)CCO1 67168,C1(NC(CC(C)(C)N(C(c2c(C)coc2)=O)C)=O)CN(C)CC1(F)F 67169,C(=O)(CCN(C)C(C1(C)CC1)=O)NCC1C(C(=O)OCC)C1 67170,C1(CC)CN(C(c2cnc(=N)[nH]c2)=O)CC1C(=O)NC1CC=CC1 67171,C1(COC)(NC(c2coc(C3CCC3)n2)=O)CCN(C(C2COC2)=O)C1 67172,Cc1cccnc1C(C(C)(C)C)NC(C12CC(n3cc(C4CCC4)nn3)C1C2)=O 67173,C(C)(CCCCNC(c1cc(C(N)=O)co1)=O)NC(CC(C)O)=O 67174,C1(NC(C2(C)CCCCCC2)c2n(CCOCC)nnn2)CCCC(C)(C)C1 67175,N1(C(CNC(CCC(C)C)=O)=O)CCC(NC(=O)CC2CNC(=O)C2)C12CCC2 67176,c1(C(=O)NCC(=O)N(CC(N2CCCC2Cc2cccs2)=O)C)c(N)cccc1Cl 67177,N1(C(Cc2c(C)occ2)=O)CC2CN(C(=O)COc3ccc(F)cc3)CC2(C)C1 67178,c1(C(=O)NC2CC(CNC(C3CCCC3(F)F)=O)C2)ccc2nc(S)oc2c1 67179,C1(C(N(CC(CCC)O)C)=O)CCN(C(=O)C#CC2(C)COC2)C12CCC2 67180,C1(=CC(=O)NCC(CN(C(C(CC)O)=O)C)O)CC2CCC(C1)N2C 67181,N(C(=NCCCN(S(C)(=O)=O)C)NCC1CCCCO1)C(CC)C 67182,CC1=C(C(=O)NC2CC3CC(NC(C4CC(C(C)C)=NO4)=O)CC3C2)CCCC1 67183,CC1CCCN(C(=O)Nc2ccccc2NC2(C)CCCO2)C1 67184,c1(C(N2CC(CNC(c3n(CC)nnc3C)=O)OCC2)=O)c[nH]c(C)cc1=O 67185,Cc1c(C(N2CC3(CC3)CC2CNC(=O)CNC(N)=O)=O)sc2ccccc12 67186,C(CC(C(=O)N1CC(O)C(O)C1)NC(C1SCC=C1C)=O)SC 67187,c1(CNC(C(C)NCCC)=O)nc(CO)n[nH]1 67188,C1(C)(CNC(CC2C=NN(C)C2=O)=O)CN(c2cccc(C(F)(F)F)n2)CCO1 67189,CC1CCN(C(c2c(Cl)cncc2Cl)=O)CC1NC(c1ccnc2[nH]ncc12)=O 67190,c1(CC(=O)NCC(C)NC(=O)Cc2cncs2)ccnc(O)c1 67191,C1(CNC(C(C)OC)=O)CCCC1NC(C1CCC2CC12)=O 67192,c1(C(N2CC3C(CCNC(c4ccon4)=O)(CC3)C2)=O)ccc(F)cc1[N+](=O)[O-] 67193,c1(C(N2CC(CNC(C(S(C)(=O)=O)C3CC3)=O)OCC2)=O)cc2ccccc2s1 67194,C1(CNC(CC=CC)=O)CC(NC(c2cn(C)cn2)=O)C12CCC2 67195,N1(C(C2CCOCC2)=O)CCC(N(C2(C3CCCO3)CC2)C(C2CC2)=O)C(F)C1 67196,C(=O)(CC1C(=O)N(C)c2ccccc21)NCC1(CNC(CCC(=O)OC)=O)CC1 67197,N1(C(C2(CNC(c3cc(C)c(O)nn3)=O)CCCCC2)=O)CCCC2(C)CCC12 67198,C1(NC(c2ccc(I)c(Br)c2)=O)CN(C(=O)Cn2cc(Cl)cn2)CC1(F)F 67199,c1(CN(CCC)C(=O)Nc2nc(C(C)C)ns2)cc(Cl)ccc1Br 67200,C(=O)(C(F)C(CC)CC)N1CCN(CC(C)NC(c2nc(CC)oc2)=O)CC1 67201,C(=O)(C1=CS(=O)(=O)CCC1)N(CC(C)(C)NC(=O)COc1cccc(O)c1)C 67202,n1(CC)cnc2nc(N3CCN(C)C4(CCC4)C3)nc(N(CC(F)(F)Br)C)c12 67203,CCC(CC(C)CO)NC(=O)N(C1CCSC1)C 67204,CCS(=O)(=O)CC(=O)NC(CNC(=O)C1=CCC1)CC 67205,CCC(CC1CCCCC1)C(=O)NCCC(C)CCNC(=O)Cc1csnn1 67206,C1(CNC(C(C)(O)CCc2ccccc2)=O)CC2CCC1N(C(=O)CCF)C2 67207,C1(NC(CSCC(=O)OC(C)(C)C)=O)CCCN(Cc2ccc(O)c(O)c2)CC1 67208,C1(NC(CN(C(C(c2ccccc2)N(CC)CC)=O)CC)=O)(CC)CCN(C)C1 67209,c1(C(=O)NCCC(=C)CNC(c2c(CC)nn(C)c2Cl)=O)ccnc2c1CCC2 67210,C(=O)(CN=c1[nH]c(C)cs1)N1CCC(F)(CNC(c2cnc(OC)c(C)n2)=O)C1 67211,N1(C2CN(C(=O)NC(c3ccco3)C#C)C2)CCCS1(=O)=O.C1CC1 67212,c1(NC(=O)COC(C2CCOC2C(F)F)=O)ccc(C(F)(F)F)cc1Cl 67213,C1(CCC)CN(C(=O)CC(C)C)CC1C(=O)NCC(C)(O)C1CCC1 67214,C1(CC)CN(C(=O)CC(C)C2CCCCC2)CCN1C(=O)CSc1ccccc1 67215,C1(CCCOC(C)C(=O)NCCc2ccccc2)CCCN1C(=O)CC1(C)CC1 67216,C(=O)(C(F)C(C)(C)O)N(CC(CC)NC(c1cc(N(C)C)ccc1N)=O)C 67217,CN1CCC(NC(=O)CNC(=O)CNC(C2CCC(F)C2)=O)CC1=O 67218,N1(C(C(COC(C)C)(C)C)=O)CC(C#N)CC1C 67219,C(c1ccc(F)nc1)=CC(=O)NCC(CNC(c1c(C)nc(N(C)C)s1)=O)C 67220,C1(N(C(c2ccc(CNC(C)=O)s2)=O)C)CCCN(C(C2COC(=O)O2)=O)CC1 67221,C(=O)(CC(C)(C)CNC(c1cc(Cl)n[nH]1)=O)NCC(C)Cc1cn[nH]c1 67222,C(=O)(C(C)(O)C(F)(F)F)NCCC1CN(C(C2CC(OC)C(OC)C2)=O)C1 67223,C(CCC(CCC)NC(c1n[nH]c(C)c1C)=O)NC(c1cn(CCCC)nn1)=O 67224,C1(CNC(C(C)SCC)=O)(CO)CCCN(C(C2CCCN2C(C)=O)=O)C1 67225,C(=O)(CC1=CCOCC1)NCc1cn(CCNC(c2nc(C)n(C)c2)=O)nn1 67226,Cn1ccc(=O)c(C(=O)NCCCN2CCN(C(C3CCS(=O)(=O)C3)=O)CC2)c1 67227,Cc1cc2ccccc2nc1C(N1CC2CCN(C(c3csnn3)=O)CC2C1)=O 67228,C(CCCCC(=O)N1CC(NC(=O)CSC)CC(C)C1)OCC 67229,C1(CCC(=O)NCCN(C(=O)CCc2ncc(C(F)F)o2)C)CCC(C(F)(F)F)O1 67230,CC1(C)CC(CC(=O)NC(CNC(C2(CO)CCCO2)=O)C2CC2)CO1 67231,N1(C(CCS(=O)(=O)NC)=O)CCC2(CC1)CC2NC(=O)C(c1cccc(C)c1)F 67232,c1(C(N2CC(C(=O)NCc3ccc(OCC)cc3)C2)=O)cc(OC)c(C)cc1Br 67233,c1(C(N2CC(C)OC(CCNC(=O)C3=CCCC3)C2)=O)cc(C#N)ccc1F 67234,c1(C(=O)NC2(CO)CCN(C(CC3ON=C(CC)C3)=O)C2)cc(C)nc2ccnn12 67235,N1(C(c2c(C)nco2)=O)CCCC(O)(CN(C(=O)C(C)CN2CCCCC2)C)C1 67236,C1(C(=O)NC(C(=O)NC2CCCC2)c2cccs2)CN2CCCC1C2 67237,CC(CC1CCCO1)N=c1[nH]c(=NC(C)c2cn(C)cn2)[nH]c2c1CCCCC2 67238,Cn1ccc(-n2cc(C(CC(N)=O)NC(=O)CC3CCCSC3)nn2)cc1=O 67239,C1(C(=O)NC(n2ccc(C(N3CC(n4ccnn4)C3)=O)c2)C)CCOC1C 67240,c1(C(=O)Nc2cc(Br)ccc2CO)cccn2c(-c3ccnc(O)c3)cnc12 67241,C1(C(=O)NCCNC(=O)CC2CCCCC2O)CC(=O)c2ccccc2C1 67242,c1(CN2CC3CN(C(=O)CCc4ccccn4)CC32)ccc(I)c(F)c1F 67243,C(=O)(C#CC1CCCOC1)NCCOCCN(C(CC(C(=O)OC)C)=O)C 67244,CCC(C)C(C)(O)CNC(C1CCOCC1NC(=O)C(CC(C)C)OC)=O 67245,N1(CCN(C(CN(C(=O)C(C)N(CC)CC)CCC)=O)CC)CCCCC1 67246,CC1CCCC(O)(CNC(C2CC(n3cc(CC4CCOC4)nn3)C2)=O)C1 67247,N1(C(CCCN(C(C(CCC)C)=O)C)=O)CCCC(C)(CCC)C1 67248,c1(CNC(C(CO)OC)=O)ncccc1C(=O)N(CCCCN(C)C)N(C)C 67249,N1(C(c2c(CC)ocn2)=O)CC(NC(c2cc(O)ncn2)=O)C2CCCCC12 67250,Cc1ccc(Cl)c(C(=O)NCC2(O)CCCN(C(C3CC34CCCC4)=O)C2)c1N 67251,C1(OC)CC(CNC(=O)CC(C)(C)C)N(C(=O)CCn2cncn2)C1 67252,CCCC(O)C(CO)NC(c1cncc(CNC(=O)CCc2cnn(C)c2)c1)=O 67253,C(=O)(C(F)C(C)(C)O)N(C1CCN(C(=O)CCOCC(C)(C)C)C1)CC 67254,N1(C(c2c[nH]c(=NC)s2)=O)CCC(C2CC2)C1CNC(c1cc(F)n(C)n1)=O 67255,N(C(=NCc1cccs1)NC1CC12CCCC2)CC(F)F 67256,CCCC(CCO)NC(=O)CC1(N(C(=O)C(CC)OC)C)CC1 67257,c1(OC)cc(C(=O)NCc2ccccc2C(C)(F)F)cc(C)c1 67258,c1(CC(N2CC(OCC)C(CNC(=O)CC(C)(C)O)C2)=O)ccc(Cl)cc1Cl 67259,C12(CNC(C(C(C)O)C)=O)CC(NC(=O)C3=CCCC3)(C1)C1(CCOCC1)O2 67260,N#Cc1cc(C(N2CCC(F)(C(=O)N(C3CCOCC3)C3CC3)C2)=O)cs1 67261,C1(NC(=O)C=C2CCCCC2)(CF)CCN(C(=O)C(c2cccc(F)c2)O)C1 67262,N1(C(C2(CCCC)CC2)=O)CCCC(C2CCCN(C(C3C4COCC34)=O)C2)C1 67263,N1(C(CP(C)(C)=O)=O)CCOCC(NC(c2ccccc2Cl)=O)C1 67264,N(C(=NCCC1CCC1)NCCC(N1CC(C)OC(C)C1)=O)C1C(C)CSC1 67265,CS(=O)(=O)c1cnn(CC(=O)NC2CCCC(NC(=O)CSC(F)(F)F)CC2)c1 67266,c1(-n2cc(CC(N3CCC(N(C)Cc4ccccc4)C3)=O)nn2)cncc(Cl)n1 67267,C1(C(N2C(CCNC(c3cnco3)=O)CCC2)=O)CC(F)(F)C12CCC2 67268,Cc1cc(C(F)(F)F)cc(CN2CCC2Cn2cc(C3CCCC3O)nn2)c1 67269,CCCC(CC)CC(=O)N1CC2CCC(C1)N2c1nc(Cl)nc(C)c1F 67270,C1(CNC(C2(OCC)CC2)=O)CN(C(=O)C(C)C(F)F)CC1(F)F 67271,N1(C(C2C(C)(Br)C2)=O)CC23CCCC2(C1)CN(C(=O)CCC1CCCC(O)C1)C3 67272,C1(NC(c2nccc(OC)c2)=O)CN(C(=O)C(C)(C)N(C)C)CCC1C(F)(F)F 67273,C1(COC)CC(CNC(C2CC2C(C)(C)C)=O)N(C(=O)CNC(N)=O)C1 67274,c1(CN(C)C(C23COCC(C2)C3)=O)ccccc1CNC(C1(F)CC=CCC1)=O 67275,c1(C(N(CC(CNC(C2(COC)CCCOC2)=O)C)C)=O)nnn2c1COCC2 67276,C(=O)(C(C)(C)C1=CCSCC1)NC(C1OCCN(C(c2c(CC)cco2)=O)C1)C 67277,Nc1ncc(C(F)(F)F)cc1C(N1CC(CCNC(C2CC(F)C2)=O)C1)=O 67278,c1(C(=O)NC(CN(C(=O)C=Cc2cnc[nH]2)CC)C)nccc(N)c1Cl 67279,c1(C(N2CCN(C(=O)OC(C)(C)C)CC2C(F)F)=O)cc(F)cc2nccnc12 67280,Cc1ccc(F)c(CN2CCN(Cc3cnc(Cl)c(Cl)c3)CC2)c1Br 67281,C1(C(=O)NCC2CC(OC)C2)(NC(=O)CCC2(C#N)CCC2)CCSC1 67282,C(=O)(C(C)(C)C(=O)NC(C1CCCCN1C(c1cc(Cl)n(C)n1)=O)C)OCC 67283,C1(N(C(=O)C2CC2)CC)CCN(C(=O)CC(=O)NC(=O)CN(C)C(C)C)C1 67284,Cc1cc(Cl)c(Cl)cc1C(N1CCCCC1C1(NC(=O)CSC2CC2)CC1)=O 67285,C1(C(=O)NCCCN(C(=O)CC(C)(C)C2CC2)CC)CC(C2CCC2)C1 67286,c1(CC)ccoc1C(=O)NC(C)(CNC(=O)CCOCCOCCCO)CC 67287,Cc1[nH]nc2c1CC(C(=O)NCC1CC(C)(C)CN1C(c1ccoc1Br)=O)CC2 67288,C=CCC(C(=O)N1CC(CNC(c2cc(Br)cnc2C)=O)(OC)C1)C(C)C 67289,c1(CNC2CN(C(CCc3c(C)noc3C)=O)CC2C)cc(F)cc(C#N)c1 67290,c1(N2CCC(NC(CC3(OC)CC3)=O)C2)cc(SC(C)C)nc(C)n1 67291,N1(C(C(C)N2CCCC2)=O)CCCCC(CNC(=O)CN(c2ncccn2)C)C1 67292,N1(C(C(CC)CC)=O)CC(CNC(c2cc(Br)ccc2C)=O)C2(CC2)C1 67293,C1(N(C(c2cc(OC)ns2)=O)C)CCN(C(c2cccc(C)c2O)=O)CC12CC2 67294,C1(CNC(C2(OCC)CCOC2)=O)(CNC(=O)CC(F)F)CC12CCC2 67295,C(CCC(C)(C)C(=O)Nc1cnc(F)nc1)NC(C=Cc1cc(C)no1)=O 67296,N1(C(CC2CC(C(=O)OC)C2)=O)CCCC(N(C(=O)C=CSC)C)C1 67297,c1(NC(=O)Nc2ccccc2)ccccc1OC1CC(c2nccc(C(F)F)n2)C1 67298,CC(C)CCC(C(=O)NCc1ccnc(F)c1F)NC(c1cnn[nH]1)=O 67299,CC1CN(C(C2(Cl)CC2(F)F)=O)CC1NC(c1cc(CC(F)(F)F)nn1C)=O 67300,c1(C(=O)NC2CCN(C(c3cc(C)c(C)o3)=O)CC2C)cccc2c(C)csc12 67301,N1(C(CCOC(C)C)=O)CCC2CCN(C(c3cc(C(F)(F)F)n(C)n3)=O)C2C1 67302,c1(CNC(=O)Cc2cccc(C3CC3)c2)ncc([N+](=O)[O-])cn1 67303,c1(OC)cccc(CN2CCC(CNC(c3csc(C)n3)=O)C2)n1 67304,c1(C(=O)NCC(C)(C2CC2)NC(c2nncs2)=O)ccc(-n2ccnn2)cc1 67305,n1(CC(N2CCC(C(C)NC(C3CC(N=[N+]=[N-])C3)=O)CC2)=O)ncc(O)nc1=O 67306,C(CCN(C)C(c1ccc(OC)o1)=O)(C(C)C)NC(c1cc(SCC)on1)=O 67307,Cc1csc2ccc(CC(=O)NC(C)CCCNC(C3CCC(O)C3)=O)cc12 67308,C(N=c1cc[nH]cc1S(=O)(=O)NCC1CN(c2ccccc2Cl)C1)c1c(C)non1 67309,C1(C(=O)NC23C(CN(C(C4(CC=C)CCC4)=O)C2)C3)COc2ccc(F)cc2C1 67310,C1(C(=O)NCCCN(C(=O)CN(C)CCOC)CC)CC=CCC1 67311,C(CC(C(C)(C)C)NC(c1ccnc(C(F)F)c1)=O)N(C)C(C1CC=CCC1)=O 67312,N1(C(C2C=C(C)CS2)=O)CC2(C)CC1(C(=O)N(C1CCN(C(C)C)C1)C)C2 67313,Cc1ccc(C(N)=O)cc1C(=O)NC1CCC(C)(CNC(=O)CC2CS(=O)(=O)C2)C1 67314,Cc1nc(CCC(N2CCC(CF)(NC(=O)CC3CC34CC4)C2)=O)oc1C 67315,C#Cc1ccc(C(=O)NCCC(CNC(=O)CN2CCC(=O)CC2)OC)cc1 67316,C1(OC)CCC(CC(N2CC(n3cc(CN(C)C(C)=O)nn3)C2)=O)CC1 67317,Cc1cc(F)c(F)cc1C(N1CC2CC2(C(=O)Nc2ncc(Br)nc2Cl)C1)=O 67318,c1(CN2CC(C(=O)NCc3c(C)cccc3)SCC2)cc([N+](=O)[O-])cc(O)c1O 67319,C1(CC)CN(C(=O)Cc2cccnc2)CCC1NC(c1sncc1C)=O 67320,N1(C(c2cc(S(=O)(=O)NC)oc2)=O)CCOC2(C1)CN(C(=O)C(C)CC1CC1)C2 67321,c1(C(N(CC(O)CN(C)C(C2CCCN2N=O)=O)C)=O)ccn(C)c(=O)c1O 67322,C1(CC(=O)NCC(CO)NC(=O)CNc2ccccc2)CCCCCC1 67323,Cc1cccc(CNCC2COCCN2C(c2ncc(Br)cc2Cl)=O)c1F 67324,C1(C(=O)OCC)CC2(CCCN2C(=O)NC(C(F)F)C2CCC2)C1 67325,N1(C(CCN(C)CC)=O)CCC2(CCCCN(C(C3(Cl)CC3(C)C)=O)C2)C1 67326,N1(C(c2c(C)ncs2)C(=O)NC(C)(C)C)CC(C)(C)OC2(CCOC2)C1 67327,c1(C(N2CC3CN(C(C(C)(C)O)=O)CC3C2)=O)nc2ccc(Cl)nn2n1 67328,N1(C(c2c(CC)csc2)=O)CC2CS(=O)(=O)CC2(NC(c2ccc(=N)[nH]c2)=O)C1 67329,N1(C(C2(F)C(C)OCC2)=O)C2CCC1CN(C(C1(CO)CC(F)(F)C1)=O)C2 67330,c1(OC)c(C(=O)NC2(C)CN(C(C3(C)CC3(F)F)=O)C2)ccnc1Cl 67331,C1(NC(Cn2c(C)nnn2)=O)CC2CC(C1)N(C(=O)CC1CC(F)(F)C1)C2 67332,Cc1cc(C(F)(F)C(=O)N(CC(O)CNC(C2CCC(C)O2)=O)C)cc(C)c1 67333,C1(C(=O)NC2CC3CC(NC(C(COC)COC)=O)C2C3)CCC(=C(F)F)CC1 67334,c1(C(=O)NC(C2(O)CCN(C(=O)CN3CCOCC3)C2)C)nccc2nn[nH]c12 67335,c1(NC(C2CSCCN2C(=O)Cc2ccc(Br)nc2)=O)cnc(Br)nc1 67336,c1(C(=O)NC2(CCNC(CCc3cn(C)nc3)=O)CC2)cnc2[nH]ccc2n1 67337,C(CN=C(NCC(c1cnccn1)(F)F)NCCOc1ccccc1)C1CC(F)C1 67338,C1(C(=O)NC)CN(C(C2CCN2C(=O)CCC(C)SC)=O)CCO1 67339,CC(C)C(C)C(CNC(=O)CCOCC(F)(F)F)NC(c1cc(C#N)on1)=O 67340,c1(NC)cccc(C(N2CC(O)(C(F)C(=O)NCCCC(=O)OC)C2)=O)n1 67341,C(C(N=c1[nH]c(=NCc2cnn(C)c2Br)[nH]c2c1CCCC2)C1CC1)OC 67342,c1(C(=O)NC2CCN(C(c3n(CC)nnc3C)=O)C2)cc(C)cc(Br)c1O 67343,c1(C(N2CC(CN(C(C(CCC)C)=O)C)OCC2)=O)cnc(O)c2ccccc12 67344,N1(C(C(c2cn(C)nc2)O)=O)CCC2(CC1)CC(NC(=O)C=CI)C2 67345,c1(CCCC)c(C=O)cnn1-c1ccccc1.N(C1=NCCS1)CC1CC1 67346,c1(C2(C(=O)NCC(CC=C)NC(c3c(C#C)c[nH]n3)=O)CC2)cccc(Cl)c1F 67347,C1(C)(CC)CC(C(=O)NCCN(CC(C)C(=O)OC)CCOC)C1 67348,c1(CC(N2CC(C)C(NC(c3nc(=O)n(C)[nH]3)=O)C2)=O)ccc2sccc2c1 67349,N1(C(CSCC=C)=O)CC2=C(C1)CN(C(c1cc(C)sc1Br)=O)C2 67350,CC(CCO)C(=O)N1CCCCC1Cc1cn(-c2cccc(F)n2)nn1 67351,C1(C(C2CC2)NC(N(CC=C)CC=C)=O)CCCCO1 67352,N1(C(CC2CCN(C(c3cc(OC)ncc3)=O)C2)=O)CC2CCCCC2C1 67353,C1(C(=O)NC2(CC(=O)NC3CCCC(CO)C3)CC2)(OC)CCCCC1 67354,c1(SCC(=O)NC(CNC(c2c(CC)non2)=O)C)ccc(O)cc1 67355,N1(C(C2(COCC)CC2)=O)CC2CCN(C(c3ccc(CC)nc3C)=O)CC2C1 67356,O=C(C1=NOC2(CCC2)C1)N1CC(C2CC2C(=O)NCC23CCC(CC2O)C3)C1 67357,c1(C(N2CCC3(N(C(C4C(C(C)C)C4)=O)CCC3)C2)=O)ccc2nc(=N)[nH]n2c1 67358,C(c1cncnc1O)=CC(N1C(CNC(C(CC)n2ccnc2)=O)COCC1)=O 67359,C1(C2CCN(C(CCC=C)=O)CC2)CC(N=c2[nH]c3ccc(N)cc3s2)CCO1 67360,C12(C(=O)NC(C(=O)NCC(C)(C)O)CC3CCOCC3)CCC(CC1)C2 67361,CCS(=O)c1ccccc1C(=O)N(C(C)CNC(c1cc(OC)n[nH]1)=O)C 67362,c1(C(N2CCC(CNC(C(c3cccc(Cl)c3)CC)=O)C2)=O)ccc(F)c(N)c1 67363,c1(CC(N2CCCC(NC(C(C)OCC)=O)C2)=O)ccc2nsnc2c1 67364,Cc1ccc(CC(=O)NCC2CCN(C(=O)CN3CCCCC3)CC2)c(F)c1F 67365,C=CCC(C)C(=O)N(CCCCNC(C1(COC)CCCOC1)=O)C 67366,CCC(O)C(C)(C)C(=O)NCC1(O)CC(C(=O)N(CCC(F)(F)F)C)C1 67367,C(=O)(CC(C)(C)C(F)F)NCC1N(C(c2c(Cl)cn(CCC)n2)=O)CCN(C)C1 67368,Cc1c(C(=O)NCC2CN(C(=O)C=CC3CC3)CC2O)noc1-c1ccccc1 67369,C1(CNC(c2c(C)cco2)=O)CC2CCC(C1)N2C(=O)C(C)Oc1ccccc1 67370,c1(C(=O)NCC23CC(NC(C(C)OCC4CC4)=O)(C2)C3)ccc2nccn2c1 67371,C1(C(N(CCC)C)=O)CCCN1NC(=O)C1CN(C(C)=O)CCO1 67372,c1(CC(=O)NC(C)(C)CCNC(C23CCCC2C3(F)F)=O)c[nH]c2cnccc12 67373,N1(C(c2c(NC)cccc2)=O)CCC2C(CCCN2C(C2(C)CCCC2)=O)C1 67374,CC1(F)CCC(C(=O)NC2C3CN(C(=O)CC4CC=CCC4)CC23)CC1 67375,C1(C(=O)NCCN(CCC)C(c2cc(C)ccc2OC)=O)CCC2C1C2(F)F 67376,CC1CN(C(C2OCCCC2(C)C)=O)C(C)CN1C(C1CN2CCCN1CC2)=O 67377,N1(C(C(=O)NCCCOCC)C)CCC(C)(NC(c2sccc2Cl)=O)C1 67378,c1(N(C(C2CCC(C(C)C)CC2)C(=O)NC(CC)C)C)ccc(F)c(Cl)c1 67379,C1(NC(C(CN(C)C)O)=O)CN(C(c2cc(F)c[nH]2)=O)CCC1CO 67380,C(=O)(C1CCc2c(Cl)cccc21)N1CCCC(N(C(c2c(C)cco2)=O)C)CC1 67381,N1(Cc2cn(-c3n(C)nnc3)nn2)CCN(C(C2CC(=O)N2)=O)CC1 67382,C1(CC)CN(C(=O)CSc2nncn2C)CCC1NC(=O)Cc1cc(Cl)cs1 67383,N1(C(CNC(CC)=O)=O)CCC(C(C)C)CC1CNC(=O)C=CBr 67384,C(=O)(CCCCC(C)(C)C)NC(C(=O)N(C)Cc1c(C)ccs1)Cc1ccco1 67385,C=CCC(CC)C(=O)NCC(c1ccccc1)CNC(C1(O)CC(C)(C)C1)=O 67386,C(C)(CCC1CCCC1)(c1n(CC(=C)C)nnn1)NCCC1CCCO1 67387,CN1CCC2CCN(C(=O)C(O)CCCNC(c3ccc(F)c(F)c3)=O)C2C1 67388,N1(C(Cn2cc(CCCC=C)nn2)=O)CCC(O)C1C(C)(C)C 67389,C(C)(C)(CCCCC(=O)NCC1CCC1NC(c1ccoc1Br)=O)OC 67390,C=CCCCCC(=O)NC(CC(=C)C)C(=O)NCCc1cn(C)nn1 67391,C(C(=O)N1CC(F)(F)C1C(C)C)(C(C)(C)C)n1cc(-c2c(C)nccc2)nn1 67392,Cc1c(Br)ccc(F)c1C(=O)NC(C)CCNC(=O)CC1C=CCC1 67393,N1(C(CC2CC(=O)NC2=O)=O)CC(NC(=O)Cc2ccon2)CC(F)C1 67394,O=C1CN(C(=O)NN2CCN(CCc3ccccc3F)CC2)C2CCCCC2N1 67395,C1(C)(C(N2CC(SC)C(n3cc(CC4CCOC4)nn3)C2)=O)CCCCNC1=O 67396,C(CC(C)C)(C(=O)NC1(CF)CCN(C(c2cscc2C(F)(F)F)=O)C1)OC 67397,C1(OC)CN(C(=O)CCc2ccccc2)CC1NC(=O)CC(C)n1cccn1.C1(C)CC1 67398,N1(C(C2CC(F)CN2C(=O)Cc2ccc(Cl)c(F)c2)=O)CCCC2CCCCC12 67399,c1(CC(N2CCC(CC(=O)Nc3c(CC)ncs3)C2)=O)ccc2nc(Br)sc2c1 67400,C(=O)(C(F)C(C)(F)F)NCc1ccc(C(N(CC)CC2CCOC2)=O)s1 67401,C1(NC(=O)OC(C)(C)C)C2CC3C1C3C2NC1C(F)(F)C12CCC2 67402,C1(C(=O)OC)CCCC(C(N2CCC(F)(C(N3CCOC(CO)C3)=O)C2)=O)C1 67403,C12(CC(N3CCC4(CCC4)C3)=O)CCC1CN(C(c1cccc(CO)n1)=O)C2 67404,C1(C)(C(=O)NCC2(O)CC(C)(C)C2)CCCN(C(=O)Cn2cnc(C#N)n2)C1 67405,c1(C(=O)NCC2N(C(C(c3ccncc3)C)=O)CC2)c(F)cccc1Cl 67406,C(=O)(C(F)(F)Cn1cc(Br)cn1)NCC1(c2ccc(C(=O)O)cn2)CC1 67407,C(=O)(CN=c1ccc(Cl)n[nH]1)N1CC(CNC(c2ccc(C)o2)=O)CC12CCC2 67408,CCC(C)C(C(=O)NCCc1cnc(C)o1)N(C(=O)CCCC1CCC1)C 67409,C#CCC(C)(C(=O)NCC(C)N(C)C)NC(=O)CC1CC(=O)NC1=O 67410,c1(-c2c(C)ccc(CN3CC4CC4C3)c2)cc(NC(C)(C)C)cc2c[nH]nc12 67411,C1(C2CCN(C(C3CCCO3)=O)C2)(NC(c2cccc(C(C)C)n2)=O)CC1 67412,C1(CNC(CCCC=C)=O)CN(C(=O)CN2CCC(=O)NC2=O)CC1(C)C 67413,c1(C(N2CCCC(NC(c3cn(CC(F)(F)F)nn3)=O)C2)=O)c(F)cncc1Cl 67414,C1(C(=O)NC2CCC(NC(C3CC34CCCC4)=O)CC2)CC2CSCC(C1)C2 67415,N(C(=NCCC1CCOC1)N(C)Cc1cc(F)ccc1C)Cc1cc(C)on1 67416,C#CC1(C(N2CC(C(C)(C)C)C2)=O)CCN(C(c2nn(C)cc2Cl)=O)C1 67417,Cc1c(Br)noc1C(N1CCC(n2cc(CNC(=O)N(C)C)nn2)C1)=O 67418,C1(NC(=O)CC2CCOC2)CC=CCC1C(N1CC(Cn2ccnn2)C1)=O 67419,c1(C(=O)NCC(CNC(c2cc(CCC)nn2C)=O)(C)C)cc2occc2[nH]1 67420,N1(C(C(C)CC(N)=O)=O)CCCCCC(Nc2ncnc(C(C)(C)C)n2)C1 67421,N1(C(CCC#C)=O)CCCC(CCCCNC(C2(Cl)CC2(F)F)=O)C1 67422,c1(C(=O)OC)c(NC(=O)CC2CCCN2S(=O)(=O)CCCl)cccc1F 67423,c1(N(CCNC(=O)Nc2cc(C)c(C)o2)C)ccn2nccc2n1 67424,CC(C)CC(C)(CNC(c1ccc(OC(F)F)cn1)=O)NC(C1CC1(C)C)=O 67425,c1(CN2CCC(NC(C(C)OCCC=C)=O)C2)ncc(Cl)n1C 67426,c1(N2CCCC(CNC(C)=O)C2)ccc(S(=O)(=O)N(CCCCO)C)c(Cl)c1 67427,CC(C)(C)C#CC(=O)NCCCC1CCCCN1C(=O)CC1CCC(=O)O1 67428,N1(C(C(CCC)OC)=O)CC2CCCC1(CNC(C1CC13CC3)=O)C2 67429,N1(C(C(C)NS(C)(=O)=O)=O)CC2(C1)CN(C(=O)Cc1cccc(Cl)c1)CC2CO 67430,Nc1c(C(=O)NC2CC2NC(C2CCC(NS(N)(=O)=O)CC2)=O)cccc1[N+](=O)[O-] 67431,c1(CC(=O)N(CC(CNC(C2CCN(CC)CC2)=O)C)C)c(C)nn(CC)c1C 67432,C=C(C)C(O)CC(=O)NCCC1CN(C(=O)CCCc2nc(CC)no2)CCO1 67433,c1(C(=O)NCC(CC)(CC)NC(C2C(=C)CC2)=O)cc2n(n1)CCNS2(=O)=O 67434,c1(CCC(=O)NCC2CCCN(C(C(CC)(C)O)=O)CC2)nc2ncccn2n1 67435,c1(NC(C2C3(CN(C(c4cncc(C)n4)=O)C3)C2)=O)cc(C(F)(F)F)ccc1I 67436,C(=O)(CC(CC)CCCC)NC(CCC#C)C(=O)NC(C)Cc1ncn(C)n1 67437,C(=O)(C(F)CCC(C)(C)C)NCC1(OC)CCN(C(C(CC)F)=O)C1 67438,C#CCC(CC(F)F)C(=O)NC(CCC)CC(=O)NC1(C(F)(F)F)CC1 67439,N1(C(C2(COC)CC2)=O)C(C(=O)Nc2sncc2C#N)CC2CC12 67440,CN=c1ncc(-c2cnc(F)c(C(c3c(N)cccc3Br)=O)c2)c[nH]1 67441,c1(CC(=O)NC2CC(NC(c3ccsc3)=O)CC2O)n[nH]c2ccccc12 67442,c1(C(=O)NC2CCC23CN(C(=O)CCC2CCCO2)C3)[nH]nc2ncccc12 67443,c1(CC(=O)NCCC(C)NC(c2c(F)ccc(CC)c2)=O)cnn2c1CCCC2 67444,C(=O)(C(C)(CC#C)N)N.C(=O)(C(=O)CCC=CC)C(CC=C)CC 67445,CC1=C(C(=O)NCC(C)NC(C2(C)CNC(=O)N2)=O)SCCO1 67446,c1(NC(=O)OC)nc(C)c(C)s1.n1(CCC)nnnc1C1C2CC(C2)N1 67447,N(C(=NCCN(C(C)C)Cc1ccc(N(C)C)cc1)Nc1ccc(Cl)cc1)CC 67448,Cc1cccc(C)c1C(=O)NC(C)CC1CCN(C(C2CCC2(F)F)=O)CC1 67449,Cc1ccccc1-n1cc(C(=O)NCC2CC2NC(C2CC(C)(C)CO2)=O)nn1 67450,c1(C(=O)NC(CN(C(C(CC)n2nccc2C)=O)C)C)cnc2c(C)nsc2c1 67451,Cc1cccc(N2CCC(C(=O)NCC3CC3c3ccc(C)s3)C2=O)c1 67452,C(F)(c1ccccc1)=CC(=O)NCCC(C)(C)NC(C1CCC(F)(F)C1)=O 67453,c1(C(C(N2C(CN(C(c3c(CC)ocn3)=O)C)CCC2)=O)C)ccncc1C 67454,N1(C(CC(CC)O)=O)CC2CC(NC(=O)C3=CCCCCC3)CC1C2 67455,CC(C)C(C)(C)C(=O)NCCN(C(C1CC(S(C)(=O)=O)C1)=O)C1CC1 67456,C(CN=c1cc[nH]c(-c2nccs2)n1)C1N(C(C2(C#C)CCCC2)=O)CCCC1 67457,c1(C(=O)NC(C)CCN(C(=O)C(C(C)O)NC(N)=O)C)cnc(N)c(Cl)c1 67458,N1(C(=O)NCC2(CNC(=O)OC(C)(C)C)CC23CCC3)CCC2(CC2CO)C1 67459,C(=O)(C1=NOCC1)N(CC(=O)NC(c1nc[nH]n1)CC)CCOC 67460,c1(CCC(=O)N(C(=O)CCC2(C(=O)O)CCN2)C(C)(C)C)cccc(C#N)c1 67461,CCC(C#N)C(=O)NC(C1CN(C(=O)CCOc2cccc(OC)c2)C1)C 67462,C12(C(=O)OC)CCCC(CNC(=O)NCC3(C)C=CCC3)(C1)OC2 67463,C(CCS(C)(=O)=O)(C(=O)NCCCN(C(c1ncccc1O)=O)C1CC1)OC 67464,C12(NC(CNC(=O)OC)=O)CCCC1CN(C(=O)C(C)CN1CCOCC1)C2 67465,Cc1ccccc1CN1CCCC(C(=O)ONC(C)Cc2cncnc2)C1 67466,C1(OC)(CNC(=O)C=C(C)Cl)CCN(C(C2(Cl)CC23CCC3)=O)CC1 67467,Cc1ccc(C)c(C(=O)NCC2(C)CN(C(c3nn(C)cc3Cl)=O)CCO2)n1 67468,C1(CNC(C(CC=C)OC)=O)COC(C)(C)CN1C(c1ncc(F)cc1F)=O 67469,Cc1cc(C(=O)N(CC(O)CNC(=O)C=CC2CC2)C)cc(O)n1 67470,c1(C(N(CCN(C(C2CCC(C)NC2=O)=O)C)C)=O)cccc2c1CCN2 67471,n1(CC(N2CCC(N(C(CCNC(C)=O)=O)C)C2)=O)nc(C)oc1=O 67472,c1(C(=O)NC(CCOC)CNC(C2(C3CCC3)CCC2)=O)cc(C)c(OC)c(Cl)c1 67473,C(=O)(CCS(=O)(=O)Cc1ccccn1)N(CCCCNC(=O)C#CC1CCC1)C 67474,Cc1cc(CC(=O)NC(C2CCOC2)CNC(C2CC(C#N)C2)=O)on1 67475,N1(C(C(C(C)(C)C)O)=O)CCC(C2CC2)(CNC(=O)CC2CC2)C1 67476,C1(CNC(COCC)=O)COC(CNC(c2c[nH]nc2C(F)(F)F)=O)C1 67477,CCCCS(=O)(=O)CC(=O)NCCCCC1CCN(C(=O)C(O)C(C)C)CC1 67478,C1(C(N(CC(C)N(C(Cc2scc(C)c2)=O)C)C)=O)C(C)(C)C1(F)F 67479,c1(SCC(=O)N(C(=O)NC(CCC=C)C(=O)OCC)CC)nc2ccccc2s1 67480,C(=O)(CC(C(C)OC)NC(C1CC=CCC1C)=O)N1CCC(C#C)C1 67481,c1(N2C(CNC(c3ccc(F)cc3)=O)CC(F)C2)nc2cc(F)cc(F)c2o1 67482,N1(C(c2cn(CCN(C)C)nn2)=O)CC2CCC1CN2C(C1(C)CCC(=O)C1)=O 67483,CCCC(O)C(=O)NCC(F)CNC(c1sc(COC)nc1C)=O 67484,n1(CC#C)c(C)cc(C(N2CC(CCNC(c3cc(C(C)C)no3)=O)C2)=O)c1C 67485,C1(NC(C(C2CCC2)OC)=O)CN(C(=O)C2=COCCC2)C2CCCCC12 67486,c1(C2C(NC(C3(c4ccccc4)CC3)=O)C2)ccc(Br)cc1F 67487,C(c1ccc(C(C)C)cc1)=CC(=O)NCC1(CO)CN(C(C(CSC)OC)=O)C1 67488,c1(CN2C(C)(CC)CC(NC(=O)OC(C)(C)C)C2)ccn2nccc2n1 67489,CCC(CC)C(C)C(=O)NC(COC)CNC(c1csc(C)n1)=O 67490,N1(C(C(N2CCCC(O)C2)C)=O)CCCC(CNC(C2CCCCS2)=O)C1 67491,C(CS(=O)(=O)CC(=O)N1CC(NC(c2cc(C)sn2)=O)CC12CCC2)OC 67492,C1(NC(C(C2CC2)SC)=O)(CO)CN(C(c2ccc(C(C)=O)o2)=O)C1 67493,c1(C(C(=O)NCC(C)C)N(C2CCSCC2)C)nnc2n1CCC2 67494,CC1CCCC(C)N1C(=O)C(N1CCC(CN(C)C(c2cc(Br)n[nH]2)=O)CC1)=O 67495,N1(C(N(c2c(OC)ccc(OC)c2)C)=O)CCCC12CCOCC2 67496,c1(CCC(N2CC(O)(CN(C(C(C)OCCCC)=O)C)C2)=O)ccnc(C)n1 67497,c1(OC(C)(C)C)cccc(Cl)c1NC(=O)C(CC(C)C)OC(=O)Nc1ccccc1 67498,C1(CNC(c2csc(C)c2C2CC2)=O)C(C)CCCN1C(c1cnns1)=O 67499,c1(CC(=O)NCC2N(C(CC(=C)Br)=O)CC2)csc2nc(C)cn12 67500,c1(NC2CCC(SC)CC2)ccncc1S(=O)(=O)NCC1CCCC1 67501,CC(C(C)(C)NC(=O)CCCn1cncn1)NC(=O)COCCc1ccccc1 67502,c1(N(CCCC=C)C)nnc(-c2ccc(C)o2)n1CCc1cccc(O)c1 67503,C(=O)(C1=CCCCC1P(C)(C)=O)NCC(C)(C)NC(CC(C)n1cccn1)=O 67504,c1(C(=O)NC2C(NC(C3(CC)COC3)=O)C2)ccc2ccn(C)c2c1 67505,N1(C(CN(CCC#C)C)=O)CC(NC(c2cnc3cc[nH]c3c2)=O)C(C2CC2)C1 67506,C1(NC(Cc2nc(C)oc2)=O)C2CC1N(C(=O)Cc1c[nH]nc1OC(C)C)C2 67507,Cn1nnc2c1CCN(C(=O)CCCCCNC(=O)C(C)(F)C(C)(C)F)C2 67508,Cc1c(C(=O)NCC(C)NC(C23CC2COC3(C)C)=O)cncc1Cl 67509,C1(C(=O)OC)C(C)CCN1C(C1CC(NC(=O)CSC(F)F)CCO1)=O 67510,C1(C(N2CC(O)(CNC(C3C(COC)C3)=O)C2)=O)CCc2cnn(C(C)C)c2C1 67511,c1(OCC(=O)NCC(C(C)C)NC(=O)C(O)c2cnc[nH]2)cccc(Br)c1 67512,N1(C(C(C=CC)O)=O)CCC(NC(c2cccc(Br)c2)=O)C1(C)C 67513,N1(C(CC23C(CN(C(Cc4c(CC)con4)=O)C2)CC3)=O)CC(=O)NCC12CC2 67514,c1(C(=O)NC2CC(CNC(C3CC(CCC)OCC3)=O)C2)ccc([N+](=O)[O-])s1 67515,N1(C(C(c2cccc(Cl)c2)(C)C)=O)CC2CCN(C(C3CCCS3)=O)CCC2C1 67516,C1(NC(c2c(OC)n[nH]c2)=O)CCN(C(=O)Cn2ccc(C(F)(F)F)n2)CC1O 67517,C1(C(=O)NCCc2onc(C)n2)CC(C)CN1C(=O)CN1CCCC1C 67518,C1(C(=O)NCc2scc(CNC(C(C)SCC)=O)n2)CC2CCCC(C1)C2 67519,c1(-n2ccc(C(=O)NC3C(NC(=O)C=Cc4cscn4)C3)n2)ccccc1Cl 67520,c1(C(=O)NC(CC)CN(C(C2CN(C(C)C)C2)=O)CC)c(C)noc1C1CC1 67521,C(CCCCCCC(=O)N1CC2CC(NC(=O)CCc3ccccn3)C1C2)SC 67522,c1(C(=O)NC2C3CC(NC(C(C)SCCCC)=O)CC32)cc(C)cc(C)c1N 67523,C#CCC(CC(=O)NC1CCC(NC(=O)C=CC(C)(C)C)C1)c1ccccc1 67524,C(=O)(CCCC(C)(C)C)N1C(CCNC(c2cnn(CC)c2C)=O)COCC1 67525,c1(C(N(CCNC(c2c(O)cc(C)nn2)=O)C2CC2)=O)c(C)nc2ccccn12 67526,CCCCC(O)CNC(=O)CC1CN(C(c2cccc(C3CC3)c2)=O)CC1C 67527,CC1CCCCCC1NC(c1cc(CNC(c2cnc(CN)nc2)=O)nn1C)=O 67528,c1(NC(=O)C(N2CCCCC(CO)C2)=O)cc(N2CCCC2)cc(F)c1 67529,N1(C(CC(C)(C)OC)=O)CC(C)N(C(C2(C)CC3CCC2O3)=O)C(C)C1 67530,C1(C)(SC(C)(C)C)CCC(NC(N2CC(CCS(C)(=O)=O)C2)=O)C1.C12CN(C1)C2 67531,c1(C(=O)OCC)ccc(Cl)c(NC(c2oc(C(=O)OC)nc2C)=O)c1 67532,c1(OC)cc(OC)cc(NC(=O)CN(C)Cc2cnc(C(C)C)s2)c1 67533,C1(NC(=O)CCc2cccc(Cl)c2)CN(C(c2cc(F)n[nH]2)=O)CCC1O 67534,CC1(C(=O)O)C=CCN1C(C1COCCC1NC(=O)CC12CCC(CC1)C2)=O 67535,c1(CNC(C2(C)CCCN2C(C2CCCC2)=O)=O)cnc(O)nc1O 67536,C1(C)(C(N(CC(CC)NC(=O)CCOCCN(C)C)C)=O)CC2CC2C1 67537,c1(C(=O)NCCCN(C)C(c2csc(Cl)n2)=O)nccc2c1NCCC2 67538,CCC(CC)(CCNC(c1cnc(COC)s1)=O)NC(=O)CC1CCCOCC1 67539,CCC(C)CCCCC(=O)N1CCC(NC(C2CCCC(C)(C)C2)=O)C(C)(C)C1 67540,N1(C(C(C(C)C)c2cccnc2)=O)CCOCC(NC(c2cccnc2)=O)C1 67541,C1(C(N2CC(c3ccccc3)(NC(CC(C)OC)=O)C2)=O)CCCCC1(C)C 67542,c1(N2CCC(CC)OCC2)nc(N2CCSC(c3ccccc3)C2)c2c(n1)CCS2 67543,Cc1nc(NC2CCc3n[nH]cc32)cc(C#N)n1 67544,c1(C(N2C(C(C)(C)NC(=O)CCC3CCC3)CCC2)=O)ccc2nc[nH]c2c1F 67545,C1(N(C(CSCCCC)=O)C)CCN(C(=O)CCCc2cccs2)C1 67546,C(C(F)(F)C(C)(C)O)NC(C1(CNC(C(CN(C)C)O)=O)CC(C)(C)C1)=O 67547,CC(O)(C(=O)NCC12CC(NC(=O)CN3CCCNS3(=O)=O)(CO1)C2)C(F)(F)F 67548,CCCCCCCC(=O)NCCCC(C)NC(C1CCCC1CC)=O 67549,CCCCCC(F)C(=O)NC(C)(C)CCNC(=O)Cc1cnn(C)c1C 67550,CN1CCCc2cc(C(=O)Nc3nnc(CF)s3)ccc21 67551,N1(C(CC)=O)C2CCCC1CN(C(c1c([N+](=O)[O-])c(C(F)(F)F)nn1C)=O)CC2 67552,CC1(C)CCN(C(c2cc(F)ccc2N)=O)CC1NC(C1COCCO1)=O 67553,CCC(O)C(C)(C)C(=O)NCC(CC(=O)N(CC(C)(CC)OC)C)OC 67554,n1(CC2C(C)CCCC2)ncc2cc([N+](=O)[O-])ccc2c1=O 67555,c1(C(=O)NCC2(O)CN(C(C(C(C)O)C)=O)C2)cn2cc(Cl)cnc2n1 67556,C1(COC)(NC(c2ccc(C#N)cc2)=O)CCN(C(C23CC(F)(CO2)C3)=O)CC1 67557,C1(C(=O)NCCCC(C)NC(=O)CCC#N)(CO)CCCCO1 67558,Cc1ccccc1-n1cc(CN2CCC(O)CC2)cn1.N12CCC(CC1)NC2=O 67559,CC#CCC(C(=O)Nc1cnccc1OC)NC(=O)C(CC1CCC1)OC 67560,O=C(CC=C(Cl)Cl)NC1CCCC1CNC(=O)C=Cc1cc[nH]c1 67561,c1(C(N(C2CN(C(=O)CCCC#N)CC23CC3)C)=O)cc2ccsc2n1C 67562,N1(C(C(c2cncnc2)C)=O)CCC(NC(=O)C=Cc2ccco2)C12CC2 67563,N1(C(CC)=O)CCC(C)C1C(=O)N(C)Cc1ncc(Br)cn1 67564,C1(C)(C(N(CCC)CCNC(=O)CC2CCCC2)=O)CCCC1O 67565,S(=O)(=O)(c1ccc(NCC(c2ccccc2F)OC)cc1Br)NCC=C 67566,c1(C(N2CCN(C(c3c(C(C)C)nns3)=O)CC2)=O)cccc(Cl)c1O 67567,C(CNC(c1c(C)noc1CC)=O)(C(C)C(C)C)NC(CCCC=C)=O 67568,C#CC1(C(=O)NCC(c2ccnn2C)O)CCN(C(c2csc(C)n2)=O)C1 67569,C1(CNC(C(CCOC)NC(c2cnncc2O)=O)=O)CC2CCCC2C1 67570,Cc1ccc(C#CC(=O)NCC2CCOCO2)cc1 67571,C1(NC(c2cncc(OC)c2)=O)CN(C(C2CCSC2)=O)C2CCCC12 67572,C12(C(=O)NCc3cncc(C)c3)CC(CN(C(C3(n4cnnn4)CC3)=O)C1)C2 67573,O=C(C1=NOC2(CCOC2)C1)N1CCC2CCN(C(=O)C(F)(F)C(F)(F)F)CC12 67574,c1(OCC(=O)NCC2CN(C(C=CC(=O)OC)=O)C(C)C2)ccc(Br)c(F)c1F 67575,c1(CNC(CSCCC)=O)cnn2c1CN(C(c1cncc(C)c1C)=O)CC2 67576,N1(C(COCC#C)=O)CC(CNC(=O)C(F)(F)CO)OC(C)(C)C1 67577,c1(SC)nc(=NC2CC(NC(c3cncnc3)=O)C2)s[nH]1 67578,Cc1c(Cl)sc(Cl)c1C(=O)NCCCC1C=CCC1 67579,C1(CC(=O)N(C2CCN(C(c3cc(C(C)=O)c[nH]3)=O)C2)CC)CC2CCC1CC2 67580,N1(C(c2cc(OC)n[nH]2)=O)CCCC(CNC(=O)C(O)Cc2cnc[nH]2)C1 67581,C1(CC=C)(C(=O)NC2(CCO)CCC2)CCN(C(=O)CN2CCNC(=O)C2)C1 67582,c1(NC(C2CCCN(C(c3c(C)ncn3C)=O)C2)C)cc(=O)n(C(C)C)c(O)n1 67583,N1(C(CN(CC)CC)=O)CC(CNC(=O)CCc2ccc(SC)cc2)C2(CC2)C1 67584,N1(C(C(C#N)=CC(C)C)=O)C2CCC1CC(NC(c1c[nH]nc1C1CC1)=O)C2 67585,N1(C(C2CC(OCC)C2)=O)CCN(C(c2cc(C(F)F)[nH]n2)=O)C2(CC2)C1 67586,C1(NC(C2CC(CC)C2)=O)COCCN(C(c2c(N)cccc2Cl)=O)C1 67587,CC1CCOC(C(=O)NCCN(C2CCCCC2)C(c2cc(=O)cc[nH]2)=O)C1 67588,C1(NC(c2ccnc(N3CCCC3)n2)=O)CCCN(C(c2ccoc2)=O)C1 67589,C1(C(=O)NCC2CCC(C)C2)(OC)CCN(C(=O)C=NOC)C1 67590,N1(C(CC=CC)=O)CC(CNC(c2cc(CO)[nH]n2)=O)CC1(C)C 67591,C(=O)(CCCCC1CC1)NC(c1ccccc1)CNC(c1ncc(CC)s1)=O 67592,N1(CCOCCCC)CC(=O)N(CCN2CCCS2(=O)=O)C1=O 67593,N1(C(C2C(C)C2)=O)CC2(C=C(C(=O)NCP(C)(C)=O)CO2)C1 67594,N1(c2cc(COC)ncn2)CCCN(CCC(=O)N(C)C(C)C)CC1 67595,c1(OCC(=O)N(CCCCN(C(C(CCC)O)=O)C)C)c(C)cccc1Cl 67596,c1(CCN(CC(O)CN(C(=O)C(F)C(F)(F)F)C)C)ccc(C#N)cc1 67597,C1(NC(=O)C=CC=C(Cl)Cl)CC2(CCCCN2C(=O)CCCC2CC2)C1 67598,N1(C(=O)COCc2nc[nH]n2)CCC2(CCCN(C(=O)CC3CCOC3=O)C2)C1 67599,CCC(C)C(=O)N(C1CCCC1)CCNC(=O)C(C)(O)C1CCOCC1 67600,C(=O)(C1=CCCOCC1)NC1(C(=O)NCc2ccsc2)C(C)CCC1 67601,N1(C(CNC(=O)CC2CC(F)(F)C2)=O)CCOCC1C(=O)NCc1ccccc1 67602,N1(CC)C(=O)CCC1CC(=O)N(CC(O)CNC(=O)C(Cl)=CCl)C 67603,C1(CNC(C(CC=CC)C)=O)CN(C(=O)COC2(C)CCCC2)CC1(C)C 67604,N1(C(CSCCCC)=O)CCCCC(CCC(N2CCC(F)(C#N)C2)=O)C1 67605,c1(C(=O)NC2CN(C(C3C(=C)CC3)=O)C(C)CC2)cn(C(C)C)c(=O)nc1O 67606,c1(NC(N(C)C)=O)cccc(C(N2CCOC(C(C)(C)C)C2)=O)n1 67607,S(=O)(=O)(c1cc(F)c(F)c(F)c1)N1CCC(C)(C(=O)Nc2ccc(O)cc2O)C1 67608,C1(NC(Cc2n(C(C)C)cnn2)=O)CCC(C)N(C(=O)CC2(C)OCCO2)C1 67609,N1(C(c2cc(CC)[nH]n2)=O)CCC(NC(c2ccc(C(C)C)s2)=O)C(C(C)C)C1 67610,CC1=C(C(=O)NC2CCN(C(=O)C3CC3)C(C)C2)C(C)n2nnnc2N1C 67611,CCCCCCC(C)NC(=O)C(C)=CCNC(c1coc(C2CC2)n1)=O 67612,N1(C(CCN(C)CC)=O)CCCC(CCNC(c2n[nH]c3c2CCC3)=O)CC1 67613,c1(C(N2CC3(CCCN(C(C4C(C)C4)=O)C3)C2)=O)ccc2c(Cl)nccc2c1 67614,C(=O)(CCC(F)(F)C(F)F)NC1CN(C(c2ccn(CCC)n2)=O)CC(O)C1 67615,c1(CNCc2cccc(OC)c2OC(F)F)ccc(C)c(F)c1F 67616,c1(OC)ccc(C(N2CC(O)(C3CCCN3C(=O)CC(C)OC)C2)=O)cn1 67617,C12(C(=O)NCC(C)CNC(=O)Cc3ccsn3)CCCCC(F)(C1)C2 67618,c1(C(N2CC(C)C(CNC(=O)CCn3cnnn3)C2)=O)nn2c(c1Br)CCC2 67619,c1(C(=O)NC2C(C)CN(c3nccc(Br)n3)C2)cc2ccccc2cc1O 67620,C12(C(N(CC(C)NC(C3C(OCC)CC3)=O)C)=O)CC3CC(C(=O)N1)C2C3 67621,C(=O)(C1CC(=O)c2ccccc21)NCC(C)C(=O)OC(C)(C)C 67622,C1(NC(=O)Cn2ccnn2)C=CC(CNC(c2csc(O)n2)=O)C1 67623,c1(OC)ccc(CC(N2CC(NC(c3ccc[nH]3)=O)CC(C)C2)=O)c(F)c1 67624,C1(NC(CCCCSC)=O)CCC2CN(c3cc4nnc(C)n4cn3)CCC2C1 67625,c1(OCC)cc(C(C(=O)Nc2ccccc2Cl)N(c2cccc(Cl)n2)C)ccn1 67626,C(CC(=O)Nc1cccc(Cl)c1O)(C(C)(C)C)NC(c1cnc(C)o1)=O 67627,CC(C)CC(C(=O)NC1C2CN(C(C3CCCC(C)(C)CC3)=O)CC12)C(N)=O 67628,CCC(O)(C(=O)NCCN(C(=O)CC(C)(O)c1ccccc1)C)c1ccccc1 67629,C(CC(=O)N(CC(O)C1CC1)C)N(CC(C)C)C(C)=O 67630,Cc1c(C(N2CCCC(C(C)C)C2)C(=O)NC2CCCCC2)cccc1Cl 67631,C1(N(C(C(C)NC(CC)=O)=O)CCO)CCCN(C(c2cc(CF)on2)=O)C1 67632,c1(-c2cn(C(C(=O)NCC(CC)N(C)C)C)nn2)cccc2ncoc12 67633,N1(C(CCCCC=CC)=O)CCC(NC(=O)COc2cccnc2)C(CO)CC1 67634,N1(C(c2ccc(C(C)C)cn2)=O)CC(CNC(=O)CP(C)(C)=O)C2(CCC2)C1 67635,c1(CC(=O)NCC2C(NC(c3c(CC)csc3)=O)CCC2)ccc(OC)c(Cl)c1 67636,C1(C(=O)NC(c2nc[nH]n2)CC)CCCN1C(=O)CC1CCSC1 67637,N1(C(C2(C)CCC(=O)N2)=O)CCC2CC(NC(c3ccc(F)cc3)=O)CCC2C1 67638,C1(NC(=O)CC2CC2(Cl)Cl)CN(C(C2CCC(F)(F)CC2)=O)C2(CCOCC2)C1 67639,c1(C(N2CC(N(C(=O)Cc3cccc(O)c3)C)C2)=O)ccnn(C)c1=O 67640,C1(N(C(C=CC(=O)OCC)=O)C)CCCCC1N(C)C(C1CC1F)=O 67641,c1(SC(C)C(=O)NCC(C)(O)CNC(=O)CCc2ccn(C)n2)ccccn1 67642,n1(CC(=O)NC(N2CCN(C(C3CCC3)=O)CC2)C)ncc2ccccc12 67643,N1(C(C2CN(C(c3cc(C(C)C)[nH]n3)=O)CC(F)C2)=O)Cc2ccccc2C1 67644,C1(C(=O)NC2CCCN(C(c3ccc(C(C)C)s3)=O)CC2)CC2(CCCC2)CO1 67645,Nc1cc(Cl)cc(F)c1C(N1CCCN(C(c2cccc(O)n2)=O)CC1)=O 67646,CC1CN(C(c2c(Cl)ccnc2O)=O)c2cnccc2NC1=O 67647,C1(CN(C(=O)CN2CC(=O)NC2=O)C)COCCN1C(C1(C)CC1(F)F)=O 67648,C(=O)(C(C)CCCC(C)C)NCCN(C(c1c(N)ccc(OCC)c1)=O)C 67649,N1(C(Cn2ccc(C)n2)=O)CCC12CCCN(C(c1n[nH]c(C)c1C)=O)C2 67650,c1(C(=O)NCCOC2CCN(C(CC(C)SC)=O)CC2)ccc(C)cc1[N+](=O)[O-] 67651,c1(C(N(CCCCN(C)C(C2CC(F)C2)=O)C)=O)cc(N)cc(F)c1 67652,CCC(C)CCCC(=O)N1CC2CCC(C1)N2C(c1cnsn1)=O 67653,c1(C(C)OCC)nc(C)c(CS(=O)(=O)Cc2csc(-c3ccsc3)n2)s1 67654,C(=O)(C(CS(=O)(=O)C(C)C)NC(=O)C=Cc1cccc(OC(C)C)c1)OC 67655,C(C)(CC(=O)NCC1CC(F)CN1C(=O)Cc1ccccc1F)(C(F)F)N(C)C 67656,N1(C(C2C(C(=O)NC(CCC)C)C2)=O)CCN(c2ccc(Cl)nn2)CC1 67657,N#CC1(C(N2CCC(NC(C3CCCC(C(N)=O)C3)=O)C2)=O)CCCO1 67658,N1(C(C(=O)NCC)=O)CCC(O)(C2(NC(c3cnc4ncnn4c3C)=O)CC2)CC1 67659,CN1CCCCCC1C(=O)Nc1ccc(Oc2cccc(C#N)c2)cc1 67660,c1(C(=O)O)ccnc(CNC(CC2CCCC2)Cc2ccc(F)cc2)c1 67661,C#CC1(C(=O)NCC(C)S(N)(=O)=O)CCN(C(C2CC2(C)C(F)F)=O)C1 67662,C1(NC(c2ccc3ncc(Br)cc3c2)=O)CCOC2(CCCOC2)C1 67663,C1(NC(C(C=C)O)=O)CCCC12CCN(C(=O)COCC(=O)OC(C)(C)C)CC2 67664,CC1CN(C(=O)C2=COCC2)CC1CNC(C1OCCC1c1cnn(C)c1)=O 67665,c1(C(N(CCCCNC(C2COCC(C)O2)=O)C)=O)ccnc(C(F)(F)F)c1F 67666,c1(C(=O)NCC(C)N(C)C(c2ccnc(Cn3cnnc3)c2)=O)nnn(C)c1N 67667,N1(CC(=O)NCCC(C)N(C(=O)C=Cc2cscn2)C)CCC(CO)CC1 67668,C12(N)CC3CCC(C1C2)N3CCC.C12(C(C(C(COC)OC)=O)=O)CCOC(C)(C1)C2 67669,c1(OCC)cc(C(N2CCC(C(=O)NC3CC3(F)F)C(O)C2)=O)ccc1OC 67670,Cc1nccnc1C(=O)NC(CC1CCCC1)C(=O)NC(C)CC(F)(F)F 67671,c1(CC(=O)NCCC(C)NC(=O)Cc2ccc(F)cc2)ccc(C#N)nc1 67672,C#Cc1cccc(CC(N2CC3CC(N(C(=O)Cc4cc[nH]n4)C)C2C3)=O)c1 67673,C1(NC(C(C2CC2)OCC)=O)CCN(C(c2ncc(C)cc2OC)=O)CC1CC 67674,c1(C(c2nnnn2CC(F)F)NCC(=C)CC)c(N(C)C)ccnc1Br 67675,N1(Cc2nc(C)sc2C)CCC(NC(c2cccc([N+](=O)[O-])c2)=O)CC(C)(C)C1 67676,C(CCN=c1[nH]c2cc(C(N)=O)ccc2s1)Oc1c(OC)ccc(CN)c1 67677,C12(C(=O)NCC3C(NC(CCC(=C)Cl)=O)CCCC3)CCCCC1C2(F)F 67678,N12CC3(CC(C3)CC(=O)N(C)CC3(CC(=C)C3)C1=O)C2.c1(CC)nc(C)no1 67679,N1(C(CC(=O)NC)=O)CC(C)CN(C(c2ccc(NC)cn2)=O)CC1C 67680,C1(C(c2ccccn2)Nc2ccc(CC(C)C)cc2)CCC(F)(F)CC1 67681,c1(N(C(c2c(CNC(c3c(CC)nc(C)o3)=O)cc[nH]2)=O)CC)ccc(C)c(C)c1 67682,c1(NC2CCN(CC=C)CC2)nc(N2CCC3(CCCN3C)C2)nc2sccc12 67683,c1(C(=O)NC(C2N(C(CCc3nc(C)sc3)=O)CCC2)C)cc(C)c(C)o1 67684,C1(CNC(Cn2ncc(CC)c2)=O)CN(C(=O)CSC(F)F)CCC1C 67685,CC1(C)C(Nc2ccnc(N3CCC(c4ccc(Cl)cc4)CC3)n2)CC1O 67686,C(=O)(CC(C)CCC=CC)NC(CCCC)CNC(=O)Cc1cc(C2CC2)no1 67687,CCC(C)C(=O)C(=O)N1CC(C(=O)NC2CCN(C3CC3)C2=O)C(F)(F)C1 67688,C1(NC(C(CN(C)C)O)=O)(CO)CCCN(C(=O)CCCC2CCCC2)C1 67689,c1(N(C(CC)=O)CC)ccc(O)c(C(N2CCN(C(=O)Cc3ccco3)CC2)=O)c1 67690,C1(C(=O)NCC2N(C(c3c[nH]c(=N)s3)=O)CCC2)CCN(CCF)CC1 67691,C#CCCC(C(=O)NCCC(C)C(=O)OC)NC(c1cc(F)ccc1C)=O 67692,c1(CC(=O)NCC2(O)CCN(C(C(C)CF)=O)C2)ccc(Br)c(F)c1 67693,C=CCC(CC(=O)N1CCN(C)C(CC)C1)NC(c1c[nH]nc1Cl)=O 67694,N1(C(C2CCN(C(C3(COCC)CCCC3)=O)C2)=O)CCC(CC(C)O)CC1 67695,C1(C(N(C)CC2CN(C(c3cnn(C)c3N)=O)CCO2)=O)CCN2CCOCC12 67696,C1(NC(c2n(CC)ccn2)=O)COC2(C1)CN(C(c1c[nH]c(C#N)c1C)=O)C2 67697,N1(C(CNC=O)=O)CCN(C(CNC(=O)CC2CCC(=O)N2)C(F)F)CC1 67698,C1(N(C)C)CCCN(C(=O)C(O)C2CN(C(C3(O)CCCCC3)=O)C2)CC1 67699,CC1CCCCC1NCCNCCCCCCNC(=O)OC(C)(C)C 67700,Cc1nnc2n1CC(C(=O)NCCCOCCNC(c1ccncn1)=O)C2 67701,C1(C(=O)Nc2ccc(OC)c(N3CCOC3=O)c2)Cc2ccc(F)cc2C1 67702,C1(NC(CCc2n(C)ccn2)=O)CCCCC1NC(=O)CCN1C(=O)CCC1=O 67703,c1(COC)nn(C)cc1C(=O)N(CCNC(=O)CN1CCC(C)C1)CC1CC1 67704,c1(C(=O)NCC(C(=O)NCC(COC)O)C)cnn2ccccc12 67705,N1(C(C2ON=C(CC)C2)=O)CC(C(N2CCCC(OC(C)C)C2)=O)C2(CCC2)C1 67706,C1(COC)(CNC(=O)C=CC(C)C)CCCN1C(=O)CCc1nnc(C(F)F)o1 67707,C1(CNC(CCC(=C)Cl)=O)C(C2CC2)CCN1C(c1ccc(C2CC2)nn1)=O 67708,c1(C(N2C(C)CC(CNC(=O)CCc3cnn(C)n3)C2)=O)cc2ncccc2o1 67709,N1(C(CNC(C(CC)CC)=O)=O)CCC(NC(c2coc(O)n2)=O)C(C)C1 67710,c1(C(=O)NC23CC(NC(C(CCSC)O)=O)(C2)C3)ccn2cc(C3CC3)nc2c1 67711,N1(C(C(CCOC)OC)=O)CCN(C)CC1C(=O)NCc1ccnc(O)c1 67712,c1(CCC(=O)NCC2CCN(C(C(C3CCC3)OC)=O)CC2)c(F)cccc1Cl 67713,C=CC(C)(CCOC)C(=O)NCC(C)NC(=O)CCC1CC1 67714,N1(C(c2cc(CC)[nH]n2)=O)CCCC(C)(C)C1C(=O)NCC(CC(C)C)C(C)C 67715,CCS(=O)CCNC(=O)CC1(N(C)C(c2cccn2C2CC2)=O)CC1 67716,c1(C(=O)OCc2ccc(C3CCC3)cc2)c(F)ccnc1F 67717,Cc1coc(CNC(C2CC(NC(C3CCCO3)=O)C2)=O)c1 67718,N1(C(COC)=O)C(C)C2CC1C2NC(c1sccc1C1CC1)=O 67719,C1(NC(c2cc(C)ns2)=O)CCC2CCN(C(=O)CCc3ccccc3Cl)C1C2 67720,Cc1[nH]c(=NCCc2cn(C(C)C)nn2)ccc1C#N.C12CCC(NC1=O)CN2 67721,N1(C(C2N(CC)CC2)=O)CCC(=CCNC(=O)CCCCN2CCOCC2)CC1 67722,N1(C(c2ncc(C)c(C)c2)=O)CC2CCC1CC2NC(c1cnsn1)=O 67723,C1(C(=O)NCC(C(=O)NC2CC(O)C2)O)Cc2nccn2C1 67724,Cn1nnc2c1CCN(c1nnnn1C1CCC(Cc3ccccc3)C1)C2 67725,C1(NC(C(F)=CC)=O)CCN(C(c2ccc(C)cc2C(C)=O)=O)CCC1CO 67726,c1(CCN(C(=O)N)CCO)ccc(F)c(Br)c1.c1(N2CCOCC2)ncc(Br)s1 67727,N1(C(c2cnc(OC)s2)=O)CCC(C(C)NC(C2CCCOCC2)=O)CC1 67728,c1(C(=O)NC(C(C)NC(c2ccc(C(C)C)cc2)=O)CO)cc2occc2n1C 67729,C1(C(=O)NC(c2ccncn2)C)CN(C(=O)CCC2CCCOC2)C2(CCC2)C1 67730,C(C(=O)N1CCCC1C(C)NC(=O)COC1CCC1)(C(C)C)SC 67731,CC1(C)OCc2c1n[nH]c2C(=O)NCC1CCC1NC(c1csc2nnsc12)=O 67732,CC(CCC(=O)NC1CC1)NC(C1CCCN1C=O)=O 67733,N1(C(C2(C)C(C)(C)C2)=O)CC2CC2(CNC(c2cccc(-n3cncn3)c2)=O)C1 67734,C(=O)(C=CS(F)(F)(F)(F)F)NCCN(C(CC(CC)(C)C)=O)CC 67735,C1(NC(c2n(C)c(S)nc2)=O)CN(C(C2CCCS(=O)(=O)C2)=O)C2CCCC12 67736,N(C(=NCCc1cnccn1)N)C1C(C)C1.c1(C2CCCC2)ccc(=N)[nH]c1 67737,C1(CC(N2C(CN(c3ccncn3)C)CCC2)=O)CCC2CC12 67738,N1(CC)C(C)CN(C(C2CC(O)CN2C(=O)C(c2cnn(C)c2)C)=O)CC1C 67739,C(C)(CCC(F)(F)F)NC(CC1(NC(c2n(CC)c(O)nc2)=O)CC1)=O 67740,c1(C(=O)Nc2cn(C)c(C(=O)O)n2)c(CN2CCCC2CO)ccc(Cl)c1Cl 67741,CCN(OC)C(=O)C(C1CCCC1)NC(c1sc(F)cc1C)=O 67742,c1(OC(C)C)ccc(C(=O)NCC2C=CCN2C(=O)C(F)C(C)C)nc1 67743,c1(NCCC2CCN(CC(=O)NCC(N3CCCC3)=O)CC2)cc(O)cc(O)c1 67744,C(=O)(C(C)(C)CS(N)(=O)=O)NCCOC1CCN(C(c2c(SC)cnn2C)=O)C1 67745,Cc1[nH]nc(CO)c1C(=O)O.N1(CC(=O)NC(C(N)=O)C2CCCC2)CCC(N)CC1 67746,c1(C(=O)NC2C(C)CN(C(=O)CCP(C)(C)=O)CC2)ccc2c(c1)NC(=O)CO2 67747,CCCC(CC(=O)NC1CCC(=O)NC1C)NC(=O)Cc1cnsc1 67748,CC1CN(C(C2CCN2C(C)(C)C)=O)CC1CNC(=O)C(c1ccccc1)O 67749,N1(C(c2ccc(N3CC(O)C3)cc2)=O)CCN(Cc2ccc(I)c(O)c2)C2CC12 67750,c1(C(N2CCC(N(C(=O)CCn3ccnc3C)CC)C2)=O)cc(Cl)cc(F)c1N 67751,c1(C(=O)OC)cnc(COC(=O)NCC2CC(OC)C2)n1C 67752,C(=O)(CCCCC(N)=O)N1CCC(C)C1CNC(c1cnc2[nH]cnc2c1)=O 67753,C1(CNC(Cn2cc(COCC(=O)OC)nn2)=O)OCCNC(=O)C1 67754,C1(OC)CC(CNC(=O)Cc2cc(C3CC3)on2)N(C(C2CCC(F)(F)C2)=O)C1 67755,c1(CN(C)CCN(C(C(C)OCCOC)=O)C)nnc(C)cc1O.C(C)(=O)O 67756,c1(C(N2C(CNC(COCCC)=O)C=CC2)=O)nn(C(C)C)cc1Br 67757,CC1C(NC(=O)C2=COCCC2)CCCN1C(c1ncc(F)cc1N)=O 67758,N1(C(C2(C)CC2Br)=O)CCCC(n2cc(C(=O)NCCSCCCO)nn2)C1 67759,n1(CC(N2CCC(NC(C3C(OCC)C3)=O)(CF)C2)=O)ncc2cc(C)cnc12 67760,C(CC(=O)NCC(F)CNC(c1cc(C)ccn1)=O)(C(C)C)OCC 67761,C1(C)(NC(C(C)SCCCC)=O)CCCN(C(=O)Cn2ccc(C)cc2=O)C1 67762,N1(C(c2cnccc2Cl)=O)CCCC12CN(Cc1ccc(Cl)nc1Cl)C2 67763,C1(C(C)C)CN(C(=O)CCCn2cccc2)CCCN1C(=O)CS(C)(=O)=O 67764,c1(NCCN(C(C)C2CC2)CC)ccc(S(=O)(=O)NCCO)c(Cl)c1.C(C)(CC#N)N 67765,c1(C(N(C(C)CNC(c2cnc(C)n2C)=O)CC)=O)cc(C)c2nc(C)cn2n1 67766,C1(C(=O)NC2COC2)CN(CCNC(CCCSCC)=O)CCO1.C1CS1 67767,c1(CC(N2C(C(C)(C)NC(CCCCOC)=O)CCC2)=O)cccc(O)c1C 67768,N1(C(COC)=O)CCC2(CCN(C(c3ccc(C(=O)OC)s3)=O)CC2)C1 67769,C1(NC(C(CC)F)=O)CCOC12CCN(C(c1nc(C)c(C)nc1C)=O)CC2 67770,O=C(CCCC(F)(F)CO)NC1CC2CCC(C1F)N2C(C1CC2(CCC2)C1)=O 67771,CC(O)C(C)(C)CNC(c1cc(CNC(=O)C(O)CCN(C)C)no1)=O 67772,c1(CC)nn(C)c(C(N2CCC(CO)(NCc3ccccc3Br)CC2)=O)c1Br 67773,C1(C)(C(=O)NC2(CN(C(=O)CC(F)(F)F)C)CC2)CCOC12CC2(F)F 67774,CC(C)(C)C(=O)N1CSCC1C(N(CC(c1cccs1)=O)C)=O 67775,CCCCCCC(C)C(=O)NC(CN(C(c1cn2c(n1)CCC2)=O)CC)CC 67776,c1(C(N2C(CNC(CC=C(C)C)=O)C=CC2)=O)ccc(C)c(S(C)(=O)=O)c1 67777,C1(C(N(CCCC)C)=O)OCCC1CNC(C1CC1C)=O 67778,Cc1cc(Br)cc(Cl)c1NC(=O)NCc1nccn1C 67779,c1(C(C(=O)NC)N(C(C)CCO)C)ccc(Cl)c(C)c1 67780,c1(SCC(=O)NC2CC(NC(=O)CC34CCCC3C4)C2)cc(Cl)ccc1Cl 67781,N1(C(C(C)C(=O)N2CCOCC2)=O)CCCCCC(NC(C2CCOCC2)=O)C1 67782,N1(C(C2(COC)CN(C(COCCC#C)=O)C2)=O)CCCCC(OC)C1 67783,C(=O)(CC(C)(C)CNC(c1scc(C)c1C)=O)N1C(C(N)=O)CC(OC)C1 67784,CC1(CNC(C2CCNC2=O)=O)CCN(C(C2SCCCS2)=O)C1 67785,CCC(C)CCCCC(=O)NCCCCCN(C)C(C1(OC)CCC(C)(C)C1)=O 67786,C(=O)(C1=CCCOC1)NC1C(CC)N(C(c2cnc(CC(C)C)[nH]2)=O)CC1 67787,N1(C(CCC=CC(C)C)=O)Cc2[nH]nc(C(N3C(C)CCC3(C)C)=O)c2C1 67788,C1(NC(CCS(=O)(=O)NC)=O)(CNC(c2ncccc2C)=O)CC2CCC1CC2 67789,c1(OC)ccc(OC)c(CCC(=O)N2CCC2CNC(C2Cc3nccn3C2)=O)c1 67790,C12(C(=O)NCc3ccc(COC)c(F)c3)CC3CC(C1)C(=O)C(C3)C2 67791,C1(OCC)CN(c2ccc(N3CCN(C)CC3)nn2)CC1c1nn[nH]n1 67792,N1(C(c2cccc(NC(C)=O)c2C)=O)CCCC12CN(Cc1ncsc1C)C2 67793,C1(C)(OCC(=O)NCC(C)CNC(C2CCCSC2)=O)CCOCC1 67794,N1(C(C2(n3cc(C(c4ncc[nH]c4=O)N)nn3)CC2)=O)CC2CC1CCN2C(N)=O 67795,c1(C(N2CC(c3cn(CCN4CCOCC4)nn3)C2)=O)cnc(O)o1 67796,C1(NCCN(C(CCCC)=O)CC)CCCCN1C(=O)Cc1scnc1C 67797,CCC(CC)C(C(=O)N1CCC(C(=O)NCCCSC)(CC)CC1)OC 67798,CC1CCN(C(c2cnn(C)c2C(F)F)=O)CC1NC(C1CC(F)(CO)C1)=O 67799,c1(C(N2CCCC2CCNC(C2CC(O)C2)=O)=O)cc(Cl)c2[nH]c(O)nc2c1 67800,c1(C(N(C)Cc2c(C)cco2)=O)ccnc(CNC(=O)COc2ccsn2)c1 67801,c1(C(c2n(C3(C)CC3)nnn2)NCC2CCC3(CC3)C2)cccc2sccc12 67802,c1(C(N(C)CCOCCNC(=O)Cc2cccs2)=O)ncc(Cl)s1 67803,c1(C2C(NC(=O)C(N3CC(O)(C(F)F)C3)=O)C2)cc(F)ccc1F 67804,c1(C(N(CCCCNC(C(C(COC)C)C)=O)C)=O)cnn(C)c1S(N)(=O)=O 67805,C1(C(=O)NC2(C)CN(C(=O)CO)C2)C2Cc3ccccc3C12 67806,c1(C(=O)NCC(CNC(Cc2cn(CC)nc2)=O)(C)C)noc2cc(F)ccc12 67807,CC(CC(=O)NC1COCC1CNC(=O)CC1CCCSC1)N(C)C 67808,CCCC(CCC)C(=O)N(C1CCN(C(C2(CCOC)CCCC2)=O)C1)C 67809,c1(OC)ccc(CCC(N2CCC(NC(=O)C(O)CSC)C2(C)C)=O)cc1OC 67810,c1(C(=O)NC(C2(CNC(C3(O)CC3)=O)CC2)C)cc2c(cc1N)CCCC2 67811,C1(NC(=O)CC2CCCNC2=O)CN(C(=O)CSC2CC2)Cc2nccn2C1 67812,CC(C)C(C)(O)CNC(c1sccc1CNC(=O)C=Cc1cccnc1)=O 67813,Cc1nc2c(s1)CCCC2CN(C)C(c1cnccc1C1OCCO1)=O 67814,C1(C(=O)NCCCN(C(CSCC#C)=O)C2CC2)CC(C)CC(C)C1.C(=O)NC 67815,C#Cc1cn(C)nc1C(N1CCC1CNC(c1cccc(O)c1C)=O)=O 67816,c1(C(N(CCOCCC(=O)N(CCCC)CCO)C)=O)cc(C(F)(F)F)n[nH]1 67817,n1(CC(N2CC(C)(NC(CC=C)=O)C2)=O)cc(C)c(O)nc1=O 67818,C(=O)(CCC(C)(C)[N+](=O)[O-])NC(C(=O)NCC(CC(C)O)(C)C)CCN(C)C 67819,C(=O)(CCCCC(C)C)NCCNC(C1CC(CCC)OCC1)=O.CC 67820,N1(C(CCCOC)=O)CCN(C(=O)CCc2nnc(S)nc2O)CC12CC2 67821,C1(CC)CN(C)CCCN1C(=O)C(C(C)C)NC(c1c[nH]c(=NC)s1)=O 67822,C=CC1CCCN(C(=O)COC2CC(CNC(c3coc(C(N)=O)c3)=O)C2)C1 67823,CCCCC(C)(F)C(=O)NCC(C)(CNC(=O)CC1(n2ccnc2)CC1)OC 67824,N1(C(c2ccc(SC)o2)=O)CC(C(=O)NCC(c2ccccn2)N(C)C)C2(CC2)C1 67825,Cc1cc(N(C(=O)CC2(NC(c3cnc(S)nc3)=O)CC2)C)cc(C)c1 67826,c1(C(N2CC(CNC(C3(Cl)CC3)=O)C(O)C2)=O)cc(F)c(C(F)(F)F)c(F)c1 67827,C=CCC(CC)C(=O)NCCC(O)C(=O)N(C)C(c1ccccn1)C 67828,C1(N(C(=O)C(C)(C)CC(F)F)C)CC2CCCC1N2C 67829,CCCC(C)CC(=O)NCC(C)(CC)C(=O)NC1CC(O)CC1O 67830,n1(CC(=O)NCCCCNC(C2CC2F)=O)nnc(-c2ccccc2)n1 67831,CC(CC1CCC1)C(=O)NC1CCN(C(C2CC(F)(F)C2)=O)C1 67832,c1(OC)ccc(C(=O)NC(CNC(=O)CC(C)(C)C#N)C(C)(C)C)cc1F 67833,c1(C(=O)NCCCN(C(C(C)OCCC#C)=O)C)c(OC)ccc(F)c1Br 67834,CC1(C)OCCC1C(N1CC(OC2CCN(C(=O)COCC3CC3)CC2)C1)=O 67835,c1(C(=O)NCC2(COC)CCN(C(C(C=C)C)=O)C2)cnc(O)c(F)c1 67836,N1(C(C(c2cccc(Cl)c2)CC)=O)CCCCCC1CNC(c1cnc(S)[nH]1)=O 67837,C1(CNC(c2nc(CCC)sc2)=O)CN(C(c2nocc2Cl)=O)CCC12CCC2 67838,C1(C(=O)NCC=CCNC(COC(C)C)=O)CCCC(C2CC2)O1 67839,N1(C(C2N(CC(c3ccc(O)cc3)=O)CCOC2)=O)CCOC(C(F)F)CC1 67840,c1(C(=O)NC)ccc(CN2CC3C(NC(C4CCCC4)=O)C3C2)cc1 67841,C(CC(=O)NC1CCCC2(C1)N=N2)(C(F)(F)F)NC(C(CC)=CCCC)=O 67842,C(C1CCCN1C(=O)C=CC(=O)OC)=CC(N1CC(C)(NC(=O)C=CCF)C1)=O 67843,c1(C(=O)NC2C3(CCN(C(CCC)=O)C3)CCC2)ccc2ccc(Br)cc2n1 67844,N1(C(C2(C)C(C)OCC2)=O)CCC(CNC(C2(c3ccno3)CC2)=O)C(O)C1 67845,C(CCCC(=O)N1CCOC(C2CC2)C1)N(C)C 67846,c1(CNC(C2C(CNC(c3c(C(N)=O)c[nH]n3)=O)C2)=O)ccnc(F)c1F 67847,C1(CCC(N2C(C(=O)NC)CC2)=O)CCC(NC(c2cc(C(C)=O)on2)=O)C1 67848,c1(-c2cn(CCN(C(C3C(=C)C3)=O)C)nn2)cccc(Cl)c1Cl 67849,S(=O)(=O)(c1cccs1)NC(C)C(N1CCOC(CNC(C2(Cl)CC2)=O)C1)=O 67850,C1(CNC(CCCc2scc(C)n2)=O)CN(C(=O)C(F)(F)C(F)F)CCC1(C)C 67851,C1(OC)COCCC1CC(=O)NCC(C)(C)CNC(c1scc(C)c1Cl)=O 67852,C1(CC(=O)N(C2(CC)CC2)C)CN(C(=O)C(CO)NC(N)=O)CC1C 67853,CC(CN(C)C)CC(=O)NC(C)(C)C(=O)NC1CC(=O)N(C(C)C)C1 67854,C1(NC(c2ccc(Cl)o2)=O)C2CN(C(=O)Cc3ccccn3)CC12 67855,C(c1ccc(OC(=O)NNC(C2CC3(CC3)C(=O)O2)=O)c(OC)c1)=CC.C1CN1 67856,N1(C(CN(CCCCCC)C)=O)CC2CC1C2CNC(=O)CC(C)(C)O 67857,c1(OCC)nc(C(=O)NC2(C(=O)NC3CC(C(N)=O)C3)CC2(C)C)co1 67858,CC(C)C(CNC(C12CC(C)(C1)C2)=O)NC(C1C(C)C1(F)F)=O 67859,N1(C(C2=CC(C)(CC)C2)=O)Cc2ccccc2C(NC(C2(F)CCCC2)=O)C1 67860,CC1CN(CCNC(N2CC(C)(C)CC2CO)=O)S(=O)(=O)C1 67861,N(C)(C1CCc2c(Cl)cccc21)C(c1ccc(OC)c(F)c1)C(=O)NC(C)C 67862,C1(NC(C(C2CC2)NC(C2OCC(C)(C)C2)=O)=O)CCCN(O)C1=O 67863,c1(C(N(CC(C)N(C)C(C2CC2CF)=O)C)=O)ccc2c(c1)C(=O)CCS2 67864,C1(C2CC2)(CNC(CC2C(C)(C)CC2)=O)CCN(C(c2ccc(Cl)cc2O)=O)C1 67865,C1(NC(c2ccn(CCCC)n2)=O)CN(C(=O)CCn2cccnc2=O)CC1O 67866,c1(C(N2CC(O)CC2C2CCCCC2)C(=O)NCCCSC)ccccc1Br 67867,c1(CN2C(C(=O)Nc3nc(-c4ccccc4)cs3)CCC2)ccc(Br)cc1O 67868,C12(CNC(C3C(C=C)CC3)=O)CCC(CC1)N(C(C1CC3CC3C1)=O)C2 67869,C(=O)(CC1CCc2ccccc21)NC(C1(CNC(c2cc(C)c(C)o2)=O)CC1)C 67870,C1(C(=O)NCCC(CC)O)CC2CC2N1C(C1COCC(C)O1)=O 67871,c1(CC(=O)NC2C(NC(C3(C(N)=O)CC3)=O)C2)ccc(Br)cc1Cl 67872,C(=O)(CC(C(F)F)C(C)(C)C)NC(CNC(c1c(N(C)C)cccn1)=O)C1CC1 67873,c1(OCC)ncccc1C(N1CCC(C)C1C(=O)NOCc1ccncc1F)=O 67874,N1(C(C=CCC)=O)CCN(C(=O)CNC(N)=O)CC1CC 67875,c1(NC2C(NC(C(C)SCC)=O)CCCC2)ncnc2cnccc12 67876,c1(NC(=O)NCC(c2ccc(C)o2)C)ccc(-c2ccccc2)nc1 67877,C1(CC=C)(NC(=O)Cc2cccc(Cl)c2)CCCN(C(c2cocc2C)=O)C1 67878,C1(CNC(CC2CC(C)(C)OC2)=O)CC2CCC(C1)N2c1nc(C(F)(F)F)ns1 67879,c1(N(C)CC2CCCN2C(=O)CC2CCOCC2)ncccc1S(C)(=O)=O 67880,C1(c2n(C)nnn2)(NCCOCC2CC2)CC2COC1C2 67881,C(=O)(CC1=NNC(=O)C1)NC1CCN(CCNC(C2(C=C)CCC2)=O)CC1 67882,c1(C(=O)NCC(C(C)C)NC(C2(O)CCSC2)=O)cscc1S(C)(=O)=O 67883,C(C)(C(C)(C)C(=O)NC1C(C)(C)C1(C)C)NC(c1ccc(CC)s1)=O 67884,N1(C(c2c(C)snc2)=O)CCC2CCN(C(c3cc4n(c3)CCCC4)=O)C2C1 67885,CC1Cc2cccc(C(=O)NC3(CNC(c4ccc(F)cc4)=O)CCC3)c2O1 67886,N1(C(Cc2cccc(C)n2)C)CCC(O)C(C(=O)N(C)Cc2cccc(F)c2)C1 67887,C1(NC(=O)Cc2c[nH]nc2O)C=CCN(C(C2(F)CC2c2ccccc2)=O)C1 67888,C(CN=c1[nH]c(=NC(C)c2cc(C)on2)[nH]c2c1SCC2)SCCOC 67889,CCC(O)CC(=O)N1CC(CF)(NC(c2cccc(C(F)F)c2)=O)C1 67890,N1(C(=O)OC(C)(C)C)CCCC12CCN(Cc1c(F)cc(I)cc1F)CC2 67891,C1(NC(Cc2c(C)nc(Cl)cc2)=O)CN(C(=O)C(C)(C)NC(N)=O)CC1C1CC1 67892,C(=O)(CCC(C)(C)c1ccccc1)N(C1CCCC(O)C1)CC 67893,c1(C(=O)NC2CN(C(c3c(CC)noc3)=O)C(C)CC2)cnc(O)c([N+](=O)[O-])c1 67894,C(=O)(C1=CC(O)C(C(=O)N)C1)N1CCC(C(C)N(C)C)CC1.N1(CCS)CCS(=O)CC1 67895,c1(C(=O)NC(CCNC(CCSC)=O)(C)C)cn(C)c(-c2ccccn2)n1 67896,CN1CC2CN(C(=O)NCc3cn4c(n3)CCCC4)CC2(C)C1 67897,N=c1ccc(C(=O)NCC=CCNC(C2CCCN(c3ccccn3)C2)=O)n[nH]1 67898,N1(C(C2CN(C(C3CC4(CSC4)C3)=O)CCO2)=O)CCc2nn[nH]c2C1 67899,CCS(=O)C1CCCCC1NC(=O)C(=O)N(C1CCOC1)C 67900,N1(C(CCC#CC)=O)CCN(C(=O)C=C(C)C(C)C)CC2CCCCC12 67901,N1(C(c2cn(CC=C)nc2)=O)CCC2(CCN(C(=O)C(F)=C3CCCC3)C2)C1 67902,C1(CNC(CC(=O)OC)=O)CN(C(=O)C(n2nccc2C)C)CC12CCC2 67903,C(=O)(C(O)C1CN(C(c2ccoc2)=O)C1)NCC(=C)Cl 67904,c1(CNc2cn(CCOc3c(F)cccc3)cn2)ccc(Br)c(Cl)c1F 67905,c1(C(C(=O)NCC(=C)CCNC(C2CC(C)(F)C2)=O)(C)C)cccc(C)c1 67906,c1(C2(NC(=O)Nc3cc(C)ncc3)CC2)cc(F)ccc1F 67907,C1(C(=O)NC(C(=O)NCC(C(C)C)(C)F)CCC2CCC2)CC2(CCC2O)C1 67908,C(=O)(CC1=CCOCC1)NCC1C(C(=O)NCc2cccc(OC)n2)CC1 67909,N#Cc1ccc(Br)cc1CNCC12CC1CN(C(c1c(F)cc(F)cc1Cl)=O)C2 67910,c1(C(N2C3C(CNC(c4cnn[nH]4)=O)C(C3)C2)=O)cc(Cl)cc(Cl)c1OC(F)F 67911,C1(C(=O)NC2(CC)CC2)CC2(C1)CN(C(c1csc(CO)n1)=O)C2 67912,c1(NC(C2CC3C=CC2C3)=O)cnc2ncc(-c3ccc(OCCO)cc3)cn12 67913,C(C(C(=O)NCC1(F)CC(CO)C1)N(C)C)NC(C1C(C)CC1)=O 67914,c1(-c2cn(CC3(C)CCC3)nn2)nc2ccccc2s1 67915,CC1CCC(NC(c2nc(Cl)ccc2F)=O)CN1c1ncc(F)cn1 67916,CCCCCCC(CC)(CC)C(=O)N(C)CC1CCCN1C(=O)C(F)C(C)(C)O 67917,N1(C(C2C(NC(c3ncn(C(C)C)c3)=O)C2(C)C)=O)CC(S(N)(=O)=O)C1 67918,CC(=O)N1C(=O)C(CCCCNCCC23CCCN2CCC3)c2ccc(Br)cc21 67919,c1(C(N(CC(CNC(c2nc(C)sc2C)=O)C)C)=O)cc(N)cc(O)c1C 67920,C(=O)(C1=Cc2ccc(Cl)cc2OC1)N(C1CCN(C(C2CC(=O)NCC2)=O)C1)CCO 67921,c1(OC)ccc2c(c1)CC1(CC1)N(C(C1C3CC(N)CC13)=O)C2 67922,C(=O)(CC(O)CC(C)C)N(C1CCN(C(c2c(C)cccc2Cl)=O)CC1)CCO 67923,C(=O)(Nn1cnnc1COC)C1N(C(Cn2ncc(CC)c2)=O)CCCC1 67924,CCC(C)CCCCC(=O)NCCN(C(C1CC2CCC1C21CC1)=O)C1CC1 67925,C1(C(=O)NCC(C)Cn2cccn2)CC(=O)CN1C(C1OCCC1(C)C)=O 67926,N1(C(COCCC)=O)CCC(CNC(=O)CCCN=[N+]=[N-])C(C)C1 67927,c1(C(=O)OCC)cn(C)nc1NC(=O)CCN(CC(C)C(C)C)C 67928,N1(C(CN(CC#C)C(C2CN3CCN2CC3)=O)=O)CC2CC(N(C)C)C(C2)C1 67929,c1(CC)cc(C(=O)NCC(C)N(C)Cc2cccc(Cl)c2F)cc(O)n1 67930,C1(C)(C(=O)NC(CC=CC(N2CCCC(CCOC)C2)=O)(C)C)CCC(=O)CC1 67931,C(=O)(CC(C(F)F)NC(=O)Cc1ccns1)NCC(C)SC 67932,Cc1ccc(-c2cc(C(=O)NCCCCC(C)NC(=O)CC(C)(C)F)on2)cc1 67933,c1(CN(CC(CN(C)C)OC)CC=C)cccc(OC)c1 67934,Cn1cncc1CC(N1CC(O)(C(C)(C)CNC(C2CC2F)=O)C1)=O 67935,c1(C(=O)NC2CN(C(C(CCC)N(C)C)=O)CC2C)cncn(C)c1=O 67936,C1(C(N2CC=CC2)=O)CN(C(c2ccc(CO)nc2)=O)CCO1 67937,c1(C(=O)NCC(CNC(C(F)=C(C)C)=O)(C)O)c[nH]nc1[N+](=O)[O-] 67938,CCCC(C)(C)C(=O)NC1CCCC(CNC(c2c[nH]c(Br)c2)=O)C1 67939,c1(C(CNC(=O)CC2CC(C)(C)C2)NC(c2c(C)snc2)=O)ccc(F)cc1F 67940,Cc1cc(NC(N2CCCC2Cc2ccncc2)=O)c(C)n1Cn1cncn1 67941,CC(C)C(F)C(=O)NC12CC1CN(C(c1cnn(C)c1CN1CCOCC1)=O)C2 67942,N1(C(C2C(C(=O)OC)C=C2)=O)CCN(C(=O)Cc2ccccc2F)C(COC)C1 67943,c1(C(N(CC(C)NC(c2cn(CC)nc2C)=O)C)=O)c(C)ccc(N)c1C 67944,C1(NC(c2ccc(F)cc2Cl)=O)CCN(C(=O)CCC2CC2(Cl)Cl)CC(O)C1 67945,C1(NC(C(CCC)OC)=O)CN(C(c2scc(C)c2Cl)=O)CC1N=[N+]=[N-] 67946,C(=O)(C#Cc1ccc(Cl)cc1)N1C(C#N)CCCC1.C12CCCN1C2=O 67947,c1(OC)cc(C)c(CN2CC(C(=O)NCC3CCCO3)CC2CO)cc1OC 67948,C1(NC(c2coc(Br)c2)=O)CCC2CCN(C(=O)CCC3CCCC3)C12 67949,CC1=C(CNC(C2CN(CC(F)F)C2)=O)SCCO1 67950,c1(C(=O)NCC2(C)CCN(C(C3C(C#C)C3)=O)CC2)cc(C)c(F)cc1F 67951,c1(C(N2C(CNC(C(C)OC3CCCC3)=O)CC2)=O)ccc(O)cc1[N+](=O)[O-] 67952,N1(C(Cn2c(C)nnn2)=O)CCN(C(=O)COc2ccc(O)cc2)C(CCO)C1 67953,C1(C(=O)NCC(=O)OCCCC)CC(O)CN1C(c1ccn(C(F)F)n1)=O 67954,C(=O)(C(C)(C1CC1)N(C)C(=O)NC1CCN(C)C1)N(CC)CC1CCCO1 67955,N1(CCOCC)C(=S)NC(c2csc(CN(C)C)n2)C2=C1CCN(C)C2=O 67956,CC1CN(C(=O)CCC(F)(F)F)CC1(C)CNC(=O)CC1(C)CCC1 67957,C12(OCC)CCC(C(N3CCC(CF)(NC(=O)CSCC(N)=O)C3)=O)(CC1)C2 67958,N1(C(Cn2c(C)ccn2)=O)CC(=O)NCC1C(N1CC(CO)CC1CO)=O 67959,N1(C(=O)NC(CC)C)CC(NC2CCCCC2N2CCCC2=O)CCC1C 67960,c1(C(N2CCC(C(CNC(CC(C)SC)=O)F)CC2)=O)n[nH]c2c1CCCCC2 67961,c1(OCCOC)ccc(NC(=O)C(c2cnn(CC(C)C)c2)C)cc1 67962,C1(CN(C2(c3nnnn3CC(F)F)CCCC(C)C2)CC)C2CC3CC(C2)CC1C3 67963,c1(C(N2CCC(N(C(=O)CN3CCC3C)CC#C)CC2)=O)ccc(O)c(F)c1 67964,C12(C(=O)NC(C)CN(C)C(c3ccccc3CO)=O)CC1COC2(C)C 67965,Cc1nn2cc(C(=O)NCC3CN(C(=O)C(C)N4CCC4)C(C)(C)C3)nc2s1 67966,C1(O)(CC)CCN(C(C2C(NC(=O)Cc3cc[nH]c3)C2(C)C)=O)CC1 67967,C1(C(N2CC(CC#C)OCC2)=O)CCN(C(C2CC23CCOCC3)=O)C12CCC2 67968,C1(N(C(=O)NC2CN(CC)C2)C)CCCN(C(c2cc(C)oc2C)=O)C1 67969,C(CC(=O)NCCS(C)(=N)=O)(CC(C)C)NC(c1c(C)cc(C)nc1)=O 67970,C(=O)(CC(C)C(C)(C)C)N1CCC(F)(CNC(c2c(C)n(C)cn2)=O)CC1 67971,C=CCC(CC)C(=O)NCC1(NC(=O)CC2(O)CCOCC2)CCOCC1 67972,c1(C(=O)NCC2(C)CCC(NC(C(=C(C)C3CC3)F)=O)C2)ccc2cc[nH]c2n1 67973,CCC(C(=O)N(CCCN(C)C(c1cc(O)cs1)=O)C)OC1CCCC1 67974,C(=O)(C(C)(C)N(C)C)N1C(C(=O)NC(C=C)C2CCC2)CC1 67975,N1(C(C2C(C)CC2)=O)CCC(CO)(CNC(C2CC(n3cnnc3)C2)=O)CC1 67976,N1(C(COC2(C)CCC2)=O)CC(NC(=O)Cn2cc([N+](=O)[O-])cn2)C2(CC2)C1 67977,C1(CNC(C=CC(C)NC(C=CC(C)(C)SC)=O)=O)CCOC(C)C1 67978,C(=O)(C1=CC2(CCOC2)C1)N1CC2C(CNC(c3c(C)nncc3)=O)C2C1 67979,N1(Cc2c(Br)ccc(OCC)c2)CC2CCN(C(c3cc(C(F)(F)F)c[nH]3)=O)C2C1 67980,c1(C(N2C(C)CCC(NC(c3csc(C#N)c3)=O)C2)=O)ccn2nccc2c1 67981,c1(OC)cc(NC(C23CC2CN(C(c2ncccn2)=O)C3)=O)c([N+](=O)[O-])cn1 67982,C1(CNC(C(c2cccc(F)c2)C)=O)CN(C(C2CC(=O)C2(C)C)=O)CCCO1 67983,Cc1cnc(C)c(C(=O)NCCC(C)CCNC(=O)C(N2CCC(O)CC2)C)c1 67984,N1(C(c2ccc(-c3csc(C)n3)s2)C(=O)NC)CCCN(C2CC2)CC1 67985,Cc1ccncc1C(N1CCC(N(CC(N2CCC(C(=O)N(C)C)CC2)=O)C)C1)=O 67986,c1(C(=O)NC(C(N)=O)C2CCCO2)ccc2nc(S)[nH]c2c1 67987,CC(C)CN=C(NCC(C)(C)C(C)(C)C)N1CCC(C)(F)C1 67988,n1(CCC(=O)N(C(C)CNC(=O)Cc2cnsc2)C)cnccc1=O 67989,c1(C(=O)NCC(CNC(C2CCCC(F)(F)C2)=O)OC)cc(N)ccc1O 67990,CCCCC(C(=O)N1CC(CNC(c2cccnc2N)=O)C1)NC(N)=O 67991,C1(CC(=O)NCCS(CC)=O)N(C(=O)C2=CCCC2C)CCC1(C)C 67992,C(=O)(CCC(F)(F)C(F)F)NCCCNC(CCc1nc(C)sc1)=O 67993,c1(CC)ccc(C(=O)NC(CNC(C2CC2(F)F)=O)CC)cc1[N+](=O)[O-] 67994,c1(OC)cccc2c1C(C(=O)NCC1CC1NC(c1ncccc1OC)=O)CC2 67995,C1(CCNC(C2C(CCOC)C2)=O)(OCC)CN(C(=O)C(c2ccn(C)c2)C)C1 67996,CC(C(=O)NC1CC(CNC(=O)C=Cc2cnc(C(C)(C)C)s2)C1)S(N)(=O)=O 67997,C(=O)(CCCCCOC)NCCn1cc(C(=O)NC(CC)(C)C(N)=O)nn1 67998,CC1(C(=O)NC(C2CCCCC2)CNC(C2CCCCS2)=O)CC2(CCC2)C1 67999,O=C1CCC(O)CN1Cc1cn(CC2CCN2C(C2CC2c2cccnc2)=O)nn1 68000,CCC(C)CC(C(=O)NCCCn1cc(C)cn1)NC(c1cnc2n1CCC2)=O 68001,C(N=c1[nH]ccnc1F)C1CN(C(C2(C)CCCOC2)=O)CC1C(F)(F)F 68002,C12(NC(c3cc(Br)co3)=O)CCCN(C(c3cc4cccnc4[nH]3)=O)CC1C2 68003,N1(C(CN(C)C)=O)CCC12CN(C(=O)CCc1ccc(Cl)cc1Cl)C2 68004,CC(C)CC(O)CC(=O)NC1CC(CCNC(C2CC2C(N)=O)=O)C1 68005,C1(C(=O)NC(CNC(COC(C)(C)C)=O)C2CCC2)CC2(C1)CC21CCC1 68006,N1(C(C(C(C)C)O)=O)CC2(C1)SCCC2NC(c1ccc(-n2cncn2)nc1)=O 68007,C1(C(=O)NCCN(C(=O)Cc2sccc2Cl)CCC)(N(C)C)CCCCC1C 68008,CCC(C(=O)N(C)CCOCCCN(C(=O)C(C1CCCCC1)OC)C)OC 68009,C1(CC=O)CC(O)CN1C(=O)CCc1cnn[nH]1.O=C(CCN1CCC1)N 68010,C1(C(=O)NCC2(F)CCC(NC(CCCC#CC)=O)C2)CCCCC12OCCO2 68011,CCC(O)C(=O)N(C1CCN(C(=O)CCN(CCCO)C(=O)OC(C)(C)C)C1)C 68012,C(=O)(C(C)C(O)CCCC)NC(C(=O)N1CCC(CC#C)C1)CCCC=C 68013,c1(CNC(c2c(CCC)n[nH]c2)=O)ccnc(C(=O)N(C(C)CSC)C)c1 68014,N1(C(CCc2cnn(C)n2)=O)CCC2CCCN(C(=O)C=Cc3ccsc3)C2C1 68015,N12CCC(C3(CC3)C(=O)N1)CC2.C12(c3nnc(N4CC(C=C)C4)o3)CCOC(C)(C1)C2 68016,C=C(C)C1OCCC1N=c1nc2c(ncn2C)c(NCC2CCCC2)[nH]1 68017,c1(CC(=O)NCC(c2ccccc2F)NC(CC=C=C)=O)cn(C)nc1C(F)F 68018,c1(OC)ccc(C(N2CC(NC(C3CC(O)(C(F)F)C3)=O)C2)=O)cc1 68019,C=C1CCN(C(c2cccs2)=O)C(C(=O)NCc2cc(C)ccc2O)C1 68020,C#CCC(C)C(=O)N(CC(C)(C)NC(c1cn(CC2(CC)COC2)nn1)=O)C 68021,c1(C(N2CC3C(C2)N3C(c2cnnc(Cl)c2)=O)=O)cc(Cl)c2cn[nH]c2c1 68022,c1(CCCC)cc([N+](=O)[O-])c(NC(=O)NCC(O)C2CC2)cc1OC(C)(C)C 68023,C#CCC(O)C(=O)N1CC(C(=O)NCc2nc(C)c(C)o2)C(CC)C1 68024,CCCCC(CC(=O)NCC(C)(O)C(C)CC)NC(c1ccccn1)=O 68025,C1(C(N2CCC(NC(c3cc(OC(F)F)cc(F)c3)=O)C2)=O)CCC2(CCC2)C1 68026,N1(C(c2cc(C)[nH]c2)=O)CCCC(O)(CNC(c2c[nH]cc(F)c2=O)=O)C1 68027,c1(C(N2CC(N(C(CC=C=C)=O)C)C(O)C2)=O)ccc(F)cc1CC 68028,c1(C(=O)NCCC(C)CCNC(=O)COCP(C)(C)=O)cc(Cl)c(F)cc1O 68029,c1(C(N2CCCC(NC(c3c(OC)oc(C)n3)=O)C2)=O)c(C)cc(C)cc1C 68030,CC1(CNC(c2cc(Br)c[nH]2)=O)COCCN(C(c2cc(C#N)c[nH]2)=O)C1 68031,c1(C(=O)NCCC(C)NC(C(CC)N(C)C)=O)cnc2ccnn2c1 68032,c1(CC)cccc(CC)c1C(N1CC(O)CC1C(=O)NC(C)C)=O 68033,CC1(C)CCCCC1=CC(N1CCOCC1CCNC(C1(C)CCNC1=O)=O)=O 68034,C1(C(N2CCCC(N(C(=O)Cn3cnnn3)C)CC2)=O)CCC(C2CCCO2)O1 68035,C1(C(C)NC(C2CC2c2ccco2)=O)CCN(C(=O)Cc2cc[nH]c2)CC1 68036,C1(c2ccccc2)(NC(c2n(CCC)nnn2)c2nccn2CC)COCCO1 68037,c1(C(N2C(C)(CNC(COCC)=O)CCC2)=O)ccc(=O)n(C)n1 68038,Cn1[nH]c(=NC(=O)C2CCCN(C(c3cc(CCO)on3)=O)C2C)cc1C(N)=O 68039,C1(NC(Cc2scc(C)n2)=O)CC(NC(=O)Cc2ccn(C)n2)C12CCOCC2 68040,c1(C(N2CC(C(C)NC(=O)CCc3ccccc3F)C2)=O)ccc([N+](=O)[O-])o1 68041,N1(C(CCC2(C)CC2(F)F)=O)CCC12CCNC2=O 68042,c1(C(C)NC(c2cccc(Cl)c2)C(=O)OCC)ccccc1I 68043,C1(C2CCN(C(=O)Cc3cccnc3N)C2)(NC(c2c(C)ncs2)=O)CC1 68044,C1(C)(CNC(C2CC(N(C)C)C2)=O)CCCN(C(=O)Cc2cc(C3CC3)on2)C1 68045,Cc1ccc(CC(=O)NC(C)(CNC(C2CCC(C)O2)=O)C2CC2)c(Br)c1 68046,C1(CC(=O)OC)CC2(CC2)CN1C(=O)OC.C1CC(C(C)C)Sc2cn1nn2 68047,C1(NC(Cn2c(C)nc(C)n2)=O)COC2(CCN(C(c3nnn(C)c3C)=O)C2)C1 68048,C(N=c1[nH]c(N2CCC3OC(=O)OC3C2)nc(=N)[nH]1)C1(SC)CC1 68049,C(=O)(C1=Cc2ccccc2C1)NC1C2(CCN(C(CCSCC)=O)C2)C1 68050,C(c1ccc(-c2ccccc2)cc1)=CC(=O)NC1CC(NC(C=CS(C)=O)=O)C1 68051,C(=O)(C1CCCc2ncccc21)N1CC=C(CNC(C2C(C)CCCC2)=O)CC1 68052,C1(NC(c2c(CC)ocn2)=O)CCN(C(=O)C(C)c2ccsc2)CCC1(F)F 68053,N1(C(C(CC)(C)O)=O)CC(N(C)C(c2cc(C)c(Cl)cn2)=O)C2(CC2)C1 68054,C=CCC(C)(C)CC(=O)N1CCN(C(c2cncc(N)n2)=O)CC1CC(=O)NC 68055,N1(C(c2c[nH]c(=NC)o2)=O)CCC2(CC2C(N2CCC(C)CC2)=O)C1 68056,CC1(CNC(=O)CC2CCOC2)CCN(NC(=O)CCCc2csc(C)n2)CC1 68057,c1(CCC)c(C(=O)NC2CCCC2NC(=O)CCN2C(=O)CNC2=O)cnn1C 68058,N12C3CCC(CC1CC3)COC2=O.CC(C)(C)NC(=O)NC(C)(C)C 68059,C1(c2nc(C)on2)CCCN(C(C2CCCCCC2)C(=O)NC2CCC2)C1 68060,C(=O)(NNC(=O)C(N)c1cccc(I)c1)c1ccc(OC)c(Cl)c1 68061,N1(C(CC(CC#C)NC(=O)C(CC=C)NC(C)=O)=O)CCn2nccc2C1 68062,N#Cc1cccc(OCC(N2CCCC2c2ccnn2C2CCOCC2)=O)c1 68063,Cn1nc2c(c1NC(C1CSCCN1Cc1cc(F)ccc1Br)=O)CCC2 68064,N1(C(C(C2CC2)OC)=O)CC(O)(C2(CNC(C3(Cl)CCC3)=O)CC2)C1 68065,C(=O)(C1=CC(C)(CC)C1)NCC(CN(C(=O)Cn1cc(C)cn1)CC)(C)C 68066,C(CCCCC(=O)N1CC(NC(=O)C=Cc2ccccn2)C(C)C1)=CC 68067,C1(O)(CN(C(C2(OC)CC2)=O)C)CCN(C(C2CCCOC2C)=O)CC1 68068,C1(C(=O)NCC(CNC(c2cccc(C3CC3)c2Cl)=O)CO)CC2CCC1CC2 68069,C(=O)(CCCC(F)F)N1C(C2(O)CN(C(C3N(CCC)C(=O)CC3)=O)C2)CCC1 68070,C1(NC(C2C(C)(C)N(C(c3cc(Cl)ns3)=O)CC2)=O)CCCOC12CCC2 68071,C(C)(c1cccnc1)=CC(=O)NCCN(C(=O)C(F)C(F)(F)F)CCC 68072,S(=O)(=O)(c1[nH]c(=NCc2c(C)cccc2Cl)ccc1Br)NCCS(CCOC)=O 68073,C(=O)(CC(=O)N1CCC(N(C(=O)C(C2CCCC2)OC)CC)C1)NCC#C 68074,C(=O)(CN=c1ccc(C#N)c[nH]1)N1CCCC(N(C(C(CCC)C)=O)C)C1 68075,C(=O)(CC(F)(F)C(F)(F)F)N1C(CNC(c2cncs2)=O)CCC1 68076,CCC(CC(=O)NC1CC(CNC(c2cnns2)=O)C12CCC2)CC(C)C 68077,CC(CCNC(c1cc(Br)n[nH]1)=O)CCNC(C1CCS(=O)CC1)=O 68078,CCCCC(C)CCC(=O)NCC1CCC(C(=O)NC(C2CCCC2)C)O1 68079,O=C1COC2CCN(C(c3cccc(C(F)(F)F)n3)C(=O)NC3COC3)CC2N1 68080,C1(F)(CNC(C2(C)C(C)C2)=O)CCC(NC(=O)CCc2ncc(F)cn2)C1 68081,N1(C(C(C)N(C(C)=O)C)=O)CC=CC(C(N2CCC2(C(=O)O)C(=O)O)=O)C1 68082,Cc1c(C(=O)NC(CNC(=O)C(CC(C)C)C(N)=O)C(C)C)sc2nnc(S)n12 68083,C(CC(C)C)(C(=O)NC1CCN(C(=O)CCc2c[nH]c(=N)[nH]2)C1(C)C)OC 68084,C1(CCC)(NC(c2ccc(CO)s2)=O)CCCN(C(c2cccc(C)n2)=O)C1 68085,C12CCN(C1CCOC)C(=O)c1ccoc1CC(=O)N2.N1(CC)CCC1C(N)=O 68086,c1(C(=O)OCc2c(F)cc(C)c(F)c2)ccc2nnc(C(F)F)n2c1 68087,C(C(CNC(C1(CC(C)C)CCC1)=O)OC)NC(C1C(CCC)C1)=O 68088,N1(C(C(CC2CCC2)NC(c2ccco2)=O)=O)CCC(C(F)F)CC1 68089,C1(C)(NC(C2C(C(=O)NCC#C)C2)=O)CCN(C(c2oc(C)nc2CC)=O)CC1 68090,CC(C)C(CCNC(=O)C(N)=O)NC(=O)C(C(C)O)c1ccccc1 68091,CC1CN(C(C2(F)CCOCC2)=O)CCC1N=c1[nH]c(Cl)ncc1Br 68092,c1(C(N(C2CC(NC(c3cnc(=N)[nH]c3)=O)C2)C)=O)cccc(F)c1C(F)F 68093,C1(NC(CCN(CC#C)C(C2CC(C)(F)C2)=O)=O)CC2(CC2)C1 68094,S(=O)(=O)(c1ccccc1F)NCCC(=O)N1CC(CNC(C2C(CC(C)C)C2)=O)C1 68095,c1(CC(=O)N(CC(C)O)CCNC(C2CCN(C(CC)=O)C2)=O)ccccc1F 68096,CC1=C(C(=O)N(CCNC(c2cc(F)ccc2Br)=O)C2CC2)SCCO1 68097,Cc1nc2c(N3CCN(C(c4c(F)cncc4F)=O)C4CC34)ncnc2[nH]1 68098,N(C1CCc2ccccc21)C(CCCCNC(CC=C)=O)=O 68099,c1(C(N2CCC(OCC(N3C(C)CC3CO)=O)C2)=O)cc(C#N)n(C)n1 68100,c1(C(N2C(CC)CCC2)=O)cccc(S(=O)(=O)NCc2cc(O)no2)c1 68101,c1(C(=O)OCC)nc(C(N2CCC(C(C)NC(=O)CC3CCC3)C2)=O)cs1 68102,c1(C(N(C2CCCN(C(C3(C(F)F)CCC3)=O)C2)C)=O)nn(C)nc1C(F)(F)F 68103,c1(N2C(C)CCC(NC(c3c(OCC)ccnc3)=O)C2)nc(OC)c(F)c(C)n1 68104,N1(CCCC)CCN(C(c2c(C)cnn2COC)C(=O)NC)CC1 68105,Cc1ccc(C#N)c(NC(C2CN(C(C3CCCCC3n3cccn3)=O)C2)=O)c1 68106,N1(C(C(=O)Nc2ccc(F)cc2)c2csnn2)CCc2ccc(Cl)nc2C1 68107,c1(OC)c(C)csc1C(N1CC(F)CC1CN(C)C(c1cnc(C)[nH]1)=O)=O 68108,c1(C(=O)NC(C2CN(c3snc(C(C)(C)OC)n3)C2)C)ncc(F)cc1F 68109,c1(SCC)ccc(C#N)c([N+](=O)[O-])c1.C(=O)(COCCOCCN)OC.C1CO1 68110,C1(NC(C(C=C)(C)O)=O)CCC2(CC1)CN(C(c1cccc(C(=O)OC)c1)=O)C2 68111,C1(CNC(CSCC(C)C)=O)CCC(C)N(C(c2ccc(CC3CC3)nc2)=O)C1 68112,CCC(C(=O)OC)C(=O)NC(C)(C)CN(C(=O)C(COC)OC)C 68113,c1(OC)ccc(C(=O)NC2CCC23CN(C(=O)CC2(OC)CC2)C3)c(F)c1Cl 68114,C(=O)(CC(CNC(C1CSCC(=O)N1)=O)C1CCC1)NCc1c(C)nsc1 68115,C12(C(=O)NC3CCC(NC(CCCC#N)=O)C3)CC3CC1(CO)CC3C2 68116,c1(C(=O)NCC(C)(C2CC2)NC(c2cc(SC(F)(F)F)c[nH]2)=O)ncc(F)cn1 68117,N1(C(CCN(C)CCO)=O)CCC2CCN(C(=O)COCC3CCC3)CC12 68118,C12(C(N(CCNC(=O)CCSCC(C)C)CC)=O)CC(C)C1C2 68119,c12cnc(F)cc1C(=O)NC1CCN(CC1O)C(=O)N2.c1(OC)ccccn1 68120,C12CN(CC1F)C2=O.C1(CC)CCC(NC(=O)CCCC2CC2C)C1 68121,C1(O)(C(C(=O)NC2C(O)CC2O)NC(N)=O)CCCCC1 68122,C(=O)(CCCCCC(C)(C)C)NC12C(CN(C(CS(CCC)(=O)=O)=O)C1)CCC2 68123,CC(CCCNC(c1csc(O)n1)=O)NC(c1csc(O)n1)=O 68124,c1(C(=O)NCCC(=C)CNC(=O)CC2CCCOC2)ccccc1SC 68125,C1(C(N(C2CC(OC)C(N)C2)C)=O)(N(C)C)CCC(F)(F)CC1 68126,C(CCC(C)CC(=O)N1CC(NC(=O)CCc2cnn(C)c2C)C1)=C(C)C 68127,N1(C(C=CCCC)=O)CCC2(CCCC2NC(c2cnc(N(C)C)o2)=O)C1 68128,c1(CC(N2CC(C)C(CNC(c3cc(Br)c[nH]3)=O)C2)=O)nn(C)c2ccccc12 68129,C1(C(=O)NC2C(CNC(=O)CC3(O)CCC3)CC2)(NC(N)=O)CCCCC1 68130,C(=O)(C1c2c[nH]nc2CCC1C)NC1C(S(CC)=O)CCC1 68131,CN1CC(NC(c2cccc([Si](C)(C)C)c2)=O)Cc2ccccc21 68132,C(=O)(C(O)CNC(C1CC1(C)C(F)F)=O)N(C(C)CO)C1CC1 68133,n1(C(CC)C)nc(C(=O)NC(C)CNC(=O)C=Cc2csc(C)n2)cc1C 68134,C(=O)(C(F)C(C)CNC(=O)C(C)(C)C(F)F)NC(c1c(C)ncs1)C 68135,c1(C(=O)NC2CN(C(C3CCC(OC)CC3)=O)C(C)CC2)csc2cccnc12 68136,c1(NC(C2CCN(c3ccccc3Cc3nn[nH]n3)C2)=O)nc(Cl)c(Br)cc1O 68137,c1(N(C2CCCN(C(CCC(C)SC)=O)C2)C)snc(C)c1C#N 68138,C1(N(C)C)CN(C(c2cocc2Br)C(=O)NC2CCOCC2)CC12CC2 68139,c1(C(N2CC(C(N3CCC(F)C(F)(F)C3)=O)NCC2)=O)ccc2c(c1)CCC2 68140,c1(NC(C2(O)CCN(C(=O)CCc3cc(F)ccn3)C2)=O)cccc2[nH]ccc12 68141,Cc1c(CN(CC(C)NC(c2ccccc2C(F)(F)F)=O)C)cccc1O 68142,C(N=c1[nH]c(=NCCC(C)C(F)F)[nH]c2c1SCC2)C1N(C(C)=O)CCC1 68143,c1(C(N2CCC(NC(CCCCSC)=O)CC2)=O)ncc2ccccn12 68144,C1(NC(c2c(C)onc2)=O)(CNC(C2(C)CCCO2)=O)CC2CCC1CC2 68145,C1(COC)CN(CC2CC2n2cnc(=N)[nH]2)CCN1CC(F)F 68146,C1(C(=O)NCC(n2cccn2)C)CCOCCN1C(c1ccc(C#N)o1)=O 68147,c1(C(=O)NCC2C(NC(C3(C)C=CCCC3)=O)CCC2)cc(F)c(F)c(O)c1F 68148,c1(C(=O)NCCN(C(C2CCC(=O)NC2)=O)CC)coc2ccccc12 68149,C=Cc1cc(C(=O)NCC2(C)CCN(C(c3ccnc(OC)c3)=O)C2)cc(F)c1 68150,c1(COC)nn(C)c(Cl)c1C(N1CCCC1CNC(C1CC(C)(C)C1)=O)=O 68151,Cc1ccc(C=CC(=O)NCC(C2CC2)NC(=O)C(n2nccc2C)C)cc1Cl 68152,C1(CC(=O)NCC(CC)C(C)C)CCN(C(=O)CCC2CCC(=O)C2)C1(C)C 68153,c1(Sc2nc(CCC(CCC)O)on2)cc(C(N)=O)cc2cccnc12 68154,N1(C(CSC)=O)Cc2ccccc2C(CNC(c2cnc(NC(C)=O)o2)=O)C1 68155,C1(CNC(C=C(C)C(C)(C)C)=O)CC2CN(C(C3(C#N)CC4CC4C3)=O)CC12 68156,CCC(CC(=O)NCCC(=O)NC(C)(C)CC(C)C)CC(C)C 68157,N1(C(=O)Cn2cnc(Br)c2)CCC2CCCC(C1)N2C(C1C2COCC12)=O 68158,C1(C(=O)NC(C)C(C)(C)NC(=O)CCN2CCOCC2)CS(=O)(=O)CCO1 68159,C1(C(N2CC(C(C)NC(C=CCC)=O)C2)=O)CC(C2CCOCC2)=NO1 68160,CC(C)(O)C(F)C(=O)N1CCOC(c2ccccc2)C1.c12cn(nn1)CC2 68161,N1(C(c2ncn(CC)c2)=O)CCC(C2CCN(C(c3cc(C)ccc3C)=O)C2)C1 68162,CC1(C)CN(C(c2ccon2)=O)CC1NC(c1cc(-n2ccnc2)cs1)=O 68163,CCCCS(=O)(=O)NC(N(C)CCCc1cn(-c2ccccc2Cl)nn1)=O 68164,N1(C(C(C)C2CC2)=O)CC2(CCC2NC(=O)Cc2nn(C)cc2Br)C1 68165,C1(NC(C(CSC)(C)C)=O)CCCN(C(c2cc3sccc3s2)=O)CC1 68166,CN1CCC(N(C(=O)C(c2cccn2C)=O)C)C1 68167,C1(C2CCN(C(C3(C)CC(C)=NO3)=O)C2)(NC(c2cc(OC)n(C)n2)=O)CC1 68168,CC1CCCC(C(N2CCC(CC(F)(F)F)CC2)C(=O)NCC2CCOCC2)C1 68169,CC1(C(=O)NCc2cccc(Cl)c2F)CCCN(Cc2nccs2)C1 68170,c1(CC(=O)NCCNC(CCCN(CCOC)C)=O)ccc(OC(F)F)c(F)c1 68171,c1(C(=O)NCCn2cc(C(C3CCN(CC(F)(F)F)C3)=O)nn2)nc(Cl)sc1Cl 68172,c1(NC(C2N(Cc3ccc(OCC#C)cc3)CC(F)C2)=O)nc(Cl)cnc1Cl 68173,N1(C(c2cc(C)n(C)c2)=O)CC(N=[N+]=[N-])CC1C(=O)N(CC(O)CN(C)C)C 68174,N1(C(C)=O)CCCC(O)(CC(N2CC(O)(CNC(c3cc(OC)ns3)=O)C2)=O)C1 68175,CCC(CC)CC(=O)NCC1CN(C)CCN1C(c1cc(C)nn1C(F)F)=O 68176,n1(CC)nccc1C(N1CCC(N(C(=O)COCc2ccnn2C)C)C1)=O 68177,N1(C(CC(C)(C)C)=O)CC2(CCC2)CC1CNC(c1ccnc2c1CCC2)=O 68178,C(=O)(CC(=O)NCC1CC(NC(c2c[nH]nc2C(C)(F)F)=O)C1)N(C)C 68179,N1(C(C)=O)CCN(C(=O)CCCn2cc(CCOC(N)=O)nn2)CC1 68180,Cc1nn(C)c(C)c1C(N1CC(NC(=O)CCN2CCCS2(=O)=O)CC(O)C1)=O 68181,N=c1[nH]cc(C(=O)NCC(O)CNC(c2cscc2F)=O)c2cc[nH]c12 68182,C1(C(NOCC(COC)O)=O)CCC(O)CN1C(c1cnncc1OC)=O 68183,N1(CC(N2CCN(C)CC2)C)CC2(CCC1CO)CC2 68184,c1(C(N2CC(NC(CCOCC#C)=O)C(O)C2)=O)cc(=O)c(OC)cn1C 68185,c1(NC)snc(C)c1C(=O)NCCOCCNC(=O)C(C)CCc1cccc(F)c1 68186,c1(C(N(CCN(C(CCC2CC(OC)C2)=O)C)C)=O)ccc(N)c2ccncc12 68187,C1(C2(O)CCOCC2)(C(N2C(C(=O)OCc3ccccc3)C(O)CC2)=O)CC1 68188,c12cccc(c1)C=CC2.c1(OC)ccccc1SC1COC1 68189,c1(C(=O)NC)cccc(CCNC(=O)NC2CCC2C(C)(C)C)c1 68190,Cc1cnc(C(C)NC(=O)C(C2CCCCC2)C)s1 68191,C1(CCC)CN(C(=O)CCc2ncccn2)CCN1C(=O)CCCCNC(N)=O 68192,C(=O)(C(C)(CC)CO)N(CCC)CCc1nc(C(=O)OC)nc(O)c1 68193,CC1CCCN(C(C)CN(c2ccccc2)C(=O)Nc2conc2C2CCCO2)C1 68194,C(=O)(C(O)C(C)(C)C)N1CC(C)C(NC(=O)Cc2ccncc2Cl)C1 68195,C#CC1(C(=O)OC)CCN(C(=O)C(N)Cc2nonc2C)C1 68196,C(c1ccc2occc2c1)=CC(=O)NC1C(NC(C(C(C)O)(C)C)=O)CCC1 68197,C(=O)(CC(C)CC(F)(F)F)N1C(CCNC(C(=C(C)C2CC2)F)=O)CCC1 68198,CCC(CC)(CCO)NC(c1cncn1C(C)C)c1nnnn1C 68199,C1(C(=O)OC)COCC1C(=O)N(CCCCN(C(=O)C(C1CC1)NC(C)=O)C)C 68200,c1(NC(C(=O)NCCN(C(CC)C)C)=O)ccc2c(c1)C(=O)OC2(C)C 68201,C(CNC(=O)CCc1ccccc1)(CC(F)(F)F)NC(C(C)OCCOC)=O 68202,c1(C(N2CCC(C(=O)OCC)CC2)=O)ccc(F)c(-c2c(C)cccc2F)n1 68203,c1(C(C(=O)NCC=C)N(C2CCC2(C)C)C)nnc(-c2ccccc2)s1 68204,C1(NC(c2nnc(C)s2)=O)CN(C(=O)C2=CCC(C)(C)CC2)C2(CCCCC2)C1 68205,c1(C(=O)NC(CCCNC(C2C(=C)C2)=O)C)cc(CC)nn1C 68206,N(C(=NCc1ccc(O)cc1)N1CCc2nn(C)c(=O)cc2C1)C(COC)C 68207,Cc1cc(C)n2nc(CNC(C)(C)COc3cccc(Br)c3)nc2n1 68208,c1(SCC)ccc(Cl)cc1C(=O)N(CC(CC)NC(=O)C(F)CC1CCC1)C 68209,C12(NC(C(COC)COC)=O)CCC(F)(F)CC1CN(C(=O)C(F)C(C)(C)O)C2 68210,c1(C(=O)NC2CC(NC(c3nc(C)sc3C)=O)C2)ccc2nn[nH]c2c1O 68211,c1(C(=O)Nc2ccc(-c3cc(OC(C)C)ncc3)s2)cc(Br)cn2ccnc12 68212,C1(NC(C(C)C)=O)CCN(C(c2csc(C(F)F)c2)=O)CC1C(C)C 68213,C#CCCCCCC(=O)NCC1(F)CN(C(c2c(C)csc2C)=O)C1 68214,C12(CNC(C3N(C)CCC3)=O)CCCC(CN(C(=O)C(F)C3CCC3)C1)C2 68215,O=[N+]([O-])c1ccc(C(F)F)cc1OC(c1cc(Cl)ccc1F)=O 68216,c1(C(=O)NCC2N(C(Cn3c(=O)sc(C)c3C)=O)CC2)c(F)ccc2c1OCO2 68217,C12(CNC(C=CCOC)=O)CC1CN(C(C1CC(C)CCO1)=O)C2 68218,C(=O)(CCCCCOCC)N1CCC(C(C(N2CCC(=C)C2)=O)C)C1 68219,c1(C(=O)NCCC(C(C)C)NC(=O)Cc2cn[nH]c2)cc(=O)c2ccccc2[nH]1 68220,C1(NC(C(C2CC2)OC)=O)COCC1NC(c1ccoc1I)=O 68221,CC(Cc1ccccc1)(C(F)F)NC(=O)OCC(F)(F)F 68222,c1(C(=O)NC2CN(C(CC(C=C)C)=O)CC2O)n[nH]c2c1CS(=O)(=O)CC2 68223,c1(C(N2CCCC(CNC(CCC3CC(C)C3)=O)C2)=O)cn(C)c(=O)n(C)c1=O 68224,N1(C(C=C2CCC(C)CC2)=O)CCC(O)(CNC(=O)CC(C)(F)F)CC1 68225,c1(Cc2nnnn2C2COC2)cc(CNC(C)CCC(C)C)ccc1C#N.CC 68226,C#CC1CCC(NC(=O)COc2ccccc2F)CC1 68227,CC(C)(C)C(CNC(c1ccn(C(F)F)n1)=O)C(=O)NCCC1(C)CC1(F)F 68228,C1(C(N(C)CC2CC2)=O)CN(Cc2cncn2C2CCCC2)CCC1O 68229,c1(C(=O)NCC=CCNC(=O)CC2(O)CCOCC2)cnn2c(=O)cc[nH]c12 68230,C1(CNC(C2(C)CC(C)C2)=O)CC2(CCN(C(=O)CNc3ccccn3)C2)CO1 68231,Cc1[nH]c(C)c(C(=O)NCC2=CCN(C(=O)C(C)Cc3cnc[nH]3)CC2)c1C 68232,C1(CNC(C(CC)COC)=O)CCC2(CCC2)CN1C(c1cncn(C)c1=O)=O 68233,C1(CCNC(CCOCCCOC)=O)CN(C(=O)CC2CS(=O)(=O)C2)CCO1 68234,c1(OC)cc(C(=O)NC2CC(C)CN(C(=O)OC(C)(C)C)C2)ccc1C 68235,N1(C(C(CCOC)OC)=O)Cc2ccccc2CC1CNC(=O)CC1CCCC1 68236,c1(C(C(=O)NCC(Cn2cc(C=CC)nn2)(C)C)(C)C)ccc(C#N)cc1F 68237,Cc1nocc1CCC(=O)NC1CC(CNC(c2csnc2Br)=O)C1 68238,C1(C(=O)NCCc2ccc(O)cn2)CCc2nnc(-c3ccccc3)n2C1 68239,c1(CC)oc(C(=O)NCC2CN(C(=O)C(CC3CC3)CC3CC3)CC2C)cc1C 68240,C1(COC)(CNC(=O)CCc2cc(C)no2)CCCN1C(C1CCCC1)=O 68241,c1(CCC(=O)NCC(CNC(c2cc(CC)on2)=O)(C)O)c(C)n[nH]c1C 68242,C1(CC(=O)NC(CC2CCCO2)CO)CC2(C1)CN(C(=O)CCc1cccs1)C2 68243,N1(C(c2c(C)nncc2)=O)CCN(C(c2ocnc2C)=O)CC(O)C1 68244,c1(N(C)C)nccc2c1CCN(Cc1ncsc1Br)C2 68245,C(C)(C)(CCCNC(C1CCC(C)O1)=O)NC(c1c(C(C)C)ncs1)=O 68246,C1(CCNC(C(C=CCCC)O)=O)CCCN(C(=O)CNC(=O)CCC(C)C)C1 68247,N1(C(C(C=C)(C)O)=O)CC(NC(C2CC3(CCOCC3)C2)=O)CC2(CCC2)C1 68248,C1(NC(C=C(C)C(C)C)=O)CCN(C(C23CCCC2C3(F)F)=O)CC1CO 68249,Cc1cc(C(c2ccco2)NCc2cn(C3CCOC3)nn2)on1 68250,c1(N2C(CC(=O)Nc3cc(CCC)no3)COCC2)ncc2cccc(Br)c2n1 68251,C1(C)(C(=O)OC)CC12CCN(C(c1ccc(Nc3cn[nH]c3)cc1Cl)=O)CC2 68252,c1(C(N(C(CNC(C(C)CC2CCC2)=O)C)C)=O)c[nH]c2nccc-2c1 68253,C1(CNC(c2ccn(CC)n2)=O)CC(NC(=O)C(O)CC2CC2)C(O)C1 68254,N1(C(CCN(C)CC)=O)CCN(C(C23CC(C2)S(=O)(=O)C3)=O)CC1C 68255,c1(C(N(C2CCN(C(=O)C3=NNC(=O)CC3)C2)C)=O)cc(F)c2cn[nH]c2c1 68256,Cc1nc(CC(=O)NC2(C(=O)N(C)C(C)C3CC3)CSC2)cs1 68257,N1(C(C2(CC(C)C)CCNC2)=O)CCC(C#N)(NC(N)=O)C1 68258,c1(C(N2C(CN(C(CC3N(CC)CCC3)=O)C)CCCC2)=O)cc(N)nc(Cl)c1 68259,N1(C(CNC(CCC(C)C)=O)=O)CCC(C(=O)N(C)Cc2ccsc2)C(C)(C)C1 68260,CC1(CO)CCCN(C(C2CCCN2C(c2scnc2Cl)=O)=O)C1 68261,c1(COC)cnc(OC)c(C(=O)NCC(C)CNC(=O)COC2CCCOC2)c1 68262,C(=O)(C1=C(Cl)CCCC1)NC1(O)CCN(C(CCOC(CC(C)C)C)=O)CC1 68263,CCC(CC)C(C)C(=O)NCC(C)(CC)NC(=O)CSc1nncn1C(C)(C)C 68264,c1(-c2cn(C(COCC)C(=O)NC3(SC)CC3)nn2)ccc(-c2cncnc2)cc1 68265,N1(C(c2scc(C)c2Cl)=O)CCC(CCNC(C2C(C)C2C)=O)C(F)(F)C1 68266,c1(C(N(C(CNC(C2C(c3cn(CC)nc3)OCC2)=O)C)C)=O)ccnnc1C 68267,C(=O)(C1CCc2ccccc21)NCc1c(C(=O)NC2(C(C)(F)F)CCC2)con1 68268,N1(C(c2cnc(CC(C)C)s2)=O)CC2CC(NC(=O)CC3=NNC(=O)C3)CC1C2 68269,CCCC(C)(CC)C(=O)N1CCCCCC(NC(C2(O)CCC2)=O)C1 68270,O=C(C1=COCC1)NCC1CN(C(=O)Cc2cccc(OC3CC3)c2)CCO1 68271,C1(C(=O)NCC(C)CN(C(=O)C(C)(C)F)C)(Cc2ccccc2)CCOCC1 68272,C1(OC)CCC(C(=O)NC2(CNC(=O)CCc3ccc(C)cc3)CCOC2)CC1 68273,C12(C(=O)NCC3C4CN(C(C(C)(C)N(C)C)=O)CC43)CCC(C)(C(=O)O1)C2(C)C 68274,Cc1nc(N2CCC3(CC3C(=O)NC(C)CCO)C2)c2sccc2n1 68275,c1(CNC(C)C)cccnc1C(=O)N(C)CCN(C(=O)C(CO)N(C)C)C 68276,CC1CC(NC(=O)CC2CCC(=O)N2C)CCN1Cc1cncs1 68277,C1(C(N2CCC(C)(NC(c3nc(C(C)C)oc3)=O)C2)=O)CC12CC(F)(F)C2 68278,N1(C(=O)NC2CC2)C(C(c2cc(C)n(-c3nccs3)c2C)=O)CC2OCCC12 68279,C1(NC(c2ccc(N(C)C)nc2)=O)CN(C(C2CC2C(F)(F)F)=O)CC1C1CC1 68280,C(=O)(C(O)CCC(F)(F)F)NC(C1CCCC1)CNC(CC(COC)(C)C)=O 68281,c1(C(N2CC(NC(Cc3c(C)cccn3)=O)C(C)C2)=O)c(C)nc2cccnn12 68282,C1(CNC(c2ccc(Cl)cn2)=O)C2CN(C(=O)CCc3cncc(F)c3)CC12 68283,N1(C(c2cncc(C3CC3)c2)=O)CCC(O)C(O)c2ccccc21 68284,c1(C(N2CC(CNC(c3ccc(OC(C)=O)s3)=O)C2)=O)c(F)cccc1Br 68285,Cc1ccc(C=CC(N2CCCN(C(=O)CCCC3CC3)CC2CO)=O)cc1Cl 68286,C1(N(C(Cn2ncc(CC)c2)=O)CCO)CCCN(C(=O)CCC2CCCC2)C1 68287,CCCCC(CC)CC(=O)N1CC(F)CC1CN(C(=O)CC(C)(C)C(F)F)C 68288,C1(NC(C2C(C)CN(C(c3cnc(O)n3C)=O)C2)=O)CCN(C)CC1C#N 68289,C(CC(C(=O)NCCSCCNC(=O)C=Cc1ccco1)N(C)C)SC 68290,C(=O)(CC1=NNC(=O)C1)N1C2C(NC(CN(C)C(N)=O)=O)C(C2)C1 68291,O=C(C#CC1CCOC1)NCC1CCN(C(=O)CCOC2CCCC2)CC1O 68292,C=CC1(CC(=O)N(CC(=O)NC)C(C)C)CN(C(=O)CC(CC)SC)C1 68293,C(CC(=O)NC1CN(C)CC1O)(C(C)OC)NC(CCOC)=O 68294,C1(c2n(CC(=C)C)nnn2)(NCc2ccccc2-n2cncn2)CC(C)N(C)C1 68295,c1(C(=O)NCC(C(=O)NCC(COCC)C)O)ccc2[nH]ccc2c1 68296,Cc1cscc1C(=O)NC(C(=O)NCCc1cn(C)nn1)C1CCCO1 68297,c1(NC(CN(C2CCC2)C(c2c(CC)cco2)=O)=O)ccc(O)c(OC)c1 68298,N1(C(Cc2cc(C)no2)=O)CCCC(CC(N2CC3CC3(CO)C2)=O)C1 68299,c1(C(=O)N(C2(CNC(C3CN(S(C)(=O)=O)C3)=O)CCOC2)CCO)c(C)ncn1C 68300,C(=O)(C(C(=O)NCC12CC1CN(C(C1CCC1COC)=O)C2)C(C)C)OCC 68301,c1(C(=O)NC2CN(Cc3cn(C(C)C)nc3)C2)cccc(=O)n1O 68302,C1(CC)COCCN(C(C2CCCN(C(c3cnn(CC)c3C)=O)C2)=O)C1 68303,c1(C(=O)NC2CCCCN(C(C(C(C)C)(C)C)=O)C2)cc2c(nc1N)CCC2 68304,c1(C(N2CCC(NC(C=C(CC)C)=O)C(F)C2)=O)cnc2c(N)cccc2c1 68305,N1(CCC)CC(C(N2CC=CC(NC(=O)CSC(C)C)C2)=O)CC1=O 68306,C1(C(=O)NCc2c(C(=O)NCC(C3CC3)SC)con2)CCC(C)=C(C)C1 68307,C1(C(COC(n2cccc2N(C)C)=O)=O)CCCN(C(=O)C(C)(C)C)C1 68308,C(C(O)C(=O)NC1CC(F)(CNC(c2csnn2)=O)C1)SC 68309,C1(C(=O)NCC2(C(C)(C)O)CN(C(=O)CC(O)C3CCCC3)C2)CC12CCCCC2 68310,C(=O)(C(C)(C)CS(N)(=O)=O)NCC1(F)CC(NC(CC(=O)NCC#C)=O)C1 68311,C(=O)(CC1=CCN(C(C2OCCC2(C)C)=O)CC1)N(C(CSC)C)C 68312,Cc1cccc2nc(C(=O)NCC(O)CNC(C34CCCCC3C4)=O)cn12 68313,C1(F)(CNC(C2C(OCC)C2)=O)CC(CNC(C2(O)CC2)=O)C1 68314,c1(OCC(=O)N(C2CCN(C(CC(=C=C)C)=O)CC2)CCO)cc(F)cc(F)c1 68315,c1(CC)ncc(C(N2CCC(CC(N3CCNC(=O)C3CC)=O)C2)=O)c(C)n1 68316,CC1CCN(C(c2cc3n(n2)CCC3)C(=O)NCCCOC(F)F)CC1C 68317,c1(CC)nn(C)c(C(=O)NC2CCN(C(=O)C(C)(C)C)C2)c1Cl 68318,N1(C(CC2CC(=C)C2)=O)CCN(C(=O)CCC2CCCN2CC)CC1 68319,CCC(C)C(CC(=O)N1CCn2nncc2C1)NC(=O)CSCC(F)F 68320,c1(NC(=O)NC2C(CC(=O)OC)COCC2)ccc(F)c(F)c1 68321,C(=O)(CCCCNC(N)=O)NCC(C)(C)CNC(C1(C)CCNC1=O)=O 68322,C1(NC(C2N(C)CCC2)=O)CCN(C(=O)CC2CCC(O)C2)C12CC2 68323,C=CC(C)CC(=O)NC(CNC(=O)CC1CNC(=O)O1)C(C)C 68324,C1(CC(=O)NC2CCC(CCNC(CCC)=O)C2)CC(=O)NC(=O)C1 68325,N1(C(C2CCC(NC(C3CC(F)C(=O)N3)=O)CC2)=O)CCCC(OC(F)F)C1 68326,Cc1ccc(-n2nnnc2N2CC(NC(C3(C)CCC(C)C3)=O)CC2C)cc1 68327,c1(N2CCC(C)C(NC(=O)CN3CCCS3(=O)=O)C2)ncnc2cnccc12 68328,c1(C(=O)NCC2CC(C)N(C(=O)CCC3CCCCO3)C2)ccc(Cl)nc1O 68329,c1(OCC)ccc(CN2CC3C(C2)N3C(=O)C(C(C)C)OCC)c(O)c1 68330,C1(C(=O)NC2(CO)CN(C(C(=Cc3cnc[nH]3)C)=O)C2)CCS(=O)(=O)N1 68331,C1(C(N2CCCCC(CNC(=O)C=C3CCSCC3)C2)=O)COCC2(CCC2)O1 68332,CCC(F)(C(=O)OC)C(=O)NCCNC(c1ccc(CCF)cc1)=O 68333,N1(C(C(C)CCN(C)C)=O)CCC(C2CC2)C1CNC(=O)C=CC1CC1 68334,Cc1noc(C)c1C(C)C(=O)N(CCNC(=O)Cc1ccc(C(N)=O)nc1)C(C)C 68335,C12(COC)CCC(C(=O)NC3CCC3NC(C3CCCC(=O)O3)=O)(CC1)CO2 68336,CN1CC(C)(C(N2CC=CC(C(=O)NCC(N3CC=CC3)=O)C2)=O)CC1=O 68337,C1(CN2CC(c3nc(C(C)C)[nH]n3)OCC2)CCCCCCC1O 68338,c1(CNC(CC(C)CC2CCC2)=O)ccccc1[N+](=O)[O-] 68339,C1(C(N2CCC(CC(F)(F)F)CC2)=O)COC2(CNC2)C1 68340,C12(NC(C3CCCOC3)=O)CC3CCC(C1C2)N3C(c1c[nH]c2nccc-2c1)=O 68341,N1(C(C2CC=C(C)CC2)=O)CCC(C)(C(=O)Nc2ncc(C)c(Cl)n2)CC1 68342,CN1CCCC1(C)C(=O)NCC1CC1C(N1CCC12CCC2)=O 68343,C(N=c1[nH]cnc(Cl)c1C(C)=O)C1(NC(c2ccc(C(=O)NC)nc2)=O)CCCC1 68344,n1(C(C(=O)N(CC(CC)NC(=O)C(O)C2CCCC2)C)C)nc(C)cc1C 68345,N1(C(CCCC#C)=O)CCCC2C(NC(c3cc(O)cc(C#N)c3)=O)C(C)(C)C12 68346,C=CCCC(=O)N(CCCCCNC(=O)C=CC(=O)NC1CC1)C 68347,c1(COC)ncc(C(N2CCN(C(=O)COc3cnc(N)cn3)CC2)=O)c(O)n1 68348,c1(C(N(CCC)CCNC(C2(CCC)CCC2)=O)=O)cc(Cl)cc(Cl)n1 68349,c1(CC(=O)NC2CN(C(c3c(OC)nsc3)=O)C3C2C3)cc2ccccc2o1 68350,c1(C(=O)NC2COCCN(C(C3CC(C(C)C)C3)=O)C2)cn2ccccc2n1 68351,N1(C(C=CC(=O)NCC2(c3cccs3)C(C)(C)C2)=O)CC2C(NC(=O)C(N)=O)C2C1 68352,C(=O)(C(C(C)(C)C)NC(N)=O)N(CC(C)NC(=O)C(=O)Cc1cccs1)C 68353,c1(C(N2CC(O)CC(NC(C3SC4C=CC3CC4)=O)C2)=O)cnn2c(Cl)cccc12 68354,C(=O)(C#CC1CCCC1)NCCC1(OC)CN(C(c2cnn(CC)c2Br)=O)C1 68355,CCC(C)C(C(=O)NCC1CCC2(CC1)CC2)N(C(=O)CN1CCOCC1)C 68356,c1(C(=O)NCCC2CN(C(C3C(C(=O)OC)CCC3)=O)C2)c(C)cccc1O 68357,C1(C(NC=O)=O)CCCN1NCC1(F)CC1.C1C(=O)N1 68358,C(C(=O)NC)(C1=Cc2cc(Br)ccc2OC1)N(CC(CC)C)C1CC1 68359,Cc1c(C)n(C)c2ccc(C(=O)NCC3CN(C(=O)CO)CCC3C)cc12 68360,C1(N(c2c(F)cccc2Cl)C(=O)CCc2cnccn2)CC2(CCNCC2)C1 68361,N1(C(C(c2ccccc2)SC)=O)C2CCCC1CN(C(=O)C(C)NC=O)C2 68362,Cc1cncc(C(=O)NC2CC(C)N(C(=O)COCCC(C)C)C2)c1 68363,C(=O)(CCC(CC)NC(c1cc(OC)ccn1)=O)N1C(C=C)CCC1 68364,C1(N(C)C(=O)NC2C(C)(C)C2(F)F)CC(=O)N(Cc2ccccc2)CC1 68365,C1(NC(Cn2nc(C)c(Br)c2)=O)CN(C(c2cnc(N)cn2)=O)CC1(C)C 68366,CCC(C(=O)NCC(C)(C)NC(C1CC1c1cncn1C)=O)SC 68367,C1(NC(C2CC3(CCC3O)C2)=O)CCC(O)CN(C(c2cc(CO)on2)=O)C1 68368,Cc1ccc(F)cc1C(=O)C(=O)NCC1(F)CC(NC(c2cnc(C)n2C)=O)C1 68369,c1(C(N2C(CN(C(COC(CC)C)=O)C)CCCC2)=O)ccnc2ncsc12 68370,C(=O)(CN=c1[nH]cnc2c1CCCC2)NC(C(C)C)C(F)(F)F 68371,C1(NC(CCCC)=O)CCC2(CC1)CC2NC(C1CCC(=O)N1C)=O 68372,C(=O)(CC(C)(C)NC(=O)Cc1ccccn1)NC(C(=O)OCC)C 68373,C#CC1CN(C(=O)CC2CC(F)CN2C(=O)CC2CNC(=O)O2)CCN1C 68374,C1(NC(c2c(C(C)C)noc2)=O)CN(C(C2COC(=O)N2C)=O)CC1O 68375,CC(C)(C)CCCCCC(=O)N1CCn2ncc(C(=O)NC34CC(F)(C3)C4)c2C1 68376,N1(C(c2ccc(F)cc2)CC)CCC2(CCCN(C(c3cncc(F)c3)=O)C2)C1 68377,C(=O)(CS(=O)(=O)CCC(F)(F)F)N1CCN(C(c2n(C)nnc2)=O)C2C1C2 68378,C1(O)(CCNC(Cc2ccc(C)nc2)=O)CCN(C(=O)C(C)(C)CC#N)CC1 68379,N1(C(c2cc(Cl)c(Br)c(Cl)c2)=O)CCC2C(CCN2Cc2cc(I)ccc2F)C1 68380,C1(C(=O)NC2C3CN(C(CC(CC)CC)=O)C2C3)CCc2nnnn2CC1 68381,Cc1nn(CC(=O)NC(C)(CO)C(=O)NCCC(O)C(C)C)c(=O)o1 68382,n1(CCOC)nnc(-c2nc(COC)nn2CC(C)(C)C)c1C 68383,C=CCC(C)C(=O)NCc1ccc(CC(C)NC(c2cnn(C)c2SC)=O)cc1 68384,c1(C(N(C)CC2(NC(C(F)=CCC)=O)CC2)=O)cn2c(n1)CCC2 68385,C1(C(N(CCNC(C=COCC)=O)C(C)C)=O)C2CC1(c1ccccc1C)CO2 68386,C1(C(N(CCC(C)NC(c2cc(C3CC3)ccc2F)=O)C)=O)CCC(C)(C)CO1 68387,C1(C(N2CCN(C(Cn3c(C)nnn3)=O)CC2CCO)=O)CC2CC(O)C(C1)C2 68388,Cc1cnc(C(=O)NCc2ccc(C(=O)NC3CC(CC#N)C4CC34)nc2)cn1 68389,Cc1cncc(C(N2CCCC2CCCNC(=O)C(C)OCC2CC2)=O)c1C 68390,Cc1ccc(Cl)cc1NC(=O)C(C)(C)C1CCCN1C(=O)CSC(F)F 68391,c1(CCCC(=O)N(CCNC(C=CC=CC)=O)C(C)C)cccc(Cl)n1 68392,c1(CC(=O)NCC=CCNC(C2C(COC)C2)=O)ccc(F)c(Cl)c1 68393,N1(C(C(CCC)NC(c2nn(C)cc2C)=O)=O)CCC2(CCCOC2)C1 68394,Cc1nc(NCCS(C)=O)cc(N2CCCC(C(F)(F)F)C2)n1 68395,C1(C(=O)NCC(C)CN(C)C(c2cnccc2Cl)=O)CCN(C)S1(=O)=O 68396,c1(C(N2CCC(NC(COCC#C)=O)CC2C)=O)cc2nc[nH]c2cc1F 68397,C(=O)(C(C)(F)C(=O)N1CC=CC(C(=O)N(C)CCc2ccccn2)C1)OC 68398,C1(CC)CC(C)(C)CN1N1CCCC1(C)Cc1c(F)cccc1F 68399,N1(C(CCC2CC(OC)C2)=O)CCCC2CN(C(C3CCCCC34CC4)=O)CC12 68400,C1(NC(C2(Cl)CC2(F)F)=O)COC2(C1)CN(C(=O)CCOC1CCCC1)C2 68401,c1(C(=O)NC2(COC)CC(OC)C2)csc(N=S(C)(C)=O)n1 68402,C#Cc1ccc(C(N2CCC3(CC(NC(=O)CCCCSC)C3)C2)=O)cc1C 68403,N1(C(=O)NC2CC(CCC)C2)CCN(C(c2csc(S)n2)=O)CC1.C(=O)N 68404,N1(C(C=CCC)=O)CCCC(O)(CCNC(=O)CNC(c2cccc(Cl)c2)=O)C1 68405,c1(C(=O)OC)ncc2c(n1)CN(c1cc(SC)nc(C)n1)C2.C1CN1 68406,c1(C(=O)NC(C2CCN(C(C3=C(C)OCC3)=O)C2)C)cc(C)cc(Cl)c1N 68407,C1(C(C)C)CC(NC(C2CC(C)(C)O2)=O)CO1 68408,Cc1cccnc1CCC(=O)NC(CN(C)C(c1cnc[nH]1)=O)(CO)CO 68409,c1(-c2c(OC)ccc(-c3nccn3CC(O)CO)c2)cc2cccc(OC)c2o1 68410,C(CC(C(=O)N1CC(C(=O)NCC2(F)CCCCC2)(SC)C1)OC)OC 68411,c1(SC)ccccc1CC(=O)NCC1CCN1C(c1cccc(NC(C)C)n1)=O 68412,N1(C(c2c(N(C)C)nccc2)=O)CCN(C(=O)C=CCF)CC1C1CCC1 68413,C(CCCCCCC(=O)N(CCNC(=O)CC1CC2CCC1O2)CC1CC1)SC 68414,C1(CNC(CC)=O)CC2(CN(C(=O)C(C)O)C1)CC2(F)F 68415,C1(NC(=O)CCc2cncs2)C=CCC(C(=O)NCCCCn2ccnc2)C1 68416,Cc1ccc2ccccc2c1-c1nnc(Sc2nnc(C3CC3)n2C)o1 68417,n1(CC(=O)NCC(C)(C(C)C)NC(C(c2cccnc2)SC)=O)nc(C)c(C)c1C 68418,C1(CC)CN(C(C2CNC(=O)N2)=O)CC1C(=O)Nc1c(C)nsc1C 68419,N1(C(CCCCCOC)=O)CC2CCOC2(CNC(=O)Cc2c(C)noc2C)C1 68420,c1(OCC)ccc(N(C(=O)CC)CC(=O)Nc2ccccc2N=[N+]=[N-])cc1OC 68421,c1(C(N2C(C)CC(CNC(C3(C=C)CCC3)=O)C2)=O)sc2ncccc2c1N 68422,N1(C(C(CC)CC)=O)CCCC(C)(C)C1CNC(c1c(C)ncnc1C)=O 68423,c1(-c2cn(C)nc2)ccc(C(=O)OC(C)(C)C)cc1.C1(=O)CC(c2ccccn2)N1 68424,CC(CC(C)(F)F)C(=O)NC(c1cn(CCN2CCNC2=O)nn1)(C)C 68425,Cc1cnncc1C(=O)NC(Cc1cccs1)CC(=O)NCC(N1CCOCC1)=O 68426,C1(C(N(C2CC2)CC)=O)Cc2nccnc2CN1C(c1snnc1C1CC1)=O 68427,c1(C(N2CCCC(OC)CC2C)C(=O)NC(CC)C)cc(Cl)c(OC)cc1F 68428,c1(OC)cc(CN2CCCC2)ccc1OCCON=NC1CC(C[Si](C)(C)C)C1 68429,c1(C(C(=O)NCC(CCOC)NC(c2sccc2C)=O)(F)F)ccc(C)cc1 68430,N1(C(C2=C(C)OCCC2)=O)CCOC2(C1)CN(C(=O)CC13COC(CF)(C1)C3)C2 68431,c1(NC(C2CC(c3ccccc3)CN2C(c2ccsn2)=O)=O)ncc(Br)cc1Cl 68432,N1(C(C(C)NC(=O)NC)=O)CCSCC1CCNC(c1oc(SC)cc1C)=O 68433,c1(C(=O)NCC(CNC(CC2(C=C)CCC2)=O)OC)cnnc(O)c1 68434,Cc1nc2ncnn2cc1C(=O)NC1CCCCC1NC(=O)Cc1cccnc1 68435,C1(C(=O)NCCC2C(C)CN(C(c3csc(C(N)=O)n3)=O)C2)COCC(C)(C)O1 68436,c1(C(N(C(C)CNC(=O)Cc2ccncc2Cl)C)=O)ccc(S(N)(=O)=O)cc1Cl 68437,C1(CC)(NC(=O)C(C)C(C)(F)F)CCN(C(=O)C(C)Cc2ccncc2)CC1 68438,C1(CNC(c2ccc3[nH]ccc3n2)=O)CCCC2CN(C(c3nncs3)=O)CC12 68439,C1(CC)CN(C(c2ccccc2Br)C(=O)Nc2cccc(OC)c2)CCO1 68440,C(C(O)C(=O)NC1(C)CC(NC(c2cc(C3CCC3)[nH]n2)=O)C1)=CC 68441,c1(N(C)C)cncc(C(=O)NC2CC(CO)N(C(=O)C(N3CCOCC3)C)C2)c1 68442,CC1CCc2nc(N3CC4CSCC(C4)C3)[nH]c(=NCC(Cl)(Cl)Cl)c2C1 68443,c1(C(=O)NC2C(C(N(CCCC(O)CO)C)=O)COCC2)ccc([N+](=O)[O-])[nH]1 68444,c1(C(=O)NCCC(C)N(C(C(CC)OC)=O)C)ccn(C)c(=O)c1 68445,CC(C)C(CC(=O)NCC1CC2CCC1CC2)NC(C1CC2(CCO1)CC2)=O 68446,c1(C(N2CCC(c3sc(C(=O)OCC)c(C)n3)C2)=O)c(F)ccc(O)c1O 68447,C1(CC)CN(C(c2cc(-c3cccnc3)no2)=O)CCN1C(=O)C1=CCC1 68448,C(=O)(C1CCc2nccn21)N1CC(C)C(NC(=O)CC2(n3cccn3)CC2)C1 68449,C(=O)(C(CN(C)C)CC)NCCCOCCNC(C(C)OCCCC)=O 68450,c1(C(C(=O)NCC(CCN(C(CC=C)=O)CC)O)CC)ccc(C(F)(F)F)cc1 68451,C(CC(C)CC)(C(=O)NCCC(=O)NCC)NC(CCCC)=O 68452,c1(NC)nc(C(C)C)nc2[nH]ccc12.C12(CCC1)N(C(C1(CCOC)CC1)=O)C2 68453,N1(C(C2(NC(C(C)OCC#C)=O)CCOCC2)=O)CC2CC(C)C2C1 68454,C(=O)(CCCC(=O)NC1CCOC(c2cccnc2)C1)c1ccc(OC)cc1 68455,c1(OCC)ccccc1CC(C)=CC(=O)NC1CC1NC(c1nocc1C)=O 68456,C(C1=NOC2CN(C(C3CS(=O)(=O)C3)=O)CC12)NC(c1cc(OC)ncc1Cl)=O 68457,C1(N(C)S(N)(=O)=O)(CO)CCN(C(C2CC23CC(F)(F)C3)=O)CC1.C1(=O)CN1 68458,C(C(C)(C)C(=O)OC)(c1n(CCCC)nnn1)NCC1CC(c2ccccc2)C1 68459,c1(C(N2CCC(C)(CC(=O)NC(CCO)C3CC3)C2)=O)cc2ncccc2[nH]1 68460,C1(NC(C(C)(C)OC(C)C)=O)C2CCC(C2)C1C(=O)N(CC(=O)N(C)C)C 68461,c1(C(=O)NC2CC(CCNC(C3(Cl)C(C)(C)C3)=O)C2)cc2cn[nH]c2cn1 68462,c1(N2CCC(CC(=O)NCC(C(=O)NC)C)C2)cc(C(=O)OCC)ncn1 68463,c1(CNC(C(C2CN(C(c3oc(CC)c(C)c3)=O)C2)OC)=O)ccc(C)nc1O 68464,C1(C)(NC(C(C2CCCCC2)NC(c2c(C)snc2)=O)=O)CCC2(CC1)CC2 68465,C1(C(=O)NC2CCC(NC(CCC)=O)C2)COCCN1C1CCCC1 68466,C1(C(=O)O)CN(C(c2nccs2)=O)CC12CN(Cc1cc(Br)cc(Cl)c1F)C2 68467,C=C1CC2CC1CN2C(=O)C(C1(O)CN(C(=O)CC2CCC2)C1)F 68468,c1(-n2ccc(C(N(CCN(C(C(F)OC)=O)C)C)=O)n2)cccc(F)c1 68469,C(CC(=O)N1CCCC1)N(C(C1CC1OC(=O)C=CCBr)=O)CC.C(C)(=O)O 68470,C(c1ccc(F)c(F)c1)=CC(N1C2C(NC(C(C(C)C)F)=O)C(CC2)C1)=O 68471,N1(C(c2cc3sccc3s2)=O)CC2(CCN(C3CCc4ccc(Cl)cc43)C2)C1 68472,c1(C(=O)NCC(CC)NC(C2CCCCC2C(N)=O)=O)ccnc(OC)n1 68473,N1(C(C2(CCNC(=O)CC3CCCOC3)CC2)=O)CC2CCCC1C2CO 68474,N(C1CCc2cc(CNC(=O)COC(F)F)ccc21)C(C1(C)CCC(=O)NC1)=O 68475,N1(C(C2(CC)CCCO2)=O)CC(CNC(c2cc(C)ncn2)=O)C(O)C1 68476,Cc1nc2n(c1CC(=O)OC(C)(C)C)CCCC2.C1(C)(c2nn[nH]n2)C(C)CO1 68477,c1(C(=O)NC2CN(Cc3c(C(F)(F)F)nn(C)c3Cl)C2)cccc2c1CCCO2 68478,Cc1nnc(CCC(=O)NCC(O)CN(C)C(C2CCC(O)C2)=O)n1C 68479,N1(C(C2C(Cl)(C(=O)OC)C2)=O)CC2CCC(CNC(C3CC(C(C)C)C3)=O)(C2)C1 68480,C(=O)(C(CC(F)F)N(C)C(c1ccc(F)cc1F)=O)N(CCCSC)C 68481,C1(NC(c2ccc(-c3ccccc3)s2)=O)CCCN(C(c2ccncc2)=O)C1 68482,C1(c2nc(C(N3CCC(C)CC3)C)on2)COc2ccccc2C1 68483,N1(C(C(CC2CCOCC2)NC(c2cnsc2)=O)=O)CC2COCC2C1 68484,N#CC1(CC(N2CC3(CCN3C(=O)C=Cc3cccnc3)C2)=O)CCOCC1 68485,C=C(C)CCC(=O)N1CCC(N(C(=O)C(=Cc2cnc[nH]2)C)C)CC1 68486,C#CC1(C(=O)N(CC(C)COC)C)CN(C(=O)C(=C2CCCCC2)F)C1 68487,C1(F)(CNC(C(C)NC(C)(C)C)=O)CCN(C(=O)CC2OCCCC2(C)C)CC1 68488,N1(CCC(NNC(C(C)Oc2ccccc2)=O)=O)C(=O)Cc2ccccc2C1=O 68489,N1(C2CN(C(C3(Nc4scc(C(C)C)n4)CCCC3)=O)C2)CCN(C)CC1 68490,C1(CNC(N(C(C)C2CC2)C2CC2)=O)CCCC(C(F)(F)F)C1 68491,c1(N2C(C)CCC(NC(c3c(C)ccnc3)=O)C2)ncc2ncnc-2[nH]1 68492,c1(C(=O)NC2C(CNC(COC(C)=O)=O)COC2)cccc2c1CC(C)(C)C2 68493,Cc1ccc(Cl)c(C(N2CCC(NC(c3nc(=O)n(C)[nH]3)=O)C(CO)C2)=O)c1N 68494,C1(c2cn(C)nc2)CN(C(C2CC23CCCCC3)=O)CCN1C(=O)CCC(F)(F)F 68495,C1(C(=O)NCC2(C)CCCN2C(c2ccncn2)=O)Cc2ccccc2S1(=O)=O 68496,N1(C(C(C(=O)OC)(C)C)=O)CC2CCCCCC2(C#N)C1 68497,C1(NC(CCC=C)=O)CCCC12CN(C(c1cc(Cl)cc(F)c1F)=O)C2 68498,C(=O)(CC(C(=O)NC1CC(C)(NC(C2CCOCC2)=O)C1)NC(C)=O)OC 68499,c1(NC(c2ccccc2C)c2n(C(CC)C)nnn2)cncc(C(=O)OCC)c1 68500,Cc1cc2[nH]c(C(N3CC4=C(C3)CN(C(C3(C)CCCCO3)=O)C4)=O)cc2s1 68501,c1(C(=O)NCC(C)NC(=O)CC2COC(=O)N2)ncc(Cl)nc1Cl 68502,Cc1cccc2c1CC(C(N1CC3CN(C(=O)C(C)C(F)F)CC3C1)=O)O2 68503,CCCC(O)CN=c1[nH]c2cc(Cl)c(S(=O)(=O)NC(CSC)CC(C)C)cc2s1 68504,C(=O)(C1=NNC(=O)CC1)NC(CCCC)CNC(c1cnc2n1CCS2)=O 68505,C=CCC(CNC(=O)OC)NC(=O)C(N(C)CCN(C)C=O)OC.C(C)(C)C 68506,N1(C(=O)CCC2CCOC2)CCCCC(C(=O)NC2(C3CC3)CCCC2)C1 68507,N1(C(C2(CC)CC2)=O)C2CCC1C(C(=O)NCc1ncn(C3CC3)n1)C2 68508,c1(C(N2CC3C(NC(=O)Cc4cscn4)(CCC3)C2)=O)cnc(O)c2cncn12 68509,Cc1csc2c(N(C3CCNCC3(C)C)CC=Cc3ccc(O)cc3)ncnc12 68510,N1(C(c2cscn2)=O)CCN(C(C2CC3(CCC3)CO2)=O)C(CF)C1 68511,N1(C(c2ccc(Cn3cc(C(=O)OC)nn3)cc2)=O)C2CCC1CC(F)(F)C2 68512,c1(NCC2(OC)CCOC2)[nH]c(=NC(C)c2cnn(C)c2)nc2sccc12 68513,Cc1cc(C(N2CC3(CC(NC(c4cnsn4)=O)CO3)C2)=O)c(Cl)cc1Cl 68514,c1(N2C(C)(C)C(NC(=O)Cn3cncn3)CC2)cc(C#N)ccc1[N+](=O)[O-] 68515,N1(C(c2ccn(CCC)n2)=O)CCN(C(c2cc(CN(C)C)on2)=O)CC1CF 68516,C(C)(CC(C)NC(c1ccnn1C1CC1(F)F)=O)NC(CNC(=O)OCC)=O 68517,c1(C(=O)NCC(CNC(c2cncc(OC)n2)=O)C)cc(C)nc(O)n1 68518,N1(C(C2C(CCOC)C2)=O)CCN(C)C(C(=O)NCC2(CO)CC3CC3C2)C1 68519,Cc1ccc(F)c(C(=O)NCC2C=CCN2C(=O)Cn2nc(Cl)ccc2=O)c1 68520,Cc1[nH]c(C#N)cc1C(=O)NC(c1nocc1C(=O)NCCOCC(F)F)C 68521,C1(C(N2C(C(C)NC(Cn3c(C)c(Cl)cn3)=O)CCC2)=O)CCn2cnnc2C1 68522,N1(C(c2scc(C)c2C)=O)C2CCCC1CC(NC(C1C=CCCC1)=O)C2 68523,N1(C(C(CC)O)=O)CC2(CCC2)CC1CNC(c1ccnc(-c2ncc[nH]2)c1)=O 68524,Cc1cc(C)n(CC(=O)N(C)CC2(O)CCN(C(c3[nH]c(O)nc3C)=O)C2)n1 68525,C1(C(=O)NC(C2(C(=O)OC)CC2)C)C=CCN(C(=O)CC23CCC(CC2)C3)C1 68526,N1(C(CC(C)=C(C)C)=O)CCCC(C)(C(=O)Nc2cccc(Cl)c2)C1 68527,C(CC)(CC)(CCNC(c1c[nH]cc1-c1cc(C)no1)=O)NC(C=COCC)=O 68528,C1(CNC(c2ccc(CC(=O)OC)cc2)=O)CN(C(c2ncoc2C)=O)CC1(F)F 68529,Cc1cccc2c(C(=O)NCC34CC(NC(=O)Cc5ccn(C)n5)(C3)C4)coc12 68530,CCC(F)(C(=O)OC)C(=O)NCCC12CCC(CC1)N(C(c1cn[nH]c1)=O)C2 68531,Cc1cncc(C(N2CCC(CCNC(c3nncs3)=O)C2)=O)c1 68532,C1(NC(c2c(CC)[nH]nc2Cl)=O)CCN(C(=O)C=Cc2cncc(O)c2)CC1C 68533,c1(C(N2CCC(N(C(COCC(C)C)=O)C)C2)=O)cc(N)cc(F)c1 68534,CCCCC(O)CC(=O)N1CC2C(CNC(=O)C=C(Cl)Cl)C2C1 68535,Cc1ccc(F)c(CNC(C2(CNC(C3CCS(=O)CC3)=O)CCOCC2)=O)c1 68536,C1(NC(CN(C)CCO)=O)CCN(C(=O)Cc2cnn(C(F)F)c2)CCC1CO 68537,c1(C(=O)NC2(NC(CC3(C(=O)OC)CC3)=O)CCC2)ccc(N(C)C)cc1F 68538,N1(C(C2C(C)CC2)=O)CCCC2CCN(C(=O)C=Cc3nccs3)CC12 68539,C1(NC(COc2c(C)cccc2)=O)CCCN(C(c2cccc(F)c2F)=O)C1C 68540,C1(NC(=O)C=Cc2ccccc2F)CCSC12CN(C(C1OCCO1)=O)C2 68541,C(CCCCN1CCCC1)NC(=O)NC(c1ccccc1)C(=O)NC1CCCO1 68542,Cn1cc(C(=O)NCC2(NC(=O)CC3=CCOCC3)CC2)c2ccccc12 68543,CC(c1ccccc1F)=CC(N1CC(N(C)C(C2COCCN2C)=O)C1)=O 68544,C1(CNC(C2(C(C)C)CCOCC2)=O)CNCC(C)(C)C1 68545,N1(C(C2OCC(C)C2)=O)CC2CCC1CC2NC(=O)CCNC(=O)CO 68546,C1(C(CO)NC(C2(NC(=O)COCC3CCC3)CC2)=O)CCCCC1 68547,c1(C(C)=O)ccc(C(=O)NC2CCC2NC(c2ccncc2)=O)cc1[N+](=O)[O-] 68548,C1(CNC(=O)NCC2CN(C3CC3)C2)CC2CCC(C1)S2 68549,c1(C(C(N2CC(C(C)NC(=O)C(CC)N3CCCC3=O)C2)=O)C)c(C)noc1C 68550,C1(NC(=O)CC2(O)CCC2)CC2CCC1CN2C(C1CNC(=O)N1)=O 68551,C#CCCC(C(=O)Nc1cccc(C#N)c1)NC(c1[nH]nnc1C)=O 68552,C(=O)(CC(C)CC(C)(C)C)NCCC(=O)NCc1ncc(C)cn1 68553,Cc1ccc(C(=O)NC2CCOCC2NC(C23CC(F)(C2)C3)=O)c(F)c1F 68554,N1(C(C(C(C)NC(=O)C(N2CCNC2=O)C)(C)C)=O)CCC2CCCC2CC1 68555,C1(C(=O)NCC23C(CN(C(CNC(=O)OC)=O)C2)C3)CCc2nc(C)[nH]c2C1 68556,Cc1nc(CNC(=O)CC2C3CN(C(=O)CCc4ccccc4F)CC23)oc1C 68557,c1(C(N(C(C(=O)NC(CCC)c2nn[nH]n2)C)C2CC2)=O)snc(C)c1N 68558,CN1CCC(NC(=O)C(C2(C)CC2)NC(c2cc3n(n2)CCC3)=O)C(C#N)C1 68559,C(=O)(C(F)(F)C(C)O)NCCOC(CNC(C=C(C)c1ccco1)=O)(C)C 68560,c1(C(=O)NC2C(NC(c3ccoc3)=O)CC2)c(F)cc([N+](=O)[O-])cc1Br 68561,c1(C(N2CCCC(CCNC(C(C)=CC)=O)C2)=O)cccc2c1OC(C)C2 68562,CCC(C)(C(=O)N1CC(CO)(NC(c2cocn2)=O)C1)OC 68563,N1(C(c2c(CC)ocn2)=O)CC(NC(=O)C=Cc2cccc(F)c2)CC1(C)COC 68564,CC(C(C)(C)NC(=O)CCC1CC1(F)F)NC(=O)CSCC(N)=O 68565,c1(C(=O)NCC(C2CC2)NC(=O)COc2ccccn2)cc2cc(F)ccc2o1 68566,O=C(C#CC1CCOC1)NC1CN(CC2CCc3ncnn32)C1 68567,N1(C(C(CC)N(C)C(c2ncnc(C)c2C)=O)=O)CCCC(C)(C)C1C 68568,N1(CC)CC2CCC1CN2C(C1CC(NC(=O)OC(C)(C)C)CCO1)=O 68569,N1(C(C2(CC=C)CCN(C(=O)C(C)OCCC(C)C)C2)=O)CCC(O)CC(C)C1 68570,N1(CC)CCN(C(C2CCN(C(=O)C(Cl)Cl)C(C)C2)=O)C(C)C1 68571,c1(SCCCC(=O)NC2CCCC(CNC(CSC)=O)C2)ccc(C#N)cc1 68572,N1(C(c2c(C)nc(O)[nH]2)=O)CC(CNC(=O)C2=NOC(C)C2)CC1(C)C 68573,CCCCCCOCC(=O)NCC1(NC(=O)CCc2cnc(O)[nH]2)CCOC1 68574,CN1CCC(C(N2CCC(N3CCCC3)C2)C(=O)NCc2ccco2)CC1 68575,c1(OC)cc(C(CO)NCc2cc(Cl)ncc2NC(=O)OC(C)(C)C)cc(F)c1 68576,C1(NC(=O)CC2CC3(CCC3)CO2)CN(C(c2cncc(F)c2)=O)C2(CCC2)C1 68577,C1(CN(C(=O)C=CC(F)(F)F)CC)CCCN1C(=O)C(F)OC 68578,C1(C2CC2)(CNC(C2(OC)CS(=O)(=O)C2)=O)CCN(c2nc3ccccc3o2)C1 68579,c1(C(=O)NC2C(CNC(COCC(=O)NC)=O)C2)cc2ccc(Cl)c(F)c2[nH]1 68580,N1(C(CC(=C)C)=O)CCCC2CN(C(C3CCc4c(nnn4CC)C3)=O)CCC12 68581,C1(C#CC(=O)N2CCCC(CNCC34COC(C3)C(OC)C4)CC2)(CC)COC1.OC 68582,N1(C(C2C(C)(C)CCN2C(C2CCCOC2)=O)=O)CCCC2C(=O)NCC12 68583,Cc1cccc(C)c1C(=O)NC(C1CCCN(C(=O)CC(C)(C)C#N)C1)C 68584,c1(CC(N2CCC(C(C(C)C)NC(=O)CC(F)F)CC2)=O)c[nH]c2ncccc12 68585,Cn1c(O)nc2cc(C(=O)NC3CN(Cc4ccc(Br)cc4)CC3(C)C)ccc12 68586,Cc1noc2ncc(C(N3CC(NC(c4ccc(Br)o4)=O)C4CC4C3)=O)cc12 68587,CC1(C)CC(O)(CC(N2CC(CCCCNC(c3nn[nH]c3Cl)=O)C2)=O)CO1 68588,c1(S(CCOC)=O)cc(Br)ccc1S(=O)(=O)N1CCOC(OC)C1 68589,Cc1ccc(CN(C)Cc2cn(-c3cc(Cl)cc(Cl)c3Cl)nn2)c2cccnc12 68590,C(=O)(CC(C)CC(F)(F)F)NC1(CNC(C2ON=C(C(C)C)C2)=O)CCCCC1 68591,Cc1cc(C(=O)NCCCCNC(=O)CC2COC3CC2C3)oc1Br 68592,C(=O)(C1=CC2C=CC1C2)N(CCC(=O)Nc1cccc2c1OCC2)CCCO 68593,C1(NC(CN(C(C)=O)C)=O)CCC(C)(CNC(=O)Cc2csnc2C)C1 68594,C1(=CC(=O)NC(CCC)CCCNC(=O)C(C)CF)CC2CCC(C1)N2C 68595,C#CCCCCCCC(=O)NC1CC(NC(c2ocnc2CC)=O)CC1O 68596,N1(C(CNC(=O)CC(F)(F)F)=O)CCN(C(=O)C=CC2CCOC2)C2CCCC12 68597,C(=O)(C1=CS(=O)CCC1)NC12CCC(CNC(c3n(CC)nnc3)=O)(OC1)C2 68598,c1(C(N2C(CCNC(CC3ON=C(C)C3)=O)COCC2)=O)ccc(Cl)cc1O 68599,c1(C(N(C)CC2(NC(=O)CCc3cn[nH]c3)CC2)=O)ccnc(Cl)c1Cl 68600,c1(C2(OC)COC2)cccc(C(=O)NCC(c2cccc(Cl)c2)O)c1.CCC(C)C 68601,N1(C(C(C(C)C)n2ccc(C)c2)=O)CC(O)C(O)C(O)C1c1noc(C2CC2)n1 68602,C1(C(C)C)COCCN(C(=O)CCOCCN(C(=O)C(O)C(C)(C)C)C)C1 68603,c1(N(C(C)(C)C)C(N2CCOCC2)=O)ccc(F)c(OC(C2CN(S(N)(=O)=O)C2)=O)c1 68604,c1(C2CC(CNC(C(c3cccc(F)c3)N)=O)C2)ccc(F)c(F)c1 68605,c1(CC(N2CC(F)(CNC(C3(COC)CCCC3)=O)C2)=O)cc(F)ccc1C 68606,C1(C(=O)OC)CN(C(N2CCCC2CC2CC2)=O)CC1(C)C(F)(F)F 68607,C1(C2CC2)(C(N2C(C)CC2(C)C)=O)CN(C(=O)CC2CC3C=CC2C3)C1 68608,c1(C(=O)NC2CC(C)(NC(=O)CC3CCC(F)(F)CC3)C2)ccc2nonc2c1 68609,CC(C)(C)CC(O)CC(=O)NC1CCCCC1NC(c1cc2cccnn2c1)=O 68610,C(C)(N=c1ccnc(NCC2CC2(C)C)[nH]1)c1ccc(SC)cc1 68611,CCC(C)CCC(=O)NCC(C)(CNC(c1ccc(F)cn1)=O)OC 68612,CCC(CC(=O)NCC(O)CNC(C1CC(C(F)F)C1)=O)C(F)F 68613,C(=O)(C#CC(C)(C)CNC(=O)C(C)CC)NC(CCC)CC 68614,C(=O)(C1=C(Cl)CCC1)N1C(C(C)NC(=O)CCOCC(F)F)CCC1 68615,C1(n2cc(C(C3CC(=O)NC3=O)C)nn2)CCN(C(=O)CC2CCCOC2)CC1 68616,CCCCC(C(=O)NCC1(CC(C)C)CCC1)NC(c1cn(C)nn1)=O 68617,CC(C)CCCC(C)C(=O)N(C)C.C12Cc3cc(ccc3O1)C(=O)OC2 68618,N1(C(CN(C2CCC2)C)=O)CCN(C(C2CC23CCOC3)=O)CC(O)C1 68619,Cc1c(N(C(=O)OC(C)(C)C)C(C2CC3(CSC3)C2)=O)cncc1N 68620,C=CCCCCCC(=O)NC1(C2CC2)CCN(C(c2ccc[n+]([O-])c2)=O)C1 68621,N1(C(c2c(C)ccc(=N)[nH]2)=O)CC2CCCC2(NC(=O)CCC2CCOC2)C1 68622,C1(C(N(C2CCN(C(=O)CCC(C)N(C)C)C2)CC)=O)C(C)(C)C1(C)C 68623,N1(CCc2cn(CC(C)NC(C3CC(F)CS3)=O)nn2)CCS(=O)(=O)CC1 68624,C1(CCC)COCCN1C(C1CCCCC1NC(c1ccncc1OC)=O)=O 68625,Cc1cc(=N)[nH]cc1C(=O)NCC1CCCCC1NC(=O)C(C)(C)C(C)C 68626,c1(CC)nc(C(=O)NCCC2CCN(C(C3(CC)COC3)=O)C2)c(C)o1 68627,N1(C(c2c(OC)nn(C)c2)=O)CCC(NC(c2cc(F)ccc2OC)=O)C(C)C1 68628,C(C1NC(=O)c2ccccc21)NC(=O)Nc1cc(C(F)(F)C(F)(F)F)on1 68629,N1(C(CC2C(=O)OCC2)=O)CC(O)(C2CCN(C(=O)CCC3CC3)CC2)C1 68630,N1(C(C2CN(C(c3c(C)nc(O)s3)=O)C(C)(C)C2)=O)C2CCC1CC(=O)NC2 68631,C1(CNC(C2CCOC2)=O)CN(C(=O)CCCNC(C2CCCC2)=O)CC12CC2 68632,N1(C(c2c(OC)nsc2)=O)CC2=C(C1)CN(C(=O)CC1C=NN(C)C1=O)C2 68633,c1(NC(=O)Nc2cc(C)sn2)cccc(CC2CC2)c1 68634,C1(NC(C(C)(C)NC(C=COC)=O)=O)CN(C(c2cnc(C(C)C)s2)=O)CC1F 68635,C1(C)(CC)CCC(C(=O)NC2CC(NC(=O)C3=C(Cl)CC3)C(O)C2)O1 68636,c1(OC)cc(NC(C2CN(C(c3c(Cl)ccnc3Br)=O)CCS2)=O)nc(Br)c1 68637,C12(C(=O)NC3C(C)(C(=O)NCc4ccc(OC)cn4)CCC3)CC(C)(CCO1)C2 68638,c1(C(=O)NC2(CNC(CNS(CCC)(=O)=O)=O)CCC2)cc([N+](=O)[O-])ccc1O 68639,C(=O)(C#CC1CCCC1)NCCN(C(C(CCC)(F)F)=O)CC 68640,C(C(C)(C)CC(=O)NCCOc1ccccc1)NC(C(C1CCC1)OC)=O 68641,C#CC(C(C)(C)C)NC(=O)C(C(C)O)NC(=O)C=CC(C)CC 68642,C1(NC(c2ccc(CC)cc2)=O)CN(C(=O)CNS(=O)(=O)CC)C2CCCCC12 68643,N1(C(c2cnc(CC)s2)=O)CC2CC(NC(=O)CNS(=O)(=O)NC)C2C1 68644,c1(C(=O)NCC(CC(F)(F)F)NC(C(C)(F)F)=O)ccc(P(C)(C)=O)cn1 68645,Cc1nn(C)c(C)c1NC(C1CCN(C(c2ccc(Cl)cc2Br)=O)C1)=O 68646,C1(NC(C(C2CC2)NC(CCOC(C)=O)=O)=O)CN2CCC1(C)CC2 68647,N1(C(COCCCCC)=O)CCc2sccc2C1CNC(C12CC(CCO1)C2)=O 68648,CC1CN(C(=O)C#CC(C)(C)C)CCC1NC(c1cccc(NS(N)(=O)=O)n1)=O 68649,c1(C(=O)NCC2(C)CC(NC(c3cc(Cl)ccn3)=O)C2)cc2n(n1)CCCC2 68650,N1(C(CCC2(NC(CSCCC(C)C)=O)CCC2)=O)CCOC(C(C)C)CC1 68651,c1(C(N2CCC(NC(c3c(C)[nH]cc3)=O)C2)=O)cc(C)n(C2CC2)c1C 68652,C(=O)(C1=NOC(C2(O)COC2)C1)NC(C)CNC(=O)CC(C)(C)c1ccc(F)cc1 68653,C1(CNc2ccc(N3C(=O)OCC3)cc2)CC2OC1C1CC21 68654,Cc1cccc(C(N2CCN(Cc3ccc(F)c(F)c3)C(C)C2)=O)c1C 68655,c1(OC)cc(C(=O)NC(C)C(C2CCCCC2)NC(=O)CSC(F)F)on1 68656,C(C(C(=O)NC1CCC1C)C(C)C)NC(CCC(=O)NCCC)=O 68657,C1(NC(c2cccc(C3CC3)c2)=O)CC1C1CCCN(C(c2cccnn2)=O)C1 68658,c1(OC(C(=O)N(CCN(C(c2cc(CCC)on2)=O)C)C)C)ccc(Cl)cc1C 68659,C1(OC)CC(CNC(=O)CN2CCN(C)CC2)N(C(C2CCC2CF)=O)C1 68660,N1(C(C=CCN(C)CC)=O)CC2CCCC2(CNC(=O)CCCCN(C)C)C1 68661,c1(C(N(C2CCCN(C(C3CCCC4CC34)=O)CC2)C)=O)nc2ncccn2n1 68662,N1(Cc2cncc(-c3c(CC)ncs3)c2)CCC(N(C)CC)CC1C 68663,c1(OC)ccc2oc(C(N3CC4CC3C4C(=O)Nc3ccc(O)nc3)=O)cc2c1 68664,c1(OCC(=O)NC(CC(C)C)C(=O)NCC2CSC2)ccccc1[N+](=O)[O-] 68665,N1(C(C#C)=O)CCn2cc(C(=O)NCCOCC)nc2C1 68666,CC1CC(CNC(c2cnc[nH]c2=N)=O)CN1C(=O)CCc1cnccn1 68667,O=Cc1cccc(CN2CC3(CCC(C(=O)NC4CSC4)O3)C2)c1Br 68668,C1(C2CC2)(CNC(C(c2cccs2)NC(=O)CC2CC=CC2)=O)CCCO1 68669,c1(CS(=O)(=O)NC(c2nncs2)CC)cccc(F)c1 68670,N1(C(C2CC(C)(C)NCC2)=O)CC(C)(C)C(O)C1(C)C 68671,C12(NC(c3c(C(N)=O)csc3)=O)CCC(CC1NC(c1ccc(F)c(O)c1)=O)C2 68672,C1(N(C(=O)C(F)CC)CC#C)CCN(C(=O)C(C2CCOCC2)F)CC1 68673,C1(CC(=O)OC)(NCC(c2ccc(C)cc2)O)CS(=O)(=O)C1 68674,c1(CN2CCC(NC(c3cccc(C(F)(F)F)c3)=O)CC2)c(Cl)cc(Cl)cc1Cl 68675,C(=O)(C1=NOC2COCC12)N1C2C(NC(CCNC(=O)CO)=O)CC(C2)C1 68676,c1(COC)nc(Cl)cc(=NCCOC)[nH]1.C12(C(=O)N)CCC(C1)OC2 68677,CC1CCN(C(C2CCCC2(C)C)=O)CCN1C(c1cnco1)=O 68678,CCCCC(C(=O)NCCC1CCCCN1C(=O)CN(C)C)C(C)C 68679,n1(CC(=O)N(C(c2ccccc2)CNC(c2cnnn2C)=O)C)nnc(C2CC2)n1 68680,C(CCCCCNC(c1c(Br)nnn1C)=O)NC(CC1ON=C(C)C1)=O 68681,C(CCCC(=O)OC)(C(=O)NCc1cccc(Br)c1)N1CCCC(COC)C1 68682,C1(C(=O)NC(C)(C)C(O)CO)CN(C(=O)CSC(F)(F)F)CCC1(C)C 68683,Cc1cc(C(=O)NCC(=O)N(CCCN(C(=O)C(F)CC2CC2)C)C)c(C)o1 68684,C(=O)(C1CCc2c(Cl)cccc21)N(C(Cc1ccc(C)cc1)C(=O)O)CCN(C)C 68685,N1(C(C2C(C=C)OCCC2)=O)CCC2(CCCN2C(=O)Cc2c[nH]nc2C)CC1 68686,CC1=CCCN(C(=O)C(Cc2ccco2)NC(C2CCN(C)CC2)=O)C1 68687,S(=O)(=O)(c1cn(-c2ccccc2)nn1)NCC1(CO)C(C)(C)C1 68688,C(=O)(C(O)CC(C)(C)C)NCC1C(NC(c2c(C)[nH]c(C#N)c2)=O)CC1 68689,C1(C(=O)NCCOCC)CCOCC1NC(C1OC2CCC1C2)=O 68690,c1(C(=O)NC2C(CNC(C3(Br)C(C)(C)C3)=O)C2)ccn2c(O)nnc2c1 68691,C(C(COC)C(=O)NC(CO)C(C)NC(C1(N(C)C)CCC1)=O)OC 68692,c1(CN(C(c2nc(C)cs2)C(=O)NC(C(=O)OC)C)C)ccc(Cl)cc1F 68693,C12(COC)CC(CNC(c3ccc(Cl)o3)=O)(CN1C(C1(C(F)F)CCCO1)=O)C2 68694,C1(NC(C(C2CCOC2)NC(CCC(CC)OC)=O)=O)CC2CC1C(O)C2O 68695,C1(C(C)NC(c2cc(C(C)=O)on2)=O)CN(C(C2CCS2(=O)=O)=O)CCO1 68696,N1(C(c2ccc(C3CC3)nc2O)=O)CC2CCCN(C(=O)Cc3cccs3)C2C1 68697,Cc1cc(C(=O)N(CC(C)CNC(c2c(C(F)F)cnn2C)=O)C)sc1C 68698,C(C(=O)NCc1cn(C2CN(C(=O)CC(C)C)C2)nn1)(C(C)(C)C)NC(C)=O 68699,N1(C(C(C(C)CNC(C23CC(F)(C2)C3)=O)F)=O)CCCCN(C)CC1 68700,c1(-c2scc(CC(=O)NCCN(C(c3c(CC)nco3)=O)C)n2)ccc(O)cc1 68701,Cc1cc(CC(=O)NC2CCCC2n2cc(C3CC34CC4)nn2)cc(C)c1Br 68702,C1(NC(C2C(OCC)C2)=O)CN(c2nnco2)C1 68703,c1(C(=O)NC2C(NC(c3sc(CC)c(C)c3)=O)CC2)ccc(F)c(F)c1C 68704,C1(C(=O)NCCN(C(CN2CCN(CC)CC2)=O)C)CC(C2CCCC2)C1 68705,c1(C(N(CCOC)CCNC(=O)Cn2cnccc2=O)=O)cc(O)cc(N)c1C 68706,C(=O)(C(CCNC(c1ccc[n+]([O-])c1)=O)OC)NCC1CCN(CC)C1 68707,C=CCC(C)C(=O)NCC1(CC(=O)NC(CCOC)C(C)C)CC1 68708,N1(C(CSSC)=O)CCC2(CCCCC2NC(c2nncs2)=O)CC1 68709,N1(C(C2(C=C)CCN(C(=O)CN(C3CCC3)C)C2)=O)CC2CC(C)(C)C2C1 68710,O(C=CC(O)(Cn1cc(CN)nn1)C(F)(F)F)CC.C1(=O)C(C)(COC)N1 68711,c1(OC)c(C(=O)NC(C2CCCCN2C(=O)CCN(C)CCO)C)cccc1F 68712,Cc1cc(C(N2CC(NC(C3C4COCC34)=O)C(n3cccn3)C2)=O)nc(C)n1 68713,C(C)(CNC(C1(C)CC1(F)F)=O)(CC(C)C)NC(C=CCCC)=O 68714,Cc1nc(C(C)(C)C)nc(O)c1C(=O)NCC1CC(F)CN1C(c1ccsc1)=O 68715,c1(C(C)=O)nc(N2CCOC(C(C)NC(=O)C3=C(C)OCC3)C2)ncc1Cl 68716,CC(=O)CCCC(=O)N1C(C(=O)N(C)CC2(N(C)C)CCC2)CCC12CC2 68717,C#CC1CCCC(NC(C2CC(F)(F)CN2C(=O)CCOCC(F)F)=O)C1 68718,N1(C(c2csnn2)=O)CC2CCC2(CCNC(C23CC(CC(F)F)(C2)C3)=O)C1 68719,N1(C(C(C)NC(N)=O)=O)CC(CNC(=O)Cn2nccn2)C(c2ccccc2)C1 68720,C(=O)(C1=NOC2COCC12)N1CC=C(C(=O)NCCC(C=C)C)CC1 68721,c1(CC(N2CC(OCCNC(COCCC(C)C)=O)C2)=O)ccc2ccoc2c1 68722,C1(NC(c2c(CC)scc2)=O)C(C)CN(C(=O)CSCCOC)CC1C 68723,C(CSC)(C(=O)NC1CCCC1NC(c1coc(C)c1)=O)OC 68724,S(=O)(=O)(c1cccc(Br)n1)N1C(C)(C(=O)NCc2cncc(Br)c2)CCC1 68725,C1(NC(C(CCC)C)=O)CCC12CCN(C(c1c[nH]c(=NC)s1)=O)CC2 68726,C1(NC(=O)OC(C)(C)C)CCCC2CN(C(c3noc4cc(F)ccc34)=O)CC12 68727,N1(C(COCCOCC#C)=O)CC(C)CCC1CNC(=O)C(=O)NC1CC1 68728,CCCCCCC(=O)N1CCCC1CNC(c1cccc(Cl)c1OC(F)(F)F)=O 68729,C1(OC)COc2c(C(N3CCCC3CN(C)C(c3scnc3Cl)=O)=O)cnn2C1 68730,O=c1cc(-c2ccccc2)oc2cc(F)c(OCCN3CCCC3)cc12 68731,Fc1cncnc1Cc1nnc(N2CC3CCC2C3)n1CC(c1ccccc1)F 68732,c1(OC)ccc(C(=O)NCC2CC(OC)CN2C(=O)Cc2cc(C)cs2)cc1Cl 68733,c1(C(=O)NC2CC(C(N3CCC(C4CCCO4)C3)=O)C2)ccnc(CO)c1 68734,Cc1nc(Cl)nc(N2CCC(NC(C3CCCC(F)(F)CC3)=O)CC2)c1[N+](=O)[O-] 68735,CC(C)(C#N)CCC(=O)NC1(CNC(c2cc3ccccc3o2)=O)CCOC1 68736,C1(C(C)C)CN(C(C2(Cl)CC23CCC3)=O)CCN1C(c1sccc1CC#N)=O 68737,C1(C(NOCC(CC)C)=O)CCC(C)N1C(c1ccc(C)n1C)=O 68738,c1(C(=O)NCC2C(NC(C3CC=C(C)CC3)=O)C2)cn(C)cc(Br)c1=O 68739,C=CC(C)(C)CC(=O)NC1(CNC(=O)COCc2ccnn2C)CCCCC1C 68740,c1(C(=O)NCC2N(C(Cc3cn(CC)nc3)=O)CCC2C)cc(Cl)c([N+](=O)[O-])[nH]1 68741,CC1=NOC(C)(C(N2CC3C(NC(c4cn(C(F)(F)CO)nn4)=O)C3C2)=O)C1 68742,c1(C(c2ccccn2)NC(c2ccc(C3CC3)cn2)=O)ccccc1F 68743,CC1CC(NC(C2(F)CC2)=O)CCN1C(c1ccc(-c2ccccc2)cc1F)=O 68744,c1(NCC2(NC(C(C)C3CC3)=O)CCC2)ccc(Cl)cc1Cl.C1(C=O)C2CCCC12 68745,C(C(O)C(=O)NCCN(C(=O)C(C)N(C)C)CCSC)SC 68746,C1(CC)CN(C(C2CC3CC3CC2C)=O)CCN1C(c1ccccc1CC#N)=O 68747,C1(CC(C)NC(C=C(C)C(C)C)=O)CCN(C(c2cc(C3CC3)no2)=O)CC1 68748,CCC(CCCC(=O)NC1(C)CCCC1(F)F)NC(c1c(C)ccn1C)=O 68749,C#Cc1ccc(CC(N2CCC(F)(C(N3CCC(F)(CO)C3)=O)CC2)=O)cc1 68750,C1(C(=O)NC(C)CC2CCOCC2)CC(F)CN1C(=O)CCOC1CCCC1 68751,C=CCCCC(C(=O)NCC(C)(O)CC)NC(=O)Cc1cc(C)on1 68752,n1(CCOC)nnnc1C1(NC(C)Cn2cncn2)CCC1 68753,c1(C(N(CC(C)NC(c2n(CC)c(O)nc2)=O)C)=O)cc(S(=O)(=O)N(C)C)c[nH]1 68754,c1(C(=O)NCC(=O)NCCC(C)NC(c2cccc(=O)o2)=O)ccc(N)cc1 68755,C(C)(C)(C(C)CC(=O)N1CCC2CC12)NC(CC(C)CN(C)C)=O 68756,Cn1c(NCC2CC(NC(=O)CN3CCCC3=O)C2)c(C#N)c(=O)n(C)c1=O 68757,CCCC(C)CC(=O)N(CCNC(C1(c2ccccc2C)CCCC1)=O)C(C)C 68758,C1(CCC(=O)NC2(COC)CCC2)CCN(C(=O)CCn2ccnn2)C1 68759,Cc1cc(-n2cc(CONC(C3CCCC(NC(N)=O)CC3)=O)nn2)cc(C)c1 68760,C1(NC(c2scc(OC)c2OC)=O)CC2(C1)CN(C(C1CC1(C)C)=O)C2 68761,C1(OC)CCC2(CCN(C(c3ccc(CNC(=O)C4=CCOCC4)s3)=O)C2)C1 68762,c1(C(N2C(C(N3CC(C=C)C(O)C3)=O)C(CC)CC2)=O)cccc2ccoc12 68763,c1(COC)csc(C(N2CCC(CNC(C3CC3(Cl)Cl)=O)C2)=O)c1 68764,C(=O)(CS(=O)c1ccc(Cl)cc1)N1C(CNC(CSCC)=O)CN(C)CC1 68765,c1(C(C)(C)C)ccc(C(N2CCCC(N(CCO)C(c3cscc3Cl)=O)C2)=O)cc1 68766,CN1CCN(C(=O)CCCCc2ccc(C#N)cc2)CC1CNC(C1(F)CC1)=O 68767,C1(CNC(C2CCC2)=O)CC(CNC(=O)C(C)OC2CC2)CO1.CCSC.C 68768,Cc1cc(Cl)n[nH]c1=NC(=O)C1CC(O)CN1C(c1cccc2c[nH]nc12)=O 68769,N1(C(C2(COC)CC=CC2)=O)CC2(CC(NC(=O)CN3CCOCC3=O)CO2)C1 68770,C1(C)(NC(C2CC(=O)N(C)C2c2ccccc2)=O)CCc2ccccc2C1 68771,n1(CCC(=O)NCCOCC(=O)NCC(C)(C2CC2)OC)ccnc1C 68772,N1(C(C(CC)C)=O)CCC(NC(=O)CN(C2CCCC2O)C)C1C 68773,Cc1ccc(C)c(CNC(=O)C(C2CCN(C(=O)Cn3nccc3C)CC2)C)c1 68774,C1(CN(C(C2CCC(C)S2)=O)C)CCN(C(=O)CCc2cccnc2)CC1 68775,N1(C(CCN(C)CC)=O)CCC(C)(CNC(C2CCC(F)C2)=O)CC1 68776,C1(NC(COCCOCCOC)=O)CN(C(=O)Cc2ccccc2)CC1O 68777,CON1CC(C(=O)NC2CCCCC2NC(=O)C(F)(F)c2ccncc2)CC1=O 68778,C1(NC(=O)Cn2ncnn2)COC2(C1)CN(C(c1cc(CCCO)on1)=O)C2 68779,CC1(NC(C2CC2C(F)(F)F)=O)CCCN(C(C23CC4CC2C3C4O)=O)C1 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68798,C(CC(C)C)(C(=O)NC(C(=O)N(CC1=CCCOC1)C)C1(O)CCC1)OC 68799,CN1CCC(C(=O)N(C)CC2CC(F)(F)C2)(NC(=O)Cc2cnn(C)c2)C1 68800,Cc1[nH]nc(Cl)c1C(c1nnnn1C)NCCCc1cnoc1 68801,C1(NC(C2C(CC)CCC2)=O)CC12CCN(C(=O)CCc1ccccn1)C2 68802,N1(C(CC2CC(SC)C2)=O)CC2CCC1CC2NC(c1ncnc(C)c1C)=O 68803,C1(CC(=O)NC)(CC)CCCN(C(=O)OC(C)(C)C)C1.N12CCC1C2=O 68804,c1(C(=O)NC2C(CSCC)C2)ccc(OCc2cnn(C)c2)nc1.C1C(=O)N1 68805,N1(C(c2c(OC)scc2)=O)CC(C(=O)NCC2(C)CCC2)C(C(C)C)C1 68806,Cc1cnc(CCC(=O)NC(C2CCCN2C(c2nnn(C(C)C)n2)=O)(C)C)[nH]1 68807,c1(C(=O)NC2CCC(NC(C3N(C(CC)=O)CSC3)=O)C2)cnccc1Cl 68808,Cc1c(F)cc(C(=O)N(CC(C)NC(=O)C(C)(C)C2CC2)C)c(F)c1N 68809,c1(C(=O)NCCn2cc(C(N(C)Cc3nc(=O)o[nH]3)=O)nn2)cc(C#N)cn1C 68810,c1(CN(C(C)C)C)ccc([N+](=O)[O-])cc1.c12ccccc1-c1cc(ccn1)NC2 68811,C(CC(=O)N(C1CN(C(c2cncn2C)=O)CC1O)C)(C(F)(F)F)OC 68812,O=C(C1=C(Cl)CCC1)NC(Cc1ccco1)C(N1CC2(CCC2)C1)=O 68813,CC1CCCN(C(c2c[nH]nc2C(F)F)=O)C1CCNC(c1ccc(C#N)[nH]1)=O 68814,C1(C2CCCCO2)(C(N(C)CC2CC2)=O)CCCO1 68815,C1(CC)CCCC1C(=O)NCc1ccc(C(=O)N(CCCF)CC)o1 68816,C1(C(=O)NCC(=O)NC(C)C)CCN(C(=O)COc2ccn(C)n2)C1C(C)C 68817,c1(OC)ccnc(C(N2CC(NC(c3cn(CCO)nc3C)=O)C(C)C2)=O)c1O 68818,C(=O)(CCCC(C)c1ccccc1)N(CCNC(C1(OC)CCSCC1)=O)CC 68819,c1(C(N2CCC(CNC(CCc3scc(C)c3)=O)C2)=O)ccnc(C)n1 68820,N1(C(C(C)=CC=Cc2ccccc2)=O)CCOCC(CNC(=O)C=CS(C)=O)C1 68821,C1(CC(N2CCN(C(C(C)OC)=O)C(C)C2)=O)SC2=NCCN2C1=O 68822,c1(C(=O)NCCCN(C(CCc2onc(CC)n2)=O)C)ncnc(O)c1Br 68823,c1(CC(N2CCC(CCCNC(C=C(CC)C)=O)CC2)=O)ccc(F)cc1F 68824,C(=O)(CC(C)CC(=O)OC)N(C(CC)C(=O)NC1COCC1O)C1CC1 68825,c1(C2(C(N(CCNC(CC3(C(=O)OCC)CC3)=O)C)=O)CC2)cccc(Cl)c1 68826,c1(NCC2CC(C)N(C(c3csc4ccccc34)=O)C2)ncnc2c1ncn2C 68827,C=CCC(CC(C)C)C(=O)N1CC2(C1)CN(C(C1CCCCC1CC)=O)C2 68828,C12(C(=O)NC3(CC=C)CN(C(=O)CCCCn4ccnn4)C3)CCC(C)(C1)OC2 68829,N1(C(C=C=C(C)C)=O)CCCC(C)C1CNC(c1c(Cl)sc(C)c1C)=O 68830,c1(-c2scc(C(=O)OCC3CCC(C)CC3)n2)c(F)cccc1F 68831,N1(C(C2CCc3nnc(O)n3C2)=O)CCC2C(CCCN2C(C2CC(F)C2)=O)C1 68832,C(=O)(C(=O)N=c1ncn(-c2ccccc2)[nH]1)NC1C(C)C2CCC1C2 68833,Cc1ccc(CNC(=O)CC2(CNC(C3CCC3C)=O)CC2)cc1F 68834,C1(N(C(=O)C(C)OCC(F)(F)F)CC)CCCN(C(=O)Cc2nccn2C)CC1 68835,C12(NC(C(C)OC)=O)CCCC1N(C(=O)CCc1cn[nH]c1)CC2 68836,Cn1nc(O)cc1C(=O)NC(C)(C)CNC(=O)Cc1csc(-c2ccoc2)n1 68837,C=C(C)C1OCCC1CNC(=O)CN(C(=O)Cn1ccc(C)n1)C1CCC1 68838,Cc1ccc2c(C(N3CC(CN4CCN(C(=O)C(C)(C)CO)CC4)C3)=O)csc2c1 68839,c1(OC)cc(C(C)=O)ccc1-c1cc(N2CCN(CCO)CC2)ccn1 68840,C(=O)(C(F)(F)F)NCC(=O)NCCCN(C(=O)CNc1cccnc1)CCO 68841,C=CC1CN(C(=O)C(C)P(C)(C)=O)CC1NC(c1cnc(C2CC2)nc1)=O 68842,c1(C(=O)NCCCCNC(C2(C)C(C)CCCC2)=O)cccc2c1ncn2C 68843,C1(NC(CCc2onc(C)n2)=O)COCCN(C(C2CNC(=O)N2)=O)C1 68844,N1(C(CC2C(COC)CC2)=O)CCCC(O)(CNC(c2cn(C)nc2OC)=O)C1 68845,O=C(NNc1cccc2c1CCCC2)c1cnc2ccccc2n1 68846,c1(C(N(CCCN(C(c2c(C)sc(O)n2)=O)C)C)=O)cnc(Cl)c(N)c1 68847,N1(C(C(C2CCCC2)OC)=O)CCCC2(C1)CN(C(=O)COC1CCCO1)C2 68848,C12(C(=O)NCC3(CCNC(C(C4CC4)OCC)=O)CC3)CC(C)(C1)OC2C 68849,C12(C(=O)NCC3CN(C(CCc4c[nH]c(=N)[nH]4)=O)C3)CCCC(=O)N1CCC2 68850,C1(CNC(C(C)c2cc[nH]n2)=O)CC2(C1)CN(C(=O)CC1CCCCC1(C)C)C2 68851,N1(C(C=C(CCC)CCC)=O)CC(C)N(C(=O)CC(C)C(F)F)C(C)C1 68852,C1(C(=O)NC2(CO)CCN(C(C34CC(C)C3C4)=O)C2)CC2C(C1)C2(F)F 68853,C1(NC(C(CC)NC(N)=O)=O)CC(OC)CN(C(=O)Cc2c(O)ncnc2O)C1 68854,C1(C(C(=O)N(CC(CC)O)CC)F)CCN(C(=O)CC2(CC)CCC2)C1 68855,Cc1cnc(NC(C2CCN(Cc3ccc(Cl)cn3)CC2O)=O)nc1Cl 68856,c1(OCCN=[N+]=[N-])ccc(C(=O)OC2(CC(N)=O)CCCC2)cc1 68857,c1(C(N2CC(COC)(NC(c3c(C)noc3C)=O)C2)=O)c(O)cc(O)cc1O 68858,CC(C)CC(CC(C)C)C(=O)N1CC2(CCCC2NC(c2ccncc2N)=O)C1 68859,c1(SC)cc(C(=O)N(C)CC2CCCN(C(=O)CC3COCC3O)C2)nn1C 68860,c1(CC(C)C)nncn1CCNC(=O)CC1CCN(C(=O)COCCN(C)C)C1 68861,N1(C2CN(C(C3C=CCC3)=O)C2)CC(NC2(C(=O)C3CC3)CCCCC2)CC1=O 68862,Cc1ccc(C(=O)NCCCOC2CCN(C(=O)C3=CCCO3)CC2)nc1F 68863,N1(C(C(C)(Cl)Cl)=O)CCC(c2cn[nH]c2)(NC(c2ccon2)=O)C1 68864,C(=O)(CCCC(F)(F)F)N1CC(O)(CNC(C23CCCCC2C3(F)F)=O)C1 68865,N1(C(c2cn(CC=C)nn2)=O)CC2CCC1CN2C(=O)C=CC(=O)NC1CC1 68866,N1(C(C(=O)Nc2c(OC)nsc2)=O)C(CO)CCCC1c1ccccc1 68867,c1(C(=O)NCC2N(C(CC(C(C)C)O)=O)CCN(C)C2)ncn2ccccc12 68868,c1(-c2ccc(F)c(C)c2F)cccc2c(C(=O)Nc3cc(Br)ccc3F)c[nH]c12 68869,c1(OC)ncc(C(=O)NC2CCC(NC(c3scc(C)c3Cl)=O)C2)cc1Br 68870,N1(C(C(CC(=O)OC)OC)=O)CC=C(CC(=O)N2CCOCC(C)(C)C2)CC1 68871,N1(C(c2c(C)noc2C)=O)CC2CC(O)C1C2NC(c1ccc(CO)cn1)=O 68872,C=CC(F)(F)C(=O)NC(CNC(=O)C(CC)=CCCC)C1CC1 68873,C1(O)(CC(=O)N(C2(C(=O)NCC3(CC=C)CC3)CC2)C)CCCC1 68874,C1(NC(C=CC=CCC)=O)CC2CC(NC(=O)COC3CCCOC3)CC12 68875,C=CCCC(F)(F)C(=O)N1CCC(C)(NC(=O)COC2CCC(C)CC2)CC1 68876,CC1c2nncn2CCN1C(c1ccc(CNC(=O)CSc2cn[nH]c2)s1)=O 68877,C1(C(N(C)CC2(OC)CCCCC2)=O)CCN(C(=O)C(C)C(O)C(C)C)O1 68878,C=CCCC(CC(C)C)C(=O)N1CCC(C)C(CNC(=O)COCC2(F)CC2)C1 68879,N1(C(c2cc(C(F)(F)F)c[nH]2)=O)CC2(C1)CN(C(C1(N3CCCC3)CC1)=O)C2 68880,C(C(C)(C)CC(=O)NC(C)CCO)NC(Cn1c(C)nc(C)n1)=O 68881,c1(CC)cccc(N(C)C(C2COCC2NC(=O)CCc2ccn(C)c2)=O)c1 68882,N1(CCC)CCCC(C(=O)NC(C)(C)C(C)NC(=O)CC2CC(C(F)F)C2)C1 68883,S(=O)(=O)(c1c[nH]c(=NCCC#N)cc1C)NC(CC)C(C)O 68884,CN1CC2CCCN(C(=O)CCn3cc(CN4CCOCC4)nn3)C2C1 68885,C1(C(=O)NCC(C(C)C)NC(=O)CCCC2CC2)CCC(C(=O)N(C)C)CC1 68886,CC(C)(C)C#CC(=O)N(CC(=O)NCC1OC(=O)CC1(C)C)CCO 68887,c1(SC(c2cccc(C3CC4(CC(C)OC4)C3)c2)=O)ccc2c(c1)CN=S2(C)=O 68888,c1(C(N2CCC(O)(CNC(C3CCCN(C(C)=O)C3)=O)C2)=O)c(C)cc(C)nc1O 68889,C1(C(=O)NCCC2(C(=O)NCCCCCO)CC2)(OC)CCC(C)C1 68890,C12(CNC(=O)CCN3CCCCCC3)CCC(CC1)N2C(=O)Cc1ccon1 68891,c1(CC(=O)NC(CN(C(c2csc(C3CC3)n2)=O)CC)C)ccccc1C 68892,C1(CNC(=O)CCF)CCCC2CN(C(=O)Cc3ccnc(F)c3F)CC12 68893,N1(C(C2CCCN(C(C3CC4CCCC4C3)=O)CC2)=O)CCOCC(C2CC2)C1 68894,c1(CC(C)C)cccc(C(N2CCC(C(C)(C)NC(c3c[nH]c(Br)c3)=O)C2)=O)c1 68895,C(C)(C)(CCCNC(=O)C=CC=C(Cl)Cl)NC(C(CC)n1ccnc1)=O 68896,C1(C)(COC)CCCN(C(=O)CC2(O)CCCN(C(=O)Oc3ccccc3)C2)C1 68897,C1(NC(CCC2C(C)(C)C2)=O)C2CC1N(C(c1ccc(O)cn1)=O)C2 68898,Cc1cc(CN(C)CC2CCCC(c3ccccc3)C2)ccc1F 68899,c1(C(=O)NC(C2CCCN(C(CNC(CC)=O)=O)C2)C)c(F)c(F)cc(F)c1F 68900,C(CC(C)C)(CC(C)C)NC(CCNC(CN(C(COC)=O)C)=O)=O 68901,C(=O)(C(CC(C)C)C(N)=O)NC1N(C(C(CC#C)C2CNC(=O)O2)=O)CCOC1C 68902,N1(C(C(=O)N(CCn2cccn2)CC)=O)CCCC(CN(c2cccn2C)C)C1 68903,N1(C(Cc2cc(C)nn2C)=O)CCC2CN(C(=O)CCS(N)(=O)=O)C(C)C12 68904,c1(OC)ccc2c(c1)C(C)(C)CC2NCC(=O)Nc1nccnc1C 68905,CCCCCCC(C)CC(=O)NC1(C)CN(C(c2c[nH]nc2CC)=O)C1 68906,C1(N(c2cc(C(F)(F)F)ncn2)C(C2(C)CC2)=O)CC12CCNCC2 68907,CC(C)(C)CCC(=O)NC1(c2ccccc2)CCN(C(=O)C2=CCC2)C1 68908,c1(C(=O)NCC2CC(NC(C(C)C3CCCO3)=O)C2)cc(Br)cs1 68909,CC(c1ccc(F)cc1F)=CC(=O)N(CCCCNC(C1CC2CC2C1)=O)C 68910,C#CC1(C(N2CCC(C(C)O)CC2)=O)CCN(C(c2cc(Cl)c[nH]2)=O)C1 68911,C(CN=c1cc(Cl)nc(C(C)C)[nH]1)N(C(c1cccc2nc(O)n(C)c12)=O)CC 68912,c1(C(CC)=O)cccc(NC(N2CCCC(CN(C)C)C2)=O)c1 68913,c1(CC)cccnc1C(N1CCC(CCC(=O)NC2CN(C(N)=O)C2)C1)=O 68914,CCC(C)C(CC(=O)N(C1CCOCC1C)C)NC(c1conc1C)=O 68915,N1(C(C(Cn2cncn2)NC(c2c[nH]nc2Cl)=O)=O)CCC2(CC1)CC2CO 68916,c1(OCCCC)ccccc1NC(=O)NCCC1(O)CCOC1 68917,C1(CNC(=O)C2CC2)CC2(CCN(C(=O)CCOc3ccccc3)C2)CO1 68918,C=CCC(C(=O)NC1(C)CC(NC(C2CC2c2ccc(F)cc2Cl)=O)C1)C(C)C 68919,N1(C(C(C=CCCC)O)=O)CCC(O)(CCNC(c2c[nH]c(C)cc2=O)=O)CC1 68920,C(C(O)C(F)(F)F)N(C1CCC1)C(C1C(CNC(c2cc(C)[nH]c2)=O)C1(C)C)=O 68921,c1(OCC)cc(C(=O)NCC(CNC(=O)CCC(C)OC)CO)ccc1C 68922,CC(CC(=O)NCC(N1CCN(C(=O)CN2CCCCC2)CC1)C)P(C)(C)=O 68923,C(=O)(CCCCCCNC(C(F)(F)F)C1CCCC1)OC(C)(C)C 68924,C1(NC(c2c(CC)nns2)=O)CCCC12CN(C(c1cc(O)c(F)cc1N)=O)C2 68925,C(=O)(C(CNC(c1ccsc1)=O)CC(C)C)NC(c1nc[nH]n1)CC 68926,c1(-c2c(C(=O)NC(C)C)cccc2)ccc(C(N(CC#CC)C)=O)c(F)c1 68927,N1(C(C(C(=O)OCC)C2CC2)=O)CC(n2cc(CC3OCCO3)nn2)C2(CCC2)C1 68928,Cc1nc(O)sc1C(=O)NC(Cn1cccn1)C(=O)NCCC(C)(C)C1CC1 68929,CC1CN(CCO)CC1Cc1ccccc1NCCNS(C)(=O)=O 68930,c1(C(C(=O)NC(C)(C)CC)N(N2CCCC2)CCC#N)ccc([Si](C)(C)C)s1.CC 68931,C1(C(=O)NC(C)CCCNC(=O)C(C)OCC2CC2)C(C(F)(F)F)C1[N+](=O)[O-] 68932,N1(CC(N2CCC(SCc3nn[nH]c3C(=O)O)C2)=O)CCC(C)(C2CC2)C1 68933,C=CC(C)(O)CC(=O)N(C(CNC(=O)C(C)Sc1ccccn1)CC)C 68934,N1(c2nnn(C)n2)CCN(C(c2ccnc(-c3ccco3)c2)=O)CC(O)C1 68935,CCN=C(NCc1ccc(N2CCCC2=O)cc1)N1CCC2CCCOC2C1 68936,C1(N(C(C(=O)Nc2cccc(OC)c2)C2CC=CC2)CC)CC2CCCC(C1)C2 68937,C(C)(C)(CCC(=O)N1CCC(C)(C(=O)NCC2(C)CCC2)C1)N(C)C 68938,C=CC1COCC1NC(C1CSCN1C(=O)C(C(=O)OC)OC)=O 68939,C1(NC(C=Cc2scc(C)n2)=O)CCCC12CCN(C(=O)CCc1cnco1)C2 68940,N1(C(C(=O)NCC2CC2)=O)CCC2CC12C(N1CCN(CCF)CC1)=O 68941,c1(C(C)=O)ccc(C(=O)NCC2CCCN2C(=O)Cc2cc(C)no2)cc1 68942,C1(C(=O)NC2CCN(C(C3COC(=O)O3)=O)CC2)CCc2ncncc2C1 68943,C1(CNC(C(c2cn(CC)nc2)(F)F)=O)CC(C)N(C(=O)CN(C)C(C)C)C1 68944,C1(C(=O)NC2C(C=C)CN(C(=O)CC(=C)Br)C2)CCCCCS1(=O)=O 68945,C1(CC)CC(N=c2cc(C)nc(N3CC=CCC(C)(C)C3)[nH]2)C1 68946,N1(C(c2c(C)cn(C)c2)=O)C2CCC(C2)C1CC(=O)NCCOCC(F)F 68947,c12ccc(Cl)cc1NC2=O.Cn1cc(-c2cn(CO)nn2)c(C2CC2)n1.C(C)(C)C 68948,c1(C(=O)NCCC(=C)CNC(C2OCCC2C)=O)cccc2c(C)[nH]nc12 68949,C1(N(C(=O)CC2(O)CCC2)CC)CCCN(C(c2ccc(Br)nc2C)=O)CC1 68950,C(=O)(C1c2c[nH]nc2CCC1C)NC1(c2c(C)cccn2)CCCCC1 68951,C1(OC)CN(C(C23CC(C2)C3)=O)CCC1NC(c1cc(B(O)O)co1)=O 68952,N1(C(C)=O)CCC(c2ccccc2)(NC(C2(C)CCCC2)=O)C1 68953,CCCC(C(O)C(=O)NCC1C=CCC1)NC(=O)C(CC)(CC)CC 68954,N1(C2(C(=O)NCC3C(NC(C4CC=CCO4)=O)CC3)CC2)CCOC1=O 68955,C12(C(=O)NC3(C)CCN(C(=O)CC4CC(=O)NC4=O)C3)CCC(CF)(C1)OC2 68956,C1(C(C)NC(c2ocnc2C2CC2)=O)CCN(C(=O)CSc2cn[nH]c2)CC1 68957,N1(C(c2ccc(C(C)C)cc2)=O)CCCC(NC(c2cn(C)nn2)=O)C(F)C1 68958,C1(C)(C(=O)NCCNC(c2cc(SC)oc2)=O)CCCCCC1 68959,c1(C(=O)NCCN(C(=O)CC2(O)CCCC2)CCC)ncc(C(C)(C)C)o1 68960,C1(CC(=O)NCCCOC=C)CCN(Cc2cn(C)nn2)C1 68961,CCCCCCC(=O)N(CC(=O)NC(CC)C(=O)OCC)CC1CC1 68962,Cc1ncc(CC(=O)NC2CC2NC(c2sccc2SC(F)F)=O)s1 68963,c1(NC(C)=O)ccc(F)c(C(=O)NC2CC3CNC(C2)C3)c1 68964,C1(CNC(c2c(C)n[nH]c2C)=O)CCN(C(=O)CCSc2nccn2C)CC1C 68965,C1(C(N2C(C)(C)CC(NC(=O)CC3(C(F)F)CC3)C2)=O)CSc2ccccc2O1 68966,C1(NC(COCCOC)=O)CS(=O)(=O)CC1NC(C1(c2ccccc2F)CC1)=O 68967,C1(CC)CCCCCN1C(C(=O)NCCCOC)C1CC1(C)C 68968,c1(C(N2CC(NC(Cc3ccc(C#C)cc3)=O)C(O)C2)=O)ccc2c(c1)CCO2 68969,N1(C(N2CC(C)C2Cc2ccno2)=O)CCCCC(CCC(=O)OC(C)(C)C)C1 68970,C1(COC)CC(C)(C)CN1OC(=O)C(C)CCSC1CCC1 68971,C(CCC(C)CC(=O)N1CC(NC(C2CCOCC2)=O)C2CC2C1)=C(C)C 68972,C1(CNC(c2c(CC)occ2)=O)CN(C(=O)C(O)Cc2ccccc2Cl)CC1C 68973,C1(Cc2cn(CC)nn2)CN(C(=O)NC2(c3ccccc3C)CC2)CCO1 68974,N1(C(c2c(CSC)ccc(F)c2)=O)CC2(CCCC(NC(=O)OC(C)(C)C)O2)C1 68975,C1(NC(C2(C)CC(C)(C)C2)=O)CCN(C(=O)CC2CC(F)(F)C2)CC1O 68976,CSC1=C(C(=O)NC2CN(C(=O)Cc3nonc3C)CC(C)(C)C2)CCCC1 68977,c1(N2CCC(CC=C)(NC(C3NC(=O)CC3C)=O)C2)nc(Cl)nc(C)c1[N+](=O)[O-] 68978,C1(CN(C)C(C2(CO)CC2(F)F)=O)COCCN1C(=O)CCC1CCN(C)CC1 68979,C1(c2c(OC)cccc2)C(NC(c2cccc(C3COC3)c2)=O)CC(=O)N1C 68980,N1(C(c2n(CC)ccc2)=O)CC(NC(=O)CSc2nncn2C)C(C(F)(F)F)C1 68981,c1(CCCC(=O)NCC2(O)CCN(C(=O)C3CC3)CC2)c[nH]c2ccccc12 68982,C1(NC(c2cn3ccnc3s2)=O)CN(C(C2CC=CC2)=O)C2(CCCOC2)C1 68983,C(=O)(C=C1SCC(=O)N1C)NC12CCCN(C(CC3C(C)CCCC3)=O)CC1C2 68984,C(=O)(C(C)(C)CC(F)F)N(C(CNC(CCCC(=O)NCCC)=O)C1CC1)C 68985,C1(NC(C(C)(C)Cc2cccc(Cl)c2)=O)CC2CC(C1)N(C(=O)CCC1CC1)C2 68986,c1(CC)ccc(NCC(=O)N(C2(CC)CCOC2)CC)cc1 68987,c1(C(=O)NC2CCCC(NC(CCN(C)CCO)=O)C2)cc(Cl)c(F)cc1F 68988,N1(CC)CCOC(C(=O)NCC#CCNC(=O)CCc2cncc(OC)c2)C1 68989,C1(O)(C(C)NC(c2cncnc2)=O)CCN(C(c2ccc([N+](=O)[O-])[nH]2)=O)CC1 68990,Cc1cc(=NC2CC(C)N(C(=O)CCOCC(F)F)C2)[nH]c(C(F)(F)F)n1 68991,CC1(C)CN(C(C23CC2CCN3C(c2n[nH]c(=N)[nH]2)=O)=O)CCC1O 68992,C1(CC(=O)NCC2C=CCC2)CCCC1NC(c1cc(CO)on1)=O 68993,CN(C)NC(=O)CCC(=O)N1CC=CC(NC(=O)CC2C=CS(=O)(=O)C2)C1 68994,c1(OCC(=O)NC2CC(NC(C(C)Cc3cccnc3)=O)C2)ccc(Cl)c(F)c1 68995,c1(C(N2C(CCC(N3CCC(=O)NCC3)=O)CCC2)=O)ccc2c(c1)CCCO2 68996,C(C(C(C)C(C)C)NC(C1(C(F)(F)F)CC(F)(F)C1)=O)NC(CCOCC#C)=O 68997,CCC(C)CCC(=O)NCC(C)C(=O)NC1(CC)CCOCC1 68998,c1(NC(CC2CC(C)C(C)CC2)=O)cccc2c1C1CCC2CC1 68999,C(=O)(C1CCc2ccccc21)N1CCCC(C)(CNC(CCC(C)(C)O)=O)C1 69000,C12(CNC(c3c(COC)scc3)=O)CCCC1CN(C(=O)CCC(C)(C)F)C2 69001,Cc1cccnc1C(=O)NC(c1ccccc1F)CNC(=O)C=Cc1cocn1 69002,N1(C(CC2OCCN(C(C3C(C)C3C)=O)C2)=O)CC2CCC1C(CO)C2 69003,C(=O)(C(CC(C)C)C(N)=O)NCCCN(C(C(CC)N(C)C)=O)CCO 69004,C1(C(N2C3(CNC(CC4CCN(C(C)=O)C4)=O)CC(C2)C3)=O)CCOCC1(C)C 69005,N1(C(C(CC)C)=O)CCC2(CCCN(C(=O)Cc3ccc(OC)c(OC)c3)C2)C1 69006,Cc1nccc(C(=O)N(C2CCN(C(C3CCCC34CCC4)=O)C2)C)c1N 69007,c1(CN2CCC(C(N3CC4(CCC4)C3)=O)C2)c(O)cccc1F 69008,N#CCCCCC(=O)N1CC2C(NC(=O)CCc3ccccc3Br)C2C1 69009,C#CCC(CC(F)F)NC(c1cn(CCNC(=O)OC(C)(C)C)nn1)=O 69010,C1(CNC(C2N(C)C(=O)CC2)=O)CCCN(C(=O)C(F)(F)c2cncs2)CC1 69011,c1(C(=O)NCC2=CCCN(C(C3(NC(C)=O)CCC3)=O)C2)cn2ncccc2n1 69012,c1(C(=O)NC2C=CC(CC(=O)NC3(C)CCCC3O)C2)cc(C#N)ccc1N 69013,CON=Cc1ccc(C(=O)NCC(C)NC(=O)CC2CCCC23CC3)cc1 69014,c1(C(N2CCN(C(CCC#CC)=O)C(CCO)C2)=O)ccc(C)c(S(N)(=O)=O)c1 69015,c1(C(=O)NCC2CN(C(CCCOCC=C)=O)C2)ccc(=O)n(C(C)C(C)O)c1 69016,Cc1[nH]c2ccc(F)cc2c1C(=O)NC(c1cn(C2COCCC2O)nn1)C 69017,c1(C(N2CCC(O)(CNC(Cc3nn(C)c(Cl)c3)=O)C2)=O)cc(N)cnc1Cl 69018,CC1CCCc2nc(C(=O)NC(CNC(=O)CCNC(N)=O)CC(F)(F)F)cn21 69019,C1(C(=O)NCC2(C)CCN(C(=O)C=CC3CCCO3)C2)CC(C2CCCC2)C1 69020,N1(C(C2CC(C(F)(F)F)(OC)C2)=O)CCC2(NC(c3cccc(=O)o3)=O)CC2C1 69021,C1(C(=O)NC(CC)CN(C(=O)CCC2(C)CC2)C)CCN(c2ncccn2)C1 69022,C1(CC(N2CCC(N(C(=O)CCOCC)CC)C2)=O)CCc2ccccc2C1=O 69023,C(=O)(CCCCCC#N)N1C(C)CC(CCNC(=O)CCC(N)=O)CC1 69024,C(=O)(CCCN=[N+]=[N-])NC1(C)CCN(C(c2csc(-c3ncc[nH]3)n2)=O)C1 69025,Cc1cc(NCC2CC(C)(C)CCC2NC(=O)CCC2CCC2)ccc1[N+](=O)[O-] 69026,C(C(=O)NCCC(C)C(F)(F)F)(C(C)(C)C)NC(C(OCC)OCC)=O 69027,c1(C(=O)NCC(NOCC)=O)cccnc1CNC(=O)Cc1cccn1C 69028,Cc1cc2ncc(C(N3CCC(C)C(NC(c4nocc4Cl)=O)C3)=O)cn2n1 69029,C(=O)(N1CC(O)CCO1)C1(C)CC(NC(C2CC(=C3CCC3)C2)=O)C1 69030,c1(C(=O)NCCC2CCCN(C(c3ccn(CC#N)n3)=O)C2)ccc(Cl)cc1O 69031,C(N=c1ccc([N+](=O)[O-])c(O)[nH]1)C1(NC(c2c(CC)nc[nH]2)=O)CCCCC1C 69032,c1(C(N2CC(CCOC)N(C(c3cc[nH]c3)=O)CC2)=O)cc(C)cc2ccoc12 69033,N#Cc1ccc(C(=O)NCCCCCNC(c2cnc(Br)s2)=O)cc1O 69034,c1(OCC(=O)NC(CCCC)CNC(=O)CC2COC(=O)N2)cc(Cl)ccc1C 69035,C(=O)(C(Cc1ccccc1)C(F)(F)F)NC1CN(C(C=C(C)C(F)F)=O)CC1(C)C 69036,c1(CNC(NC(C2CCC2)C)=NCC23CCCCC2C3)ccc2c(c1)OCC2 69037,CC1CC=C(C(=O)NCc2ncccc2O)CC1 69038,c1(NC(C)=O)ccc(F)c(C(=O)NCC(CC)NC(=O)CCc2cnn[nH]2)c1 69039,c1(C(=O)NC(CC)CNC(=O)CC2CCCC3(CC3)C2)c(F)ccc(CC)c1F 69040,C(C(C(C)C)NC(=O)CCN)NC(C1CCC1)=O.C(COC)SC 69041,C1(C(=O)NC(CNC(c2c(OC)cc(C)cn2)=O)C(C)C)CCCC1S(C)(=O)=O 69042,c1(C(=O)NC2CN(C(C3C(C)CCC3)=O)C2)nn(C)cc1N 69043,N1(C(CCSCC)=O)CCN(C(c2cnn(CC)c2)=O)CC1COC 69044,C1(NC(CC)=O)CCC2CN(C(C3(c4cccc(Br)c4)CC3)=O)CCC2C1 69045,c1(C(C)(C)C)cc(Br)cc(Br)c1C(=O)NCc1n[nH]cc1C(=O)O 69046,C=CCCCC(C(=O)N1CC(CC(C)(C)C)C1)NC(=O)CN1CCN(C)CC1 69047,Cc1ccc(SCC(=O)NC2CCN(C(C3(CCF)CC3)=O)C2C)cc1C 69048,c1(C(=O)NC(C(C)C)CNC(c2cncc(C(F)F)c2)=O)cc2ncccc2o1 69049,C1(C(=O)NCC(CC)(C)C(N)=O)CN(C(c2cccc(O)n2)=O)CC(C)(C)C1 69050,N1(CC)CCOC(C(=O)NCCC2(OC)CN(C(=O)C(CCSC)OCC)C2)C1 69051,S(=O)(=O)(c1cnc(N2CC(CCO)C2)c(Cl)c1)NC1C(C(C)C)C2CCC1C2 69052,c1(C(C)C)c(C(N2CCCC(NC(=O)C=CCF)C2)=O)cnn1CCO 69053,CC1(C)CCN(C(=O)CC2CCSC2)C1CC(=O)NC1(C)CC2(CC2)C1 69054,Cc1cc(C)c(C(=O)NCC2CC(NC(C3(CF)CC3)=O)C2)c(Cl)n1 69055,C1(NC(C(c2ccc(OC)cc2)=O)=O)CC2CC1CN(C(C1CC1C)=O)C2 69056,N1(C(C(CCOC)C)=O)CCC(CNC(=O)Cc2nc[nH]n2)(OC)CC1 69057,Cc1nc(C)c(C(=O)NC(C2CN(C(c3cocc3C)=O)C2)C)[nH]1 69058,N1(C(CC2COCC(C)(C)O2)=O)CC2CN(C(=O)CSC3CC3)CC2(C)C1 69059,c1(C(N2C(C)(CC(N3CC(F)(CO)C3)=O)CC2)=O)ccc(=N)[nH]c1 69060,c1(Cn2c(-c3cncc(CC)c3)nc(CC(C)C)n2)cnc(O)nc1O 69061,C(C(CC1CC1)C(=O)NCC1CC=CC1)NC(CC1N(C)CCC1)=O 69062,CC1(CC(F)(F)F)CN(C(=O)C(C2CCCC2)NC(C2CC2C(F)F)=O)C1 69063,C1(N(C(C(CCNC(c2c(CC)cc[nH]2)=O)O)=O)C)CC2CCC1CC2 69064,Cc1ccc(Cl)c(C(=O)NC2(C)CC(NC(=O)COc3ccc(F)cc3O)C2)c1 69065,c1(CC)nc2sc(C)cn2c1C(=O)NCC1CC2(CCNC2)CO1 69066,N1(C(C(n2cc(-c3ccc4c(c3)OCO4)nn2)C)=O)CC(CO)Oc2ccccc21 69067,N#Cc1cccc(F)c1CC(N1CC2CC(NC(=O)C#CC3CCC3)C1C2)=O 69068,C1(C(N2CCC(C(C)NC(c3cnc(C(F)(F)F)s3)=O)C2)=O)CCS(=O)(=O)N1 69069,C1(CC)CN(C(=O)CCOCC2CC2)CCC1NC(=O)CC1CCC=CCC1 69070,Cc1ccc(C)c(NC(=O)C(CO)NC(=O)Cc2cc(C)[nH]n2)c1 69071,N1(C(C(=O)NC2CN(c3cccnn3)C2)=O)CCc2nc(O)cc(O)c2C1 69072,N1(C(C2(C)CCCO2)=O)CC2(CC(CC(N3CCCC3CF)=O)C2)C1 69073,c1(C(=O)NC(CCCCNC(c2c(C)ccs2)=O)C)cc(F)c(F)c(F)c1F 69074,C1(NC(C2(C)CC2(F)Cl)=O)CCC(CNC(=O)CSCc2ccc(O)cc2)CC1 69075,C(C)(C)(C(=O)NC1CC(CCNC(C2CSCN2C(=O)C(C)(C)C)=O)C1)N(C)C 69076,C(C)(C(=O)N1CC(OC2CCOCC2)C1)(C(C)C)NC 69077,c1(C(C)(C)C)nocc1C(=O)NC1CCCC1NC(=O)C(C1CCC1)C1CCC1 69078,c1(OCC)ccc(Cl)cc1C(N1CC(OCCNC(c2cc(N)ccn2)=O)C1)=O 69079,Cc1nc2ccccc2nc1NC(c1ccc(CN2CCOC(C)(C)C2)cc1)=O 69080,C(=O)(C(C)CC(F)(F)F)N(C(C1CN(C(c2ccnc(C3CC3)n2)=O)C1)C)C1CC1 69081,c1(C(=O)NCC(C)N(C)C(c2nnsc2C(F)F)=O)cnc(O)n(C)c1=O 69082,N1(C(=O)OC(C)(C)C)CC(N=c2ccn3ccnc3[nH]2)CC2(CCC2)C1 69083,C1(c2nnnn2CCOC)(NCCCC(C)(C)C)CCCC(C(F)(F)F)C1 69084,c1(C(=O)NC2C(CNC(c3ncc(NC)nc3)=O)C2)ccc(F)c(Cl)c1F 69085,C1(C(N2CCCC(CC(=O)O)C2)=O)CCCC(NC(COC(C)(C)C)=O)C1 69086,C(=O)(CCC(C)(C)C#N)N(c1ccc(C)cc1)CC(=O)NC(COC)C 69087,C(CC1=CCOCC1)NC(=O)CC(O)CNC(=O)CN1CCCCC1 69088,Cc1ccn2cc(C(=O)NC3CN(C(C4CCC(N=[N+]=[N-])C4)=O)CC3(C)C)nc2c1 69089,N1(C(CC2(C)CC2)=O)CC2CCCC(C1)N2C(=O)CC1CCCCCC1(F)F 69090,CC1CS(=O)(=O)CC(C)N1C(C1SCCCS1)=O 69091,C1(C(N2CCN(C3CC(N)C3)CC2)=O)CCC2(CCC2)C1O.c1(O)ncccc1S 69092,C(=O)(C1=CCOCC1)NCC1CC(NC(=O)C=Cc2cscn2)CC1O 69093,c1(C(N2CCCC(OC3CC3)C2)C(=O)NC2CCC2)ncccc1F 69094,C1(CC)CN(c2nnc(CSCCO)n2CC(=O)NC)CC(C)O1 69095,c1(C(=O)NC2CN(C(c3ccc(F)c(F)c3Cl)=O)C2)cc(Cl)c2cn[nH]c2c1 69096,c1(OCCNC(c2c(OC)cccn2)=O)c(F)cccc1Cl 69097,c1(CC(C)C)ccccc1C(=O)NC(C)(C)CNC(=O)CCN1CCNC(=O)C1 69098,c1(C(=O)NC2CCCN(Cc3ccc(O)cc3)C2)csc2ccc(Cl)cc12 69099,N(C(=NCCn1cccn1)NCc1ncccc1O)CC1N(CC)CCC1 69100,c1(OC(C)C)c(F)cc(-c2nc(NC(=O)CNc3nccs3)cs2)cc1F 69101,c1(C(=O)NCCN(C(N)=O)CC)cc(F)c(F)cc1NC(=O)Cc1cnns1 69102,N1(C(=O)NCCCc2c(C)cccn2)CCN2CCOCC2C1 69103,C(=O)(C(=O)CC(C)CC)NC(C(=O)N(C1CC(=C)C1)C)c1cccs1 69104,Cn1c(C(N2CCC(O)(CNC(=O)CC3CCCOC3)CC2)=O)cc2sccc12 69105,N1(C(C=CC=CCC)=O)CCC2OCCN(C(C3CCC(F)(F)CC3)=O)C2C1 69106,c1(C(=O)NC2CCN(C(C(C)NC(=O)C3CC3)=O)C2)ccnc2ccc(Cl)cc12 69107,C(=O)(C(CC(C)C)C(N)=O)NC(C1N(C(C(CCC(C)C)F)=O)CCC1)C 69108,N(C1CCCc2n[nH]cc21)C(C(N(C(=O)CCn1cnc(=N)[nH]1)C)C1CC1)=O 69109,c1(CNC2CN(C(C3=CC=NC(=O)C3)=O)CC23CC3)cccc2nccnc12 69110,N1(C(c2ccc(Cl)s2)=O)CC(CNC(C23COCC2C3)=O)C2(CCC2)C1 69111,Cc1nc(-c2cn(CC(C3CN(C(=O)CCc4nccs4)C3)F)nn2)sc1C 69112,C1(NC(c2n[nH]c(=N)s2)=O)CCCC2CN(C(C3CCCC(F)(F)CC3)=O)CC12 69113,O=C(N1CC(n2cc(C3CCCCO3)nn2)CO1)c1cncc(C2CC2)c1 69114,Cc1nc(O)ccc1C(N1CCC(C(=O)NCCc2c(C)n[nH]c2C)C1)=O 69115,c1(CC=C)ccccc1C(=O)NCCCCCNC(=O)C(COC)N(C)C 69116,C=CCC(CNC(=O)CN(C)C(N)=O)C(=O)NCc1nnn(C)c1C 69117,C1(C(C(=O)NC2(c3ncc[nH]3)CC2)NC(c2ccc(CO)s2)=O)CCCCC1 69118,Cc1cccc(C)c1COC(c1ccnc(-n2cccn2)c1)=O 69119,C1(NC(c2n(C)c(S)nn2)=O)CCCC(C(N2CCCC2(C)CO)=O)CC1 69120,C1(C(N2CC(NC(=O)C(C)(C)C#N)CC(C)(C)C2)=O)Cc2cc(Br)ccc2O1 69121,N1(C(CSC)=O)CC(NC(=O)CSc2cccc(Br)c2)CCC1C 69122,c1(CC)ccc(N(CCO)C(c2c[nH]nc2CNC(C2CC(C)(O)C2)=O)=O)cc1 69123,CC(C)(C)C(C(=O)NCCCC1OCCO1)n1cc(Cc2ccc(F)cc2)nn1 69124,N1(C(c2c(C)ccnc2C)=O)CC2CCC(C1)C(NC(c1ccoc1C)=O)C2 69125,N1(C(=O)CC2CCCCC2NC(C2(CO)CCCCO2)=O)CC2(CCOCC2)C1 69126,CCC(CC)C(=O)NC(C)(CNC(c1cccc(C(=O)N(C)C)c1)=O)C(C)C 69127,C1(CC)CN(C)CCCN1C(C1CC1C1CN(C(C2CC3(CCO2)CC3)=O)C1)=O 69128,C1(N(C(C2CCCOC2)C(=O)NC)C)CCC(OC)CC1 69129,C(C)(C)(CCCC(=O)NC(C1CCCC1O)C)NC(c1c(C)cc(O)nc1)=O 69130,N1(C(CC2(COC)CC2)=O)CCC(NC(=O)CCCN2CCCC2)C1(C)C.C1CC1 69131,C1(NC(c2cnn(C(C)C)n2)=O)CC(C(=O)NCc2snnc2C)C12CCC2 69132,N1(Cc2c(C(=O)OCC)n[nH]c2)CC2CN(C(c3cc(B(O)O)co3)=O)CC12 69133,Cc1ccccc1C(C)C(=O)NCC(C)CN(C(=O)C(C1CCC1)C1CCC1)C 69134,Cc1cc(-n2cccn2)nc(=NCC2C(C)CCCN2C(=O)C(C)CN(C)C)[nH]1 69135,c1(C(N(CC(C)NC(=O)CCCC#N)C)=O)ccc(-n2cccn2)cc1 69136,c1(N2CC(C)=C(C)C2)ccc(S(=O)(=O)NCC2Cc3ccccc3CO2)cc1Cl 69137,c1(C(N(CCC(C)NC(=O)CC2CCN(C)C2=O)C)=O)cc(N)c(F)c(F)c1F 69138,c1(OC)cc(OC)c(C(=O)N(c2ccccc2)C)cc1N.C12C=CC(C1)C(=O)N2 69139,Cc1nc(-c2ccc(C(=O)Nc3ccccc3)cc2)ccc1C(=O)NC1COC1 69140,N1(c2n(CC=C)c(-c3nccn3C)nn2)CC(C(N)=O)OC(C)C1 69141,C(C)(C)(CC(=O)NC(CNC(=O)Cc1ccno1)CC(C)C)OC 69142,C12=C(Cl)N=CNC1=NCC1(F)CC(C1)NC2=O.c1(C(C)=O)coc(SC)c1 69143,c1(C(=O)NC2(C)CCN(C(c3ccc(N)cc3Cl)=O)C2)ccn2nnnc2c1 69144,C#CC(C(C)OC)NC(C1(C(C)NC(C2CC(CC)C2)=O)CC1)=O 69145,CC(CCCC(F)(F)F)(c1nnnn1Cc1ccccc1)NCc1cccnc1 69146,Cc1nn(CC(=O)NC(C)C(C)NC(=O)C(CO)c2ccccc2)cc1Cl 69147,C1(C(N2CCC(O)(C(F)(F)F)C2)=O)CN2CCN1CC2 69148,c1(C(N2CC3CC(C2)N(C(=O)Cc2ccncc2)C3)=O)ccc2nc(Br)sc2c1 69149,N1(C(C23OCC(C(C)C)(C2)C3)=O)CCC(C)(NC(=O)CCS(N)(=O)=O)CC1 69150,Cc1cc(C)c(C(=O)NCC2C(C)CCN2C(=O)CCc2csc(=N)[nH]2)o1 69151,c1(C(N2CC(SC)C(NC(=O)C=CSC)C2)=O)ccn(CC(F)(F)F)c(=O)c1 69152,C1(O)(CN(C)C(c2ccoc2)=O)CCN(C(C2CCC(c3ccccc3)C2)=O)C1 69153,C(C)(C(CCc1cn[nH]c1)NC(c1[nH]c(O)nc1C)=O)NC(CSC)=O 69154,C(N=c1[nH]c(N(CC(C)C)C)nc2c1SCC2)C1CCN(S(C(C)C#N)(=O)=O)C1 69155,N1(C(C2C3CC(=O)CC32)=O)CC2C=CC1C(C(=O)NCC1(O)CCOC1)C2 69156,N1(C(C2(CC)C=CCC2)=O)CCC(CN(C(=O)COC2(C)CCC2)C2CC2)CC1 69157,C(=O)(C#CC1CCOCC1)N(C)CC1N(C(C(C)Cn2ccnc2)=O)CCC1 69158,C1(C(N2CCC(C#N)C2)=O)CN(C(C2(C(F)(F)F)CC2)=O)CC12CC2 69159,C(C)(CCC(=O)NCCCNC(=O)C(C)(C)N1CCOCC1)OC 69160,C1(C(=O)NC(C#C)CC2CCC2)CC2CC2N1C(=O)CNC=O 69161,N1(C(C(CC)OC2CC2)=O)CCN(C)CC1CNC(=O)C=CC(=O)OC(C)(C)C 69162,n1(CC)nc2c(c1C(N1CCC(C(C)NC(=O)C(O)C(C)C)CC1)=O)CCCC2 69163,N1(C(C=CC)=O)CCC(NC(=O)C=Cc2cc[nH]n2)C(C)C1 69164,CN1CC(F)CC1C(N1CCC(NC(=O)CCCc2cncs2)C1)=O 69165,C1(CC(=O)NC2CN(C(c3cc(F)c[nH]3)=O)CC2CO)CCCS1(=O)=O 69166,C1(C)(CNC(CC=C=C)=O)CCN(C(=O)C(O)C(C)c2ccc(C)cc2)CC1 69167,CC(C)C(C)(O)C(=O)NCC1CC(NC(c2coc(Br)c2)=O)CC1O 69168,C1(NCCCC(=O)NCC(CO)OC)CCN(C(=O)OC(C)(C)C)C1C(C)C 69169,C(=O)(C(C)(O)C(F)(F)F)NCC(C)(C)NC(=O)C(O)CC1CCOCC1 69170,c1(C(N2CCC(NC(C(COC)C)=O)C23CC3)=O)ccc2cccc(C)c2n1 69171,CCS(=O)CC(=O)NCCC1(C)CN(C(=O)COCCN(C)C)C1 69172,C1(CS(C)(=O)=O)CSC(NC(=O)CCC2CCCO2)=N1 69173,c1(ONC(C23N(C(c4ccccc4)=O)CC(C)(C2)C3)=O)cccc2c1OCO2 69174,c1(NC(C2CC(O)(CNC(C3(C=C)CCOCC3)=O)C2)=O)ccc(F)c(C)c1F 69175,C12(c3c(C(=O)NCC(=O)N4CC=CCO4)cccc3)CC3CC(CC(C3)C1)C2 69176,C1(CNC(CSCC#C)=O)(OC)CCN(C(c2ccc(NC(C)=O)s2)=O)CC1 69177,C1(CNC(C(c2cccnc2)OC)=O)CC(C)(C)CN1C(c1ccc(F)nc1)=O 69178,c1(C(=O)NCC2C(NC(CC(CC)SC)=O)CC2)cccc(F)c1NC 69179,c1(CC)nc2sc(C)cn2c1C(=O)NC1CCC1NC(c1ccoc1CC)=O 69180,C1(NC(CC(C)(O)c2ccccc2)=O)CC2(C1)CC2N=c1[nH]nc(C#N)s1 69181,c1(CNC(CC(COC)(C)C)=O)nc2c(s1)CN(C(c1ccnnc1)=O)CC2 69182,c1(CCC(=O)NC2CN(C(C3C(OCC)C3C)=O)C2)ncccn1 69183,c1(NC(=O)CC2CCC(NC(c3nc[nH]n3)=O)CC2)cc(Br)nc(Br)c1 69184,N1(C(C(c2ccc(C)o2)C)=O)CC2(C1)CN(C(C13CC1COC3(C)C)=O)C2 69185,N#Cc1ccccc1C(=O)NCCc1cc(C(N2CCC(F)(F)C2)=O)no1 69186,C(=O)(C(C)(O)C(F)(F)F)NCC(C)(CO)NC(c1ccc(-n2cncn2)cc1)=O 69187,C(=O)(CCC1CCc2ccccc21)NC1(C)CCCN(C(C2(F)CCOC2)=O)C1 69188,C(=O)(CC(C)C(C)C)NC1C(CNC(C(c2ccc(C)s2)C)=O)CCCC1 69189,N1(C(C2OCCN(C)C2)=O)CC2CC1CN2C(=O)COCc1ccccc1 69190,c1(C(=O)NC2CC(CNC(C3C(C(=O)OCC)C3)=O)C2)cccnc1S 69191,C(=O)(C(CC)C(C)C)NC(CC=C)CNC(c1cnn(C)c1COC)=O 69192,c1(CC)ccc(C(=O)NC2COCCC2NC(=O)Cc2ccc(C)cc2)c(O)c1 69193,c1(C(=O)NCC(CCNC(c2nnn(C)c2N)=O)O)ncc(F)cc1F 69194,C12(C(N3CCC(C)(C)C3)=O)CCC(CN(C(=O)CC3CCCO3)C1)C2 69195,N1(CCC(=O)NCC2(F)CN(C(C3C(OC)C3)=O)C2)CCSC(C)(C)C1 69196,Cc1ccc(CC(=O)NC2CCC(NC(C3CCC4C3C4(F)F)=O)CC2)cc1Cl 69197,N1(C(Cc2nnc(C)o2)=O)CC2CC1CN2C(c1ccnc(O)c1)=O 69198,c1(OC)cnnc(C(=O)N(CCCOCCNC(C2(N=[N+]=[N-])CC2)=O)C)c1 69199,C1(CNC(c2scc(OC)c2)=O)CCC2CN(C(=O)CCc3cc(C)[nH]n3)CC12 69200,c1(C(=O)NC(C)(C)CNC(C2CCCCS2(=O)=O)=O)cc(Cl)cc2ccncc12 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69271,C(C)(CCN=c1[nH]c(Cl)ncc1C)NC(C(c1cccc(OC)c1)C)=O 69272,N1(C(C(C)NC(CC)=O)=O)CC=CCC1C(N1CCN(C(C)C)CC1)=O 69273,c1(NC(C(=O)N(C(c2ccccn2)C)CCO)=O)ccc(C2CCC(=O)N2)cc1 69274,C(=O)(C(O)C(C)(C)C)N(CCN(C(c1sc(CCC)c(CC)c1)=O)C(C)C)C 69275,c1(CC(=O)NCC(CO)NC(CCc2ncc(C)[nH]2)=O)ccnc(Cl)c1F 69276,C12CCN(C1)C2=O.c1(C(C)(C2CC2)Nc2nccs2)nnnn1CCF 69277,C1(NC(C(COCC)CC)=O)CCN(C(=O)CCCN(C)C)CC1(C)C 69278,N1(C(C2C(C)(CC)C2)=O)CCOC2(C1)CN(C(C1(SC)CC1)=O)C2 69279,N1(CCC#C)CCC(C(N2CCN(C(=O)C3CC3)CC2)C(=O)NC)CC1 69280,C(=O)(C1=NOC2(CCOC2)C1)NCC(CNC(CC1CC(NC(C)=O)C1)=O)OC 69281,C1(C(=O)NC(c2ncccn2)(C)C)CCC2(CC2)N1C(=O)CCC1CCC1 69282,C1(NC(C(C(CC)C)OC)=O)CCCC12CN(C(c1ccsc1SC)=O)C2 69283,CC(C)C(C)C(=O)N1CC2CC2(NC(C2(c3ccccc3F)CCC2)=O)C1 69284,CCC(C)(C)C(=O)NCC1CC(NCC2(CC(=O)OC)CC2)C1 69285,C(=O)(C#CC1CCC1)NCC(C)CN(C)C(C1C2CCCC12)=O 69286,CC1CC2(CCN(c3nnc(-c4ccon4)s3)CC2)CN1C(C1CCC2CC12)=O 69287,n1(CC)nncc1CN1CCC(N(C)C(=O)O)C1.C(C)(C)(C)OCC 69288,c1(C(N2CCN(CC(N)=O)CC2)C(=O)NCCCSCC)ccc(C)c(F)c1 69289,C1(C(N2CCCC(F)(CNC(C3SCCCS3)=O)C2)=O)CCC2(CCCC2)C1 69290,N1(CCCc2cn(C=C)nc2)CCCCC(C)C1.c12cn(nn1)C(C)C(=O)N2 69291,C#CC1(OCC(=O)NCCNC(=O)C(c2cnn(C)c2)O)COC1 69292,C1(N(C)C(C23CCC2C3)=O)CC2CCC(C1)N2C(=O)Cc1cccc(Cl)c1 69293,CCCCCC(O)CC(=O)N(C(CC(F)F)C(=O)N(CC1=CCSC1)C)C 69294,c1(NCC2CC=C(C)CC2)ccc(S(=O)(=O)N2CCC(C)(C)C(C)C2)c(Br)c1 69295,C1(CC=C)(NC(=O)CCCc2cccs2)CCN(C(=O)CCOCCOC)C1 69296,N1(C(CC(=C)C)=O)CCC2(CC1)CC(NC(C1NC(=O)CC1C(F)(F)F)=O)C2 69297,C(c1cnn(-c2ccccc2)c1)=CC(=O)NCC(CC)NC(=O)COCC(F)F 69298,C1(NC(c2c(C)nco2)=O)CN(C(=O)CC(N2CCCCC2=O)C)CC1C(F)F 69299,c1(-c2c(-c3n(Cc4c(N)sc5c4CCC5)ccn3)cccn2)cc2c(cc1O)OCO2 69300,N1(C(C(C=C=C)C)=O)CC(C(=O)N)C(C)(C)C1.C(C)COC 69301,Cc1ccc(C(N2CC3CC3(NC(=O)OC(C)(C)C)C2)=O)c(N)c1 69302,CC(C)CC(C)(O)C(=O)N1CCCC(O)(CNC(=O)CC(F)F)C1 69303,CC1CN(C(c2nc(Br)c[nH]2)=O)CCC1N(C(=O)Cc1cccc(F)c1)C 69304,N1(C(C(C(C)C)O)=O)CC2CCN(C(c3cc(C(F)(F)F)ccc3N)=O)C2C1 69305,N1(CCC)CCCN(C(=O)Nc2ccc(F)cc2C(F)(F)F)CC1 69306,CCCCC(O)CC(=O)NCC(c1cccc(C)c1)NC(=O)CCCC#N 69307,C#CCC(C)(CC)C(=O)NC(CC(=O)N(C(C)COC)CC)C(F)(F)F 69308,C1(C(N(c2ccccc2)CC)=O)CCCN1NC(=O)CCc1cccn1C 69309,c1(CC)ccc(S(=O)(=O)N2CC(F)CC2C(=O)Nc2cc(F)c(F)cc2Br)cc1 69310,CC1(CNC(c2ccc(F)c(O)c2)=O)CCN(C(C2SCCCS2)=O)CC1 69311,c1(-n2cc(C(=O)NCC(CNC(CN(C)CC)=O)C)nn2)ccccc1C 69312,c1(NCCc2cc(C(=O)OC)no2)nccc(=NCC2CCCO2)[nH]1 69313,N1(C(C(C)(C)OCC)=O)CC2CCOCC2(NC(c2nc(C(C)C)oc2C)=O)C1 69314,c1(C(N2C(C(=O)NC(c3ccsc3)C)CC(O)C2)=O)cccc([N+](=O)[O-])c1 69315,C12CN(CC1O)C(=O)CCNC2=O.C1(C(C)C)CC1NC(=O)OCC(C)(C)C 69316,C1(NC(C2(F)C(C)C2)=O)CC2(C1)CN(C(c1cc(F)ccc1OC(C)C)=O)C2 69317,c1(C(N2C3CC(CNC(CC(C)SC)=O)C2CC3)=O)coc2c(F)cc(Cl)cc12 69318,N1(C(C(CC)SC)=O)CCCC(C2CCN(C(=O)C(F)=CC3CC3)CC2)CC1 69319,CC(C)(CO)C(=O)NCCCN(C(=O)CCc1cc[nH]n1)CC1CCCC1 69320,N1(C(COC(C)C)=O)CC=CC(NC(c2ccc(OCc3cscn3)cc2)=O)C1 69321,O=C(CC(C(F)(F)F)NC(C1CC1(F)Cl)=O)NCCCOCC(F)F 69322,C1(C(N2CCC(c3ncco3)C2)C(=O)NCC(C)C)CCC(CCC#N)CC1 69323,C1(C(=O)NC(C(=O)N2CCC(C(=O)OC)C2)CCC2CC2)CCCC(=O)CC1 69324,CCCCC(CNC(=O)CCN(S(C)(=O)=O)C)NC(c1cc(COC)cn1C)=O 69325,C=C(Cl)C(C)(C)C(=O)NCC1(C(C)NC(=O)CN2CCNC(=O)C2)CC1 69326,CC(C)S(=O)(=O)CC(=O)N1CCC2CC1CN2C(=O)CSc1ccc(F)cc1 69327,N1(C(c2[nH]ccc2C2CC2)=O)CCN(C(C2CCCCC2)=O)C(C(F)(F)F)C1 69328,N1(OCC)CCC(NC(=O)C(C)(C)C2CCN(C(=O)CCCN(C)C(C)=O)C2)C1 69329,N1(C(C(C)OC(C)(C)C)=O)CCC(NC(=O)COc2ccccn2)C12CCC2 69330,c1(CC(=O)NCC2C(CNC(=O)CCCC3CCCC3)C2)cn2c(n1)CCCC2 69331,c1(C(C)(C)C)ncc(C(=O)NCC2CC2NC(=O)CC(C)(C)C2CC2)cn1 69332,c1(CCCC(=O)N(C(C)CCNC(=O)C(F)(F)CO)C)nc2ccccc2s1 69333,CC1CN(C(c2cc(C3CCC3)no2)=O)CCC1CNC(=O)CCNC(N)=O 69334,C1(C)(C(N2CCC(C)(CNC(c3c(C)n(C(C)C)nc3)=O)C2)=O)CCCN(C)C1 69335,C1(NC(C2N(C(C)=O)CCC2)=O)CC2(CCCN(C(c3cnc(C)s3)=O)C2)C1 69336,C1(C(=O)NCC(CNC(C=CC=CCC)=O)CO)CC(C(C)C)=NO1 69337,C1(C(C)C)CN(C(c2cc(F)cc(F)c2)=O)CCN1C(=O)C1=CCCO1 69338,c1(NC(C)=O)cc(F)ccc1C(=O)NCC1(NC(c2[nH]cnc2C)=O)CCOC1 69339,CC(C)(CNC(C1CC2(C1)CC2(F)F)=O)CC(=O)NCCC(F)(F)F 69340,C=CC1CN(C(=O)C(CC2CC2)OC)CC1NC(c1cc(C(F)F)ncn1)=O 69341,c1(OC)cccc(C(=O)NCC23CC2CN(C(c2cnc(Br)s2)=O)C3)c1OC 69342,c1(N(CCCNC(Cc2c(C)cccc2C)=O)C)nc2cc(F)ccc2o1 69343,CC(C)C(C(=O)N1CC(CCNC(c2ccnn2CCF)=O)C(C)C1)C1CCC1 69344,CC(CCCNC(=O)Cc1nc(C(C)(C)C)n[nH]1)NC(=O)CC(=O)NCCOC 69345,c1(OC(C)C)ccc(N)c(C(=O)NCC2CN(C(c3cncs3)=O)CCC2C)c1 69346,C12(NC(c3cc(F)cnc3Cl)=O)CCCN(c3nccc(C4CC4)n3)CC1C2 69347,c1(-n2c(-c3c(N)non3)nc(-c3ccncc3)n2)cccc(C#N)c1 69348,C12(NC(c3c(C)ocn3)=O)CCC1CN(C(c1ccc(-n3cccc3)cc1O)=O)C2 69349,N1(C(CCOCC#C)=O)CC2CCC2(CC(=O)NC(C)Cc2ccccn2)C1 69350,CON1CC(C(=O)NC2CCN(C(c3cncc(C)n3)=O)C2(C)C)CC1=O 69351,c1(C(c2ccccc2)NCC(=O)Nc2nnc(CCC(C)C)s2)ccccc1F 69352,O=S(=O)(C1CCCCCC1)C1CCN(S(=O)(=O)c2cc(F)c(Br)cc2F)CC1 69353,c1(C(=O)NCC2CC(NC(CCCC=C)=O)CC2O)cc2occc2s1 69354,C(N=c1nc2c(ncn2C)c(NC(C)Cn2ccnc2)[nH]1)c1n(CC)ncc1 69355,C1(C(C(c2cc(F)cc(Cl)c2)C(Cn2cc(CC(C)(C)C(N)=O)nn2)=O)=O)CC(=O)NC(=O)N1 69356,C1(OC)CN(C(=O)C=Cc2ncc[nH]2)CCC1NC(=O)Cc1ccsc1C 69357,C1(C(=O)NC(c2ccccc2)C(=O)NCCCC(O)CO)CC12CCCCC2 69358,Cn1c(O)nc(N2CC3(CCCC3NC(c3cnn4cccnc34)=O)C2)cc1=O 69359,C12(C(N3CCN(C(CCN(CCC)C)=O)CC3)=O)CC3CC1C2C3O 69360,N1(C(C2(C(=O)OC)CC2C)=O)CCN(C(C2CCN(CC3CC3)CC2)=O)CC1 69361,N1(C(C(COC)C)=O)CC2CCC(C1)N2C(c1cccc(C)c1NC(C)=O)=O 69362,C(=O)(CCCC(C)(C)CC)N(CC(C(=O)N1CC(CCC)C1)(C)C)C 69363,CCCCCCCN(C(=O)C(CCSC)NC(c1cc(C2CC2)on1)=O)C 69364,C12(NC(CNC(CCC)=O)=O)CN(C(=O)C3=CCS(=O)(=O)C3)CC1CS(=O)(=O)C2 69365,c1(OC)ccc(CC(=O)NC2CCC(N(C(=O)CCn3cncn3)C)C2)cn1 69366,N1(C(c2c(OC)n[nH]c2)=O)CCCC2CN(C(C34CC(C#N)(C3)C4)=O)CC12 69367,N1(C(C2OCC(C)C2)=O)CCC(NC(c2ccc([N+](=O)[O-])o2)=O)C12CCC2 69368,c1(C(N2CCCC(CNC(c3sccc3C3CC3)=O)C2)=O)cnn2c1CCCC2 69369,c1(C(N2CC(CNC(C(CC)C)=O)C2)=O)cc(F)cc(Br)c1 69370,Cc1nc(NC(c2c(CO)cccc2C)=O)ncc1Br.C12CCC(CC1)C(=O)N2 69371,N1(C(c2cncc(COC)c2)=O)CCN(C(c2ccc(C)cc2)=O)CC1COC 69372,CCCC(C)CC(=O)NCc1ncccc1CNC(C12CCN(CC1)CC2)=O 69373,N(C(=NCCCOC(C)C)NC(C)Cc1ccc(C)s1)Cc1c(C)cnn1C 69374,O=C(CCCCN1CCCC1)NCCC1CN(C(=O)Cn2cccn2)CCO1 69375,N1(C(C(CC)OC)=O)C2CCC1C(NC(C1(c3cc(Cl)cc(Cl)c3)CC1)=O)C2 69376,C=CCCC(O)CN(C)C(C1CSCCN1C(C1SCC=C1C)=O)=O 69377,C=CCC(CC=C)C(=O)NC1CCOCC1NC(C1(CCF)CC1)=O 69378,N1(C(C2(CC#C)CCOCC2)=O)CCCCCC(NC(c2ccoc2C)=O)C1 69379,c1(C(=O)NC(C)CCCNC(c2ccon2)=O)cc(C2CCCC2)n(C)n1 69380,c1(CN(C(C(C2CCCC2)NC(C2C(NC(C)=O)C2)=O)=O)C)ccc(O)cc1 69381,C(=O)(C(F)(F)C(F)(F)C(F)F)N1CCC(N(C(C2CC23CCOCC3)=O)CC)C1 69382,C1(CNC(=O)Cc2ccsc2)CCC2(CCC2)C1NC(=O)CC1CCOCC1 69383,Cc1cc(=NC(C)CN(C(=O)Cc2ncncc2Cl)C)[nH]cn1 69384,O=C(C1=CCCN(Cc2c[nH]c3ccccc23)C1)N(c1ccc(F)cc1)CCO 69385,C1(C(=O)O)C[Si](C)(C)CN1C(=O)NCCCOCNCc1ccccc1 69386,N1(C(CCSCCC)=O)CC(NC(C2CCCC(=O)C2)=O)C(C)C1 69387,CCCCC(C)CCC(=O)NC(C)C(C)(C)NC(=O)Cc1ccc(O)c(C)c1 69388,C1(C(N2CCOCC2c2nn[nH]n2)COC(F)F)(OC(C)(C)C)CCS(=O)(=O)C1 69389,C(=O)(CC1C(=O)Nc2c(F)cccc21)N1CCN(C(CSCC)=O)C(C)C1 69390,C(=O)(C(C(C)CC)NC(N)=O)N1CCC(O)(CNC(C(C)=CC)=O)C1.C1CC1 69391,N1(C(COCCCOC)=O)CCC(C)C(NC(=O)C(F)=C(C)C)C1 69392,c1(C(N2C(CN(C(C(CC=C)C)=O)CC)CCC2)=O)ccc(NC(C)=O)cc1Cl 69393,CCCC(C(=O)OC)C(=O)N1CC(C)CC1C(=O)NCCCC(C)C 69394,Cc1ccc(NC(=O)C=C2CCN(Cc3c(Br)cnn3C)CC2)c([N+](=O)[O-])c1 69395,C1(C(=O)NCCC(=C)CNC(c2cnnn2C2CC2)=O)CCCC(C)(C)O1 69396,c1(NCc2nc(C)[nH]n2)cc(=NC(C)c2cc(Cl)cc3c2OCC3)[nH]c(C)n1 69397,Cc1cc(C(=O)NC2CC2NC(=O)C2=C(Cl)CCC2)cc(O)n1 69398,N1(C(Cc2c(C)c[nH]n2)=O)CCCC(Cc2cn(CC3CCOCC3)nn2)C1 69399,CC1CCOC1CCC(c1nnnn1CCOCC1CC1)NCC1CC(Cl)(Cl)C1 69400,c1(C(N2CC(CCC)N(C(c3cnnn3C)=O)CC2)=O)ccn2cccc2c1 69401,Cn1ccnc1C(N1CCC(C(=O)NCCOc2cccnc2)C1)=O 69402,C=C1CCN(C(c2nc(C)sc2C)=O)C(C(N2CCCC(C(C)C)CC2)=O)C1 69403,C1(C(=O)NCC(CNC(=O)C(C2CCOCC2)C)CO)(CC)CCCC1 69404,CCC(C(=O)NC(C)CCNC(C1(F)CC=CC1)=O)OC 69405,C(C(CC(C)C)NC(c1cnc(C)s1)=O)NC(c1n(CC=C)ccc1)=O 69406,CC(F)(F)CCC(=O)N1C2CCC1C(CNC(c1ccnn1CC1CCC1)=O)C2 69407,N1(C(CCC2N(C(c3c(CC)cco3)=O)CCC2)=O)CCC(C)C2(CCC2)C1 69408,c1(CN(CCCCOCCS)C)csc(-c2cnn(C)c2)n1 69409,CC1CN(C(=O)CC(O)C2CCCC2)CCC1NC(c1cn(C)ccc1=O)=O 69410,C1(NC(C2CC2O)=O)CCN(C(c2ccc(C3CC3)nn2)=O)CC1CO 69411,C1(NC(CN(CC)CC)=O)CC2(C1)CC(C(=O)NC1CCC3CCC13)C2 69412,N1(C(C(C)OC)=O)CCC(F)(F)C(N=c2nc(C)nc3[nH][nH]cc2-3)C1 69413,N1(C(CNC(=O)OC)=O)CC2CCC2(CC(=O)NC2CC(=C3CC3)C2)C1 69414,C1(O)(SCC)CCN(C(=O)C(C)C(=O)OC(C)(C)C)C1.C1(C2(CC)CC2)C(=O)N1 69415,Cc1cc(C(N2C(C(N3CCC(F)(F)C3)=O)CC3CC23)=O)c(C)cc1Br 69416,C(=O)(C1CCCc2scnc21)N1C(C)(C)CC(NC(C2CCC(C)CC2)=O)C1 69417,C1(OC)CCC(C)(C(=O)NCCCCC(CO)NC(=O)CCF)CC1 69418,CC1CC(C(=O)NCC2(O)COC2)N(C(c2cnc(Br)s2)=O)C1 69419,c1(NC(=O)CC(F)(F)F)ccccc1NC(=O)C(=O)N(C(C)CC#N)C1CC1 69420,N1(C(COc2cccc(CC)c2)=O)CCC2(NC(=O)C(C)(F)F)CC2C1 69421,c1(NC(c2cn(CC=C)nn2)=O)cccc(CNC(=O)CC2CC2C2CC2)c1 69422,C#CCC(C)(C(=O)NCCC)NC(=O)CCC(=O)NC.C1CN2CCC1CC2 69423,N1(C(CC2CCC(OCCC)CC2)=O)CC2CC1CCC2NC(c1cnsn1)=O 69424,N1(C(Cc2c(C)ocn2)=O)C2CCCC1CN(C(C1CCCOC1)=O)CC2 69425,N1(C(=O)NC(C2CCO2)C2CCC2)CCN(N2CCC2)CC1 69426,c1(NCc2cc(C)ncc2)nc(C)nc(Br)c1F 69427,c1(C(=O)NC(CNC(c2c(C)ccnc2O)=O)C(C)(C)C)ccc2c(c1)OCC2 69428,N1(C(C(CC)C)C(=O)NCCC2CC2)CCC2(CCCOC2)CC1 69429,N1(C(c2c(OC)cc(Br)cn2)C(=O)NC2CC(F)(F)C2)CCCNC(=O)C1(C)C 69430,CC1Cc2cc(CCN=c3ccnc(N4CCC(C)(F)C4)[nH]3)ccc2O1 69431,C1(NC(C=CCN(C)C)=O)CC2CN(C(c3[nH]nnc3C(F)F)=O)CC12 69432,N(C(=NCCCC1CCC1)N1CC=C(c2cccs2)CC1)CCOC 69433,CCC(C(=O)N(C1CCCC1)CCNC(=O)COCC1CCCC1)SC 69434,C=CC1CN(C(C2CC(=O)CCO2)=O)CC1NC(C1CCCO1)=O 69435,CCC(CC(=O)NC1CCC12CN(C(=O)COc1ccc(C)c(C)c1)C2)C(F)F 69436,c1(NC(=O)NCc2[nH]nc(CSC)n2)cnc(N(C)C)nc1 69437,S(=O)(=O)(c1c[nH]c(C(=O)NC2CN(C(=O)CCc3cnn(C)n3)CC2F)c1)NC 69438,N1(C(CC=C)=O)CCCC(NC(c2nc(C)n(C3CC3)c2C)=O)C1C 69439,C(CCC(=O)NCCC1(NC(=O)CCF)CCCC1)=CC 69440,S(=O)(=O)(c1cnc(NCC2CCC2)c(Cl)c1)NCC(C(CC)CC)O 69441,N1(C(C(COC)OC)=O)CC(CNC(=O)Cc2cccc(OC)c2Cl)C2(CC2)C1 69442,CC1CCCCC1CNC(=O)CC(c1cccc(Br)c1)C 69443,Cc1ccc(F)c(C(=O)NCc2cccc(CNC(c3cn(C)cn3)=O)c2)c1F 69444,C(=O)(C(CNC(C1(CO)COC1)=O)C(C)(C)C)N(CCC)CC 69445,CC1CCC(NC(=O)Cn2cnc(=N)[nH]2)CN1C(=O)CC1(CO)CC1 69446,N1(C(C23CC(OC)C2C3)=O)CCN(C(c2cc(C3CCCC3)n(C)n2)=O)C(C)C1 69447,CC1(C(=O)NCC2(O)CCN(C(=O)CCCn3cccc3)C2)CCCNS1(=O)=O 69448,N1(C(CC(=O)OC)=O)CC(NC(C2(F)CCC2)=O)C(C)C1 69449,c1(C(=O)NC2(C)CCC(NC(C(C)(C)OC)=O)CC2)cc(C)c(F)cc1N 69450,c1(C(=O)NC(C)CN(C)C(c2cnn(C3CCOC3)n2)=O)cncc2c1CCC2 69451,c1(C(=O)NC2(C)CN(C(C(CCC)(C)C)=O)C2)n[nH]c2c(C)cccc12 69452,Cc1cccc(OCCCC(N2CC(CNC(=O)C#CC(C)C)C(O)C2)=O)c1 69453,C(=O)(CC1=CCCC1)NCC(C)CNC(c1conc1C(F)(F)F)=O 69454,c1(C(=O)NCCCCC(C)NC(=O)C(C2CC2)N(C)C)ccn2nccc2c1 69455,C1(C(N2CCOC(c3n[nH]c(CO)n3)C2)=O)CCOC2(CCC2)C1 69456,CCC(F)(F)CC(=O)N1C2CCC1C(CNC(c1ccc(OC)c(C)c1)=O)C2 69457,N1(C(CCNC(=O)OC(C)(C)C)=O)CC2CCC(NC(C3(CSC)CC3)=O)CC2C1 69458,C1(NC(CN(CCCCCC)C)=O)CC2CCCC(C1)C2NC(=O)C(C)CF 69459,C(=O)(C(C)(C)C(O)C(C)C)NCCC(CC)(CC)NC(CCC(C)SC)=O 69460,Cc1nc(=N)[nH]c(C)c1C(=O)N(C)CCNC(c1cc(F)ccc1C(F)F)=O 69461,C(=O)(CC1OCc2cc(Cl)ccc21)N1CC(CCNC(C2CCC(=O)NC2)=O)C1 69462,N#Cc1cnn(-c2ccccc2)c1NC(C1CCN(Cc2cccnc2Cl)C1)=O 69463,Cc1nc2ccccn2c1C(=O)NC(CNC(C1CCCC1C)=O)C(C)(C)C 69464,C1(NC(C2N(C)CC2)=O)CCCCC1NC(c1cnc[nH]c1=N)=O 69465,CN1CCN(C(c2ccc(O)nn2)=O)CC1C(N1CC(n2cnnc2)C1)=O 69466,c1(CC)cc(N)c(C(N2CCOC(CNC(=O)CCC(CC)SC)C2)=O)cc1F 69467,C1(CC(=O)N(CCC(N2CC(C)(CC=C)C2)=O)CCCO)CCC(=O)CC1 69468,c1(C(=O)NC(C)CCCO)ncsc1C(=O)NCCC1(CC)CCCC1 69469,C(CCCCC(C(=O)NC(C)(C)C)N1CCN(C(C)(C)CF)CC1)OC 69470,S(=O)(=O)(c1cc(C)cnc1NCC(O)C(C)C)NC(c1scc(CC)n1)C 69471,c1(OC)cc(C)sc1C(=O)NC1CC(NC(c2cc(Br)n(C)n2)=O)C1 69472,C1(CCCSCC(=O)NCC#C)CCN(C(c2ccc(NC)cn2)=O)CC1 69473,c1(NC(C(=O)N(CC(C)NC)C)(C)C)cc(N(C)C)nc(SC)n1 69474,N1(C(C=NOC)=O)CCCC2(C1)C(NC(=O)CC1CC3CC3C1)CCN2C 69475,c1(OC)cc(C2CCCN(C(C3(C4CCC4)CCC3)=O)C2)cc(F)c1 69476,c1(CC)cc(C(=O)NCC2(C(C)(C)C)CCN(C(c3csc(C)c3)=O)C2)ncn1 69477,c1(OC)nc(OC)nc(N(C2CCNCC2)C(=O)CCn2nc(C)nc2C)n1 69478,C12CC3CN(CC13)C(=O)C1CN(C1)CC(=O)N2.c1(CC)cccc(F)c1 69479,c1(CNC(C(C)CO)=O)cc2n(n1)CCN(C(c1cc3n(n1)CCCO3)=O)C2 69480,C12(C(=O)NC(C3CCCOC3)(C)C)CC(CO)(CN1C(c1ccncn1)=O)C2 69481,Cc1ccc(CC(C)NC(=O)NCc2cccc(-c3ccccc3)n2)c(C)c1 69482,N12CC3CC1CN3C2=O.c1(C(C(C(=O)OC)C)=O)ccc(C(C)(C)C)cc1 69483,c1(CC(=O)NC(C2(O)CCN(C(=O)C3=CCOC3)C2)C)cc(F)cc(F)c1 69484,C1(C(=O)NCC(C(=O)OC)(C)O)CCN(C(C2(C)CC3C=CC2C3)=O)C(C)(C)C1 69485,CC1CC(NC(c2cn(CCO)nn2)=O)CN(C(=O)Cn2ccccc2=O)C1 69486,Cc1cc(NC(=O)C(=O)Nc2cccc(C(C)C)c2)nc(-c2cnccn2)n1 69487,n1(CC)cccc1CCNC(=O)NCCCC(=O)N(C)C(C)C 69488,C(=O)(CC(O)CNC(=O)C(C)(CO)NC(=O)C(n1ccc(C)n1)C)OC 69489,c1(SC)cccc(CC(=O)NCC(C)(CC)NC(=O)Cc2cnc[nH]2)c1 69490,C1(CNC(CC2(COC)CC2)=O)CN(C(=O)C(C)C2CCC2)C2COCC2O1 69491,c1(C(N2CC3(CCN(C(c4cnc(C)s4)=O)C3)C2)=O)cccc2nc(O)oc12 69492,C1(CC)CN(Cc2ccc(Br)c(O)c2)CCN1C(c1cccnc1SC)=O 69493,N1(C(c2n(C(C)C)cnc2)=O)CCN(C(=O)C=Cc2nnn(C)n2)C(CO)C1 69494,N1(C(C=Cc2cccc(OC)c2)=O)CCC(NC(C2COC(=O)C2)=O)C(C)(C)C1 69495,c1(C(=O)OCc2cc(C(=O)NC)c(F)cc2)cnc(C)c(C#N)c1 69496,C1(CCCNC(C(C)Cc2ccco2)=O)CN(C(=O)CN(C)C(N)=O)CCCO1 69497,c1(OC)ccc(OCC(N2CCC2CNC(=O)CC2COCC(C)O2)=O)cc1C 69498,N1(C(=O)OCC)CCCCCCC1NCCCc1cscn1 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70010,N1(C(C(C(CC)O)C)=O)CCCC2(C1)CN(C(=O)CCc1ccccn1)CCO2 70011,c1(C(N2CC3CC(CNC(C(C)(C)OC)=O)C3C2)=O)coc(S(=O)(=O)N(C)C)c1 70012,c1(NC(C(C)NC(c2ccc(C)[nH]2)=O)C(C)C)cc2nn[nH]c2cc1[N+](=O)[O-] 70013,C(=O)(C(C)(O)CC(F)F)N(CCCNC(c1ccc(CN(C)C)o1)=O)C1CC1 70014,c1(CCNCC(COCC(C)C)O)coc(-c2ccccc2)n1 70015,O=C1Cc2cccc(C(=O)NC3CCN(C(c4c(F)cccc4Cl)=O)C3)c2N1 70016,C(=O)(N(CCC(=O)N1CCCC(C(C)C)C1)OC)C1C(CC)CCOC1 70017,N1(C(C2(OCC)CCC2)=O)C2CCC1C(CNC(=O)Cc1cccnc1Cl)C2 70018,N1(C(C(COC)O)=O)CCC(CC(=O)O)(NC(=O)OC(C)(C)C)C1 70019,c1(C(=O)NCC(C2CCCC2)NC(c2csnn2)=O)cccc2c1OCCO2 70020,c1(N2C(Cc3scc(C)n3)CCC2)ncc2cc(C)ccn12 70021,c1(C(N2C(CN(C)C(C3CCCOCC3)=O)COCC2)=O)cnn2ccncc12 70022,CCC(C(=O)NCCOCCN(C(=O)CC1CCC(O)C1)C)C(C)C 70023,c1(C(=O)NC2C=CC(C(=O)NC3(C#C)CC3)C2)cnn(C=C)c1N 70024,C(=O)(C1=CCN(C(c2coc(C)c2)=O)CC1)N(C1COCC1O)CC 70025,C1(O)(C(N2CCN(CCNC(=O)Cc3ccco3)CC2)=O)CC2CCC1C2 70026,N1(C(C2(C(=O)OCC)CC2)=O)CC2CC(C1)N(C(C1(F)CCC(C)(C)CC1)=O)C2 70027,N1(C(C(=O)NCc2ncc(Br)cc2C(F)F)=O)CCc2ccc(F)cc21 70028,C(CC(C)C(=O)N1CCC(C)(CNC(c2nn(C)cc2SC)=O)C1)=CC 70029,N#Cc1cccc(NC(=O)C(=O)NC(C2CCOC2)CO)n1 70030,C(=O)(C(C)CC(C)(F)F)NCCCCCN(C(C1CC=C(C)CC1)=O)C 70031,C1(C(=O)CN2CCCC2)CNc2ccccc2C1Cn1cc(I)cn1 70032,Cc1ccc(C(=O)NCC2C=CC(NC(C3CC(CC4CC4)C3)=O)C2)o1 70033,c1(CC(=O)N(CC(CC)NC(=O)CCN2CCC(F)C2)C)ccccc1F 70034,C(=O)(C=CS(=O)(=O)CC)N1CC(C(Cn2cc(CC(C=C)O)nn2)F)C1 70035,c1(C(=O)NC(C2N(C(CC(=O)OCC)=O)CCC2)C)cc(C)nc(O)c1 70036,c1(SCC#C)cccc(C(=O)NC(CNC(=O)C(c2cccs2)SC)CO)c1 70037,c1(OC)nc(C2=CCNCC2)ccc1C(=O)Nc1cnn(CC(F)F)c1 70038,N1(C(=O)NC2(C(=O)O)C(C)C2)CCN2CCN(C(C3CCC(=O)N3C)=O)CC2C1 70039,C1(CNC(CS(C(C)C)(=O)=O)=O)CCC2CN(C(C3CC4CC4C3)=O)CCC2C1 70040,N1(C(C)C)CC2CN(CC34CCCC3C4)CCC12 70041,C1(NC(c2c(CC)nco2)=O)CCN(C(c2c[nH]nc2-c2cccs2)=O)CC1F 70042,c1(C2CCN(CC(F)F)C2)nc(C2OCCc3ccccc32)nn1C1CCSC1 70043,C1(C(N(C)Cc2ccc(F)cc2)=O)CC(C)(C)CN1C(C1CC2(CC2)CO1)=O 70044,c1(C(N2CCC(C)C(N(C(=O)CC3CCCOC3)C)C2)=O)cc(C#N)ccc1F 70045,Cc1nnc(O)c(C(=O)NCC(C)N(C(=O)C(C)Cn2cccn2)C)c1C 70046,N1(C(C(N2CCCC(C)C2)=O)=O)CCC(NC(=O)C(F)(F)c2cncs2)C1(C)C 70047,N1(C(CN(C(=O)OCC)C)=O)CCC2(CC1)CC2C(=O)N(C)CC1CCCOC1 70048,c1(SC)cc(Br)c(F)cc1NC(=O)NCc1cn(-c2cc(F)cc(Br)c2F)nn1 70049,c1(CC)cc(=NC(=O)C2CC(NC(=O)CC3CCCCC3O)C2)[nH]n1C 70050,C1(OC)CC(CNC(=O)Cc2occc2C)N(C(=O)Cc2ccccc2F)C1 70051,C12(C(=O)NC3(C4N(C(CC5(OC)CC5)=O)CCC4)CC3)CCN(CC1)C2 70052,c1(CN2C(C(N3CCC(C(N)=O)CC3)=O)CC2)c[nH]c2cccc(F)c12 70053,c1(C(N2CCC(NC(C(C)SC)=O)C(C)C2)=O)cccc2c1NCC2 70054,C(=O)(C(C(C)CC1CCOCC1)N(C)CC1CCCN(C)C1)NCC=C 70055,C(=O)(C1=CC2(CCOCC2)C1)N1CC(C)(CNC(=O)C2=CS(=O)CCC2)OCC1 70056,Cc1nnccc1C(N1CCC(CNC(=O)CN2CCCNC2=O)C1)=O 70057,N1(C(Cn2cc(C(C)O)nn2)=O)CC(NC(=O)CC(C)(F)F)CC1C 70058,C1(C(=O)NC(C)CCNC(=O)C(O)C2CCCC2)CCC(N=[N+]=[N-])CC1 70059,N1(C(C2=C(C)CC2)=O)CC2(C(N3CCOC(CCO)C3)=O)CC1CO2 70060,C1(C(=O)NC(CNC(c2cc(OCC)ncc2)=O)(C)C2CC2)CC2(C1)CC(F)C2 70061,C1(CCC)CN(C(=O)C(=O)NCC2CC2)CCN1C(=O)COc1cccc(F)n1 70062,C1(C(=O)NC2(C)CN(C(CC(C(C)C)OCC)=O)C2)Cn2c(C)nnc2CN1C 70063,C1(CNC(C(C)OC)=O)CN(C(C2CCN(C(=O)OC(C)C)CC2)=O)CCN1C 70064,CC1CCN(C(=O)COCC2CC2)CCN1C(=O)C(C1(O)CCCC1)F 70065,C1(CC(=O)N(CCN(C(C(C(C)C)OCC)=O)CC)CC)CCCC2(CCC2)O1 70066,C1(CC)CCC(C(=O)NCCC2CN(C(=O)Cc3ccsc3C)C2)C1 70067,C1(C(=O)NC(CC)CO)C(CNC(c2ccoc2Cl)=O)C1(C)C 70068,c1(C(=O)NC2CC(C)(NC(CC(C)CF)=O)C2)nc[nH]c2ncnc1-2 70069,c1(CC(C)N(C(c2ccc(C(Cl)Cl)cc2)C(=O)NC)C)c(C)nn(C)c1C 70070,CC(N=c1[nH]c2c(c(=NCCOc3ccc(Cl)cn3)[nH]1)CCCCC2)C1CC1 70071,C1(NC(C=CC=CCCCCC)=O)CN(C(c2csnc2C)=O)CCC1CO 70072,c1(NC(c2ccccc2I)=O)ccccc1N1CCCCC1 70073,C=CC(C)(O)C(=O)NCCCN(C)C(C1(c2cccs2)CC1)=O 70074,C1(NC(c2cccc(C3CCC3)c2)=O)C2CCN(C(C3CC=CCC3)=O)C12 70075,N1(C(COC)=O)CCN(C(C2CC(=O)N(c3ccc(Cl)c(F)c3)C2)=O)C(CF)C1 70076,Cc1cc([N+](=O)[O-])cnc1C(=O)NC1CC1NC(c1cnc2ccc(F)cn12)=O 70077,Cc1cc(C)c(C(=O)NCc2cc(C(=O)Nc3ccccc3)n[nH]2)s1 70078,c1(C(=O)NCC(C)(C)OCCNC(C(CC(C)C)OC)=O)c(C)ccc(C)c1C 70079,c1(C(=O)NCCCN(C(c2cccnc2)=O)CC)cccc2scnc12 70080,C1(NC(COC2(C)CCC2)=O)CC2CC(NC(=O)CSc3n[nH]c(=N)s3)C2C1 70081,C(=O)(CC(F)(F)F)N1C(CN(C(C(n2ccc(C)n2)C)=O)C)CCC1 70082,C1(C(=O)NCCCCCN(C(=O)C(C)(C)C(N)=O)C)CNc2ccnn2C1 70083,C1(C(=O)NCCN(C(=O)C(=O)Nc2ccccc2)CC)COCCN1C 70084,CCCC(CC(=O)NCCN1CCCCC1)NC(C1CC(CF)C1)=O 70085,C(CC(=O)N1CCCC(CCO)CC1)(C(F)F)NC(C1C(CC(C)(C)C)C1)=O 70086,C1(C)(C(N(CCC)C2CC2)=O)CC12CCN(C(C)Cc1cccc(Br)c1)CC2 70087,C1(C(=O)Nc2c(C(=O)OC)cc[nH]2)CC2(CCC2)CN1C(c1ncccc1F)=O 70088,N1(C(COC(C)(C)C)=O)CCC2CN(C(=O)C=Cc3cccs3)CC2C1 70089,CCCCCCC(C)(CC)C(=O)NC1CCC(NC(=O)CCc2nncs2)C1 70090,c1(C(=O)NC2(CNC(c3c[nH]nc3F)=O)CCOC2)cc(Cl)c(Br)[nH]1 70091,N1(C(C2C(NC(c3c(Cl)ccc(OC)c3)=O)C2)=O)Cc2ccc(Br)cc2C1 70092,C(C(=O)N1OC2CCC1C2)C1CCN(C(C(N=S(C)(C)=O)=O)=O)C1 70093,C1(C2CC2)(NC(C(C)OCCCC)=O)CCN(C(=O)C(C)(C)C(=O)OCC)C1 70094,c1(SCC(N2CCC(N(C(=O)CN3CC4CC4C3)CC)C2)=O)c(O)nc(=N)[nH]c1C 70095,C1(CCN(C)C(c2ccc(F)cc2)=O)CCCCN1C(c1n[nH]cc1Cl)=O 70096,c1(CNC(c2c(C)ncnc2)=O)nc(CNC(=O)CN2CCOCC2)cc(O)n1 70097,C(=O)(C1=Cc2ccccc2C1)N1CC(F)(CNC(=O)C2=CC3(CCOC3)C2)C1 70098,CCS(=O)(=O)CC(=O)NCC1(C(=O)NCC(C)(CO)CO)CC12CCC2 70099,CCCC(CC(C)C)C(=O)NCC1(NC(=O)COC(C)CC)CCOCC1 70100,C(=O)(C1=CS(=O)CCC1)NC(CC)CNC(=O)C(c1ccc(F)c(F)c1)C 70101,C(CCN(C(=O)CC1CC=CCN1C)C)(C(C)(C)C)NC(C1CC(OCC)C1)=O 70102,C1(O)(CNC(C(C)N(C(C2(CCC=C)CC2)=O)C)=O)CCCCCC1 70103,N1(C(C2CCC(CC)O2)=O)CCCN(C(c2cnc(O)cc2C)=O)C(CO)C1 70104,N1(C(c2ccno2)=O)CC(C2CCCN(C(C3CC3F)=O)C2)C1 70105,N1(C(CCOCCN(C(C=C(C)C(F)F)=O)C)=O)CCCC(C)(C#N)C1 70106,CC1C(C(=O)Nc2cccnc2F)CCCN1C(C1CC2(C1)CC2(F)F)=O 70107,C1(C)(NC(C(CSC)O)=O)CCCN(C(c2nc(C(F)(F)F)oc2C)=O)C1 70108,c1(Nc2cccc(Nc3ncc(OC)cn3)c2)ccc(S(C)(=O)=O)cc1C 70109,C1(NC(CCn2ccc(C)n2)=O)CN(C(c2ccsc2)=O)CCC1F 70110,C1(C2N(C(C(C)N3CCCC3)=O)CCC2)CCN(C(=O)C=C2CCOCC2)CC1 70111,c1(COC)cc(C(N2CCOCC2CNC(C2(O)CC(C)(C)C2)=O)=O)n(C)c1 70112,C12(NC(C3=NOC(C)C3)=O)CCCC1(F)CN(C(c1ccncc1Cl)=O)C2 70113,N1(C(C(CCC)O)=O)CCC(O)(C(C)NC(=O)CN(S(C)(=O)=O)C)CC1 70114,C(CC(C(=O)N(C1CCC(CO)CC1)C)NC(C1(C(C)C)CCCO1)=O)SC 70115,c1(OC)cc(F)c(C(=O)NC2CC(F)(CNC(=O)CC3COCCO3)C2)c(F)c1 70116,N1(C(C(C2CC2)SC)=O)CCC(C(=O)N(C(C)C(F)F)C)(CF)C1 70117,c1(C(N2CC(C)(OCC(N3C(C)(N(C)C)C=CC3)=O)C2)=O)cc(=O)n(C)cn1 70118,C(=O)(C(=O)NCCNC(C)=O)NCCN(C(=O)Cn1ncnn1)CCOC 70119,N1(C(c2c(C3CC3)ccc(C)c2)=O)CCC2CCC(C1)N2C(=O)CCC#N 70120,N1(C(CCc2ccc(C(=O)OC)cc2)=O)CCN(C(C2CSC2)=O)CC1CCO 70121,N1(C(CN(C(C)C)CC)=O)CCC(C(C)(C)NC(=O)C(O)CC2CC2)CC1 70122,c1(C(N2CCC(C)(NC(=O)CC3CCOC3=O)C2)=O)cc(S(N)(=O)=O)ccn1 70123,S(=O)(=O)(c1c(F)cc(F)cc1F)N1CC2CN(C(C(C(C)(C)C)O)=O)CC(C1)O2 70124,N1(C(c2ccn(CC)n2)=O)CC2CC(C1)C(CO)C2NC(C1CC1F)=O 70125,CC1CC(C(=O)NCCn2cncn2)CN(C(=O)Cc2ccon2)C1 70126,N1N(CCc2cn(-c3ccc(OC)cc3)nn2)CCOC2(CCOC2)C1 70127,C(CCN=C(NCc1cccc(O)c1)NC1CCCC1)c1c(C)cccc1 70128,c1(-c2cn(C3CN(C(CCOCC)=O)C3)nn2)sc(OC2CCCOC2)nc1Cl 70129,C12(C(N3CC(NC(c4ccc(CO)o4)=O)C3)=O)COCC1CS(=O)(=O)C2 70130,C1(C(=O)NC(C(=O)NCCc2c(C)ocn2)CN(C)C)CC2CCC1O2 70131,C1(NC(C(C)=C2CC2)=O)CN(C(C2(C)CCCS2)=O)CC2(CCOCC2)C1 70132,Cc1nccc(C(=O)NC2CC(C(=O)NCCN(C)C(C)C)C23CCC3)c1C 70133,CC(CS(N)(=O)=O)NC(=O)CC1CCC(NC(C2(C)CC=CCC2)=O)C1 70134,C(C(CC1CC1)C(=O)N1CC2CC2(CO)C1)NC(C1CC(=C2CC2)C1)=O 70135,NC(=O)CC(O)C(=O)N1CCC(NC(=O)CCOc2ccc(Cl)c(Cl)c2)C1 70136,c1(CN2CCC(C(=O)Nc3c(C)nn(C)c3C)C2)ccc2c(c1)CCCO2 70137,C=CC(C)(O)CC(=O)NCCC1(C(=O)NCC2CCSCC2)CCC1 70138,N1(C(C(CC)NC(C)=O)=O)CC(C(=O)N(CC(F)(F)F)Cc2ccoc2)C(C)C1 70139,c1(C(=O)NCC(C2CCOC2)NC(=O)COC2CCC2)ccc(CO)nc1 70140,CC(CCC(C)(C)C)C(=O)NC1CCN(C(=O)CCc2cnn[nH]2)CC(O)C1 70141,N(C1CCc2cc(CO)ccc21)C(=O)Nc1cnc(O)c(N2CC(OCC)C2)c1 70142,C=CC(CC)CC(=O)N(CCC(C)NC(=O)CCNC(=O)OCC)C 70143,C1(CC(=O)NC(CSC)C)CCCC(NC(=O)C(C)c2cc[nH]n2)C1 70144,CC1CCCC(C(=O)NC(C)(C)CC(=O)NCc2nn(C)c(=O)o2)C1 70145,C1(CC(C)NC(C2(C3CC3)CCCO2)=O)CCN(C(c2ccco2)=O)CC1 70146,C#Cc1cccc(C(=O)NC2CN(C(C3COCCN3C)=O)CCC2(C)C)c1C 70147,C(CC(C(C)C)NC(C1(CNC(=O)CC2CSCCO2)CC1)=O)OC 70148,C1(C(=O)NCC2(C)OCCN(C(CC(=O)NCC)=O)C2)CCn2c(O)nnc2C1 70149,C#Cc1ccc(Br)c(C(=O)NCC(=O)N=S(C)(C)=O)c1 70150,N1(C(c2scnc2C)C(=O)NC)CCC(O)CC12CC2 70151,N1(C(CC2(C)CCCCC2)=O)CCC=C(CNC(c2cccnc2)=O)C1 70152,C(c1cnn(C)c1C)=CC(N1CCC(NC(C2CCC(=C)CC2)=O)C1)=O 70153,c1(C)cccc(C(F)F)c1.C12(C(F)F)CN(C1)C(=O)N2.C1(OC)=CCC1 70154,C1(CCOC)CN(C(=O)C(N2CCN(C)CC2)(C)C)CCN1C(c1csnn1)=O 70155,CC(C)CC(CNC(C1(F)CCC1)=O)NC(=O)CC(=O)NC1CC1 70156,C1(CNC(c2ccc(C(C)=O)s2)=O)CC(C)N(C(=O)Cc2cnn(C)c2)C1 70157,Cc1cccc(C=CC(=O)NC2CC(O)C2CC(=O)NCC(F)(F)C(N)=O)c1 70158,C1(C(COC(c2ncn(CCC)n2)=O)=O)CC(=O)N(c2ccc(SCC)cc2)C1 70159,c1(C(=O)NCC2C3CN(C(C45COC(CCO4)C5)=O)CC23)ccc2cc[nH]c2n1 70160,CC1CC(CNC(=O)CC(C)(C)O)CN1C(c1cnco1)=O 70161,C#CCC(CC#C)C(=O)NCC(CC)(CC)NC(=O)CCC1CC2CCC1C2 70162,N1(C(CCC(=O)NC)=O)CCC2(CCN(C(=O)C(C)OCC3CCCO3)C2)C1 70163,c1(N(CCCC)Cc2ncc(-c3c[nH]c(=N)c(C)c3)cn2)cccc(O)c1OC 70164,c1(C(N2C(CO)CC(NC(C(C)S(C)(=O)=O)=O)C2)=O)ccc(F)c(Cl)c1F 70165,Cn1ccc(C(=O)NC2CC(CNC(C3CC(C(F)(F)F)C3)=O)C2)c1C1CCC1 70166,CC(C)CC(C(=O)NCc1ccc(CO)o1)N(C(=O)CC(C)C1CC1)C 70167,C(=O)(C(CCC=C(C)C)N(c1ccccc1Cl)C)NC.C1CC(=O)N1 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70185,C#CC1(C)CCN(C(c2c(C)noc2C)C(=O)NC)CC1 70186,c1(C(N(C(C)C)Cc2ccc(F)cc2F)=O)cccc2c1CCC(=O)N2 70187,C12CCCC(C1)NC(=O)N2.C(CC(=O)N(CC(C)C)C(C)C)NC(COC)=O 70188,c1(CC(N2CC(CCNC(C3CC(CC4CC4)C3)=O)(OC)C2)=O)ccccc1F 70189,N1(C(C2CCCN(CC)C2)=O)CC2(CC(CC(=O)NC3(CCF)CC3)C2)C1 70190,N1(C(C2N(C)S(=O)(=O)CC2)=O)CCCC2(CCCN2C(C2CC(O)C2)=O)C1 70191,c1(C(N2C3C(NC(c4n(CC)nc(C)c4)=O)C(CC3)C2)=O)ccc2nonc2c1 70192,N1(C(C=Cc2ccc(C(N)=O)o2)=O)CCCC(C2CN(C(=O)C3=COCC3)C2)C1 70193,C(=O)(CCC(C)(C)OC)NC(CC)(C)CNC(=O)CCC=CC(C)C 70194,C1(=CC(N2CC(CNC(CC3(C#N)CCC3)=O)C3C2C3)=O)CCCCC1(C)C 70195,C(=O)(C(F)C(F)(F)F)NC1C(C(N2CCOC(CCCNC(C)=O)C2)=O)C1(C)C 70196,N1(C(C(C)CC(F)(F)F)=O)CC2(C)CN(C(C3CC4(C3)CC(O)C4)=O)CC2(C)C1 70197,N1(C(c2cn(CC(=O)N(C)C)nn2)=O)CC2CC2(CNC(=O)C(F)(F)C2CC2)C1 70198,N1(C(c2cc(C#N)no2)=O)CCC2CCN(C(=O)COCCF)CC12 70199,C1(F)(C(=O)NC(C(C)C)CCN(C(=O)C=Cc2nnn(C)n2)C)CC2(CCC2)C1 70200,c1(CNC(=O)NC2(C3CC3)CCCCC2)cccc2c1OCCC2O 70201,N1(C(C2(CO)COC2)=O)C(C(N2CCC2NC(=O)NC2CC2)=O)CCC1C1CC1.CO 70202,CCCC(O)C(CO)NC(=O)C1=NOC(CNC(C2CC3(CC3)C2)=O)C1 70203,C1(C(=O)NC2CCCCCC2)CC2(CCC2)CN1C(c1cscc1Cl)=O 70204,c1(CN2CCC(C(C)=O)C2)cccc(Cn2nc(C)cc2C)c1 70205,C(=O)(C(C(C)C)NC(=O)COC1CC(n2cc(COC3CCCC3)nn2)C1)OC 70206,C12(CNC(C(C)OCCCCCC)=O)CC(CN1C(=O)C(O)Cc1cnc[nH]1)C2 70207,N1(C(CC(=O)NCC#C)=O)CCC(C)C(NC(=O)C(CC)n2cccn2)C1C 70208,C=CC1CN(C(=O)COCC2CCOC2)CC1NC(C1CC2CC2C1)=O 70209,c1(C2N(C(c3c(OC)oc(C)n3)=O)CCC2)cccc(Cl)c1Cl 70210,C1(NC(C(n2cc(C3CC3)nn2)C)=O)CCN(Cc2ccccc2)C1C(C)(C)C 70211,c1(N2CCN(C(=O)NOCC(F)(F)F)CC2)ncnc2ccccc12 70212,C(=O)(C=C=C(C)C)N1C(C(=O)NCCC2(COC)CC2)CC1C 70213,CCCC(C(=O)OC)C(=O)N1CCC2(C1)CN(C(C1CCCS(=O)(=O)C1)=O)C2 70214,N1(C(Cn2c(CCC)ncc2)=O)CCC(O)C(N(C(=O)C(F)C2CCC2)C)C1 70215,Cc1cc(O)cc(O)c1C(=O)NC1CC(C)CN(C(=O)C2=CCCC2)C1 70216,C#CC1CCC(C(N2CCOC(C(C)NC(=O)COc3cn[nH]c3)C2)=O)CC1 70217,c1(C(=O)NC(C)CNC(C2(O)CC3CCC2C3)=O)ccc(F)c(F)c1F 70218,C(=O)(C1CC(=O)Nc2cc(F)ccc21)N1CC(NC(=O)CCF)C2C1CCCC2 70219,C(C(C)(O)C(=O)NCc1cccc(F)c1)OC.C12CC(C1)NC(=O)CCNC2=O 70220,CCC(C)(C)C(=O)C(=O)NC1(CO)CCCN(C(=O)Cc2ccc(C)cc2)C1 70221,c1(C(=O)NCC2(C)CN(C(C3CC4(CSC4)C3)=O)CCO2)cccn2cnnc12 70222,CC(CC(F)(F)F)C(=O)N1CCC(C(C)(C)C(=O)NC23CCC(CC2)C3)C1 70223,c1(C(=O)NC(C(C)NC(c2cnn(C(C)(C)C)c2)=O)C)cc(Cl)n(C)n1 70224,C1(NC2(c3nnnn3Cc3ccco3)CC(F)C2)Cc2nc3ccccc3n2C1 70225,C1(CCC(C)C)CCN(CC(=O)NCCC2CCCCC2)CC1 70226,c1(-n2cc(C(C)(C)NC(CC(=O)NC)=O)nn2)cccc2cnccc12 70227,c1(OC(C(=O)NCC2CN(C(CC3C(C)C3)=O)C2)C)cccc(Br)c1 70228,Cc1cc(C=CC(N2CC(NC(C3CC3C(F)F)=O)C3(CCC3)C2)=O)c[nH]c1=N 70229,C1(C(N(C)CC2N(C(c3cc(C)c(C)o3)=O)CCC2)=O)CCC2C(CC1)C2(F)F 70230,Nc1sc2c(c1C(N1CC(O)(CNC(C3C4CCCC34)=O)C1)=O)CCC2 70231,CCC(CNC(C12CC(C)(C1)C2)=O)(CC)NC(=O)CCn1cccc1 70232,C(=O)(CS(=O)(=O)CC(C)C)NCC1CCN(c2snc(SC)n2)CC1O 70233,C1(C(=O)NC(CC)CN(C(=O)COC2(C)CCOCC2)CC)CN2CCN1CC2 70234,c1(C(N2CCOCC(NC(C)=O)C2)=O)cnc2[nH]ncc2c1 70235,C1(OC)(CNC(=O)CC2(C)CCN2C(=O)C(C)OCC(C)C)CCOC1 70236,N1(C(c2cc(CC)cc(Cl)n2)=O)CCC2(CCOCC2)C(NC(=O)C2CC2)C1 70237,C1(C(=O)NCC2CC(NC(c3ccnnc3O)=O)C2)OCC2CCCCC12 70238,C1(COC(C2CCS(=O)CC2)=O)CCCC(C(F)(F)F)C1 70239,C1(C(N2CC(CCCCNC(C(C3CCOC3)OC)=O)C2)=O)CN2CCC1CC2 70240,C1(CNC(CCC2CCC(=O)N2)=O)CC2(CC2)CN1C(c1nc(Cl)c(Cl)s1)=O 70241,C(=O)(C(F)(CNC(=O)C(CCC)N(C)C)C(C)C)NCCCCCC 70242,C1(C)(CC(=O)NCCN(C)C2CC2)CCN1C(=O)CC1CC(F)(F)C1 70243,c1(C(N(CCOCCCNC(C(C=C)O)=O)C)=O)c[nH]cc(C)c1=O 70244,Cc1cc(CC=O)cs1.C(=O)(CNC(C)(C)C)N(CCN(C)C)CC 70245,c1(CN2CCC(c3ccc(OC)cc3)C2)cc(Cl)ccc1N1CCOCC1 70246,N1(C(=O)C2=CCCSC2)CCC2(CCC(NC(C3CC(O)C3)=O)C2)C1 70247,N1(C(c2scc(CC)n2)=O)CCC(CO)C(O)C1.c12ccc(C)cc1[nH]c(=O)[nH]2 70248,c1(CC)ccc(OCCCC(=O)NC(C)C(C)(C)NC(=O)CN2CC(C)C2)cc1 70249,C=CCCCCCC(=O)N1CCN(C(c2ccc(C(F)(F)F)nn2)=O)C(C)C1C 70250,CCS(=O)CC(=O)NC1CC1NC(c1ccc(NC(=O)NC2CC2)nc1)=O 70251,C1(C2CCN(CC(=O)N(C)CC)C2)CCCCN1C(=O)CN1CCOCC1 70252,C(=O)(CC(CC(N)=O)c1ccc(F)cc1)N(CCCNC(C1COC(=O)O1)=O)C 70253,c1(C(=O)NC2CCC(C)(NC(c3cc(C)sn3)=O)CC2)ccnc2c1CCO2 70254,c1(C(=O)NCC2OCCN(C(c3cc(C(C)C)[nH]n3)=O)C2)ncccc1N=[N+]=[N-] 70255,C1(NC(CCCC(C)C)c2ccccc2)Cc2cccnc2C1 70256,c1(CCCC(=O)NCC(C)N(C(C(C)OCC2CC2)=O)C)cccc(Cl)c1 70257,C1(C(N(C2CCCN(CC3CCOCC3)CC2)C)=O)CC2CC2CC1C 70258,C(=O)(C(O)CC(C)(C)C)NCC(CCNC(CSc1ccc(C)cc1C)=O)O 70259,CCC(C)CCCCC(=O)NC1CC(C)N(C(c2ccc3oc(O)nc3n2)=O)C1 70260,C(c1ccc(OC)c(F)c1)=CC(=O)NCC1N(C(C(CC#C)O)=O)CC=C1 70261,c1(C(C)NC=O)ccc2ccn(C)c2c1.C(C)(C)(C)OC(=O)NC(C1CC1)C 70262,O=S(=O)(c1cc(F)cc(F)c1)Nc1ccc(Br)c(Cl)c1F 70263,c1(C(N(CC(C)NC(c2ccc(=NC)[nH]c2)=O)CC)=O)ccn2nnnc2c1 70264,C1(C(N(CCN(CC(COCCOC)O)C)C)=O)(OC)CCCCC1 70265,C1(NC(c2cccc(N(C)C)c2)=O)C2CCC1CN(C(C1CC(=O)N1)=O)C2 70266,C=C1CCN(C(=O)CC2CC2(C)C)C(C(=O)NC2CNC(=O)C2(C)C)C1 70267,c1(CSC)nc(-c2c[nH]ccc2=O)n(CC2CCCOC2)n1 70268,C(C(=O)NCCN1CCN(C(=O)C(=O)NCCC(N)=O)CC1)(C(C)(C)C)OC 70269,Cc1ncc(NC(=O)COC2(C)CN(C(C3C4CCCC(=O)C34)=O)C2)c(C)c1C 70270,c1(C(N2CC(OCCNC(CC3C(C)CCO3)=O)C2)=O)c(Cl)csc1Cl 70271,CN1CCCCC1C(=O)NC1(CNC(c2cccc(C3(C#N)CC3)c2)=O)CC1 70272,CC(C)CC(C(=O)N1C2CCCC1CC(NC(=O)Cc1cn(C)cn1)C2)C(C)C 70273,C1(C(=O)NCC(C)N(C(c2ccc(F)cc2F)=O)CC)CN(CP(C)(C)=O)C1 70274,N1(C(C(C)=CC)=O)C2CCC1C(CNC(=O)CCC(=O)NCc1ccccc1)C2 70275,c1(C(C)NC(=O)NC(C(=O)OC)C)cccc(F)c1 70276,C(C(CC(=O)NCC1CCC1C(=O)NC(C(C)C)C(C)C)C1CCC1)OC 70277,C#CCCCCCC(=O)NCc1cc(C(=O)NCC(C)C(C)CC)n[nH]1 70278,CCCCCC(C)CC(=O)NCC1CCCN1C(c1cnn(C)c1C(C)(F)F)=O 70279,C(CC1CC1)(CC(=O)NCC1CC1c1ccoc1)NC(C=C(CCC)C)=O 70280,CCC(CC(=O)NC1COCCOC1)NC(=O)C(C)C1(O)CCC1 70281,C#CCCC(C(=O)NC(CO)C(C)C)NC(=O)C(C)NC(C)(C)CC 70282,C1(C(=O)NCCC(=O)NC(CC)C)CCN(C(C2CC2Cl)=O)C12CC2 70283,C1(C(=O)NCC=CCNC(C2(CC=C)CCCC2)=O)Cc2nnc(C)n2C1 70284,C1(NC(CCOCC)=O)CCC(C(N2CCC2CF)=O)C1 70285,c1(C(N2CCC(N(C(=O)CCC(C)C#N)CC)CC2)=O)cc2n(n1)CCCC2O 70286,C1(NC(=O)C2=CCOC2)CCN(C(c2cc(C3CCC3)no2)=O)CC12CCC2 70287,c1(-c2cncc(NS(CCOC)(=O)=O)c2)ccc(F)c(NCC2CCCCO2)c1 70288,c1(C(N2CC(NC(c3cn(CCC)nc3C)=O)C2)=O)ccc([N+](=O)[O-])cc1F 70289,C12(C(=O)NCC(=C)CCNC(C3NC(=O)OC3C)=O)CCCCC(=O)N1CCC2 70290,N1(C(C(CC)n2nccc2C)=O)CCC(NC(c2cnc(C)cn2)=O)C(C)(C)C1 70291,Cc1cc(C(N2CC3CC(NC(c4nnc(O)cc4O)=O)C2C3)=O)c(C)cc1Cl 70292,C1(CNC(C2CC3CC3C2)=O)C2CCC1CN(C(c1c(F)cc(F)cc1F)=O)C2 70293,N1(C(C(C)c2cc[nH]n2)=O)CC(CNC(c2cc(C(N)=O)no2)=O)C2(CC2)C1 70294,C1(C)(C(N2CC(CC(NOCC(CC)C)=O)OCC2)=O)CC2C=CC1C2 70295,C12(CC(=O)N(CCCN(C)C)CC)CCC1CN(C(=O)CCc1cccn1C)C2 70296,c1(C(N(CC(O)CN(C)C(c2ccc(O)c(N)n2)=O)C)=O)ccc2c(c1)CC2 70297,CC#CCC(C(=O)N(CC(C)(CO)CO)C)NC(=O)CC(=O)OC 70298,c1(C(=O)NC2C=CCN(C(Cc3cc(C)ncc3)=O)C2)c(C)ccnc1O 70299,C1(CNC(CC(C(=C)C)OCC)=O)CC2CCC1N(C(C1(Cl)CC1)=O)C2 70300,c1(C(=O)NC2(COC)CN(C(=O)CN(C)C3CC3)C2)cccc2ccsc12 70301,N1(S(CC)(=O)=O)CCC2(CC(C(=O)Nc3cccc4c(O)cccc34)=NO2)C1 70302,C1(NCC2CCN(C(C)C)CC2)CC2CC(CNc3ccc(F)c(F)c3)CC12 70303,N1(C(CC(COC)C)=O)CCC2(CCCN2C(=O)CCc2nc(=N)[nH][nH]2)CC1 70304,c1(C(N(CCNC(CC2(COC)CC2)=O)C2CC2)=O)cnc2ncnc(O)c2c1 70305,C(=O)(C1CCCn2c(C)nnc21)N(CCN(C(C#CC1(CC)CC1)=O)C(C)C)C 70306,N1(C(C(CC)NC(N)=O)=O)Cc2occ(C(=O)NC(C)C(C)(C)CN(C)C)c2C1 70307,Cc1nc(N(C2C3CNCC23)C)c2sccc2n1 70308,Cc1ccc(F)c(C(=O)NC(Cc2cc[nH]n2)C(=O)NCc2ccc[n+]([O-])c2)n1 70309,C12(NC(CCSC)=O)CN(C(c3nc(C)n(C)c3C)=O)C(COC)(C1)C2 70310,c1(C(=O)NC2CCCC(N(C(CN3CC(CC)C3)=O)C)C2)cn2nc(C)sc2n1 70311,C1(CC)COCCN1CCn1cc(C(=O)N(C)CC)nn1.C12CCC(O1)C(=O)N2 70312,C1(C(N2CC3C(CNC(C4CCCC4)=O)(C3)C2)=O)CCN(CCO)C(=O)C1 70313,CCC(CC(=O)NCC(C)(C)C#CC(=O)N(C1CCCC2(C1)N=N2)CC)C(F)F 70314,CCCCCCCCCC(=O)NCC1CN(C(=O)C2=NNC(=O)CC2)CCO1 70315,c1(N2CCCC(CC(C)(C)C)C2)nc(=N)[nH]c(=NCc2nccs2)[nH]1.C1(N)CCC1 70316,C(C(COC)CC(=O)NCCCC(=O)NCC1COCC1O)OC 70317,c1(C(=O)NC(CC)CN(C(=O)C(O)C2CCCC2)C)ncn(-c2ccccc2)n1 70318,C1(C2CCCO2)(C(=O)Nc2ncc(C#C)cn2)CCCO1 70319,C(=O)(C(C)(C)C(C)O)N1CCCC(CN(C(c2c(C)oc(Cl)n2)=O)C)C1 70320,c1(C(=O)NCC(C)N(C(C2(SC)CC2)=O)C)cc(C)c2[nH]nnc2c1 70321,Cc1nc(CC(=O)NCC2CCCN2C(=O)C(c2ccnn2C)C)sc1C 70322,C1(C2CC2)(C(=O)NC2CC(CCNC(C34C=CC(CC3)C4)=O)C2)CCOCC1 70323,c1(CN(C(C)(C)C)Cc2nnnn2C)cccc(C(N)=O)c1.C(C(F)(F)F)S 70324,Cc1ccc(F)c(CC(=O)NC2(CCCNC(C3CC4CC3CC4O)=O)CC2)c1 70325,C1(CNC(C(C=C)O)=O)CCCC2CN(C(=O)CCCCC(=O)NC)CC12 70326,c1(C(N2C(CNC(CC(CCC)(C)O)=O)CC2)=O)cc(F)cc2nccnc12 70327,C1(NC(c2c(C)cc(C)[nH]2)=O)CS(=O)(=O)CC1NC(=O)CCC1CCCCC1 70328,C#CCC(C(=O)NC1(C)CCN(CCCCC)C1)NC(=O)CCCNC(C)=O 70329,C1(NC(C(CSC)O)=O)CN(C(c2ccc3ncncc3c2)=O)CC1S(C)(=O)=O 70330,C(=O)(C(O)C(F)(F)F)NCCSCC(=O)NCCc1csnn1 70331,c1(C(N(C(CN(C(C(COCC)C)=O)C)C)C)=O)cc2n(n1)CCCC2 70332,N1(C(C2CCN(C(c3cc(OC)ncc3Br)=O)C2)=O)CCc2cccc(F)c2C1 70333,C(CN=c1[nH]c(Cl)ncc1C)C1CC(NC(C2(CC)CCNC2=O)=O)C1 70334,C=CCC(C(=O)NCC1CC(F)(F)CN1C(=O)Cc1cc(F)ccc1Cl)C(C)C 70335,c1(C(=O)NCCCN(C)C(C2CC(O)(C(F)(F)F)C2)=O)ncn2c1CCCC2 70336,C1(NC(CCc2cnc(C)nc2O)=O)CN(C(=O)Cn2ncnn2)CC1C1CC1 70337,N1(CC(=O)NC(=O)NC)CCC(C2CN(C(c3cccnc3)=O)C2)C1 70338,N1(C(=O)C(F)C2CC2)CCN(C(=O)CCCn2ccnn2)C(CC2CCOCC2)C1 70339,Cc1cc(C(N2CCCC(N(C)C(c3cc(O)nc(O)n3)=O)CC2)=O)cnc1O 70340,N1(C(=O)CC2(O)CC2)CCC2C(C1)CN2C(C1CCOCC1)=O 70341,c1(CC(=O)NC2CCCC(NC(COCCC#C)=O)C2)noc2ccc(F)cc12 70342,Cc1nc(C(N2CCC(C(C)NC(=O)CCCc3cccnc3)C2)=O)c(C)s1 70343,N1(C(c2c(F)cccc2Cl)=O)CCC2C(CCN2C(=O)CCCCCO)C1 70344,C=CCC(C)C(=O)N(C1CCC(NC(C2(OC)CCOCC2)=O)CC1)C 70345,c1(N(CC(=O)NC2(CO)CN(C(C3C4CCCC34)=O)C2)C)ccc(Cl)cn1 70346,C1(C2CC2)(CNC(c2c(C(C)C)ccs2)=O)CCN(C(=O)C(O)C2CCC2)C1 70347,N1(C(C23N(C(CN(C)C)=O)CCC2CCC3)=O)CCC2(CCCCC2)C1 70348,c1(CC(=O)NCCCN(C(=O)C(O)c2ccco2)CC)cncnc1 70349,C1(CCNC(C2CC23CCCC3)=O)CCCN(C(C2(F)CC2)=O)C1 70350,CC1C(=O)NC(=O)CN1C(C1(C)CN(C(c2cc([N+](=O)[O-])n[nH]2)=O)C(C)(C)C1)=O 70351,Cc1nn(C)c(CNC2CC(N(C)C)C2)c1S(N)(=O)=O 70352,CCC(CO)C(=O)N1CCC(n2cc(CNC(=O)Cn3nccn3)nn2)CC1 70353,C1(CC)CCN(C(C2CC23CCC3)=O)C1C(=O)NCC(=O)NC(C)C 70354,CC(CC=Cc1ccccc1)C(=O)N1CCC(NC(C2OCCO2)=O)C1 70355,C(C)(CCCC(=O)NCC1OCC2CCC1C2)NC(C(C)(C)NC(C)=O)=O 70356,C12(NC(c3ccc(F)c(O)c3)=O)CCOCC1CN(C(C1(Cl)CC1)=O)C2 70357,C(=O)(C1CCCn2ccnc21)N1CCCC(O)(CNC(CCCS(N)(=O)=O)=O)C1 70358,c1(C(N2CCC(O)(CNC(C(C)NS(CC)(=O)=O)=O)C2)=O)ccc2c(n1)CCO2 70359,C(CCC(=O)NCC(N1CCC(OCCOC)C1)=O)NC(COCC)=O 70360,C(c1ccc(C(C(=O)N(CCCN(C(C(C)CO)=O)C)C)=O)cc1)=CC(=O)NC 70361,CC(CNC(C1(C)CCN(C)C1)=O)CC(=O)NCCCC(F)(F)F 70362,C1(NC(CCC(=O)NC)=O)CC(O)CN(C(=O)CCCNC(N)=O)C1 70363,c1(C(=O)NC2C(N(C(=O)CCC3CCOC3)C)CCCC2)cccc2nc[nH]c12 70364,c1(C(=O)Nc2scc(-c3c(C)ccs3)n2)cc(F)c(F)c(Cl)c1 70365,C1(CCC(=O)NC2CC(C)OCC2)CCCCN(C(C2(O)CCOC2(C)C)=O)C1 70366,C1(NC(C2(OC)CC2)=O)CC2C(NC(=O)C(c3ccccc3)C)C2C1 70367,N1(C(C(CC)NC)=O)CC2CN(C(c3cnc(Cl)c(C)c3)=O)CC12 70368,Cn1nnc2c1CCC(C(=O)NC1CCC13CCN(C(=O)C(C)(C)CF)CC3)C2 70369,N1(C(C(CCC)(C)O)=O)C2CCC1C(C)C(NC(C1CCC(C(C)C)CC1)=O)C2 70370,c1(NC(N2CC(CCN3CCOC3=O)C2)=O)cc(Cl)ccc1I 70371,N1(CC)CCCCC1C(=O)NCCCC(=O)N(CCCC(C)O)C 70372,CC(C)CC(CNC(C1CC2CC2N1C(C12CCC(CC1=O)C2)=O)=O)CO 70373,C1(OC)CC1C1CCCN(C(=O)Cc2cc(C(F)(F)F)n[nH]2)C1 70374,C1(NC(COCC(=O)OC)=O)CN(C(c2cn(C3CC3)nn2)=O)C(C)(C)C1 70375,C(=O)(CS(=O)(=O)c1ccccc1F)N1CCC(NC(C2CCC(O)C2)=O)(CO)C1 70376,CCCC(O)C(=O)NC1CN(C(=O)C(c2ccc(F)cc2)(C)C)CC1OC 70377,Nc1cc(C(=O)NCCOC2CN(C(=O)CCc3ccncn3)C2)cc(Cl)n1 70378,C1(C(N2CCCC(Cn3ccnn3)C2)=O)Cc2ccc(O)cc2CN1 70379,C#CCC(CC#C)C(=O)N1CCC(C(F)CNC(=O)C(F)n2cccn2)CC1 70380,c1(C(=O)NCCN(CC(=O)NC2CC2)C2CC2)ccoc1I 70381,c1(CN2CCN(C3CCN(C(C4CC5(CC5)CO4)=O)C3)CC2)cc(Cl)cc(Cl)c1 70382,C12(CC)CCC(C(=O)NCC(CC(F)(F)F)NC(=O)Cc3ccno3)(CO1)C2 70383,c1(C(N2C(CCCNC(CN(C(C)=O)C)=O)CCC2)=O)cc(C(F)F)ccn1 70384,C#Cc1ccc(F)cc1C(=O)NC1CN(C(=O)CC(C)F)CC1n1cccn1 70385,C(=O)(C(C)C(CC)CC)N1C(C(=O)NCC(=C)Br)CC(=O)C1 70386,c1(C(=O)NCC(CN(C(COCC)=O)C)O)cc2sccc2n1CC1CC1 70387,C(CNC(c1cnc(C#N)s1)=O)(C(C)(C)C)NC(C1(COC)CC1)=O 70388,C=C(C)C(C)(C)C(=O)NC1CN(C(=O)C(=O)NCC2CC2)CCC1CO 70389,c1(C(=O)NC2(CCNC(CCC#CC)=O)CCC2)ccc2ccnc(Cl)c2n1 70390,c1(C(N2CCN(C(c3c(OC)c(Cl)sc3)=O)CC2)=O)n[nH]c2c1CCC2 70391,C#CCC(C)(C)C(=O)N1CC(C(=O)Nc2cncc(N(C)C)c2)C(C(C)C)C1 70392,C(=O)(CCCCCn1cc(CCCO)nn1)NC(C)CC(N1CCC(C#N)C1)=O 70393,C1(C(=O)NC2C(NC(c3c(Cl)cn(CCC)n3)=O)CCC2)CCc2nncn2C1 70394,C1(CNC(CCCN(C(C)=O)C)=O)CC(C(=O)N(C)Cc2ccncc2F)=NO1 70395,c1(C(N2CC3C(CNC(CC(=C=C)C)=O)C3C2)=O)cc[nH]c2nccc1-2 70396,CC(C)C1=NOC(C(N2CCC(C(C)NC(C3CC(=O)C3)=O)C2)=O)C1 70397,C=C=CCCC(=O)NCCC1CCC(NC(=O)CCS(C)=O)C1 70398,C1(NC(CNC(C=C)=O)=O)CN(CC2CCC(=O)NC2)CC1C#N 70399,C1(NC(C=CC(C)(C)SC)=O)CCCC1NC(=O)C(C)CC1CC1 70400,N1(C(c2cc(C)ncc2)=O)CCC2CC2(C(N2CCC(OC(C)C)CC2)=O)CC1 70401,c1(N(CCSC)C)ncnc2c1ncn2CC(c1ccccc1)(C)O 70402,c1(CC(=O)NCCC(CCNC(C(C)NC(=O)NC)=O)C)c(C)nn(C(F)F)c1C 70403,N1(C(COCC(C)(C)O)=O)CCCC(C2CCN(C(=O)COC(F)(F)F)CC2)C1 70404,c1(C(=O)NC2(CNC(CCCOCC=C)=O)CCCC2)ccc(OCC)c(F)c1 70405,c1(OC)ccccc1NC(=O)C(C(C)C)N1CCN(S(=O)(=O)C(C)C)CC1 70406,C(=O)(C(O)C(C)(C)C)N1CC(C)C(CNC(C2(C)CC(O)CN2C)=O)C1 70407,C1(NC(c2cc3ncccc3o2)=O)CC2CC1CN(C(c1cc(Cl)sc1Cl)=O)C2 70408,N1(C(C2C(C)=CCS2)=O)CC2(CC(C(=O)NC3COC(C(C)C)C3)CO2)C1 70409,c1(C(C)O)ccc(C(N2CCCC2CNC(c2coc(Cl)n2)=O)=O)cc1 70410,C(CC(=O)NC1CCC12CCCC2)(C(C)OC)NC(C(COC)(C)C)=O 70411,C1(F)(NC(C2(OC(C)=O)CCC2)=O)CCCN(C(=O)CCOC2COC2)C1 70412,C(=O)(CCCCCN(C)C)NC(CNC(C1(C#C)CC(=O)C1)=O)CC=C 70413,c1(OC)cc(C)cnc1C(N1CCC(O)(CCNC(C2C(C)C2C)=O)CC1)=O 70414,CC1(C)C(=O)NCC1NC(C1CC1NC(c1cccc(O)c1O)=O)=O 70415,C(=O)(CCC(=O)NC1CCC1NC(c1cccc(F)c1)=O)N(CCC)CCC 70416,C1(CC)CCCC(C(=O)NCC2CCC(C(=O)NCC3(CC(C)C)CC3)C2)C1 70417,C(=O)(CCCCNC(c1snc(C)c1N)=O)NCC(C(=O)NC)C 70418,N1(C(C(CC(C)C)N(C)C)=O)CCC2(CC(C(N3CC(O)CC3(C)CO)=O)C2)C1 70419,N1(C(c2cncc(NC)c2)=O)CC(O)C(O)C1CNC(C1CC1OC)=O 70420,N1(C(C=C(C)C2CC2)=O)CCN(C(C2CC3CC23)=O)CC1 70421,C(=O)(C(C(C)(C)C)SC)NCC1CN(C(c2c(COC)ncs2)=O)C1 70422,C(=O)(C(CO)C(C)(C)C)NC(C(N1CC(C(C)C)N(C)CC1)=O)CCC#N 70423,CCCCS(=O)(=O)NCC(=O)NC1CCCC1NC(C1CCN1CC)=O 70424,C1(NC(=O)NCC(CC2CC2)OC)CC2CC1CC2(C)OC 70425,c1(CCC)ccc(C(N2CCCC2C(N2CCCC2)=O)=O)cc1S(N)(=O)=O 70426,C1(C(=O)NCCOC2CN(C(CCc3cnc(C)s3)=O)C2)CN(C)CCO1 70427,C=CCC(F)(F)CNC(C1(CO)CCN(C(c2ccc(CC)[nH]2)=O)C1)=O 70428,N1(C(c2ccc(Cc3cn(CCC(F)(F)Cl)nn3)o2)=O)CC2CN2C=NC=CC1 70429,Cc1cc(C(=O)NC(CO)C(C)NC(C2(C3CCCCO3)CCC2)=O)nn1C 70430,c1(C(N2CC(CNC(c3c(OC)ccs3)=O)C(C)(C)C2)=O)ccc2snnc2c1 70431,C1(NC(C2N(C(C)=O)CCC2)=O)CC(C(=O)NCc2c[nH]nc2C)=CC1O 70432,CC1(C)CNCC1OCC(=O)N(CC(c1ccccc1)CO)CCO 70433,C1(NC(c2c(C)cc(CNC(C(C)=CC3CC3)=O)o2)=O)CCCC1C1CC1 70434,C1(CC(=O)N(c2ccccc2)C(CC)C)CCCN(C(=O)Cn2nnnc2C)CC1 70435,c1(NC(N(CCC(C)C)CCO)=O)cnc(-c2ccncc2)s1 70436,c1(NC(CC2CCN(Cc3c(CN)cccc3)C2)=O)cc(F)c(F)cc1Cl 70437,c1(CN(C(=O)C(N2CCCCC2c2nnc(C)o2)=O)CCOC)ccc(F)cc1F 70438,C1(NC(CCN(C(COCCCC#C)=O)CC2CC2)=O)CCN2CCCC2C1 70439,C(=O)(CC(C)C(F)F)NC1CN(C(c2nc(C)oc2C)=O)CC1C 70440,Cc1cc(C(=O)NC2CCCCC2NC(c2cccs2)=O)nn1CC(F)(F)F 70441,c1(NC(CN(C(=O)C(N2CCOCC2)C)CC#C)=O)cnc(C)c(C#N)c1 70442,C1(CC)CCN(C(C2CCC2COC)=O)C(C(=O)NC2C(O)CC2O)C1 70443,n1(CC(N2CC(CNC(COc3cccc(C)c3)=O)C2)=O)cc(P(C)(C)=O)cn1 70444,c1(CC)c(C(N2CCN(C(=O)Cc3cc(C4CC4)no3)C3CC23)=O)cccc1C 70445,N1(C(CC2(C#N)CC2)=O)C2CCC1CN(C(C1Cc3cccnc3C1)=O)C2 70446,CC1(C)OC2CC(C(=O)NC3(CNC(C4OCC5CCCCC45)=O)CC3)CC2O1 70447,Cc1ccc(-c2cc(-c3nccn3C3CCSC3)nn2C)c(C)n1 70448,n1(CC(N2C(C)CC(CNC(=O)CSC3CC3)C2)=O)ccc(O)nc1=O 70449,c1(OC)cc(O)nc(NC(C2CCN2C(c2ccc(NC(C)C)cc2)=O)=O)n1 70450,C1(C(=O)NC2C(N(C)C)CN(C(CCCCCSC)=O)C2)CC1C1CCCCC1 70451,N1(C(C(CC#C)O)=O)CCC(C2CCC2)(CNC(=O)C(C(C)C)OC)CC1 70452,C1(CNC(c2ccc(C(F)(F)F)[nH]2)=O)CN(C(C2CSC2)=O)C2CC12 70453,N1(C(c2c(N)ccc(Cl)c2)=O)CCCN(C(C2(CO)CC2(F)F)=O)CC1CO 70454,c1(C(=O)NC(C2(O)CCN(C(=O)C=C3CCN(C)C3)C2)C)cccc(C2CC2)c1 70455,CC(O)C(F)(F)C(=O)NC1CC(C)(CNC(=O)CCc2ccccc2F)C1 70456,C1(CC(=O)N(C(C)CNC(C2CCC(N(C)C)CC2)=O)CC)CCS(=O)(=O)C1 70457,c1(C(=O)NCCN(C(=O)CC2CC(F)C2)C)cn(C)cc1C(F)(F)F 70458,c1(C(N2CCC(C)(NC(c3ccc(CCC)[nH]3)=O)C2)=O)ccc(F)c(F)c1F 70459,Cc1cc(CC(=O)NC2CCCC(NC(=O)CCOCC(C)C)C2)cc(C)c1 70460,c1(CCC)nc(C)c(C(N2CCC(NC(C3CC3C)=O)C2C)=O)s1 70461,c1(C(=O)OCC2CC3(CCC3)C2)ccc([N+](=O)[O-])c(O)c1 70462,Cc1c(Br)ccc(O)c1C(N1CC(NC(=O)CCC2CCC(C)O2)C1)=O 70463,C1(CC)CC(C(N2CCC(F)(CNC(c3cc(F)n(C)n3)=O)C2)=O)CC(=O)N1 70464,O=C(C(O)CC1CC1)NC1CC(F)(CNC(c2csc(Br)n2)=O)C1 70465,C1(C)(CNC(C2(OC)CC2)=O)CCC(NC(c2cc(CCO)on2)=O)C1 70466,C(=O)(CCS(C)=O)N1CC(C(C)NC(=O)C(C)(C)N2CCOCC2)C1 70467,C1(NC(=O)CC2CCCC2)CCCC12CCN(C(=O)CC1CC3(CC3)CO1)CC2 70468,C1(NC(c2cc(O)nc(C3CC3)n2)=O)CC2CN(c3cc(Cl)ncn3)CC2C1 70469,N1(C(CNC(=O)NC)=O)CCN(C(=O)CC(C)(C)C2CC2)C(CO)C1 70470,C1(CC#C)(C(=O)N(C)CCN(C(=O)CCOCC2CCC2)C)CCOC1 70471,C1(C(=O)NCCC(C)NC(=O)CNC(=O)N(C)CC2CCCC2)CCCCN1C 70472,N1(C(=O)C=Cc2ccco2)CC23CCCC2(C1)CN(C(c1cc[n+]([O-])cc1)=O)C3 70473,C1(NC(C2(F)C(C)C2)=O)CCC(C)N(C(=O)Cc2ccc(C(F)F)cc2)C1 70474,CC(C)C(C)C(CNC(C1CCC1)=O)NC(c1ccc(CCCN)cc1)=O 70475,c1(SC)cc(C)ccc1C(=O)NCC1(O)CCN(C(c2nn(C)cc2C)=O)C1 70476,C1(CNC(C2CN(C(C)=O)C2)=O)CC(NC(c2n[nH]cc2Br)=O)C1(C)C 70477,c1(CN2CC(CC(N3CCS(=O)(=O)CC3)=O)C2)ncccc1[N+](=O)[O-] 70478,C(C1c2ccccc2CCN1C(C1C(C)C1)=O)N(c1cccnn1)C(C1CC1F)=O 70479,c1(OC)cccnc1C(N1CCCC(CN2CCCCC2)C1)C(=O)NCCC#N 70480,c1(C(=O)NCCCN(C(c2nccs2)=O)CC)ccncc1OCC(F)(F)F 70481,N1(Cc2cn(CCC(C(=O)OCC)C)nn2)CCC12CCSCC2 70482,C1(NC(c2ccc(S)cc2)=O)CN(S(=O)(=O)c2cccs2)CC1(F)F 70483,c1(CC(=O)NCCCC(C(=O)N2C(C(=O)NC)C=CC2)O)csc2nc(C)cn12 70484,c1(N(C(=O)CC2CCN(C(=O)Cn3cnnn3)CC2)C)ccccc1Cl 70485,C1(C(=O)NCC2CCN2C(=O)CSC(F)(F)F)CCCC1C(F)(F)F 70486,c1(C(=O)NC2CN(C(C#CC3(CC)CC3)=O)CC2O)cc2n(n1)CC(F)C2 70487,CC1CC(c2nnnn2CC2CCOC2)(NCC(C)(C)CO)CC(C)O1 70488,N1(C(c2c(C)n(C)cn2)=O)CC(C(=O)NCc2cnn(C)c2O)CC1(C)C 70489,C(C#Cc1cccnc1)NC(C1CCN(C(c2cccn3cncc23)=O)C1)=O 70490,N1(C(C(=O)NCCN(C(C2CC(OC)C2)=O)CC)C)CCCC(O)C1 70491,c1(CCC(=O)NC2C(NC(CCNC(=O)NC)=O)C2)cc(C)on1 70492,N=c1ncn(CC(=O)NCC2(C(=O)NCc3nc(C4CC4)no3)CCCO2)[nH]1 70493,C(C1=CCN(C(=O)CC2CCCS(=O)(=O)C2)CC1)NC(CC1CCC(C)CC1)=O 70494,N1(C(=O)OC(C)(C)C)CCC(C(=O)N(C2CCC2)CC2CC2)C1 70495,C1(C)CCC2CC2C1.C1(N(C(C2C(C(=O)OCC)C2)=O)CC)CCN(C=O)C1 70496,C1(C(N2C(C(=O)OC)C=CCC2)=O)CCN(C(=O)CC(C)(C)SC)C(C)(C)C1 70497,N1(CC(=O)NC(C2CN(C(C3CCOC(=O)CC3)=O)CCO2)C)CCSC(C)(C)C1 70498,C1(CNC(c2c(C)nsc2)=O)CCCCN(C(=O)CCc2ccccc2)C1 70499,N(C1CCCn2nccc21)C(C1(C=C)CCN(C(c2n[nH]c(C)c2O)=O)C1)=O 70500,Cc1ccc(C(C)CC(=O)NC(C)C(C)(C)NC(c2ccsn2)=O)cc1 70501,c1(OC)ccc(C(C)C(=O)NC(C)COc2ccc(F)cc2)cc1F 70502,c1(OC)ccc(C(N2CCCCC2COCC2CC2)C(=O)NC(C)C)cc1OC 70503,c1(C(N(C2CCN(C(C3(C#N)CC3C)=O)CC2)CC)=O)cc2ccsc2s1 70504,CCC(CC(=O)NC(C(=O)N(C1CCCC1C#N)C)C(C)O)C(F)F 70505,C12(C(=O)NCC(C)(C)O)CC(CN(C(C3C4CCC(F)C34)=O)C1)C2 70506,C1(C(=O)NCc2cc(C)c(C(=O)NC3(C4CC4)CCCC3)o2)CCCC(C#N)C1 70507,N1(C(c2c(CC)cco2)=O)CCCN(CCNC(=O)Cn2cncn2)CC1 70508,Cc1c(C(=O)NCC2CC(NC(C34CC(C)(C3)C4)=O)C2(C)C)cccc1O 70509,C#CC(C)(C)C(=O)NCc1nc(C(=O)NC(C)CC)c(C)o1 70510,C(C)(CN=c1nc(C#N)[nH]cc1C)(C(C)C)NC(c1c(C)nc2ncnn2c1C)=O 70511,C#CC1(NC(=O)C(C)(C)CN(C)C(c2ccc(C(N)=O)o2)=O)CCOC1 70512,N1(C(=O)COC2CCOC2)CCCC(C2CCCN(C(c3ccc[n+]([O-])c3)=O)C2)C1 70513,C1(NC(CN(C)S(N)=O)=O)CCCC12CN(C(=O)CCn1cc[nH]c(=O)c1=O)C2 70514,c1(C(=O)Nc2nc(-c3c(F)cccc3F)cs2)cc(F)c(Br)c(F)c1 70515,C(=O)(C(C)CC(C)C(C)=O)NCCn1cc(C(N2C(C)(CCC)CC2)=O)nn1 70516,C1(CC(=O)NC2C(CNC(C(COCC)(C)C)=O)CCCC2)CC2CCC1CC2 70517,c1(C(N(C(CNC(c2cc(C)cc(C)n2)=O)C2CC2)C)=O)ccc2[nH]ccc2n1 70518,N1(C(C(COC)(C)C)=O)CCC2(CC1)OCCCC2NC(=O)CSS(C)(=O)=O 70519,c1(CN(C)C)ccc(C(N2CCC2CNC(c2csc(=N)[nH]2)=O)=O)[nH]1 70520,C#CCC(C)C(=O)N1CCC(C(C)NC(c2ccc(C3(C)CCO3)cc2)=O)CC1 70521,c1(C(C(C)C)NC(CCc2cn(CC)nc2C)=O)ccc2ncccc2c1 70522,N1(C(C2N(CCC)CCCC2)=O)CCC(F)(CNC(=O)CC(C)(C)O)CC1 70523,C12CCC(C1)NC2=O.c1(C(=O)NCCNC(C2(Br)CC2)=O)ccco1 70524,c1(C(N(C)CC2CN(C(c3ccn(C)n3)=O)CCO2)=O)ccc(C2CC2)c(Cl)c1 70525,C(C)(C)(C=CC(=O)NC1(CC(=O)NCC(C)SC)CCC1)SC 70526,C(CCC(C)CCC)c1nc(-c2ccc(OCC)cn2)on1 70527,c1(CC)nn(C)cc1C(N1CC(C(O)C(N2CCCC(C(N)=O)C2)=O)C1)=O 70528,C1(C(N2C(CNC(c3n(C)cc(C#N)c3)=O)CC(F)C2)=O)CNC(=O)C(C)(C)C1 70529,C(C(=O)N1CC(NC(=O)Cc2ccc(C(N)=O)nc2)C(C)C1)(C(C)C)OCC 70530,c1(-c2nc(C(C)SC)nn2C(c2cncc(F)c2)C)cc2c(OC)cccc2[nH]1 70531,C1(NC(c2c(C)ocn2)=O)CN(C(=O)C(C)OCC(C)C)CCC1F 70532,C(CCCCC(=O)NCCOCCNC(C1CCC(N(C)C)C1)=O)SC 70533,Cc1nn(C)c(N)c1C(=O)NCC(C)NC(c1cccc(C(N)=O)c1C)=O 70534,CC(C)C(C(=O)NC1C=CCN(C(=O)CCSc2ccccn2)C1)NC(N)=O 70535,C#CC1(NC(=O)CCOCCN(C(=O)C2=NOCC2)C)CCOC1.OCC 70536,CCCCC(CNC(c1ccc(F)s1)=O)NC(=O)C(O)C1CCC1 70537,N1(C(c2c(C(C)C)ncs2)=O)CCC12CN(C(C1CCCCN1C)=O)C2 70538,Cc1c(C(=O)NCC2COC(C)(C)CN2C(=O)C=CC2CCC2)nc2sccn12 70539,c1(CCCNC(CN(CCOC)C(C2C=CCS2)=O)=O)nc[nH]n1 70540,n1(C(CC)C)nc(C(=O)NCCC(C)(C)NC(C2CC3C=CC2O3)=O)cc1C 70541,N1(C(c2cc(C)no2)=O)Cc2ccc(O)cc2CC1C(N1CC(F)CC1C#N)=O 70542,C1(CNC(c2cc(Br)cnc2O)=O)CCN(C(=O)NC(=O)C(Cl)(Cl)Cl)CC1(F)F 70543,c1(C(N2CC(NC(C3C(C)CC(C)O3)=O)(CO)C2)=O)ccc(S(=O)(=O)C(F)F)cc1 70544,N1(CC)CC(C(=O)N(CC(C)(C)NC(=O)C=Cc2cncc(O)c2)C)CCC1=O 70545,C(C)(CCS(C)(=O)=O)(c1n(CCSC)nnn1)NCC1(C)COC1 70546,CC(C)CC(C)C(=O)N(C1CN(C(=O)CC2COCC2(C)C)C1)C 70547,C1(NC(c2cn(C)nc2O)=O)CC(NC(=O)CC2(c3ccon3)CC2)C12CCC2 70548,Cc1cc(C)c(NC(=O)CC23CCC2CN(C(=O)C2=CCCCO2)C3)c(C)n1 70549,c1(C(N2CCCC(OC3CC3)C2)C(=O)NCC)nc(Br)ccc1OCC(C)C 70550,C(=O)(CC(P(C)(C)=O)P(C)(C)=O)N(C(CNC(C(CCC)O)=O)C)C 70551,c1(C(N2C(C)CCC(CNC(=O)CCC(C)(C)C)C2)=O)ccc2n[nH]cc2c1 70552,c1(C(=O)NCC(CC)N)ccc(C(N)=O)o1.c1(C(N2CC(C)C2)=O)ccn(CC)n1 70553,C(CC)(CCC(=O)N(c1ccc(OC)cc1)C)NC(C(CC)CC)=O 70554,C12(NC(c3cc4n(n3)CC(F)C4)=O)CCCC1CN(C(c1cc(O)cs1)=O)C2 70555,C=CCC(C)C(=O)N(C(C)(C)CC(=O)N1CC(F)C(F)C1)C 70556,c1(C(=O)NC2CCN(C(c3ccc(OC)s3)=O)CC2F)ccc2nc(O)sc2c1 70557,Nc1ccc(C(=O)NCC(CO)NC(C2CCCN2C=O)=O)c(Cl)c1 70558,c1(CNC(C(=O)NCC)=O)cccc(CNC(C2CCC(F)C2)=O)c1 70559,N1(C(C=Cc2cn(C)nc2)=O)CC2COCCC2(NC(=O)C(F)=C2CCCC2)C1 70560,C1(CNC(C2(CC#C)CCC2)=O)CCN(C(=O)CN2CCCCC2C)CC1 70561,c1(C(=O)NC(C2CCOC2)CNC(C(C)=C2CC2)=O)ccc(CO)nc1 70562,CCCC(O)C(=O)N1CCC(OCCNC(c2coc(C#N)c2)=O)C1 70563,c1(C(N(C(CC(=O)NCC(CC=C)(C)C)(C)C)C)=O)cc(F)cnc1O 70564,c1(CNC2CCN(c3c(C(=O)O)ccs3)C2=O)noc2cc(Br)ccc12 70565,C(C(C)N=c1nc(OC)cc(OC)[nH]1)NC(CCC(=O)NC)=O 70566,CC(C)C(C(=O)N1CC(NC(=O)CSC(F)(F)F)C(C)C1)NS(=O)(=O)C1CC1 70567,CC1CN(C(C2CC(C)(C)CO2)=O)CC1C(=O)NC1C=CCC1 70568,C1(NC(c2ccn(CC)c2C)=O)CN(C(C23CCCC2C3)=O)C2(CCCCC2)C1 70569,C(CC(C(=O)NCC1CCCCO1)NC(=O)CC1CCC(=O)C1C)OC 70570,C(CCCC(=O)NC(CNC(=O)CCN1CCC(F)C1)(CC)CC)OCCC=C 70571,C=C=C(C)CC(=O)NC(C1CCCN1C(=O)CCSc1nccn1C)C 70572,C(=O)(C1=CCCCO1)N(C1CCCN(C(C2(CC=C)CCOC2)=O)C1)CC 70573,N1(C(CCCOCCOCC)=O)CCN(C(=O)CN2CSCCSC2)C2CCC12 70574,C1(CC=C)(NC(C2CCCO2)=O)CN(C(C2CC(C)(O)C2)=O)C1 70575,c1(OC)ccc(C(C)NC(=O)NC(C)C(c2ccc(F)cc2)O)cc1C 70576,N#CC1CN(CCN(C(=O)CC23CC(C2)C3)Cc2ccncc2)CC12CCC2 70577,C1(NC(C2CC(NC(c3ccoc3)=O)C2)=O)CCCC(O)CC1 70578,CC(C)(CCCO)CN=c1[nH]c(=NCc2ccc(C(F)(F)F)s2)c2sccc2[nH]1 70579,c1(C(N(CCCCCNC(c2nc(=O)n(C)[nH]2)=O)C)=O)[nH]c2ccccc2c1Cl 70580,CCCC(C(=O)NC(C1CN(C(c2coc(C#N)c2)=O)C1)C)S(N)(=O)=O 70581,c1(CN(C(C2CCC(C)(C(=O)OC)N2)=O)CC)cc(Br)ccc1C 70582,c1(OC)cc(C)cnc1C(=O)NC(C(C)NC(c1cn(C2CC2)cn1)=O)C(C)C 70583,N1(C(C=C(C)C)=O)CCC2CN(Cc3c(C)cccc3Br)CC12 70584,Cn1cnc2ccc(C(=O)NCC3CC4CCC3N4C(c3cc(Cl)on3)=O)nc12 70585,Cn1ncc2c(NC3CCN(C4CCCC4)CC3)[nH]c(=NCCc3nc[nH]n3)nc12 70586,CP(C)(=O)c1ccc(C(=O)NCC(C2CCC2)NC(c2ncccc2F)=O)cc1 70587,CC(C)(CNC(C1CC2CC1CC2O)=O)CC(=O)NCCC1(CO)CC1 70588,N1(C(C=CCNC(=O)CCC2OCCO2)=O)CC(O)CC12CCC2 70589,N1(C(CC2CN(C)CC2O)=O)CC(NC(c2ccoc2Cl)=O)C(C)(C)C1 70590,C(=O)(CC(=O)NCC(c1ccccc1)NC(C1CCOC1C(C)C)=O)NCC 70591,C1(C(N2C3(C(N4CCC(O)(C(C)C)C4)=O)CC3CC2)=O)C2CCC(C2)C1C 70592,c1(C(=O)NC2CC(CCC(=O)NC3(CCCC)CC3)C2)cnc(C)n1C 70593,Cc1c[nH]c(C(=O)NCC2CCC2C(=O)NCCC2CCCN(C)C2)c1C 70594,N1(C(C(=O)NC2C(NC(CCCC)=O)COC2)CC)C(=O)CCC1=O 70595,N1(C(C(C)N(C(C2CC(=O)CC(=O)C2)=O)CC)=O)CC(C)CCCC1C 70596,C=CCC(CNC(=O)C(C)(C)N(C)C)NC(=O)C(C)=C1CC1 70597,C(C(C)C(=O)NCCNC(N)=O)N(C(C(C)SCC)=O)C 70598,c1(C(=O)NC2C(CNC(CCC#CC)=O)C2)cc(F)cc(Br)c1F 70599,C1(C(N(CCN(C(c2ccsc2)=O)CC)CC)=O)CC2(C1)CC(F)(F)C2 70600,c1(C(=O)NC2CCC2)ccccc1F.C(C1(C)CN1)NC(C1(C(=O)NC)CC1)=O 70601,C(=O)(C(CNC(C1CC=CCC1)=O)C(C)(C)C)N(C(CCSC)C)C 70602,C1(NC(=O)CCC2CCOC2)CC(O)(CNC(c2ccc(CO)s2)=O)C1 70603,N1(C(CC2CC(OC)C2)=O)CCC2CN(C(=O)C=CI)C2C1 70604,N1(CC(=O)NCC(CO)NC(COCCOC)=O)CCS(=O)(=O)CC1 70605,N1(C(CC(CC)C)=O)CCC(C2CC2NC(c2cc(C)cc(Cl)c2)=O)CC1 70606,N1(C(c2cnc(CCC)s2)=O)CCCCC(NC(C2(C)C=CCC2)=O)C1 70607,c1(OC)cc(C)c(NC(CCC(F)F)C(N)=O)cc1OC.c12ccnc(n1)N2 70608,N12CC3CCC(C3C1)N(C)CC(C)(C)CC2C.c1(N)ccccc1.CS 70609,C(=O)(C1=CCCN(C(C2(COC)CCCO2)=O)C1)NC(CCCC)(C)C 70610,CCC(CC(=O)NCCCCn1cc(CC(C)(O)c2cccs2)nn1)CC(F)(F)F 70611,S(=O)(=O)(CC(=O)NC1C2CC1N(C(c1ncccc1COC)=O)C2)NCC 70612,N1(C(CC2CC(OC)C2)=O)CC2CCCC(NC(c3cc(CO)ccn3)=O)(C2)C1 70613,C1(C(N2CC(C(N(C(CO)C3CC3)C)=O)OCC2)=O)CC(=O)NC1(C)C 70614,C(=O)(C(C)S(N)(=O)=O)N1C(CNC(c2c(C)[nH][nH]c2=N)=O)CC1 70615,c1(NS(=O)(=O)Cc2ccncc2)ccnc(Oc2ccccc2)c1 70616,c1(C(C(=O)NC(C)(C)C)N(C(C(C)SC)C)C)ccn(C(C)C)c1 70617,C1(C(=O)NC2CON(CC)C2=O)CC(C)(C)CCN1C(C1CCN1C)=O 70618,C1(C(N2C(C(=O)NC)CC2)=O)CN(C(=O)CCc2ccccc2)C2(CCC2)C1 70619,c1(C(=O)NCC(CO)NC(C(C)(CO)NC(C)=O)=O)cc(Cl)c(F)cc1F 70620,c1(C(=O)NCC2C(NC(C3(C)CC4CC4C3)=O)CCCC2)ccc2c[nH]nc2c1 70621,N1(C(C(C)CC2CC2)=O)CC2(C)CC1(C(=O)NCCC1(C)CCOC1)C2 70622,C(C(CC1CC1)C(=O)N1CCC1(C)CC1CCC1)NC(C1CC(N(C)C)C1)=O 70623,C=CCC(C)C(=O)NCCCC1(NC(=O)C2=CCOC2)CC1 70624,CC(C)(CCC(=O)N1CC(C(=O)NCC(c2cnc[nH]2)O)C(F)C1)[N+](=O)[O-] 70625,c1(NC(C(CC=C)CNC(C2CN3CCC2CC3)=O)=O)cnc(C)c(C)c1C 70626,c1(CC)ccccc1CC(N1CC(C)(NC(C2CC(C)CO2)=O)C1)=O 70627,C=CC(C)C(=O)N(CC(C)N(C(=O)Cc1c[nH]nc1O)C)C 70628,c1(C(=O)NC2(C)CCN(C(=O)CCc3cnoc3)C2)nccc2ccsc12 70629,C1(C(N2CCN(CCCNC(=O)CC3CC(F)(F)C3)CC2)=O)CC(=O)C12CCC2 70630,C12(C(=O)N(CC(N3CC4C(CO)C4C3)=O)CCO)CCCC1C2(F)F 70631,N1(C(C(=O)NCCOC)=O)CC2CC(NC(=O)Cc3cccc(Cl)c3)C2C1 70632,c1(SCC(=O)N(CCC(C)NC(C(CCSC)O)=O)C)ncnc2[nH]cnc12 70633,CCC(O)C(C)(C)C(=O)N1CCOC(CC(=O)NC2(C)CCCC2)C1 70634,c1(OC)ccc2c(c1F)CCC2NCCc1cncc(Br)c1 70635,c1(C(=O)OC)ccc2nc(Oc3ccc(C(=O)OC)cc3[N+](=O)[O-])sc2c1 70636,C1(CNC(CC2(C=C)CCC2)=O)CCN(C(c2ccc(N)c(O)c2)=O)C12CCC2 70637,CC1CN(C(C2CCN2C2CCCC2)=O)CC1NC(C1(C)C=CCC1)=O 70638,C1(C)(C(=O)NC(c2cnc(C)s2)C)C=CCN1C(c1cnn(C)c1Cl)=O 70639,C(=O)(C(F)(F)C1=CCOCC1)N1CC(CC(C)(C)CNCc2cc(N)c(Cl)c(O)n2)C1 70640,c1(C(N(CC(C)O)CCNC(C(C)OCC)=O)=O)cnc(CC(C)(C)C)o1 70641,C(c1ccc(F)cc1)=CC(=O)NCC1(C(=O)Nc2ccc(F)c(F)c2)CC1 70642,c1(C(=O)NCC(CC=C)NC(C2CC3CC3C2)=O)ccc(C(F)(F)F)cc1Cl 70643,CC(C#N)C(=O)NC(Cn1cccn1)C(=O)N(C)Cc1ccsc1 70644,C(C(C)CC(C)C)NCc1nnc(SC)s1 70645,n1(CC(=O)NCC(Cc2cccnc2)C(=O)O)cc2ncccc2n1 70646,c1(C(N(CC(CC)NC(=O)CC2CNC(=O)C2)CC)=O)ccc(C2CC2)cc1 70647,C1(C(N2CCN(c3cccc(OC)c3)CC2)C)CCC(F)(F)CC1 70648,C1(CC(C)NN(C)Cc2ncoc2C(F)F)Cc2ccccc2O1 70649,CC1C(NC(C2CCCO2)=O)CCN1C(=O)Cn1ccnn1 70650,C1(C(=O)NC2C(C=C)C2)C(C2CC2)C1(F)F 70651,c1(NC(C2N(C(CCS(C)(=O)=O)=O)CC=C2)=O)ccc2nc(Cl)sc2c1 70652,c1(C(=O)NCC2N(C(CC3CCC(=O)C3)=O)CC(F)(F)C2)nc2c(s1)CCCC2 70653,N1(C2C(NC(C3CCOCC3)=O)CCC2)CCN(C(C23CCCC2C3)=O)CC1 70654,CC(C(=O)NCC1(CNC(=O)CCn2cncn2)CC12CCC2)S(C)(=O)=O 70655,c1(C(=O)NC2(C)CC(NC(C(C)Cc3cnc[nH]3)=O)C2)cnc2c[nH]nc2c1 70656,Cn1nc(C(=O)NC2CN(C(=O)CC3CCOCC3)C3CC23)c2ccccc12 70657,c1(C(=O)NCC2N(C(C(CC)NC(C)=O)=O)CCCCC2)cccc2scnc12 70658,O=C(CC1=CCCCC1)NC1CCCN(C(=O)Cn2ccnn2)CCC1 70659,C1(C(C)C)CN(C(C2CCCCCCC2)=O)CCN1C(C12COC(CF)(C1)C2)=O 70660,C(=O)(CC(C)(C(F)(F)F)N(C)C)N1CCC(N(C(=O)C=C(C)CC)CCC)CC1 70661,C1(C)(NC(=O)NCCCC(=O)N(C(CF)CF)C)C=CCCC1 70662,C(=O)(CC(P(C)(C)=O)P(C)(C)=O)NC1CN(C(C2C(C)N(C)CC2)=O)C1 70663,N1(C(c2ccn(C)n2)=O)CCC2OCCN(C(=O)C(O)C(F)F)C2C1 70664,Cc1ccc(F)c(C(=O)NC(C2CCN(C(c3ccn(C)n3)=O)C2)C)c1 70665,Fc1cncc(SCc2nc(-c3cccc(Cl)c3)nn2Cc2ccccn2)c1 70666,c1(CNC(C(=O)NCC(n2cccn2)C)=O)ccc(CN2CCNC(=O)C2)cc1 70667,CC(CC(=O)NCC(CC(=O)N1CC(N2CCNC2=O)C1)C1CCC1)C(F)F 70668,C(=O)(C(C(C)C)C(C)C)NC1C(NC(c2c(Cl)c(C)n(C)n2)=O)CCCC1 70669,Cc1nscc1C(=O)NC1(CCNC(=O)C(C2CCCCC2)F)CCC1 70670,N1(C(CC2CN(C)C2)=O)CC(NC(=O)COC2CCCC2(C)C)C2(CCC2)C1 70671,C1(CNC(C2CC(=O)NC2)=O)CC(C(F)(F)F)CN1C(=O)CCc1cnccn1 70672,C1(CNC(C2(N(C)C)CCCC2)=O)CCC(NC(=O)Cc2cnccn2)CC1 70673,c1(SC)cc(N2CCC(NC(=O)C(C)NC(=O)NC3CC3)C(F)C2)nc(SC)n1 70674,CC1(C)C2CCC(C(=O)NCC3(O)CCN(C(=O)CNC=O)C3)C1C2 70675,C1(CNC(c2c(CC)cco2)=O)COC(C)(C)CN1C(c1cc(N)nc(Cl)c1)=O 70676,c1(CC)cnc(C(=O)NC2(CN3CCN(C(C4CCC(F)C4)=O)CC3)CC2)cn1 70677,c1(OC)nc(=NC(C)CCNC(C2(C)CC2(F)F)=O)[nH]c2ccccc12 70678,N1(C(C(C)OCC)=O)CC(NC(=O)Cc2cccc(NC(N)=O)c2)C(C)C1 70679,c1(C(=O)NCCOC2CCN(C(CC3C(C)C3)=O)C2)cc(C#N)ccc1F 70680,C1(CC(N2C(CO)CC2C)=O)(OC)CN(C(=O)C=Cc2ccoc2)C1 70681,c1(N2CC(CNC(=O)Cn3nnnc3C3CC3)OCC2)ncnc2[nH]cnc12 70682,C1(c2n(CC=C)nnn2)(N(CCC2CC2)CC)CC2(C1)CC(C)(C)OC(C)(C)C2 70683,C1(CC)C(NC(=O)CCOC(C)CC(C)C)CCN1C(c1cnc(O)s1)=O 70684,CC1(C(=O)NC(C)(CNC(c2ncccc2C2CC2)=O)C2CC2)CCOCC1 70685,c1(C(N(C2CN(C(CCC=C)=O)C2)C)=O)cccc(OC)n1 70686,C#Cc1ccc(NC(=O)C#CC(C)(C)CNC(c2cncnc2C)=O)c(C)c1 70687,C(=O)(CCCC(=O)NC1CCOC(c2ccccn2)C1)N(CC)CC 70688,CN1CCC(C(=O)NC(C(=O)NCC2(C(N)=O)CC2)C2(C)CC2)C1=O 70689,c1(CN(C(=O)CCN2CCC(F)C2)C)ccccc1CNC(=O)CC(F)(F)F 70690,c1(C(=O)NCC(C)NC(C(COC)C)=O)ccccc1-n1cnnn1 70691,N1(C(COCCCCC)=O)CCC(C(=O)Nc2cccnc2C)CC1C 70692,C1(C)(CNC(C(CC)CCOC)=O)CN(C(C23CC(C2)C3)=O)C(C)(C)C1 70693,N1(C(c2c(C)csc2)=O)CCC(n2cc(-c3cscn3)nn2)C(O)C1 70694,N1(C(c2cc(CC)n(C)n2)=O)CC(NC(=O)Cc2nccn2C)C(C)(C)C1 70695,N1(C(CCC(=O)C2C(C)C2)=O)CC2(CCN2C(C2(N3CCOCC3)CC2)=O)C1 70696,c1(C(=O)OC)cc(S(C)(=O)=O)cc(F)c1NC(=O)NCC1CCC2(C1)CC2(F)F 70697,CC1(C)CC(NC(=O)C(=O)NCC(F)(F)F)CN(C(=O)C(C)(C)S(C)(=O)=O)C1 70698,c1(C(=O)NCCOCCN(C(=O)C(C2CC2)C2CC2)C)ccc(Cl)s1 70699,C(=O)(CC(C)CNC(C1COCCN1C(c1coc(C2CC2)n1)=O)=O)OC 70700,C1(NC(=O)COC2CCOCC2)CCC(C(=O)NCCOc2ccc(Cl)nc2)CC1 70701,C1(C2CN(C(=O)CNc3ccccn3)C2)CN(C(c2ccc(CO)s2)=O)CCO1 70702,O=C1CCc2nc(NC3CCC(NC(c4cc5n(n4)CCC5)=O)CC3)ccc21 70703,N(C1CCc2cccnc21)C(=O)COCc1c(OC(F)F)cccc1F 70704,c1(C(N2CCC3C(NC(C4(F)CCCCCC4)=O)C3C2)=O)ccn2cncc2c1 70705,S(=O)(=O)(c1ccc(N(C)Cc2ccc(Cl)cc2)cc1Cl)NC(C)CCCO 70706,C1(NC(CCc2nc(C)sc2)=O)CC2CC1N(C(=O)CC1(C#N)CC1)C2 70707,c1(C(=O)NCC2(F)CN(C(C3C(CC)CCC3)=O)C2)cc(Br)cnc1S 70708,c1(CCC(=O)NCC(C2CCOC2)NC(=O)CC2CSC2)nc(C2CC2)no1 70709,C1(CCN(C(=O)Cc2cccnc2Cl)C)CCCCN1C(=O)CC1CCC1(C)C 70710,C(=O)(C(O)C(F)(F)F)OCC(C)O.C1(=O)CO1 70711,CCCC(C)CC(=O)NC(CNC(c1cc(C)cnc1Cl)=O)CC(C)C 70712,C1(NC(c2c(C#C)c[nH]n2)=O)CCCCCCC1NC(=O)CCCCOC 70713,N#Cc1ccccc1C(N1CCN(C(c2ccncn2)=O)C(CC2CC2)C1)=O 70714,c1(C(N(C2CCN(C(=O)C=NOC)C2)CC)=O)cn(C)nn1 70715,C1(C2CC2)(C(=O)NC(CC(=O)NC)C2CC2)CN(C(C2CC(SC)C2)=O)C1 70716,C(=O)(CC(C)(O)C(F)(F)F)N1CC(C)(NC(=O)Cc2csc(=N)[nH]2)C1 70717,c1(C(N2CCOC(CNC(c3cc(CO)[nH]n3)=O)C2)=O)ccc(Cl)c([N+](=O)[O-])c1 70718,C1(C(=O)NC2(CCNC(CN3CC(CC)C3)=O)CC2)CCN(C(C)=O)CC1 70719,c1(CNC2CC(CN=[N+]=[N-])C2)cc(O)c2ccccc2c1 70720,C1(C(N(CC(O)CO)C(C)C)=O)CCCC2C1C2(F)F 70721,c1(C(N2CC(NC(CCS(C)=O)=O)C(CO)CC2)=O)cnc2c(c1)NC(=O)CS2 70722,Cc1cccc2cc(C(=O)N(CC(C)(C)NC(c3occc3Cl)=O)C)cnc12 70723,C=CC1(C(=O)N(CCCN(C(=O)C(C)Cc2ccncc2)C)C)CCC1 70724,c1(C(N(CCCNC(CCCC)=O)C)=O)ccc2ccc(Br)cc2n1 70725,O=C(C1=CCCCO1)NCCCOCCNC(C1COC2(CO)CC1C2)=O 70726,C1(C(=O)NC2CCOCC2C)(CC)CCN(C(c2csnn2)=O)C1 70727,CC1(C)CC(C(=O)NCC2CN(C(=O)C3CC3)CC23CC3)CCO1 70728,O(NC(=O)C(O)C1CCCCC1)CC(=O)N(CCOC(C)=O)C(C)C 70729,C#CCCC(=O)NCCCOCCN(C(=O)C(O)C=C)C 70730,C1(NC(C(NC(C)=O)=CC2CC2)=O)CC2CCC(C1)N2Cc1ccccc1O 70731,C(=O)(C(C(C)C)C(C)C)NCC1CCN(C(c2cccc(CC(=O)OC)c2)=O)C1 70732,c1(C(=O)NC(CC)CNC(=O)CCCCOC)ccnc2[nH]ncc12 70733,C1(NC(c2n(C)ncc2Cl)=O)CCC2CN(C(C3(C#N)CCCOC3)=O)CC2C1 70734,c1(CC(=O)NCC(CNC(CCSCC(N)=O)=O)O)ccc2nonc2c1 70735,N1(C(C(C)C#N)=O)C2CCC1CC(CNC(c1cc(Cl)ccc1OC(F)F)=O)C2 70736,C1(CNC(C2CC(OC)C2)=O)CN(C(C2CCN2C2CCCC2)=O)CCO1 70737,c1(NCC(C(C)C)(C)NC(c2ccc(F)nc2F)=O)ncnc2c1nnn2C 70738,C12(NC(c3n(CC)ncc3)=O)CCC(C(N3CCC(C)(O)C3)=O)(CC1)CC2 70739,CCCC(CCCNC(=O)COc1ccc(F)cc1)NC(c1nc(O)sc1C)=O 70740,c1(SCC)ccc(Cl)cc1C(=O)Nc1c(OCC)cccc1F 70741,c1(C(=O)NCCOCCN(C(C(CC#C)C)=O)C)cc2c(nn1)CCCO2 70742,Cc1cc(C(=O)NC2CCCCC2NC(C2CCC(=O)O2)=O)cc(C)c1Br 70743,Cn1cc(Br)c(C(=O)NCC2(CCNC(=O)Cn3cccn3)CC2)cc1=O 70744,Cc1cc([N+](=O)[O-])c(N2CCC(C(F)(F)F)C2)cc1Br 70745,C#CC1CC2(CC2)CN1C(=O)C(C(C)CC)N(C)C(c1oc(C)cc1C)=O 70746,c1(CNC(c2ccccc2Cl)c2n(CC)nnn2)ccc(Cl)nc1 70747,c1(NC(C(=O)NCC(=C)F)=O)cc(C(F)(F)F)ccc1OC 70748,c1(NC(=O)Cc2noc(-c3ccccc3)n2)cc(N2CCOC2=O)ccc1F 70749,C(=O)(C(O)CC(F)(F)F)NC1(CC(N2CCC(C(=O)OC)CC2)=O)CCC1 70750,N1(C(C(C)=C2CC2)=O)CCCN(C(=O)CCN2CCNC(=O)C2)CC1 70751,C1(C(C)C)(NC(=O)NCC2(CN(C)C(=O)OC(C)(C)C)CC2)CCC1 70752,C1(CC(=O)NCCN(C(C(c2cncnc2)C)=O)C2CCCC2)CCC(C)(C)O1 70753,C1(NC(c2cn(CC)nc2)=O)CCC(NC(=O)C(C)Sc2ccc(F)cc2)CC1 70754,N1(C(CCC#CC)=O)CCC(CNC(=O)C(CCC)NS(C)(=O)=O)C(O)C1 70755,N1(C(C2(C(C)C)CCN(C(c3ccsn3)=O)C2)=O)CCC12CCSCC2 70756,C(CCCCC(=O)N1CCCC(C(C)(O)CNC(c2cc[n+]([O-])cc2)=O)C1)OC 70757,C1(C(=O)NC(C)CCNC(c2occc2F)=O)C2CCCOC12 70758,N1(S(C(C)C)(=O)=O)Cc2ccc(NC(=O)C(C)OCc3ccccc3)cc2C1 70759,C1(C(C(=O)NCC=C)N(C)CCc2noc(C(C)C)n2)CCSCC1 70760,Cc1ccc(CCC(N2CCN(C(c3nnc(O)nc3O)=O)CC2)=O)cc1Cl 70761,CN1CC(=O)N(CC(=O)NC2CC(NC(=O)Cc3cn(C)cn3)C2)C1=O 70762,C1(C(N2C(CNC(c3cc(CC)on3)=O)CC2)=O)CCOCC12CCC2 70763,Cc1[nH]c2ncccc2c1C(N1CCN(C(=O)CC2CCCO2)C(CF)C1)=O 70764,N1(c2cc(C)nc(N3CCC(c4ccc(S(N)(=O)=O)s4)C3)n2)CC2CN(C)CC2C1 70765,c1(NCC2CC3CN(C(C(C)OCC)=O)CC32)nc(C)nc2sc(C)c(C)c12 70766,c1(C(C(=O)NC2C(CNC(c3nccc(C(C)(C)C)c3)=O)C2)O)cc(Cl)cc(Cl)c1 70767,N1(C(C(=O)Nc2ccccc2)=O)CC2CCNCC12.c12ccc(cc1)OCCC2 70768,C1(CC(=O)NC(CC)(C)CO)CN(C(C2C=CCS2)=O)CCO1 70769,N1(C(C(C(CC)O)C)=O)CC2CCN(C(c3scc4c3OCCO4)=O)CC12 70770,Cc1cc(C(N2CCC2C(=O)Nc2cnn(C3CCS(=O)(=O)C3)c2)=O)n(C(F)F)n1 70771,c1(SC)cccc(CC2CCCC2)c1.C12CC(C)N(C1)C(=O)CN(CO)C(=O)C2 70772,C(=O)(C1=CC(C)(C)C1)NCC1(CN(C)C(C2(Cl)CC2(F)F)=O)CC1 70773,c1(-c2cn(C3C(C)CN(C(=O)C(F)C4CCC4)C3)nn2)cc(Cl)cc(Cl)c1Br 70774,C1(NC(C2N(C(c3cnn(C=C)c3N)=O)CCCCC2)=O)C(=O)OC2CCCC12 70775,C=Cc1cnn(C)c1CNC(=O)N(C)CC1(O)CCOCC1 70776,C1(NC(c2ccc(CCC)cc2)=O)CCN(C(c2cnc(N)c(O)c2)=O)CC1F 70777,C(C1=CCSC1)(c1n(CC(=C)C)nnn1)NCC1CC(=O)N(C2CC2)C1 70778,C1(NC(C2CCN(c3ncccn3)C2)=O)CC1C1CC1 70779,C1(NC(C2(CC)CN(C(C(CCCC)C)=O)C2)=O)CCCCC12CCC2 70780,C1(CNC(c2scnc2Cl)=O)CN(C(c2cn[nH]c2)=O)C2(CCOCC2)C1 70781,N1(C(C(C)(C)NC(=O)OC)=O)CCN(C(=O)C(C)c2cccs2)C(CN(C)C)C1 70782,c1(CC(=O)NC(CC#C)COC)nc(C)ccc1Br 70783,c1(C(N2CCC(NC(c3c(OC)scc3)=O)CC2C)=O)cc(C)cc2ccoc12 70784,c1(C(=O)NCCC(CNC(C2(CCC)CCC2)=O)O)cc(Cl)c2[nH]c(O)nc2c1 70785,c1(C(=O)NCC(CNC(C2CCN(C(CC)=O)C2)=O)OC)cc(C)n(C2CC2)c1 70786,C1(C(=O)NC(C)CCNC(c2ccnc(Cl)c2N)=O)CC(C(C)(C)C)=NO1 70787,C(C(C)(C)C(=O)N1CCC(OCC2CCC2)C1)N(C(CN(C)C)=O)C 70788,C(C(=O)N1CCOC(CC(N2CC(O)CC2CN(C)C)=O)C1)(C(C)C)OCC 70789,c1(CC)cccc(OCC(=O)NCCC(C)(C)NC(C2CCC(C)O2)=O)c1 70790,c1(NC(C(CC)C)=O)ccc(SCCC(N2CCC(C)CC2)=O)cc1C 70791,C(=O)(C(C(C)C)N(C)C)NC1C(NC(C2(COC)CCC2)=O)CC1 70792,c1(N(C(C2N(C(CCC)=O)CC3(CC3)C2)=O)C2CC2)cn2c(n1)CC(OC)CC2 70793,C(=O)(C(C)(C)CCCNC(=O)CCc1nccs1)NCC(c1cnc[nH]1)C 70794,C(=O)(N=c1[nH]nc(CC#N)s1)N1CCC(CN(CCC)CC)C1 70795,C1(C(CNC(C(C)(C)n2ccnn2)=O)(C)O)CCN(C(C2CCCCC2)=O)CC1 70796,CN1CC(NC(c2cc(CNC(c3ccc(O)nn3)=O)ccn2)=O)CC12CCC2 70797,CCCCC(CC)N.N12CCCC(C1)COC2=O.c1(O)ccccc1Br 70798,C#Cc1cc(C(N2CCC(F)C(NC(c3cc(Br)n(C)c3)=O)C2)=O)cc(N)c1 70799,N1(C(C2(COC)CC=CC2)=O)CCC(F)(CNC(C2(COC)C=CCC2)=O)CC1 70800,c1(OC(C)C)cccc(CC(=O)NC2CC2)c1.C1CC1NC(C1(C)CC1)=O 70801,O=C(CCC[N+](=O)[O-])N1CCCC(CCNC(C2(c3ccccn3)CC2)=O)C1 70802,CC1CCC(CCC(N2CC(O)(CN(C(=O)CC34CC(C3)C4)C)C2)=O)O1 70803,N1(C(c2c(C(C)C)con2)=O)CCCC(C)(C(=O)NC2CCCC2)C1 70804,CCCCC(C(=O)N(CC(C)NC(c1nn(C)nc1C(=O)OC)=O)C)C(C)C 70805,c1(C(N(C)CC2CCN(C(C(CCC)O)=O)C2)=O)cnn2c1N(C)CC2 70806,c1(C(=O)NCCN(CCC)C(c2c[nH]nc2CC)=O)c(C)csc1Cl 70807,C1(CNC(c2cnc(O)o2)=O)CC2(CCC2)CN1C(c1ncoc1C1CC1)=O 70808,C(=O)(CC(C)(C)C(=O)N1CC2CC(NC(=O)C(c3ccccc3)C)CC2C1)OC 70809,N1(C(Cc2ccn(C)n2)=O)CC(NC(C2(c3cncs3)CC2)=O)CC(F)C1 70810,CC#CCCC(=O)NC1(C(N2CCOC(COC)C2)=O)CC1 70811,c1(CCC(=O)NCC(C)N(C(=O)C(F)(F)c2cscn2)C)ncc(C(C)(C)C)o1 70812,C1(CC)CC(NC(=O)Cn2cc(-c3csc(-c4ccc(Cl)cc4)n3)nn2)C1(C)C 70813,CCC(CC)C(F)C(=O)N(CCNC(C1CCCC(C)(C)O1)=O)CC 70814,C(CC1CC1)(C(=O)NCC=CCNC(c1cc(Br)co1)=O)OC 70815,C=C(C)C(CC(=O)NC(C)(CNC(c1cc(O)ccc1O)=O)C1CC1)OCC 70816,C1(CCC#C)CCCN(C(=O)C(C)(CO)NC(=O)C(C)N(C)C(C)=O)C1 70817,C1(C(=O)NC(C(C)C)(C)CNC(=O)CN2CCC(=O)CC2)CCCCC1(F)F 70818,C1(C(=O)NC(C(=O)NC2(C(COC)O)CC2)CCC2CC2)C2CCC(C2)C1C 70819,c1(CC(=O)NC2CC2NC(C2CC3OC(=O)CC23)=O)nc([N+](=O)[O-])n[nH]1 70820,N1(CCn2c(C)csc2=O)CCCN(C(c2c(Cl)nn(C)c2Cl)=O)CC1 70821,c1(NC(C2CCN(c3cn(C)nc3)C2)=O)cc(Br)cnc1S 70822,CC(C)CC(O)CN=c1cc[nH]cc1S(=O)(=O)N1CCc2c(C)cccc2C1 70823,c1(OCC)ccc(NC(c2nnnn2C2CC(F)(F)C2)(CC)C2CC2)c(F)c1 70824,c1(CN(C)C(C2CN(c3ccncc3)C2)=O)ccnn1C 70825,CCC(C)C(O)C(=O)NC1(CO)CN(C(=O)C(C)(O)C2CC2)C1 70826,CN1C(=O)OCC1C(N1CCC(F)(C(=O)NC2CC2)C1)=O 70827,N(C(=NCCC(C)C)NCC(C1CCOCC1)(F)F)Cc1c(CC)cccc1 70828,Cc1cnn(C(C)C(=O)NC(c2cccnc2)C(=O)NC2CC(C(N)=O)C2)c1 70829,N1(C(CC=C(C)C)=O)CCN(C(c2ccc(C(F)F)o2)=O)CC1c1cn[nH]c1 70830,C(CO)(CCCCN(C(c1ccc(C(C)C)cc1)C)CO)NC(=O)OC(C)(C)C 70831,c1(N(c2nccc(C(C)C)n2)C(C2CCCNCC2)=O)ncc2ccccc2n1 70832,Cc1cc(C(N2CCC23CN(C(=O)CCC(C)(F)F)C3)=O)c(O)c(C)c1 70833,N1(C(C2(C(=O)OC)CC2)=O)CCCCC(c2nc(-c3ccc(OC)cc3)no2)C1 70834,C(C(C(=O)N1CC2CCOC2C1)NC(C1C2CC3C(C2)C13)=O)c1cnn(C)c1O 70835,c1(OC)cc(C)cnc1C(=O)NCCCOC1CCN(C(=O)C(C)C(C)C)CC1 70836,Cc1cc(C)c2nc(N3CCN(c4c(F)ccc(F)c4C#N)CC3)sc2c1 70837,Cc1ncc(C(C)NC(=O)CCCN(C(=O)NCC2(C)CC2)C)s1 70838,c1(C(=O)NCC2CN(C(C(C(C)C)F)=O)CC2(C)C)cnc2n1CCCCC2 70839,CCC(C(=O)NC1CC(C)N(C(=O)Cc2cc(C)n(C)n2)C1)C(C)(C)CC 70840,c1(CC)ccnc(NCC2CCCC2NC(=O)CCCN2CCCC2)n1 70841,c1(N2C(C)CCN(C(=O)Cc3cc(F)cc(F)c3)CC2)nc2cccc(F)c2o1 70842,C1(CNC(C(C#C)(C)C)=O)CN(C(=O)Cc2cc(C)on2)CCCO1 70843,Cc1cc(Br)cc(C)c1C(=O)NCCN(C(=O)Cc1c(O)ncnc1O)C 70844,N=c1[nH]c2ccc(C(=O)NCC3CCCC3NC(=O)CCc3ccoc3)cc2o1 70845,c1(CN(C(COCCNC(c2ccc(CC)[nH]2)=O)=O)C)ccc(C)cc1 70846,c1(COC)ccccc1NC(C1CC1C(=O)Nc1cc(CS(C)(=O)=O)on1)=O 70847,c1(-c2nc(N(C(C=CC)C)CCC3CC(C)(C)NC3=O)sc2)cc2ccccc2o1 70848,O=C(C(F)(F)CO)N1CCC(OC2CN(C(=O)Cn3ccc(C4CC4)n3)C2)CC1 70849,CCCC(C)(C)C(=O)NCC(C)N(C(c1ccc(OC2CC2)cc1)=O)CC 70850,c1(OCCOC)cncc(C(=O)NC2CC(CNC(=O)C(Br)=C(C)C)C2)c1 70851,C(CC(=O)N(CC(C)CO)C)(C(C)CC)NC(C(CCC)N(C)C)=O 70852,C1(C(N2CC(F)(CC)C2)=O)COCCN1C(=O)CC(C)=C(C)C 70853,C(C(=O)NCC1CC12CCCCC2)(C(C)(C)C)NC(C1N(C)C(=O)CC1)=O 70854,c1(C(=O)NC2CN(C(CC(C(C)C)C)=O)CC2(C)C)c2c(nn1C)CCCC2 70855,c1(C(N2CC(NC(C3(C)CC4CC4C3)=O)C(C)(C)C2)=O)ccc2oc(=N)[nH]c2c1 70856,c1(C(N2CCC(C)(CNC(=O)CC3CCC(=O)N3)C2)=O)cc2c(Cl)cncc2s1 70857,N1(C(C(C)OCC(C)C)=O)CC(C2CCCN(C(c3cc(CO)[nH]n3)=O)C2)C1 70858,c1(C(=O)NCc2cc(C(=O)NCCC(COC)O)n(C)n2)ncc(F)cc1N 70859,CC1CC(CNC(=O)C=CC2CCCCCC2)CCN1C(c1nn(C)cc1Cl)=O 70860,C1(C(N2CC(F)(C(N(c3ccc(OCC)cc3)C)=O)C2)=O)CC(=O)OC1(C)C 70861,c1(CN(CCCC)S(C)(=O)=O)ccccc1-c1ccc(NC(c2nc[nH]n2)=O)s1 70862,CC1CN(C(c2cc(Cl)ccn2)=O)CC(C)C1NC(c1cc(N)nc(Cl)c1)=O 70863,C(=O)(C#CC1CCOC1)NC1(COC)CN(C(c2ccc(C(F)F)cc2)=O)C1 70864,Cc1ccc(CNC(=O)C(CC2CC2)NC(c2cnn(C)c2)=O)s1 70865,C1(CCC)CCCCCN1C(c1cc(Br)ccc1N1CCNC1=O)=O 70866,C(=O)(C1CCCn2nncc21)Nc1n(C)c(-c2cncnc2O)nn1 70867,c1(C(=O)NCCCN(C(=O)C=C(C)COC)CC)ncncc1OC 70868,N1(C(C2N(C(c3cccc(C)c3O)=O)CCC2O)=O)CC2(CCOCC2)C1 70869,N(C)(C(=NCC1CC2CC1C2)NCC(C)(C)C)CCCOC 70870,C(CCCCCNC(c1sccc1C1CC1)=O)N(C(CC=C)=O)C 70871,c1(C(N2CCN(C(C=CCOC)=O)C(C)CC2)=O)ccc2c(c1)C(C)CO2 70872,c1(C(N(C(C)CNC(C2CC2(C)CC)=O)CC)=O)ccccc1S(=O)(=O)C(F)F 70873,CC1SCCCC1C(=O)N(C1CCC(CNC(=O)CSC(C)(C)C)CC1)C 70874,N1(C(CC(=C)Br)=O)CCC2(CCN(C(c3cccc(C(C)C)n3)=O)C2)C1 70875,c1(C(=O)NCC(C2(O)CCN(C(COCC=C)=O)C2)C)cc(N(C)C)nc(Cl)c1 70876,n1(CC(=O)NCC(CC(C)C)NC(CSCCCC)=O)cc(F)ccc1=O 70877,C1(C2CCC2)(NC(C(C2CCN(C(c3csc(F)c3)=O)C2)C)=O)CC1 70878,c1(C(N2CCN(CCN(C3CN(C(C)=O)C3)CC)CC2)=O)cnn2cccc2c1 70879,c1(C(=O)NC2C(C(=O)NCC(F)(F)F)C2)cccc(Cc2ccccn2)c1 70880,CCCCC(CNC(C1CCC(OCC)CC1)=O)OCCC.C1(=O)CCCCN1 70881,C1(C(N(CCC)CC)=O)C=CC(N(C(=O)COC)CC2CC2)C1 70882,C1(C#CC(=O)NCCn2cnc(C(=O)NC(C)(C)CC(C)C)c2)(CC)COC1 70883,C(=O)(C1CCOc2ccccc21)N1C2CN(C(c3nnc4ccccn34)=O)C(C2)C1 70884,C(=O)(CCC(=O)Nc1ccc(C(C)Nc2cn(-c3ccccn3)nn2)cc1)OC 70885,C1(NC(CC(C)C)C(=O)C(=O)CCn2cnc(=N)[nH]2)CCC2CCCC1O2.N 70886,N1(C(CC=C)=O)CCC(NC(=O)CCc2ccc(C)nc2)C(CC)C1 70887,C1(CN(C(=O)C(C)n2cccc2)CC)CCN(C(=O)C(C)Cc2ccco2)CC1 70888,N1(C(CC2CCN(CC)C2)=O)Cc2ccc(F)cc2CC1C.N12CC(CC1=O)C2 70889,N1(C(C2(NC(C)=O)CCC2)=O)C2CCC1C(NC(c1ccc(Cl)cc1)=O)C2 70890,Cc1ccccc1C=CC(=O)NCc1occc1C(=O)NCC1CC2(CCC2)C1 70891,c1(OC)cc(C(F)(F)F)ccc1CNC(=O)C(c1ccc(OC)nc1)N 70892,CCCC(C)(CC)C(=O)NCC(C(=O)N(C1CCCC1C#N)C)N(C)C 70893,N1(C(C(=O)OCC)=O)CC(OC)CC1CCNC(=O)CSc1ccccc1OC 70894,c1(N(C(c2cc(C)c(O)nn2)=O)OC)ccc([N+](=O)[O-])cc1C#N.C1(C)(CN)CC1 70895,C1(C(N2CC(CC(C)NC(CC3CC(SC)C3)=O)C2)=O)Cc2nccn2C1 70896,C1(C(=O)NCC2(CCNC(COCCCC#C)=O)CC2)CCC(C2CC2)C1 70897,C1(CNC(CN(C)CCO)=O)CCC12CN(C(=O)CCCn1ccccc1=O)C2 70898,N1(C(c2nc(C)oc2C)=O)CCc2sccc2C1CNC(C12CCC1C2)=O 70899,C(C(CCC)C(=O)NCc1nc(N(C)C)no1)NC(C=C(CC)CC)=O 70900,Cn1ncc(Cl)c1C(=O)NCC12CC(NC(C3CCCN(CC=C(C)C)C3)=O)(C1)C2 70901,c1(C(N2CCC(C(=O)OC)(C(C)C)C2)C(=O)NCCSC)ccc([N+](=O)[O-])cc1 70902,C(CC(C)(C)C)(C(=O)NC1CCCCC1N=[N+]=[N-])NC(CCC#C)=O 70903,C1(C(N2CCC(N(C(C3CC(OCC)C3)=O)C)C2)=O)CC2(CCC2)C1 70904,Cc1cc(C(N2C(C(=O)NC(C)C(C)F)CC2C)=O)cn1C 70905,Cc1cc(Cl)ncc1CC(N1CCN(C(=O)CC(C)C2CC2)C(C)C1)=O 70906,C(=O)(C(C(C)(C)C)NC(N)=O)NC1CC(CNC(C(=O)NC(C)C)=O)C(O)C1 70907,c1(OC)cc(C(=O)NCC(C)N(C(=O)CCC2CCCCN2C)C)cc(C)n1 70908,c1(NC(=O)NCCCNS(C)(=O)=O)ccc(C2CCCNC2)cc1 70909,C1(C(=O)NCC(CC)CC(C)C)CCCN1NC(=O)c1cccnc1C 70910,CC(C)C(C(=O)NCC1(NC(c2ccc(-n3cnnn3)cc2Cl)=O)CC1)C(C)C 70911,C1(C(N2CCCC(C)C2)=O)CN(C(=O)CCc2ccc(N(C)C)cc2)CCC1O 70912,Cc1cc(F)c(C(=O)NCC2CCN(C(c3cnc(O)c(Cl)c3)=O)C2)c(Br)c1 70913,CC(CC(=O)NCC(C(=O)N1CCc2ccsc2C1)C(C)(C)C)CC(C)(C)C 70914,c1(CNC(c2cc(OC)ns2)=O)cccc(C(=O)NCC2OCC(CC=C)C2)c1 70915,C1(CNC(CN(CCC)C)=O)C(C)CCCN1C(=O)C(C)N(CC(F)(F)F)C 70916,C1(CN(C(=O)C=CCOCC(F)(F)F)C)COCCN1C(C1CC2CC2C1)=O 70917,C(=O)(C(C)CC(F)(F)F)N(CCC(C(C)C)NC(CCCCC=CC)=O)C 70918,C1(C(=O)NCC=C2CCN(C(C3CC(=C4CC4)C3)=O)CC2)CCC2(CCC2)CO1 70919,c1(C(N2CC3=C(CN(C(=O)CC(F)(F)C(F)F)C3)C2)=O)coc2ccc(F)cc12 70920,c1(C(N2CCC(OC)CC2)C(=O)NC2(C)CC2)cc2cccc(Cl)c2o1 70921,CCC(c1ccccc1)=CC(N1CCC(N(C(=O)COC2CCC2)C2CC2)C1)=O 70922,N12CC(C(O)C1)C2=O.c1(NC(C)C)nc[nH]n1.C12(CC1)N(C)C(=O)COC2 70923,N1(C(CC2C(OC)CC2)=O)CCCC1C1(NC(c2sccc2C(C)=O)=O)CC1 70924,c1(C(N2CCC(C(C)NC(C(C)OCC#C)=O)CC2)=O)cc(Cl)c([N+](=O)[O-])[nH]1 70925,CC(C)CC(=O)N1CCC(C(=O)NCC2C(CO)C2(F)F)C1 70926,c1(C(=O)NC(C)C(C)C(N2CCC(C)(C#N)C2)=O)cccc2[nH]ccc12 70927,N1(C(c2scnc2Br)C(=O)Nc2c(C)cc(F)cc2)CCN(C(=N)NC(=N)N)CC1 70928,CC1(C(N2CCC(OCC3CC3)C2)=O)CCCN(C(c2ncccn2)=O)C1 70929,N1(C(=O)Nc2ncc(CCOC)s2)CC(CO)OC(C)(C)C1 70930,C1(NC(Cc2c(C)nsc2)=O)C=CCN(C(=O)C(c2cccc(F)c2)(C)C)C1 70931,C12(NC(CN(CC(=O)NC(C)C)C)=O)CCOCC1CN(C(=O)CS(C)(=O)=O)C2 70932,C1(NC(c2c(CC)cco2)=O)CCC(C)N(C(c2cnn(C)c2Br)=O)C1 70933,N12CCCC(F)(C1)CCCN(C(CC1CCC1)CO)CCC2=O.C(CO)OC 70934,C#CCC(CC(F)F)C(=O)N1CC(CC(=O)NC2(CC=C)CCCC2)CC1C 70935,c1(SC)cc(C)c(C(N2CC(NC(c3cc(CCO)on3)=O)C(C)C2)=O)o1 70936,C1(C(N2C(C)(CC(=O)NC(C#C)(C)C3CCC3)CC2)=O)CCCC(=O)C1 70937,CS(=O)(=O)c1ccc(CCOC(C2CC2c2cccc3ccccc23)=O)cc1 70938,N1(C(c2c(C)scc2)=O)CCCCCC1C(=O)NC(c1nn[nH]n1)C1CC1 70939,C#CC1(C(N2CCC=C(Cl)C2)=O)CCN(C(c2cncc(C#C)c2)=O)C1 70940,N1(C(C=CCOC)=O)CCOCC1CCNC(=O)C(c1ccn(C)n1)C 70941,c1(C(=O)NC2CCN(C(c3ncn(CC)c3)=O)C2)ncc(P(C)(C)=O)cn1 70942,C1(C(N(CCCN2CCCC2)C)=O)CC12CCN(C(C1CCC(C)CC1)=O)C2 70943,c1(CN(CCN(C(COC)=O)C(C)C)C)nnc(-c2cccs2)o1 70944,c1(CN2CC3(CC)C(C)(C2)C3)cc2ccoc2cn1.c12ccc(cc1Cl)[nH]c2=O 70945,CC1(CNC(C2CC(NC(=O)Cn3cccc3)CCO2)=O)NC(=O)NC1=O 70946,c1(C(=O)NCC23N(C(C=CSC)=O)CCC2CCC3)ccc2c(c1)CCCO2 70947,c1(C(=O)NCCNC(=O)CSCC2CCCO2)cc(=O)n2ccccc2n1 70948,N1(C(C=CSC)=O)CCOC(CCNC(C2(C3CC3)CC2C(F)(F)F)=O)C1 70949,c1(CC(=O)NC2CN(C(C3(CC#C)CCCCO3)=O)CC2F)ccc(C)c(F)c1 70950,c1(OC)ccc(Cl)c(C(=O)NC2CC(F)(CNC(=O)C(F)(F)C3CC3)C2)c1N 70951,c1(N2CCC(=C)C2)nc2ccc(S(=O)(=O)N3CC(C#N)C4(CCC4)C3)cc2s1 70952,Cc1cc(OCC(N2CC3CCOC3(CNC(=O)CC3CC3)C2)=O)cc(C)c1Cl 70953,c1(CN2CCC(O)(C(=O)NCC(C)OC)CC2)c[nH]c2ncc(Br)nc12 70954,CCC(C)C(C(=O)N1CCCN(Cc2ccc(C(C)C)cc2)CC1)OC 70955,c1(C(N(C(C(=O)NCCC(C)OC)=O)C)C)ccc2c(c1)OCCO2 70956,CCC(C)(COC)C(=O)NC1CC(NC(=O)C(C)N(C)C)C(O)C1 70957,c1(C(=O)NC(C2(O)CN(C(=O)CCNc3ccccn3)C2)C)ccoc1Br 70958,c1(OC)cc(CN2CC(F)(F)CC2C(=O)Nc2cc(Br)ccc2I)c(Br)cn1 70959,Cc1nn(C)c2c(NCCN3CCCOCC3)nc(=NCC(C(C)C)N(C)C)[nH]c12 70960,N1(C(c2n(Cc3nc(C)on3)nc(C)c2)=O)CCC(O)CC1C(=O)N(C)C 70961,Cc1c(C=CC(N2CCC(CCNC(C3CC4C=CC3O4)=O)CC2)=O)cnn1C 70962,Cn1cc(C(=O)NCCCC(c2ccccc2)NC(C2(F)CC=CC2)=O)nn1 70963,N1(C(C2(CCC=C)CCCC2)=O)CCN(C(=O)Cc2cnn(C)c2)CC1CCC 70964,c1(C(=O)NC2CC(N(C(Cn3c(C)ccc3C)=O)C)C2)ccc(P(C)(C)=O)nc1 70965,c1(C(=O)NCC(CCNC(C(C)CS(C)=O)=O)(C)C)scc2c1OCCO2 70966,CC(CNC(c1cc(O)cc(F)c1)=O)C(F)C(=O)NCC1(C(F)(F)F)CC1 70967,c1(C(N2CCC(OCCNC(C(CC#C)O)=O)CC2)=O)ccc(C(C)=O)nc1O 70968,N(C(=NCc1ccn(C)c1)NCc1cccc(OCC(F)(F)F)n1)C(C)C1CC1 70969,N1(C(C(C)SCC)=O)CCC2(CC1)CCN(C(c1cnncc1O)=O)C2 70970,c1(OC)nc(C(=O)NC2CCC(NC(c3cc(Cl)cs3)=O)CC2)cc(O)n1 70971,N1(C(CNC(=O)OC)=O)CCCC(C)(C(=O)NC(c2ccncc2)C)C1 70972,c1(CNC(C(C)OC)=O)ccc(CCNC(=O)CC(C)(C)c2cccs2)cc1 70973,Cc1nc2ccccc2n1CC(N1CC(C(C)NC(c2ccnnc2)=O)C1)=O 70974,CCC(C)(CNC(=O)C(F)C(C)C)C(=O)N1CC(O)(C(C)C)C1 70975,C1(C(C)NC(c2c(CC)ocn2)=O)CN(C(=O)C(C)(C)c2cccs2)CCO1 70976,CCCCC(CNC(c1cnccc1N)=O)NC(c1cc(C(F)(F)F)c[nH]1)=O 70977,N1(CC(=O)N(C2CCc3ncsc3C2)CCCCCC)CCc2cc(F)ccc2C1 70978,CCCCC(C)N=c1cc(NCCCCCOCC2CC2)nc(C)[nH]1 70979,c1(NC(C)=O)ccc(C(N2CCC(CNC(=O)Nc3cncc(C)c3)C2)=O)nn1 70980,C1(CC)CN(C(=O)C(=O)NC2CC2)CCC1NC(=O)C(c1cnn(C)c1)O 70981,CC(C)CC(C)CNC(c1csc(-c2cnn(C)c2)n1)=O 70982,N1(C2(C(=O)NCC(CNC(CC=CCC)=O)OC)CC2)CCCCC1=O 70983,C1(C(N(CCC(=O)NOCCC2CC2)CC#C)=O)CC2C=CC1CC2 70984,CS(=O)(=O)C(C(=O)OCCCCCCCCSC)C1CN(C(=O)OC(C)(C)C)C1 70985,c1(C(=O)NCC(C)(CO)NC(CCSC)=O)cccc(-c2noc(C3CC3)n2)c1 70986,c1(CN(C(C(OC)OC)=O)CCCNC(C2(C)CSC2)=O)ccccc1 70987,C(=O)(CCCC(C)(F)F)NC1(CCOC)CCN(C(=O)C(C)C2(O)CCC2)C1 70988,c1(OCC(N2C3CC(NC(COCC)=O)C2CC3)=O)ccc(C#N)cc1Cl 70989,C1(C(N2CCC(C#CC)C2)=O)CCC2CCC1N2C(c1coc(C)c1)=O 70990,C(=O)(C1=CCC2CCC1N2C(c1coc(C(F)F)c1)=O)NCCCOCCCC 70991,C(=O)(C#CC1CCCO1)N(CCC)CCNC(C1(NC(=O)C2CC2)CCCCC1)=O 70992,N1(C(C=C(C)CNC(C2CC(=O)N(C)C2)=O)=O)CCc2cc(F)ccc21 70993,C#CCC(C(=O)NC1COCC1F)NC(c1ccnc(C)c1)=O 70994,N1(C(C(C(C)C)SC)=O)CCCN(C(C2(c3ccc(Cl)c(Cl)c3)CC2)=O)CC1 70995,C#CC(C)(C)C(=O)N1CCC(C(=O)NCCC(=O)NC(C)C)O1 70996,c1(N(C)C)cc(C(=O)NC2CCC2C2CC2)nn1-c1ccc(Cl)cc1 70997,c1(CSCCC(=O)NCC#CCNC(C2C(C)(C(C)C)C2)=O)ccc(Cl)cc1 70998,C1(CNC(=O)CCC2CCCN2C(=O)CC2CCOC2)CCC=CCC1 70999,Cc1nn(C)c2sc(N3C(C(=O)C(=O)NCCC(P(C)(C)=O)c4ccccc4)CC3)cc12 71000,c1(C(=O)NC2CCN(C(c3cc(OC)c(F)cc3)=O)C2)cn(C)cc(Br)c1=O 71001,C1(N(C(=O)CC2CCOC2)CCC)CCN(C(=O)Cc2cc[nH]n2)CC1 71002,C1(C(=O)NCC2CC(C)N(C(c3cnc[nH]c3=N)=O)C2)CCCC(C)(C)O1 71003,C1(C(N(CCN(C(=O)CC(C)n2cc(Br)cn2)C(C)C)C)=O)CNC(=O)C1 71004,Cc1sc(O)nc1C(N1CC(F)(C(=O)NC2CCOCC2F)C1)=O 71005,N1(C(CC(=O)NCC)=O)CCC(O)(C2(NC(=O)C(C)C(C)(F)F)CC2)CC1 71006,c1(CC(C(=O)OC)N(c2cccc(N(C)C)c2)CCF)ccc(F)cc1 71007,CCC(C)C(C(=O)N1CCC(NC(=O)C(Cl)=CCl)C(O)C1)NC(=O)OC 71008,C1(OC)CN(C(=O)C=Cc2ccccc2)C(C)(CNC(c2nncs2)=O)C1 71009,c1(C(=O)NC2CCc3n(C)cnc3C2)ccc2c(=N)[nH]cnc2c1 71010,C1(C(=O)NCC2CCCN(CC(=O)NCC)C2)CCCCC1(C)C 71011,C#Cc1ccnc(C(=O)NC(CC=C)C(=O)N2CCOCC2CCO)c1 71012,C1(C(=O)NC2CSCC2C)(NC(c2ccc(CC)o2)=O)CC(F)(F)C1 71013,C1(C(N(CC(=O)NCCC)C)=O)CCCC(NC(C2CCO2)=O)CC1 71014,c1(C(=O)NCc2cccc(NC(C(CC)F)=O)c2)cc2cc(C)[nH]c2cc1Cl 71015,C(CC(C)CCNC(=O)CCC1CCCO1)NC(C1N(C(C(C)C)=O)CCC1)=O 71016,C1(NC(C2(CC=C)CC2)=O)CCC(O)CN(C(C2CC23CCSCC3)=O)C1 71017,CCC(CC)C(C(=O)N1CC(O)(C2CCCN2C(=O)C=Cc2ccc(C)o2)C1)OC 71018,C(C(CN=c1[nH]c(Cl)nc2ccc(Br)cc12)c1ccc(Cl)cc1)OC 71019,N1(C(C(COC)C)=O)CCOC2(CCCN(C(c3ccc(CN(C)C)[nH]3)=O)C2)C1 71020,C(=O)(C(C)(C)CC(C)(C)C)NC(CC)CN(C(=O)C1=CCCC1(F)F)C 71021,C1(CCCC)CCC(C(N2CCC2C(O)C(=O)OCC)=O)C1 71022,Cc1cc(C)c(C(N2CCCC(NC(C3(C)CC3(F)F)=O)CC2)=O)c(S)n1 71023,C=CCCC(C(=O)OCCCN=[N+]=[N-])NC(=O)CN(C1CCOC1=O)C(C)=O 71024,C1(C(=O)Nc2ncccc2C2CC2)CC(F)CN(C(=O)CC2CCSC2)C1 71025,C=CCC(C(=O)N1CCC1(C)CC(=O)NC1CC(C)C12CC2)OC 71026,c1(C(=O)Nc2cnn3cccnc23)ccc2c(N3CCOCC3)nccc2c1 71027,C1(C(=O)OC)CCn2cc(C(N3CCC(N4CCCC4=O)C3)=O)nc2C1 71028,c1(C(C)C)ncc(C(N2CCC(F)(C(N3CCOC(CF)C3)=O)C2)=O)cn1 71029,C1(NC(c2nc(C)n(C)n2)=O)C(CNC(=O)C(C)(C)CO)CCC12CCC2 71030,CCCC(C)(C)C(=O)N1CC(NC(C2CC2c2cccc(C)c2)=O)CC(F)C1 71031,Cc1nsc(N)c1C(N1CCC(CC(=O)NC2CC(C(C)O)C2)CC1)=O 71032,C12(C(=O)NCC(C)(C3CC3)NC(=O)CC3CC4CCC3O4)CCCC1C2(F)F 71033,c1(C(=O)NC2CCCC(CNC(C3C(CC)CCO3)=O)C2)ccn2cccc2c1 71034,c1(C(=O)NC2CN(C(CC(=O)OC)=O)C2)coc2cc(C)c(C)cc12.C12CC(C1)C2 71035,C(=O)(CC(C)CC)NC1(C)CN(C(COCCC#C)=O)C1 71036,Cc1cc(C2CC2)ncc1C(=O)NCC1CCC(C)CN1C(c1cnccn1)=O 71037,C1(C(=O)NC2(CNC(C3CC(C)(CC)C3)=O)CCCC2)CCC2(CCOCC2)O1 71038,CC1CCN(C(C2CC23CC(O)C3)=O)CCN1C(=O)CCC1CC1(F)F 71039,N1(C(CCC2(C)CC2)=O)CCC2(CO)CN(C(C3C4CC5C(C4=O)C35)=O)CC2C1 71040,N1(C(c2nn(CC)nc2C)=O)CCC(C(N2CC(O)CC2COC)=O)C(C)(C)C1 71041,CC1C(NC(=O)COc2ccc(Cl)c(Cl)c2)CCCN1C(=O)COCC(C)(C)C 71042,N1(C(c2ccc(SC)o2)=O)CCCC(CC(=O)NC(c2nn[nH]n2)(C)C)C1 71043,N1(C(C(C)OCOC)=O)CCOC(C)C1C(=O)NCCC(O)C(F)(F)F 71044,c1(C(=O)NC(CNC(c2ccc(NC(=O)OC)cc2)=O)(C)C)nn(C)c(Cl)c1Cl 71045,CCCC(CC)CC(=O)NCC1COCCN1C(=O)CN(C)CC 71046,N1(C(CCc2ccc(C)cc2C)=O)CC2(NC(C3CC3C(F)F)=O)CCC1CC2 71047,N1(C(=O)C=C2CCC2)CCCC2C1CCCCN2C(=O)CCF 71048,C1(C2(O)CN(C(C3CC3C)=O)C2)(CNC(Cn2nc(C)c(Br)c2C)=O)CC1 71049,C1(N(C)C(C2CC(C#N)C2)=O)CCCN(C(=O)Cn2cc(Br)cn2)C1 71050,C1(CNC(=O)C=CCN2CCCCC2)C=CCN(Cc2ccc(Cl)o2)C1 71051,C1(NC(c2cc(C)n(C)c2C)=O)CCC2(CC1)CC(NC(=O)C(F)(F)C(C)O)C2 71052,C(=O)(C#CC(C)(C)Cc1ccccc1)NC(c1c(C)nccn1)C 71053,c1(C(=O)NCC(CO)NC(CC(=O)NCC)=O)csc2c(Br)cccc12 71054,c1(C(=O)NC(CNC(c2c(CC)noc2)=O)(C)CO)ccc(C)c2c1CCC2 71055,N1(C(C2C(C)CC(C)O2)=O)CC2CCN(C(c3ccc(=O)n(C)c3)=O)CCC2C1 71056,Cc1scc(C(N2CC(NC(=O)Cc3ccc(C(N)=O)cc3)CC2CO)=O)c1C 71057,Cc1ncc(C(=O)NC(C)(C)CCNC(C2CC(C3CC3)=NO2)=O)cc1N 71058,C1(C(N2C(C(=O)Nc3cccc(OC)c3)(CC)CCC2)=O)OC(C)(C)OC1(C)C 71059,CCC(C(=O)OC)C(=O)NC(C(N1CC(C)(F)C1)=O)C1CCCC1 71060,N1(C(CCCOCC)=O)CCOCC(C(N2CCN(C)C(C3CC3)C2)=O)C1 71061,C(=O)(CCCCCNC(c1ncncc1C)=O)N1C(CC)CC1 71062,C(C(F)(C(=O)NCCC1CCCC1(C)C)C(C)C)NC(c1nc(OCC)oc1)=O 71063,c1(OC)ccncc1NC(=O)C(N1CCC1CNC(=O)C(C)NC(=O)C(C)(C)C)=O 71064,CC(C)CCC(O)C(=O)NCCCCCCNC(c1cn(C(F)F)nc1C(F)F)=O 71065,C1(C)(C(N(CC)CC2CCC2)=O)CNC(C)(C)C1 71066,c1(CC)cc(=NCC(C2CC2)NC(=O)CCCCc2ccccc2)[nH]c(C)n1 71067,c1(C(=O)NCC(CC)NC(c2ncn(C)n2)=O)noc2cc(F)ccc12 71068,c1(C(N(C(C)C(N2CCN(CCF)CC2)=O)C2CC2)=O)cn(C)ccc1=O 71069,C1(C(N(CC#C)C)=O)CCN(C(=O)C(C)COC(C)=O)CCO1 71070,C1(C(=O)NCC(C(C)C)OC)(NC(c2cc(O)nc(C)n2)=O)CCC(C)(C)C1 71071,C(=O)(C1CCOc2ccc(Cl)cc21)NC1CN(C(CCC(N)=O)=O)C2(C1)CCC2 71072,c1(C(C(=O)NCC(COC)NC(c2c[nH]nc2C(C)(C)C)=O)C)cccnc1 71073,C#CC1CCCC(CNC(C2(F)CN(C(C3CCC(C)(C)C3)=O)C2)=O)C1 71074,C12(NCc3c(C(=O)OCC)n[nH]c3)CC1CN(C(C1CCC(CC)CC1)=O)C2 71075,C12(CNC(C(CC)O)=O)CCC(CC1)N2C(C1CCC(=C2CCC2)CC1)=O 71076,C=CC1(NC(C2N(C(C3CCC3OC)=O)CCC2(C)C)=O)CCOCC1 71077,CC1(C)CC(C(=O)NCC(c2ccsc2)O)CCN1C(=O)Cc1ccon1 71078,c1(C(C(=O)NC(C2CCN(C(C(CSC)C)=O)C2)C)C)ccccc1C 71079,c1(-n2ccc(C(=O)NCCC(C)(C)N)n2)ccc(Cl)c(F)c1 71080,Cc1ccc(OCC(C)NC(C2CCN(C3CC3)CC2)=O)c(F)c1 71081,Nc1nc(C(=O)NCC2CC(F)(CNC(=O)C(F)n3cccn3)C2)ccc1O 71082,CCCC(CC(C)C)C(=O)NC1CN(C(c2ccn(C)c2)=O)CCC1O 71083,c1(NC(c2cnc(Br)s2)=O)ccnc(C(=O)NCc2ccccc2CO)c1 71084,c1(C(=O)NC(CNC(c2c(CCC)cccc2)=O)C)ccnc(F)c1N 71085,Cc1csc(=O)n1CC(=O)N(C1CCN(C(C23CC(C#N)(C2)C3)=O)CC1)C 71086,C1(C(N(C2CCN(C(C3(C#N)CC=CC3)=O)C2)CC)=O)CCCCC1O 71087,c1(C2N(C(C3N(C(c4ccc(=O)oc4)=O)CCOC3)=O)CC2)c(Cl)cc(Cl)cc1Cl 71088,c1(CNC(C(CO)N(C)C)=O)ccc(C(N2CCC(C)(CO)C2)=O)cn1 71089,C(=O)(C1COc2ccccc21)NCCN(CCC)C(C1(C)CC(F)(F)C1)=O 71090,n1(CC(=O)NCC2(F)CN(C(C(C)C(F)F)=O)C2)cnc2ccccc12 71091,C(=O)(CC1=CCCCC1)N1C(C(c2[nH]ccc(=O)c2C)N2CC(C#C)(O)C2)CCC1 71092,C(C(=O)N(CCCNC(C1CC1F)=O)C)N(C)CC 71093,CCC(C)CC(C(=O)NC1CC1)NC(=O)C=CCN(C)Cc1noc(C)n1 71094,c12ccc(cn1)CN2C.c1(SCC)c[nH]c(C#N)c1.C1(OC)CCCC1CNC(=O)N 71095,N1(C(C(C)CC(C)(C)C)=O)CCC2(CCCN2C(=O)C(C2CCOCC2)O)C1 71096,CCCCCCN(CC(=O)NCC(C)(CC)NC(c1coc(SC)c1)=O)C 71097,c1(C(N)=O)ccc(Cl)nc1NC(C1CCCC1NC(c1ccnc(O)c1)=O)=O 71098,O(C1CCCc2nc(C)sc21)C(C=Cc1ccc(C(CC)(C)C)cc1)=O 71099,C(=O)(C(O)C(F)(F)F)NCCN(CCOC)C(C1CCCOC1)=O 71100,c1(C(N2CC(CNC(C(CN(CC)CC)F)=O)(OC)C2)=O)cccc(F)c1C 71101,CC1CCc2[nH]c(C(=O)NCCCN(C(=O)CC(C)(C)O)C3CCCC3)cc2C1 71102,N1(CCNC(CCCCC)=O)CCCN(C(=O)Cn2cc(C(C)O)nn2)CC1 71103,C1(C)(CCNC(c2c(OC)ccs2)=O)CCN(C(C2(O)CCSC2)=O)C1 71104,C1(C#N)(C(N(CC=CC(=O)NC2CN(CCC)C2)C)=O)CC2CC2C1 71105,N1(C(CC)=O)CCc2cc(C(N3CCC(F)C(NC(=O)CSC)C3)=O)ccc21 71106,c1(C(N(C2C(N(C(c3c(CC)nc[nH]3)=O)C)CCCC2)C)=O)ccc(C)nc1C 71107,N1(c2n(CC=C)c(-c3cc4n(n3)CCCC4O)nn2)CC2NC(=O)C(=O)NC2C1 71108,C(C1C(C(=O)NCC2CN(C(=O)Cn3cnnc3)CCO2)C1(C)C)=C(C)C 71109,c1(C(=O)NCC2(NC(=O)CC(F)(F)C(F)(F)F)CC2)cc(Cl)cc2ccncc12 71110,c1(C(=O)NCC(CNC(=O)CC2C=CS(=O)(=O)C2)OC)ccc2cncn2c1 71111,C1(C2CC2)(NC(C(C)SCC)=O)CCN(C(=O)Cc2ccc(C#N)nc2)C1 71112,c1(C(N2CC(F)(C(=O)NCc3n(CC)cnc3)C2)=O)cc(Br)c(C)cc1O 71113,C(C(C)(C)CC(=O)N1CC(CC(=O)NC(c2[nH]c(C)nc2C)C)C2(CC2)C1)OC 71114,c1(CC(=O)NCCN(C(c2cc(C)n(C3CC3)n2)=O)C)c(F)cccc1F 71115,N1(C(C2CC(C#N)(OC)C2)=O)CCOCCC1C(=O)NC1(CF)CC1 71116,S(=O)(=O)(c1ccc(N(C)CCF)c(F)c1)NCC1OCC(C)C1 71117,C(=O)(C#CC1CCCOC1)N(C1CCCCN(C(C=C(C)C(F)F)=O)C1)C 71118,C1(CC(=O)N(CC#CC)C)CCCCN1C(c1cn(C)nn1)=O 71119,c1(CNC(C(CC)C)=O)ncccc1CNC(c1cc(Br)nn1C)=O 71120,C1(CCC(=O)N(CCN(C)C)C)CN(C(=O)OC(C)(C)C)CCO1 71121,C12(C(=O)N(CCNC=O)CC3CC3)CCC(CF)(CC1)CC2.C1(CO)(CO)CCCO1 71122,CC(C)(C)C(C(=O)N1CC(C#N)(c2ccccn2)C1)N1CCCC1=O 71123,c1(C(=O)NC2(CO)CN(C(C3(F)CCCOC3)=O)C2)ccc2nccn2n1 71124,c1(C(=O)NCCCN(C(C)C)C(C2CCC3CC23)=O)ccc2c(c1)CCOC2 71125,CC(CCCNC(c1cccnn1)=O)NC(C1CCCC1c1nc[nH]n1)=O 71126,n1(CCNC(c2coc(CO)c2)=O)cnc(CNC(c2nocc2C2CC2)=O)n1 71127,C(=O)(CC(O)CC1CC1)NC(C)CCCNC(=O)C(F)CNC(=O)OC(C)(C)C 71128,N1(CCC)CCC(C(=O)NCCN(C(=O)CCC2CCCO2)CC(C)O)CC1 71129,N1(C(C2C(CNC(CNC(CCC)=O)=O)OCC2)=O)CCOCC(C(C)C)C1 71130,c1(C(N2C3CN(C(C(C#C)(C)C)=O)CC2CC3)=O)ccc2c(n1)CCC(C)C2 71131,N1(C(CCc2n(C)ccn2)=O)CCCCN(C(c2cccc(O)c2)=O)C1.CC=CC#N 71132,N1(C(c2cc(Cl)nc(=N)[nH]2)=O)CCCC2(CCN(C(c3cnc(Cl)cn3)=O)C2)C1 71133,Cc1nnc2n1CCC(NC(=O)NC(C)(C)C(C(=O)O)c1ccccc1)C2 71134,c1(NC(C)CN(C)C(C2CCS2(=O)=O)=O)ncc(O)cn1 71135,C1(C(C)C(=O)N(CC(C2CCCC2)O)C)CCN(C(=O)CC2CCSCC2)C1 71136,N1(C(CCN(C(C)=O)C)=O)CC2(CC(NC(=O)C(C)(C)C(C)O)CO2)C1 71137,C(=O)(C(C)Cc1cnc[nH]1)NC1C(NC(CSCCC)=O)C1 71138,C12(C(=O)NC)CCC(C(=O)O)C1CC2.C12CC(C1(C)C)N2 71139,C(=O)(C(O)C(F)(F)F)N1CC2C(CNC(C(CCO)N(C)C)=O)(C2)C1 71140,CCCCC(CNC(C1CC(N(C(=O)CC2(OC)CCC2)C)C1)=O)CC 71141,N1(Cc2c(OC)cccc2C)CCC2(CCN(C(=O)Cn3cc(Cl)cn3)C2)C1 71142,CCCC(CCC)CC(=O)NCC1CN(C(c2ccsc2CC)=O)CC12CCC2 71143,c1(NCC(CC(=O)NCC2CN(C(C)=O)C2)O)cccc(F)c1C 71144,CN1N=C(C(=O)NCC2COC(C)(C)CN2C(=O)C=C2CCC2)CCC1=O 71145,N1(C(c2[nH]nc(OC)c2Cl)=O)CC2(CCC2NC(c2ccc(CO)cc2)=O)C1 71146,C1(C(=O)NCC(C)NC(c2c(OC)cnc(Cl)c2)=O)CCOCC12CCC2 71147,c1(C(=O)NC2CCCN(C(c3c(Cl)ccc(C)c3)=O)C2C)cc2cccnn2n1 71148,N1(C(C2CC(OC)C2)=O)CC2OCCN(C(=O)CCC(=O)NC3CCCC3)C2C1 71149,C1(C(N2CC(C#N)C(NC(c3csc(Br)n3)=O)C2)=O)CCc2ccccc2C1 71150,C1(O)(CNC(c2cc(C)nn2C(F)F)=O)CCCN(C(C2CCOC2)=O)C1 71151,c1(C(N2C3C(NC(C4CS(=O)(=O)C4)=O)CC(CC3)C2)=O)cccc2c1CCCC2 71152,C(=O)(C(C)(C)CCCNC(C1(C#N)CCCO1)=O)N1CC(CCC#C)C1 71153,CC1CCCN(C(=O)C(=O)NCC2CC(NC(=O)C(C)(C)C3CC3)C2)C1 71154,CCC(C)(C(=O)N1CCC(O)C(NC(=O)Cc2ccc(C)nc2)C1)C(N)=O 71155,Cc1cc(C(=O)NC2C3CCC2N(C(C2(CCN(C)C)CC2)=O)C3)ncc1CO 71156,c1(CC(N2CCC(F)(C(=O)NCC(C)(C)N(C)C)C2)=O)cc(Cl)cc(Cl)c1 71157,c1(CCC(=O)NC(C(=O)NC(C)CCn2cncn2)c2cccs2)nccn1C 71158,CCC(O)C(C)(C)C(=O)NCc1ncoc1C1CN(C(C23CCC(C2)C3)=O)C1 71159,CCCCCS(=O)(=O)CC(=O)N1CCCC(NC(=O)Cn2cnnn2)C1C 71160,Cn1c(C(N2CCC(C(F)F)(CNC(=O)CC(F)F)C2)=O)cc2cc(Cl)ccc12 71161,N(C1CCCn2ncnc21)C(C(CNC(c1ccc(CC)[nH]1)=O)OC)=O 71162,Cc1ccc(Br)c(CN(C=O)CC(C)(C)C(O)c2ccccc2)c1 71163,N1(C(C(C)Cn2ccnc2)=O)CCN(C(c2ccc(Cl)cc2I)=O)CC12CC2 71164,c1(CSCCNC(c2cn(CC)nn2)C)ccnc2c(Br)cccc12 71165,c12cc(OC)ccc1O2.C(C(=O)NCCOCCNC(C1CC1C)=O)SC 71166,c1(C(=O)NCC2(C)N(C(c3cc(OC)nn3C)=O)CCC2)cc(O)nc(O)c1 71167,C1(CC(=O)NCCCNC(Cc2[nH]c(=N)sc2)=O)CCCC12NC(=O)NC2=O 71168,C(C)(C)(C(C)CC(=O)N1CCC(CC(C)O)CC1)NC(C=C(COC)C)=O 71169,C=CCCCCCN=c1nc2scnc2c(NCCc2ccn(C)n2)[nH]1 71170,N1(Cc2cncc(C)c2)CCC(O)CC1C(=O)NCC1CCOCC1 71171,C1(CC#C)(C(=O)NC(CNC(c2cnn(C(C)C)c2F)=O)CO)CC=CCC1 71172,c1(C(=O)NC2CN(C(c3c(C)nsc3C)=O)CC2O)cccn2ccnc12 71173,N1(C(c2c(C)nsc2)=O)CCC2CN(C(=O)C(O)CC3CCCCC3)CC12 71174,C1(C(=O)OC)CN(C(N2CC3C=CC3C2)=O)CC1C(=O)OCc1ccccc1 71175,Cc1cc(C(N2CCSCC2C(=O)N=c2cc[nH][nH]2)=O)ccc1F 71176,c1(C(N2CCC(C)C(NC(c3nsnc3O)=O)C2)=O)ccc(C#N)c(Cl)c1 71177,C1(C(=O)NCC2C(NC(C3C(=C)C3)=O)CCC2)C(C)(C)C1(C)C 71178,N1(C(C=CC(C)C)=O)CC(O)(C(C)NC(=O)CNC(C2CCC2)=O)C1 71179,CCCCCC(CC)C(=O)N1CC(C)CC1C(=O)NOCC1CCCCC1 71180,c1(C(C)=O)c[nH]c(C(N2CCC(N(C)C(c3cc(C(N)=O)[nH]n3)=O)C2)=O)c1C 71181,C(=O)(C1CSc2ccccc21)N(C)CCNC(=O)COC(F)F 71182,C1(C(=O)NC(CNC(CN2CC(C)C2)=O)(C)C2CC2)CC(c2ccccn2)=NO1 71183,C#CC1(C(=O)NC2CCS(=O)CC2)CCN(C(=O)C(F)n2ccnc2)C1 71184,N1(c2n(CC=C)c(C(O)CC3CCCCC3)nn2)CCC2(CCOCC2)C1 71185,Cc1ccc(C(=O)NC2CCCC2NC(c2scnc2C2CC2)=O)o1 71186,C1(NC(CCc2n(C)ccn2)=O)CC12CCN(C(=O)CC1CC(F)(F)C1)C2 71187,c1(C(=O)NCC2OCCN(C(Cc3ccn(C)n3)=O)C2)cc(Cl)cc(Cl)n1 71188,N1(C(c2c(C)ncnc2)=O)CC(C2(NC(C3CC4(C3)CC(C)C4)=O)CC2)C1 71189,c1(-c2c(C)ccc(CO)c2)cnc2[nH]cc(C(=O)Nc3ccnn3CCO)c2c1 71190,CCC(C)C(O)C(=O)N1CCCC1C(C)NC(=O)C=CC=Cc1ccccc1 71191,C1(N(C(CC=CC=C)=O)CC)CCN(C(=O)CC)CC1.C1(=O)C(C2CC2)N1 71192,Cc1ccc(C(=O)NCC2C3CN(C(=O)Cc4c(C)cnn4C)CC23)c(O)n1 71193,C12(C(N(C3CN(C(C4(O)CCC4)=O)CC34CC4)C)=O)CCC(C)(CC1)CO2 71194,c1(C(=O)NC(C(CO)NC(c2cc(C)no2)=O)C)cnc2n1CCC(C)C2 71195,C1(CN(C=O)CC(c2cc(C)c(F)cc2)O)CCS(=O)(=O)C1(C)C 71196,Cc1cc2cc(C(=O)NC3CC4(C3)CC4C(=O)NC3CCC3)oc2cc1C 71197,C(=O)(C#CC1CCCCO1)NC1CC(C)(C)CN(C(=O)CC(F)(F)F)CC1 71198,c1(C(=O)NCC2(OC)CCN(C(CC(C=C)(C)C)=O)C2)ccc2c(C)[nH]nc2c1 71199,C1(CC)(NC(=O)CSS(C)(=O)=O)CCCN(C(c2cncc(OC)c2)=O)C1 71200,C(c1ccncc1)=CC(=O)NCC(C(=O)NC(c1nc[nH]n1)CC)N(C)C 71201,N1(CCNC(C2(CCCC)CC2)=O)CCCN(C(=O)CC2CC2C(F)(F)F)CC1 71202,c1(COC)nc(C)ncc1C(=O)NCC1CCC1NC(c1ccc(CF)cc1)=O 71203,CC(C)(C(=O)NCC1CCN(C(C2(c3cccnc3)CCC2)=O)C1)C1CCCC1 71204,c1(NCC2(C)CCN(C(C3CC(CCC)OCC3)=O)C2)cc(C)nc(Cl)n1 71205,c1(C(c2n(C3CC(F)(F)C3)nnn2)NC2CC2C(F)(F)F)cccc2c[nH]nc12 71206,c1(C(C)C)nnsc1C(C)NC(=O)NC(CCCCOC(C)(C)C)C 71207,N1(C(c2occ(S(C)(=O)=O)c2)=O)CC2CCCN(C(c3n[nH]c(=N)s3)=O)C2C1 71208,c1(C(C(N2C(CNC(C3(OC)CC3)=O)CCCC2)=O)O)ccc(Cl)cc1F 71209,CCCC(C)(O)C(=O)N1CCC(C)(CC(=O)NCC2(O)CCN(C)C2)C1 71210,N1(C(c2scc(C)n2)C(=O)NC2CCCC2)CCc2cc(O)ccc2C1 71211,C1(C(=O)NC2C(C)CN(C(=O)CCc3cncc(F)c3)C2)CCC2C(C1)C2(F)F 71212,CC(C)CC(O)C(C)C(=O)N1CC(F)(F)CC1C(=O)NC1C=CCCC1 71213,C1(C(N2CCC(OCCNC(=O)CSC(F)F)C2)=O)C(C(F)(F)F)C1[N+](=O)[O-] 71214,N1(C(c2cnc3cnccn23)C(=O)NCC2CC2)CCc2c(Br)cccc2C1 71215,c1(C(OC)OC)ccc(C(=O)NC(C2CCOC2)CNC(=O)CN(C)C)c(O)n1 71216,c1(C(N2CCC3C(NC(C4N(C)C(=O)CC4)=O)C32)=O)cccc2c1nc(O)n2C 71217,C1(CC(=O)NC2(CN(C(=O)CP(C)(C)=O)C)CC2)CCC12CCC2 71218,CCCCCCCC(C)CNC(=O)NC1CCN(c2ccc(Cl)cc2)C1 71219,C12CC(C)N(C1)C2.c1(C(=O)NC(CSCC(=O)OC)=O)n[nH]c(CO)n1.C(C)C 71220,c1(CC(=O)NC(CC)CNC(C2SCCS2)=O)ccc(C)nc1 71221,c1(CC)ncnc(N2CCSC(C(=O)Nc3sccc3OC(F)F)C2)c1F 71222,Nc1c(O)ccc(Cl)c1C(=O)NCC1CCCN(C(=O)C=CC2CCC2)C1 71223,C1(C)(C(=O)NCCN(CCOC)C(c2ccc[n+]([O-])c2)=O)CNC(=O)C1 71224,C(=O)(C(F)(F)C(F)(F)OC(F)(F)F)NC1CN(C(C2CCN(C)C2)=O)C(C)(C)C1 71225,Brc1ccc(C2CCN(CCCCc3nccs3)CC2)nc1 71226,O=S(=O)(c1ccc(Br)c(Cl)c1)Nc1cc(-c2ccc(CO)nc2)ccn1 71227,c1(C(N2C(C(C)NC(=O)CO)CCCC2)=O)cnc2c(c1)NC(=O)CS2 71228,c1(C(=O)NC2CN(C(C3(COC)CC3)=O)CC(O)C2)cnc2cc(C)nn2c1C 71229,C1(NC(Cc2c(C)nn(C)c2)=O)CC2CCC1N(C(c1nnc(O)nc1O)=O)C2 71230,Cn1cnc2sc(C(=O)NC3CC4(C3)CN(C(=O)C(=O)NCC(F)(F)F)C4)cc12 71231,c1(COC)nc(NCc2cccc(F)c2Br)cc(N2CCN(CCF)CC2)n1 71232,C1(C(=O)Nc2ccc(-c3cn(CCC(=O)NC)nn3)cc2)CCCCC1(C)C 71233,C(CC(C)C)(C(=O)NCC(C)n1cncn1)ONC(=O)C1(CCCC)CC1 71234,c1(OC)ncccc1S(=O)(=O)NC(=O)C=C1CCC(C(C)(C)C)CC1 71235,N1(C(CCCNC(N)=O)=O)CC2CC1CCC2NC(C1C2C3CCC(C3)C12)=O 71236,Cc1cc(O)cc(=O)n1CC(=O)N(C)CC1CCN(C(C2C=CCC2)=O)C1 71237,n1(CC(=O)NCCNC(C2CCC3(CCOC3)O2)=O)sc2ccccc2c1=O 71238,C(=O)(C(F)(F)Sc1cnn(C)c1)NCCOCCN(C(=O)Cc1ccn(C)n1)C 71239,C(CCNC(C1(C)CS(=O)(=O)C1)=O)(C(C)C)NC(C(COC)O)=O 71240,c1(C(=O)NCCN2CCC(NC(C(CC)C)=O)CC2)ccc(Cl)c(Cl)c1F 71241,C(=O)(C(C(C)(C)C)OC)N1CCC2(C1)C(=O)NO2.C1(C(=O)OC)CC2C(C1)C2(C)C 71242,C1(NC(c2ccc(-n3cncn3)cc2)=O)CCCC(C(=O)Nc2ncc(F)s2)C1 71243,Cc1csc2nc(CN3CCC3C(=O)N=c3ccc(Br)n[nH]3)cc(=O)n12 71244,Cn1c(C(N2CCCC2C2CCCN(C(=O)CSC(F)F)C2)=O)cnc1Cl 71245,c1(CNC(C23CCC2C3)=O)ccc(C(C)=O)c(N)c1.C12(CCC1)C(=O)NC2 71246,c1(C(=O)NCC2(O)CN(C(=O)Cc3cccc(Cl)c3)C2)cccc2oc(O)nc12 71247,N#CCCC(=O)NC(CC(N)=O)c1cn(C2COCC2n2cccn2)nn1 71248,N1(C(CCCNC(N)=O)=O)CCCC2CN(CCCC3CCOC3)CC12 71249,C(=O)(CS(=O)CCC(F)(F)F)N1CCC(N(C(CCC2CCN(C)CC2)=O)C)C1 71250,C#CCC(C)(C(=O)N(CC(O)CCC)C)NC(=O)C1=CC(C)(C)C1 71251,C1(CNC(CC(C)C)=O)CN(C)CCN1C(=O)CCc1ccc(Br)s1 71252,C1(NC(c2cccc(OC)c2)=O)CN(C(c2cc(C)ccc2N)=O)CC2(CC2)C1 71253,c1(C(=O)NCC2C(NC(CSCCC(C)C)=O)CCC2)ccc(Cl)c(Cl)c1 71254,N1(C(C2CCSC2(C)C)C(=O)NC)CCNC(=O)CC12CCC2 71255,c1(C(N2CC(CN(C(C(C)OCCOC)=O)C)C2)=O)n[nH]c2c1CCCCC2 71256,C1(CN)CCCN(CC(O)CC2CCCO2)C1 71257,N1(C(c2cnc(Br)n2C)C(=O)Nc2c(C)cccc2)CCCN(C)C(=O)C1 71258,CC1CCSCCN1Cc1cccc(-c2ccc(F)cc2)c1 71259,CC(C(=O)NCCC1CN(C(=O)CCc2nncn2C)CCO1)C(F)(F)C(F)F 71260,C1(OCC)(CNC(c2sc3nccn3c2C)=O)CCCS(=O)(=O)C1 71261,C1(CNC(C2(CC(C)=O)CC2)=O)(CNc2ccncn2)CC12CCC2 71262,CC(C)CC(C(=O)NC1CC(C)OC1=O)NC(C1CNC(=O)O1)=O 71263,C(=O)(C1=CCOC1)NC(C)CC1CN(C(=O)C(C)c2cccs2)C1 71264,C1(NC(C2(CC=C)CN(C(c3cc(CO)oc3C)=O)C2)=O)C2CCC(C2)C1(C)C 71265,CC(CNC(=O)CC1(N2CCCC2)CC1)(CO)NC(=O)CCC1CCC(=O)C1 71266,CC(C)(C)CCCCNC(C1COCCC1NC(=O)Cc1cccnc1F)=O 71267,CCCC(F)C(=O)N1CCC(CC(C)NC(C2(CCC)CC2)=O)CC1 71268,N1(C(CCc2cc(C)on2)=O)CCC2CCC(NC(=O)CCc3cnc[nH]3)C1C2 71269,N1(C(=O)NC2C(CC=C)COC2)CCC(F)C(F)C1 71270,N1(C(=O)CCC(F)F)CCN(C(=O)CSc2cccc(F)c2)C(CO)C1 71271,c1(C(=O)NCC2N(C(C3CCCCS3)=O)CCC(C)C2)cc(S(N)(=O)=O)ccn1 71272,C1(COC)(NC(=O)Cc2csnc2C)CN(C(C2CC(OC)(OC)C2)=O)C1 71273,C1(CNC(C(C)O)=O)CC2(CCN(c3ncc(S(C)(=O)=O)cc3Cl)CC2)CO1 71274,C1(NC(c2cc(-c3nc(C)sc3)sc2)=O)CN(C(C2COC(=O)C2)=O)CC1F 71275,Cc1c(C(=O)NCC2CC(C)N(C(c3ccoc3Cl)=O)C2)cccc1C#N 71276,C1(NC(=O)COCCOCCO)CCCC(CNC(=O)CC2CCSCC2)C1 71277,c1(C(N(C2CCCN(C(CCNC(COC)=O)=O)C2)C)=O)ccc(S(N)(=O)=O)[nH]1 71278,c1(NC(C2C(NCc3c(C#N)c(F)ccc3)CCC2)=O)c(O)cccc1[N+](=O)[O-] 71279,c1(C(N(C)CCNC(c2ccccc2C2(C)CC2)=O)=O)ccc(Cl)c(O)c1 71280,c1(C(N2C(CN(C(=O)CC3CCC4CC4C3)C)CCC2)=O)cc2sccc2s1 71281,C1(NC(C=CC)=O)CC(C)CN(c2nccc(Oc3ccccc3)n2)C1 71282,O=C1CCCCCN1Cc1cn(CC2CCN2C(=O)CC2CSCCS2)nn1 71283,N1(C(c2c(CC)n[nH]c2)=O)CC(OC)CC1C(N1CCC(O)(CN(C)C)C1)=O 71284,c1(COC(C2C(Nc3nc(C)nc(O)c3)CCCC2)=O)[nH]c2ccccc2c1Cl 71285,c1(OC)cccc(OC(=O)N(CC(C)C)CC2CC(F)(F)C2)c1 71286,CCCCCC(CC)C(=O)OC(C1CCOCC1)COC 71287,N1(c2c(F)cnc(OCC)n2)C2CCC1CC(NC(c1cc(F)ccc1I)=O)C2 71288,Cc1ccc(O)c(CNC(=O)CCN(C(C2CC3CC3C2)=O)C2CC2)c1 71289,N1(C(COC(C)C)=O)CCN(C(C2CCC(N(C)C)C2)=O)C(C(C)(C)C)C1 71290,N1(C(c2c(C(C)(C)C)noc2)=O)CCCC(C2CN(C(=O)C=CCF)C2)C1 71291,C1(O)(C(N2CCC(O)(C(C)NC(C(C)CC(F)F)=O)C2)=O)CN2CCC1CC2 71292,N1(C(c2cc(C)ns2)=O)C2CCC1CC(NC(c1cncc(N3CCCC3)c1)=O)C2 71293,c1(CC(N2CC(NC(C3N(CCC)CCCC3)=O)C2)=O)cc(Br)ccc1OC 71294,C1(NC(CCC(C)(C)OC)=O)CC2CCC(C1)N2C(C)C 71295,C1(OC)(CNC(=O)C(c2cccnc2)C)CCN(C(=O)CC2CCCS2(=O)=O)C1 71296,C#Cc1cn(C)nc1C(=O)NCC(CC)NC(c1ccc(N)cc1Cl)=O 71297,C1(NC(C)=O)CCC(C(N2CCC(C)(NC(=O)CCCNC(N)=O)C2)=O)CC1 71298,C1(CNC(c2csnn2)=O)(CO)CCN(C(c2occc2C2CC2)=O)C1 71299,Cc1cccc2c1CCOC2C(=O)NC1CCCN(C(c2nn(C)cc2Cl)=O)C1 71300,c1(C(=O)NCC2(CN=c3cc(COC)nc[nH]3)CC2)ccc2c(c1)COCC2 71301,c1(NC(C2COCCN2C(=O)CCCCC2CC2)=O)cncc(CO)c1 71302,c1(CC)ccc(CC(=O)NCC(c2cccc(Cl)c2)NC(=O)CP(C)(C)=O)cc1 71303,c1(C(=O)NC(CC)CN(C(=O)CC2CC2(C)C)C)cnc(-c2cccnc2)s1 71304,c1(C(N2CCCC(N(C(c3c(COC)cc[nH]3)=O)C)C2)=O)ccc([N+](=O)[O-])[nH]1 71305,C(C1CCN(C(=O)C2=CCCCO2)CC1)=CC(=O)NCc1cc2n(n1)CCC2 71306,CCC(O)(CNC(=O)CC(C)(C)NC(=O)C(C)(O)C1CC1)CC 71307,c1(CC)ccc(C(N2CCC(OC3CCC3)C2)=O)cc1C#N 71308,c1(NC(c2cc(Sc3ncccn3)on2)CC)cccc(NC(=O)NO)c1 71309,N1(C(C=CCN(CC#C)C)=O)CCN(C(=O)Cc2ccc(SC)cc2)C(C)C1C 71310,N1(C(C(C)C2CC2)=O)CC2CCN(C(C34CCC(C(F)F)(CC3)C4)=O)CC2C1 71311,c1(N(CCNC(c2c3c(nn2C)CCCC3)=O)CC)ncnc2c1c(Br)nn2C 71312,c1(N2CC(CN(C(C3C(C)C3)=O)C)C2)nc(Cl)nc2[nH]ccc12 71313,C(c1nccs1)=CC(=O)NCc1nc(C(=O)NC2COC(C(F)F)C2)co1 71314,C1(C)(CCC(=O)N(CCCC)CCCO)CN(C(=O)Cc2csc(C)n2)C1 71315,C1(CNC(C(CC)=CC)=O)C2CCC(C2)N1C(=O)CCC1CCCC1 71316,C12(C(=O)NC(CNC(C34CCC(OCC)(CC3)C4)=O)(C)C)CCCN1CC(O)C2 71317,CS(=O)CC(S(C)(=O)=O)NC(c1cccc(Cl)c1)c1nocc1C(C)(C)C 71318,C1(C(=O)NCCC2(C)CCN(C(CSCC)=O)C2)CCc2nc(C)nn2C1 71319,C(=O)(CC(CC)C(C)(C)C)NC1C(CCC)CN(C(=O)CONC(=O)OCC)C1 71320,C1(C(C(=O)NC(C(C)C)CN(CC(=O)N(C)C)C)C)CCCC(F)(F)C1 71321,C1(CCCNC(C2(C(C)(F)F)CC2)=O)CCN(C(c2ccncc2O)=O)CC1 71322,C12(CN(C)C(=O)NCc3cnn(C)c3)CCCC1OCC2 71323,c1(NC(C(=O)NCC2C(OCC)COC2)=O)ccc(Br)cc1[N+](=O)[O-] 71324,n1(CC)nc(C(=O)NC2CCCN(C(C3(CCOCC)CCC3)=O)C2)cc1C 71325,c1(OCC(N2CCC(C)(CNC(COCCCOC)=O)C2)=O)ccc(F)c(F)c1 71326,C(=O)(CCP(C)(C)=O)NC(C(C)C)C(=O)NCCC1(C)CCCO1 71327,n1(CCC(=O)N(C)CC2N(C(C(C)C#N)=O)CCCC2)cc[nH]c(=O)c1=O 71328,c1(CCC(=O)NC(CNC(Cn2c(C(C)C)ncc2)=O)C(C)C)ccccc1Cl 71329,C1(C(=O)NC(C)C(=O)NCCO)CCC2(CO1)CN(C(=O)OC(C)(C)C)C2 71330,C1(C(=O)OC)CN(Cc2cc(C3CC3)ccn2)CCC1C(F)(F)F 71331,C1(C(=O)Nc2scc(C)c2C(N)=O)CCN(Cc2cnn(C)c2C)CC1O 71332,c1(CCC(=O)O)ccc(CNC2(c3ncccc3F)CCOCC2)cc1 71333,c1(Nc2ccc(C(N(C)C)=O)cc2)ccc(S(=O)(=O)CCS(C)(=O)=O)cc1 71334,c1(OCC)cc(C(=O)NCCN(C(=O)C2=CCSC2)c2cccc(Cl)c2)ccn1 71335,Cc1cc(C(N2CC3CC2CN3C(=O)C(n2ccnc2C)C)=O)c2[nH]cnc2c1 71336,c1(C(=O)NCC(CNC(c2c(C)ncs2)=O)(C)F)c(C)nn2ccccc12 71337,CC(C)(CS(C)(=O)=O)C(=O)NCC1CCC(NC(c2cc3n(n2)CCCN3)=O)C1 71338,C=CC1CCCCN1C(C1(C)CCN(C(c2nnn(C)c2C)=O)CC1)=O 71339,Cc1noc2ncc(C(=O)NC3CC(CNC(c4cccc[n+]4[O-])=O)C3)cc12 71340,C(=O)(C(C)(C)C(O)C(C)C)N(CCC(=O)NC(CC)CC(F)(F)F)CC=C 71341,c1(NC(c2nnnn2C(C)C)(COC(C)=O)C)cc(C(C)(F)F)ccc1Cl 71342,c1(C(N(CCN(C(C(C(C=C)C)C)=O)C)C)=O)ccc2c(=N)[nH]cnc2c1 71343,Cc1cc(C(=O)NCC2(C)CCCN2C(=O)CC(C)C2CCCC2)c(O)nn1 71344,CC1(C)CN(C(=O)CCCS(N)(=O)=O)CC(CNC(C2CC3(CSC3)C2)=O)O1 71345,CC1=CCC=CC1C(N1CCC(C(C)NC(C2CCC(=O)N2)=O)CC1)=O 71346,N1(C(c2nc[nH]n2)CC)CCc2cc(F)c(F)cc2C1 71347,c12cc(oc1C)NC2=O.C1(CNC(COCC=C)=O)COC(C(=O)OC)C1 71348,C=C1CCN(C(=O)CCCCSCC)C(C(=O)N(C(CC)CO)C)C1 71349,C1(NC(=O)CC2CCCCC2)CN(C(=O)C(F)n2cccn2)C2CCCCC12 71350,C1(C(N(C)CC2(CNC(c3c(C)scc3)=O)CC2)=O)CCc2nncn2CC1 71351,c1(C(N2C(C(N3CCN(S(C)(=O)=O)CC3)=O)CC3CC32)=O)ccc(F)c(F)c1Cl 71352,N1(C(C)C)CCCC1C(=O)NC1CCCC1NC(=O)C(C)(C)c1ccnn1C 71353,N1(C(C2C(C)C2C)=O)CCCOC(CNC(c2cc(Br)cn2C)=O)C1 71354,CC1(C)CC(=O)NCC1C(N1CCC(OCCNC(C2CC(=O)N2)=O)C1)=O 71355,N1(C(CC(=C=C)C)=O)CCN(C(=O)Cn2ccc([N+](=O)[O-])n2)CCC1C 71356,N1(C(CC2ON=C(CC)C2)=O)CCCCCC1C(=O)NCCc1cnc(C)[nH]1 71357,C12(NC(c3ncn(CC)c3)=O)CCCC1N(CC1CCCCO1)CC2 71358,C(=O)(CC(C(F)(F)F)NC(C1CC2CC2C1)=O)N(CCCCOC)C 71359,N1(C(CC2ON=C(C)C2)=O)CCC(NC(C2CN(c3nnnn3C)C2)=O)C(C)(C)C1 71360,CC1CC(N(C(=O)C(c2ccoc2)NC(=O)COCCCN=[N+]=[N-])C)CCO1 71361,N1(C(c2c(OCC)cccc2Cl)=O)CC2(CCCN2C(C2(C)CCCCC2)=O)C1 71362,c1(-n2c(C(c3cc(=NC)[nH]cc3)NCCC(F)F)nnn2)ccc2c(c1)CCC2 71363,C1(C(=O)Nc2cc(-c3cc(F)cc(F)c3)[nH]n2)CCC(O)C(O)CC1 71364,N1(C(CCC(C)(C)C)=O)CCC2(CCC2NC(c2csc(C(F)F)c2)=O)CC1 71365,C(=O)(C1CCCc2nncn21)NC1CCCCN(C(c2c(=N)[nH]cnc2)=O)C1 71366,C12COCCN(C1)C2=O.C1(C)(NC(C=CC(=O)N(C)C)=O)CCC1 71367,n1(CC)cnc2nc(N3CCC(C)(CC)C3)nc(NCC3CC(C(F)(F)F)C3)c12 71368,N1(C(c2cncc(C)c2)=O)CCC(C)C(N(C)C(c2cn(C3CC3)cn2)=O)C1 71369,Cc1cc(=NC2CCCc3n[nH]cc32)[nH]c(N2CCC(F)(CF)C2)n1 71370,N1(C(C2(C)CCCC2)=O)CC(NC(C2(Cc3cnn[nH]3)CCC2)=O)C(CO)C1 71371,C1(NC(CC2C(C)(C)C2(C)C)=O)CCCN(C(c2nc(F)ccc2Cl)=O)CC1 71372,N1(C(c2cc(C)nn2C)=O)CCC(CNC(=O)C(O)CC(C)(C)C)C(F)(F)CC1 71373,c1(C(N2C(C(=O)NC(CC)C(C)O)CC(O)C2)=O)cc(F)cc(Br)c1F 71374,CCN=c1[nH]cc(C(=O)NC(C)(C)CNC(=O)Cc2ccc(OC)cc2F)s1 71375,c1(CNC(CC(C(C)C)O)=O)cnn2c1CN(C(c1cncc(O)c1)=O)CC2 71376,C12CCC(CC1)N(c1nnc(O)s1)C2=O.C1(c2cccs2)(C(=O)OC)CCCC1 71377,C1(C)(CC=C)CN(C(=O)CCC2CCC(NC(=O)C(C)SCC)C2)C1 71378,c1(CC)nc(C(=O)NCC2CCN(S(C)(=O)=O)C2)c(Br)s1 71379,C1(C(=O)NCCn2cc(C3CCOC3)cn2)CCN(CCn2cncn2)CC1 71380,C1(C(N(CCC(=O)NC2CC23CCC3)CCCO)=O)CC(C2CC2)=NO1 71381,Cc1cccc(Cl)c1C(=O)NC1CS(=O)(=O)CC1NC(C1CC2(C1)CC(C)C2)=O 71382,c1(C(=O)NCC2OCCC(NC(C3C(C)C3)=O)C2)ccnc2c1CCC2 71383,N1(C(C(c2n(C)ccc2)=O)=O)CC2CCC2(C(=O)Nc2ccc(O)cc2Cl)C1 71384,c1(CN2CCC(C(N(CCC(=O)OC)C3CC3)=O)CC2)cc(Br)c(O)c(Br)c1 71385,Cc1ccccc1-n1nnnc1C(c1cc(OC)ns1)OC(F)F.c1csnc1C 71386,C1(CNC(C)=O)C2CCC1CN(C(=O)Nc1c(C)nn(Cc3ccccc3)c1Cl)C2 71387,N1(C(CONC(C2OCCN(C)C2)=O)=O)CCC(O)CC1C(N)=O 71388,c1(C(=O)NC)ccc(C(=O)NC2CC2NC(c2cccc(C)c2C)=O)cc1F 71389,[N-]=[N+]=NC1CCN(C(=O)C(O)CCNC(c2ccc(O)cc2F)=O)C1 71390,C(c1ccc(F)cc1F)=CC(=O)NC(C(C)NC(=O)CC(C)(C)O)CO 71391,c1(OC)ccc(C2(C(=O)NCCCN(C(=O)C=Cc3cncs3)C)CC2)cc1 71392,c1(C(N2C(CNC(CCCC=C)=O)C(C)CC2)=O)cc(Br)c2ncccc2c1 71393,C1(CN(C(C(N2CCC(C)C2)=O)=O)C)CCCCN1C(=O)CC1CC1 71394,c1(C(=O)NC(CNC(C(C(C)C)OC)=O)C(C)C)cncc(P(C)(C)=O)c1 71395,c1(NC(CC(C2CC2)NC(c2cccc(C)c2O)=O)=O)cccc2c1CCO2 71396,N1(C(C2(NC(CC(COC)C)=O)CCN(C)C2)=O)CC(=O)NCC12CC2 71397,C1(NC(CCC=C(C)C)=O)CCCCN(C(C23COC(CF)(C2)C3)=O)C1 71398,C1(COC)(NC(C2CCSC2)=O)CCN(C(=O)CCCSC)C1 71399,C1(NS(CC2CCC(C)(C)CO2)(=O)=O)CCCC2(CCC2)C1 71400,C(=O)(CCC(=O)N1CCN(C(=O)CCC2NC(=O)NC2=O)CC1)N(CC)CC 71401,N1(C(CCN(C)CCNC(=O)CCC2CC2(F)F)=O)CC(=O)N(C)C(=O)C1 71402,C(c1sc2ccccc2c1Cl)=CC(=O)NCC(O)CO 71403,N1(C(CC2C(=O)NC(=O)N2)=O)CC2CCN(C(=O)CCc3cncc(F)c3)C2C1 71404,C(=O)(CCC(C)C)NC12CC(CNC(C3(CC)CCCO3)=O)(C1)C2 71405,N1(C(CCCOC)=O)CC(CNC(=O)C(C)(O)C(C)C)CC(C)C1 71406,C1(NC(C2(C)CCC(F)(F)CC2)=O)CN(C(=O)C(N)=O)Cc2nccn2C1 71407,Cc1cnc(N)c(C(=O)NC2CCC(C)N(C(c3coc(Br)c3)=O)C2)c1 71408,C=CC1(CC(=O)NCC2CN(C(=O)C=CCO)CCN2C)CCCCC1 71409,C1(C(N2CC(C)(CNC(c3c(C)nn[nH]3)=O)OCC2)=O)C2CCC3C(C2)CC13 71410,Cc1ccsc1C(=O)NC1(C(=O)NCCCC2(C)CC2)CC1(C)C 71411,CC1(N=c2[nH]c(Cl)nc3ccccc23)CC(NC(c2c(Cl)ccc(F)c2Cl)=O)C1 71412,CC1CC(NC(c2ccc(C3CC3)s2)=O)CN(C(C23CCC(CC2)CO3)=O)C1 71413,c1(OC)cc(N2CC3CC2CN3Cc2cccc(Br)c2Cl)nc(OC)n1 71414,N#CC1(C(=O)NC(CO)C(F)F)CC12CCOCC2 71415,N1(C(CSCCC(C)C)=O)CCCC(O)(CCNC(=O)CC2CCCN(C)C2)C1 71416,C1(c2ccccc2)(NC(C2C(C#C)C2)=O)CCN(C(c2cc(Cl)cs2)=O)CC1 71417,CCC(CN(C)C)CC(=O)NC1CCC(CNC(C2CCN(C3CC3)C2=O)=O)C1 71418,n1(C(C)C)ccc(C(=O)NC(C(=O)NCC2=NOCC2)C2(C)CC2)n1 71419,c1(CNC(C(C)Cn2cccn2)=O)ncc(C(=O)NCC(CO)N(C)C)cn1 71420,Cc1c[nH]c2ncnc(N3CCC(C)C3CNC(c3ccc(S(C)=O)cc3)=O)c12 71421,CC(Cn1ccnc1)C(=O)NCc1cc(C(=O)NCC(O)C(N)=O)cs1 71422,C1(NC(C(F)=CC)=O)CCOC1C(=O)NCC(C)(F)CNC(=O)OC(C)(C)C 71423,n1(C2CCN(C(=O)C(O)CN3CCCC3)CC2)cnc2c1CCN(C(=O)CO)C2 71424,C1(CNC(c2c(C)nc(O)[nH]2)=O)CCN(C(C2CCC(=O)O2)=O)C12CCC2 71425,CCC(CC)C(=O)NCc1cccc(C(=O)NCc2ncnn2C(C)C)n1 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71443,C(C(C)(C)CC(=O)N1CC=CC(O)C1)NC(C(C)OC(C)(C)C)=O 71444,C(=O)(C1=NN(c2ccccc2)C(=O)CC1)NCC1N(C(C2ON=C(C)C2)=O)CC1 71445,c1(C(=O)NCC2(CNC(C(=O)NCCC(N)=O)=O)CC2)cc(CCCO)on1 71446,N1(C(C(C)OC)=O)CCC(C)(NC(=O)CC(C)CNC(=O)OC(C)(C)C)CC1 71447,N1(C(C(CCCC)=O)=O)C(CO)CCC12CCC2.C1(CC)CCC(=O)N1 71448,C(=O)(C(C)(C)C1=CCN(OC(=O)OC(C)(C)C)CC1)NC(C)CCC1CCCO1 71449,C1(N2CC3C(C)C3C2)CCCN(CC(=O)OCCO)C1=O 71450,c1(CC(=O)NC2CCC(CNC(=O)Cc3ccc(Cl)cc3)C2)ccc(O)c(Cl)c1 71451,C(CC(=O)NNC(=O)c1ccccc1)C(=O)NC(C)CCN1CCCCC1 71452,Cc1nc(S)nc(C)c1CCC(=O)NC(CNC(C1CC(C#N)C1)=O)CC(C)C 71453,C(CCC(=O)NC(c1ccoc1)C)(C(C)C)NC(c1cc(OC)n[nH]1)=O 71454,c1(CC)cccc(C(=O)NCC2CCC(NC(C3(COC)CC3)=O)C2)n1 71455,C12(C(=O)NCC(c3ccccc3)NC(=O)Cc3ccco3)COCC1C2(F)F 71456,C(=O)(C(C)C(O)CC(C)C)N1CC(C(=O)NC23CCN(CC2)C3)(CC)C1 71457,C12(C(=O)NC(C)(C)C)CC(NC(=O)OCC(F)(F)F)(C1)C2.C1CCN1 71458,CCCCN=C(NCCC(=O)NCCC)N1CCc2ccc(F)c(F)c2C1 71459,c1(C(=O)NC(CC)CNC(C2(CO)CCCO2)=O)cc(C)cc2c1NCCC2 71460,O(NC(=O)CCCC1CCCC1)CC(=O)NCc1cc(O)cc(F)c1 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71478,Cc1cn(C)nc1C(=O)NCc1nc(C(=O)Nc2cncc(F)c2)c(C)o1 71479,N1(C(CN(C)C(c2cccs2)=O)=O)CCN(C(c2cc(Cl)cn2C)=O)CC(O)C1 71480,C(=O)(C(C(CC)CC)NC(c1occc1CC)=O)NC(CC=C)CC(=O)OC 71481,C1(C)(CCCC(=O)NCC2C(NC(c3nccc(OC)c3)=O)C2)NC(=O)NC1=O 71482,N1(C(CC(CCSC)O)=O)CC2(C1)CN(C(c1nocc1C(C)C)=O)CC2CO 71483,CCCCC(O)C(C)C(=O)NCC1CN(C(c2cc(O)ccc2C)=O)CC1O 71484,C(CCCCN=c1[nH]c(N(C)CCn2cccn2)nc(=N)[nH]1)OC 71485,CC(CO)C(=O)NCC1(C(c2ccoc2)=O)CC1.C123CC(C1)(C2)CNC3=O 71486,c1(N2CCCC(N(C(=O)CN3CCCC3=O)C)CC2)nc2ccc(F)cc2s1 71487,N1(S(CCC)(=O)=O)CCN(CC)CC1.c1(C2CC3(CC3)N2)nnnn1CCOC 71488,C(=O)(C1=COCCC1)NCCN(CCOC)C(C1CCCC1CN(C)C(C)C)=O 71489,C1(C)(C(N2C(C)CC2C(=O)NC23CC(F)(C2)C3)=O)CC(C)(C)C1 71490,C=C(CNC(=O)C=Cc1cocn1)CCNC(c1coc(-c2ccccn2)n1)=O 71491,c1(SC(C(=O)NC2(CN(C(c3cnc(SC)[nH]3)=O)C)CC2)C)ccc(C)cc1 71492,C1(C2CCN(C(c3ncn(C)n3)=O)C2)(NC(c2ncn(C)c(=O)c2)=O)CC1 71493,C1(C(N2CC(OC)C2)=O)CCC2(CC2)N1C(=O)CN1CCNC1=O 71494,C1(NC(c2c(C)sc(C(C)N)n2)=O)CC1C1CCOCC1 71495,Nc1cc(C(N2CC3CC2CC3CNC(C2CCCCS2)=O)=O)cnc1N 71496,C1(C(=O)NC2CC(C)(NC(CC3CCCC(OC)C3)=O)C2)CN2CCN1CC2C 71497,N1(C(c2cc(=O)cc[nH]2)=O)CCC2(CCCN2C(C2CCCS2)=O)C1 71498,c1(NC(C2C=CC(NC(=O)CCc3ccc(F)cc3)C2)=O)ccc(Cl)cc1F 71499,C1(NC(CC=C)=O)CC(F)CN(C(=O)Cc2n[nH]c(=N)s2)C1 71500,N1(C(C2N(C)CCOC2)=O)CCN(C(=O)CCN2C(=O)CCC2=O)C(C2CC2)C1 71501,Cc1cc(C(N2CCCC2Cc2cn(CC(C)O)nn2)=O)c(Br)s1 71502,c1(C(N2CC(N(C)C(C3CC3OC=O)=O)C2)=O)cc(C2CC2)on1.C(C)(C)C 71503,N1(C(C=CCN(C)CC)=O)CCC(NC(=O)CN2CCC(CO)CC2)C(O)C1 71504,C1(CC(=O)NC2(CC=C)CCCC2)COCCN1C(=O)CC1OCCCO1 71505,C1(O)(CN)CN(C(=O)C(C)(O)C2CCC2)C1.n1(C2(C(=O)OC)CCC2)ccnn1 71506,N1(C(C2CCN(C)CC2)=O)CC2CCCC1(CNC(c1cc3cscc3s1)=O)C2 71507,N1(C(C(CCC)OCC)=O)CC2(CCN(C(C3CCCS(=O)(=O)C3)=O)C2)C1 71508,N1(C(C2(C)CN(C(c3cccc(O)n3)=O)C2)=O)CCCN(CCO)CC1 71509,CC(CC1CC1)C(=O)NCCC(=O)N(C)Cc1ccsc1 71510,C(=O)(CC(F)(F)CC(=O)Nc1cc(C(F)(F)F)cc(C2CC2)c1)OC 71511,N1(C(Cc2c(C)cco2)=O)CCN(C(c2c(C)nn(C)c2C)=O)CC1C(C)C 71512,C1(N(C(CCCC(C)=O)=O)C)CCN(C(C2CCC(C)=C(C)C2)=O)CC12CC2 71513,C(=O)(CC(C)C(=O)N1CC2C(N(C)C(c3cnc4sccn34)=O)C2C1)OC 71514,Cc1ccc(C(N2CCC(C)C(CNC(c3ccncc3)=O)C2)=O)cc1Br 71515,Cc1cnc(CNC(C2(NC(=O)CCc3ccc(C)o3)CC2(C)C)=O)cn1 71516,c1(C(N(C(CNC(C(CC)OC2CCCC2)=O)C)C)=O)nn(CC)cc1[N+](=O)[O-] 71517,c1(CC(=O)NC(C(C(C)C)NC(=O)CCNC(=O)CO)C)ccc2nn[nH]c2c1 71518,C#CC1CN(C(=O)C(C2CC2)OCC)CCN1C(c1[nH]ccc1COC)=O 71519,C(=O)(C(CNC(=O)C(OC)OC)C(C)(C)C)Nc1c(OC)cc(C)cc1 71520,Cc1ncnc(O)c1C(N1CCC(F)(CNC(C2OCCCC2(C)C)=O)CC1)=O 71521,C1(C(N2CC=CC(NC(COCCCC(C)C)=O)C2)=O)CC(C)(C)CC(C)(C)C1 71522,n1(CC)ncc(C(=O)NC(C2(O)CCN(C(c3csc(C(C)C)n3)=O)C2)C)c1Cl 71523,c1(C(=O)NCCCNC(C(CC=C)CC)=O)ccc(N)c2ccncc12 71524,CC1CN(C(=O)C=Cc2ccoc2)C1C(=O)NCC(=O)N.c1(N)ccccc1 71525,CCC1=NOC(C(=O)NC2CCC(N(C)C(c3cnnc(O)c3)=O)CC2)C1 71526,c1(NC(CCCOC)C)cc(Br)ccc1S(=O)(=O)NC1CCC1(C)C 71527,C1(C(=O)NCCNC(N(C)C)=O)CN(C(=O)CC2CCCC2)C2(CCOC2)C1 71528,CCCC(CC)CCC(=O)N1CC(C)(C)CC1CC(=O)NCC1(OCC)CCC1 71529,CCCC(CCC)CC(=O)N1CCN(C(=O)CN(C)C(C2CSCN2C)=O)CC1 71530,N1(C(C(c2cc(C)sc2)(C)C)=O)CC(NC(c2cncn2C)=O)C(C)C1 71531,c1(C(=O)NCC(C2CCCC2)NC(=O)CC2CCCCO2)ccc2c(n1)CCCC2 71532,C1(C(=O)NC2CCC(CCC(=O)N(C3C(C)CCCC3)C)C2)CN2CCN1CC2 71533,N1(C(c2c(CC)ccs2)=O)CC2CC1CCC2NC(c1c[nH]nc1C(C)(C)C)=O 71534,C1(NC(c2n(CC)c(O)nc2)=O)CC2CCC1CN(C(=O)C(C)(F)C(C)(C)F)C2 71535,N1(C(c2c(COC)scc2)=O)CCC2CC1CN(C(=O)C=CC(=O)N(C)C)C2 71536,c1(C(=O)NCC(C)(F)CNC(=O)CC2CC3CC3C2)cnc2n1CCCC2 71537,Cc1n[nH]c(C)c1CC(=O)NCC1CC1CC(=O)N(C)C(c1ccncc1)C 71538,c1(C(=O)NCc2ccoc2C(=O)NOC2CC3CCC2C3)ccc(O)cc1 71539,C1(CC)CC(C(=O)NC2CCN(c3nnc(COC)s3)CC2)CCO1 71540,C1(NC(C2C(CCC)C2)=O)CC2CCC(C1F)N2C(=O)CCSC(F)(F)F 71541,O=C(NNC(=O)C1CC=CCN1c1nncs1)C1CCCN(c2ccc(Br)cn2)C1 71542,N1(C(CC=CC)=O)CCc2ccc(C(N3CCCC4OCCC34)=O)nc2C1 71543,c1(N2CC(CNC(C(CC)OC)=O)OCC2)nc(Cl)nc2[nH]ccc12 71544,c1(C(N2C(C)(CC(=O)N(c3c(OC)cccc3)C)CC2)=O)cc(F)ccc1O 71545,CC(C)C(N=[N+]=[N-])C(=O)NC1C=CC(C(=O)NC2(CO)CC3CCC2C3)C1 71546,CC1C(C(=O)N2CCCCC2CC(N2CC3COCC3C2)=O)=NOC1C 71547,C1(CN(C(=O)COCC(C)(C)C)C)CCCN(C(C23CCCC2C3)=O)C1 71548,c1(OC)cc(C(=O)NC2CC2CNC(c2cc(Cl)c[nH]2)=O)ccc1O 71549,C(=O)(CC(C)C(F)(F)F)NC(CNC(CC1(CC(=O)OC)CCCC1)=O)C 71550,N1(C(Cc2c(C)con2)=O)CCN(C(c2csc(S)n2)=O)CCC1C 71551,N1(C(C2N(C(C)C)CCC2)=O)CCC(F)(CNC(=O)C(C)c2cccs2)CC1 71552,C1(NC(c2ccc(C(F)(F)F)o2)=O)CCC2(CCN(C(c3ccon3)=O)C2)C1 71553,C(=O)(C1=CS(=O)CCC1)N(C(CNC(c1nnc(C)s1)=O)C)C 71554,C#Cc1ccc(C(=O)N(C(C)CCNC(C23CCC(CC2)O3)=O)C)c(F)c1Cl 71555,C1(NC(=O)CCNC(c2ccsc2)=O)CN(C(C2CC=CC2)=O)CC1C1CC1 71556,N1(C(CC(CNC(c2cn(CC)nn2)=O)OC)=O)CCC2(CCCCC2)C1 71557,n1(CC(N2C(CCNC(CCNC(=O)NC)=O)CCC2)=O)ccc(C)cc1=O 71558,CCN=c1[nH]c(C(=O)NCCCNC(c2cccc(OCC3CC3)c2)=O)cs1 71559,C1(NC(c2cn[nH]c2)=O)CCN(c2nnc(C(N3CC4CCC3C4)=O)s2)CC1F 71560,c1(CC)ccc(C(N2CCOC(CCOC)CC2)C(=O)NCCSC)cc1F 71561,O([Si](C)(C)C(C)(C)C)CC(N1CC(NC(c2c(OC)scc2)=O)C(O)C1)=O 71562,C1(CC=C)(NC(C2CSC(C)=N2)=O)CCCN(C(c2ccsc2C(F)F)=O)C1 71563,Cc1cc(C(=O)NCC2CCN(C(C3C4CCC(=O)C34)=O)CC2)cc2c1CCC2 71564,N1(CCNC(N2CCC(CN)CC2)=O)C(=O)NC2(CCC2)C1=O 71565,c1(C(N2CCC(C)(CNC(C(C(=C)Cl)(C)C)=O)C2)=O)cccc2nn[nH]c12 71566,c1(C(=O)NCCC(CNC(c2ccc(C)nc2O)=O)O)cccc(C=C(F)F)c1 71567,c1(C(=O)NC(C)CNC(=O)Cn2ncnn2)nccc2c(Cl)cccc12 71568,C=CCC(CNC(=O)C(CC)N(CC)CC)C(=O)NC1(O)CCC1 71569,c12ccccc1OCCN2.n1(CC=C)nnnc1C(CCC1CCCO1)OC 71570,Cc1cccc(CC(=O)NC2CN(C(C3(O)CCSC3)=O)CC2C)c1Cl 71571,C(=O)(CC1=Cc2ccccc2C1)N1CCC(NC(c2ccc(F)cn2)=O)C(F)C1 71572,C(=O)(CCC(C)(C)C#N)N1C(C(=O)NCC(C#C)OC)CCCC1 71573,c1(NC(C2CSCCN2C(=O)CC(F)(F)F)=O)cc(O)ccc1C(F)(F)F 71574,C1(CNC(=O)C(C2CCN(C(=O)C3CC3)C2)F)Cc2ccccc2C1 71575,C1(C)(C(N(CCCN(C(C2CCN(C)C2=O)=O)C)C)=O)CCS(=O)(=O)CC1 71576,N1(c2nnc(CC(C)C)n2CC2(C)CCCO2)CCN(C)C(=O)C1(C)C 71577,C(=O)(CS(N)(=O)=O)NC(C)CN(C)C(c1ncnn1C1CCOCC1)=O 71578,N1(C(C2CN(C)C2)=O)CCC2CCC12CNC(c1ccoc1Br)=O 71579,N1(C(C(C)O)=O)CC2COCCC2(NC(C2(c3ccccc3Br)CC2)=O)C1 71580,C(=O)(C1=CCCN(C(=O)C(=C2CCCCC2)F)C1)N(C1C(C)C1)C 71581,c1(C(CNC(=O)C(Cl)=CCl)NC(C(C)NC(=O)OC(C)(C)C)=O)ccccc1 71582,CC1CCC=C1C(=O)N(C(C)C(=O)NC1CCC12CCCC2)C 71583,N1(C(CNC(CC)=O)=O)CCC(C(=O)NCC2(C)CC3CC3C2)C(C)(C)C1 71584,C1(C(N2C(CNC(CCCC(C)=O)=O)CCC2)=O)CCc2cnn(C(C)C)c2C1 71585,N1(C(C2CC(NC(C(CCOC)OC)=O)C(O)C2)=O)CCOC2(CC2)C1 71586,c1(C(C(=O)NC2CCCC(NC(C(CC)(C)C)=O)C2)O)ccc(F)c(Cl)c1F 71587,CON(C(=O)C1=C(F)CN(C(=O)Cc2cc[nH]c2)CCC1)C1CCC1 71588,C(CCC(=O)NCC1(C(C)(C)O)CN(C(=O)C(CN(C)C)N(C)C)C1)SC 71589,c1(C(C)C)cc(NC(=O)C(=O)NCC2NCCC2C)ns1 71590,N1(C(C(CC)CCOC)=O)CCC2(CC1)CCN(C(c1ccc([N+](=O)[O-])[nH]1)=O)C2 71591,C#Cc1ccnc(C(=O)N(CCC)CCNC(=O)CCn2ccnc2)c1 71592,C1(N(C(C(C(=C)C)(C)C)=O)C)CCCC2CN(C(c3ccn(C(F)F)n3)=O)CC12 71593,C(C(=O)N=c1cc(C)n(C2CC2)[nH]1)N(C(=O)C(C)CN(C)C)CC 71594,C(=O)(C(C)NC(=O)NC(C)COC)NCCOCC#C 71595,Cc1cc(NC(=O)C(c2cnn(C(C)(C)C)c2)=O)n(-c2ccc(F)cc2)n1 71596,N1(C(C(C)Cc2ccccc2)=O)CC(NC(C2CC(CF)C2)=O)CC(O)C1 71597,CN1CCC(C(=O)N(C)CC2CCCN(C(=O)CC3CCCSC3)C2)CC1 71598,CC(C)CC(C)CC(=O)NC1CC(F)(CNC(c2ccnc(C(F)(F)F)c2)=O)C1 71599,c1(C(=O)NC(C)C(C)NC(=O)C=C2CCOCC2)ccc(-c2csnn2)cc1 71600,C1(C)(C(N(CCCC(=O)NC)C)=O)CC(O)CN1C(C1CCN(C)CC1)=O 71601,c1(C(=O)NCC23OCC(NC(COCCCC)=O)(C2)C3)cc(N)ccc1[N+](=O)[O-] 71602,c1(C(N(C2CCN(c3nnc(CC)o3)CC2F)CCC)=O)cc(C)c(C)nc1O 71603,c1(C(=O)NCC=C)cc(F)ncc1NC(c1ncccc1C(F)F)=O 71604,CC1CCCn2c(C(N3CC(CCNC(=O)C(C)c4ccsc4)C3)=O)cnc21 71605,N1(C(C(CO)C2C(C)=C2)C)CCC2CCC(C1)N2.C(CC#N)N 71606,c1(OC)ccc(F)cc1C(C1=CCCCC1)NCCN1CCOC(C)(C)C1 71607,C(C(C)(C)CC(=O)NCCCC(C)(C)C)NC(C(CC)C)=O 71608,c1(C(=O)NC(CNC(c2ccc(COC)o2)=O)(C)CO)ccncc1OC 71609,Cc1cc(C(=O)NC2CC3CCC2N(C(C2CCCSC2)=O)C3)cc(C)c1N 71610,c1(C(C(=O)NCCCOCC2CCCN2C(=O)CC2CC2)O)ccc(Cl)nc1 71611,N1(C(C(C=C)(C)CC)=O)CCN(C(c2ccsn2)=O)CC2(CC2)C1 71612,C1(COC)CN(C(=O)Cc2ncoc2C)CCN1C(=O)C1=CCCCC1 71613,c1(N2CC=CC(NC(C(CSC)C)=O)C2)nc2c(C)cc(C)cc2s1 71614,c1(OC(C)C(=O)NCC(C)(C)CN(C)C)cccnc1 71615,c1(NCC)cccc(C(=O)N(CCC(C)NC(c2snnc2C)=O)C)c1 71616,C1(C(=O)NCc2ccn(CC)n2)CC(C)(C)CN1C(=O)Cc1cncs1 71617,c1(C(N2CC(NC(C(C)OC3CCCCC3)=O)C2)=O)oc2ccccc2c1CO 71618,S(=O)(=O)(c1ccc(OC(F)(F)F)cc1)N(c1cn(CC2CCCOC2)nn1)C 71619,C1(NC(c2cncs2)=O)CCC2(CCN(C(c3cnn4ccncc34)=O)CC2)C1 71620,c1(C(C)CC(=O)NC2CC(F)(CNC(=O)Cn3ncnn3)C2)cncc(F)c1 71621,C(=O)(C(C)(C)C(F)(F)F)NC1CC(C)N(C(=O)CCCSc2ccccc2F)C1 71622,C1(C(N2C(C(=O)N(C)CC3(O)CCCCC3)(CC)CCC2)=O)CC2C(C1)C2(F)F 71623,C1(CNC(CO)CO)C2(CCC2)C12CCC2 71624,CCCCCC(C)(C)C(=O)N1CCOC(CNC(=O)CC(CC)OC)C1 71625,c1(NC(C(=O)Nc2cccc(C3CCC(=O)N3)c2)=O)cc(Cl)n2nccc2n1 71626,C1(NC(CC(COC)C)=O)C2CC3CN(C(C4CCC(COC)C4)=O)C1C3C2 71627,C1(C(=O)NCC(=C)C(F)(F)F)CN(C(c2ccn(C(F)F)n2)=O)CCC1O 71628,C(C(C)(C)OC(=O)CNC(C)=O)NC(=O)OCCN(C)C(=O)C1CC1 71629,Cc1cc(O)c(C(N2CC(F)(F)CC2C(=O)Nc2cc(O)ccc2F)=O)cc1Br 71630,c1(OCC)ccc(S(=O)(=O)N(C2CCCCCC2O)C)cc1C(=O)OC 71631,c1(C(C(N2CC(Cn3cc(C(OC)C4CC4)nn3)OCC2)=O)F)ccc(Cl)c(F)c1 71632,N(C1CCCc2c[nH]nc21)C(CC(CNC(c1cc(CC)nn1C)=O)O)=O 71633,c1(C(C)=O)cc(=NCC23CC(CNC(=O)C(C)C(C)C)(CO2)C3)[nH]cc1[N+](=O)[O-] 71634,C1(CC(=O)NCC2(OC)CCN(C(c3ccc(F)cn3)=O)C2)CC(O)C12CCC2 71635,N1(CC2CN(C(C(C)(C)N3CCCCC3)=O)C2)CCN(C(C2CCC2F)=O)CC1 71636,c1(CC(N2CCCCC(NC(c3nc(C)sc3)=O)C2)=O)ccc2c(c1)CCO2 71637,N1(C(C(CCOC)C)=O)CCC(C2CCCN(C(c3ccsn3)=O)C2)C1 71638,N1(C(C(CC(C)C)ONC(C2CC3C=CC2C3)=O)=O)CC2(CCOC(=O)N2)C1 71639,c1(CC(N2CC(C(C)NC(c3cccc(=O)o3)=O)OCC2)=O)ccc(O)c(F)c1 71640,CC1(C)CCCC1(CO)NC(=O)C1=CCN(C(=O)C=CCN2CCC2)C1 71641,N1(C(c2n(CCC)ncc2)=O)CCCC2CCN(C(c3cnsn3)=O)CC12 71642,CCCCC(C)C(C(=O)NCCCOC)N1CCC(OCC2CC2)CC1 71643,c1(-n2c(C(C)CC(F)F)nc(C(CC)O)n2)cc(C)ccc1C 71644,OC1c2ccccc2CC1NCC1(c2cccs2)CCC1 71645,N1(C(C(C=CC)O)=O)CC=C(CC(=O)NC(CCC)c2nn[nH]n2)CC1 71646,CN1CC(NC(c2c[nH][nH]c2=N)=O)C(O)C1.C1(=O)C(CC2CC2)CN1C 71647,C(=O)(CCS(=O)(=O)N1CCCC1)N1C(CNC(=O)Cn2nnc(=O)[nH]2)CC(O)C1 71648,c1(NC(C2N(C(c3ccc(OC)cc3)=O)CC=C2)=O)cccc2cc(C)cnc12 71649,C1(NC(CC(=O)N(C)C)=O)CCCC12CCN(C(=O)C(C)(C)c1nccs1)CC2 71650,c1(C(N2CCN(C(C34OC(C)C(C3)C4)=O)C(C)C2)=O)n[nH]c2c1CS(=O)(=O)CC2 71651,Cc1cncc(C(=O)NC2COCC2NC(C23CC(F)(C2)C3)=O)c1C 71652,C1(NC(c2cc(C)cc(F)c2)=O)CN(C(=O)COCC2(F)CC2)CCC1(C)C 71653,c1(C(=O)NC(CN(C(C(CC)(C)F)=O)C)C)ccc2c(c1)nc(C)n2C1CC1 71654,C(=O)(C(C(C)CC)N(C)C)NC1C=CC(C(=O)NC2CC(=C)C2)C1 71655,Cc1cc(C=CC(=O)NCC2CC3(C2)CN(C(=O)C(C)CO)C3)ccc1F 71656,N1(C(c2cn(CCC)nc2)=O)CC(NC(=O)C(C)S(C)(=O)=O)C2(CC2)C1 71657,N1(C(C(=O)NCC(CCOC)NC(c2cc(F)c[nH]2)=O)C)CCN(C)CC1 71658,c1(C(N2CC(F)(CNC(C3CCC(C)C3)=O)C2)=O)ccnc(N2CCCC2)n1 71659,C1(CNC(CC(C)(F)F)=O)CCCN(C(C2(C)CCC2)=O)CC1 71660,C1(CCNC(C(c2cccs2)NC(CCC=C(C)C)=O)=O)COC(C)(C)C1 71661,C(=O)(C=CS(C)=O)N1CC(C)(NC(C2CCN(C(C)=O)C2)=O)C1 71662,N1(C(C(C)C)=O)CCN(C(C)CNC(=O)CSC(C)C)CC1 71663,C(=O)(C1=CCC2CCC1N2C(c1occc1CC)=O)N1CC(C#C)C1 71664,C(c1ccc(CC)o1)=CC(=O)N(C)CC1CN(C(CSCC#C)=O)C1 71665,CCC(CC)(CCNC(C1C2(CC2)C12CC2)=O)NC(=O)C(C)OC1CCOC1 71666,c1(CC(N2CCC(O)(CNC(CCC(C)(C)OC)=O)C2)=O)ccc(C#N)cc1F 71667,C=CCC(C)(C(=O)N(C(C)CCNC(C1(O)CCCC1)=O)C)N(C)C 71668,C1(C(C(C)(C)C)=O)CC12CCCCC2.c1(C(=O)OC2CN(C)C2)cn(CCO)nn1 71669,c1(C(N2CCN(C(C(C)CC3CCC3)=O)CC2C)=O)cc2c(O)cccc2n1C 71670,C1(C(=O)NCCNC(C2(c3ccc(Br)nc3)CCC2)=O)CCC([N+](=O)[O-])CC1 71671,O(NC(=O)CCOCCCNC(=O)C(F)CC1CCOC1)CCN(C)C 71672,n1(CC(=O)NC2CC(N(C(Cc3cn(CC)nn3)=O)C)C2)cc(C#N)cn1 71673,c1(C2(C(N3CCC(CNC(C4CNC(=O)N4)=O)C3)=O)CCCC2)ccc(Cl)cc1 71674,C(=O)(C(C)(C)C(C)OC)OC(C(=O)N(CC=C)CC1CC1)C 71675,C(C(F)(F)C(=O)NCCOCCC(=O)NC1CCCC(O)C1)OC 71676,N1(C(COCCCOC)=O)C(C(=O)NCCCc2ccsc2)CC2CCCCC12 71677,Cn1c(C(=O)NCC2CCCCC2NC(=O)CC2CSCCS2)cc2ccccc12 71678,N1(C(CCCC(N)=O)=O)CC2CN(C(c3ccc(C4CCC4)nc3)=O)CC2C1 71679,N1(C(C(CC=CCC)C)=O)CCC2CCCC12C(=O)NC(c1nc[nH]n1)C 71680,CCC(C)C(C(=O)NC1CCC(NC(c2ccccc2NCCO)=O)CC1)OC 71681,C=CCCCCCCCCC(=O)NCCCCCCNC(=O)CCCC(=O)NCC 71682,N1(C(C(CC)NC(C)=O)=O)CCC2(CC(NC(=O)C=Cc3cnccn3)CO2)C1 71683,C(=O)(C#CC(C)(C)C)NCC1OCCN(C(c2ccn(C)c2C2CCC2)=O)C1 71684,CC1CCCN(C(=O)C(C)N(C(c2cncn(C)c2=O)=O)C2CC2)CC1 71685,C=CCC(C)(C)CCNC(c1cnn(CCNC(c2cncc(C)c2)=O)c1)=O 71686,c1(N2CC(C)C(NC(C3(CO)CCC3)=O)CC2)nc(Cl)nc2ccccc12 71687,CCCCC(CC)C(=O)NCCN(C(c1nc(Cl)sc1C)=O)CC 71688,C1(CNC(C(CCC=C)(F)F)=O)CCC2(CCN(C(=O)C(F)C(C)C)CC2)CO1 71689,N1(C(C2C(C)C2)=O)CCC(C(C)NC(C23CCN(CC2)C3)=O)CC1 71690,C1(CNC(c2c(C(=O)OC)csc2)=O)CN(C(=O)C(=O)NC2CC2)CCC1C 71691,N1(C(C2C(C=C)CC2)=O)CC(NC(c2cc(OC)ccn2)=O)CC12CCCCC2 71692,c1(C(=O)NC2CCN(C(C3C(C(=O)OC)C3)=O)C2)cccnc1F 71693,C1(CNC(COCCC)=O)CCCN(C(=O)CC2CCCS(=O)(=O)C2)CC1 71694,C(=O)(NOC(C)(C)C)C1(C(C)NC(COCCCC)=O)CC1.CCOC 71695,CCCCCCCNC(=O)C(CC1CCCCC1)Nc1ccccc1 71696,C1(NC(CN(C(C)C)C)=O)CN(C(=O)CCC2CC2(F)F)CCC12CCC2 71697,CC(C)CS(=O)(=O)CC(=O)NC1CN(C(c2ccc(F)nc2F)=O)CC(C)(C)C1 71698,C1(NC(CC(C=C)C)=O)CCC(O)CN(C(c2cc(C(C)(C)C)on2)=O)C1 71699,C(=O)(C1=CC2(CCOC2)C1)N1CCC(NC(c2c(CSC)cccn2)=O)CC1C 71700,N1(C(c2cc(C(=O)OCC)sn2)=O)CC2CC(NC(C3CC4(CSC4)C3)=O)C1C2 71701,c1(Oc2cccc(C(N3CCC(OC)C3)=O)c2)c(F)cc(F)c(N)c1[N+](=O)[O-] 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71861,CCCCC(CC(=O)NC1CCC(OC)CC1)NC(c1ccc2cc[nH]c2c1)=O 71862,c1(CC(=O)NCC(C)NC(c2occ(OC)c(=O)c2)=O)noc2ccc(O)cc12 71863,C(=O)(C(C1=CCCCCC1)N1CCCCCCCCCC1)NC(C)(C)C 71864,C12CCN(C)C1NC(=O)CN(C(C)C)C2=O.C1(OCC)(CC)CC1 71865,n1(C(CC)C)nccc1C(=O)NC(C1CCCN1C(=O)CCCNC(=O)OC)C 71866,CC1OC2(C(=O)NC3CCC(NC(c4cnc(-c5ccccc5)[nH]4)=O)CC3)CC1C2 71867,c1(CC(C)C(=O)NC2(C)CN(C(=O)CC(C)N(C)C)C2)ccc(Br)cc1 71868,N#CCCCC(N)C(=O)Nc1ccc(NCCN2CCOCC2)cc1 71869,CC12CCCC(C(N3CCC(c4cn(C5CCCC5O)nn4)C3)=O)(CO1)C2 71870,c1(OC(CCC2CN(CCC(C)C)C2)=O)cccc(Br)c1 71871,CCCC(C(=O)N1CC2CC(NC(c3coc(CC)n3)=O)CC1C2)S(N)(=O)=O 71872,CC(CC(=O)NCC1CCN(C(=O)CC=CCc2ccccc2)C1)CC(F)(F)F 71873,N1(C(C(CC)SC)=O)CC2(CCC(CNC(=O)C(O)CC3CCCC3)O2)C1 71874,C1(NC(Cc2c(F)ccc(C)c2)=O)CC12CCC(NC(=O)C(C)CF)CC2 71875,C1(CCOC)(NC(c2ccc(COC)s2)=O)CCN(C(C2CC3(CCC3)C2)=O)C1 71876,Cc1ccnc(C)c1C(=O)N(CCCCNC(C1(c2ccccc2Cl)CC1)=O)C 71877,c1(-c2nc(C3(C(F)(F)F)C(C)C3)n(CCS(N)(=O)=O)n2)ccc2ccccc2n1 71878,Cc1cc2ccccc2n1CC(=O)N(CC(C)(C)NC(=O)CC1COC(=O)C1)C 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71896,CCCCC(CC(=O)Nc1ccc(C(C)C)nc1)NC(=O)CCn1cncn1 71897,c1(C(=O)NC2CC(C)N(C(=O)Cn3nccn3)CC2)cccc2c(O)nncc12 71898,CC1CN(C(c2cc(Br)co2)=O)CC1CCNC(C1(O)CCC1)=O 71899,N1(C(C2(F)CCN(C(C3=C(C)CCC3)=O)CC2)=O)C2CCC1CC(O)C2 71900,c1(C(N(CCNC(C(OC)OC)=O)CC2CC2)=O)cc(O)ncn1 71901,C1(NC(c2cnn(C(C)C)n2)=O)CCCCCC1C(=O)NCC(c1cnc[nH]1)C 71902,N#Cc1ccc(C(N2CCC23CN(Cc2ccc(Cl)cc2F)C3)=O)c(Cl)c1 71903,CC1(NC(N2CCCC2)=O)CCCC1C(=O)O.c12ccc(cc1)oc2=O 71904,C1(NC(c2cc(CC)n(C)n2)=O)CC2(C1)CC(CNC(C1CCCCC1C)=O)C2 71905,C1(NC(Cc2nc(C)sc2)=O)CCOCC1C(=O)NCCc1ccncc1 71906,C1(C(N(C2(C(=O)NC(C#C)C(C)OC)CCC2)C2CC2)=O)CC=C(C)CC1 71907,Cc1nc(O)sc1C(=O)NC(c1ccccc1)C(C)NC(c1cn(C)nn1)=O 71908,C(CN=C(NCc1nc2c(s1)CCCC2)N(C)Cc1ccc(N(C)C)cc1)OC 71909,N1(C(c2sc3cc(C)sc3c2)=O)CCC2(C1)CN(C(c1cnn[nH]1)=O)CCO2 71910,Cc1nn(C(F)F)cc1NC(c1nnnn1C1CCCCC1)(C1COC(=O)C1)C 71911,Cc1cc(N2CCC(C)C(NC(=O)CN(C)C(N)=O)C2)nc(-c2ccccn2)n1 71912,C1(C(=O)NC(CC)CN(C)C(c2coc(C)c2)=O)COc2cccc(OC)c2C1 71913,C(=O)(C(CCC1CCC1)N1CCC(n2cccn2)C1)NCCSC 71914,c1(C(N(CC(O)CNC(=O)Cc2ccccc2)C)=O)ccc([N+](=O)[O-])n1C 71915,c1(C(C)C)ncsc1C(=O)NC(C)CN(C)C(c1ccnn1C1CC1(F)F)=O 71916,Cc1ccc(O)c(NC(=O)Cc2csc(=NCc3cccc(I)c3C)[nH]2)n1 71917,N1(C(c2cccc(OC)n2)=O)CC2CCC1C2NC(C1CC(N2CC(O)C2)C1)=O 71918,N1(C(CC(C)n2ccnc2)=O)CCC2CCCC12C(N1CCc2ccsc2C1)=O 71919,FC1(F)C2CCC1CN(Cc1nc(C3CCOCC3)co1)C2 71920,c1(C(N(CCC)CCNC(c2ocnc2C2CC2)=O)=O)c(C)cccc1F 71921,C1(CNC(c2ccoc2)=O)CCCCC1NC(C1CC(O)(C(F)(F)F)C1)=O 71922,N1(C(Cc2cccc(OCC)c2)=O)CCCC(NC(=O)CC2(C(F)F)CC2)C1C 71923,CCC(CC(=O)N1CSCC1C(N1CCC(C)(O)C1)=O)SC 71924,C(C(C)C(C)C(=O)NC1C2CC1CN(C(C1CSCCS1)=O)C2)OC 71925,C(=O)(C(C)CCCC(C)C)NC1C(NC(c2c(SC)cccc2)=O)CCC1 71926,C#CCC(O)C(=O)NCC1(C(=O)NC2(c3nc(C)no3)CC2)CCCO1 71927,c1(C(=O)NCCCCCCN(C(CC(C)O)=O)C)ccc(S(N)(=O)=O)c(N)c1 71928,C#Cc1cccc(OCC(=O)NC2(F)CCN(C(=O)CCCNC(N)=O)CC2)c1 71929,c1(OC)cc(NC(c2[nH]c(C)c(CNC(C3(C4CC4)CC3)=O)c2C)=O)cc(C)c1 71930,C1(NC(CSC)=O)C2CC3CN(C(C4C5CCC(=O)C45)=O)C1C3C2 71931,CN1C(=O)Cc2c(C(=O)NCC(C)(C)NC(=O)C(F)C(F)(F)F)cccc21 71932,C12(C(N3C4C(NC(C5C(C)(C)NC(=O)C5)=O)C(C4)C3)=O)CCC(C1)S(=O)(=O)CC2 71933,c1(C(=O)NC(CCOC)CNC(c2cnc(C(C)C)s2)=O)cncc(C)c1C 71934,c1(CC)ccc(F)cc1C(N1CCCC(C(=O)O)C1)=O 71935,Cc1cccnc1CCC(N1CC2CC2(NC(=O)CSCCC#N)C1)=O 71936,C(=O)(C1=CCCSC1)N1C(CCCNC(CNS(CCOCC)(=O)=O)=O)CCC1 71937,C1(CC(=O)NCCC2CC(NC(=O)C=CC3CCCC3)C2)CC(F)(F)C1 71938,CC1(C)CCCC(C(N2CCC(CO)(NC(C3CC(F)(F)C3)=O)C2)=O)C1 71939,c1(C(=O)OC2(CN(CC)CC)CCCC2)cc(N2CCOCC2)ccn1 71940,c1(C(c2n(CC)nnn2)NCC2CSCCO2)ncccc1C 71941,N1(C(C(CCSC)O)=O)CC2CC1CCC2NC(c1cc(C)c(F)c(C)c1)=O 71942,N1(C(CCC2CC(NC(C3C(C)CC(=O)NC3)=O)C2)=O)CCCN(C)CC1C 71943,N1(C(c2n(CC=C)ccc2)=O)CCC(C)(C)C(CNC(c2ccsc2C)=O)C1 71944,N1(C(c2cc(OC)nn2C)=O)CCC(CO)(NC(c2snnc2C)=O)CC1 71945,c1(NC(CC)=O)ncccc1C(=O)NC1COCC1n1cc(CCOC)nn1 71946,N1(C(C(C)(C)CC#N)=O)C2CCCC1CN(C(C1CCc3ccnn3C1)=O)C2 71947,c1(C(=O)NCCCCC(C)NC(C2C(=C)CC2)=O)c(O)cc(Cl)cc1F 71948,C12(NC(Cc3cc(C)no3)=O)CCC1CN(C(c1nccc(Br)c1C)=O)C2 71949,c1(NCC)cccnc1C(=O)N(CC(C)CNC(=O)C(c1cccc(Cl)c1)C)C 71950,C(=O)(CN=S(C)(C)=O)NC1(C)CCN(C(=O)CNC(C2CCOCC2)=O)C1 71951,CC1(C)C(CNC(=O)C(O)C2CCC2)CCN1C(=O)CCCn1cccc1 71952,c1(-c2c(OCCC)cccc2)cccc2c1CCN(Cc1n[nH]c3c1CCC3)C2 71953,c1(C(=O)NCC(=O)NCC(CN(C)C)O)n[nH]c(O)n1 71954,c1(C(N2CC(CNC(c3c(O)cccc3O)=O)OCC2)=O)ccc(Br)cc1F 71955,CC(C)(C)C(O)C(C(=O)NCCc1ccc(C#N)cn1)c1ccccc1 71956,S(=O)(=O)(c1cccc(Cl)c1)NCC(=O)N(C1CCN(C(=O)Cc2cccs2)C1)C 71957,C12(C(=O)NC3CCC(N(C(=O)CCNC(=O)CO)C)CC3)CC1CCC2(F)F 71958,N1(C(C2CC(C(=O)OC)C2)=O)CC2CC1C2NC(c1cnncc1C)=O 71959,N1(C(C2N(C(C)C)C(=O)CC2)=O)CC(NC(C2C(C)(C)OC2(C)C)=O)CCC1C 71960,C1(CNC(C2CCCOC2)=O)CC2COCC2N1C(C1CCOCC1)=O 71961,N1(C(C(CC#C)CC#C)=O)CCC2C(C1)NC(=O)CN2C(=O)CCCC(C)CC 71962,c1(NC(C2(C#N)CC2)=O)cnc(F)cc1C(=O)Nc1cc(Br)cc(I)c1 71963,C1(CNC(=O)C2=CCCC2)CCC12CCN(C(c1cnc3ccsc3c1)=O)CC2 71964,N1(C(C(CC)F)=O)CC2CC1CN2C(c1ccc(SC)o1)=O 71965,CCC(C)(C(=O)N(C(CC(CCC)C)=O)c1ccc(C(C)=O)cc1)C(N)=O.OC 71966,N1(C(C2CCN(C(C)C)C2=O)=O)CCC(NC(=O)C(F)=C2CCCC2)CC1C 71967,C1(CNC(CN(C(C=CCOC)=O)CC(C)C)=O)CCC2(CCC2)CC1 71968,C1(NC(c2ccncc2-n2cccn2)=O)C=CCN(C(c2ccco2)=O)C1 71969,N1(C(C(CC=CC)C)=O)CC2CC1CC2CNC(=O)CCNC(=O)CO 71970,N1(C(C(COC)NC(=O)C(C)C#N)=O)CCC(F)(CF)CC1 71971,N1(S(CC2CCC(NC(=O)C3CC3)C2)(=O)=O)CCOC(N(C)C(=O)OC(C)(C)C)C1 71972,N1(C(CC(=C=C)C)=O)CC2(CCCN(C(=O)COC(=O)Nc3ccncc3)C2)C1 71973,C1(C#N)(N(CCO)Cc2cc(C(=O)OC)[nH]c2)CCCCCC1 71974,c1(C(N2C(C(=O)NC(CSC)C)C=CC2)=O)cc(C)c(C)o1 71975,C1(NC(CC2(OC)CC2)=O)CN(C(C2(c3ccccc3)CC(O)C2)=O)CC1SC 71976,c1(C(N2C(C3(C(=O)NC(C=CS(C)=O)=O)CC3)CCC2)=O)nc2cnccc2s1 71977,c1(C(=O)NC2C3CN(C(c4cc(C)c(Cl)s4)=O)CC2C3)cn2c(n1)CCC(C)C2 71978,c1(C(=O)NCCC(C)NC(C2CC(N(C)C)CCO2)=O)ccc(C(F)(F)F)nc1 71979,c1(C(=O)NC2C(NC(c3cn(C)nc3)=O)C2)cc2cc(Br)ccc2[nH]1 71980,C1(C(=O)NC2CC3(C2)CC3NC(=O)C(F)=C2CCC2)CC12CCSCC2 71981,O=C(C1CCCc2nccn21)NC1CC1C1CCN(C(=O)C=C2CCC2)CC1 71982,c1(OC)nc(F)ccc1-c1cc(CNC(=O)C(N)=O)ccn1 71983,Cc1scc(C(=O)NCC2CCCC2NC(c2ccnc(SC3CC3)c2)=O)c1C 71984,c1(CC2CN(CC)C(=O)O2)cc(Cl)cc(OC)c1O 71985,N1(C(CCC2C(C)=NOC2=O)=O)CC(NC(c2onc(C)c2C)=O)CC1(C)C 71986,Cn1cc([N+](=O)[O-])c(C(=O)NC2CC(NC(c3coc(Cl)c3)=O)C2)n1 71987,Cc1c(C(N2CC(O)CC2C(=O)NCCCS(N)(=O)=O)=O)cc(F)cc1[N+](=O)[O-] 71988,N1(C(C2C(CC)CC2)=O)CC(n2ccnn2)CCC1(C)C.C1(C)(N)CC(CC)C1 71989,c1(NC(CCN(C(C2C(OC)(OC)CC2)=O)C)=O)ccncc1C(C)C 71990,N1(C(C(C)CCO)=O)CC(C2CCCN(C(=O)C(C)(O)C3CC3)C2)C1 71991,N1(CC(=O)NC(c2ccc(Cl)cc2)C(=O)OC)CCC(C(=O)N(C)C)CC1 71992,c1(CN(C(C2CCC2)=O)CC)c(Cl)ccc(F)c1F.C12COCCN1C2 71993,CC(CNC(=O)CCC(N)=O)C(F)C(=O)NCCCC(C)(C)C 71994,C1(C2(O)CCN(C(C3CCS3(=O)=O)=O)CC2)(NC(=O)CCc2cscn2)CC1 71995,N1(C(C=CC(F)=CC)=O)CCC(OC)CC1C(=O)OCC.OCC 71996,CCS(=O)(=O)CC(=O)NCC1(F)CCCN(C(c2cc(Br)ccc2Cl)=O)C1 71997,Cc1cc(CNC(=O)CC(O)CNC(C2CCOC2)=O)sc1C 71998,c1(CC(N2CCC(C)(CNC(C3C(C)C3C)=O)C2)=O)ccc(F)c(F)c1 71999,CC(C)C(O)CC(=O)N(C(C)CCNC(=O)Cc1ccc(Cl)cc1F)C 72000,c1(C(=O)NC2C(NC(CSC)=O)CCCC2)cc(Cl)cc(C)c1O 72001,C1(NC(c2sc(CC)c(C)c2)=O)CN(C(C2CC2C2CC2)=O)Cc2ccnn2C1 72002,CC1(CN(C(C2(c3ccncc3)CC2)=O)C2CC2)CCN(C(=O)C(N)=O)C1 72003,c1(CC(N2CCC(C)(c3cn(CC(=O)OC)nn3)C2)=O)csc2cccnc12 72004,CCC(O)C(F)(F)C(=O)N1CC2(CNC(c3cc(C)on3)=O)CC1CO2 72005,C1(NC(=O)C=Cc2ccccc2)CN(C(=O)C(O)CC2CC2)CCC1CO 72006,c1(NCC(C)Oc2cccc(OC)c2)nc(N2CCOC(C)(CO)C2)cc(C)n1 72007,C1(NC(C2(c3nc(Cl)cc(OCC)n3)CCC2)=O)CC2CCCCN2C1 72008,CN1CCOC(C(=O)NC(CCOCCO)C(=O)NC2CCC(C)CC2)C1 72009,C1(CNC(C2CCC2NC(=O)COCC2CC2)=O)CCCOC1.C1CO1 72010,N1(C(c2c(C)nc(F)cc2)=O)CCC2(CC1)CCN2S(=O)(=O)c1ccc(Cl)cc1 72011,n1(CC(C)O)nc(COc2cnn(C)c2)nc1-c1ccc(=O)oc1 72012,C(C(CC(C)C)C(=O)N1CCCCC1CCC(=O)NCc1c(C)cnn1C)OC 72013,C(C)(CN=C(NCC(=O)NC1(C)CC1)NC1CCC1)OC 72014,C#CC1(C(=O)NOCC(=O)NCCC2CCC(C)C2)CC(=O)C1 72015,c1(N(S(CC)(=O)=O)C)nnc(N2CCOC(c3nccs3)C2)n1CC1CC1 72016,N#CC1CN(C(c2ncc(F)cc2F)=O)CCN1C(c1sccc1Br)=O 72017,CC(C)C(C(=O)NCC(C)(Cn1cccn1)NC(=O)C=Cc1ccc[nH]1)NS(C)(=O)=O 72018,C1(C(=O)NCCC=C=C)(CC)CN(C(=O)C(CC)OC)C1 72019,C(=O)(CCCCC#N)NCc1cccc(C(N(C(C)C(=O)NC)CC)=O)n1 72020,Cc1cc(C(=O)N(C(C)CNC(=O)C(c2cccc(Cl)c2)C)C)oc1C 72021,C#CC1(C(=O)N(C2CCOC(C)(C)C2)C)CCN(C(=O)COc2ccsn2)CC1 72022,N1(C(c2c(NC)cncc2)=O)CCC2(COC(CNC(=O)C(C)(C)CO)C2)C1 72023,c1(-c2nc(CNC(=NCC34CC(C)(OC3)C4)NC3CC3)on2)cc(Cl)cnc1F 72024,C1(C(=O)NCC(C(C)O)C)N(C(=O)Cn2cncn2)CCC1(C)C 72025,C1(C(=O)NCC(CNC(C2N(C(=O)NC)CCC2)=O)(C)C)C2CNC(=O)C12 72026,C1(C(N(C)CC2(NC(c3ccc(N)cn3)=O)CC2)=O)CCC(F)(F)CO1 72027,C#Cc1ccc(C(N2CCC(C)(C)C2CNC(C2(N(C)C)CCCC2)=O)=O)cn1 72028,c1(C(N2CCC(C)(C(=O)NCc3ccccc3)C2)=O)cc([N+](=O)[O-])c(F)cc1Br 72029,CC(C(=O)N(C)CCN(C1(C#N)CC1)C)C1OCCc2sccc21 72030,CC1CC(N=c2[nH]c(=NCC3(CN(C)C)CCC3)[nH]c3cc[nH]c23)CCS1 72031,CCCCCC(=O)NC1CCCC(CN(C(=O)CCc2nc(C)no2)C)C1 72032,c1(C(=O)NC(C(C)C)CNC(=O)CC2(C)CC2)ccccc1-c1ccccc1 72033,c1(C(=O)NCC(=C)CCNC(C2(S(C)(=O)=O)CC2)=O)cc(Cl)ccc1Cl 72034,c1(C(=O)NCC2C(C)(C)CCCN2C(=O)CS(N)(=O)=O)ccc2nc(O)[nH]c2c1 72035,N1(C(C(COC)O)=O)CCC(C)(NC(=O)COc2cccc(NC(C)=O)c2)C1 72036,c1(C(N(CC(C)C(N2CCCC(C)C2)=O)C)=O)ccc(O)cn1 72037,c1(C(=O)NC(C)(C)CC(=O)N2CCC(CCO)CC2)ccc2c(c1)CC2 72038,CC(=O)CCCCC(=O)N1CC(C(=O)NCC2CCCC(=O)N2)CC1(C)C 72039,c1(CN2CCCC(C(C)NC(=O)COC3CCOC3)C2)ccc(F)cc1Br 72040,C1(CNC(c2cc(SC)cc(Cl)c2)=O)CN(C(C2CNC(=O)N2)=O)CCC1(C)C 72041,Cc1cn2c(n1)CCC(C(=O)NC1CC3CC1N(C(=O)CC1(C)OCCO1)C3)C2 72042,c1(C(N2CCN(C(c3c(SC)nccc3)=O)C3C2C3)=O)cc2cc(F)ccc2[nH]1 72043,C12(C(=O)NCCOCCN(C)C(c3ccc(CO)s3)=O)CCOC1CCOC2 72044,C(C(=O)NC12CC(C1)N(C(=O)C=CC(F)(F)F)C2)(C(C)C)n1ncc(C)c1 72045,c1(C(=O)NCC2CCC(NC(C3CCNC3=O)=O)C2)cc2cc(F)ccc2s1 72046,Cc1nsc(NC(C2CC(F)CN2Cc2c(Cl)cccc2Br)=O)c1C#N 72047,C(=O)(C(C)(C)C(C)(F)F)NC(C)CCNC(C1CCC2CC2CC1)=O 72048,C1(OC)CN(C(=NCCCN2CCCCCC2=O)NCCC(C)=O)CC1O 72049,Cc1ccc(NC(=O)NCC2CCCN2C(=O)CO)cc1S(C)(=O)=O 72050,C1(C(N(CCC(=O)NCC2(C)N=C(C)SC2)C(C)C)=O)OCCCC1(C)C 72051,C#CCC(C)(C(=O)NCC(F)(F)C(N)=O)NC(=O)CCC1CC1(F)F 72052,C(CCC)(C(=O)NC(c1ccnn1C)C(=O)Nc1cccc(SCC)c1)=CCC 72053,CC12CC(C(N3CCN(C(=O)CCF)C(CC(F)F)C3)=O)(C1)C1(CCOCC1)O2 72054,C=CCC(CC)C(=O)N1CC2CC(C1)N2C(C1C=CCS1)=O 72055,C#CC1CN(C(=O)C(N2CCC(C(C)C(=O)NC)CC2)=O)CCN1 72056,C1(CNC(c2c(C)cn(C)n2)=O)CC(C)CN(C(=O)C(C)NC=O)C1 72057,C12(C(=O)NC(C#C)(C)C)CCC(CN(C(=O)CC3CCC(=O)CC3)C1)C2 72058,N1(C(C(CCSC)O)=O)CC2(CCC2NC(=O)Cn2cnnn2)C1 72059,CC1CC(C(=O)NCCOC2CCN(C(=O)CCc3cnn(C)n3)CC2)C1(C)C 72060,c1(C(=O)Nc2cc(F)c(F)c(F)c2)cn2c(n1)CN(C(c1cccnc1)=O)CC2 72061,c1(C(=O)NC(C)CCCCNC(=O)C=Cc2ccccn2)ccc2c(c1)CCC2 72062,N1(CC)CCC(C(=O)NC2(C(=O)NC3COCC3CN(C)C)CSC2)C1 72063,C1(=O)C(CN=[N+]=[N-])N1.C(=O)(C(CC)n1cncn1)NCCN(CCC)C(C)C 72064,C1(OC)CC2(C1)CC(NC(C1CNC(=O)CN1C(=O)COC(C)(C)C)=O)C2 72065,C=C(Cl)CCC(=O)N1CCOC(CN(C(=O)CCc2cccc(O)c2)C)C1 72066,C1(NC(CCCC#C)=O)CS(=O)(=O)C12CCN(C(=O)C(C)CS(C)(=O)=O)CC2 72067,c1(C(=O)NCCCNC(Cc2ccn(CC)n2)=O)cc(C)oc1C(F)(F)F 72068,C1(CC)CCOCCN1C(c1ccc(C#N)s1)C(=O)NC(C)C(=O)OC 72069,C#Cc1cncc(C(=O)NC2COCCC2C(=O)NCc2cncs2)c1 72070,n1(C(C)C)c(O)nc(N2CCC(NC(c3cc(Cl)ccc3F)=O)CC2C)cc1=O 72071,c1(C(=O)NC(C2CCN(C(CC=C)=O)C2)C)ccc(F)cn1 72072,C1(C(=O)NCCCC(C)NC(C=C(COC)C)=O)CCC(=O)N(C(C)C)C1 72073,C=C(Cl)C(C)(C)C(=O)NCC1(CNC(=O)Cc2ccc(C(N)=O)cc2)CCC1 72074,CC1CCC(C(C)NC(=O)C(=O)NC2CCCC2Oc2ccccc2)CC1 72075,S(=O)(=O)(c1cccc(F)c1)N(CC(CCCCC(=O)N)C)CCN(C)C.C(C)(=O)NCCN.O 72076,N1(C(C(CC#CC)NC(=O)OC(C)(C)C)=O)CCS(=O)(=O)C(CO)C1 72077,C=CCCC(C(=O)N(CCC)CCC)NC(=O)CC(C)C(F)F 72078,C(=O)(C1=C(C)OCCS1)NC1C2(CCN(C(c3cc(CC)oc3C)=O)C2)C1 72079,C(=O)(CS(=O)(=O)Cc1ccccn1)NCC(N(C)C(C1CC(O)C1)=O)C1CC1 72080,c1(NCCNC(C2CCCN(C(CSCC(C)C)=O)C2)=O)cc(N)c(F)cn1 72081,c1(-c2scc(C(N(C)CC3CN(C(C4CC4F)=O)C3)=O)n2)ncccc1F 72082,C(=O)(CC(C)(C#N)c1ccccc1)NCCN(CCC)Cc1nccn1C 72083,C(=O)(C1=CCCCC1)NC(CSCC)C(=O)NCc1nc(C)cs1 72084,Cc1nc(C2CC2)sc1CC(=O)NC1CCCC1NC(=O)CN1CCCC1 72085,N1(C(c2c(Br)ccc(C)n2)=O)CCC2(CCN(C(C3CC3C3CC3)=O)CC2)C1 72086,C(=O)(C(C)C(F)(F)F)N1CCCC(N(C(c2c(NC(C)=O)cncc2)=O)C)C1 72087,C1(NC(c2nc(C)n(C)n2)=O)CCN(C(c2cc3c(s2)CCC3)=O)CC1(C)C 72088,C(CCN(C(=O)CCSc1nccn1C)C)(C(C)C)NC(c1ccc(CC)[nH]1)=O 72089,c1(CN2C3C(CNC(C)=O)(CCCC3)CC2)cc2cc(C)ccc2[nH]1 72090,c1(CC)c(C(=O)NCC(O)CNC(=O)COCc2ccc(OC)nc2)nnn1C 72091,C1(CNC(=O)C(c2cccnc2)O)(CNC(=O)Cn2ccnn2)CCOCC1 72092,C1(C(=O)NC(CC(=O)NC)(C)C)CC2(CCC2)CN1C(=O)C(C)N(C)C 72093,C12(C(N(CCC=C)CC)=O)COCC1CN(C(c1cc(OC)n[nH]1)=O)C2 72094,c1(C(=O)NCC2(F)CC(NC(COCC(=C)C)=O)C2)cccn(C2CCC2)c1=O 72095,Cc1cc(C(=O)N(C)CCN(C(C2CC2(F)F)=O)C(C)C)cnc1C(F)F 72096,c1(OC)nc(C)c(C(N2CCCCC2C(=O)Nc2cnn(CCO)c2)=O)s1 72097,c1(CC)nsc(CNC(=O)C(C2(O)CCC2)NC(c2sccc2F)=O)n1 72098,Cc1cnncc1C(=O)NCC(C1CCCN1C(C12CC(CO)(C1)C2)=O)(C)C 72099,c1(CC(N2CCC(N(C)C(c3n[nH]cc3F)=O)CC2)=O)ccc2c(c1)OCCO2 72100,N1(C(C2OCCC(NC(CC3C=NN(C)C3=O)=O)C2)=O)CC2CSCC(C2)C1 72101,C(=O)(CCC(=O)NC1CCCCC1NC(c1nc(C(C)C)oc1C)=O)NCCC 72102,N1(C(C23CC(CC)(OC2)C3)=O)CCN(C(=O)CN2CCCNS2(=O)=O)CC1C 72103,C1(COC)(NCc2sc(C)c(Br)c2C)CCC(C)CC1 72104,C1(C(N(CCN(C)Cc2ccncc2)CC)=O)CC2CCN(C3CCNC3)CC12 72105,CC(C)CC(C(=O)NCC12CC1CN(C(C1(N(C)C)CC1)=O)C2)c1ccccc1 72106,C1(c2n(CCSC)nnn2)(NCc2ccc(Cl)c(Cl)c2)CCOC2(CCOC2)C1 72107,N1(C(C2CC23CN(Cc2c(I)ccnc2Cl)C3)=O)CCC2(CCCO2)CC1 72108,N1(C(c2c(CC)cno2)=O)CCC2(CC1)CC2C(=O)NCC(C)S(C)(=O)=O 72109,N1(C(COc2ccc(CC(C)C)cc2)=O)CCCC(NC(=O)CS(N)(=O)=O)C1C 72110,C1(OC)CC(CC(=O)NC23CC(NC(c4cc(C(C)(C)C)on4)=O)(C2)C3)C1(C)C 72111,N1(C(C(C)NC(C)(C)C)=O)CCN(C(=O)C=Cc2cncc(F)c2)C(CF)C1 72112,c1(OC)c(C(=O)NCCC(C(C)C)NC(C2CC=CCO2)=O)c(C)nn1C 72113,C1(NC(=O)CC2(C(F)(F)F)CC2)CCN(C(c2ncc(Cl)s2)=O)CC1CO 72114,C1(C(C)NC(C2CCC3CC23)=O)CN(C(c2csc(C(C)(C)C)n2)=O)CCO1 72115,CC1CC(=O)NC1C(=O)NCC1CCCN(c2ncc(Br)cn2)C1 72116,Cn1cc(Cl)c(CC(=O)NCc2cccc(NC(C34COCC(C3)C4)=O)c2)n1 72117,N1(C(=O)OC)CCCC(C(N2CCC(OCC(c3ccncc3Cl)=O)CC2)=O)C1 72118,CC#CCCCC(=O)N1CCC1CNC(C1(CSC)CC(F)(F)C1)=O 72119,c1(C(=O)NC2C(CNC(CNC(=O)NC)=O)C2)coc(C#Cc2ccccc2)c1 72120,Cc1ccn(C)c1C(=O)N(CC(C)(C)NC(C1(c2ccccc2)CC1)=O)C 72121,c1(OC)ccc(C(=O)NC(C)CNC(c2cc(C(O)C(F)(F)F)ccn2)=O)nc1 72122,CC1CC(C(=O)NCC2CCN(C(c3cc(F)ccc3O)=O)C2(C)C)=NO1 72123,N1(C(CCC#C)=O)CCN(C(c2sccc2CN(C)C)=O)CC1 72124,Cc1c(Br)cnc(O)c1C(N1CC(CNC(C2CCCC(F)C2)=O)C1)=O 72125,O=NN1CCCC1C(=O)NC1C=CCN(C(c2ccc(-c3cn[nH]c3)cn2)=O)C1 72126,Cc1noc(C)c1CC(=O)NCC1(O)CCN(C(=O)C(C)NS(C)(=O)=O)C1 72127,n1(CC)cc(C(=O)NCC(O)CN(C(=O)CCn2ccnc2)C)c(C(C)(C)C)n1 72128,N1(C(CN(CCC)C)=O)CCOCC(F)(CNC(=O)CC2CCOC2)C1 72129,N1(C(C2CC(=O)NC2)=O)CC2CCC1C(CNC(c1n[nH]c3c1CCOC3)=O)C2 72130,C(=O)(CCCC(=O)NC1CC(=O)N(C2CN(C(c3cnccn3)=O)C2)C1)NC 72131,Cc1ccc2sc(N3CCCC3CNC(=O)C(C)CF)nc2c1C 72132,c1(CC)ccc(CC(=O)NCC2C(C)CCN2C(=O)Cc2n[nH]c(C)n2)cc1 72133,CCC(C)(C)CC(=O)NC1CC(F)(CNC(C2CCCCN2C2CCCC2)=O)C1 72134,C(=O)(CC(O)CNC(C1CN(C2CCC2)C1)=O)N(C1CC(F)(F)C1)C 72135,N1(C(CCCC)=O)CC(CN(C(=O)CNC(c2cc(Cl)ccn2)=O)C)C2(CC2)C1 72136,C=Cc1ccc(CNC(=O)N(C2CC2)Cc2ccc(F)cc2C)cc1 72137,C1(CC(=O)NC)CCCN(C(=O)Cc2ccccc2N2CCOCC2)C1 72138,c1(CN(C(=O)NCC(CC)(C)COC)C)cccc(Br)c1F 72139,CC1CCc2ccccc2N1Cc1cn(C2CCC(C(=O)NCCO)C2)nn1 72140,c1(C(=O)NCC2(F)CCC(CNC(CCSCC)=O)C2)cccc(Cl)c1F 72141,c1(C(=O)NCC(C(C)C)NC(=O)C2=CCCC2C)cc(C(F)(F)F)cc(F)c1 72142,CC(C)CC(C(=O)NC(c1cnn(C)c1)C)NC(c1cccc(Cl)c1)=O 72143,C1(OCC(=O)NCC(CC)NC(c2cc(C3CC3)cs2)=O)CCCCC1C 72144,N1(C(C(=O)N(c2cccc(OC)c2)C)=O)CC2CC2(C(N(CCOC)C)=O)C1 72145,N1(C(COCC(=O)OC)=O)CC2CCC(C1)C(NC(=O)C(C(C)C)C1CCC1)C2 72146,C(C)(CCC(=O)N1CC(OC)CC1C(=O)NCc1ncc(C)s1)OCC 72147,C1(C(=O)NC)CCCC1NC(=O)NCCCC1CCOC1=O 72148,c1(C(=O)NCC(C2(NC)CC2)O)ccc2c(c1)C(C)(C)OC2 72149,c1(C(N(C(C)CCNC(c2cnc(S)n2C)=O)C)=O)c(Cl)nc2ccccn12 72150,N1(C(C(C2CCCCC2)OC)=O)CCCC2(NC(c3cnsc3C)=O)CC2C1 72151,CCC(F)(F)C(=O)NCC1C(Cn2cc(-c3ccc(C(=O)O)nc3)nn2)C1(F)F 72152,Cc1ccnc(C(F)(F)C(=O)NCC(O)CNC(C2C=CCC2)=O)c1 72153,C1(CC(=O)NCCCNC(C2C(C)(C(F)F)C2)=O)CCSCC1 72154,N1(C(c2ccc(C)cc2)=O)CC(C(=O)N(C2CC2)CC2CC2)CC(C)(C)C1 72155,CN1CCN(C(C2(F)CCCOC2)=O)c2cnccc21 72156,C1(NC(c2ncccn2)=O)CCN(C(=O)CC23CCC(CC2)CC3)CC1F 72157,C1(Cn2cc(Cc3c(I)cn(CO)n3)nn2)CCCC12CCOCC2 72158,Cc1c(Br)ccc(F)c1C(=O)NC(C1CN(C(=O)C(C)(C)C#N)CCO1)C 72159,c1(CC)cc(C(=O)NCC(C23CCC(CC2)C3)NC(=O)C=C2CCC2)cc(C)c1 72160,c1(OC)c(C)cnc(C(c2nnnn2C)NC(c2cncc(Br)c2)C2CC2)c1C 72161,c1(C(=O)NCC2CCN2C(=O)CC2CC=CCC2)cc2c(C3CC3)cccc2[nH]1 72162,C=CCCCC(C(=O)NCCC(F)(F)Cl)NC(C1CNC(=O)N1)=O 72163,C(=O)(C(CC(C)C)NC(C1CC(O)C1)=O)NC(COC)CCO 72164,CCCCCCC(CC)C(=O)NCC12CC(C1)C(NC(=O)COC)CO2 72165,c1(C(N2CC(NC(=O)COCc3ccccn3)C2)=O)ccnnc1S 72166,CC(=O)CCCC(=O)NC1CS(=O)(=O)CC1NC(=O)C1=CCC1 72167,c1(C(=O)NC2C(NC(C(C)CC3CC3)=O)CCC2)c[nH]nc1S(N)(=O)=O 72168,C(N=c1ccnc(NC2CS(=O)(=O)CC2OC)[nH]1)c1c(CC)con1 72169,c1(NC(C)C(N2CCCCC2CNC(c2ncn(C)n2)=O)=O)ccc(Cl)cc1 72170,C1(C(=O)N)CCC(C2CCCC2)O1.CC(C)CN(CC(=O)NCN)C(=O)OC(C)(C)C 72171,C1(C(C)C)CCC(C)CC1CN(C(C(=O)Nc1cc(-c2ccccc2)on1)=O)C 72172,Cc1cc(C(N2CCC3C(C2)CN3C(=O)CN2CCC2C)=O)cc(C)c1C 72173,C1(C)(NC(C(C)N(C)Cc2ccccc2)=O)CC(NC(=O)Cn2cnnc2O)C1 72174,N1(C(c2c(C)coc2)=O)CC(CC(=O)NC2CC3C=CC2C3)C2(CC2)C1 72175,N1(C(C(C)OCCOCC)=O)CCCC2(CCN(C(C3(CC)CCC3)=O)C2)C1 72176,c1(C(=O)NCC(C2CCC2)Nc2nccc(C3CC3)n2)ccc2ocnc2c1 72177,C(=O)(CC(F)(F)C(C)(F)F)N1CCCC(C)(CNC(C=CCCC)=O)C1 72178,C1(NC(c2scc(C)c2)=O)CCC2(CC1)CC2NC(=O)Cn1c(C)c(C)sc1=O 72179,N1(C(C(C)N(C)C)=O)CC2(CCCCN(C(=O)C(C)S(C)(=O)=O)C2)C1 72180,N1(C(c2cnn(CC)c2C)=O)CC(CNC(=O)CC(F)(F)Cl)CC12CCC2 72181,Cn1nccc1CC1CCN(C(c2cc(C(C)F)on2)C(=O)NC2CCOC2)C1 72182,CCC(C)C(=O)NC1CC(O)C1CC(=O)N(C(CC)CO)C 72183,N1(C(C)=O)CCC2(CC1)CN(CC1CCC(C(F)C(=O)O)CC1)CCO2 72184,c1(SC)ncc(N)c(C(=O)N(CCNC(=O)CCc2nc[nH]n2)C2CC2)n1 72185,C1(NC(C(CSC)O)=O)CN(C(c2csc(Cl)n2)=O)CC2(CC2)C1 72186,N1(C(c2ccc(OC)c(Br)c2)=O)CC(NC(C)=O)C(C2CC2)C1 72187,N1(C(=O)NC2CCc3ncccc3C2)CCS(=O)(=O)c2ncc(Br)cc21 72188,C1(CNC(Cn2c(=N)nc[nH]2)=O)CCC(NC(c2cccc(=O)o2)=O)CC1 72189,C(=O)(CCC(C)S(C)(=O)=O)N1CCC2(CN(C(C(C)C3CCCC3)=O)C2)C1 72190,C1(C(N2CCC(COCC)C2)=O)CC12CCN(C(C1(O)COC1)=O)CC2 72191,n1(CCC(=O)NC2CN(C(C3CC34CC4)=O)C2)c(=O)oc2cc(Cl)ccc12 72192,N1(C(C(CC=C)NC(C2CC(C)N(C)C2)=O)=O)CC2(CC(F)C2)C1 72193,C1(NC(C(C)=C2CCCC2)=O)CC2CCC(C1C)N2C(c1cc2cscc2s1)=O 72194,C12(C(N3CCC(OC(C)=O)C3)=O)CCCC1CCN2C(C1CC2CC(=O)C1O2)=O 72195,c1(OC)ccc(C(=O)NC2CCCC2CNC(C)=O)c(NC(=O)C(C)(C)CF)c1 72196,C1(CC)(NC(C2CC(C)CO2)=O)CCN(C(c2cc(CC(C)C)nn2C)=O)CC1 72197,c1(C(=O)NC2CCN(C(c3c(C)cc(Cl)cc3)=O)C2C)cnc2c(c1)nnn2C 72198,c1(OC)cncnc1C(=O)NCC(c1ccc(C)cc1)NC(=O)CN(C)C(C)=O 72199,Cc1ccc(OCCC(=O)NC2CN(C(=O)CC3CCC(C)(C)CO3)C2)c(Cl)c1 72200,C1(C2CCN(C(=O)COCCN(C)C)C2)(NC(CCCC)=O)CC1 72201,CCC(CCCC(F)(F)F)NC(=O)NC1CC=CC(N)C1 72202,c1(C(=O)NC2CCC3CCN(C(=O)C4=CCSC4)C23)ccc(Cl)c2ncccc12 72203,C(=O)(C1=CCC(NC(=O)CC2CCCC(=O)C2)C1)Nc1cccc(C(C)=O)c1 72204,CC(C)(F)C(=O)NC1CCCC1CNC(c1cn(CCF)nn1)=O 72205,c1(-n2cc(CC3N(C(CC=C)=O)CCC3)nn2)ccc(F)cc1Br 72206,Cc1ccc(OCC(=O)NCC2CCC=CCC2)c(Br)c1 72207,C(C(=O)NCC1(F)CC(NC(=O)CNS(N)(=O)=O)C1)(C(C)C)OC 72208,C=CCCCCCCCCC(C(=O)NCCC)N1C2CCCC1CC(O)C2 72209,Cc1cc(=NC2CCC(N3CCOCC3)C2)[nH]c(=NCC2COC(C)(C)C2)[nH]1 72210,CC(C)C(CC(=O)NCC1(NC(=O)Cn2ccccc2=O)CCOC1)C(C)C 72211,C(c1cccc(Cl)c1Cl)=CC(=O)N(C1CCCN(C2COC2)C1c1nn[nH]n1)C(C)=O 72212,C1(NC(N(CCc2nc(C)on2)C)=O)CC2CCN(S(C)(=O)=O)CC12 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72282,N1(C(CCCCOC)=O)CC2CCN(C(=O)CC3(N(C)C)COC3)C2C1 72283,C=CCC(C(=O)N1CCOC(C(=O)NCC(C)(C)SC)C1)OC 72284,c1(NC(C2CC=CCN2C(C2CC3CC2CC3O)=O)=O)cc(F)ccc1O 72285,n1(Cc2n(CC=C)nc(-c3ccc(N(C)C)nc3)n2)ncc2cc(C)cnc12 72286,c1(OC)cc(C=CC(=O)NCC2(O)CCCCCC2)ccc1OC(F)F 72287,C(C1c2ccsc2CCN1C(=O)C=C1CCC1)NC(C1CC2CCC2C1)=O 72288,N1(C(C2(CC#C)CCCO2)=O)CCC2C(C1)CN2C(=O)CCc1nc(C)c(C)o1 72289,N1(C(C2OCCN(C(C(N3CC4CC4C3)C)=O)C2)=O)CCC(O)C(N(C)C(N)=O)C1 72290,c1(C(N2CCC(OCCNC(c3c(C)onc3)=O)C2)=O)cc2c(cn1)OCCO2 72291,N1(C(C(N2CC(CC)OCC2)=O)=O)CC(=O)N2CCc3ccccc3C2C1 72292,N#CC1(C(=O)NCC(O)CNC(=O)CCSc2ccccc2F)CCOC1 72293,c1(C(N(C)CCOCCNC(C2(C(F)(F)F)CC2)=O)=O)cc([N+](=O)[O-])c[nH]1 72294,N1(C(C(COCC)F)=O)CCCC(C2CC2NC(=O)OC)C1.C12(CC1)C(=O)N2 72295,c1(N2CCC(NC(=O)Nc3cccc(Cl)c3Cl)C2)cnnc(O)c1Cl 72296,CC1(C(=O)NC2(CCNC(C3CCC(C(F)(F)F)C3)=O)CCCC2)CCCCC1 72297,C(=O)(C1OCCc2ccccc21)NCC1N(C(COC(CC)(C)C)=O)CCCC1 72298,c1(C(N2C(C)CCN(C(=O)C=Cc3cc[nH]n3)CC2)=O)ccc2c(c1)CCCC2 72299,C(C)(C)(CCCC(=O)NCCC1CCC(C)C1)NC(C1OCCN(C)C1)=O 72300,c1(OC)ncnc(C(N2CCC(C)(CCNC(C3CC3(F)F)=O)C2)=O)c1F 72301,C1(NC(c2cnn(CC(F)F)c2)=O)CC(NC(=O)C2CC2)C12CCC2 72302,N1(C(COCC(C)C)=O)CCC(OCC2CCN2C(=O)OC(C)(C)C)CC1 72303,C(=O)(C(C(C)C)C1CCC1)N(C(c1ccccc1)CNC(C(C)(C)OC)=O)C 72304,c1(C(N2CCC(NC(=O)C(c3ccc(Cl)cc3)(F)F)C2)=O)cnn2ccsc12 72305,C1(C2CCN(C(=O)CCC3CCCOC3)C2)(NC(CCNC(=O)C=CCl)=O)CC1 72306,c1(C(=O)NCC(CN(C(C2C(C)C2C)=O)C)C)c[nH]c2nccc(Cl)c12 72307,c1(C(N(C2CN(C(C3ON=C(C)C3)=O)CC23CC3)C)=O)n[nH]c2c1CN(C)CC2 72308,C1(CC(=O)N(c2ccccc2)C)OCC2CN(C(c3cnc(O)c(Br)c3)=O)CCC12 72309,N1(C(C2CC(C#C)(O)C2)=O)CC(C)N(C(c2cnn(CC)c2C)=O)CC1C 72310,C(=O)(C(F)(CNC(=O)OC)C(C)C)NC1C(NC(CCN(CCC)C)=O)CCC1 72311,Cc1nc(C(=O)NCC(CNC(=O)CC2CC=CCC2)CO)cs1 72312,C#CCCC(N)C(=O)NCCc1nc(CN2CCNC(=O)C2)no1 72313,C1(CNC(CC(C)SC)=O)CN(C(c2cc(C#N)c[nH]2)=O)CCC1C 72314,c1(C(=O)NC2(C)CCCN(C(C(CC)(C)O)=O)C2)cccn2c(C)nnc12 72315,C=CC1CCCC(c2nnnn2CCCC)(Nc2cn(C)c(=O)cc2C)C1 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72387,C1(C(=O)NCCc2ccncc2)CN(C(=O)Nc2cnccc2Br)CC(F)(F)C1 72388,CC1CCN(C(=O)C(O)C2CCCC2)C(C)C1NC(=O)C(C)OCC1CC1 72389,c1(C(C)NCC(c2c(OC)cccc2)N(C)C)cc2cccc(F)c2o1 72390,N1(C(CCOC)=O)CC(NC(=O)Cc2cccc(C(C)(C)C)c2)C(C)(C)C1 72391,C1(c2n(CCOCC)nnn2)(NCCc2cc(C)cc(C)c2)CCC(C)(C#N)C1 72392,c1(C(=O)NC(CN(C(C2(OC)CCCOC2)=O)C)C)cc(C)ccc1F 72393,CC1CN(C(c2sccc2CNC(c2snc(Cl)c2Cl)=O)=O)CC1CCN(C)C 72394,C1(OC)CCC2(CCN(C(=O)NC3CCCCC3C(=O)Nc3ccccc3)C2)C1 72395,C1(NC(Cc2scc(C)c2)=O)CC=C(C(=O)NC2C(C)CCC2C)C1 72396,CC1(C#CC(=O)NC2CC2CNC(c2c(F)c(F)cc(F)c2F)=O)CCCO1 72397,c1(C(C)(C)C)ncc(C(=O)NCC2(O)CN(C(=O)CCCc3ccccc3)C2)s1 72398,C1(CNC(CC2C(C)=NNC2=O)=O)CCN(C(=O)Cc2cnsc2)C12CC2 72399,S(=O)(=O)(c1c[nH]ccc1=NCC1CCC(CN2CCC(SC)C2)CC1)SC 72400,C(=O)(C(C)(C)C(=O)N(C)CC1CCCC(NC(c2ncccc2SC)=O)C1)NC 72401,N1(C(CCCOC)=O)CCCC2(C1)C(NC(c1nc(C)ncc1Cl)=O)CCN2C 72402,C(=O)(CC(C)(C)O)N(C(C)CNC(=O)CN1CCCC1C)CC 72403,c1(C(N2CCC(N(C(c3c(C)nc(O)[nH]3)=O)CCO)C2)=O)cc(F)ccc1Cl 72404,Cc1cc(C(C)(C)C(=O)N(CC(=O)NC(C)(C)C)CCO)cs1 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72423,CCC(O)C(C)(C)C(=O)NC1CC(F)(F)CC1NC(=O)COCCCOC 72424,N1(C(C)CNC(c2coc(CO)c2)=O)CCN(C(C2CCCC2(F)F)=O)CC1 72425,CCCC(C(=O)NC(C)Cn1cccn1)NC(=O)CN(C)CC1CCOC1 72426,N1(C(CC2(C=C)CCOCC2)=O)CC2CC(NC(c3ccccc3C)=O)C(C2)C1 72427,N1(C(C=CCCC)=O)C2CCC1CC(NC(=O)Cn1ccc(Br)n1)C2 72428,N1(C(CSCC(=O)OC)=O)CCN(C(C2CCC2(F)F)=O)C(CO)C1 72429,C1(C)(C(=O)NC2CN(C(COC3(C#C)COC3)=O)C(CO)C2)CC2(CCC2)C1 72430,O=C(CC1=CCCCC1)NCC12CCC1CN(C(C1CC(=O)NC(=O)N1)=O)C2 72431,C(CCCC(C)(C)N(C(C1CCCN1C(=O)C1CC1)=O)CC)NC(C(C=C=C)C)=O 72432,C(C(=O)NC(C(=O)NC1CC=CC1)C1CCC1)(C(C)C)OC 72433,c1(-c2nc(CSc3[nH]n(CC(C)C)c(=O)c3)on2)ccc2c(c1)COC2 72434,CC1CN(C(c2ccccc2C2(C)CC2)=O)CCN1C(=O)COc1ccccc1 72435,Cn1nc(CC(N2CC3CC3(NC(C34CC(F)(C3)C4)=O)C2)=O)cc1C(F)(F)F 72436,N1(C(c2cccc(C)c2C)=O)CCC2CN(C(c3ccc(=N)[nH]c3Cl)=O)CC12 72437,N1(C(CCC(CC)C)=O)CCOC2(CCN(C(=O)C(C)C3CCC3)CC2)C1 72438,C(=O)(C(CC)C(=O)OCC)NCCc1ccn(CCC)c1.N1(C=O)CC=CC(OC)C1 72439,C(CCCCCNC(c1ccncc1Cl)=O)NC(C(C)ONC(=O)OC(C)(C)C)=O 72440,c1(OC)sccc1C(C(=O)NC1CC1)N(C(C)C(C)C)Cc1ccccc1 72441,Cc1c(CCC(N2CC(NC(C3CN(C4CCC4)C3)=O)C(C)C2)=O)cnn1C 72442,C=C1CCN(C(=O)CC2CCC2)C(C(=O)NC2CCN(C(C)=O)C2)C1 72443,C1(CNC(Cc2cc(C)sc2C)=O)CC(C)(C)CCC1NC(=O)CCF 72444,N1(C(C(COC)N(C)C)=O)CCCC1(C)CCC(=O)NCCc1ccc(O)cc1 72445,N1(C(C2(C(N)=O)CCC2)=O)CCN(C(=O)C=C(C2CC2)C2CC2)C(CC(F)F)C1 72446,c1(CN2CC(NC(CCc3c(C)ncs3)=O)(CO)C2)c(I)ccnc1Cl 72447,C1(NC(c2c(CC)ncs2)=O)CCN(C(c2cccc(C)c2)=O)CC(C)(C)C1 72448,S(=O)(=O)(c1cc(C(=O)OC)c(Cl)cc1Cl)N1CC(C#C)(c2ccccc2)C1 72449,N1(C(c2c(OCC#C)nccc2)=O)CCN(C(c2csc(C)n2)=O)C(CCO)C1 72450,C1(NC(C2C(C(=O)OC)C2)=O)CCCN(C(c2cc(C)co2)=O)CC1 72451,CCC(c1ccc(OC)cc1)=CC(=O)N(C)CCN(C)C(c1ccc(C)n1C)=O 72452,C=CCCC(CC(C)C)C(=O)N1CCC2(CC(NC(C3(F)CCOC3)=O)C2)C1 72453,C1(C(=O)NCCc2nc(CC)[nH]n2)N(C(=O)C(O)CSC)CC12CCCC2 72454,N1(C(C(N2CCCC(O)C2)C)=O)CC(N=c2[nH]c3c(F)cc(Cl)cc3s2)CC1C 72455,C(=O)(CCC(CC)CCC)NCC1C2CN(C(C3(C=C)CC3)=O)CC21 72456,c1(CC2(C)CCCN2C(=O)CC2(C)CC2(Cl)Cl)ccc(F)c(F)c1 72457,c1(C(C)C)nccn1CC(=O)NC1COCC1N1CCOCC1 72458,N1(C(c2c(C#C)c[nH]n2)=O)CC(C)(C)CC1CC(N1CC(N2CCCC2)C1)=O 72459,CC1(C)C(CO)CCN1C(c1ncc(C(F)(F)F)s1)C(=O)NC1CCOC1 72460,c1(C(=O)NCC2(CNC(C(CCO)N(C)C)=O)CC2(F)F)n[nH]c2c1NCCC2 72461,N1(C2C(NC(=O)COCC3CCOC3)CCC2)CCN(C(=O)C=CCO)CC1 72462,c1(C(N(CCN2CCN(C(C(C)OC)=O)CC2)C)=O)cc2cccnc2[nH]1 72463,c1(OC)ccc(C(N2CC(O)(CNC(=O)C(O)CCC(C)C)C2)=O)c2ccoc12 72464,C(=O)(C1=CC(C)(CC)C1)N1C(C(=O)NC2(C#C)CCC2)(COC)CCC1 72465,C(CN(C)C)(CN=c1ccc(Br)c(S(=O)(=O)NCC(COCC)C(C)C)[nH]1)OCC 72466,N1(C(c2c(CC)cns2)=O)CCCCC1C(=O)NCC1(O)CCCOC1 72467,C1(CC)C(NC(=O)CCc2ccccc2Cl)CCN1C(=O)C=CC1CCCO1 72468,C1(NC(C2C(=C)C2)=O)(CO)CN(C(c2coc(Br)c2)=O)C1 72469,N1(C(C2C(=O)NCC2)=O)CCC2CCCC(C1)N2C(c1cncc2sccc12)=O 72470,c1(CC(=O)NC(CNC(c2c(C)ncc(Br)c2)=O)CO)ccccc1[N+](=O)[O-] 72471,c1(C(=O)NCCC2CCN(C(c3cc(N(C)C)ncc3)=O)C2)c(F)cncc1Cl 72472,c1cc(P(C)(C)=O)cs1.c1(C(CCO)N(CC)C)ccccc1 72473,N1(C(C2C(C)C2)=O)CCN(C)C(CNC(C2(c3ccc(Br)cc3)CC2)=O)C1 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72631,CCC(CC)(CO)C(=O)N1CCC(NC(C2CCn3cncc3C2)=O)CC(O)C1 72632,Cc1nccc(C(N2CC(c3ocnc3CNC(=O)CCCF)C2)=O)c1N 72633,N1(C(C2(C)CC=CCO2)=O)CC2=C(C1)CN(C(=O)CCNC(c1cccs1)=O)C2 72634,C(CC(C(=O)NC1(C)CC1)NC(=O)C(F)C(C)C)OC 72635,C1(CCCNC(CC2CCC(C)O2)=O)CCN(C(=O)COc2ccccc2)CC1 72636,c1(C(=O)NC(C(C)C)CNC(=O)C=CC2CCCC2)cc2scnc2[nH]1 72637,C1(C(=O)NC(C(=O)NCCC)CC)C2CCC(C2)N1C(=O)CCC1(C#N)CCC1 72638,C1(N(C(Cc2ncc(C)o2)=O)C)CN(C(=O)CC2CN(C)C2)CC1F 72639,CC1(C)OCCOC1C(N1CCC(F)(CNC(c2cc(O)ccc2F)=O)CC1)=O 72640,CS(=O)c1ccc(C(=O)NCCC2CCCN2C(=O)Cc2ccc(Cl)cn2)cc1 72641,c1(CNC(C2(NC(C3CC3C(F)(F)F)=O)C(C)(C)C2)=O)ccccc1O 72642,CCC(CC(=O)N1CCC(NC(C23CCCCC2C3)=O)C1C)C1CCC1 72643,C1(C2CC2)(C(=O)NCC(CNC(CCC)=O)OC)CCOCC1 72644,C(=O)(CCC1=CCCCC1)N1CCN(C(CCCC#CC)=O)CC1CC(F)(F)F 72645,c1(CC(=O)NCC(C)NC(=O)CCc2ccc(Cl)nc2)cccc(F)c1 72646,C1(NC(=O)CC2CCCCC2)CC12CCN(C(c1ncc3[nH]ncc3n1)=O)CC2 72647,O=C1CSc2cc(C(N3CCC34CN(Cc3cnc(O)c(Cl)c3)C4)=O)ccc2N1 72648,C1=C(C)C(=O)NC(C(C)C)C(=O)NCCCn2cc1nn2.c1(SC)ccccc1 72649,C1(CNC(CCC2CCN(C(c3c(CC)cco3)=O)C2)=O)CCC(C)N1C 72650,N1(C(C(OC)OC)=O)CCCC(CCNC(=O)CCCc2cccc(Cl)c2)C1 72651,C1(NC(C2CN(C)C2)=O)CN(C(c2cccc(CC#N)c2)=O)C2CCCCC12 72652,C(C1CCCCCC1)=CC(=O)N(CCCCN(C(C1CCC(OC)C1)=O)C)C 72653,N1(C(C(CC)NC(N)=O)=O)CCC2C1CCCN2C(c1cc(Br)cc2[nH]ncc12)=O 72654,C(=O)(CC(C)C(=O)OC)NCCC1(O)CCN(C(C2(OCC)CCOCC2)=O)C1 72655,C1(C2CN(C(=O)C(C)Cn3ccnc3)C2)(NC(Cc2c(C)n[nH]c2)=O)CC1 72656,C1(CCN(C(=O)CSCC2CCCCO2)C)CCCCN1C(c1cc[nH]n1)=O 72657,c1(C(=O)NCC(CCNC(CCC(=O)NCC)=O)O)cnc(C)cc1Cl 72658,Cc1nn(C)cc1S(=O)(=O)N1CC(N2CCN(C(c3sccc3I)=O)CC2)C1 72659,C1(OC)CC2CC1CN(C(C1CCCCC1(C)NC(c1cn(C)c(C)n1)=O)=O)C2 72660,Cc1ncnc(O)c1C(=O)NC1CCN(C(C2CCC3(CCC3)O2)=O)C1 72661,CC(C)(C)C(CNC(=O)Cc1nc(=N)[nH][nH]1)NC(C1CC1Sc1ccccc1)=O 72662,c1(C(=O)NCCC2(C(=O)NCC3(OC)CCC3)CC2)nc(C)sc1C 72663,C(=O)(C(O)(C(F)(F)F)c1ccccc1)N1CCC(CCNC(C2(F)CC2)=O)C1 72664,C(=O)(C1CCCc2n[nH]cc21)NCCCC(C)NC(C1CC1(F)F)=O 72665,N1(C(CC(C)O)=O)CCC(F)(F)C(CNC(c2cc(C3CC3)n(C)n2)=O)C1 72666,Cc1nnc(NC2CC(NC(c3sccc3C)=O)C2)nc1C 72667,c1(N2CCN(C(CCC)=O)CC2)cc(C)nc(C)c1[N+](=O)[O-] 72668,C1(C(=O)NC(C2(OC)CCC2)C)CC2CN(C(c3ncn(C)n3)=O)CC2C1 72669,C(C1CCCN1C(c1coc(CO)c1)=O)=CC(=O)N(C)Cc1ccco1 72670,N1(C(C#CC2(CC)CC2)=O)CCCC2CN(C(C3(CO)CCC3)=O)CC12 72671,S(=O)(=O)(C1=Cc2ccccc2CCC1)N(C(C)C(=O)O)CC=C 72672,Cc1c(C(=O)NCc2ncc(C(N3CC(C)CC3C)=O)cn2)c[nH]c1C#N 72673,CCC(C)C(O)CC(=O)N1CCOC(CC(=O)NCC(C)(F)C(C)(C)F)C1 72674,c1(C(N2CCC(CN(C(C(N3CCC(O)CC3)C)=O)C)C2)=O)cccc(Cl)c1Cl 72675,N1(C(CC(C=C)C)=O)CCN(C(=O)CCc2cc(OC)no2)CC2(CC2)C1 72676,N1(C(C=CC=CC)=O)CCC(NC(c2cn(C)nc2CCC(F)(F)F)=O)C1C 72677,c1(C(C)(C)C)nc(Cl)cc(=NC(CO)C2CCN(Cc3ccccc3)CC2)[nH]1 72678,N1(C(CSCC#C)=O)CCCC(C(C)(C)C(=O)NCc2cnn(CCC)c2)C1 72679,C1(NC(=O)C=Cc2ccncn2)CCN(C(C2CC2(F)F)=O)CC1CO 72680,C(=O)(C(F)(F)C(F)(F)F)N1CC(NC(=O)Cn2ncc(O)nc2=O)C(O)C1 72681,C1(C(N(CC(=O)N(CCCC(C)C)C2CC2)C)=O)CNC(=O)CC1C 72682,c1(NCCN=C(NCc2c(C)nn(C)c2)NC2CC2C)ccc([N+](=O)[O-])c(F)c1 72683,n1(CCC(=O)NC2C=CCN(C(CSCC#C)=O)C2)nc(O)c2ccccc12 72684,C1(C(N2C(C)(COC)CCC2)=O)CC2CCCC2N1C(=O)C1=C(C#N)CCC1 72685,N1(C(C(c2cn(C)nn2)NC(CC=CC)=O)=O)CCC(C(C)C#N)CC1 72686,N1(C(c2cncc(C)c2)=O)CCN(Cc2cccc(C)c2O)C2CC12 72687,C(=O)(CCCC(=O)NCC1CN(C(=O)CC2CCCCN2C(C)C)CCO1)OC 72688,N1(C(Cc2nc(C)c(C)s2)=O)CC2CC1CN(C(C1CCC(C)O1)=O)C2 72689,C(=O)(CS(N)(=O)=O)NC1(C(N2C(C(C)O)CC2)=O)CCC1 72690,N1(C(C(=O)NCCC(C)c2ccco2)=O)CCC(NCC(F)F)CC1 72691,C(C(CC)(CC)C(N)=O)NC(C1C(CNC(CCC=C=C)=O)CCC1)=O 72692,N1(C(CS(C)(=O)=O)=O)Cn2cc(C(=O)O)cc2C1 72693,c1(SC)cc(NNC(=O)NC2COC3(CCNCC3)C2)ncn1 72694,CCCCCCC(=O)NC(C(=O)N(C)CC1CCOCC1)c1cccs1 72695,n1(CCOCC)nc(-c2cccc(C(F)(F)F)c2)nc1CCCC1CCCCC1 72696,CCC(C)C(=O)C(=O)NCC1C(C)CCCN1C(c1cnn(C(C)C)c1)=O 72697,C1(NC(C(C)CO)=O)CCC2(CC1)CN(C(c1cc(C3CCOCC3)[nH]n1)=O)C2 72698,Cc1cc(NC(=O)CN(C(=O)C(F)C(C)(C)O)C(C)C)cc(C)c1O 72699,c1(CC(=O)NCC(CNC(C(C)OCC(C)C)=O)CO)ncc(F)cc1F 72700,C(=O)(C1=CC(O)C(NC(C2(C)COC2)=O)C1)NC1(CO)CC(OC)C1 72701,c1(OC(C)C)ccc(COC(c2ccccc2CS(C)=O)=O)c(Cl)c1 72702,C1(NC(C2OCCN(C(C=CCOC)=O)CC2)=O)CCCCN(C)C1=O 72703,C1(C(=O)NC(CNC(c2c(SC)csc2)=O)C2CC2)CCCCCCC1 72704,N1(C(C(COC)(F)F)=O)CCCC2(CC(NC(c3cc(Cl)ccc3Cl)=O)CO2)C1 72705,C1(NC(CC=C)=O)CC2(CCN(C(c3cc4sccc4cn3)=O)CC2)C1 72706,N1(C(C(C)=C(C)C)=O)CCCC1CCNC(c1ccco1)=O 72707,N1(C(c2[nH]cc(CC)c2)=O)CC(C2CCN(C(=O)Cn3[nH]cnc3=N)CC2)C1 72708,N1(C(c2cc(C)cc(F)c2)=O)CCC2(CC2)CC1C(=O)NC(C)C(C)(C)O 72709,c1(C(=O)NCC(C)NC(Cc2c(C)cco2)=O)cc2c(n1C)CCOC2 72710,C(=O)(CC(CC(C)C)NC(=O)CCn1cnc(=N)[nH]1)Nc1cn(CC)nc1 72711,N1(C(c2ccc(N(C)C)cc2O)=O)CC(C2CC2)C(F)(C(=O)O)C1 72712,C1(C(N2CC(NC(c3c(CC(C)C)cccc3)=O)C(O)C2)=O)CCN(C)S1(=O)=O 72713,C1(CCNC(CC)=O)CCCN(C(=O)CSCC(N2CCCC2)=O)CC1 72714,c1(C(N2C(CO)CC(NC(c3cc(C)oc3C)=O)C2)=O)ccc2c(c1)NCCC2 72715,C=C(C)C(C)(C)C(=O)NC1CCCC(CNC(c2ccc(C(F)(F)F)nn2)=O)C1 72716,C1(C(=O)OCC)CN(C(=O)C=CC(=O)NCC2(F)CCCC2)CC12CCOCC2 72717,C1(N(c2cccc(-n3cnnc3)c2)C(c2c(C)noc2)=O)CCNCC12CC2 72718,c1(C(c2n(CC)nnn2)OC(C2CCCCC2)CNCC)nccc(Cl)c1C 72719,Cc1cnc(C(=O)NCC2(C(=O)NCCC3(C)N=N3)CCCCC2)c(C)c1 72720,C1(CC(=O)N(CCCCN(C(=O)Cc2cnco2)C)C)OCCC1(C)C 72721,S(=O)(=O)(c1cccc(C(=O)NC(c2ncccn2)(C)C)c1)N(C(CC)C(N)=O)C 72722,c1(C(=O)NC2C(C)CN(C(C34CC(CC(F)F)(C3)C4)=O)C2)cc([N+](=O)[O-])ccn1 72723,N1(C(CCCC#C)=O)CCOCC(NC(=O)CCCn2cc(C)cn2)C1 72724,C1(C(=O)NCC2(O)CN(C(CNC(C(CC)C)=O)=O)C2)CNC(=O)C(C)(C)C1 72725,CC(C)C(F)(CNC(C1CCCC12CCC2)=O)C(=O)N(C)CC1CCOC1C 72726,C(=O)(C(C)(C)CC(=O)NC(c1ccccc1F)CNC(=O)C(C)CF)OC 72727,c1(C(=O)NC2C(OC)CN(C(c3cccn3C)=O)C2)ccc2c(N)nccc2c1 72728,N(C1COc2cc(Br)cc(C)c21)C(=O)Nc1ccc(-c2nc(C)[nH]n2)cc1CO 72729,C=CCCC(C(=O)NC1CCCN(CC2CCC2)C1)CC 72730,N1(NC(c2nc(CC)on2)=O)CCCC(n2cc(C(C)(C)F)nn2)CC1 72731,c1(C(C2(C)CSC2)NC(COC)(C)C2CC2)nnnn1CSc1ccccc1 72732,CC1C(C)N(C(=O)CC23CCC(CC2)OC3)CCN1C(=O)C(C)OCCN(C)C 72733,C1(N)(CCC)CCN(Cc2cn(Cc3ccccc3)cn2)CC1 72734,c1(C(=O)NCCC(=O)OCC)cnn2cccc(-c3ccc(C#N)c(F)c3)c12 72735,c1(C(=O)NCCC2CC(NC(CC#N)=O)C2)ccc2c(c1)S(=O)(=O)NC2 72736,C(=O)(C(C)(C)CCC#N)NC1COCC1C(NOC(C=C)C)=O 72737,c1(NCC(C)(C)OC)nc(C)cc(=NC(C)c2ccc(C#N)c(C)c2)[nH]1 72738,C(=O)(C(O)CC[S+](C)C)N(CCCNC(C(C)OCCC=C)=O)C 72739,C1(NC(c2n(C)nnc2)=O)CCCC(NC(C2CC=CCC2)=O)C1 72740,C(=O)(NN1CCCC1C(=O)N(C1CCCC1)C)C1CC(N(C)C)C1 72741,c1(OC)cc(C2(C(=O)NCC(C)(O)CNC(=O)CC3CC(F)C3)CC2)ccc1C 72742,c1(COCCNC2CCN(C(C(c3ccccc3)SC)=O)C2)ccnc(F)c1N 72743,N1(c2cc(C)ncn2)CCCCC(NC(=O)Cc2c(F)cccc2F)CC1 72744,c1(CCC(=O)NC2CCC(CNC(C3(C)CC3)=O)C2)cc(Cl)ccc1Cl 72745,n1(C(C(=O)NC(C(C)C)c2nn[nH]n2)C)cc(C(C)CC2CCC2)nn1 72746,CCC(C)(O)CCNC(C1(NC(C2C3CCCOC23)=O)CCSC1)=O 72747,Cc1ccc2ncc(C(N3CCCC(N(C)C(c4coc(C)n4)=O)C3)=O)n2c1 72748,c1(CN2CC(O)(C(=O)NC3CCC3)C2)cccc2c1oc1ccccc21 72749,C(=O)(CCCCCF)NC1C(C)CN(C(c2cnc(C(C)(C)C)[nH]2)=O)C1 72750,C1(C(N2CC(C)C(C(=O)N(c3ccccc3O)C)C2)=O)CCCCCN1C 72751,CC12CN(C(=O)Cc3ncc(Cl)s3)CC1CN(C(c1coc(C(F)F)n1)=O)C2 72752,c1(NC(CSCCC(=O)NCc2n[nH]c(O)n2)=O)cccc(C(F)F)c1 72753,C1(NC(c2c(OC)csc2)=O)CCCC(CNC(=O)C(C)C2CCC2)C1 72754,C(CNC(=O)C=Cc1ccnn1C)(C(C)C(C)C)NC(Cn1c(C)cnc1)=O 72755,c1(C(=O)NC(C2CCCN2C(=O)CS(=O)(=O)N(C)C)C)cc(C(=O)N(C)C)oc1C 72756,c1(N2CCCC(NC(C(c3cn(C)nc3)O)=O)CC2)ncnc2c1ncn2C1CC1 72757,N1(C(C(C)=CC2CC2)=O)CCC2(NC(c3conc3C)=O)CC2C1 72758,C1(NC(c2ccc(C(N)=O)[nH]2)=O)CCN(C(C2CN(C3CCC3)C2)=O)CC1F 72759,c1(C(=O)NCC2(F)CC(CNC(C(CC(=C)C)C)=O)C2)cncc(S(C)(=O)=O)c1 72760,c1(C(=O)NCC2N(C(C3CCC(C)(C)CO3)=O)CC2)c(Cl)cccc1[N+](=O)[O-] 72761,c1(CC(=O)NCC(=O)NC2CCC2CNC(=O)Cc2cnns2)ccccc1 72762,N1(C(CCOCCOC)=O)CCC(C2(NC(c3ccc(N)c(C)c3)=O)CC2)CC1 72763,CC(C)CCCCCC(=O)NCC1C2CC1N(C(c1coc(Cl)n1)=O)C2 72764,C(=O)(C(C)(C)n1cccn1)NCCN(C(CCNC(COC)=O)=O)C 72765,c1(CNC2CC(C(=O)Nc3ccco3)OCC2)ccc(-c2cncnc2)cc1F 72766,c1(CN2C(C(N3CCCC3)=O)CC(OC)C2)c(Cl)nc(SC)nc1Cl 72767,c1(CN(C(=O)CSc2nc[nH]n2)CCNC(CC2(SC)CC2)=O)ccccc1 72768,CC1CN(C(=O)CC(C)CN(C)C)CCCN1C(=O)CCn1cccc1 72769,c1(OC)cccc(Cl)c1C(N1CCC(CO)(Nc2ccncn2)CC1)=O 72770,N1(C(C2(CC)CCC2)=O)CCCC(C(C)C(=O)NCCN(C)C2CC2)C1 72771,C(CN=c1[nH]c(N2CCN(CC(F)(F)F)CC2)nc2c1CCC2)SC 72772,c1(C(=O)NC2C(NC(C(C)CN(C)C)=O)COCC2)ccc(Cl)c2ccccc12 72773,c1(N(C)Oc2ccc3c(c2)OCO3)nc2c(c(=NCCCP(C)(C)=O)[nH]1)COC2 72774,c1(OCC)cccc(C(N2CC(O)CC2C(=O)Nc2nc(C#N)cs2)=O)c1 72775,C1(NC(CCP(C)(C)=O)=O)CCN(C(=O)COC2CC(F)(F)C2)CCC1CO 72776,c1(COC(c2ccc(-c3ccccn3)o2)=O)cccnc1F 72777,c1(OCC)cccc(OCC(N2CC(C)(NC(C3(C)CC3Br)=O)C2)=O)c1 72778,c1(C(N2CCCC2Cn2cncn2)C(=O)NC(C)C)ncc(C(C)C)s1 72779,c1(OC)ccc(Br)cc1CN1CCCC1C(=O)Nc1cnc(C)nc1 72780,c1(C(=O)Nc2cc(C)c(C(F)(F)F)cc2)cccc(S(=O)(=O)NCCN(C)C)c1 72781,C(CC)(CCCC(=O)N(C)CP(C)(C)=O)NC(C1C(=C)C1C(=O)OC)=O 72782,CCCCCC(C)CC(=O)N1CCC(NC(=O)CCc2ccc(O)nn2)C(F)C1 72783,C(=O)(CC(C)CC(C)(C)C)N1C(C(=O)NC(C)C(=O)NO)CSCC1 72784,C(=O)(CC(F)(F)Cl)NCC(c1ccc(F)cc1)NC(CCNC(CC(C)C)=O)=O 72785,N1(C(CN(C(=O)OC)C)=O)CCC2(CCN(C(=O)CCC(C)OC)C2)C1 72786,C#Cc1nccnc1NC(C1CCCN1C(=O)CCNC(c1ccc[nH]1)=O)=O 72787,N1(C(CC(CC)C)=O)CC(NC(c2cc(C)cc(C)n2)=O)CC(O)C1 72788,N1(C(COCCCC#C)=O)CC2CCC(CNC(=O)C(O)CC(C)C)(C2)C1 72789,CC(Cl)(Cl)C(=O)N1CC(C(N)=O)(CNC(c2ccc(C(N)=O)o2)=O)C1 72790,C1(CNC(C23N(C(c4cc(C)ncc4)=O)CC(C2)C3)=O)OC(=O)CC1(C)C 72791,c1(NC(c2n(C)cc(NCc3ccc(Br)[nH]3)n2)=O)ccc(Br)cc1C(C)(C)C 72792,c1(OC)ccc(C(=O)NC2CCN(C(c3cc(C)ccn3)=O)C(C)C2)c(F)c1Cl 72793,C1(C(N2CCN(CCN)CC2)=O)C2CC(O)C(C2)N1C(=O)C(F)CC1CCC1 72794,N1(CCNC(C(c2cccc(Cl)c2)(C)C)=O)CCC(NC(C2CC(F)C2)=O)CC1 72795,N1(C(C2(c3c(C)cccc3)CC2)=O)C2CCCC1CC(NC(=O)C(C)(C)Br)C2 72796,c1(C(N2CC(C(=O)NCC)C2)=O)cnc(CNC(=O)CC2CCC(=O)C2)nc1 72797,N1(C(C(C)C2(O)CCC2)=O)CCN(C2CN(C(=O)COC3CC(F)(F)C3)C2)CC1 72798,c1(C(=O)NC2CC(n3cc(-c4cncc(Cl)c4)nn3)C2)c[nH]nc1[N+](=O)[O-] 72799,C1(CNC(CCC(=C)Cl)=O)CC2(CCN(C(C34CCC(F)(CC3)C4)=O)C2)CO1 72800,c1(OC)ccc(CCNC(N2CC(F)(F)C2C(=O)N(c2ccccn2)C)=O)cc1 72801,C1(C(=O)NCCCCN(C(COCCN(C)C)=O)C)CCCCN1C1CCCC1 72802,c1(C(=O)NC2CCCC(CNC(C(=O)NCC)=O)C2)c(C)cnnc1O 72803,c1(C(N2CC3CC(NC(C4CCC5CC5C4)=O)C3C2)=O)ccc2n[nH]cc2n1 72804,C(=O)(CCCC(C)(C)C)NCC1C(CNC(c2ccc(CNC(C)=O)o2)=O)C1 72805,c1(CNC(=NCC=C)NCC(C)C#N)ccc(S(=O)(=O)N2CCCCC2C)cc1 72806,C1(C(=O)NC(=O)C(c2cccc(F)n2)(F)F)CCC(N2CCCC2)CC1 72807,C12(CNC(C3CC4(CCC4)C3)=O)CCCC1CCN2C(c1cc2c(s1)CCC2)=O 72808,C(=O)(CC(C)(C)C1CC1)NCCCC(C)NC(=O)CC1C=NN(C)C1=O 72809,CC1CCCn2cc(C(N3CCCC4(NC(C5CCCCC5)=O)CC4C3)=O)nc21 72810,c1(C(N2CCC(O)(CCNC(c3c(C)onc3O)=O)C2)=O)ccc(F)cc1O 72811,C1(COCC)CCN(C(=NCC2CCC2)NCC2CCCOC2(C)C)C1 72812,N1(CCCNC(c2cccn(C)c2=O)=O)CCC2(CCCCC2)CC1 72813,C1(NC(C(C)=CC2CC2)=O)CC(C(=O)N(C)Cc2cnccn2)C1(C)C 72814,C#CCCCC(C)C(=O)N1CCC2(CC2NC(=O)C(c2ccccc2F)C)C1 72815,C=C(C)C(C)(O)C(=O)NC1CCC(NC(c2csc(CC(C)C)n2)=O)C1 72816,CCC(C)CCCC(=O)NCCC1CC(C(=O)NCCOCC(N)=O)C1 72817,CS(=O)(=O)c1ccc(C=CC(N2CC3CC(C2)CN(C(=O)CC#N)C3)=O)o1 72818,Cc1ccc(C(N2CCCC(N(C)C(c3cc(N)ccc3C)=O)C2)=O)c(F)c1 72819,N1(C(C2CCC(NC(c3cn(C(C)C)nc3)=O)CC2)=O)C2CCC1COC2 72820,C1(C(=O)Nc2c(C)nco2)C2CN(C(c3coc(C(N)=O)c3)=O)CC12 72821,N1(C(=O)C2=CCCCC2)CCC2CCCC12C(=O)NCC12CCC(CC1O)C2 72822,C1(CNC(=O)CN2CCCS2(=O)=O)C(C2CC2)CCN1C(=O)Cc1ccc(Cl)s1 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72840,CCC(O)CCNC(=O)CC1(CNC(=O)Cc2ccsc2C)CC1 72841,C1(C(N2CCC(F)CC2)=O)CC12CCN(Cc1ccc([N+](=O)[O-])o1)C2 72842,N1(C(C2C(OC)CC2)=O)CCCC2(NC(c3coc(C(C)C)n3)=O)CC2C1 72843,c1(C(N2CCC(C)C2)=O)c(CNC(c2cc(Cl)cs2)=O)cnn1C 72844,c1(SCC(=O)NC23CC(NC(C4CCC(CC)C4)=O)(C2)C3)nnc2ccccn12 72845,c1(C(=O)NC(CC)CN(C)C(c2cc(Cl)n(C)n2)=O)cccc(F)c1C#N 72846,C(C(C)(CC)CC)(c1n(CCCOC)nnn1)NCc1cn2ccsc2n1 72847,C1(C(=O)NC2C(C(N(C(C)C(F)F)C)=O)CCC2)CCCC(=O)N1C 72848,C(=O)(C1=CCCOC1)NC(C(C)(C)C)CNC(=O)CC1OCCO1 72849,C(=O)(C1CCOc2ccccc21)NCC(CNC(c1c(C)[nH]nc1Cl)=O)O 72850,c1(C(=O)Nc2cncnc2Br)cn2c(n1)CN(Cc1c(F)ccc(O)c1F)CC2 72851,c1(C(=O)NCCC2CCCN(C(c3cnc(O)s3)=O)C2)ccc2cccnc2n1 72852,N1(CC(=O)N(C(C)CNC(C2CC23CCOC3)=O)C)CCS(=O)(=O)CC1 72853,N1(C(c2cnc(C)[nH]2)=O)CCN(C(C2CC=CCO2)=O)CC1CS(C)(=O)=O 72854,CCC(CC)C(C)C(=O)NC(CCOCCO)C(=O)Nc1ccc(F)cc1C 72855,CN1CCC(C(=O)NC2CC2NC(=O)C=Cc2cccc(CO)c2)S1(=O)=O 72856,c1(NC(C2CCCN2C(=O)CC2(N3CCCC3)CC2)C)ncncc1Cl 72857,N(C1CC2(CN(C(C3CC(C)N(C)C3)=O)C2)n2ccnc21)C(C(C(=C)C)(C)C)=O 72858,O=C1CCC(NC(=O)CC2CC3(CC3)CN2C(c2ccc(F)s2)=O)C(=O)N1 72859,N#CC1CCCC1NC(=O)CC1CCN1C(C1CCCSC1)=O 72860,C(CCCCC(=O)NCC(C)(C)C(=O)NCCCc1nccs1)N(C)C 72861,C1(NC(c2cccc(O)c2F)=O)CC2CN(Cc3ccccc3)CC2C1 72862,Cc1nc(C(C)(C)C)sc1C(=O)N(CCC(C)NC(=O)CCC(C)N(C)C)C 72863,CN1C(=O)CN(CC(N2CCN(C3CN(C(=O)C4=C(Cl)CCC4)C3)CC2)=O)C1=O 72864,c1(C(=O)NCC(CNC(CNS(NC)(=O)=O)=O)F)ccc(C(F)(F)F)nc1 72865,S(=O)(=O)(c1ccc(C#N)c(N(CC(C)OC)C)c1)N1CC(CC)C2(C1)OCCO2 72866,c1(N)cnc(N)c(Br)n1.c1(SC)ccccc1C(C(C)N)C(C)=O 72867,Cc1c(C(=O)NCC2(NC(C3C(Cl)(Cl)C34CC4)=O)CC2)sc2ccsc12 72868,C(=O)(CCS(=O)(=O)C(F)(F)F)NCC1N(C(c2cc(C(C)=O)sc2)=O)CC=C1 72869,N1(C(C2(CN(C)C)CCCC2)=O)CCCC(CO)(NC(C2CC(CF)C2)=O)C1 72870,C(CC(F)F)(C(=O)N(C)Cc1ccsc1)NC(C1C(C)C1)=O 72871,C1(C(N2C(C)C(C)(C)CC2)=O)C(C2CC2)CCN1C(c1cc(C#N)cn1C)=O 72872,C1(NC(CNC(=O)NC)=O)CCC2(CC1)CN(C(=O)C(C)(CC)CO)CCO2 72873,N1(C(CCC=C)=O)CCC(C(=O)NC2CN(CCC)C2)=C(F)C1 72874,O=C1NCC2(CCN(C(C3CCCN(C(=O)C4CCc5nccn54)C3)=O)C2)N1 72875,C(=O)(C#CC(C)(C)O)NC(C(NC[Si](C)(C)C)=O)C1(O)CCC1 72876,c1(C(=O)NCCCC(C(=O)OC)O)nc2ccccc2nc1O 72877,c1(C(N2C(CNC(C(CCC)C)=O)CC(OC)C2)=O)sc2ccccc2c1C 72878,c1(C(=O)NC(CC)CN(C(=O)C=C(CC)CC)C)ccnc(N2CCCC2)n1 72879,N1(C(c2c(OC)cc(Br)c(S(N)(=O)=O)c2)=O)CCn2cccc2C12CCNCC2 72880,C1(CNC(C(C)OCC#C)=O)CCN(C(c2cc(C)nn2C2CC2)=O)CC1(F)F 72881,C(C(=O)NCCCCC(C)NC(=O)C(C)Cc1cnc[nH]1)(C(C)C)SC 72882,c1(CC)cccc(C)c1C(=O)NCc1ccc(CNC(C2CSC2)=O)cc1F 72883,C=C(CNC(=O)NCCCc1ccc(C)nc1)c1ccccc1F 72884,C(C(C)(O)C(=O)NC(C)C=CC(=O)NCCCn1cc(C)cn1)OC 72885,C1(C(=O)NC(c2ncc[nH]2)C)CCCCCN1C(C1CC2(CCC2=O)C1)=O 72886,C1(C)(C(=O)NC2CCC(NC(CCNC(C)=O)=O)C2)CCNC1=O 72887,C1(CC(=O)N(CC(C)(C)C#N)C)CC(C)(C)CN1C(c1ccc(=O)n(C)n1)=O 72888,N1(C(c2ccc(C(N)=O)[nH]2)=O)CC2CCN(C(=O)C(C3CCOCC3)F)C2C1 72889,C(CCCCCN(C)C(C1CC=C(C)CC1)=O)NC(C(C1CC1)OCC)=O 72890,Cn1ccc2ccc(C(=O)NCC3CN(C(C4(C)CCOC4)=O)CC3(C)C)cc12 72891,N1(C(c2cc(OC)n[nH]2)=O)CCN(C)C(CNC(=O)COCCc2cccs2)C1 72892,N1(C(C(C=C)CC)=O)CC(C(=O)NCc2cc(C)nc(O)c2)CC12CCC2 72893,C(C(C)(CC(C)C)NC(=O)Cn1cc(CO)nn1)NC(c1[nH]nc(OC)c1Cl)=O 72894,c1(CCN(C(=O)NCc2c(OC)nn(C)c2)C)ccc(OC)c(OC)c1Cl 72895,c1(C(N2CCC(CCNC(c3cnc(OC)nc3)=O)C2)=O)ccsc1S(C)(=O)=O 72896,C1(CC)(NC(=O)CCCc2ccncc2)CCN(C(=O)C(O)C2CCCC2)CC1 72897,c1(CNCC2(C)N(CC(c3cccc(C(C)C)c3)C)CCC2)cc(O)ncc1Br 72898,C1(C(=O)NCCC(N)=O)CCN(C(c2ccc(C3CC3)nc2)=O)C12CCC2 72899,C1(NC(c2ccc(Br)cc2)=O)CCC(O)CN(C(c2sccc2F)=O)C1 72900,c1(CC)ccc(OC)cc1.C12CC=CC(C1)CN(CC(O)(COC)CO)C(=O)N2 72901,c1(N2CCN(C(c3cc(OC)c(F)cc3)=O)C(C)C2)cc2ncnn2cn1 72902,c1(CC(=O)NC2C(NC(c3cncc(C)n3)=O)C2)ccc(C)c(F)c1 72903,Cc1cc(Br)ccc1NC(=O)C(C1CCSC1)N(C1CCSC1)C 72904,c1(C(=O)NCC2C(C)CCCN2C(C2CC(O)C2)=O)cnn2c1CCCC2 72905,c1(CC(=O)NC2(CC=C)CCN(C(C3CC3C)=O)C2)c[nH]c2cc(F)ccc12 72906,C12(NC(c3c(N)ccc(Cl)c3)=O)CCCC1CN(C(=O)CCCC1CC1)C2 72907,CC1CC(C#N)(C(=O)NCC2(F)CC(CNC(=O)CCC3CCC(=O)NC3)C2)C1 72908,c1(C(N2CC(CNC(=O)Nc3cccc(C)c3C)C2)=O)cc(F)c(Cl)nc1Cl 72909,O=[N+]([O-])c1cc(NCC2OCC3CCCCC23)cc([N+](=O)[O-])c1 72910,C(=O)(NNC(=O)CCCn1cc(C2CCCO2)nn1)c1c(O)ccc(OC)c1 72911,CS(=O)CCC(O)C(=O)NCC12CC(NC(=O)CCCC3CC3)(C1)C2 72912,c1(C(=O)NC2CC(CC(=O)NCc3cn(C4CC4)nn3)C2)c[nH]c(=S)cn1 72913,c1(C(N(CC(=O)NCC)C(C2C(C(CC(=O)N)C)C2)=O)C)cccc(OC)c1.OC 72914,Cc1cc(C(=O)NCC2CCN(C(=O)C=Cc3ncc[nH]3)C2)nc(C(F)(F)F)n1 72915,C(=O)(C1CCc2ccccc21)NCC(CC(=O)N1CC(C#N)C1)OC 72916,CC1(C)C(NC(C2CN3CCC2C3)=O)CC1C(=O)NC1CCCC1CF 72917,N1(C(CN(CCOC)C)=O)CC2(CCN(C(=O)C(c3cscn3)N(C)C)C2)C1 72918,CCC(CC)C(F)C(=O)N1CCN(C(C2CC2(Cl)Cl)=O)C(C2CC2)C1 72919,C(=O)(CS(=O)(=O)C(C)C)NCC(CCCC)NC(=O)CC1CCCO1 72920,N1(C(c2ccc(C(C)(C)C)s2)C(=O)N(C2CCCOC2)C2CC2)CCC(O)CC1 72921,C(=O)(C(O)C1=CCCCC1)NC(CC=C)CNC(c1cnn(CC(C)C)c1C)=O 72922,C1(OCCCNC(=O)CC2CCCOC2)CCN(C(C2CCC3(CC3)C2)=O)CC1 72923,Cc1[nH]c(C)c(C(=O)NCCC2CCC(NC(=O)CCNS(C)(=O)=O)C2)c1C 72924,N1(C(Cc2c(C)nccc2)=O)CCN(C)CC1CF 72925,c1(OC)ccc(F)c(C(N2C3CN(C(c4ccno4)=O)CC23)=O)c1F 72926,CC1(C)CCN(C(=O)C(CNC=O)CC2CC2)C1c1ccccc1.C(C)(C)(C)O 72927,c1(OC)cc(CCNC(=O)N(C(C)CC(C)C)C)ccc1O.C1C(=O)N1 72928,N1(C(C2CN(C(c3c(C)ccc(F)c3)=O)CC(C)O2)=O)CCC(C)(C2CC2)C1 72929,N1(C(CN(C)CC)=O)CCCC(CNC(=O)CCOc2ccccc2C)C1 72930,C(CN=C(NCC(C)(COC)COC)NC1CCCC1)OC 72931,N1(C(CCOCCOCC)=O)CC(NC(C2CCCN2C=O)=O)C(C)C1 72932,c1(CN2CCC(C(c3cn(CCCCCO)nn3)C)C2)ccc(CC(N)=O)cc1 72933,c1(C(=O)NC(C(C)C)C(N2CCC(N=[N+]=[N-])C2)=O)coc2c1COC2 72934,C1(CC(=O)NCC(C2CCCCC2)NC(CC(=O)OC)=O)CCC(OC)CC1 72935,CCCCC(CC)CC(=O)NCc1c[nH]nc1C(=O)N(CCO)CC 72936,C=CCCCCCCC(=O)NC1CCN(C(c2coc(O)n2)=O)C(C2CC2)C1 72937,c1(C(N2CC(C)C(NC(=O)CC3CCC(F)(F)CC3)C2)=O)onc2ccccc12 72938,C1(NC(C2CCC(C)(C)C2)=O)CC2CCC(C1)N2C(c1cnn(CCO)c1N)=O 72939,CC1CCc2[nH]c(=NC(C)c3cnn(C)c3)[nH]c(=NCCCCC(F)(F)F)c2C1 72940,C(C)(C(=O)NOCC(=O)OC)(C1CCC1)NC(C(C=C)CC)=O 72941,C1(CNC(C2CC(C)(C)C2)=O)CC(O)CN1C(c1ccnc(C2CC2)c1)=O 72942,C1(OCC#C)CCN(C(=O)CCC2CC2C(=O)OC)C1 72943,C(=O)(CS(=O)(=O)N1CCOCC1)NCC(C)N(C)C(c1ccc(C(C)O)cc1)=O 72944,c1(C(=O)OCC(C2CCN(C)C(=O)C2)=O)cnc2ccnn2c1O 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73122,C12(CNC(=O)C(F)n3ccnc3)CCC(CC1)N(C(c1cc(F)cnc1O)=O)C2 73123,C1(C(N2CC(n3cc(CNC(CNC(C)=O)=O)nn3)C2)=O)CCCC(C)(C)CC1 73124,c1(C(=O)NCC2CC(NC(C3(C#N)CC(C)C3)=O)C2)c[nH]c2cccc(Cl)c12 73125,C(=O)(C1=COCCC1)NC1C(C(=O)NCCn2c(C)ncc2)CCOC1 73126,C12(NC(c3cccn4ncnc34)=O)CCCC1N(C(=O)C1=NOCC1)CC2 73127,N1(C(c2ccc(N)cc2F)=O)CC2CCC(C1)N2C(C1CCCC(F)(F)C1)=O 73128,c1(CC(=O)NCCC(C)NC(=O)C(C)(C)n2cnnn2)ccc2nn(C)cc2c1 73129,Cn1cncc1C=CC(=O)NC(C1CCCCC1)CNC(C1COC(=O)O1)=O 73130,N1(c2nc(=NC3C(C(C)C)C3)nc(N3CCOCC3)[nH]2)CCc2[nH][nH]c(=N)c2C1 73131,N1(Cc2cnn(CCC)c2C)CCC2CN(C(=O)C(C)CNC(=O)OC)CCC12 73132,c1(CNC(=O)NCC(N(OC)C)=O)cc(F)ccc1N(C=O)C1CC1 73133,N1(C(=O)NC(c2ccccc2)Cc2cn(C)nc2)CCC(CO)(CO)CC1 73134,N1(C(C(C)(C)OC(C)C)=O)C2CCCC1CN(C(=O)CC(C)(O)C(F)(F)F)C2 73135,C(=O)(C1=NOC2COCC12)NCC(CC(=O)Nc1ccc(C)nc1C)O 73136,C#CC1(C(=O)NCc2ccccc2CC)CN(C(c2cn(C)cn2)=O)C1 73137,c1(CC(N2CCC(CNC(CSC)=O)C2(C)C)=O)ncn2c1CCCC2 73138,C1(C(N2CC(C(C(=O)NCc3cccc(O)c3F)OC)C2)=O)CCOC(C)(C)C1 73139,c1(C(=O)NCC(CN(C(c2c(OC)c(Cl)sc2)=O)C)O)ccc(F)c2[nH]ccc12 73140,CC1CC(N(C(=O)C(=O)NCc2cccc(C(C)(C)C)c2)CCO)CCO1 73141,CCCC(C)(O)C(=O)NC1CCCC(NC(C2CC(F)(F)C2)=O)C1 73142,N1(C(CN(CCOC)C)=O)CCCC(OC)C1.C1(=O)C(CC)OCC2(CC2)CN1 73143,C1(C(N2CC(C3(NC(CCOCCC)=O)CC3)C2)=O)CC2OC(C)(C)OC2C1 73144,c1(CCC(=O)NCCCCN(C)C(c2cnn(C3CC3(F)F)c2)=O)cnc(O)[nH]1 73145,N1(C(C(C)Cn2ccnc2)=O)CC(NC(c2c(Cl)cnn2C(C)C)=O)C(O)C1 73146,c1(OCC(=O)NCC2CCN2C(=O)C(CO)N(C)C)nc(O)nc(O)n1 73147,C1(C)(C(=O)NC2C(NC(Cc3ccn(C)n3)=O)CC2)CCC12CCC2 73148,CC1(CNC(C2CC(NC(=O)CCN=[N+]=[N-])C2)=O)CCCCO1 73149,N1(C(c2ccc(CCC)s2)=O)CCCCCC(Nc2ncc3ncnnc3n2)C1 73150,c1(CC)nc(Cc2cc(C)oc2C)n(-c2c(C)noc2C)n1 73151,C1(O)(CNC(CNC(C(CC)C)=O)=O)CCCN(C(C23CC(CC)(C2)C3)=O)CC1 73152,Cc1cccc(C(=O)NCC(C2CC2)N(C)C(c2cc(Cl)n[nH]2)=O)c1N 73153,c1(CC(N2CCCN(C(C(C)NC(CC)=O)=O)CC2)=O)coc2ccccc12 73154,c1(C(=O)NCC(Cn2cc(COC3CCCOC3)nn2)OC)cc(C)ncn1 73155,c1(C(=O)OCC)cnc(N2CCCC2CN(C(=O)CC2CCCCO2)C)nc1 73156,C(=O)(CCCS(N)(=O)=O)NCCC(C)N(C(Cn1nc(C)n(C)c1=O)=O)C 73157,c1(C(N2CCOCC(F)(CNC(CSCC=C)=O)C2)=O)cccc2c1CNC2=O 73158,N1(C(c2cn(CC=C)nn2)=O)CCCCCC(NC(C2(COC)CCCC2)=O)C1 73159,C1(C(=O)OC)(C(N2CCC(C(C)C(=O)N(C)CCOC3CC3)C2)=O)CCCC1 73160,c1(CC(=O)NC(C2CCN(C(CCCNC(C)=O)=O)C2)C)ccc(Cl)cc1 73161,C1(C(N2CC(CC(C)NC(C3CCCCC3O)=O)C2)=O)C2CC3CC(C2)CC1C3 73162,C1(NC(c2c(CCC)occ2)=O)CC(C)CN(C(c2ccn(CCO)c2C)=O)C1 73163,N1(C(C2C3(CC(OCC)C3)C2)=O)CC2CC(NC(=O)C(=O)C(C)(C)C)C1C2 73164,CC(C)(CC(F)C(=O)NCC1CNC(=O)O1)NC(=O)CCC1CCC(=O)C1 73165,c1(C(=O)NCc2cc(Br)ccc2-n2cccc2)cc2ccc(Cl)nc2s1 73166,c1(OC)ncncc1NC(=O)C(=O)Nc1cnn(C)c1 73167,c1(C(N(C2CCN(C(=O)CC3CCC(C)C3)C2)CC#C)=O)ccc(OC)c(Cl)n1 73168,CCC(CC)(CC)C(=O)NCC1CC1NC(c1ccc(S(N)(=O)=O)s1)=O 73169,c1(OC)ccc(C(=O)Nc2ccc(C(=O)C(F)(F)F)cc2)c(O)c1F 73170,c1(SC)nc(N2CCOCC2CNC(c2cc([N+](=O)[O-])cs2)=O)ncc1Br 73171,c1(C(C)C)sc(Cl)nc1C(N1CC(N(C(=O)CCC2CCOCC2)C)C1)=O 73172,C(CNC(=O)CC1CC2(CC2)CO1)(CC(=O)N(C)C(C1CCCC1)C)OC 73173,C1(C)(C(=O)NCC(C)(CNC(=O)C(C)=C(C)C)OC)CCC(C)C1 73174,CC(CC(F)(F)F)C(=O)N1CC(CC(=O)NC2(C(O)CO)CC2)CC1(C)C 73175,c1(C(=O)NC2C(NC(c3ccn(C)c(=O)c3)=O)CCCC2)c[nH]nc1S(N)(=O)=O 73176,N1(C(CN(C(C(CC)OCC)=O)CCOC)=O)CCCC(CC2CC2)C1 73177,c1(C(=O)NC(C)CCCCNC(c2ccon2)=O)c(Cl)oc2ccccc12 73178,c1(OC)ncnc(C(=O)NCC2CCCCC2NC(=O)Cn2cnnc2O)c1F 73179,C(=O)(C(CO)C(C)(C)C)NCC1(C)OCCN(C(c2cnc(C(C)(C)C)[nH]2)=O)C1 73180,N1(C(C(CSC)C)=O)CCC2(CC1)CN(C(=O)Cc1nn(C)cc1Cl)CCO2 73181,N#CCCCCCC(=O)NCCC1CN(C(=O)Cn2ccccc2=O)CCCO1 73182,c1(C(=O)NC2CN(C(c3ccc(C)cn3)=O)C(C)C2)cc(C(F)(F)F)ccc1O 73183,CC1CCCC(N)(C(=O)NC2CCC(C(=O)O)C2)C1 73184,c1(C(N2C(CNC(CC3CC(OC)C3)=O)CCC2)=O)ccc(N)c(F)c1Br 73185,c1(OC(C(N2CC(NC(C(C=CC)O)=O)C2)=O)C)cc(Cl)cc(Cl)c1 73186,Cc1cccc(C(C)C(=O)NC2CCC2NC(c2cnn(-c3nccs3)c2)=O)c1 73187,C(=O)(CCC(C)(C)[N+](=O)[O-])N(C)Cc1nn(C)cc1Br 73188,c1(NC(C2CC(O)(CNC(c3cscc3C3CC3)=O)C2)=O)ccc(CCO)cc1 73189,N1(C(=O)C(C2CCCCC2)O)CCN(C(c2ccn3cccc3c2)=O)C2(CC2)C1 73190,C#CC(C1CCc2ccccc21)Nc1nccc(SC)n1 73191,c1(C(=O)NC(CCCNC(COCCOCC#C)=O)C)ncnc2cc[nH]c12 73192,C1(CNC(C=C(C)C(C)C)=O)CCCCN1C(C1CN(C(=O)OC(C)(C)C)C1)=O 73193,C(=O)(C1CCCc2scnc21)NC1C(CNC(c2c[nH]c(=NCC)s2)=O)CCC1 73194,CC1COCCN(C(=O)C(C(C)(C)C)NC(=O)C2=CCCC2)C1 73195,CCCC(C)CCCC(=O)NCC1(F)CCC(NC(=O)CC2(O)CCCC2)C1 73196,C(=O)(C(C#N)(CC)CC)NCC1CCC(CN(C(C(CC)OC)=O)C)CC1 73197,c1(C(N2CCN(C(c3c(C)nn[nH]3)=O)CC2C#N)=O)cc2cc[nH]c2cc1F 73198,C1(N(C)C(c2coc(C(F)F)n2)=O)CCCC(NC(C2CC(C)(C)C2)=O)C1 73199,C1(CNC(=O)CCCc2cnccn2)C(F)(F)C12CC2 73200,c1(NC(CC=C)C)[nH]c(=NCc2cnc[nH]2)nc2c1cnn2C 73201,O=S(=O)(c1nccs1)NCC1(F)CCN(Cc2ccc(I)c(F)c2)CC1 73202,C1(N(C(c2cc(SC)cs2)C(=O)NCCCSC)C)CCC2(CC2)C1 73203,C(CC(CNC(c1cc(C)co1)=O)NC(=O)C=CC1CCCO1)OC 73204,CCCCC(C)(F)C(=O)NC1CCCCC1NC(c1ccc(F)cc1)=O 73205,C1(C(=O)Nc2ccc(C(C)C)cc2)CN(C)CCN1C(=O)C(F)C(F)(F)F 73206,C(=O)(C1=CC2(CCOC2)C1)NC(C(=O)N(C(C#C)C1CCC1)C)CC1CC1 73207,c1(C(N(C)CC2CCCN(C(=O)CCC3CCC3)C2)=O)n[nH]cc1[N+](=O)[O-] 73208,C(=O)(C1=CS(=O)CCC1)NCC12CC(NC(CC(=O)N(C)C)=O)(C1)C2 73209,CCC(C)C(C(=O)NCC(C)(C)CCOC)NC(c1ccccc1NC)=O 73210,c1(C(C)NCc2ccc(OCCO)cn2)cccc2c1CCC2 73211,N1(C(C(C)N(C(C)=O)C)=O)CCC(C2CCN(C(C3(F)CCCC3)=O)CC2)CC1 73212,N1(C(C(C)(C)SC)=O)CCCN(C(=O)Cc2ncc(Cl)s2)C(C)C1 73213,CCC(C(=O)NCC1(F)CCN(C(c2cc(OC)n[nH]2)=O)CC1)C(C)O 73214,CC(C)(C)CCCN=c1ccc(S(=O)(=O)NCCCCC2CCCC2)c[nH]1 73215,c1(C(=O)NCCN(C(C(C)NC(CC)=O)=O)CC)c(C)nc2cc(O)nn2c1C 73216,CCC(C(=O)N(CC(C)(C)CNC(=O)C(Cc1ccsc1)NC=O)C)C(C)C 73217,c1(OC)cc(C(=O)NCC2CCCCN2C(=O)CC(C)(C)C)cc(Cl)c1O 73218,C(=O)(CS(=O)(=O)C1CC1)NCC1N(C(C2CNC(=O)N2)=O)CC(F)C1 73219,c1(C(=O)NC2C=CCN(C(c3n[nH]c(C)c3N)=O)C2)cnn2c1CCCC2 73220,C(C)(Cc1ccccc1)(CC(C)C)NC(C(C=C)CC)=O 73221,C(=O)(CC(C)(C)CC(F)F)N1CCN(C(c2sc(C)c(O)n2)=O)CC(CO)C1 73222,c1(OC)ccc(O)c(CNC2CCN(C(c3ccc(OC(C)C)cn3)=O)C2)c1 73223,N1(CCc2cn(CC(=O)N(CC(N)=O)CC)nn2)CCN(C(C)C)CC1 73224,C(=O)(C(C)CS(C)(=O)=O)NC1CCCCN(C(CSCc2ccc(C)cc2)=O)C1 73225,N1(C(CN(C)CC)=O)CCC(NC(=O)CS(=O)(=O)N2CCOCC2)CC1C1CC1 73226,C1(NCc2c(C)c(C(F)(F)F)n[nH]2)CC2(CCC2)C12CCC2 73227,S(=O)(=O)(c1ccc(N2CCC3(CC=CCO3)C2)nc1)NC(c1cccc(Br)n1)C 73228,N1(C(CCC2(NC(c3cncc(O)c3)=O)CCC2)=O)CC2C(CO)C2C1 73229,C1(NC(=O)Cc2ccccc2CO)CN(C(=O)C=CC2CCCCC2)CC1(F)F 73230,c1(C(N(CC(C)NC(c2cnc(C3CC3)s2)=O)CC)=O)ccc2ncn(C)c2n1 73231,C12(C(N3CCN(C(C)C)CC3)=O)CCN(C(=O)CNC(N)=O)CCC1C2 73232,c1(OC=O)n[nH]cc1-c1ccncc1.C(C(=O)NCCC1(N)CC1)OCCOCC 73233,c1(C(=O)NC(CN(C(CN(C2CC2)CC)=O)C)C)cnn(C)c1S(C)(=O)=O 73234,c1(OC)ccc(NC(C2CC(F)(F)CN2Cc2scnc2C)=O)c(Cl)n1 73235,C(=O)(C(O)C(C)C)NC(CC)(C)CNC(=O)C(C)(C)c1ccccc1 73236,N1(S(CC)(=O)=O)CCCC(C(=O)N(CC(O)COC)CC)C1 73237,Cn1ncc(C(c2nnnn2CCC2CC2)NCC2(CSC)CCCC2)c1Br 73238,c1(C(CNC(C23CC(C)C2C3)=O)NC(=O)Cc2cn(C)nn2)cccc(Cl)c1 73239,CC(CC(C)(C)O)C(=O)NCCNC(c1ccc(-n2cncn2)c(F)c1)=O 73240,c12ccc(cc1Br)S(=O)(=O)N2CCNc1nnnn1C1CCC1.CC=C=CCC 73241,c1(C(=O)OC)cc(NC(=O)C(F)(F)C(O)C2CC2)n2ccccc12 73242,CCC(C(O)C(C)C)NC(c1ccc(NC(=O)N(C2CC2)CC)cc1)=O 73243,CCCCCCCCCCCCNC(c1ccc(OCC(=O)O)cc1)=O 73244,C1(NC(C2(CC)CC2)=O)CN(C(c2cccc(OC)n2)=O)CC2CCCC12 73245,N1(C(c2ccc(NC(C)=O)s2)=O)CCC(C)(C)C1CNC(C1CC(=O)N(C)C1)=O 73246,c1(CN(C)Cc2cc3ccccc3s2)cc2ccnc(Cl)c2o1.C12CCCN1C2 73247,C12(C(=O)NCC3C(NC(CNS(NC)(=O)=O)=O)CC3)CCC(=O)N1CCS2 73248,c1(C(C)C)c[nH]cc1C(=O)NCC(C(N1CCCC1)=O)C1CC1 73249,C(=O)(C(C)CC(F)(F)F)N1CC(C(=O)NCCc2noc(CC)c2C)(CC)C1 73250,CC1(C)CCCC(O)(CNC(=O)Nc2ccc3ccoc3c2)C1 73251,CC1CCN(CC(=O)N(CCCNC(C2(C)CC2c2ccccc2)=O)C)CC1 73252,C1(CCC(=O)NC(C)C(C)NC(=O)CN(C)C(=O)OC(C)(C)C)CCCOC1 73253,N1(C(C(C)CC(F)F)=O)CCC2C(CCCN2C(C2(O)CCCCC2)=O)C1 73254,c1(CNC(NC(COC)C)=NCC2CN(C)CCO2)nc2c(s1)CCC2 73255,N1(C(C2CCC(CC)O2)=O)CC2CCC2(CC(=O)NCCc2ccc(C)cn2)C1 73256,c1(C(CCC)C)cn(CC(=O)OC)nn1 73257,CCS(=O)c1ccccc1C(=O)NCCOC1CCN(C(=O)CSC(F)F)CC1 73258,C1(NC(C(c2cc(C)oc2C)C)=O)CC2CN(C(=O)CCc3cn[nH]c3)CC2C1 73259,C(CCCC(=O)NC12CC(C(=O)NC3CCC(C#N)C3)(C1)C2)OC 73260,C1(C(N2CC(NC(C3(C)CCCC3)=O)C2)=O)CCC(N=[N+]=[N-])C1 73261,CN1C(=O)Cc2c(C(=O)NCC3C4CN(C(=O)Cn5cnnn5)CC34)cccc21 73262,c1(N2CC(NC(c3c(C)cn(C)c3)=O)C(C)(C)C2)c(F)cccc1[N+](=O)[O-] 73263,C(=O)(C(C)CCC(C)(C)C)NCC1(F)CCN(C(C(C)NC(CC)=O)=O)C1 73264,C1(CC=C)CCCCN1C(c1cn(CC)nn1)C(=O)NC(C)(C)CC 73265,C1(CN2CC(NC(C(C)(C)C3CC3)=O)C(c3cncn3C)C2)CCCNC(=O)C1 73266,C1(N(C(C2CCN(CC(C)C)C2)=O)C)CN(C(=O)CCc2ccco2)CC12CC2 73267,C1(C(=O)NC2CCCC(O)C2)CN(C(c2ccnn2C2CC2)=O)CC1(F)F 73268,N1(C(C2(N(C)C)CC2)=O)CCC(CC2(N)CCC2)C1 73269,c1(C(=O)NCC2C(NC(c3c(C(C)C)c[nH]n3)=O)CC2)ccc(N(C)C)cc1 73270,N(C1CCCc2c[nH]nc21)C(c1nccc(CNC(=O)Cc2cc[nH]n2)c1)=O 73271,c1(-c2nc(-c3scc(C)n3)nn2C2CCCCCC2)cc(S(N)(=O)=O)c(C)cc1C 73272,N1(C(C(CC)CC)=O)CCC(C2(CNC(=O)C3CC3)CCOCC2)CC1 73273,N12CCc3sccc3C1CNC(=O)C(F)(F)C(C1CC1)C2=O.N1(C2CC2)CCCC1 73274,C1(C(N2CCC(C(F)(F)F)(OC)C2)=O)CCN(C)CC1C(F)(F)F 73275,CC(C)CCC(CO)NC(C1CC(N(C)C(c2coc(CO)c2)=O)C1)=O 73276,N1(C(Cc2c(C)nsc2)=O)CCC(C)C(CNC(C2(C(C)C)CC2)=O)C1 73277,C1(NC(CCN2C(C)(CC(C)C)CCC2)=O)CCC(F)(F)CC1 73278,C(=O)(C(C(C)(C)C)c1cc[nH]n1)N(CCN(C(=O)CCOCC1CC1)C)C 73279,c1(NC(C)C(C)(C)F)cccc(C(F)F)n1 73280,CC(C(O)C(=O)N1CC(F)(CNC(=O)C(F)=C2CCC2)C1)c1ccccc1F 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73543,N1(C(C(C)n2ccnc2)=O)CCCC(C)(C)C1CNC(C1CC1C1CC1C)=O 73544,C(=O)(CN=S(C)(=O)c1ccc(Cl)cc1)NC1(C)CCCC1C(=O)OC(C)(C)C 73545,c1(OC)ccc(OC)c(S(=O)(=O)NCC(=O)Nc2ccc(OC)cc2)c1OC 73546,Cc1cc(CCN2CCN(CC(C)O)CC2)cc(O)n1 73547,C(CCCC(C)NC(C1CCOCC1)=O)NC(c1nc(C(=O)OCC)sc1)=O 73548,c1(C(=O)NC(COc2c(OC)cccc2)C)c(Br)ccc2c1CCC2 73549,N1(C(Cc2c(C(C)C)cccc2)=O)CC2COCC2C1 73550,C1(C(N2CC(CC(C)NC(=O)CCSCC(N)=O)C2)=O)(OC)CCOCC1 73551,c1(C(C)(C)C)ccc(C=CC(=O)NCCN(C(c2ccccc2)=O)C2CC2)cc1 73552,N1(C(C2NCCN(C(C(c3ccc(OC)cc3)C)=O)C2)=O)CCc2n[nH]cc2C1 73553,C(=O)(C1=CS(=O)(=O)CCC1)NCC(C)(CNC(C1(O)CC2CCC1C2)=O)OC 73554,N1(C(c2c(C)coc2)=O)CCN(C(=O)C(F)(F)Oc2ccccc2)C(C)C1 73555,c1(C(=O)NCC2C(NC(CCn3ccc(C)n3)=O)COC2)ccn2nncc2c1 73556,Cc1nc(-c2c[nH]cc2C(=O)NCCN(C)C(c2sccc2CC#N)=O)cs1 73557,N1(C(CC(C)OC)=O)CCC(C)C1C(=O)NCCc1ccc(C)nc1 73558,C1(N(C(CCSCCNC(CC(C)SC)=O)=O)C)CCC(CO)CC1 73559,CC1CC(NC(=O)Cc2nncn2C)CN1C(=O)COc1ccc(F)cc1 73560,C(c1c(C)coc1C)=CC(C1(C2N(C(Cc3cnc(C)o3)=O)CCCC2)CC1)=O 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73631,C1(O)(CNC(C2CC2CF)=O)CCN(C(=O)CCC=CBr)CC1 73632,Cc1cc(C(N2CC3C(CNC(C4(C)CCN(C)C4=O)=O)C3C2)=O)cc(C)c1 73633,C1(OC)CN(c2cc[nH]c(=N)n2)CC1NC(=O)NCCCl 73634,CC(=O)CCCC(C)C(=O)NC1(C(N2CCC(CF)C2)=O)CC(F)(F)C1 73635,C1(C(N(C2CCN(C(C3(C)CC=CC3)=O)C2)CC)=O)COCC1(C)C 73636,c1(C(=O)NC2C3CCC2N(C(c2occc2F)=O)C3)cc2ccc(F)cc2o1 73637,Cc1cc(C(N2CC(C(C)NC(=O)CC3(C)CC3(F)Cl)C2)=O)on1 73638,N1(C(C(c2ncc(C)s2)C)=O)CC(O)CC1CC1CCNCC1 73639,c1(C(N2C(CN(C(CNC(=O)OC)=O)C)CCC2)=O)cc(Cl)cc(F)c1F 73640,c1(C(=O)NCC2CCN(C(C(CC=C)CC)=O)C23CC3)cc2ccccc2cn1 73641,C1(CC(=O)NCCc2ccns2)CN(C(=O)C=Cc2cc[nH]n2)CC12CC2 73642,C1(C(=O)NCCN(C(=O)CN(C)CCO)CCOC)CCCSC1 73643,c1(C(N(CC(CNC(c2c(C(C)C)occ2)=O)C)C)=O)cnc2[nH]ncc2c1 73644,N1(C(C2C(=C)C2)=O)CCN(C(=O)CCc2ccc(Cl)cc2)CC1CF 73645,c1(CC)cc(N2CC3C(CNC(=O)C(C)Cn4ccnc4)C3C2)ncn1 73646,c1(CC(C(=O)NCCC2(O)CN(C(C3(OC)CC3)=O)C2)O)cc(Cl)sc1Cl 73647,C1(C(=O)NCCCN(C(c2cccc(C)c2O)=O)CC)CC12CCC(F)(F)CC2 73648,O=C1CC(C(=O)OC(C(=O)NCc2cccc(Br)c2)C(F)(F)F)C2(CCC2)C1 73649,c1(C(=O)NC2C=CCN(C(C3C(C)CC(=O)NC3)=O)C2)cc2ccc(Cl)cc2[nH]1 73650,C(=O)(C(F)CC(C)C)N(C1CCCN(C(c2n(CC)ccc2)=O)C1)C 73651,C1(C(=O)NCC(=O)N(CC)CC)CCC(CNC(=O)Cn2cc(C#N)cn2)CC1 73652,C1(C)(CC)CCN(C(C2(CO)CCN(C(=O)C(CO)NC(=O)OC)C2)=O)CC1 73653,C(=O)(CCCCCCCC)N1CC(CNC(C(CC#C)(C)CC)=O)C(O)C1 73654,c1(CNC(C2(CCNC(=O)CNC(=O)CCn3cccn3)CC2)=O)cccs1 73655,C12(C(=O)NCC3N(C(COCC)=O)CCC3)CCOC1CCOC2 73656,N1(C(C(F)=CC)=O)CCOC2(CCN(C(c3cscn3)=O)C2)C1 73657,C1(NC(c2cncnc2C2CC2)=O)CC12CCN(C(C1CCC3CC13)=O)CC2 73658,C1(C(=O)OC)CCCN(CCO)C1C.c1(S)cc(F)cnc1Oc1ccccc1Br 73659,N#CC1(C(=O)NCCCNC(=O)CC2CCC23CCC3)CCOC1 73660,c1(OC)c(C(=O)NC2CC(CNC(=O)C(C)n3ccnc3)C2)csc1C 73661,CN1CC(O)CC1(C)C(=O)NCC1(CCNC(C2CNC(=O)C2)=O)CC1 73662,C#CC1(O)CCN(C(=O)CC2N(C(c3ccsn3)=O)CCC2(C)C)C1 73663,C1(OC)CC(F)CN(C(c2cnn(C3CCOCC3)c2)C(=O)NC(C)(C)C)C1 73664,CCCCC(CNC(=O)C(CC(F)F)N(C(=O)CN1CC2CC2C1)C)CCC 73665,N1(C(c2c(C)noc2C)=O)CC(C)(C)OC2(C1)CN(C(=O)CCc1cnn[nH]1)C2 73666,N1(C(C2C(CC)OCC2)=O)CCN(C(=O)C=Cc2cccc(F)c2Cl)C2CCC12 73667,CCC(C)C(C)N=c1[nH]c(=NCC2(c3cnccn3)CCC2)[nH]c2c1COCC2 73668,C=CCC(CC(=O)N1CC=CC1CN(C)C)NC(=O)CC(C)(C)O 73669,C(=O)(CS(=O)(=O)CCOC)N1CC(CC(=O)NC2C(OCC)CCC2)OCC1 73670,N1(C(C2C(C(C)=O)C2(C)C)=O)CCC(N(C(=O)C(=O)NC2CC2)C)C(C)C1 73671,c1(C(=O)NCCSCC(=O)NC(C(C)(C)OC)C)c[nH]c(=S)cn1 73672,c1(CC)nc2ccccc2c(C(=O)NC2CN(C(=O)C(C)(C)C)C2)c1C 73673,C1(C(N(C(CSCCCC)C)C)=O)C=CCN(C(C2(C(N)=O)CC2)=O)C1 73674,N1(C(C(CC(=C)C)NC(=O)Cc2ccon2)=O)CCN2C(=O)OCC2C1 73675,c1(CCCC(=O)NCC2CCN2Cc2ccccc2Br)ccccc1Cl 73676,c1(OC)ccc(Cl)nc1C(N1CCC(CN(C)C(C2OCCC2C(C)C)=O)C1)=O 73677,C=C1CC2(C1)CC(C(=O)NC(C1CCCN(C(c3cc(N)cc(F)c3)=O)C1)C)C2 73678,C1(NC(c2ccc(C)cc2)=O)CCCC12CN(C(C1(C)CSC1)=O)C2 73679,c1(C(=O)NC(C2CCCC2)CNC(C2CC(OC)C2)=O)sc(SC)cc1C 73680,c1(C(=O)NC(C)CCNC(=O)CCC2CCCO2)ccccc1CO 73681,c1(CC(=O)NCC(C)(CO)NC(C(=Cc2cccnc2)C)=O)c(C)ncnc1O 73682,Cc1cnc(Cl)c(S(=O)(=O)Nc2ccc(C(=O)Nc3nccc(Br)c3O)nc2)c1 73683,c1(C(N2C(C(=O)NCc3nnc(C)n3C)CC3CC32)=O)cc(F)c(F)cc1F 73684,Cc1ccc(C(O)C(N2CCC(CCC(=O)N(CCC(C)C)CC(C)C)C2)=O)cc1 73685,c1(C(=O)NCC2(C)CCN(C(=O)CC3COC(=O)N3)C2)ccc2nc(O)sc2c1 73686,c1(NC(c2cncc(NC(c3c(C)cccc3)=O)c2)=O)ccc([N+](=O)[O-])c(Cl)c1Cl 73687,C1(CC(C)NC(C2CC(OC)(OC)C2)=O)CCN(C(=O)CC2CC=CCC2)CC1 73688,N1(C(C(C=C)(C)CC)=O)CCN(C(=O)C(CCC)N(C)C)CC(C)(F)C1 73689,N1(C(c2c(OCC)scc2)=O)CCC(NCC(=C)Cl)C(C)C1 73690,Cc1[nH]cnc1C(=O)NCc1ncoc1C1CN(C(C2CC(CF)C2)=O)C1 73691,CCCCC(CNC(c1cncc(OC)n1)=O)NC(=O)C(CC)n1cc(Br)cn1 73692,C1(NC(C(C=CCCC)O)=O)CCN(C(c2ccncc2)=O)C12CCC2 73693,n1(C)cc(CC(=O)NC2(C(=O)N)CC2)cn1.C1(C(C)C2CC2)CCN(C(N)=O)C1 73694,CCCCCC(C)(C)C(=O)ON1CCOCC(O)(C(F)(F)F)C1 73695,Cc1cc(C#N)ccc1S(=O)(=O)N(C)C(C1(S(C)(=O)=O)CC1)C 73696,N1(C(C2(C#N)CC=CC2)=O)CC2CCN(C(=O)CC3CC3c3ccccc3)C2C1 73697,C(=O)(CC(C)CC(C)(C)C)N1CC(NC(Cc2cc(OC)c(O)c(OC)c2)=O)C1 73698,c1(C(N2C3C(C(N(C4(CCO)CC4)C)=O)C(C3)C2)=O)cc(O)nc(O)n1 73699,N1(C(C(=O)NCCCOC)c2cccs2)CCC(C)C(O)C1 73700,C=CC(C)CCN=c1nc(-c2ccccc2)[nH]c(=NCc2ccc(Br)s2)[nH]1 73701,c1(C(=O)NC2C(NC(c3cc[nH]n3)=O)CCC2)ccnc2ccncc12 73702,N1(c2ccc(S(=O)(=O)NCC3OCCN(C)C3)s2)CCN2C(=O)CCC2C1 73703,C12(CSC)CC(C(=O)NCC(C(C)C)NC(=O)C=Cc3cncs3)(CO1)C2 73704,FC(F)(F)C1c2ccccc2OCCN1S(=O)(=O)CC1CC2(CCOCC2)CN1 73705,c1(NCCNC(C)=O)ccc(S(=O)(=O)Nc2nc(Br)co2)cc1Cl 73706,CC(C)(CCC(=O)N1C2CCC1CC(C(=O)NCc1cnccn1)C2)[N+](=O)[O-] 73707,CC(C)C(C#N)C(=O)NCCCC(=O)NCCC1CCC(C)O1 73708,C(=O)(C1Cc2ccc(F)cc21)NCC(CNC(C1(CCOC)CCCC1)=O)(C)O 73709,C1(O)(CNC(CCc2ccnc(C)n2)=O)CCN(C(=O)C2=CCCCO2)CC1 73710,C(CC(C)C)(C(=O)N1CC(C)CCC1CO)NC(C(C)NC(C)=O)=O 73711,C1(CNC(Cc2cc(C)no2)=O)CN(C(C2CCCC(=O)CC2)=O)CCCO1 73712,c1(C(=O)NC2CCCC(OCC)CC2)ncc2cc(Cl)ccn12 73713,CON(CCC(=O)NCc1cc(F)ccc1F)C(=O)C(O)c1cncn1C 73714,Cc1nnccc1C(=O)NC1CCCCC1CNC(=O)CC1CC2CCC1C2 73715,C(=O)(C(C)(C)C(C)C)NCCCC1OCCN(C(c2c(C)[nH][nH]c2=N)=O)C1 73716,N1(C(C)(C)C)CC2CC1CN(Cc1coc(-c3ccc(Cl)c(Cl)c3)n1)C2 73717,N1(C(CCC)=O)CCC(NC(c2ccnc(N3CCCC3)c2)=O)C(F)C1 73718,N1(Cc2ccc(COCC)o2)CC2CN(C(c3ccccc3I)=O)CC2C1 73719,c1(C(=O)NC(c2n(C)ncc2)C(=O)NCCn2ccnc2)ncnc(O)c1F 73720,CCCCCCC(C)C(=O)NC1CC(C(F)F)(NC(=O)CCCN=[N+]=[N-])C1 73721,c1(-c2c(CN3CCN(c4cn(C)nc4)CC3)csc2)cnn2c(Br)c[nH]c12 73722,C1(NC(=O)Cn2nccn2)CC2CC(NC(=O)CNC(=O)Cc3ccsc3)C1C2 73723,N1(C(C(COC)C)=O)CCC(NC(=O)Cc2csc(-c3ccco3)n2)C1C(C)C 73724,N1(CCNC(C(C)OCC2CCCO2)=O)CCN(C(=O)CC=C(Cl)Cl)CC1 73725,N1(C(c2c(OC)scc2)=O)CC2(CCN(C(=O)C(F)C(C)C)CC2)CC1C 73726,c1(C(=O)NC(CSC)CO)coc2cc(O)ccc12 73727,c1(CSC)noc(CCC(=O)NC2CC2CNC(=O)CC2CCCCO2)n1 73728,N1(C(CNC(CC)=O)=O)CCC(C(=O)Nc2ns[nH]c2=O)CC1 73729,C(C(C(=O)NCCc1cn[nH]c1)C(C)(C)C)NC(CC(C)n1cccn1)=O 73730,CS(=O)(=O)c1ccc(C(O)CNC(=O)NCc2c(O)cccc2Cl)cc1 73731,CC12CCC(CNC(N3CCCOC(CCO)C3)=O)(CO1)C2 73732,c1(C(C)C)cnn(C)c1C(N1CCCC1CC(=O)NCCc1ccncc1F)=O 73733,c1(CNC(C(C)(C)OCC)=O)ccc(CNC(=O)CCC2CCC(=O)NC2)cc1 73734,C=CCC(C)C(=O)N1CCC(N(C(c2ccc(N(CCCC)C)s2)=O)CC)CC1 73735,c1(CC(=O)N(CCCNC(=O)Cc2ccsn2)CCC)nnc(C)o1 73736,C1(NC(COCCN(C)C)=O)CCCC(NC(=O)C2=COCCO2)CC1 73737,C1(C(=O)NC(C)(CN2CCCC2)CO)CCCC2(CC(NC(=O)OC(C)(C)C)C2)C1 73738,c1(OC)cccc(C(CNC(=O)C(Cl)=CCl)NC(=O)Cc2c[nH]nc2O)c1 73739,c1(CC(N2CC(CC)N(Cc3ccc(=O)n(C)n3)CC2)=O)ccc(C)c(F)c1F 73740,N1(C(=O)OC(C)(C)C)CCC(C2CCC(CNC(=O)NOc3n[nH]c(=N)s3)O2)CC1 73741,c1(C(=O)NCC(C)(CC(C)C)NC(CCOCCC)=O)ccn2ccnc2n1 73742,c1(OC)cc(C(N2CC3CC(C2)N3C(C)=O)=O)cc(SC)c1.c12nccc-1n2 73743,c1(C(N(CC(CC)NC(CC(=O)OCC)=O)C)=O)cc(SC)cc(Cl)c1 73744,c1(CN2CC(C(=O)Nc3ccc(Cl)c(Br)c3)C(O)CC2)ccc2c[nH]nc2c1 73745,N=c1[nH]c2c(s1)CCCC2C(=O)N1CCCC1C(=O)NCC1(CO)CCOCC1 73746,C#CCCCCCC(=O)N(CCCCC(=O)N(C)Cc1ncnn1C)C 73747,CC1(C)COC(C(=O)NCCC2CN(C(=O)COC3CCCCCC3)C2)C1 73748,c1(N(CC(=O)NCC(O)CNC(=O)COCCc2nccs2)C(C)C)ccccc1 73749,c1(OC)cnc(C(=O)N(CCC(=O)NCc2sccc2C)C)cn1 73750,C1(CC(=O)NCC23CCN(CC2)C3)C2CCCC2N1C(=O)Cc1cn[nH]c1 73751,Cc1cc(Cl)ccc1NC(C1CC(CCNC(c2ccsc2C(F)F)=O)C1)=O 73752,C1(C(N2CC(n3nnnc3C(C)C)C2)=O)(CC)CCN(Cc2noc(C)n2)C1 73753,C1(CNC(=O)C(=CC2CCCCC2)F)C2CC1N(C(C1C(F)(F)C13CC3)=O)C2 73754,c1(CC(N2CCC(CCNC(C(C=C)OC)=O)CC2)=O)ccc(C#N)cc1 73755,N1(C(C=CC)=O)CCN(C(c2cnc(-c3ccccc3)c(F)c2)=O)CC1COC 73756,C(=O)(C(C)=NOCC#N)N1C(C(=O)NCCC(=O)OCC)CC1C 73757,C(Cc1ccc(OC)nc1)(N=c1cnc(OC)c[nH]1)c1ccc(CC)cc1 73758,N1(CNc2cc(C=O)no2)CCCOC(CNC(c2cc(COC)[nH]n2)=O)C1.OC 73759,N#Cc1cc(Cl)c(C(=O)NC2CCN(C(C3CN(C4CCC4)C3)=O)CC2)s1 73760,CC1(C(=O)NCc2ccnc(OC3CCCCC3)c2)CC12CCN(CCCO)CC2 73761,C1(CCC)CC1N=c1[nH]c(N(C)CC2(N(C)C)CCCC2)nc2c1COC2 73762,c1(NC(C2N(c3ncc(C(=O)OCC)cn3)C3C(C2)C3)=O)ccnc(Cl)c1C 73763,N1(C(C(C)n2ccnn2)=O)CCC2(CC1)CC(C(=O)Nc1nn[nH]n1)CO2 73764,N1(C(COCCC(C)C)=O)CCS(=O)(=O)C(CCNC(C2CC3(CC3)CO2)=O)C1 73765,c1(C(N(CC(C)NC(=O)C(c2ccnn2C)C)CC)=O)cc(Cl)c(Br)[nH]1 73766,CC(O)CCCN=c1ccc(S(=O)(=O)NCc2nc(-c3ccccc3)no2)c[nH]1 73767,N1(C(c2ncn(C(C)C)n2)=O)CCC2C(C(=O)NC3CN(C(N)=O)C3)C2C1 73768,N1(C(CC2CC(=O)NCC2)=O)CCC2C(C1)CN2C(=O)CCc1ccoc1 73769,c1(C(=O)NCC2CN(C(C(CO)N(C)C)=O)CC2(C)C)csc2c1CCCC2 73770,c1(C(N2CC(CC(=O)NC(C#C)C3CCC3)OCC2)=O)cnn2c1OCC2 73771,c1(CC(C(=O)N(C)Cc2nc[nH]n2)NC(C(C)CC2CC2)=O)cnn(C)c1O 73772,C1(NC(CCCCNC(C(CC)(C)O)=O)=O)CCCC(C)CC1 73773,C(c1ccccc1C#N)=CC(=O)NC(C1(CNC(C2CCC(=C)CC2)=O)CC1)C 73774,n1(-c2cc(C)on2)c(C)cc(C(N2CC=CC2CNC(c2cnsc2)=O)=O)c1C 73775,CC(C)CC(CNC(=O)CC1(O)CCCCC1)NC(=O)CCc1cn[nH]c1 73776,C1(NC(=O)C#CC2CC2)CCN(C(C2CCC([N+](=O)[O-])CC2)=O)C12CCCC2 73777,c1(C(N(CCNC(C(C)(C)SC)=O)C)=O)ccc2c3c(cccc13)CC2 73778,C1(NC(=O)CSc2cccc(F)c2)CN(C(C2CCC3(CC3)C2)=O)CC2CC12 73779,c1(C(=O)NCC(CNC(c2cc([N+](=O)[O-])c[nH]2)=O)OC)cc2ccc(C)cn2c1 73780,C12(C(N3CC4(C(C(N5C(C)CCC5C)=O)C4)C3)=O)CCC(CC1)CC2 73781,N1(C(CCCOC(C)=O)=O)CCCC1(C)CNC(C1CC1(c1ccccc1)C)=O 73782,C1(C(N2CCC(C)(NC(c3ccc(CO)nc3)=O)C2)=O)(OCC)CCOCC1 73783,C1(NC(c2cc(OC)ncn2)=O)CCN(C(c2cnc(Cl)s2)=O)CCC1CO 73784,N12CCC(N=[N+]=[N-])(C1)C(=O)NCC(C)(O)C2=O.C(C)(C(=O)OC)OCCCC 73785,c1(C(=O)NCC(C(C)(C)C)NC(=O)CCc2ccco2)nnn2c1CCCC2 73786,C(=O)(CCCCCN(C)C)NCCCCNC(C(C)NC(c1ccco1)=O)=O 73787,c1(OCC)nc(C)ccc1C(=O)NC(C1CCOC1)CNC(=O)CCC(C)C 73788,c1(C(=O)NC2CCC(CNC(C3CC(Cl)(Cl)C3)=O)C2)ccc(-n2cccn2)cc1 73789,C1(CNC(CCc2n(C)ncc2)=O)CCN(C(C2C3CCCOC23)=O)CC1 73790,c1(C(N2C(CNC(c3ccoc3Br)=O)CC(OC)C2)=O)ccc(N)cc1O 73791,C1(C)(CNC(C(c2n(C)ccc2)=O)=O)CCCN(C(c2cnncc2O)=O)C1 73792,N1(C(C(C)OCC2CC2)=O)CCC(CNC(c2ccc(Cl)o2)=O)CC1C 73793,C1(CC(=O)NCCCN2C(C)CCC2)CC(F)CN1C(=O)CCCN(C)C 73794,N1(C(c2c(C(C)(C)C)n[nH]c2)=O)CC(NC(c2ccc(Cl)o2)=O)C2CC2C1 73795,N1(CC)CC(C(N2CCOC(CNC(C3CC4CC(=O)C3C4)=O)C2)=O)CCC1=O 73796,c1(NC2C3(CC(NC(CC4(C(=C)F)CCC4)=O)C3)C2)nc2ccc(Br)cc2s1 73797,c1(C(=O)NC(CC)CNC(=O)CSC(C)C)cc([N+](=O)[O-])cc2c1OCCO2 73798,C(=O)(CC(=O)NCCN(C(=O)CNC(c1ccccc1)=O)CC)NCC#C 73799,N1(C(CC2C(C)(C)OCC2)=O)C2CCC(C(=O)NCC3CC(CF)C3)C1CC2 73800,N1(C(c2c(CC)nn(C)c2)=O)CC(O)CC1(C)C(=O)NCC1CCSCC1 73801,C=CCC(C)(C)CC(=O)N1CCCCCC1C(=O)NC1(CO)CC(F)C1 73802,N1(C(CC(C=C)(C)O)=O)CCC(F)(F)C(CNC(=O)CC(C)(C)OC)C1 73803,C1(C2CCC(=O)NC2)(C(=O)NC2C(C)CN(C(=O)C(F)(F)C(C)(C)O)C2)CCC1 73804,N1(C(CCC(=O)N(C)C)=O)CC(NC(c2cnc(=N)[nH]c2)=O)CC12CCCCC2 73805,Cc1cc(C#N)nc(=NC(C)CCNc2ccc(C(F)(F)F)cc2[N+](=O)[O-])[nH]1 73806,N1(C(CNC(c2ccc(F)c(F)c2)=O)=O)CC2CC(C(N3CCOCC3)=O)C(C2)C1 73807,c1(NC(C(c2ccco2)NC(C(C)OCCCC)=O)=O)cccc2c1CCC2 73808,C1(NC(c2cncc(OC)c2)=O)CC2CN(C(c3cc(F)ccc3Cl)=O)CC2C1 73809,N1(C(Cc2c(C)cnn2C)=O)CCC(N(C(=O)Cc2ccc(Cl)cn2)C)C(C)C1 73810,c1(CNC(CS(=O)(=O)NCC)=O)n[nH]c2c1CN(C(c1cnccn1)=O)CC2 73811,c1(C(N2C(C(C)NC(C3(C(F)F)CCCC3)=O)CCC2)=O)cccc(=S)n1O 73812,S(=O)(=O)(c1cccnc1N(C)CCSC)NC1CCN(CC)C1 73813,C1(CCC)CCN1.C1C(=O)O1.C(=O)(COCCCOCC)OCC=C 73814,N1(c2nc(NCC=C)c3c(n2)n(C)nc3)CCc2oc3ccccc3c2C1 73815,C(=O)(CCCc1ccccc1)N(C(C)CNC(C1CC(O)(C(F)F)C1)=O)CC 73816,C(CCC)(C(=O)N1CCC(NC(C23CC(C#N)(C2)C3)=O)C1)=CCC 73817,C(=O)(C(C)(C)C(=O)NC1CC1CNC(=O)CNC(c1ccccn1)=O)NC 73818,N1(C(C(C(C)C)NC(C)C)=O)CCN(Cc2sccc2Cl)CC1C#N 73819,N1(C(C(=O)NCCCOC)c2cocn2)CCc2nn(C)c(=O)cc2C1 73820,CCCC(C)CCCNC(C1CCCCC1)C#N 73821,CN=c1nc(N2Cc3cnn(CCO)c3C2)[nH]c(=NCCC2CC2(Cl)Cl)[nH]1 73822,Cc1ncc(C(=O)N(CC(C)(C)CNC(=O)CC2CCCC2O)C)cc1N 73823,C=C(Br)CCC(=O)NC1CCN(C(c2cc(C(N)=O)ccn2)=O)C1 73824,C12(NC(c3nc(C(=O)OC)sc3)=O)CCC(CNC(=O)CCC(C)SC)(C1)OC2 73825,c1(C(C(=O)NCCC(C)CCNC(c2ccncc2Cl)=O)O)cc(Cl)cc(Cl)c1 73826,C1(C2(O)CCOC2)(C(=O)NCCC(C)NC(=O)CCN2CCCC2=O)CC1 73827,C(C(C)(O)C(=O)NCC1(C)CCCN1C(C1CCC(C)C1)=O)OC 73828,c1(C(C(=O)NC2C(NC(CCCC)=O)CC2)(C)C)c[nH]c2ccccc12 73829,C1(NC(C(C#C)(C)C)=O)CC2CCC(C1C)N2c1ccnc(-c2nccs2)n1 73830,N(S(=O)(=O)NC(C)C)(CC)CC1OCCC1c1cnn(C)c1 73831,N1(C(C(C)NC(C)=O)=O)CC(NC(c2cnc(C3CCOCC3)nc2)=O)C(F)C1 73832,c1(NC(C2CCC(C(=O)Nc3c(C(=O)OCC)c[nH]c3)C2)=O)cc(C)cnc1Cl 73833,C1(C)(CN(C)C)CCCN(C(=O)C=CC(F)(F)F)C1.c12ccccc1CNC2=O 73834,N1(C(C(CO)OC)=O)CC(NC(=O)CCCC2CCC2)CC12CCCCC2 73835,N1(CC)CCOC(C(=O)NC2CN(C(=O)CSc3c(C)n[nH]c3C)CC2OC)C1 73836,C1(CNC(c2cnc(C)[nH]2)=O)C2CN(C(=O)Cc3ccnc(Br)c3)CC12 73837,Cc1ccc(C(F)(F)F)cc1C(N1CCCC(CNC(=O)C2=CCSC2)CC1)=O 73838,C(CCCS(=O)(=O)CCO)NC1CCN(C(N2CCc3sccc3C2)=O)C12CC2 73839,C1(NC(C(C(C)(C)C)SC)=O)CN(C(=O)CC2(O)CCCC2)CC(C)(C)C1 73840,C1(C(=O)NC2CN(C(c3ccc(C(C)C)cc3)=O)C(C)C2)CC2(CCCO2)C1 73841,Cc1ncc(N)cc1C(=O)N(C)CC1CCN(C(=O)C(C)c2ccsc2)C1 73842,C(=O)(C1COCc2ccccc21)N1CCCC(N(C(CCCC#CC)=O)CC)C1 73843,c1(OC)cccc(CCC(=O)NCC(C)NC(=O)CCc2cccc(Cl)c2)c1F 73844,N1(C(c2c(SC)cn(C)n2)=O)CC(CNC(=O)C=C(Cl)Cl)C(C)(C)C1 73845,C12(CC(=O)Nc3c(C)ccnc3)CCC1CN(C(c1cc(F)n(C)n1)=O)C2 73846,c1(NC(C)=O)cccc(C(=O)N(CC(C)NC(=O)Cc2csnn2)C)c1 73847,C1(C(N(C2CC3CC3C2)C)=O)CC2(CC(NC(c3c(F)cncc3F)=O)C2)C1 73848,Cc1ccn2c(C(N3CCC(C(=O)O)CC3)=O)nnc2c1C 73849,c1(C(=O)NCC(c2cccs2)O)n[nH]c2c1CN(C(=O)Cc1cccc(F)c1)C2 73850,C1(NC(c2ccc(COC)cc2)=O)C(C)CN(C(=O)CCCC2CCC2)CC1C 73851,C1(OCC)(CNC(=O)Cc2cccnc2)CCN(C(=O)CC2CCCOC2)C1 73852,C1(CNC(CN(C(=O)Cn2[nH]cnc2=N)CC#C)=O)CCCC(C)(C)O1 73853,c1(C(=O)NCCCC(C)(C)NC(c2ccc[nH]2)=O)cc(Br)cc([N+](=O)[O-])c1 73854,c1(CC(N2CCC(O)(CNC(C(Br)=C(C)C)=O)C2)=O)ccc(F)c(Cl)c1 73855,C(=O)(C1=CCCCCC1)NCC(CNC(C(C(C)C)NS(C)(=O)=O)=O)F 73856,O=C(CCCC(F)(F)F)NC1CN(C(C2(F)CC(NC(=O)NC3CC3)C2)=O)C1 73857,c1(C(N2CC(O)(CCNC(CC(C=C)C)=O)C2)=O)nc(C)ncc1Br 73858,N1(C(C2(F)CC2)=O)CCc2cc(C(=O)NCc3cncc(Br)c3)ccc2C1 73859,c1(C(=O)NCCCOCCNC(=O)CCCC2CCCO2)ccc(O)cn1 73860,Cc1c(C(=O)NCC=CC(N2CCCC3CC23)=O)cnn1C 73861,c1(CC)c(C(=O)NCCOC)nnn1CC.C12CCCN1N1CCC2C1.C(=O)COC 73862,Cc1noc(-c2cn(CC(=O)Nc3ccnn3Cc3ccccc3)cn2)n1 73863,N1(C(C(CC=C)(C)C)=O)CCN(C(=O)Cc2nnc3n2CCCC3)CC(C)(F)C1 73864,Fc1cccc(Cl)c1CC(CNC1CCCC1F)Cc1ccccc1 73865,CC(CN(C)C)C(=O)NCCCN(C(=O)CC(O)c1ccccc1)C 73866,C1(C(N2CC(CNC(c3c(C(C)(C)C)ocn3)=O)C3C2C3)=O)CCC(C)(C)CC1 73867,c1(C(N2C3(CNC(c4cccc(F)c4F)=O)CC(C2)C3)=O)nccn2ccnc12 73868,c1(C(CC(=O)O)NCC(=O)NCC)ccccc1F 73869,c1(CNc2c(C(N3C4CCC3CC4)=O)scc2)cnc2c(Br)cc(Cl)cn12 73870,C(C(C)C(C)C(=O)N(CCNC(=O)C=CC(N1CCOCC1)=O)CC1CC1)OC 73871,N1(C(C(=O)NCC(=C)C)CC2CC(F)(F)C2)CCOC(C)(CC)C1 73872,c1(NS(CC)(=O)=O)cnc2c(c1)CN(C(C1(C(=O)OC)CC1)=O)CC2 73873,C1(C(N(C(C)CC(=O)N(C)CC2CCCC3CC23)C)=O)CC2(CCO1)CC2 73874,C1(NC(=O)NCC(CC)(C)O)CC(F)CN(C(=O)OC(C)(C)C)C1 73875,N1(C(C(COC)n2cc(CCN(C)S(N)(=O)=O)nn2)=O)CCN(C(C)=O)C(C)C1 73876,c1(OC)ccc(C(c2nnnn2C)NCCN(C)C(C)C)cc1C#N 73877,C1(NC(=O)C=CCC2CC2)CCCCC1NC(C1CCOCC1)=O 73878,CC1COc2ccccc2C1C(=O)NC1CC(NC(=O)COc2cnn(C)c2)C1 73879,C1(NC(C(COC)(F)F)=O)CC2CCC1N(C(=O)Cn1ccc(O)nc1=O)C2 73880,c1(CN(C2CCOC2C)CCCOC)ccc(SC)s1 73881,Cc1c(F)ccc(Cl)c1C(N1CCN(C(=O)C=Cc2ccco2)C(C2CC2)C1)=O 73882,C(=O)(CS(=O)(=O)C(C)(C)C)NCCCC(C)(C)NC(c1n(CCC)ncc1)=O 73883,Cc1ncc([N+](=O)[O-])cc1NC(C1C=CCN1C(=O)Nc1cccc(C)c1C)=O 73884,C1(CC)CCC(NC(c2cc(Br)c(Br)o2)c2nnnn2C2CC2)CC1 73885,C1(NC(C2(OCC)CCC2)=O)COC2(CCN(C(=O)C3=C(CC)OCCS3)C2)C1 73886,c1(OCCCN(C(C(=O)NCCCSC)Cc2ccco2)C)cccc(Cl)c1 73887,c1(C(N2CCC(NCCC)C2)C(=O)NCCSC)cccc(Cl)n1 73888,CCC(CC(=O)NC(CNC(C1(C)CCC1)=O)CCOC)C(C)C 73889,CCCCC(CC(=O)NC1C=C(C)CCC1)NC(=O)Cc1cc[nH]n1 73890,C#Cc1cc(C(=O)NCC(O)CNC(=O)C(C)(CCC)OC)cc(N)c1 73891,Cc1cc(C(N2CCCCC23CC3)C(=O)NC2CCCC2)cnc1C 73892,c1(OC)cncc(C(=O)N(C(C)(C(=O)NCC(c2ccncc2)C)C2CC2)C)n1 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73997,C1(C(N(C2CC2)CC)=O)CCCCC1NC(c1cc(C)nn1-c1ccncc1)=O 73998,C1(C(=O)N(CCCCNC(c2ccc(Cl)cc2)=O)C)(CC)CCCCO1 73999,N1(C(C2C(C)OC(C)C2)=O)CC2(C1)C(NC(c1cccs1)=O)CCS2(=O)=O 74000,C#CC1(N(C)C)CN(C(C2CC=CCN2C(=O)CC2COCC(C)O2)=O)C1 74001,N#CC1(C(=O)NCC2CC(NC(c3ccc(CO)nc3)=O)C2)CCOC1 74002,c1(C(=O)NCC2CC(NC(C(C)C(F)(F)F)=O)C2)csc2c(O)ccnc12 74003,CC1Cc2cc(CC3CCN(C(=O)C(N4CCNC(=O)CC4)=O)CC3)ccc2O1 74004,Cc1[nH]nc(C(N2CC(O)CC2C(=O)NC(CO)C2(C)CC2)=O)c1O 74005,CON1CCC(CC(=O)NCC(CNC(c2c[nH]ccc2=O)=O)CO)CC1 74006,CC1(C)CCCCC1C(=O)NCC(=C1CN(C(=O)CCCO)C1)F 74007,c1(C(N(CCNC(C(C(C)C)F)=O)C2CC2)=O)c(F)ccc2nc[nH]c12 74008,CC1CCN(C(C2CC(CCNC(c3ccc(O)nc3)=O)C2)=O)C(C)C1 74009,C1(O)(COCC)CN(C(C2(NC(=O)CCc3nc(O)n[nH]3)CC2C)=O)C1 74010,CCC(C)(C)C(C)CC(=O)NC1CCC(NC(=O)C=CCOC2CCOCC2)C1 74011,CCC(CC(=O)NC1CN(C(=O)C2=C(Cl)CC2)CCC1CO)C(C)(C)C 74012,CC1CN(C(C23CC(NC(=O)CC4CCCOC4)(C2)C3)=O)Cc2nncn21 74013,n1(CCCCNC(c2ccc(C#C)o2)=O)c(C)cc(C(=O)O)c1C 74014,c1(C(N(C)CC2CC(NC(=O)CC3(C)CC3)C2)=O)ccc(F)c(F)c1 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74033,c1(SCC)cccc2nonc12.c12cncnc1-c1ccccc1CN(C)C2=O 74034,C1(CC(=O)NC2C(NC(Cc3cn(C)nc3C(F)(F)F)=O)C2)CCCS(=O)(=O)C1 74035,c1(SCC)cnccc1C(=O)NCCC1CN(C(=O)C(O)C2CC2)CCO1 74036,C1(C(=O)NCC23CCC(CC2)C3)CC(O)CCN1C(C1CC12CCOCC2)=O 74037,CCCCCC(C(=O)NCC1c2ccccc2CN1C(c1cnns1)=O)C(C)C 74038,CCC(CC(F)F)C(=O)N1CCN(C(=O)C=Cc2ccc(SC)cc2)C(CO)C1 74039,c1(C(=O)NC2CCCN(C(CC3(C=C)CC3)=O)C2)cnc(N)c(CO)c1 74040,N1(CCNC(c2c(C)cccn2)=O)CCCN(C(C2(C)CCOCC2)=O)CC1 74041,Cc1nc(C(=O)NC(CNC(c2ccc(F)s2)=O)C(C)C)c(C)n1C1CC1 74042,C(C(F)(F)CC(O)CO)NC(N(C)Cc1cccc(Cl)c1Br)=O 74043,c1(C(=O)NCCN(C(=O)C(C)(F)C(F)(F)F)C)cc2ccc(Cl)cc2s1 74044,CC1(C)CN(c2nc(=N)nc(N3CCC(c4ccccn4)C3)[nH]2)CCS1(=O)=O 74045,n1(CC)ccc(C(=O)NCC2CCCN2C(=O)Cc2ncc(F)cc2F)cc1=O 74046,n1(CC(N2CC3C(NC(c4ccc(CC(C)C)s4)=O)(C3)C2)=O)cnc([N+](=O)[O-])c1 74047,N1(C(CC=CCC)=O)CCN(C(c2cnc(C)nc2CC)=O)CC1CC(F)F 74048,c1(OC)ccc(C2(C(=O)NCC3CCCN3C(=O)Cc3cc(C)no3)CC2)cn1 74049,Cc1cc(C)n2ncc(C(=O)NCC3CN(C)CCN3C(=O)C3CC3)c2n1 74050,c1(C(C(=O)NC2COC2)N(CC(C)SC)C)c(Cl)nc2sccn12 74051,CS(=O)C=CC(=O)N1CCN(C2CN(C(C3C(F)(F)C34CC4)=O)C2)CC1 74052,C1(C(=O)NCC2CC(NC(=O)CC3(O)CCOC3)C2)CN2CCCN1CC2 74053,c1(C(=O)NC(CC)C)n[nH]cc1CNC(=O)CN(C)C1CC1 74054,c1(C(=O)NCC2N(C(C34CCC(OC)(CC3)C4)=O)CCC2)c(F)ccc(N)c1F 74055,N1(C(CCc2ccc(OC)cc2)=O)CCN(C(c2ccc(F)o2)=O)CC(CO)C1 74056,c1(OC)ccc2cc(C(=O)NCCCNC(=O)C(C)N(C)C(C)=O)ccc2c1 74057,C(=O)(CC(C)(C)COC)N(CC(CC)NC(C1CC1c1cccc(O)c1)=O)C 74058,Cc1ccc(-c2cn(-c3ccc(C(=O)N(C)CC4CCO4)cc3)nn2)c(F)c1 74059,c1(N2CCN(C(c3c(C)ccnc3C)=O)CC2C(C)C)ncnc2n[nH]cc12 74060,CC1CC2CC(C(N3CCCN(C(C4CCCC(=O)O4)=O)CC3)=O)(C2)O1 74061,N1(C(C(C)NC(C)=O)=O)CCOC2(C1)CN(C(C1CC1C(=O)OC(C)(C)C)=O)C2 74062,C1(CNC(Cc2ccc(C)o2)=O)CN(C(c2cc(CO)[nH]n2)=O)C2(CCC2)C1 74063,C1(C(=O)NCC(C(C)C)NC(c2ccncc2F)=O)CCC2(CCOCC2)O1 74064,CC(C)C(C)C(CNC(=O)C(F)n1cccn1)Nc1ncc(O)cn1 74065,Cc1c(C(=O)NCC2CC3CCC(C2)C3)c[nH]c1C#N 74066,C1(C(=O)NCC2C(NC(c3c(CC)c(C)sc3)=O)C2)COc2ccc(Cl)cc2O1 74067,CN1CCCN(C(=O)CC(C(F)F)NC(C2(C)CCN(C)C2)=O)CC1=O 74068,N1(C(c2c(C)cn(C)n2)=O)CCN(C(=O)CCCc2ccc(Cl)cc2)CCC1C 74069,c1(N2CC3(CCN(C(CC(=O)N(C)C)=O)C3)C2)nc(Cl)nc2[nH]cnc12 74070,c1(NC(C2N(Cc3cccc(C(N)=O)c3)CCOC2)=O)ccc2ncsc2c1Br 74071,C(Cn1ccnn1)(C(=O)NOCCCOC)NC(C(CC)O)=O 74072,C1(NC(=O)CCn2cc(-c3ccc(C(=O)O)o3)nn2)CNC(=O)OC1 74073,C1(OC)CN(C)C(C)(C(=O)NCC2(Cc3cn(COC4CCC4)nn3)CC2)C1 74074,Cc1ccc(F)cc1CC(N1CC=CC(NC(c2ocnc2C(F)F)=O)C1)=O 74075,Cc1ccc(C=CC(N2CC(F)CC2CNC(C2(C3CC3)CCCO2)=O)=O)o1 74076,C1(NC(c2n(CCCC)nnn2)c2ccncc2)CNC(=O)OC1 74077,c1(CC)nc2ccc(Br)cn2c1C(N1CCC(C(C)NC(=O)C(C)C)C1)=O 74078,c1(CC)cc(C(=O)NCC2CN(C(=O)C(C)n3cccc3)CC2C)cn(C)c1=O 74079,n1(CC(=O)NC2CCC(NC(c3ncn(CC)c3)=O)C2)cnc2sccc2c1=O 74080,C1(CNC(=O)CC2CC3(CC3)CO2)CCN(C(c2cnccn2)=O)C12CC2 74081,CC(=O)C(C)CC(C)C(=O)N1CCCCC(C(=O)NC2CC3(C2)CC32CCC2)C1 74082,c1(NC(C)=O)ccc(C(=O)NCC2CCN2C(C2CCCCC2F)=O)cc1 74083,C1(C(N2CCC(C(=O)NC)C2C)=O)C2CCC(C2)N1C(c1cc[nH]c1C1CC1)=O 74084,c1(C(N2C3CC(NC(C4(CC#C)CCC4)=O)C2CC3)=O)c[nH]c2ccc(Cl)cc12 74085,C1(C(C)C(=O)NC(C)Cc2ccnn2C)CCN(C(C2(F)CCOC2)=O)CC1 74086,Cc1nc(C(C)C)[nH]c(=NC2CC(NC(=O)C(C(C)C)c3cccnc3)C2)c1Br 74087,C1(NC(C(=O)NCC(C(=O)OC)C)=O)CC2(CCCC2)C1 74088,c1(CC(CNC(CCC)CO)O)cccc(F)c1 74089,C1(N(C(C(OCC)OCC)=O)CCN(C)C)CCN(C(=O)CCCCC)CC1 74090,N(C)(C(=NCC(O)c1ccccc1Br)NCc1ccnn1C)CCCC 74091,N1(C(C=CSC)=O)C2CCC1CC(N(C)C(c1ccc(C3CCC3)cc1)=O)C2 74092,c1(CC)nc(C(=O)N(C)CC2CCCN2C(=O)C=C(C)C(C)(C)C)cs1 74093,C1(C)(CN(C)NC(COCC)=O)CCC(NC(=O)CCc2cccc(OC)n2)C1 74094,C1(C)(C(=O)NC(C2(O)CN(C(=O)CC3=CCCCC3)C2)C)CCOC12CC2(F)F 74095,N1(C(c2c(NC)scn2)=O)CCC(O)(CC(=O)NC(C)CN(C)C)CC1 74096,c1(NC(N2C(c3c(C(=O)OC)[nH]nn3)CCC2)=O)cc(C(F)(F)F)c(Cl)cn1 74097,Cn1ccc2c(C(N3CC4CCC4(NC(=O)CCC(=O)N(C)C)C3)=O)ccnc12 74098,NC(=O)CCC(=O)NC1CCCC(CNC(=O)Cc2coc(-c3cccs3)n2)C1 74099,N1(C(c2nc(C)n(C(F)F)c2)=O)CCC(C)(NC(=O)C(C)C(F)(F)F)CC1 74100,C1(=CC(=O)N(CC(C)NC(=O)C2=CC(O)CCC2)C)CCCCCC1(F)F 74101,c1(C(N2CC(C(C=O)OC)C2)=O)nnc(S)n1C.N1CC(F)(CF)C1 74102,CC(CC(C)(F)F)C(=O)N1CC(F)(F)CC1CCNC(=O)C(C)(C)c1cccs1 74103,C1(C(=O)Nc2cn(CCCC#N)nn2)(C(C)C)CCN(CC2C(CC(C)C)C2)C1 74104,C#Cc1cnncc1C(=O)NCC1(C)CCN(C(=O)C(C(C)C)SCC)CC1 74105,N1(C(C=Cc2n(CC)ccn2)=O)CCN(C(=O)CC2CCC(O)C2)CC2(CC2)C1 74106,C1(NC(CCc2c(OC)cc(Cl)cc2)=O)CC(C)(C)C12CCC2 74107,C(=O)(C(O)CC(C)(C)C)N(C(C(=O)NC1(CCCC)CC1)C)C 74108,Nc1ccc(C(N2CC3CC3(C(=O)NCC3NC(=O)NC3=O)C2)=O)nc1 74109,S(=O)(=O)(c1ccc(=NCCF)[nH]c1)NC1C(C(C)C)CCCC1 74110,CC(C(=O)OCCNC1CCN(Cc2ccc(Cl)cc2)C1)C(C)(F)F 74111,C1(CNC(c2c(C)csc2)=O)(NC(=O)Cc2ccc(Cl)c(Cl)c2)CCCCC1C 74112,CCCC(C)(C)CC(=O)N1CCOC(C(=O)NC(C)(CO)CCC)CC1 74113,c1(C(N(CC(CC)NC(c2ccn(C)c2)=O)C)=O)coc(C)c1 74114,c1(C(N2C(CC)CN(C(=O)C(C)(C)C(=O)NC)CC2)=O)cc(C)c(C)cc1C 74115,c1(CC)cccc(OCC(N2CC(O)(CCNC(=O)C=CC(C)CC)C2)=O)c1 74116,N1(C(C2C(CNC(=O)COc3cccnc3)OCC2)=O)CC2CCC2C1 74117,C(=O)(C1=CCCSC1)NCCN(CC(C)O)C(C1CC1c1c(F)cccc1F)=O 74118,c1(CC(=O)NCC2(O)CN(C(C(CC)OCC)=O)C2)c[nH]c2cccc(Cl)c12 74119,N1(C(C(CC)(C)O)=O)CC2CCC2(CNC(=O)Cc2ccnnc2O)C1 74120,CC1CN(C(C2(C(F)F)CC2)=O)CC(C)N1Cc1cn(-c2ccccc2Cl)nn1 74121,C1(C)(C(=O)NC(C2CCCN(C(c3ncc(OC)cn3)=O)C2)C)CCN(C)CC1 74122,C1(CC(=O)NC)CN(C(c2ccc(C)nc2)=O)CCN1C(=O)C#CC1CCC1 74123,c1(C(=O)NCC(=O)N(C2CN(C(C(CCC)O)=O)C2)C)cccc(C#N)c1 74124,C(C(CC(=O)NCC1(C#N)CC1)C1CCC1)NC(c1c(C)[nH]cc1)=O 74125,c1(NC(C2CN(S(c3ccc(C)nc3)(=O)=O)C2)=O)c(C)cc([N+](=O)[O-])cc1Br 74126,C(=O)(CS(=O)(=O)N(c1ccccc1O)CC)OC1COCC1n1cc(CN)nn1 74127,C1(C(=O)NC(C)CCNC(C2(C)CCC2)=O)C2CC1N(C(=O)OC(C)(C)C)C2 74128,c1(C(N2C(CNC(c3cn(CC)nc3)=O)CCC2)=O)cc(N)cc2c1OCCO2 74129,C1(NC(C2OCCN(C)C2)=O)(CNC(=O)CSc2cccs2)CCC(C)(C)CC1 74130,N1(C(CCc2cc(C)no2)=O)CC2CC(N(C)C(c3ncn(C(C)C)n3)=O)C1C2 74131,C(N=c1[nH]cnc2c1CCC2)C1C(C)CCCN1C(=O)CCC1(C)CC1 74132,c1(C(N2C(COC)(CNC(=O)CC3CC3(C)C)CCC2)=O)ncn2cccnc12 74133,C1(CNC(COc2c(C)cccc2)=O)N(C(=O)C(CO)NC(N)=O)CCC1(C)C 74134,N1(C(CC(C)(C)C2CC2)=O)CC2CCC(C(=O)NCC3COC(=O)N3)(C2)C1 74135,C1(NC(C)=O)CCC(CC(=O)NCC(C2CCN(C(=O)C(C)(Cl)Cl)CC2)C)CC1 74136,C(=O)(C)NCCCNC(C)(C)C1(C(=O)OC)CC1 74137,C(=O)(C1=NNC(=O)CC1)N(CC(C)(C)NC(c1ccns1)=O)C 74138,C1(C(N2CC3(N(C(C(CC)n4ccnc4)=O)CC3)C2)=O)CCCCC(F)(F)C1 74139,N1(C(C2(CNC(=O)CC3(O)CCCC3)CC2)=O)CC2CC2C2CC12 74140,C(=O)(C(C)(C)CS(N)(=O)=O)N1CC(CCO)(NC(C=Cc2c(C)cncc2)=O)C1 74141,C1(NC(C2C(F)(F)C23CC3)=O)CN(C(=O)CC2CCCC2)CC1CC1CC1 74142,c1(C(=O)NC2C(C)CN(C(=O)C#CC3CC3)C2)ccc2ccoc2c1 74143,CCCCC(C(=O)NCC(C(C)(C)C)OC)NC(c1cc(C)c(C)[nH]1)=O 74144,c1(N(C)C)cc(N2CCC(NCc3conc3C(C)(C)C)C2C2CC2)ncn1 74145,Cc1nc(C(N2CC(CNC(=O)C(=Cc3c[nH]cn3)F)C2)=O)nn1C 74146,C1(CC(=O)NC(CCC=C)C)CC(C)N(C(=O)CC2CCCCC2)C1 74147,N1(C(COc2ccc(CC)cc2)=O)CC(NC(=O)CC2CCOCC2)CC(C)C1 74148,N1(C(C(C)(C)C#N)=O)CC2(CCC(CNC(C3CCC4CC34)=O)O2)C1 74149,C(CC(C)(O)CNC(C1(CNC(=O)COCc2nc[nH]n2)CCCO1)=O)OC 74150,CC1CCCn2c(C(N3CCC34CN(C(=O)COC3(C)CCC3)C4)=O)cnc21 74151,C(CCC(C)C)(C(=O)NCCC(C)(C)C)NC(c1c(C)cccn1)=O 74152,c1(CCC(=O)NCC(C(C)C)NC(c2c[nH]c(=N)o2)=O)cc(F)cc(F)c1 74153,Cc1nc(N(C(C)C(F)(F)F)c2ccccc2)ccc1C(F)(F)F 74154,n1(C(CC)CC)nc(-c2cccc(N)n2)nc1C1CC1OC(C)(C)C 74155,c1(C(N2C(C)(COC)CC(NC(=O)CC(C)C)C2)=O)[nH]c2cc(C)ccc2c1C 74156,N1(CCC=CCC)CCC(F)(F)C(CNC(=O)CC(C)CC)C1 74157,c1(NC(=O)NC(c2ccc(OC)cn2)C)nc2c(s1)CCc1ccccc1-2 74158,C1(C(N2CC(C(C(=O)NCC3(CO)CC(C)C3)O)C2)=O)CN(C)CCO1 74159,c1(C(=O)NC2CCCN(C(c3nc(C(C)C)sc3)=O)CC2)cc([N+](=O)[O-])nn1C 74160,c1(C(=O)NCCC2(O)CN(C(c3ccon3)=O)C2)cc(Br)ccc1Cl 74161,c1(C(=O)NC(CC)(CNC(C23CCCC2C3)=O)CC)cn2nc(OC)ccc2n1 74162,CCCCC(CC(=O)NCC1(CO)CCCC1)N.C1(=O)CC2(CC2)CNC1=O 74163,S(=O)(=O)(c1ncn(-c2ccccc2)n1)N(CC)Cc1ccoc1 74164,C1(C(=O)OC)CCC2CCN(C(=O)C(=O)NC(CC(F)F)=O)C12 74165,CCC(C)(C)NC(C)C(=O)NC1CC(NC(=O)CC2(C)CC2)C1 74166,N1(C(CCCOCC=C)=O)CCCC(O)(CCNC(=O)CCC(C)(F)F)C1 74167,c1(C(N(CC(CC)NC(=O)CCCC2CC2)CC)=O)cccc2ccc(C)nc12 74168,N1(C(c2cc(C(=O)OC)cn2C)C(=O)NCc2cccs2)CC2(C1)CC2(F)F 74169,C1(C)(CNC(CNC(C)=O)=O)CN(Cc2ccc(Cl)cc2Cl)CCO1 74170,Cc1ccc(F)c(CC(=O)NC2CCN(C(=O)C(C)CC(N)=O)CC2O)c1 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74453,c1(C(=O)NCC(C(C)C)NC(C2CC(N(C)C)C2)=O)ccc2c(c1)N(C)C(=O)C2 74454,c1(C2(C(=O)NCC3(C(C)(C)OC)CC3)CCCCC2)ccc2c(c1)OCCO2 74455,C1(C(=O)NC2CN(C(=O)Cc3cscn3)C3CC23)CN2CCCN1CC2 74456,c1(CC(=O)N(CCNCC)NC(=O)C(C2CC2)C2CC2)cccc([N+](=O)[O-])c1 74457,c1(CC)cccc(OC(C)C=O)c1.c1(C(=O)NCC2NCC2)ccc(OC)nc1 74458,N1(C(C(CC=C)C)=O)CC2CC(N3CCC(CC)CC3)C1C2 74459,C12(CC(=O)NC3CC(N(C(C(C)N(C)C)=O)C)C3)CC3CC(C1)CC(F)(C3)C2 74460,c1(C(N2C(C(N(CCCO)CC)=O)CSCC2)=O)ccc(O)c(C)c1 74461,c1(OC)ccccc1CNC(=O)C(C1CCC(C)(C)C1)N(CC(F)F)C 74462,C1(OC)CC2CCC1CC2C(N1CCN(C(c2cccc3nccn23)=O)CC1)=O 74463,C(=O)(C(C)(O)CC(C)C)NC(c1c(C)cccc1Br)C(=O)NCC=CC1CC1 74464,C1(C(=O)NC(C(C)NC(C(c2ccc(F)cc2)CC)=O)(C)C)CC2(C1)CC(O)C2 74465,N1(C(C2CCCN(C(c3c(C)nc(C)o3)=O)C2)=O)CC(CO)OC(C)C1 74466,C1(C(=O)NCC2CC(SC)C2)CC12CCN(C(C1(CCCF)CC1)=O)C2 74467,C1(CNC(C2CCC(C)C2)=O)CN(C(C2CCS(=O)(=O)C2)=O)CCN1C 74468,N1(C(C2CC(CC)C2)=O)CC2(CNC(=O)Cc3cc(Cl)cs3)CC1CO2 74469,C1(c2cn(CCNC3CCC(CCC(C)C=O)CC3)nn2)CC12CCOCC2 74470,c1(C(=O)NC2CN(C(CCC3CC(OC)C3)=O)C(C)CC2)c(F)ccc(Cl)c1N 74471,c1(NC(=O)NCC(Cc2cccc(C)c2)CO)ccc2c(c1)OC(C)(C)O2 74472,Cn1cccc1C(=O)NCC1(CNC(c2n[nH]cc2CN(C)C)=O)CC1 74473,c1(C(=O)NC2CCNC2)cc(C2CC2)nn1C(F)F.O=C(C=CCO)C1CC1 74474,C(CCC(=O)NC(c1cn(C(C)C(=O)OC)nn1)C)=CCC=C 74475,C12(CNC(c3ccc(Cl)o3)=O)CN(C(C3CC4(CCO3)CC4)=O)CC1CCO2 74476,c1(CC)nc(C)ccc1NC(=O)CC1COCCN1C(=O)C=Cc1cscn1 74477,C12(C(N3CC(CC)OCC3)=O)COCC1CN(C(=O)Cc1[nH]cnc1C)C2 74478,c1(C(N2CC(O)(CNC(C(C(CC)O)C)=O)C2)=O)cc2sccc2n1C 74479,c1(C(N2C3CC(NC(C(C4CC4)OCC)=O)C2CC3)=O)c(F)cccc1[N+](=O)[O-] 74480,C1(CC(=O)NC(CC)CNC(C2CCCCS2)=O)CCC2(CC1)CC2 74481,C1(CN(C)C(C2CCCN(C(N)=O)C2)=O)CCN(c2ncncc2Cl)CC1 74482,c1(N2CC(C)C(C(F)(F)F)C2)nccc(=NCc2cncn2-c2ccccc2)[nH]1 74483,C=CCCCCCC(C)OC.C1(=O)C(CCCC)N1 74484,Cc1ncnc(C)c1C(N1CCN(C(=O)CC(=O)NCC(F)(F)F)C(C)C1)=O 74485,c1(C(N2CCC(NC(CC(=C=C)C)=O)C(C)C2)=O)cc(N)c(Br)c(F)c1 74486,Cc1cc(CC(=O)NC2(CNC(c3nocc3C)=O)CCC2)cc(F)c1 74487,C1(C(=O)OCC)(CC)CCN(CC(=O)NC(C)CNC(C2CCOC2)=O)CC1 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74684,C(N=c1nc(C)c(Br)c[nH]1)C1(O)CN(C(CSc2nc(C)cc(C)n2)=O)C1 74685,C1(C(N(CCC#C)CCOC)=O)C=CCN(C(c2ccc(C(N)=O)[nH]2)=O)C1 74686,C1(OCC)CC2(C1)CC2C(=O)NCC1CCN(c2nnc(C(C)(C)CC)o2)CC1 74687,C1(CCc2n(-c3n(C)ccn3)nc(C(F)F)n2)CCc2ncsc2C1 74688,C1(CNC(C2(COC)CCC2)=O)CCCCCN1C(c1ccc(O)nn1)=O 74689,N1(C(c2ccc(CCCC)cc2)=O)Cc2ccc(-c3ccc(O)cc3C)cc2C1 74690,C1(C2CC2)(CNC(C2N(C)CC3(CC3)C2)=O)CCN(C(C2(C)COCCO2)=O)C1 74691,C1(CNC(CCCc2ccc(C)cc2)=O)C(C2CC2)CCN1C(c1cnco1)=O 74692,C(=O)(C(CC(C)C)C(C)C)NCC1CC2CN(C(Cn3c(C)cc(C)n3)=O)CC21 74693,C(=O)(CCCN=c1nccc[nH]1)NCC(CNC(=O)Cc1ccn(C(F)F)n1)F 74694,N1(S(c2ccc(N(CC(C)O)C)nc2)(=O)=O)CC2(CCOCC2)CC1C 74695,c1(SC)ccccc1CC(N1CC(NC(=O)C(F)(F)CN(C)C)C1)=O 74696,Cc1cc(C(=O)NCc2ncoc2CCNC(C2CCC(=O)C2)=O)c(Cl)cc1F 74697,CC1Oc2ccccc2OC1C(=O)NC1COCCN(C(=O)CN(C)C)C1 74698,CC(C)CC(F)C(=O)NC1(C)CN(C(C23CC4CC2C3C4)=O)C1 74699,c1(C(N2CC=CC(NC(C=C(C)Cl)=O)C2)=O)cc(F)cc2nccnc12 74700,C1(C(=O)NC(CN(C(C(CC(C)C)=O)=O)C)C)CCOC2(CCC2)C1 74701,Cn1ccc2cc(C(=O)NC3CC(NC(=O)CSC4CC4)CC3O)ccc12 74702,c1(C(=O)NC2(CNC(CC3C(C)C3)=O)CC2)cccc2[nH]ncc12 74703,C1(C(N2CC(CNC(=O)CC3CSCCO3)C(C)C2)=O)(CC)CCNC1=O 74704,C1(NC(c2c(C)c(N)ccc2)=O)CC2CC1CN(C(C1CC1C(N)=O)=O)C2 74705,c1(CN2C(C)(C(=O)Nc3cc(OC)c(Br)nc3)CC2)ccc(F)c2ccccc12 74706,C1(OC)CCN(C(C2CCN(C(=O)CCc3cc(C)on3)C2)=O)C1C 74707,C1(C(N2CC(CNC(c3ccc(C(=O)CF)cc3)=O)C2)=O)CC2(C1)CC(F)C2 74708,Cc1ccc(C(N2CC3C(NC(=O)Cn4cnnc4O)C3C2)=O)cc1S(C)(=O)=O 74709,C(CCCC(C)NC(c1conc1CN)=O)NC(COC(CC)C)=O.CC 74710,c1(OC)c(C(N2CC(NC(c3cc(C)c(C)o3)=O)C(C)(C)C2)=O)cc(Cl)cc1Cl 74711,C1(C(C)C)OCCC1CNC(=O)C(CO)NC(C1CC(C)(C)C1)=O 74712,C(=O)(CCN(OC)C(=O)C1CN(C)CCO1)NC(CC)C(N)=O 74713,c1(C(N2C3(CC)COC(C2)C3)=O)ccc(-n2cc(C(=O)O)nn2)cc1CC1CC1 74714,C(=O)(CC(CC)CC)OC(CCC)CN1C2CCC1COC2 74715,C1(NC(C2N(C(C)=O)CCC2)=O)C=CCN(C(=O)CSc2cnn(C)c2)C1 74716,C1(NC(CC(COC)C)=O)CN(C(c2conc2C2CC2)=O)Cc2ccnn2C1 74717,C1(NC(c2cc(Cl)c([N+](=O)[O-])[nH]2)=O)C2CCN(C(=O)Cc3ccncc3)CCC12 74718,C1(CC(=O)N(CCNC(=O)CC(O)c2ccccc2)CC)OCCC1(C)C 74719,C1(N(CCOC)C(c2ccoc2C2CC2)=O)CCN(C(=O)CC2CCC2)CC1 74720,c1(C(C)C)ncncc1C(=O)NC1CN(C(=O)C(O)CN(C)C)CC1C 74721,N1(C(C(c2ccn(C)c2)C)=O)CCC(C(=O)NC2CC23CCCCC3)C(O)C1 74722,CN1CCn2ncc(C(=O)NC3CC4(C3)CN(C(c3nnn(C)n3)=O)C4)c2C1 74723,C1(C(N(CC(=O)N(CC)CC)C)=O)CC(NC(=O)CCc2cnco2)C1(C)C 74724,N1(C(C(F)=C(C)C)=O)CCC(C)C1CNC(=O)C(C)Oc1ccccc1F 74725,c1(N2CC(N(C(=O)CC3CC=CC3)C)C2)c(Cl)cncc1[N+](=O)[O-] 74726,Cc1ccnc2c(C(N3CC(OCCNC(=O)CCCCCF)C3)=O)cccc12 74727,CC1=C(CNC(c2cc(F)cnc2Cl)=O)SCCO1 74728,N1(COC(C2CC(F)CN2)=O)CCCC1c1ccc(Br)s1 74729,c1(N(C2CC3CNC2C3)C(c2cc(C)nn2C)=O)ccc2ncnn2c1 74730,C1(NC(c2ccc(CO)nc2)=O)CCN(C(C2CCCOCC2)=O)CC1F 74731,N1(C(Cc2c(C)ccs2)=O)CCC2(CCCCN(C(=O)C(O)CC(N)=O)C2)C1 74732,N1(C(CCNC(=O)NC)=O)CCCC(CO)(NC(c2ccc(N)nc2)=O)C1 74733,CC(Cc1cnco1)C(=O)NCCC1(CNC(=O)CCc2cccs2)CC1 74734,C1(C(C)C)CN(C(c2n[nH]cc2-c2ccc(OC(F)(F)F)cc2)=O)CCO1 74735,c1(C(C)C)ccccc1C(=O)NCC1CC(O)CN1C(c1cc(Br)nn1C)=O 74736,c1(C(=O)NC2C(CNC(C3(Cl)C(C(C)=O)C3)=O)CCC2)ccc(C)nn1 74737,N1(C(c2cn(CC)nc2)=O)CCC(NC(=O)C2=CC(O)CCC2)C(C)(C)C1 74738,N1(C(C(C)N2CCC2)=O)CC2(CCCC2NC(=O)CC2CCC3CC23)C1 74739,N1(C(C=CCC)=O)CCN(C(c2ccccc2-c2nc(C)no2)=O)C(CC)C1 74740,c1(N2CCN(C(C3(COC)CCCO3)=O)CC(O)C2)cc(Cl)nc(S(C)(=O)=O)n1 74741,C(CC1(C)CC1)(C(=O)NCC1CCC1)N(C(C)C)C1CC1 74742,C1(NC(c2c(C)ccc(C)n2)=O)CC2CC(C1)N(C(c1ccc(=O)oc1)=O)C2 74743,C1(CNC(c2c(C)cncn2)=O)CN(C(C23CC(C)(CCO2)C3)=O)CCC1C 74744,c1(C(N2CC3C(NC(c4ccc(C(C)=O)o4)=O)(CC3)C2)=O)cc2n(n1)CCCC2 74745,c1(C(C)NCC(C2CCCOC2)OC)cn(C)c2cc(Cl)ccc12 74746,N1(C(C(c2cn(C)nn2)NC(C(CCC)N(C)C)=O)=O)CC2CC1C1CC21 74747,CCCC(CNC(=O)CC1CCCOC1)NC(c1ccoc1CC)=O 74748,C1(CNC(C2(C)CC2Br)=O)CN(C(c2nc(Cl)c(Cl)s2)=O)CCO1 74749,CON(C)CCNC(=O)C(C1CCN(C(=O)CN2CSCC2=O)C1)C 74750,N1(C(C2CN(C(C)=O)C2)=O)CCC(NC(=O)CNC(C2CCCCC2)=O)C(C)C1 74751,C12(C(=O)NCC3(OCC)CN(C)C3)CCC(CC1NC(=O)CN1CC=CC1)C2 74752,C(=O)(C(C)(C)C(C)NC(=O)C=CC(=O)N(C)C)N1CCC(NC(=O)OC)C1 74753,c1(CNC(C2(F)CN(C(c3cnc(C)nc3)=O)C2)=O)cccc(F)c1C 74754,Cn1cc2c(n1)CCC(COC(C1CCCC(CC(N)=O)C1)=O)C2 74755,CN1CCOC(C(=O)NC2CCC(CNC(=O)C(F)C3CCOC3)C2)C1=O 74756,C(=O)(C1OCCn2ccnc21)NCCC(C)NC(c1cn(CCC2CC2)nn1)=O 74757,N1(C(CCC(=C)Cl)=O)CCC2(C1)CN(C(C1CCCC(C)O1)=O)CCO2 74758,c1(OC)cc(-c2cnc(OC)c(C(=O)NCC(F)F)c2)cc(F)c1F 74759,N1(Cc2ncc(OC)nc2)CCN(C(=O)C=Cc2ccc([N+](=O)[O-])o2)C2(CC2)C1 74760,N1(C(c2c(C)ocn2)=O)CC(C(N2CCC3(CCCC3)C2)=O)CCC1(C)C 74761,C(=O)(C(O)CC(C)(C)C)N1CC(C)C(C(=O)NCCCN2CCC(O)CC2)CC1 74762,c1(CC)ccc(F)c(C(N2CCCC(F)(CNC(c3ncc[nH]c3=O)=O)C2)=O)c1 74763,C1(CC(NOCCC(C)O)=O)CN(C(c2csc(F)c2)=O)C(C)(C)C1 74764,C1(OC)CC2(C1)CC(C(N1CC(NC(=O)C=CC3CC3)C(F)C1)=O)C2 74765,C(=O)(CC1=CCCCC1)NC1(COC)CN(C(C2CC(C)CC(C)C2)=O)C1 74766,Cc1ocnc1CC(=O)NCC(c1ccccc1)CNC(C1CC(C)(C)C1)=O 74767,CC(C)(F)C(=O)N1CCCC1C1(O)CN(C(=O)CSCC2CCCCO2)C1 74768,c1(OC)cccc(C(N2CCC(C)C(NC(=O)C(F)C(F)(F)F)C2)=O)c1F 74769,C1(NC(c2n[nH]c(C)c2C)=O)CCCC12CN(C(=O)C#CC(C)(C)O)C2 74770,CN1C2CCC1CC(=CC(N1CC(F)CC1CNC(=O)CC1CCC(=O)O1)=O)C2 74771,Cc1cc(CCC(=O)NCCC(C)NC(c2cccc(CS(C)=O)c2)=O)c(C)o1 74772,CC1CCC(CNC(c2cc(Cl)c(Cl)s2)=O)N(C(c2cnn(C)n2)=O)C1 74773,N1(C(CC(CC)C)=O)CCCC2(COCC(=O)N2)C1 74774,CC(C)(CC1CCCN(C(=O)NCCC2CNC(=O)C2)C1)C(N)=O 74775,N1(C(C2CN(C)C(=O)N2)=O)C2CCC1CC(NC(c1cc3cccnc3s1)=O)C2 74776,C1(C(=O)NC(C=C)COC)(CNC(C2CCC(C)O2)=O)CC(C)(C)C1 74777,C1(C(=O)NC(C(=O)NCc2cnccn2)C2(C)CC2)CC2C(C1)C2(C)C 74778,N1(C(c2cc(C#C)cc(F)c2)=O)CCC(C2CCN(C(=O)CC3CC3)CC2)CC1 74779,c1(CC(=O)NC23CC(C(N(C(C)(C)C)CCN)=O)(C2)C3)cc(F)cc(Br)c1 74780,c1(CNC(c2cnns2)=O)ccc(CCNC(C2CCO2)=O)cc1 74781,Cc1ccnn1C(C)C(N1CCCC1C1(C(=O)NC2(C(C)C)CC2)CC1)=O 74782,N1(C(COCC)=O)CCC(CC)(NC(=O)C(O)CCSC)CC1 74783,c1(C(=O)NC2CC3CN(C(c4c(OC)ccs4)=O)CC32)csc2c1CCC(C)C2 74784,C1(C(=O)NC2CCC(N(C)C(c3cnc(O)n3C)=O)CC2)CCC2(CCC2)CO1 74785,N1(C(C2C3CN(C(CCCC=C)=O)C2C3)=O)CCC2(C=CCO2)C1 74786,CC1(CNC(=O)CN2CCCC(C(F)(F)F)C2=O)CCCN(C(=O)C(N)=O)C1 74787,CCC(O)C(F)(F)C(=O)N(C)CCN(C1CC(=O)N(c2nccs2)C1)CC1CC1 74788,C1(C(=O)NCC(COC)NC(c2csc(C)c2C)=O)CCCCC(=O)N1 74789,N1(C(c2n(CCCC)ncc2)=O)CCC2(CCC2)C(CNC(c2ccon2)=O)C1 74790,N1(C(C(C)(C)OCC)=O)CC2COCC2(C(=O)N(C)CC2(COC)CC2)C1 74791,Cc1noc(C)c1C(=O)NCC(C)(C(C)C)NC(C1CC(F)(F)CS1)=O 74792,CC(C(=O)OCC(c1cnc(C(F)(F)F)s1)=O)=C(Br)Br 74793,C1(SCc2c(C)nncc2)CCCCN(c2nc(C3CCC4(CCC4)O3)no2)C1 74794,N1(C(C(C(=O)OC)OC)=O)CCC(CNC(c2cccc(Cl)c2OC)=O)C12CC2 74795,C1(NC(C=NOC)=O)CCCC(CNC(=O)CNc2ccnc(C(F)(F)F)c2)C1 74796,C1(C(=O)NCC2(NC(C(C)c3cc[nH]n3)=O)CCOC2)CC(S(C)(=O)=O)C1 74797,CC1(C)CCN(NC(=O)C2CC3CNCC(C2)C3)CC1 74798,C1(CN(c2nncs2)C)CCCN1C(=O)C(F)C1CCOC1 74799,c1(OCCNC(N(C(CSC)Cc2cccs2)C)=O)ccccc1 74800,N1(c2ncc(C(=O)OC)cn2)CC2CCC1C(NC(C1CCN(C)C(=O)C1)=O)C2 74801,C1(CNC(C=C(C)Cl)=O)CN(C(=O)C(c2ccc(F)c(Cl)c2)C)CC(C)(C)O1 74802,CC(C(=O)NCC(C1CCCC1)NC(c1nccs1)=O)C1CCCC1 74803,N(C(=NCC(CC1CC1)CO)NC1CCC1)C(c1ccc(F)cc1)C 74804,N1(C(=O)NCCNC(=O)CO)CCCC2C1C2(F)F 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75155,C1(N=c2[nH]nc(C(F)F)o2)(CNC(C(C(C)O)C)=O)CCCCCC1 75156,C1(C(NOC2CCCCC2)=O)CN(C(=O)Cc2cnn(C)c2)C(C)(C)C1.CNC 75157,C1(CC(N2CCN(CC3(O)CN(C(C4C(C)C4)=O)C3)CC2)=O)CCCC(F)(F)C1 75158,N1(C(CN(CC)CC)=O)CC2CCCC2(NC(=O)C(C)Cc2ccc(C)cc2)C1 75159,C(=O)(C1CCc2c[nH]nc21)NCCCN(C(=O)CCn1cncn1)CCC 75160,Cc1ncc(CNC(=O)CC=CCNC(=O)Cc2cc(C)on2)s1 75161,C(=O)(C(C)CCC(C)(C)C)N1CC(O)CCC(NC(C=CCCC(C)C)=O)C1 75162,c1(CC(=O)NC2CCCC(CNC(C)=O)C2)ccc(F)cc1[N+](=O)[O-] 75163,N1(C(CCOCCCOC)=O)CCCC(CO)(NC(c2c[nH]nc2C)=O)C1 75164,N1(C(c2ccc(F)s2)C(=O)NCC)CCc2c(cc(F)c(F)c2F)C1 75165,c1(OC)ccncc1C(N1CCCC(N(C(=O)C(=O)NC2CC2)CCO)C1)=O 75166,Cc1ccc(C#N)c(NC2CC(CNC(=O)CCc3cc[nH]n3)C2)n1 75167,c1(C(N2CCC(O)(CN(C(C3CCC(=C)CC3)=O)C)C2)=O)cc2ccsc2n1C 75168,C1(O)(CNC(c2cn(CCOC)nn2)=O)CCCN(C(c2scnc2C)=O)CC1 75169,C12(NC(C)(C)C)C(NC(N(CCCOC)Cc3cccs3)=O)C3CC1C2C3 75170,Cc1c(C(=O)NC(C2CCN(C(c3occ4c3CCC4)=O)CC2)C)cncc1Cl 75171,c1(C(=O)NCCC(CNC(c2c(C)n(C)nn2)=O)O)cc(C(F)(F)F)ccc1F 75172,c1(N(CC(=C)Br)C)nc(N2CC=C(CN(C)C)CC2)nc2ccccc12 75173,n1(C(C)C)cnc2c(NCC3(C)CS(=O)(=O)C3)[nH]c(=NC3CCCCC3C)nc12 75174,C1(S(C)=O)(C(=O)OC)CCN(C(c2nnc3n2CCCC3)=O)CC1 75175,Cn1c(=O)sc2cc(S(=O)(=O)NCc3ccc4c(n3)NCCC4)ccc12 75176,C(CNC(c1cocn1)=O)(CC(F)(F)F)NC(CN1CCCC(CC)C1)=O 75177,c1(CC(C2CC2)CNC(N2CCC(C(O)CO)CC2)=O)ccc(Cl)cc1 75178,c1(SC)nc(Cl)cc(=NC(C)C(c2ccccc2)NC(c2cscc2OC)=O)[nH]1 75179,C1(NC(C(CC)=CC)=O)CCCN(C(=O)CCCC(C)N(C)C)C1C 75180,O=C(C1CCc2ccccc21)NCC1CCCC1NC(C1CCCS1(=O)=O)=O 75181,c1(C(N2C(CNC(CC(C(=C)C)O)=O)CC2)=O)ccsc1S(N)(=O)=O 75182,N1(C(C2COC3CN(C(C4COCC4O)=O)CC32)=O)CCCC(F)C(F)(F)C1 75183,C1(C(N2CC(OCCCCC)C2)=O)C=CCN1C(=O)C(n1ccc(C)n1)C 75184,C1(NC(c2ccc(C(CC)(C)C)cc2)=O)CCN(C(=O)C(C)C(C)C)C12CCC2 75185,C1(OC)CN(C(=O)CC2(O)CCCC2)CC1NC(=O)C(C)Sc1ccccc1 75186,CCC(C(=O)NCC(C1CC1)NC(C1CN(S(C)(=O)=O)C1)=O)n1nccc1C 75187,N1(C(c2c(CC)ccs2)=O)CCC(C(N2CCCCCC2)=O)C1C(C)C 75188,c1(NC(C23C(CN(c4nc(SC)nc(C)c4)C2)C3)=O)cc(F)c(C#N)cc1F 75189,C=C(Cl)C(C)(C)C(=O)N1CCC(O)(CNC(c2c[nH]c(-c3ccccc3)c2)=O)C1 75190,c1(C(=O)NC2C(NC(CCSC)=O)CS(=O)(=O)C2)ccc2ncn(C)c2n1 75191,C1(CC)CN(C(=O)CCCN(C)C)CCC1NC(C1(F)CCCC1)=O 75192,C1(CCNC(COCC(=C)C)=O)CN(C(c2cnc(NC)s2)=O)CCO1 75193,N1(C(C=CCN(C)C)=O)CCC2CCC(C1)N2C(c1cc(N)ccc1O)=O 75194,N1(C(c2cc(OC)ns2)C(=O)NCCCC2CC2)CCCc2c(C)cccc21 75195,C(C(C)N=c1[nH]c(=NCC(C)(C)COC)[nH]c2ccc(Cl)cc12)(OC)NC1CC1 75196,n1(CCC)ncc(C(=O)NC2C3CC(NC(c4nocc4Cl)=O)CC23)c1C 75197,C1(CC=C)(NC(C2CCCO2)=O)CCN(C(c2ccc(N)c(Br)n2)=O)CC1 75198,C(=O)(CC(F)(F)C(F)F)N1C(CN(C(=O)CN2CCNC2=O)C)CCC1 75199,C1(C(=O)NC(C)Cc2nc[nH]n2)(CNC(c2nonc2N)=O)CCCCC1 75200,C(=O)(CC(C(F)F)c1ccc(F)cc1Cl)N(C1CN(C(=O)C2CC2)CC12CC2)C 75201,n1(CCCC)nc(C)c(C=CC(N2CC(NC(=O)CC(F)F)C(O)C2)=O)c1Cl 75202,C(c1ccc(OCC#N)cc1)=CC(=O)NC(n1ccnc1)C 75203,N1(C(C(CC)CC2CCCCC2)=O)CC(C)(CNC(C2(O)CC2)=O)CC1(C)C 75204,C1(C(=O)NC23CC(COC)(OC2)C3)CC12CCN(C(=O)C1=CCN(C)C1)C2 75205,N1(C(CC(C#C)O)=O)CC(C)(C)CC(C)(C)C1 75206,C1(F)(C(=O)NCCc2c(CNC(CC(C)OC)=O)nco2)CCS(=O)(=O)C1 75207,C1(CNC(C(C=C)O)=O)CCN(C(c2nc(OC)c(C)s2)=O)C1(C)C 75208,N1(CC)CC(C(N2CCCC2C(=O)NCCCCCCC2CC2)=O)CC1=O 75209,CCCC(C(C)(C)C)NC(=O)CCC1CCN(C(=O)Cc2csnn2)CC1 75210,N1(C(C)C)CC(C(=O)N(C)CC2(NC(C3CC(CF)C3)=O)CC2)CCC1=O 75211,C1(CC(=O)NC2CCCC2NC(C2CC3CCC2C3)=O)CCC(F)(F)CC1 75212,c1(OC)ncc(Cl)cc1C(=O)NC1CN(C(C2(Cl)CC23CCC3)=O)CC1C 75213,N1(C(C(C=C)OC)=O)CC(O)CC1C(=O)NCCOC1CCOC1 75214,N1(C(c2cc(O)ncn2)=O)CCCC1C1CCCN1C(c1cc(O)ncn1)=O 75215,c1(C(=O)NC2(CCCC(N3CCC(OC)C3)=O)CCC2)c[nH]c(=S)cn1 75216,C=CCC(CC(=O)NCCOC)NC(=O)C(C)(C)OC1CCCC1 75217,C(=O)(CC(O)C1CCCC1)N1C(CNC(C)=O)CC1 75218,c1(C(=O)NC2CCN(C(C(C)NS(CC)(=O)=O)=O)C2)cc(N)ccc1O 75219,c1(C(=O)NCC(C)N(C(=O)CCc2cncn2C)CC)cc(F)cnc1O 75220,Cc1cnc(C)c(NC(C2CC2c2ccccc2OC(F)F)=O)n1 75221,c1(C(=O)NC2(CF)CCN(C(C(N3CCC(C)C3)=O)=O)C2)cccc2c1CCCC2 75222,C(=O)(CC1=NNC(=O)C1)N1CC(N(C)C(c2cncs2)=O)C(O)CC1 75223,C1(C(C(=O)NC(CC)C)N(CCCCO)C)C2CCOCC12 75224,N1(C(C(F)OC)=O)CCCC1CN(C(=O)C(C)(C)N(S(C)(=O)=O)C)C 75225,C1(NC(=O)CC2C=CCCC2)C2CCN(C(C3(CF)CC(F)(F)C3)=O)CC12 75226,CC(C)(C#Cc1cn(-c2ccc(F)nc2)nn1)NC(c1nsc2ccccc12)=O 75227,N1(C(CC=CC=C)=O)CCN(C(=O)Cc2ccc(C)c(OC)c2)C(C2CC2)C1 75228,C1(CC(=O)NCC(COC)C)CC2(C1)CN(C(=O)C(C)C(F)(F)F)C2 75229,c1(OC)nscc1CNC(=O)COCCNC(=O)Cc1ncoc1C 75230,C1(F)(CNC(C(CC(C)C)N(C)C)=O)CCCN(C(=O)OC(C)(C)C)CC1 75231,N1(C(c2cn(CC=C)nn2)=O)CCC(F)C(NC(c2cc(C3(C)CC3)n[nH]2)=O)C1 75232,c1(C(N2CCOC(O)C2)=O)[nH]nc2c(-c3cc(O)c(F)cc3F)cccc12 75233,c1(OCC)cccc(C2CCC2c2ccn(C(F)(F)C(F)c3ccccc3)c2)c1 75234,c1(C(=O)NCC2CC(CC)CN2C(c2cc(=O)n(C)cn2)=O)ccc(F)c(O)c1 75235,CCCCC(CNC(c1ccnc(NC(=O)C(C)OCC(C)C)c1)=O)NC(C)=O 75236,Cn1cc(C(C(=O)NCCC(C)(C)O)NC(=O)CNC(N)=O)nn1 75237,c1(C(=O)NC2(C)N(C(CCN(C)C)=O)CCC2)cc(Cl)ccc1C(F)(F)F 75238,N1(C(=O)CC2=CCCC2)CCOC2(CCN(Cc3cc4cnccc4[nH]3)CC2)C1 75239,CCC(CC)C(C)NC(C1OCCC1NC(=O)C(C)(C1(C)CC1)OC)=O 75240,Cn1ncc2cc(CNCc3ccsc3)c(Cl)nc12.C1(=O)CCCN1 75241,c1(C(=O)NCCC(C(C)C)NC(c2c(CC)nc[nH]2)=O)cccc2oc(O)nc12 75242,c1(OC2CC(NC(CCn3cc(CCCC(C)O)nn3)=O)C2)ccc(F)cc1 75243,CCCC(O)C(=O)N1CCC(C2N(C(=O)C=CC3CC3)CC2(C)C)CC1 75244,C1(NC(C2C(C(=O)OC)C2(C)C)=O)CCC(C)N(C(c2ccc(F)c(F)c2)=O)C1 75245,C1(C)(C(=O)OC)C=CCCN1C(c1cccnc1COC(C)=O)=O 75246,c1(C(=O)NCCN(C(C=C(C)c2cccs2)=O)C2CC2)cnn2c(=O)cc[nH]c12 75247,C(C(C)C(C)C(=O)NC(C1(O)CN(C(=O)C(O)C2CCC2)C1)C)OC 75248,C1(NC(c2ccc(Cl)cn2)=O)CC2CC(NC(C3(C4CC4)CC3)=O)C2C1 75249,c1(C(N2CC(O)(CNC(c3cnc(CC)nc3C)=O)C2)=O)c(C)cc(C)nc1O 75250,Cc1cc(N)c(C(=O)NC(C)(CNC(=O)C(C)(C)c2ccccc2)CO)cc1C 75251,O=C(C#CC1CC1)NCC12CC1CN(C(C1CC(=O)N(CC3CC3)C1)=O)C2 75252,N1(C(C)=O)CC(NC(C=CC(=O)NCC2(COC)CC(F)(F)C2)=O)CC1(C)C 75253,c1(C(=O)NC(C)CN(C)C(c2ncncc2Cl)=O)c[nH]cc(Cl)c1=O 75254,CC1CC(=O)NCC1C(N1CCCC1(C)CNC(C1CC(O)C1)=O)=O 75255,c1(OC)ccc(Br)nc1CN1CCCC(C)(C(=O)Nc2nc(Br)ccc2Br)C1 75256,Cc1cnoc1C(=O)N(C(C)C(=O)NC1CN(C(=O)C(N2CCOCC2)C)C1)C 75257,C#CCCCCC(=O)NC(C(=O)NCCc1cnn(C)c1C)C1CCOC1 75258,CCCCCCCCC(=O)N(C1CCCN(C(=O)CC2CCCCC2O)C1)C 75259,CCCC(CCC)=CC(=O)N(CC)Cc1cn(-c2cc(C)sc2C)nn1 75260,C1(C(N2C(C)CCC2C(=O)Nc2ccc(F)nc2)=O)CC2CCCC2C1 75261,c1(C(=O)NCCCN(C(C(CC)OC)=O)C2CCCC2)ccc(C)n1C 75262,c1(COC)ccsc1C(=O)N(C1CCN(C(=O)CCC=C(C)C)C1)CCO 75263,C12(NC(C)C(C)Oc3ccccc3)CCC1CNC2 75264,CC1(C)C(C)(C(=O)NCC2(O)CN(C(c3ccccc3CC#N)=O)C2)C1(C)C 75265,c1(C(=O)OC)ccc(C(N2CC3CC3(C(=O)OC)C2)=O)cn1 75266,C(C(=O)NNC(=O)C1=COCCO1)(c1cccc(Cl)c1)OC 75267,Cc1cc(C(=O)NC2CC(CNC(C3(c4ccno4)CC3)=O)C2)cn1C 75268,C(=O)(CC(C)(C(F)F)N(C)C)N1CCN(C(c2c(C)[nH]c(C#N)c2)=O)CC1CO 75269,N1(C(CC(=O)OCC)=O)CCN(C(C)CNC(c2cnns2)=O)CC1 75270,c1(C(N2CC(N(C(C(C)CC3CC3)=O)C)C(O)C2)=O)cc(C(F)F)ccc1Cl 75271,N1(C(c2nc(C)c(C)s2)C(=O)NCC)CC(C)C(C)C1C 75272,c1(N(CC)CC)ccc(CCC(=O)NCC(CC)NC(C2CCC2(C)C)=O)cc1 75273,CC(C(=O)NC1CN(C(C2(C3CCC3)CC2)=O)CCC1C)S(N)(=O)=O 75274,C1(C2CN(C(C3C4CC4C4CC34)=O)C2)(NC(c2ccc(O)c(Br)c2)=O)CC1 75275,C1(F)(C(C)NC(C2CCCN2C(=O)CCc2cscn2)=O)CCN(C)C1 75276,Cc1cc2[nH]c(C(=O)NC3CC4(CCN(C(C56CC(CO5)C6)=O)C4)C3)cc2o1 75277,N1(C(C2CCC(NC(COC3(C)CCC3)=O)C2)=O)CC(O)C(O)C12CCC2 75278,C(C)(C)(CC(=O)NCc1ccoc1C(=O)NCCCC(O)CO)N(C)C 75279,c1(C(=O)NC(C(=O)N(CC)Cc2cnn(C)c2)c2ccoc2)cc(OC)n(C)n1 75280,N1(C(C2(C(=O)NC3CC3)CC2)=O)CC2CCCC1CN(C(c1cnc(Cl)s1)=O)C2 75281,CC1CCN(C(c2ccc3c[nH]nc3c2)=O)C(C)C1NC(c1ccc(F)nc1)=O 75282,C1(NC(c2cc(C)nc(C)n2)=O)CC2CCC(C1)N2C(=O)C(O)c1cnc[nH]1 75283,c1(C(=O)NC2CCC(F)(CNC(C)=O)C2)ccc(Nc2ccncc2)cc1Cl 75284,c1(C(N2CC(C)C(NC(=O)C3=CCCSC3)CC2)=O)c(Cl)ccc(F)c1F 75285,C(=O)(C(F)(F)C(C)(C)O)NC1C=CC(CNC(c2cnc(C(C)C)[nH]2)=O)C1 75286,CCC(O)C(F)(F)C(=O)NCCCC1CCN(C(=O)CC(C)C(C)(C)C)CC1 75287,N1(C(CN(C(C(C)C)=O)C)=O)CCC2CN(C(=O)C(O)CC3CCOCC3)CC2C1 75288,Cc1cc(C)c(C(=O)NCCN(C(=O)CC2CC2C)C)c(C)c1 75289,N1(C(C(CCN(C)C)NC(=O)CCn2ccnc2)=O)CCC(F)(F)C(F)C1 75290,C#Cc1ccc(NC(=O)C(C)(C)CN(C(=O)CCc2ncnn2C)C)cc1 75291,O=C(C1CCc2ccccc21)NC1CN(C(C2CCC(CO)CC2)=O)CC1F 75292,CN=c1nc(N(C)Cc2ccc(=N)[nH]c2)[nH]c(=NC(C)c2ncnn2C)[nH]1 75293,C1(NC(=O)CCF)CC2CC1N(C(c1ccncc1-n1cccn1)=O)C2 75294,C1(C(=O)NC(CNC(C2C(COC)C2)=O)CO)Cc2cccc(OC(F)F)c2O1 75295,C(=O)(CCCC(F)(F)F)N1C(CCNC(C2C(C)(C(F)F)C2)=O)COCC1 75296,c1(C(N2CCN(C(CCOCC#C)=O)C(COC)C2)=O)cnc2n1CCC(C)C2 75297,C1(C)(CC)COCCN1C(=O)CC1NC(=O)NC1=O.c12csc(n1)NC(=O)C2 75298,Cc1ccc(C(=O)NCC2(NC(C3CCCCN3C)=O)CCCCC2C)c(N)c1 75299,N1(Cc2ccc(C#N)s2)CCc2cccc(C(N3CCNC(=O)CC3)=O)c2C1 75300,C1(C)(CC(=O)NC(COCC)C)CCN1C(=O)CC1(C)OCCO1 75301,C1(C(N2CCC(C(C)NC(c3cscn3)=O)C2)=O)CC1C1CC1C 75302,N1(C(c2ccccc2Cl)C(=O)NCC)CCn2c(CC)nnc2C1 75303,Cc1ccc(Cl)cc1-c1cn(C2CN(C(c3csc(CC(C)C)n3)=O)C2)nn1 75304,CC1(C)CCCCC1C(=O)NC1C=CC(C(=O)NCC2CC(O)C(O)C2)C1 75305,N1(C(c2cc(C)on2)=O)CCC(F)(C(=O)NC(C2CCCOC2)(C)C)CC1 75306,N1(C(C(N2CCOCC2)C)=O)CC(NC(c2sc(Cl)cc2Cl)=O)CC1(C)C 75307,N1(C(C2=CCCN(C(=O)OC(C)(C)C)C2)=O)CCC2(C1)CS(=O)(=O)C2 75308,C1(CC(=O)N(CCNC(c2cscc2Br)=O)CC)CC(C)(C)OC1=O 75309,C(C(C)(C)CC(=O)NCC(C1CC1)NC(C1CC(C)(C)CO1)=O)N(C)C 75310,c1(C(=O)NC(C)CN(C)C(c2cc3c(s2)CCCC3)=O)cc2cc(Cl)ccn2n1 75311,C1(O)(CNC(C2(CSC)CCC2)=O)CCN(C(=O)Cc2ccc(O)cc2Cl)CC1 75312,N1(C(CSCC=C)=O)CCCC2CN(C(=O)CCc3cnn(C)c3)CCCC12 75313,c1(C(N2CC(CC)C(NC(c3ccncc3)=O)CC2)=O)cc2nc(Cl)ccc2s1 75314,C1(C(N(CC(CCC)C)C)=O)CCC2(CC2)N1C(C1CCCO1)=O 75315,c1(CC)ncccc1C(N1CCCC1CN(C)C(c1ccnnc1)=O)=O 75316,N1(C(c2c(C)cnnc2C)C(=O)NC2CC2)CCc2cccc(CO)c2C1 75317,C1(C(=O)NCc2ccsn2)CN(C(=O)C(c2cccc(Br)c2)O)CCC1(F)F 75318,CC1CC(CN2CCCC2Cc2ccncc2)CCO1 75319,CCCCC(O)CC(=O)NCC1(O)CC(NC(=O)CCOc2ccc(C)cc2)C1 75320,C1(C)(C(=O)NC(C(CCC)C)C)CCN(C(c2ccccc2C)=O)CC1 75321,c1(C(=O)NC2CC3(CN(C(CCCCC)=O)C3)C2)c(Cl)ccc(OC)c1N 75322,Cc1cc(=NCC(CNC(=O)C(C)CC(N)=O)C(F)(F)F)[nH]c(C)n1 75323,N1(C(C(C(CC)C)O)=O)CCCC2(C1)CN(C(C1CCCN(C(C)=O)C1)=O)C2 75324,C1(C(=O)NCC(C)N(C(=O)CCC(=O)c2ccc(F)cc2)C)CCC2CCC1O2 75325,C1(OCC)CC(N(C)C(c2ccc(CO)nc2)=O)C12CCCCC2 75326,N1(C(C2(F)CCN(C(c3cnc(N(C)C)o3)=O)C2)=O)C2CCC1COC2 75327,Cc1cc(NC2CC(CNC(c3cc(C(N)=O)[nH]n3)=O)C2)nc(CC2CC2)n1 75328,C1(CNC(C=C(C)C2CC2)=O)(CNC(=O)C(C)OCC2CCCO2)CCCC1 75329,C1(CNC(c2cnc(C)s2)=O)CCN(C(=O)CC2CC(C)(C)C2)C1(C)C 75330,c1(NC)ccc(C(=O)NCCCSCCC(CO)OC)cc1 75331,C12(C(N3CCC(COC(C)=O)C3)=O)CCCC1CCN2C(=O)C1=CC2C=CC1C2 75332,N1(C(CCN2CCC(C)CC2)=O)CC(NC(C2CCOC2)=O)C2(CC2)C1 75333,C1(C(=O)NCC2COCCN(C(c3cc(OC)n[nH]3)=O)C2)Cc2ccccc2O1 75334,C1(NC(c2cc(C)n(C3CCCOC3)c2C)=O)CNC(C)(C)COC1 75335,CC1CC(NC(=O)CNC(=O)OC(C)(C)C)CN(C(c2ncccc2Br)=O)C1 75336,c1(CC)cc(NC(N2CCCC2CC(c2ccccc2)O)=O)n(C)n1 75337,N1(C(c2ccc(CNC(c3occ(C(N)=O)c3)=O)o2)=O)CC(O)CC12CCC2 75338,N1(C(C(CC)n2ccnc2)=O)CCC2OCCN(C(c3nc(=O)n(C)[nH]3)=O)C2C1 75339,CC1CCCCC1(CNC(=O)CNC(c1cnn(C)c1)=O)NC(=O)C=C(Cl)Cl 75340,c1(NC(CC(CC)C(C)(C)C)=O)cc(C)c2ncccc2c1C 75341,c1(C(N2CC(NC(C3(F)CCC3)=O)C(F)C2)=O)ccc(Br)c(Cl)c1Cl 75342,C1(S(C)(=O)=O)(C(N2CCC(F)(CNC(c3cc(C)oc3)=O)C2)=O)COC(=O)C1 75343,Cn1ncc(=NC(=O)C2C3CN(C(c4cc(Cl)cc(F)c4Cl)=O)CC23)[nH]1 75344,N1(C(c2n[nH]c(CC)c2C)=O)CCOCC(C(=O)N(CC(C)C(=O)OC)CC)C1 75345,C12(CNC(c3cn(CCOC)nc3)=O)CC1CN(C(c1ccn(CCF)n1)=O)C2 75346,C(=O)(CCC(C)(F)F)NC1(C)CC(NC(C(C2CCC(=O)NC2)OC)=O)C1 75347,C(CCOCC)(C(=O)NC1CC(NC(N)=O)C1)NC(c1c(CCCC)ocn1)=O 75348,CC1=C(C(=O)N2CCCC(C)(C(=O)NCc3ccc(C)n3C)C2)CCO1 75349,Cc1ccn(CCC(=O)NC2CC(C)(CNC(=O)Cc3n[nH]c(C)n3)C2)n1 75350,C1(NC(C(CSCC(C(=O)OC)OC)C)=O)CC2C=CCC(C1)C2 75351,C1(C(N(C(C)CNC(C2(CO)COC2)=O)C)=O)CC(=O)N(Cc2ccccc2)C1 75352,c1(N(C2CC3CCC(C2)N3)C(=O)CN2CCc3sccc3C2)ccc2ncsc2c1 75353,Cc1c(F)ccc(Cl)c1C(N1CC2CC(NC(=O)C(C)c3cccs3)C2C1)=O 75354,Cc1c(CC(=O)N(C)CCN(C)C(c2cn(C)c(C)n2)=O)cccc1Br 75355,N1(C(c2nc(C(C)O)oc2)=O)CCC2(CC1)CN(C(=O)C=CCF)C2 75356,N#Cc1ccc(NC(c2n[nH]cc2NCc2c(Cl)ccnc2Br)=O)cc1Br 75357,C1(C(=O)NCc2cc(C(=O)NCC3(COC)CCCC3)n[nH]2)CCC(O)CN1C 75358,C(=O)(CC(C)C1CCCO1)NC1(C(N(CCF)CC)=O)CCC1 75359,C(=O)(C(=O)N=c1ccn(-c2ccc(Cl)cc2C#N)[nH]1)NC(CCOC)C(C)(C)C 75360,Cn1nc(O)cc1C(=O)NCC(c1ccccc1)NC(c1nnsc1N)=O 75361,C12(NC(C=CSC)=O)CCCCCC1N(C(c1cc(F)c(N)cc1F)=O)CC2 75362,C1(C(=O)OCC)C=CC(C(=O)NC2CC(NC(c3c[nH]nc3C(C)C)=O)C2)C1 75363,N1(C(C2CC(C(C)C)C2)=O)CCC(C(C)NC(c2ncn(C)n2)=O)CC1 75364,c1(CNC(C(C)N(C)C(C2(C#N)CCCO2)=O)=O)ccccc1CO 75365,C#CC1CN(C(=O)C(C2CCCO2)NC(=O)CCN2CCOCC2)CCO1 75366,c1(SCC(=O)NC(CC2CN(C(CCC=C(C)C)=O)C2)C)nc2ccccc2[nH]1 75367,N1(C(C(C)OCCOC)=O)CCC2(CCCN(C(=O)CCCN(C)C3CC3)C2)CC1 75368,n1(CC(=O)NCC2CCN(C(CC(=O)N(C)C)=O)C2(C)C)cc2ncccc2n1 75369,Cc1ccc(C(=O)NCC2CCN(C(c3cc[n+]([O-])cc3)=O)C2)cc1O 75370,C1(C)(C(=O)NCC(C)(CO)CO)CCCN(C(=O)COCC2CCCO2)C1 75371,c1(NC(C2CCC(NCc3cnn(CCC)c3C)CO2)=O)cc(F)c(Cl)cc1F 75372,c1(NC(C(C)(C)C2CCN(C(=O)CC3(C)CCC3)C2)=O)ccc2nccn2c1 75373,C(C)(C(=O)NCC1(C(=O)NCCCOCC(C)C)CCC1)OCC(C)C 75374,C1(NC(C(C2CC2)OCC)=O)CN(C(=O)Cc2ccc3c(c2)CC3)CCC1(F)F 75375,C1(CNC(c2c(C)csc2)=O)CCC=CC1NC(=O)Cc1cnn(C)c1C 75376,c1(N2CCN(Cc3onc(C(C)OCC)n3)CC2)ncc(C(N)=O)cc1Cl 75377,N1(C(C(CC)N(C)C(c2ccc(C#N)cc2)=O)=O)CCC(F)(F)C(O)C1 75378,C(CNC(C1CC1(C)C)=O)(CO)NC(CSCC)=O 75379,C1(NC(c2n(C)ncc2)=O)CN(C(c2cnccc2Cl)=O)C2(CCCC2)C1 75380,C1(CNC(C23OC(C)C(CC2)C3)=O)CC2CCC(C1)N2C(c1cc(F)c[nH]1)=O 75381,C1(CNC(C2N(C(CC)=O)CSC2)=O)CN(C)CCN1C(C1CCC(=O)N1C)=O 75382,C1(O)(CNC(C2=CC(C)(CC)C2)=O)CCCN(C(c2cc[nH]c2)=O)CC1 75383,C(=O)(C1CCCn2cc(C)nc21)NCCN(C(=O)CCC(C)(C)[N+](=O)[O-])CC 75384,Cc1cnc(NC(C2CC2C(=O)Nc2cccc(I)n2)=O)c(C)c1 75385,CC1CC(NC(C2CC2C2CCC2)=O)CN(C(=O)Cc2nn(C)cc2Cl)C1 75386,C1(C)(NC(C(C=O)OC)=O)CCCCC1C(=O)NOCC(C)(F)F.CO 75387,c1(C(C(C)NC(=O)C(=O)NCc2cc(C3CC3)[nH]n2)OC)ccc(Cl)cc1 75388,C(=O)(C1CCCc2nc[nH]c21)NCC1CN(C(C2C(C)C2C)=O)CC1C 75389,C1(CNC(C(C2CN(C(C3CCC(CO)C3)=O)C2)OC)=O)CCCN(C)C1 75390,c1(CC(=O)NC2CC(CCNC(C3(CCOC)CC3)=O)C2)cc(F)c(F)cc1F 75391,C(=O)(C1=CN=C2N=CNN2C1)NC1CC(C)N(C(=O)C=Cc2nccs2)CC1 75392,N1(C(C(=O)NC(C)CCCNC(C2CCCO2)=O)C)CCCCCC1 75393,c1(OC)ccnc(F)c1C(=O)NC1CN(C(C2CC2(C)C)=O)CC1C#N 75394,C1(n2cccn2)(C(N2CC(C)(COC)C2)=O)CCN(C(c2ccsc2C)=O)CC1 75395,C(CC(C)C(=O)N(C)CC1CCCN1C(c1cc(-c2cccnc2)[nH]n1)=O)OC 75396,Cc1cccc(C(N2CCCC2CN(C(=O)Cn2cn[nH]c2=N)C)=O)c1O 75397,c1(C(=O)NCCCC(C)NC(=O)N(C)C)c(CNC(CC=C=C)=O)cccc1F 75398,c1(CC)c(OC)cccc1C(=O)NC1CN(C(=O)Cn2ccc(C)n2)CC12CC2 75399,CN1CCCC12CCN(C(c1nc(Cl)c(Cl)s1)=O)C2 75400,N1(C(CCOC(COC)=O)=O)C(C(=O)N(CCCCF)CC)CCC1C(C)C 75401,C(CC(F)(F)C(=O)NCCC(=O)N(C)C(C)C)n1cc(-c2cn(CC)nc2)nn1 75402,C1(NC(=O)NC(C)CN(C)C)NCC2CC12 75403,N1(C(C2C(C)CC2)=O)CCN(c2ccc(CCNC(=O)CC3(C)CC3)cc2)CC1 75404,C(=O)(CS(=O)(=O)CCOC)NCC1C(C(F)(F)F)CCN(C(C=COCC)=O)C1 75405,c1(C(=O)NCC2(NC(C3(COC)CC3)=O)CC2)cnc(C(F)(F)F)s1 75406,CC1(C(N2CC3C(CNC(c4ccc(CC5CC5)s4)=O)C3C2)=O)CC2CC2C1 75407,S(=O)(=O)(CCNC(C1CCCSC1)=O)NCC(=O)OC 75408,C1(NC(c2cn(CC(=O)OCC)nn2)=O)CCCCN(C(=O)C(C)C2CC2)C1 75409,Cc1cnc(CC(=O)NC2CN(C(c3cnnn3C3CCOCC3)=O)C2)o1 75410,C1(SC)CC(CC(=O)N(C(C)C(=O)NCCCC2CC(C)C2)C2CC2)C1 75411,c1(C(N(C2CCCC2)CCNC(C=COCC)=O)=O)cnn2c1CC(C)CC2 75412,N1(C(CS(CC)(=O)=O)=O)CC2COCC2(C(=O)NOCc2cccc(C)n2)C1 75413,c1(C(N(c2cccc(C(=O)NC)c2)C)=O)cc(C(F)F)cc(Br)c1 75414,CC(C)CC(C)NC(C1(NC(=O)CCn2cncn2)CC1)=O 75415,C1(C(=O)NCC(C)CNC(C2C3CCN2CC3)=O)CN2CCCN1CC2 75416,Cc1cn(-c2ccccn2)[nH]c1=NC(=O)N1CCC(n2ccnc2)C1 75417,N1(C(C=C(C)C)=O)CCC(NC(C2(C)CCCCC2)=O)C1C 75418,c1(C(C)=O)ccncc1C(N1CC(O)CC1CNC(=O)CCN1CCOCC1)=O 75419,c1(NC(C2CC=CCN2C(C2CCCOCC2)=O)=O)ccc(CCF)cc1 75420,Cc1ncc(C(N2CCC(N(C(=O)CC3CCOCC3)CCO)C2)=O)[nH]1 75421,CCCCC(O)CC(=O)N1CCC(C(N2CCC(O)C(CO)C2)=O)C12CCC2 75422,C1(C(N(CCCC)CC)=O)CC12CC(NC(=O)C(n1ccc(C)n1)C)C2 75423,c1(C(N2CCOCC2c2ccc(Br)cc2)=O)cc2c(Cl)c(Cl)ccc2[nH]1 75424,S(=O)(=O)(c1ccc(=NC2CS(=O)(=O)CC2O)[nH]c1)N1CCCC(C(N)=O)C1 75425,c1(C(C)NC(=O)COc2ccccc2)ncncc1OC.C(C(C)(C)C)CCN 75426,c1(N(C)Cc2ccc(CO)cc2F)nc(=NCC2CC2Cl)[nH]c2cc[nH]c12 75427,N1(C(=O)CC2C=CCCC2)CC(NC(C23CCC(F)(CC2)C3)=O)C2(CC2)C1 75428,C1(NC(=O)C2CC2)CC2CCC1CN(Cc1nc(-c3ccccc3)cc(O)n1)C2 75429,O=[N+]([O-])c1ccnn1-c1ccnc(C2CCC2)n1 75430,Cc1ccc(C(N2CC(C)(C(N3CC(CO)C(C)(C)C3)=O)C2)=O)cc1O 75431,C(=O)(CCCF)N(CC(=O)NCCOC(C)(C)C)C(C)C 75432,c1(C(N(CCCC(=O)NC(C=C)(C)C)C)=O)ccc(C#N)n1C 75433,C1(NC(c2c(C)ncc(CC)c2)=O)CCOC2(CCS(=O)(=O)CC2)C1 75434,CN1CCOCC1C(=O)NC1(CCC(=O)NC2(C)CCC2)CCC1 75435,C1(OCC#C)CCN(C(=O)CC2CCC(NC(C3CCCC3O)=O)C2)CC1 75436,c1(CCC(=O)NC(C2CCN(C(=O)Cc3cnc[nH]3)CC2)(C)C)ccc(=N)[nH]c1 75437,C(C(CC)(CC)C(=O)N1CCC(OCC(N)=O)C1)NC(Cc1cn(CC)nc1)=O 75438,N1(C(C(CNC(C=C(CC)CC)=O)N(C)C)=O)CCS(=O)C(C)C1 75439,c1(CC)ccc(Cl)c(C(=O)NC2CCC(NC(=O)C(CC)SC)CC2)c1 75440,Cc1ccc(C(N)=O)cc1C(=O)NC1CCC1NC(=O)Cc1cc(Cl)sc1Cl 75441,c1(CC(C)C(=O)NCCC(C)N(C(=O)CCc2ccccn2)C)ccc(F)cc1 75442,N1(C(c2n(CC)cnc2)C(=O)NC(C)C)CCS(=O)(=O)CC1 75443,C(N=c1[nH]c(N(C)CCc2ccccc2Cl)nc2cc[nH]c12)c1c(CC)nco1 75444,N1(C(CCC(=C)C)=O)CCC2(C1)CN(C(C1C(C)CC1C)=O)C2 75445,C1(NC(c2c(C)cc(C)o2)=O)CC2(C1)CN(C(=O)Cc1cn3ccsc3n1)C2 75446,CCC(CC)(C(=O)NC1CC(C)N(C(=O)Cc2cccnc2)C1)OC 75447,C1(CC)C(C(=O)NCCCOCCN(C)C(c2ccc(CC)[nH]2)=O)CCN1C 75448,c1(C(=O)NCCN(C(=O)CC(C)N(C)C)CCC)c(Cl)c([N+](=O)[O-])nn1C 75449,C(=O)(C(C#N)C(C)C)N(CCCNC(=O)C(O)COc1ccccc1)CC 75450,c1(C(C)C)cccc(F)c1C(=O)OCC1CCN1C(c1cc(Cl)no1)=O 75451,CCCC(C(=O)NC12CCCN(C(=O)Cc3cccc(Cl)c3)CC1C2)S(N)(=O)=O 75452,N1(C(COC(CC)C)=O)CCC2(CC1)CN(C(c1cc(Cl)c(Cl)[nH]1)=O)C2C(C)C 75453,C1(O)(CCNC(CNC(CC)=O)=O)CCN(C(=O)CCC2CCCOC2)C1 75454,C1(NC(=O)CSC2CC2)CCN(C(=O)C(O)CC(F)(F)F)CC12CCC2 75455,C1(NC(C(F)OC)=O)CCC2CC1CN2C(=O)C=CC=Cc1ccccc1 75456,Cc1nc2ccc(F)cn2c1C(=O)NC1CN(C(c2c(C)noc2C)=O)CC1F 75457,C#CC1(O)CCN(C(=O)CNC(c2ncc(OCC)cc2Cl)=O)CC1 75458,Cc1cc(C(=O)N(CCCOCCNC(=O)CC2CC2(C)C)C)nnc1O 75459,C#CCC(C)C(=O)NC1CCN(C(C2(Cl)CC2(F)F)=O)C1 75460,c1(OC)cc(CNC(C2CC(NC(=O)CCC3CC3(F)F)C2)=O)ccn1 75461,Cc1ncc(F)c(N2CCOCC2CN(C)C(c2cc(C)n(C)c2)=O)n1 75462,C1(C(=O)NCCCC(C)NC(C2C(CC(C)C)C2)=O)CCC(N(C)C)CC1 75463,Nc1ccc(C(N2CC3CC2C3CNC(C2CCC23CCC3)=O)=O)cc1Cl 75464,c1(C(=O)NC2C(NC(=O)CC3CC3C(F)(F)F)COC2)cc2c(Cl)cccn2n1 75465,C1(NC(Cc2cn(CC)nn2)=O)C=CCN(C(C23CC(C(C)C)(C2)C3)=O)C1 75466,C(=O)(C(C)(C)CCOC)N1CC(CNC(C(C)OCC)=O)C(N(C)C)C1 75467,C1(c2nc(COCC)nn2-c2ccnc(C(F)(F)F)c2)CCc2cn(C)nc2C1 75468,c1(CC)n[nH]c(=NC2CCN(C(=O)Cc3ccc(F)c(F)c3)CC2C)o1 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75556,CC1(C)CN(C(=O)Cc2csc(Cl)c2)CC1NC(=O)CC1CCOC1=O 75557,C1(NC(C(CCOC)C)=O)CCC2(CC1)CC(NC(=O)CSc1cccs1)C2 75558,C1(Cc2cnc(C)cn2)C(C)CCCN1C(=O)NCC=CCSC 75559,N1(C(C(n2ccc(C)n2)(C)C)=O)CCC2(CCC2CNC(=O)COC(C)C)CC1 75560,N1(C(c2oc(C)c(Br)c2)=O)CCC(NC(C2CC23CCC3)=O)C12CCC2 75561,c1(OC)cncc(C(N2CCC(C(N3CCC(C)(C(N)=O)C3)=O)(OC)C2)=O)c1 75562,Cc1nc(C(=O)N(C2CCN(C(=O)CC3NC(=O)NC3=O)C2)C)ccc1[N+](=O)[O-] 75563,N1(C(C2(C#C)CCC2)=O)CCCN(C(=O)C(C)C(C)C)C(CO)C1 75564,Nc1cc(Cl)nc(C(=O)NC2CCC(CNC(c3cccnc3S)=O)C2)c1Cl 75565,c1(CC)cc[nH]c1C(=O)NCCOCCCN(C)C(C1(C)CC1(Cl)Cl)=O 75566,CC1(NC(c2cn(C3COCC3F)nn2)=O)CN(C(C2(C(F)F)CCCO2)=O)C1 75567,Cc1cc2ncc(C(=O)NC3COCC3NC(c3ncccc3F)=O)cn2n1 75568,c1(C(=O)NCC2CC(NC(=O)C(=C3CCCCC3)F)C2)cnc2ncccc2c1 75569,N1(C(=O)NCC=CC=CC)Cc2nc(O)nc(O)c2C1 75570,C1(CC)CN(Cc2cc(O)ccc2Cl)c2ccccc2O1 75571,N1(C(CC(C)(C)F)=O)CCCC(O)(CNC(c2ccc(C(C)(F)F)cn2)=O)CC1 75572,C12(NC(C(N3C(CC)CCC3)=O)=O)CCCC1(F)CN(C(n1cnc(=N)[nH]1)=O)C2 75573,N1(C(C2(CCC)CC(=O)C2)=O)CCCC(CCC(=O)NCc2ccc(C)cc2)C1 75574,CN1CCN(CCc2nc(-c3cccs3)nn2CC2CCOCC2)CC1 75575,Cc1cccc(NNC(=O)C2(n3cc(N(C)Cc4ccccc4)nn3)CC2)c1Br 75576,c1(C(=O)NC2(C3N(C(C(C)OCC)=O)CCC3)CC2)ccc(CC)c(O)c1 75577,n1(CC(C)NC(=O)C(C)NC(=O)OC)cc(C(C)(C)NC(c2ccccc2)=O)nn1 75578,N1(C(C(C)CCO)=O)CCC(C)(NC(=O)COc2cccc(F)n2)CC1 75579,C1(N(C(=O)CS(C)(=O)=O)C)CN(C(=O)CSCCC#N)CC12CC2 75580,N12CC3CC1CCC3NC(=O)C=CC2=O.c1(NCO)ccccc1.C12(CC1)C(=O)N2.CCCC.CC 75581,N1(C(C2(COC)CCCCC2)=O)CC(C2CCCN(C(=O)C(C)S(N)(=O)=O)C2)C1 75582,C1(C(N(C2CCN(C(C(CC)(C)C)=O)CC2)C)=O)(CF)CC2(CCC2)C1 75583,c1(C(=O)NC2C(NC(=O)CCc3ccoc3)CC2)ccn(-c2ccncc2)n1 75584,C(=O)(CCC(C)SC)NC(C(=O)NCc1snc(CC)n1)C 75585,c1(NC2CC(CNC(C(C)CC(N)=O)=O)C2)nc2c(cc1C#N)CCC2(C)C 75586,N1(C(CCC(C)OCC)=O)CC(NC(c2cc(OC)n[nH]2)=O)CC(C)C1 75587,CC1CCC(C)(C)N1C(C1CC(NC(c2csc(Cl)n2)=O)C(O)C1)=O 75588,C(=O)(CC1=NNC(=O)C1)NC(C1CCCN(C(=O)CN2CCCNC2=O)C1)C 75589,N1(C(C2C(C)CC2)=O)CCOC(C(N2CCCC2C(N)=O)=O)C1 75590,CC(C)CC(CNC(=O)C(c1cccnc1)O)NC(c1cccc(CO)c1)=O 75591,CC(C)CCN=C(NCC1(C)CCOC1)NCc1ccc(N2CCOCC2)nc1 75592,c1(C(N2CC3(CCN(C(C(C)OCCOC)=O)C3)C2)=O)nc2nccc(C)n2n1 75593,C(CN=c1cc(COC)nc(C)[nH]1)N1CC(C)N(CC)C(C)C1.C1C(=O)N1 75594,c1(OC)cc(C(F)(F)F)nc(N2CC(NC(=O)CC3CC(C)OC3C)CC2C)n1 75595,Cc1cc(=NCC(CC(C)C)ON2CCCC2)[nH]c(Cl)n1 75596,C1(CNC(c2oc(CC)c(C)c2)=O)COC(C)(C)CN1C(=O)CN1CCCC1=O 75597,N1(C(C2C(C)(Br)C2)C(=O)NCC2CC2)CCC23CCCCC2(C1)C3(F)F 75598,c1(C(NC(=NCCCC)NCCCC2(O)CCC2)C)ccc(S(=O)(=O)CC)cc1 75599,C1(C(N(C(C)CCNC(c2cnsc2)=O)C)=O)C2CC2CN1C(=O)OC(C)(C)C 75600,C1(CNC(=O)C(c2ccc(F)cc2)CO)CCC12CCN(C(C1CCC1)=O)CC2 75601,CC(CS(C)(=O)=O)C(=O)N1CCC(Cn2cc(CN3CCOCC3)nn2)C1 75602,C1(CNC(CCC(C)SC)=O)CN(C(=O)Cc2ccnn2C)C2CCCCC12 75603,Nc1cc(C(=O)NCC23CC(NC(=O)C(O)CN4CCCC4)(CO2)C3)ccc1F 75604,C(=O)(CC(C)C(C)(C)C)OCc1ncn(CC(=O)OC)n1 75605,CC1CN(C(c2ccc(Cl)[nH]2)=O)CCN1C(C1CC(CC(F)F)C1)=O 75606,C1(NC(COC)=O)CC2(C1)CN(C(=O)CNC(c1ccc(Br)cc1)=O)C2 75607,c1(C(=O)NCC2N(C(c3cccc(C)c3C)=O)CC(O)C2)cc2c[nH]cnc-2n1 75608,Cc1cccc(CNC(=O)CCCCN(C(C2C=CCCC2)=O)C2CC2)c1 75609,C(=O)(CC(O)CC(C)C)N(CCCCC(=O)NCc1cnc(CC)[nH]1)C 75610,c1(CNCc2nc(C(C)(C)C)sc2)cc(I)ccc1F 75611,C12(CNC(C(C)(C)SC)=O)CC(CCO1)N(C(=O)Cn1cnnc1O)C2 75612,C1(NC(C2(NC(C3CC(=C)C3)=O)CC2)=O)CN2CCC1(F)CC2 75613,C(c1cccs1)=C(C)C(=O)N(C(C)CNC(=O)CCn1ccnn1)C 75614,N1(C(C2=CCCCC2C)=O)CCN(C(=O)CCc2cncnc2)C2(CCC2)C1 75615,Nc1nc(C(=O)NCCCCNC(=O)C2=NNC(C(F)(F)F)C2)ccc1[N+](=O)[O-] 75616,N1(C(CCCC#CC)=O)CC(NC(c2ccc(OC)nc2C)=O)CC12CCOC2 75617,Cc1nnc2n1C(C(=O)NC1CC(NC(C3CC3c3ccc(F)c(F)c3)=O)C1)CC2 75618,N1(C(Cc2cccc(OC)c2)=O)CCCC(NC(C2CC(N(C)C)C2)=O)CC1 75619,Cc1ccc(NC(=O)CNC(=O)CNC2CC(=O)N(C)C2=O)cc1C 75620,c1(OC)cc(=O)n(C)cc1C(=O)NCC1(F)CN(C(C2CC3CCC(C2)C3)=O)C1 75621,C1(NC(=O)CC2CC(F)(F)C2)CC2CC1CN(C(c1cccc(CO)c1)=O)C2 75622,N1(C(C2N(C)CC(C)(C)C2)=O)CC2CCCC1C2CNC(=O)CCC(C)(F)F 75623,N1(C(C(COC)OC)=O)CCC(CO)C(NC(c2ncc(F)c(OC)n2)=O)C1 75624,C1(CNC(=O)CC2CCCC2(F)F)CC2(CO1)CN(C(c1cccc(=O)o1)=O)C2 75625,C1(C(=O)NC(C2CN(C(=O)C(n3ccc(C4CC4)n3)C)C2)C)CCCC1(F)F 75626,c1(C(N2C3C(NC(C4CCCN4C4CC4)=O)CC(C3)C2)=O)ncnc2c1CCCC2 75627,CCCC(C)(C)CC(=O)NC1CCSC12CN(C(c1cc(F)ccc1NC)=O)C2 75628,N1(C(C2CC(CCC)C2)=O)CC(NC(=O)Cc2ccc(F)cc2Cl)CCC1C 75629,N(C1CCc2ccccc21)C(CC(C)CNC(c1nsnc1O)=O)=O 75630,C1(C(=O)NC(CNC(c2cnc(C(C)OC)s2)=O)(C)C)CCc2n[nH]c(C)c2C1 75631,CS(=O)(=O)C1CC(CN)C1.C1(=O)C(F)(F)C2(CCC2)N1 75632,c1(C(C)C)cccc(F)c1C(=O)NCCC(C)NC(c1cnc(Cl)[nH]1)=O 75633,C1(CCNC(C2C(C)(C)CC2)=O)(NC(C2CCC=CCC2)=O)CCOCC1 75634,c1(C(N2CC(OC)C(NC(=O)Cn3cnnc3O)C2)=O)coc2c1C(O)CCC2 75635,c1(N2CCC(N3CCCC3)CC2)nc(N2CCN(C3CC3)CC2)c2c(n1)CCS2 75636,C(=O)(C(C)(C)COCC)NC12CC(NC(CCC)=O)(C1)C2 75637,C1(NC(c2cnn(CCN(C)C)c2)=O)CCCN(C(C2(CF)CC2)=O)CC1 75638,C1(CC(=O)NCCC2N(C(CCC(=O)N(C)C)=O)CCCC2)CCCCC(=O)N1 75639,N1(C(C2CCCN(C)C2)=O)CCC2(C=C(C(=O)NC(c3cscn3)CO)C2)C1 75640,Cc1cn2nc(C(=O)NCCCNC(c3n[nH]cc3C)=O)cc2c(=O)[nH]1 75641,N1(C(CC2N(CC)CCC2)=O)CCN(C(C2(F)CCC2)=O)CC1c1nccn1C 75642,CC(CN=c1[nH]c2c(c(=NCCc3cnccn3)[nH]1)CCC2)c1ccc(Br)cc1 75643,c1(C(N2C(C)CCC(NS(CC)(=O)=O)C2)=O)ccc(Cl)c(OC)c1F 75644,c1(CCC(=O)NC(C)(CNC(=O)C=Cc2cn[nH]c2)CO)cccc(O)n1 75645,C(=O)(CC1=NNC(=O)C1)N(CCCCCCNC(c1c(OC)cc(Cl)cc1)=O)C 75646,c1(C(=O)NC(CCNC(C(C(C)C)C)=O)(C)C)ccnc2ncnn12 75647,Cc1cnccc1-c1ccc(-c2nccn2CCN(C)C)s1.c12nccn1CO2 75648,CC(C)C(O)CC(=O)NCC1CCN(CCOc2c(Cl)cccc2Cl)CC1 75649,C1(C(C)C)(C(=O)NC(C)CC(N)=O)CCCN1C(C1CN(C(N)=O)C1)=O 75650,c1(NC2C3CN(C(C4(S(C)(=O)=O)CCC4)=O)CC2C3)ncnc2[nH]cnc12 75651,C(N(Cc1ccccn1)N1CCC(c2ccccc2)C1C)c1c(C)noc1C 75652,C1(NC(c2cnc(CC(C)C)[nH]2)=O)CCCC12CN(C(c1cc(Cl)ccn1)=O)C2 75653,C12(NC(C(C)S(N)(=O)=O)=O)CCCN(C(c3cnn(C4CC4)c3)=O)CC1C2 75654,C1(C(N2C3(CNC(C4(COC)CC=CC4)=O)CC(C2)C3)=O)CCCCCS1(=O)=O 75655,Cc1ccc(F)c(C(=O)NCC2(CNC(=O)CC3CC=CC3)CCC2)c1 75656,N1(c2c(OC)cncn2)C2CCC1CC(NC(=O)C=Cc1scnc1C)C2 75657,c1(C(N(CCN(C(=O)CC(C)C2CCCO2)C(C)C)C)=O)nc2cnccc2s1 75658,c1(C(=O)NC(CCOC)CNC(=O)CN2CC(=O)NC2=O)ccc(Cl)nc1OC 75659,C1(C(N(C)CC=CC(N2CC(N(C)CCO)C2)=O)=O)CC(=O)C12CCC2 75660,C(=O)(C1SCCc2sccc21)NCC(CN(C(C(C)c1ccsc1)=O)C)(C)C 75661,c1(C(=O)NC2(CNC(c3ncoc3C3CC3)=O)CCCC2)ccc2nc[nH]c2n1 75662,N1(C(Cc2cccc(C)c2C)=O)CC2(CCC(CNC(=O)C(C)N3CCC3)O2)C1 75663,C=CCCCCC(=O)N1CC(CCNC(=O)CN2CCC(C)C2)C1 75664,C1(NC(C(F)=C(C)C)=O)CCN(C(=O)CN2CCN(C)CC2)C1C(C)C 75665,c1(CN2C(CC(N3CCC(Br)C3)=O)CCC2)ccc2ncsc2c1 75666,C(=O)(CC(C)C(=O)NC1CN(C(c2cn(CC(F)(F)F)nn2)=O)CC1(C)C)OC 75667,Cc1c(C(=O)NC(C2CCN(C(=O)CCOCC(C)C)C2)C)nn(C)c1C1CC1 75668,c1(N2CCC(CC)(CO)C2)ccc(Br)c(S(=O)(=O)NC(C)C(C)(C2CC2)OC)n1 75669,C1(C)(C(N2C(C3(NC(C4C(C=C)C4)=O)CC3)CCCC2)=O)CCN(C)C1=O 75670,N1(C(C(C(C)C)O)=O)CCN(C(C2CCC(O)CN2C)=O)C(CCO)C1 75671,c1(C(=O)NC2CN(Cc3cnc(Cl)cn3)CCC2(F)F)cc2ccc(Br)cc2s1 75672,C(N=c1[nH]c(N2CC=C(C)CC2)nc2c1CCCCC2)c1c(OC)c(Cl)ccc1 75673,C(C)(C)(CCN=c1[nH]c(N(C)Cc2nccn2C(F)F)nc2c1SCC2)OC 75674,C1(F)(CNC(CC)=O)CCC(CNC(c2sccc2-c2ccc(F)cc2)=O)C1 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75693,C1(NC(C2CCCCO2)=O)CN(C(c2ccc(C(F)F)o2)=O)CC12CCC2 75694,CN1CCN(C(c2ccccc2C2(C)CC2)=O)C(CNC(c2c[nH]nc2Cl)=O)C1 75695,c1(NC(C(CO)NC(c2cnc(OC)nc2)=O)=O)ccc(C#N)cc1O 75696,S(=O)(=O)(c1nc(N2CCC=C(Br)C2)ccc1Br)N1CCC(COCC)C1 75697,c1(CC(=O)NCC(C)NC(c2cc[nH]c(=NC)c2N)=O)ccc2c(c1)CCOC2 75698,c1(C(N2C3CN(C(C4C(OC)CC4)=O)CC2CC3)=O)c([N+](=O)[O-])c(C)nn1C 75699,C12(C(=O)NCc3c(C4CN(C(c5ccn(C)c5)=O)C4)ocn3)CCC(CC1)C2 75700,CC(C)CCCC(=O)N1CCCCC1CCNC(=O)CC1CCN(C)C1 75701,C(CN=c1nc(NCc2ccsc2Cl)c2c([nH]1)c(C)nn2C)c1ccc(C)cn1 75702,c1(CCC(=O)NC(C(=O)N2CC(N(C)CC)C2)CO)cccnc1 75703,c1(C(N(CCC(C)NC(c2ccc(CCC)s2)=O)C)=O)ccn(C)c1C1CCC1 75704,C(=O)(C1=NN(C(C)C)C(=O)CC1)NC1CCN(C(C(CC#C)O)=O)C1CC 75705,C(=O)(C(C)(C)CNC(C1CCN(C(=O)COC2(C)CCC2)C1)=O)NC 75706,CCC(C)(CCC(C)C)C(=O)N1CC(O)CC1C(=O)NCc1cccc(Cl)n1 75707,N1(C(C2(CCOC)CC2)=O)CC(CNC(=O)CC2CCCO2)OC(C)(C)C1 75708,C(=O)(CCC(C)CN(C)C)NC1CC(C(=O)Nc2c(COC)ccnc2)C1 75709,c1(C(N2CCN(C(CCOC)=O)CC2CC#N)=O)cccc([N+](=O)[O-])c1OC 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75763,c1(C(=O)NC(CCOC)CNC(=O)C=CSC)cn(C)c(=O)c2ccccc12 75764,C1(CC(=O)N(CCN(C(=O)CC(C)n2cccc2)CC)CC)CCCC(F)(F)C1 75765,Cc1c(C(N2CC(C3(N(C(=O)CN(CC(C)(C)C)C)CC)CC3)C2)=O)cncc1Cl 75766,N1(C(CSCC=C)=O)CCC2OCCN(C(c3cc(C)cnc3C)=O)C2C1 75767,Cc1ccc2cccc(C(=O)N(c3cc(O)ncn3)CC3CCNCC3)c2n1 75768,N1(C(CCCCNC(N)=O)=O)CC(C2CCCN(C(c3ccc(F)cn3)=O)C2)C1 75769,c1(C(CNC(c2coc(Cl)n2)=O)NC(=O)CC2(F)CCC2)ccccc1F 75770,Cc1nc(C)n(CCC(N2CCC(N(CCO)C(C3CC(C)(C)O3)=O)C2)=O)n1 75771,C1(NC(CC2(CC(=O)OC)CC2)=O)CCCN(C(c2ncc(OC)cc2F)=O)C1C 75772,C1(C(=O)NC2(C(=O)NCCSCc3nncs3)CCOCC2)CN2CCC1CC2.OC 75773,C1(OCC)(CNC(CC(c2ccncc2)(F)F)=O)CCN(C(=O)OC(C)(C)C)C1 75774,C1(C(N2CC(C(C)C)OCC2)=O)CC(C)CN(C(=O)C(C)(C)CC#N)C1 75775,c1(C(=O)NCC(C)N(C)C(C2(c3ccnn3C)CC2)=O)[nH]nnc1C1CC1 75776,N1(C(C2(SC)CCC2)=O)CCCN(C(C2CCN2S(C)(=O)=O)=O)C(C(C)C)C1 75777,N1(CCNC(C=CCN(C)C(c2cnc(Cl)s2)=O)=O)CCCOC1=O 75778,C#CCC(CC(=O)NCC1(CCO)CCCC1)NC(C1(C)C=CCCC1)=O 75779,Cc1n[nH]c(=NCC2CC(C)N(C(c3cc[n+]([O-])cc3)=O)C2)s1 75780,S(=O)(=O)(c1cc(C(F)(F)F)cc(Br)c1)Nc1ncc(-c2ccc(C)cc2)s1 75781,Cc1cc(Br)c(F)cc1CN1CC2C(C1)N2C(=O)C(C)(C)CCl 75782,C1(CC)CN(C(=O)CC2CC3(CC3)CO2)CCC1NC(=O)CS(=O)(=O)NC 75783,c1(C(=O)NCCCC(C)NC(C2(O)CC(c3ccccc3)C2)=O)ccc(Cl)cc1 75784,Cc1ccc(C(c2nnnn2C(C)C)NCCCCc2ccccc2)cc1Br 75785,c1(C(=O)NCC2(COC)CN(C(C3CC3C3CCCO3)=O)C2)cc(C(F)F)[nH]n1 75786,n1(CC(=O)NC2C(NC(C(c3ccccc3)OC)=O)C2)cc(SC)nn1 75787,CC1CCCC=C1C(=O)NC1CN(C(C2CCC(C)(C)CC2)=O)CC1CO 75788,N1(C(CCC=C)=O)CC2CCC1CN2C(=O)CCc1cc(F)c(F)c(F)c1 75789,N1(C(C(C)=CC2CC2)=O)CC(CNC(c2c(C)ncnc2C)=O)CC(C)(C)C1 75790,Cc1cnc(C(=O)NC2(CC(=O)N(C3CCC(C)C3)C)CC2)c[n+]1[O-] 75791,C=CC(C)(C)C(=O)N(CCC)CCNC(C1CC1Cl)=O 75792,c1(C(N(C(CCNC(c2nn(CC)c(=O)cc2)=O)C)C)=O)cc[nH]c2nccc1-2 75793,C1(NC(CCC2C(C)(C)C2)=O)CCC(NC(=O)C(O)C2CCCC2)CC1 75794,C1(CNC(CC2(CC(=O)OC)CCCC2)=O)CCC(F)(F)C(=O)N1 75795,c1(C(N2CCC(NC(CC=CCC)=O)C(F)C2)=O)c(C)cc(Br)cc1C 75796,c1(C(=O)NC(CC)CNC(C2(C)CCCC2)=O)ccc(C(=O)N(C)C(C)C)cc1 75797,Cc1cccc(C(N2CC(F)CC2CC(=O)NCCC(N)=O)=O)c1C#N 75798,N1(C(C(C(C)C)SCC)=O)CC(C)(C(=O)N(CC(=O)NC)C(C)C)CC1(C)C 75799,C1(C)(C(=O)NC2C(OC)CN(C(c3cc(C4CCC4)on3)=O)C2)CCCNC1=O 75800,N1(C(CC2CC(CC)OCC2)=O)CCN(C(C2(C#N)CC=CC2)=O)CC1CCO 75801,C(=O)(CCCCCNC(C1CC(C)CO1)=O)NCCCSC 75802,CC1(NC(c2conc2-c2ccccc2)=O)CCN(C(c2csc(=N)[nH]2)=O)CC1 75803,S1(=O)(=O)c2ccc(cc2)N1.N1(C(C)CO)CC2(CCC2)C1C(=O)NC1CC1 75804,C(C(C(C)C(C)C)NC(c1cccnc1C(F)(F)F)=O)NC(CNC(C)=O)=O 75805,c1(C(=O)NCc2cccc(NC(C3(C)C(C)OCC3)=O)c2)ccc(CO)c(Cl)c1 75806,Cc1cc(C(=O)N(CC(=O)NCCCOC(F)(F)F)CCOC)c(C)[nH]1 75807,CC(C)(CCCN=c1nc(N2CCC(C3(O)CC3)CC2)cc[nH]1)N1CCOCC1 75808,N1(C(c2c(C)cc(CC)o2)=O)CCCN(C(=O)C=Cc2cnccc2C)C(C)C1 75809,C1(C(=O)NC(C=C)C)CN(C(=O)CC(C)CCC)CC12CC2 75810,c1(SC)cc(C(=O)NCC(C)CNC(c2ccc(C(C)C)o2)=O)ccc1F 75811,c1(C(c2nnnn2C)NCc2cnc(C)s2)ccc(Cl)c(C(F)(F)F)c1 75812,Cc1n[nH]c(=NCC2CCN(C(=O)CCCOc3cccnc3)CC2C)o1 75813,C1(C(=O)NCc2c(C(=O)NCC3CCC=CO3)[nH]cc2)CC2(CCC2O)C1 75814,c1(C(=O)NCC(CC)NC(=O)CC2CCn3cncc3C2)cc(Cl)c(O)cc1C 75815,C1(O)(CCNC(CC2C(C)C2)=O)CCN(C(c2ccc(N)cn2)=O)CC1 75816,c1(C(N2C(CN(C(CC(=C=C)C)=O)C)CCCC2)=O)ccc2c(c1)CCO2 75817,C=C(Cl)C(C)(C)C(=O)N1CCCCC(NC(=O)C(C(C)C)NC(=O)COC)C1 75818,Cc1csc(C(=O)NCCn2ccc(C(=O)N(CC3=CCSC3)C)c2)c1 75819,N1(C(c2c(C)nn[nH]2)=O)CC(NC(C2CCCN2c2nccs2)=O)C2CC2C1 75820,c1(C(N(CC(CNC(c2nn(CC)c(C)c2)=O)C)C)=O)[nH]cc2c1CCS2(=O)=O 75821,c1(C(N2CCC(CN(C)C(c3ccn(C(F)F)n3)=O)C2)=O)cc2cnn(C)c2s1 75822,C1(C(N(C(CC)C(=O)NCCCNC(C)=O)C)=O)CCC(C)(C)C1 75823,C1(NC(c2c(CC)nc[nH]2)=O)CC2CC1N(C(=O)CCc1ccon1)C2 75824,c1(C(N(CC(C)NC(c2c(Cl)ccc(C)c2)=O)C)=O)cccc2cnnc(O)c12 75825,c1(C(=O)NCC(CNC(CSCC)=O)O)c(C)oc(C)c1Br 75826,c1(C(=O)NCC(C)(C2CC2)NC(c2cc(CO)[nH]n2)=O)cc2n(n1)CCO2 75827,C(c1c(C)noc1C)=CC(=O)NC(CC)(C)CCNC(=O)C(C)=C(C)C 75828,c1(C(N2C3C(NC(C(CC=C)C)=O)C(C3)C2C)=O)cc(C)c(F)cc1F 75829,C1(CNC(c2scc(C)c2C)=O)CN(C(=O)CCc2nc(O)n[nH]2)CCC1(F)F 75830,c1(CNC(=O)COC(F)F)cnn2c1CN(C(=O)CC1C=CCCC1)CC2 75831,c1(C(N2CC(F)CC(NC(CSCC=C)=O)C2)=O)ccnc(S(N)(=O)=O)c1 75832,C(=O)(C(O)C1=CCCCC1)NCC1(F)CN(C(c2ccc(C(N)=O)o2)=O)C1 75833,c1(CNCC2(NC(=O)Cn3ccnn3)COC2)c(F)cc(I)cc1F 75834,N1(C(c2oc(CC)c(C)c2)=O)CCC2(CC1)CC2CNC(c1csnc1OC)=O 75835,N1(C(c2c(C)cc(C3CC3)nc2)=O)C2CCC1CN(C(C1CCCCN1C)=O)C2 75836,c1(C(=O)NC(CC=C)CNC(=O)Cn2ccnc2C(C)C)ccc(C)cc1SC 75837,C1(C(N(CCCN(C(C2(CC#C)CC2)=O)C)C)=O)CCCCC1c1nncn1C 75838,C1(C(N(C2CCC2)CC)=O)CC(C)N1C(=O)CCc1cncnc1 75839,C1(CCNC(Cn2c(C)ccn2)=O)CC(F)(F)CN1C(c1c[nH]cc1Br)=O 75840,C(c1cccc(F)c1F)=CC(=O)NCC1(O)CCN(c2ncccn2)C1 75841,C(=O)(CCCCC(C)C)NCC1(F)CC(NC(c2cccc(CC)c2N)=O)C1 75842,c1(OC)cccc(C2CCN(C(C3CCCSC3)C(=O)NC3COC3)C2)c1 75843,c1(CSC2(CC=C)CCN2C(c2ccccc2)C)cc(C)c(OC(F)(F)F)c(C)c1 75844,CC12CCC(C(=O)NCC3(O)CN(C(=O)CC4CCCC45CC5)C3)(CC1)C2 75845,C(CCC(C)C)(C(=O)NC1CCC2CC1CO2)NC(C(C(CC)C)=O)=O 75846,CC1CC(NC(=O)Cc2cnoc2)CCN1C(C1OCCO1)=O 75847,CC(CNC(C1C(C)C1C)=O)C(=O)NC(C)C(C)F 75848,CCC(CC(=O)N1CCC1CNC(c1ccc(C(C)=O)s1)=O)C1CC1 75849,N1(C(CC=CCC)=O)CC(NC(=O)C(C(C)C)N2CCCC2=O)C2(CC2)C1 75850,c1(C(N2CC3(C)CC2(C(=O)NCCC2CCSC2)C3)=O)ccc2n[nH]cc2c1 75851,C(=O)(CCCC(C)(F)F)NC1(CNC(c2nn(C)c(=O)cc2)=O)CCOCC1 75852,c1(C(N(CC(C)NC(c2c(C)nc(C(C)C)o2)=O)C)=O)cc(Cl)c(F)cc1O 75853,CC1(C)CC(CNC(c2cn3cnnc3cn2)=O)CN(C(=O)COCCCF)C1 75854,c1(C(=O)NCC(CCCC)NC(=O)CC2CSCCS2)cccc2scnc12 75855,c1(C(N2CC(CC(=O)Nc3nccc(Br)c3Cl)OCC2)=O)cc(F)c(F)cc1O 75856,N1(C(C(C)=C2CCC2)=O)CC(O)CC1C(=O)NCC(c1ccccc1)C1CC1 75857,CC1CC(NC(C2(Nc3ccccc3)CC2)=O)CCN1C(C12CCCC(C1)OC2)=O 75858,CCC(C)C(O)C(C)C(=O)Nc1cccc(NC(C2(OC(C)=O)CCCC2)=O)c1 75859,c1(C(N(CCNC(C2CC(=O)N(C)C2)=O)CC)=O)cnc2c(C)cccn2c1=O 75860,N1(C(CC2(C)CCN(C(c3cccc(F)c3)=O)C2)=O)CCC2CCCC(C2)C1 75861,C12(C(=O)NC(C)CCCCNC(C3CSCC(=O)N3)=O)CCC(C1)C2(C)C 75862,c1(C(N2C(CCNC(c3ccc(C)o3)=O)CSCC2)=O)ccc2c(c1)OCO2 75863,C1(CC(=O)NCCOCCOCCNC(C2(F)C(C)C2)=O)COc2ccccc2O1 75864,N1(C(c2cncc(Br)c2)C(=O)NCC=C)CC(C)(C)c2ccccc21 75865,CC1C(NC2CC3(CC3)C(=O)O2)CCCC1CN 75866,N1(C(C(CC(=C)Cl)NC(=O)CCC2CCC2)=O)CCNC(=O)CC1C 75867,c1(C(N2CC=CC(NC(c3c(C)onc3Br)=O)C2)=O)ccc(Cl)c(N)c1 75868,c1(C(N2CC(C(C)(F)F)OCC2)=O)c(F)cccc1I 75869,CC1C(C)N(C(c2ccc(N)c(Cl)c2O)=O)CCN1C(C1C2CCC1CC2)=O 75870,CC1=CCSC1C(=O)NCCC1CCCN1C(=O)CC1CNC(=O)O1 75871,C#Cc1cc(C(N2CC(CO)(NC(=O)C3=C(C)CCCC3)C2)=O)cc(N)c1 75872,C1(NC(C#CC(C)C)=O)CC2CC1CC2C(N1CCOC(CF)C1)=O 75873,c12ccc(cc1F)C(=O)NNCc1cn-2nn1.N1(C(C)C)CCOCC1C1CC1 75874,c1(OC)cc(C(=O)NCC2(O)CC(CNC(C3(OC)CCSC3)=O)C2)cc(Cl)c1 75875,Cc1cc(Cl)c(C(=O)N(CC(O)CN(C)C(c2cnc(O)c(F)c2)=O)C)cc1F 75876,N1(C(=O)COC2CCCCC2)CC2CCN(C(c3c(F)ccc(O)c3F)=O)CC2C1 75877,C12(C(=O)NC3CN(C(C4(C(=O)OCC)CC4)=O)CC3C)CCOC1CC(=O)NC2 75878,c1(C(C(=O)NCC(C)NC(=O)C=Cc2ccoc2)O)ccc(Cl)c(Br)c1 75879,C=CCCCCCN(C)C(=O)NC1(c2ccccc2)CCCCO1 75880,c1(C(N2CCCCC(CNC(c3cnsn3)=O)C2)=O)cc(Cl)c2[nH]c(O)nc2c1 75881,c1(C(=O)NC2C(C)N(C(c3nc(O)sc3C)=O)CC2)ccc2c(c1)nc(O)n2C 75882,c12ccccc1C(=O)NC(C)CNC2=O.N1(C(c2cc(Cl)c[nH]2)=O)CCOCC1 75883,N1(C(C(C)NC(C)=O)=O)CCCCC1C1CCCN1CC(C)Nc1ccccc1 75884,C(=O)(CC1=CCCCC1)NC1CC(CCNC(C(C)(F)c2ccon2)=O)C1 75885,CCCCC(CNC(=O)CN1CCN(C2CC2)C1=O)NC(=O)CC1CC(OC)C1 75886,CC1CCc2[nH]c(=NCC(C)(C)CCN(C)C)[nH]c(=NC3COCC3F)c2C1 75887,C(CC(=O)N(C)CCNC(C12COCC1C2)=O)(C1=CCCC1)OCC 75888,N1(C(c2cc(C)[nH]n2)=O)CCC2(CC1)CC2NC(=O)C(C1CC(F)(F)C1)O 75889,Cn1cc(C(=O)NCC2(NC(=O)CC3CCC(C#N)C3)CCC2)c2ccccc12 75890,C1(C(=O)NCCN(C(c2cnc(C)cc2Cl)=O)CC)CCC2(CCOCC2)O1 75891,N1(C(CC2C(C)CCO2)=O)CCC(CNC(C2CCCCN2C)=O)CC1 75892,c1(C(=O)OC(C)C(N2CCN(C(C3CCOCC3)=O)CC2)=O)c[nH]c2ccccc12 75893,N1(C(CC(CCC)(C)O)=O)CCC2CCC(C1)N2C(C1(C)CCOC(C)C1)=O 75894,C#Cc1ccc(C(N2CCCC(CCNC(C3(CCO)CC3)=O)CC2)=O)nc1 75895,c1(COC)ncc(C(=O)NC2(C)CC(NC(=O)C(C)(C)c3ccno3)C2)c(=N)[nH]1 75896,c1(C(=O)NCC(C)NC(=O)C=CC2CCCO2)cnc2cc(O)ccc2c1 75897,C(=O)(CCCC1CCNCC1)OCC(=O)NCC(C)C 75898,C1(NC(c2cnc[nH]2)=O)CC2CN(C(=O)CCc3ncc[nH]3)CCN2C1=O 75899,N1(C(CCCC(C)C)=O)CCCC2C(CCCN2C(c2ccnn2C2CC2)=O)C1 75900,C(=O)(CCC(C)OC(C)=O)NC1C(C(=O)NCC(=C)CC)CC1 75901,c1(C(=O)NC2(C)CN(C(C3C(C)CC3)=O)C2)cc([N+](=O)[O-])ncc1Br 75902,N1(C(CC(C)n2cccc2)=O)CCC2CN(C(C3CC4(C3)CC(O)C4)=O)CC2C1 75903,Cn1ncc(C(=O)CC2CCCC2)c1C(=O)NCC1CCC(NC(=O)C(N)=O)C1 75904,C(=O)(C(C)(C(C)C)NC(c1cc(Cl)cc(C(F)(F)F)n1)=O)OCC 75905,C1(CC(=O)N(C)CC2CCC(NC(c3cncs3)=O)CC2)CC2(CCC2)CO1 75906,N1(C(C(Cc2c(C)cccc2)C)=O)CC2CC1CCN2C(c1ccoc1C)=O 75907,CCCS(=O)(=O)CC(=O)NCCCN(C(C1(C2CCCO2)CCCC1)=O)C1CC1 75908,c1(-c2n(Cc3cccc(C)n3)nc(-c3nc[nH]n3)n2)c[nH]c2cccnc12 75909,Cc1cc(Oc2cccnc2)ccc1NC(C1CC12CCOCC2)=O 75910,c1(OC)noc(C)c1C(=O)NCCC(C)N(C)C(C12CCCCC1C2)=O 75911,N1(C(CC2N(C)CCC2)=O)CCC(C)(C)C(C(=O)NC2(C)CCCC(C)(C)C2)C1 75912,C(=O)(C#CC(C)(C)C)N1CCN(C)C1C(=O)NCCCN=[N+]=[N-] 75913,C(=O)(C1=CCCCCC1)NC(CCN(C(c1ccc(OC)c(Br)n1)=O)C)C 75914,C#Cc1ccc(C(=O)N(CC(=O)NC(C(N)=O)C2CCCO2)C)cc1 75915,C#CCC(CC#C)C(=O)NC1(CNC(=O)Cc2c(C)n[nH]c2C)CCCCC1C 75916,c1(CSC)cc(C(=O)NC(C)CC2CN(C(=O)CCC3CCCCO3)C2)sc1C 75917,C12(CS(N3C(c4onc(C(C)(C)C)n4)CCCC3)(=O)=O)CCC(CC1)CC2 75918,C1(NC(=O)C=CC2CCCC2)CCCCC1NC(C1C(F)(F)C12CC2)=O 75919,N#CC1(C(N2CCCC(NC(c3cccc4c3CCC4)=O)C2)=O)CC2(CCC2)C1 75920,c1(C(=O)NC2CCC(C)N(C(=O)CC3CCCCC3)C2)cc2cccnn2c1 75921,C1(OC)CCN(C(=O)CC(C(C)C)NC(C2CCCN2C2CC2)=O)CC1(C)C 75922,c1(C(C(N2C(C)CC(NC(c3cnc(Cl)s3)=O)C2)=O)=O)c[nH]c2ccc(F)cc12 75923,c1(C(=O)NCC2CN(C(C3COC(=O)O3)=O)C2)ccncc1Br 75924,Cn1cc(C(=O)NCC2(NC(C3CC4C=CC3C4)=O)CCC2)c(C2CCCO2)n1 75925,C12(CC)CN(C(=O)Cc3nonc3C)C(CNC(c3cc(C)nc(O)n3)=O)(C1)C2 75926,N1(C(C2(C)ON=C(C)C2)=O)CCN(C(c2ncn3ccccc23)=O)C2(CCC2)C1 75927,c1(C(=O)NCC(CN(C)C(C2CCSCC2)=O)O)ccc2c(O)nnc(O)c2c1 75928,Cc1nccnc1C(=O)N(C(CNC(=O)CC1CC(n2cnnc2)C1)C1CC1)C 75929,C12(C(N3CCCC(NC(=O)C=C4CCCC4)CC3)=O)CCCCC1C2(F)F 75930,CC(C)(C)CC(F)C(=O)N(C(=O)CN1CCCC(O)C1)CCc1ccccc1 75931,C=Cn1nccc1C(N1CC(F)CC1CNC(c1ccccc1)=O)=O 75932,C(=O)(CCCS(=O)(=O)N1CCCC1)N1CC(NC(c2cc(O)ncn2)C)C2C1C2 75933,CCC(C)(C)CC(=O)NCC1CC(NC(=O)C(c2ccccc2Cl)(C)C)C(O)C1 75934,N1(C(C2(C)CC3CC3C2)=O)CCCCC(NC(c2ncc(Cl)cc2Cl)=O)CC1 75935,n1(CC(=O)NC23CCC(C2)N(C(C2(S(N)(=O)=O)CC2)=O)C3)nc(C)ccc1=O 75936,c1(C(N2CC(NC(C(C)(Cl)Cl)=O)C(O)CC2)=O)c[nH]c2ccc(F)cc12 75937,N1(C(CCNC(=O)NCc2cnc(C(C)C)o2)=O)CC2CCC1C2 75938,CCCCC(O)C(C)C(=O)NC(CCC(=O)NCCn1cc(CC)cn1)C(C)C 75939,c1(C(=O)NCC2(C)CCN(C(C(COC)(F)F)=O)C2)ccnc2[nH]ncc12 75940,C(CN=c1[nH]c2c(c(=NCCOc3ccncc3)[nH]1)CSC2)C1(C)CCCO1 75941,N1(C(c2c(C)n(C)nn2)=O)CCC2C(C1)CN2C(c1cc(C2CCC2)nn1C)=O 75942,C1(NC(C(CC)CC(C)C)=O)CCCCC12CCN(C(=O)CSC(F)(F)F)C2 75943,Cc1cc(O)ccc1C(=O)NC1CC(NC(=O)CSc2ccncc2)CC1O 75944,Cc1c(CC(=O)NCC(C)NC(C2CCCN2C)=O)ccc(Cl)c1Cl 75945,C(=O)(C1=CCCCC1P(C)(C)=O)N(C(CNC(c1cc(OC)c(C)cc1)=O)C)C 75946,C(=O)(C(CCCC(=O)OCC)N(C1CCOC(C)(C)C1)c1ccccc1C)NC 75947,c1(C(=O)NC2CN(C(C3CC3(Cl)Cl)=O)CC2C(F)F)cnc(O)c2ncccc12 75948,c1(C(=O)NCC(CC=C)NC(=O)CCCCOC)cc(O)cc(F)c1F 75949,N1(C(C(C)N(C(C)=O)C)=O)CC2(C1)CN(C(C13COC(CS(C)(=O)=O)(C1)C3)=O)C2 75950,N1(C(c2ccc(SC)o2)=O)CCC(F)(C(=O)NCC2(O)CSC2)CC1 75951,c1(CC(C)=CC(=O)NCCOCC(N2CCOCC2)=O)ccc(C)c(C)c1 75952,[N-]=[N+]=NCCCC(=O)NCC1(C(N2CCC(N3CC(O)C3)C2)=O)CC12CCC2 75953,C1(C(=O)NCC(c2ccccc2)CNC(C2CS(=O)(=O)C2)=O)CCOC1=O 75954,C(CNC(=O)C1=CSCS1)(C(C)(C)C)NC(C(C)OCC)=O 75955,N1(C(C(CO)NC(N)=O)=O)CC2(CCCN(C(c3cc(C4CC4)on3)=O)C2)C1 75956,C#Cc1ccc(OCC(N2CC(NC(c3cnc(C)cc3C)=O)CC2C)=O)cc1 75957,c1(C(N2CCC(N(C(c3nc(C)nn3C)=O)C)C(C)C2)=O)cccn2ccnc12 75958,c1(C(=O)NC2CCC(CNC(c3c(C)oc(Cl)n3)=O)C2)cc(O)cc([N+](=O)[O-])c1 75959,c12cc([N+](=O)[O-])c(F)cc1N2.C(=O)(COCCCF)N(CCNC(C)=O)C 75960,C(CCCCCC(=O)NCC(C)N(C)C(c1ccc(C(F)(F)F)c(F)c1)=O)SC 75961,N(C(=NCc1c(F)cccc1Cl)N(C)Cc1n[nH]cc1Br)C(C=C)C 75962,c1(CC(N2CC(CC=C)(NC(=O)CSCCN(CC)CC)C2)=O)cc(C)sc1C 75963,C1(C(=O)NC2CCN(CCNC(C(C)c3cc[nH]n3)=O)CC2)CC2CCCCC12 75964,c1(N2CCC(=C)C2)ccn2ncc(S(=O)(=O)NC3CCC4CC34)c2n1 75965,c1(N(CC(N)=O)CC2(C)CCN2)ccc2ccccc2c1 75966,c1(C(=O)NCCC(C)NC(c2c(C)noc2C)=O)ccc2nc(O)[nH]c2c1 75967,C1(CNC(C(C)NC(C)=O)=O)CCN(C(=O)Cc2ccccc2Br)CC1 75968,C12(C(=O)NCC3C(C)CN(C(=O)Cc4cnn(C(F)F)c4)C3)CCOC(C)(C1)C2 75969,c1(CC(=O)NC2CCCC(NC(=O)OC(C)(C)C)C2)c(F)cc(F)cc1Br 75970,C1(CC(=O)NCCCCC(C)NC(=O)C=CC2CCC2)CCc2ccccc2N1 75971,c1(C(=O)Nc2cnc(Cl)c(C(F)F)n2)ccc(=O)n(-c2ccccc2F)c1 75972,c1(OC)nsc(C(=O)NC2(CNC(c3nnn(C)n3)=O)CCCC2)c1Br 75973,C#Cc1cc(C(=O)NC2CS(=O)(=O)CC2NC(=O)C(C)CC(F)(F)F)ccc1C 75974,N1(C(C2CC(C)OCC2)=O)CC2(COC(CNC(c3c[nH]cc3Br)=O)C2)C1 75975,c1(OC)cccc2c(CCNC(C3(c4ccc(F)cc4)CC(C)(C)C3)=O)c[nH]c12 75976,N1(C(c2ccc(CC)c(C(F)(F)F)c2)=O)CCCC2C1CCN2C(=O)C(C)OC 75977,C(=O)(C(C)CS(C)=O)NCC1(CNC(c2c(C)n[nH]c2C)=O)CC1 75978,C(CCC(C)C(=O)N(C1CCN(Cc2csc(Cl)n2)C1)C)OC 75979,C1(C(=O)NCC(CC(C)C)(C)C)CCN(C(=O)CCC(C)(C)F)O1 75980,CCC(O)C(C)(C)C(=O)NC1CC(NC(c2cc(O)ncn2)=O)C1 75981,C=Cc1cncc(C(=O)NC(Cn2cncn2)C(=O)N(C2CCOC2C)CC)c1 75982,CC(C)C(O)Cc1cn(CC2CCCC2NC(C2CCCOC2)=O)nn1 75983,C1(C(=O)NCCC2(NC(c3nc(C(C)OC)sc3)=O)CCC2)CC12CC(F)(F)C2 75984,C(=O)(C(C(C1CC1)OC)N(C(C)(C)CC(=O)NC)C)NCCC 75985,CC(C)(CC(F)(F)F)C(=O)N1CCCC(NC(C2Cc3nncn3C2)=O)CC1 75986,N1(C(Cc2nc(C)sc2)=O)CCCN(C(=O)CNc2ccccc2Cl)CCC1 75987,C1(C(=O)NCC(=C)C)CC(N(C(=O)CCC2CCC2)C)C1 75988,N1(C(C2CC2c2cccc(F)c2)=O)CC2CC1CN2C(C12CCC(CC1)C2)=O 75989,N1(C(CCc2cn(C)nc2)=O)CCCCCC1C(N1CC(CC2CC2)C1)=O 75990,c1(C(=O)OC)c(C)[nH]c(C)c1C(=O)C(C)ON(C(C)CO)C 75991,CCCCC(CNC(C1CC(F)(F)C1)=O)NC(=O)CNC(C)=O.C(C)(C)(C)O 75992,N1(C(CNC(CNC(CCC2(C#N)CCC2)=O)=O)=O)CC2CC1CS2=O 75993,c1(CN(C2CCCCC2)CC#C)nn(C)c2c1CC(F)(F)CC2 75994,C12(NC(C(CC)NC(C)=O)=O)CCC(CC1)N(C(=O)C=C1CCCCC1(C)C)C2 75995,C1(CCC(=O)NC(CC)COC)CCCCN1C(c1ccncc1O)=O 75996,c1(C(=O)NCC2(CNC(C(C(C)O)C)=O)CCOCC2)ccc2ccoc2c1 75997,c1(CN(C(=O)C=CC(C)NCC(C)(O)C2CCCC2)CC#C)ccco1 75998,c1(C(=O)NC2C(CNC(CC(CC)OC)=O)COC2)cc(C2(C)CC2)ccc1F 75999,N1(c2cc(OC)nc(OC)n2)CCC2CN(C(c3cc(SC)nn3C)=O)CC2C1 76000,C1(C)(C(N2CC(OC)(CO)C2)=O)CC(O)CN1C(=O)C=C(C)C(C)C 76001,N1(C(c2c(C)nsc2)=O)CC(NC(=O)COCc2nc[nH]n2)CC1C 76002,C(C(C)C(C)N=c1nc(N2CCC(CCO)CC2)c2cc(Cl)ccc2[nH]1)OC 76003,C1(C(N2CCC(C(N(CC)CC)=O)C2)C(=O)NC2CC2)CC(C)OC1C 76004,CC1CCN(C(=O)C(C2CN(C(=O)CCCC3CCCC3)C2)N(C)C)C1CO 76005,c1(C(=O)NCCC(=C)CNC(c2cccc(C)c2)=O)cn2cccnc2n1 76006,C1(NC(c2c(C)cccc2F)=O)CC(C2CCN(C(=O)Cc3csc(Cl)c3)C2)C1 76007,Cc1cccc2[nH]cc(C(=O)NCCN(C(=O)C(C)n3ccnc3)CC(C)O)c12 76008,C1(OC)CC(CNC(=O)C2=CCCS2)N(C(=O)CC2(C)CCCCC2)C1 76009,C1(NC(c2cn[nH]c2)=O)CN(C(c2cncc(-n3ccnc3)n2)=O)CCC1CO 76010,N1(CC)CCC(N=c2nc(N3CC=C(CO)CC3)c3c([nH]2)c(C)nn3C)CC1C 76011,N1(C(C2(C)COCCO2)=O)CC2CC(NC(c3ccn(CCF)n3)=O)C1C2 76012,c1(CCC(=O)N(CCC(C)NC(C(CC)(C)O)=O)C)nnc(O)nc1O 76013,Cc1cc(Cl)c(Br)cc1S(=O)(=O)N1CCc2scnc2C1 76014,c1(C(CNC(C(C)OCC=C)=O)NC(=O)CCN2CCCC2=O)ccccc1F 76015,N1(C(c2nnc(C)s2)=O)CC(O)C(O)C1CNC(=O)Cc1ccc(F)cc1F 76016,n1(CC(=O)NC(CNC(CC=C=C)=O)C(C)(C)C)nc(O)ccc1=O 76017,c1(C(=O)NCC2C(C)(C)CN(C(C3CC4C=CC3C4)=O)C2)nnc2ccccn12 76018,c1(CC)sccc1C(=O)NC(C1CCCN1C(c1cnco1)=O)C 76019,N1(C(CC2N(C(C3C(OC)CCC3)=O)CCC2)=O)CCC(CO)C(F)C1 76020,CC1CN(Cc2ncccc2Br)CCN1C(c1cc(Cl)cnc1O)=O 76021,N1(C(c2cnc(CC)nc2)=O)CCC(NC(=O)Cc2ccn(CC)n2)C12CC2 76022,c1(C(=O)NCC2CC(Nc3cc(C(F)F)ncn3)C2)cn2c(n1)COCC2 76023,c1(OC)ccc(C(N2CC(CCCOC)(NC(=O)COC(C)C)C2)=O)cc1Cl 76024,Cn1cc([N+](=O)[O-])c(=NCC2(CNC(c3ccc(SC4CC4)cc3F)=O)CC2)[nH]1 76025,c1(OCC)ccc2[nH]c(=NCC(C)NC(=O)C(C)COC)sc2c1 76026,N1(C(C2(CCOC)CC2)=O)CC2CCCC(C1)N2C(C1CCCC1S(C)(=O)=O)=O 76027,Cc1csc(=O)n1CCCC(=O)NC1CC(N(C)C(c2cc(Cl)cn2C)=O)C1 76028,N1(NCc2ncn(C)c2)CCC(NC(c2ccc3c[nH]nc3c2)=O)C(F)(F)C1 76029,C12(CNC(=O)CCn3cccn3)CCC1CCN2C(=O)CNc1ncccn1 76030,c1(C(=O)OCC)coc(NC(=O)CC2CCN2C(=O)C=Cc2cn[nH]c2)n1 76031,c1(CC=C)ccccc1C(N1CC2C(NC(c3coc(CC4CC4)n3)=O)C2C1)=O 76032,[N-]=[N+]=Nc1ccccc1C(=O)NC1(CF)CCN(C(=O)Cn2cccn2)C1 76033,C1(NC(C(CC)OCC)=O)CCC2CN(C(=O)C(C)Sc3ncccn3)CC2C1 76034,C1(NC(CCC(=C)C)=O)CCN(C(C2CCC(=O)C2)=O)CC(O)C1 76035,c1(C(C)C)ccc(F)c(C(=O)NCC2C3CC2N(C(=O)C(C)S(C)(=O)=O)C3)c1 76036,c1(C(=O)NCC2C=CCN2C(c2sccc2C(F)F)=O)ccc(OC(F)F)nc1 76037,C#CCC(C)(C)C(=O)NCC1(O)CCN(C(c2ncncc2N)=O)C1 76038,C1(NC(c2c(C)ncn2C)c2nnnn2CC(F)F)CCCCCCCCC1 76039,C12N(CC1(C)C)C(=O)CC1CCCC(C1)NC2=O.c1(C=O)cccnn1.CO 76040,N1(C(C2(S(N)(=O)=O)CCCC2)=O)CCC2(CC1)OCCC2NC(C1CCCC1)=O 76041,c1(C(N2C(CNC(=O)CC3CC4(CC4)C3)CCC2)=O)cc(O)ncn1 76042,C1(CNC(c2cc(C)on2)=O)CCCCN1C(c1cocc1C(N)=O)=O 76043,N1(C(Cc2nc(C)[nH]n2)=O)CCCCC1CCCNC(=O)C(F)CC1CC1 76044,c1(CC(N2CC(OC)C(NC(c3coc(C(F)F)c3)=O)C2)=O)ccc(C)c(F)c1 76045,N#CC12CCCCCC1CN(c1ccncc1S(=O)(=O)N1CCC(F)(C#N)C1)C2 76046,N1(C(c2c(CC)nnc(C)c2)=O)CC(NC(C2CN(CC)C2)=O)CC12CCOC2 76047,c1(C(=O)OCC)cnc(NC2(CNC(c3cccc(Cl)c3F)=O)CCC2)nc1C 76048,c1(-c2scc(C(=O)NC3C(CNC(C(COC)C)=O)C3)n2)ccc2c(c1)CCO2 76049,CC1(C)NC(=O)CCC1NC(C1CCN1C(c1ccn2ccnc2c1)=O)=O 76050,CC(CNC(=O)C(C)(C1CC1)N(C(=O)CC1NC(=O)NC1=O)C)C(C)(C)C 76051,Cc1cc(C(=O)NC2CN(C(c3csc(C(F)F)c3)=O)CCC2CO)cnc1O 76052,Cc1c(C(=O)NCC(CNC(=O)Cc2nc[nH]n2)CO)sc2nnc(S)n12 76053,C1(NC(c2c(CCC)cccc2)=O)CN(C(=O)CC2CC(OCC)C2)CC12CC2 76054,N#CC1CCC(NC(c2cnn(CCN(C(C3CCCN3C(N)=O)=O)C(C)C)c2)=O)CC1 76055,C1(CNC(C(C(C)O)C)=O)CN(C)CCN1c1nc(C2CC2)nc(=N)[nH]1 76056,c1(CN(C(C(c2cn(C)nn2)NC(Cn2c(C)nnn2)=O)=O)C)ccccc1F 76057,C12(CC)CN(C(=O)CC(C)OC)C(CNC(=O)CC3C(=O)NN=C3C)(C1)C2 76058,N1(C(c2nc(CCOCC)oc2)=O)CCC(NC(=O)CSCC(C)C)CC(O)C1 76059,c1(C(=O)NC2CCC(NC(C3(Cl)CC34CCC4)=O)C2)csc2cccnc12 76060,c12ccc(nc1)C(=O)NC2.n1(CC)ccnc1NC(=O)CC1CSCCO1 76061,N1(C(C(C(CNC(c2ccnc(OC)n2)=O)C)F)=O)CCc2nc(O)[nH]c2C1 76062,C(N=c1cc(N2CCOC(C)C2)nc[nH]1)C1(Nc2c(SC)cccc2)CCC1 76063,C1(C)(C(=O)NCC2CC(C(=O)NC(c3nc(C)on3)C)C2)CNC(=O)C1 76064,C(=O)(C(C)CS(C)(=O)=O)NCCC(C)CF 76065,CCCCCCNC(c1nnnn1CCOCCO)CC1CCOCC1.C(COC)S 76066,Cc1oc(C(C)C)nc1C(=O)NC1CCCCC1NC(=O)CNC(=O)C(C)(C)C 76067,Cc1ccnc(C(=O)N(C2CCC(NC(c3sc(Cl)cc3Cl)=O)C2)C)n1 76068,CC1C(C)N(C(C2CN(C)C2)=O)CCN1C(=O)CCNC(=O)Cc1ccccc1 76069,Cc1cccc(C(N2CCN(Cc3noc(C4CC4)n3)C(C)C2)=O)c1C 76070,N1(C(CN2C(=O)COCC2)=O)CCC2CCC(C1)N2C(=O)C(N1CCSCC1)=O 76071,N1(N(CC(=O)OC)CCOC)Cc2ncsc2C1.C1(C=O)CC(NC)C1 76072,Cc1cc2cc(C(=O)NCC3CC3CNC(C3CCC3)=O)oc2cc1C 76073,c1(C(N2C(C)CC(NC(C3CC(=C)C3)=O)C2)=O)ccc2c(c1)OCCC2 76074,c1(C(=O)NCCN(C(C2CCCC(C)C2)=O)CC)nc(OC)ccc1Cl 76075,N1(C(CSC(C)C)=O)CCCC1(C)C(=O)NCCC1OCCC1(C)C 76076,C12(NC(=O)CC3CCC34CCC4)CCCC(CN(C(c3cnsn3)=O)C1)C2 76077,CN1C(=O)C2CN(c3cc(C#N)ncn3)CC2C1=O 76078,C1(CC=C)(C(=O)NCC(O)CNC(C2(C(N)=O)CC2)=O)CCNC1=O 76079,C1(N(CC#C)C(c2ccc(C(F)F)o2)=O)CCN(C(=O)CCN(CC)CC)CC1 76080,CCCC(O)C(=O)N1CCC(NC(=O)CCCNC(C)=O)C1 76081,C1(CC(N2C(CNC(C3CCCC(OC)C3)=O)CC2)=O)CCn2cncc2C1 76082,N1(C(C(C)(C)n2cccn2)=O)CC(NC(=O)CCc2cc(Cl)cs2)C(C2CC2)C1 76083,N1(C(c2cc3ccoc3cn2)=O)CCCC2C1CCN2c1ncc(Cl)cn1 76084,C(=O)(C1c2[nH]cnc2CCN1C(=O)C(CSC)c1ccccc1)OC 76085,C1(C(=O)NCCCCO)CN(C(=O)CC2CCOC2=O)CC12CC2 76086,C1(=CC(=O)NCCC2(NC(C(C)OCC3CC3)=O)CCCC2)CN2CCC1CC2 76087,Cc1cc(NC(=O)CC2CCC(NC(=O)C(C)S)CC2)c([N+](=O)[O-])cc1Br 76088,CC(O)C(C(=O)N1CCCC1CNC(=O)C1=NOCC1)NC(=O)C(C)(C)C 76089,C1CC(C)CCO1.C(=O)(C(C)C)NCC(=O)N.C(C(=O)NN)SC.C1(=O)CN1C 76090,C1(NC(CC(C)N(C)C)=O)CN(C(=O)C(C)(C)n2ccc(C3CC3)n2)CCC1(C)C 76091,C1(C(N(CCCn2cc(CCCS(N)(=O)=O)nn2)C)=O)CCOC2(CCCC2)C1 76092,C1(F)(CC(=O)NCCNC(C(n2nnc(-c3ccccc3)n2)C)=O)CCCOC1 76093,N1(C(CNC(CC)C(=O)OC(C)(C)C)=O)CCc2nc(I)[nH]c2C1.C1CNC(=O)O1 76094,C(=O)(CCN=c1nc2c(ncn2C(C)C)c(NCCCCCSC)[nH]1)NCC 76095,C=C(C)C1CCC(C)(O)C(NC(=O)NCc2nc3cccc(F)c3o2)C1 76096,c1(CC(=O)OC(c2onc(C)n2)C)csc2nccn12 76097,C(c1cncn1C)=CC(=O)NC1CC(CC(=O)N(C)CC2CCOC2)C1 76098,C1(NC(C2CC(N(C)C)C2)=O)CCCC(NC(c2ccc(=O)oc2)=O)C1 76099,C1(N(C(N(C2CCCC2C#N)C)=O)CCOC(C)(C)C)CCCCCC1 76100,C(C(C)(CC(C)C)NC(c1cc(C(N)=O)on1)=O)NC(C(C)=CC1CC1)=O 76101,c1(NC(CC2CCN(C)C2)=O)cnn(C)c1-c1cn(CC2CC3CC3C2)nn1 76102,CN=c1[nH]cc(C(N2CCC(O)(C(C)CNC(c3cn(C(C)C)nn3)=O)C2)=O)o1 76103,c1(NC(C2N(C(C(CC)(C)O)=O)CC2)=O)ccc(=O)n(CCOC)c1 76104,CC#CC1CCN(C(=O)C=CCC2(NC(=O)Cc3ccn(C)c3)CCC2)CC1 76105,N1(C(Cn2ncc(S(N)(=O)=O)c2)=O)CCC(C2(NC(C3CCCC3)=O)CC2)CC1 76106,N1(C(CCCCC=CC)=O)CCC(C2CCN(C(C3CC3(F)F)=O)CC2)C1 76107,N1(C(C(CC)(C)COC)=O)CCC2(C=C(C(=O)NCC3CSCCO3)C2)C1 76108,NC(=O)CCC(N)C(=O)N1C(C(=O)NC2COC(=O)C2)CC2CC12 76109,C=CCC(CC(F)F)C(=O)N1CCCOC(CCNC(=O)C(=O)C(C)(C)C)C1 76110,Cc1c(C(=O)NCCCCN(C(=O)CC2CN(C)C2)C)cccc1Cl 76111,C=C(C)CCCC(=O)N1CCCCCC1CNC(=O)CC1CCCCN1C 76112,N1(C(c2cnc(C)nc2)=O)CCC2CN(C(c3cnoc3C3CC3)=O)CC2C1 76113,c1(C(=O)Nc2ccc(C(N3C(CCC=C)CCC3)=O)nc2)cnnc(C)c1C 76114,C(=O)(C1c2c[nH]nc2CN1C(C1CCCCN1C)=O)N(CCC(=O)NC)CC 76115,C1(NC(C=C(C)C(C)C)=O)(CO)CCCN(C(C23CCCC(C2)OC3)=O)C1 76116,C1(C(=O)NC(CCNC(C=C(CCC)C)=O)(C)C)CC2CCC(C1)C2O 76117,C1(C(=O)NOC(C)C(=O)OC)(CC=C)CCCN1C(c1ccc(C)cn1)=O 76118,C1(C(=O)NCC2(C)CC2)CC12CCN(Cc1cccc(Br)n1)CC2 76119,Cc1cnn(CCNC(=O)CC2(NC(C3CC(F)C3)=O)CC2)c1 76120,C1(Nc2ccc(C(=O)NC(=O)NCC)cc2)CC2CCCC2C1 76121,C1(C)(C(N(CCOC)CCn2cc(C3(CCO)CC3)nn2)=O)CC(C#N)C1 76122,c1(C(=O)NC2COCCN(C(C=CC(CC)C)=O)C2)cc2c(cn1)OCO2 76123,C#CC1(C(=O)NCCN2CCCC2)CN(C(c2cnc(O)o2)=O)C1 76124,C(=O)(CC(F)(F)Cl)NCC(C(C)C)NC(=O)CC1CC(C)(C)C1 76125,C1(OC)CCCC1.C1COCCOCCNC(=O)NCCS1 76126,CCC(C)(COC)C(=O)NCCC(C)CCNC(c1ccnn1CC1CC1)=O 76127,N1(C(C)C)CCC(CC(=O)N(C)CC2CCN(C(C3C(C)C3(F)F)=O)C2)CC1 76128,C12(C(N(CC(C)NC(=O)COc3ccccc3F)C)=O)CCC(C)(C1)OC2 76129,Cc1cc(C(=O)NC(C)CN(C(=O)C(c2ccc(Cl)cc2)CO)C)n(C2CC2)n1 76130,c1(C(C)(C)C)cc(C(=O)NCCC2(NC(=O)CC3CCCC34CC4)CC2)nn1C 76131,C(=O)(C1=CCN(C(c2cscn2)=O)CC1)NCC1C(C)CCCC1 76132,c1(NC2C(C)CN(C(=O)CCCC(=O)N(C)C)C2)ncc(Br)cc1[N+](=O)[O-] 76133,C(c1cn(C)nn1)=CC(=O)NC(C(=O)NC(CC=C)CC)CC1CCC1 76134,c1(C(=O)NCC2C(CC(=O)NCc3ncsn3)C2)cc(Cl)n[nH]1 76135,N1(C(C(C)C(F)(F)F)=O)CCCCCCC1C.C(CC(F)(F)Cn1ccnn1)N 76136,C1(C(N(CCCNC(c2ccc(C)cc2)=O)C2CC2)=O)CCC2CCC1O2 76137,N1(C(CC(C)c2ccccc2)=O)CC2CC(NC(=O)Cc3ccno3)C1C2 76138,N1(C(C(=O)Nc2ccc(C)cc2)=O)CCCN(C(c2cc(C)c(C)cn2)=O)CC1 76139,C(=O)(CCCC(=O)N1CC(CNC(=O)CCC(=O)c2cccc(Cl)c2)C1)N(C)C 76140,Cc1cnc2cccc(C(=O)NC(C)C(CO)NC(=O)CSCC(F)(F)F)n12 76141,N1(C(c2cn(CC=C)nc2)=O)CCC2(CC2C(N2CC(C(C)OC)C2)=O)C1 76142,N1(C(C2C(C)=C2)=O)CC(C)OC2(CCN(c3nc4cc(C)ccc4o3)CC2)C1 76143,C1(NC(Cc2n[nH]c(=NC)s2)=O)CC2CC(C1)N(C(C1(O)CCC1)=O)C2 76144,C=CCC(C)C(=O)N1CCC(C(F)F)(CNC(=O)CN(c2ccnc(Cl)n2)C)C1 76145,c1(C(=O)Nc2cc(C)c3c(c2)NC(=O)CO3)cc2c3ccccc3n(C)c2s1 76146,C(CC(C)(C)C(=O)NCC(CNC(=O)C(N1CCC(O)CC1)C)OC)OC 76147,C1(C(=O)NC(c2ccccc2)C(=O)NCC(CC)C#N)CCOCC1(C)C 76148,c1(C(=O)NC2C(C(=O)Nc3cncc(CC)c3)CCC2)ccc([Si](C)(C)C)cc1 76149,N1(C(C(CC)(C)O)=O)CCOCC(CNC(=O)CCc2ccn(C)n2)C1 76150,CCC(CCC(=O)NCCC(O)C(F)F)NC(C1SCCS1)=O 76151,c1(CC)cccc(C(N2CCCC(NC(C3CCC4(CCC4)C3)=O)CC2)=O)c1O 76152,CN=c1[nH]c(C(N2CC3C(CNC(C4(c5cccnc5)CCC4)=O)C3C2)=O)cs1 76153,c1(Cn2cc(C(C=C)(C)O)nn2)ccc(CNC(c2ccc(C(F)F)o2)=O)cc1 76154,C1(N(CC(=O)NC(c2cn(C)nc2)CO)C(n2cccn2)=O)CCC(C2CC2)C1 76155,O(NC(=O)C(F)C1(O)CN(C(c2cn(C)c(C)n2)=O)C1)CC(=C)Cl 76156,C1(C(N(CC(=O)NCC)C)=O)CCCCCN1C(C1CC(=O)N(OC)C1)=O 76157,Cc1cc(-c2ccc(N(C)C)cc2)nc(C(F)(F)F)n1 76158,c1(C(N(C2CCN(C(C(C(C)C)OC)=O)C2)C)=O)cc([N+](=O)[O-])c(C)cc1C 76159,c1(-c2nc(-c3ccc(OC)cc3)nn2C2CC2)cnc(OC)c(Cl)c1 76160,c1(CC)ccc(C=CC(=O)NC(CNC(c2ccc(O)nc2)=O)C(C)C)cc1 76161,C1(CNC(C(c2ccccc2)N(C)C)=O)CC2CC2N1C(=O)COC1CC=CC1 76162,c1(C(=O)NC(C(C)C)C(C)NC(c2ccc(N(C)C)nc2)=O)cn(C)c(=O)n1C 76163,c1(N(C)Cc2cccc(OC)n2)ncccc1S(=O)(=O)NC12CCN(CC1)CC2 76164,C12(C(=O)NCC(C)(CNC(=O)C(C)(C)OC(C)=O)OC)CCC(F)(CC1)CC2 76165,Cc1c(C(=O)NCC(CNC(=O)C(F)(F)CN(C)C)CO)cc(C(C)(C)C)n1C 76166,C1(NC(=O)CC2(O)CCC2)CC2(C1)CN(C(C1CCN(C3CCCCC3)C1)=O)C2 76167,c1(OC)noc(C2CC2)c1C(=O)NCCC(C)NC(=O)C(C(C)C)NS(N)(=O)=O 76168,c1(CCNC(CCOCCN(C)C(C2CC2F)=O)=O)cccnc1 76169,N1(C(c2c(C)noc2)=O)CC(O)CCC1NCC(=O)N(C)C 76170,CCC(C)(C(=O)OC)NC(=O)C(CNC(c1c[nH]nc1OC)=O)OC 76171,N1(C(C(C(C)C)N2CCCC2=O)=O)CCCN(C(C2CC3(F)CC2C3)=O)CC1 76172,C1(C(=O)NC2CCC(CNC(C(C=C)(C)O)=O)C2)CCc2cncn2C1 76173,N1(C(=O)Cc2cnn(C(F)F)c2)CC2CCCC(C1)N2C(C1CCC2CC12)=O 76174,C1(OC)CNC(=O)C2CCC2(OC)CC1.C1(=O)CN1.C(C(N)=O)S.OC 76175,c1(C(N2CCC(C)(CCNC(c3occ(C)c3)=O)C2)=O)cc2scnc2[nH]1 76176,Cc1cn2cc(C(=O)N(C)CC3CCN(C(=O)C(C)(C)C)C3)nc2s1 76177,C1(O)(CNC(C2(C#C)CCC2)=O)CCCN(C(=O)Cc2ccccc2SC)C1 76178,c1(C(=O)NC(C(C)NC(=O)COCC2CC2)(C)C)ccc2c(c1)nc(O)n2C 76179,C1(CNC(c2n[nH]c(C)c2Cl)=O)CC2COCC2N1c1nnc(C2CC2)s1 76180,c1(C(=O)NC(CCNC(C2ON=C(C)C2)=O)C)ccc(C)c2c1CCCN2 76181,Cc1cc(N)c(Br)cc1C(=O)NCC1(C)CCCN1C(=O)C(C)CN(C)C 76182,c1(C(C)=O)ccc(C(N2CCN(C(=O)Cn3cnnn3)CC2)=O)cc1 76183,C1(C(=O)NC2CCC(C(=O)N(C)CC3CCCC3(C)C)C2)(CC)CNC(=O)C1 76184,C(=O)(C(CC)C(C)C)N(CCCOC1CCN(C(C2C(CCC)C2)=O)CC1)CC 76185,c1(C(=O)NC2(C)CC(NC(=O)CC3=CCCC3)C2)cnc2ccsc2c1 76186,C(C)(CC(=O)NCC(c1cccs1)O)NC(CNC(C)=O)=O 76187,c1(C(=O)NC(C(N2CCC3(CC(F)C3)C2)=O)C2(C)CC2)ncc2ccccn12 76188,Cc1cc(=NCCn2cc(C#N)cn2)[nH]c(N2CCCC3(CCN(C)C3)C2)n1 76189,C1(NC(c2ccncn2)C)CCOC1c1ccccc1 76190,C(C)(C(=O)OC(C)(C)C)(C(=O)N1CCC(CN(C(=O)C(C)C(F)F)C)CC1)OC 76191,CCCC(C)(CCC)C(=O)NCCN1CCN(C(=O)C(C)(F)C(=O)OC)CC1 76192,C1(CC)CN(C(=O)CC2(NC(C3CC(=O)CCO3)=O)CC2)CC(C)O1 76193,C1(CC(=O)N(CCCCC)C)CCCC1NC(=O)Cc1nccn1C 76194,C(=O)(CCC(C)(C)O)N1CCCC(C(C)NC(C(CC)OCC)=O)C1 76195,C1(=O)C(CC(C)C)OC=CC(=O)C(=O)CCN1CC#C.C1(N)CCCCC1O 76196,Cc1c[nH]nc1C(=O)N(C(=O)CC1CSCCS1)C 76197,c1(C(N2C3C(NC(C(C)CC4CCCCC4)=O)C(C3)C2)=O)c[nH]nc1S(N)(=O)=O 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76546,N(C1c2ccccc2CC1C)C(C(=O)NCC1(OC)CCCCCCC1)=O 76547,C12(C(=O)NCc3ccc(CNC(C(C)C)=O)cc3F)CCOC1CCOC2 76548,C(CCN(C)C(c1cccc(N(C)C)c1)=O)(C(C)C)NC(C(COC)N(C)C)=O 76549,c1(C(=O)NCCN(C(CCC)=O)C2CCCC2)nnn(C)c1C(F)(F)F 76550,C(CCSC)(CN=c1[nH]c(C)cc(=NCCN(c2ccc(Cl)cn2)C)[nH]1)OCC 76551,NC(=O)CCNC(=O)C(=O)OC(C1(C2CCCO2)CC1)=O 76552,C1(NC(CCC=C)c2nnnn2Cc2conc2C)CCC(c2nc[nH]n2)CC1 76553,CC(C)CC(CN=c1[nH]c(N2CCC(OCCO)CC2)nc2c1SCC2)N(C)C 76554,N1(C(C=C(C)c2ccco2)=O)CC(NC(=O)C2=CC3CCC2C3)CC2(CCC2)C1 76555,C1(O)(CNC(c2ccc(Br)o2)=O)CCCN(C(C2CCC(CO)CC2)=O)C1 76556,CC1COC2(C1)CN(C(C1CN(C(c3cncs3)=O)C(C)(C)C1)=O)C2 76557,C12(CC(=O)N(C3CCC3)CC(CO)OC)CCC1CN(C(c1cc(O)ncc1F)=O)C2 76558,C(=O)(C(C)(C)CCCOC)N(CCNC(c1nn(CC)nc1C)=O)C1CC1 76559,C1(CC(=O)N(CCCC(C)C)C)CC2(C1)CN(C(=O)C(O)C1CCC1)C2 76560,Cc1noc(C)c1S(=O)(=O)NCCCNC(c1c(N)ccc(F)c1C)=O 76561,c1(C(=O)NCCCC(=O)NCC2CC2NC(c2cnc[nH]2)=O)ccccc1F 76562,c1(CN(C(c2cn(C(C)C)nc2Br)C(=O)NC2(C)CC2)CC=C)nnc(C)n1C 76563,c1(C(=O)NC2CN(C(C3(C)CC3)=O)CC3C2C3)c(F)ccc2n[nH]cc12 76564,C#CCC(C)(CC)C(=O)NCCC1CN(C(=O)C=Cc2c(C)coc2C)CCO1 76565,C(=O)(C1=CNS(=O)(=O)N=C1C)NC1C(CNC(C2(COC)CCCCO2)=O)CC1 76566,N1(C(C2N(CC)CC2)=O)CCC(O)(CNC(=O)C(Br)=C(C)C)CC1 76567,N#Cc1cccc(C(N2CC3CC(NC(=O)Cc4cccnc4N)C3C2)=O)c1 76568,c1(C(=O)NC2CN(C(c3ccn(C)c3)=O)CC2F)cc(N=S(C)(C)=O)ccn1 76569,Cc1ccc(C(=O)NCCC2CC(NC(=O)C(O)Cn3cncn3)C2)cc1Br 76570,C1(N(C(=O)CCn2cncn2)CCC)CCN(CC(=O)N(C2CC2)C2CC2)C1 76571,c1(CC(=O)NCC#CCNC(C2C(C(=O)NCC#C)C2)=O)ccncc1C 76572,C1(CNC(c2[nH]c(=N)sc2)c2nnnn2CC2CCCO2)CCCC2(CCC2)O1 76573,C1(C(=O)NC(CCSC)CO)CN(C(c2ccnc(C)c2)=O)CC1(F)F 76574,c1(C(=O)NCC(C)CN(C)C(c2nccn2C)=O)ccc(F)c2c1CCC2 76575,c1(C(c2nnnn2CC2CC2)NCC=CCOC)ccc(C(F)(F)F)s1 76576,Cc1n[nH]c(C)c1CCNC(=O)CN(C(C1CCN(C(N)=O)C1)=O)C(C)C 76577,N1(C(C(C(CC)O)(F)F)=O)CCC2(C=C(C(=O)NC3CC(C4CCCC4)C3)C2)C1 76578,c1(C(N2CCC3(CC3C(N3CC(O)(CO)C3)=O)C2)=O)cccc2c1CCC2 76579,C#CCC(C(=O)NCCC(=O)NCC)NC(C1CCCN1C(C)=O)=O 76580,C1(CNC(C2(C)CCCC2O)=O)CC2CCC1N2C(=O)Cn1cncn1 76581,C(=O)(C(CNC(=O)C(C)CCOC(C)=O)C(C)(C)C)N(CC(C)(C)C)CCC 76582,C1(C(N2CC=CC(NC(CCc3cn(C)nc3)=O)C2)=O)CSC2(C)CCC(=O)N12 76583,c1(C(=O)NCC(CNC(CC(C)C2CC2)=O)F)ccncc1Cl 76584,Cc1cc(CCC(=O)NCCCCNC(=O)C(C)c2ccsc2)ccc1Cl 76585,O=S(=O)(c1ccc(Br)cc1N1CCC2(CCSC2)C1)NCCc1ccccc1Cl 76586,c1(C(N2CC3=C(CN(C(C=CC(=O)O)=O)C3)C2)=O)csc2c(Cl)cccc12 76587,CC(C(=O)OC(C)(C)C)C(=O)NC1CC(NC(=O)C(CCO)N(C)C)C(O)C1 76588,Cc1ccc(NCCC(=O)NC(C2CN(C(=O)CCNC(N)=O)CCO2)C)cc1 76589,C1(C)(C(=O)NC(C)(C)CF)C=CCN1C(C1CC1(F)Cl)=O 76590,S(=O)(=O)(CC(=O)N1CCCC1(CNC(C1CC2(CSC2)C1)=O)CC)N(CC)CC 76591,O=C(N=c1[nH]nc2ccc(Br)cn12)N1CCc2cc([N+](=O)[O-])ccc21 76592,C1(CNC(CCc2onc(C(C)C)n2)=O)CCCCN(C(c2coc(Br)c2)=O)C1 76593,C1(CCNC(C2(C#C)CC2)=O)C(C)CCCN1C(c1cccc(NC(C)C)c1)=O 76594,C1(NC(C(CC)N(CC)CC)=O)CN(C(=O)CC2COCCOC2)CCC1F 76595,C1(C(N2CC(C(=O)N(C3CSC3)C)(CC)C2)=O)CCNC(=O)C1 76596,c1(OC)ccc(C=CC(N2CC(O)(CNC(c3cccc[n+]3[O-])=O)C2)=O)cc1Cl 76597,c1(C(=O)NCC(CC)(C)NC(c2cc3ncccc3s2)=O)cncc([N+](=O)[O-])c1 76598,c1(NC(=O)C(=O)NC2CCCCC2F)c[nH]cc(Br)c1=O 76599,N#Cc1ccc(F)c(C(=O)NC2CC2CNC(c2cc3sccc3s2)=O)c1 76600,C(CC)(C(=O)N1CCC(C(C)(C)NC(=O)CC2(C(F)(F)F)CC2)C1)=CC 76601,C1(NC(C(C)C2CCCO2)=O)C2CC(NC(=O)CP(C)(C)=O)CC12 76602,N1(C(C2CC(C#N)C2)=O)CC2CC(NC(c3ccoc3)=O)CC2C1 76603,C1(NC(C(CC)CN(C)C)=O)COCCN(C(C2CN(C)CCN2C)=O)C1 76604,c1(C(C(=O)NCC(C)(C(C)C)NC(c2c(C)csc2)=O)C)c(C)nn(C)c1C 76605,c1(C(N2C(C)CCC(NC(CCOCCC)=O)C2)=O)ccc2c(c1)NC(=O)CC2 76606,N1(C(CCC)C)CCC(O)C(C(=O)N(CCCOc2ccc(F)cc2)C)C1 76607,C=CC(C)(CCOC)C(=O)N1CCOC(CN(C)C(C2CC(O)(C#N)C2)=O)C1 76608,C1(CNC(C(c2ccn(C)n2)C)=O)CC(C)N(C(=O)CC2CC3(CCC3)C2)C1 76609,c1(C(N2CCC(C(C)NC(c3n[nH]cc3Cl)=O)CC2)=O)csc2c1CCC(C)C2 76610,C12(NC(c3ccc(O)nn3)=O)CC(C1)N(C(c1cncc(F)c1)=O)C2 76611,C(CC(C(C)(C)C)NC(c1nsnc1O)=O)N(C(Cc1ncc(C)s1)=O)C 76612,N1(C(C(C)(C)SC)=O)CC2CCOC2(CNC(c2n[nH]c3cccnc23)=O)C1 76613,C1(C(=O)NC(CC)C(C)C)C=CCN(C(c2ccn(CC)c2C)=O)C1 76614,C1(O)(C(=O)NCc2c(C(=O)NCc3c(C)noc3)n(C)nn2)CCC(C)CC1 76615,N1(C(c2cccc(C)n2)=O)CCCC12CCN(C(C1CCCSC1)=O)C2 76616,C1(NC(CC(C)(C)F)=O)CC2CCC(C1)N2C(c1ccc(Cl)c(N)c1)=O 76617,C(CCCCCNC(=O)C(C)(C)CNC(C1C=CCC1)=O)OC 76618,Cn1c(C(N2CC3CC(NC(=O)CCC4CCC(=O)N4)C2C3)=O)cnc1[N+](=O)[O-] 76619,O=C(C#CC1CCOC1)NCC(c1ccccc1Br)NC(CC(O)CO)=O 76620,c1(-n2c(C3CCCN(S(C)(=O)=O)C3)nc(CS(C)(=O)=O)n2)cc(Cl)nc(Cl)c1 76621,c1(OC)cccc(F)c1C(=O)NCC1CCC(NC(c2cnoc2C)=O)CC1 76622,c1(C(N2CCCC(C)(NC(C3C(OC)CCC3)=O)C2)=O)cc(O)cc(F)c1F 76623,CC1CC(C(=O)NCCOCC2CC2)CCN1C(C1CC2CC(=O)C1O2)=O 76624,C1(N(C(=O)Cc2cnccn2)C)CC2CCC(C1)N2C(=O)Cc1nn(C)cc1Cl 76625,N1(C(CCc2scc(C)n2)=O)CCCC(C2CCN(c3cncc(Cl)n3)CC2)C1 76626,C1(C(N(C2CN(C(C3CC(=O)OC3(C)C)=O)C2)C)=O)CCCCC12OCCO2 76627,C1(C(=O)NC2CCC(CC)CC2)CCC2(CN(Cc3cnc(Cl)s3)C2)O1 76628,N1(C(c2c(C)nsc2C)=O)CC2(CCNC(C3(F)CCCOC3)=O)CCC1CC2 76629,c1(CC(N2CC=CC(NC(c3ccn(C(CC)CC)n3)=O)C2)=O)c(C)cccc1C 76630,Cc1nn(C)cc1CCC(N1CC2C(NC(C3(C)SCCCS3)=O)C2C1)=O 76631,C1(CC(=O)NC(C)CN2CCCC2)CCN(C(=O)C(C)OC(C)(C)C)C12CCC2 76632,c1(C(=O)NC(c2cnccn2)C)ccc(-c2cc3sccc3s2)c2cc[nH]c12 76633,c1(C(N(CCC(C(C)C)NC(=O)CC#N)C)=O)cccc2nc(O)n(C)c12 76634,n1(CC)cc(C(=O)NCC(O)CCNC(c2cnc(C(C)(C)C)[nH]2)=O)c(C)n1 76635,CCCC(CC)C(=O)NC1CCC(NC(c2ccc(Br)cc2N)=O)CC1 76636,c1(C(C)=O)ccc(OCCN(c2ncc(-c3cccnc3)s2)C2CC2)c(F)c1 76637,C#Cc1ccc(C(=O)NC2CC(CO)N(C(c3ccnnc3C)=O)C2)c(F)c1Cl 76638,C1(NC(C=C(CC)CC)=O)CC2CCC1N2C(c1nn[nH]c1C(F)(F)F)=O 76639,CC(CNC(=O)CC1(NC(C2CCS(=O)(=O)N2)=O)CCCCC1)CCCO 76640,c1(C(N(CCCN(C(=O)CCC(F)F)C)C)=O)cnc2ccoc2c1 76641,C1(CNC(C(C)SC(F)(F)F)=O)CC2CN(C(=O)C=Cc3ccc(Cl)s3)CC12 76642,c1(C(=O)OC)cc(C)c(C(N2CCCCC2C2CCN(C(=O)C(C)O)CC2)=O)o1 76643,c1(C(N2C3(CN(C(=O)CC(O)c4ccccc4)C3)CC2)=O)ccc(O)c(O)c1Cl 76644,C1(CCOP(C)(C)=O)CCN(C(=O)C(=O)NCC(C(F)F)c2ccccc2)CC1 76645,c1(NC(C2C(C(=O)Nc3cc(F)c(OC)c(F)c3)C2)=O)nc2cc(Br)cnc2[nH]1 76646,C1(C(=O)NCCN(C(C(C=C)O)=O)CCOCCO)CC2(CCOCC2)CO1 76647,ClCCCN=C(NN1CCC(C)C1)NC1CCCCC1.C1(CCC)CCOC1 76648,C(CC(CO)NC(=O)CC1CC(NC(C2CC2c2cccs2)=O)C1)SC 76649,N1(C(C)=O)CC(C2CC2C(=O)N(CCOC2CCOC2)C2CC2)C1 76650,Cc1cc2c(=O)n(CC(=O)NC3CCCC(CO)C3)nnc2s1 76651,C1(CNC(C(C)N(C(=O)CN(C)C(=O)C2CC2)CC)=O)COCC1(C)C 76652,Cc1cn2c(C(N3CC4(C3)CN(C(C3(C)CS(=O)(=O)C3)=O)C4)=O)c(C)nc2s1 76653,CCCC(C(=O)NC(C)CC(=O)NCC1(Cl)CC1(C)C)NC(C)=O 76654,N1(C(C2C=CC(NC(C(C)c3ccccc3)=O)C2)=O)CCCC12CCNC2=O 76655,C#CCC(O)C(=O)NCC1(CN(C)C(c2cscc2Cl)=O)CC1 76656,c1(COC)sc(N(C)Cc2ncn(-c3ccccc3)n2)nc1C 76657,N1(C(c2cc(OC)no2)=O)CCCC(C)(NC(c2nc(C)n(C)c2C)=O)C1 76658,Cc1cc(CCC(=O)NCC2CC(NC(=O)C(F)C(F)(F)F)C2)ccc1Cl 76659,c1(OC)cnc(C(=O)NCCNC(C2CC(=O)CCO2)=O)cn1 76660,CC1CN(C(=O)Cc2cn(C)cn2)CC(CCNC(=O)C(C)N2CCCC2)O1 76661,N1(C(C(F)=CC)=O)CCCC(O)(CN(C(=O)C(C)(C)CC)C)C1 76662,C(=O)(C(C(C)C)NC(=O)CC)NC(c1cn(CCCCC=C)nn1)C 76663,c1(C(N2C(C(N(C(C(=O)OC)C)C)=O)CC2C)=O)cc(C)ncn1 76664,C1(NC(c2cc(C)nc(C)n2)=O)CCC12CCCN(C(=O)C=CC1CCCC1)C2 76665,c1(C(=O)NC2CN(C(C3(CCC=C)CC3)=O)CC2F)cccc2c1C(F)(F)CC2 76666,C(Cc1ccc(OC(F)(F)F)cc1)(C(=O)N=S(C)(=O)CCN)c1cccc(C)c1 76667,C(=O)(CCCN(C)N=O)N1CC(OC)(CNC(=O)C(C)C(C)C)C1 76668,N1(C(COCCOCC)=O)CCCC(O)(CCNC(c2c[nH]c(=N)cc2C)=O)C1 76669,C1(NC(=O)Cc2nncs2)CC2CN(C(=O)CC3CCCC(F)(F)C3)CC12 76670,C1(C(=O)NCCN(c2cnc(C#N)cn2)CC)CS(=O)(=O)CC(=O)N1 76671,Cc1ccnn1CC(N1CCC(C(C)C(=O)NC2(C(C)C)CCC2)C1)=O 76672,N1(C(C2C3CN(C)CC32)=O)CC2(CCCC2NC(c2cn3ncccc3n2)=O)C1 76673,c1(COC)cc(C(=O)NC(C)C(C)(C)NC(=O)CSC(C)(C)C)ccc1F 76674,C(=O)(CS(=O)(=O)C(C)C)NC(C(C)NC(c1n(OC)cnc1C)=O)CO 76675,CCCCCCC(=O)NC1CCCN(C(c2c(CC=C(C)C)cnn2C)=O)CC1 76676,N1(C(CCCC#C)=O)CCN(C(=O)CCc2csc(Br)c2)CC1CC 76677,Cc1cc(NCC2CCC2(F)F)ncc1S(=O)(=O)NC(CO)C1CC1 76678,c1(C(=O)OC)cc(CN2CCC(C(N3CCCC(N(C)C)C3)=O)CC2)ccc1F 76679,C1(NCc2c3nc(C)oc3ccc2)CC2CC3(CC2C1)OCCO3 76680,C1(=CCNC(C(C2CCC(=O)N2)C)=O)CCN(C(=O)CCF)CC1 76681,C12(C(=O)Nc3cncc(C#C)c3)CCCC1N(C(=O)CN1CCNC1=O)CC2 76682,C12(C(=O)NC(CCC=C)C3CC3)CC1CN(C(=O)COC1CCC1)C2 76683,C(=O)(CC(C(F)F)NC(=O)CC1(NC(C)=O)CC1)NCC(=C)C(F)(F)F 76684,Cc1c(C(=O)NC(C)(C)CCNC(C2(C)CCCC2O)=O)cnn1CCC#N 76685,C1(NC(C(C)NC=O)=O)CC2C1CCN2C(C1CCOC(=O)CC1)=O 76686,c1(C(=O)NCC2(C)CCC(NC(C(C)C3CCC3)=O)CC2)cccc2c1CCC2 76687,C1(C(C)C)(CO)CCN(C(C2CC(C)N(C(=O)CSCCC#N)C2)=O)C1 76688,C1(CNC(CC=C)=O)CCC(NC(C2(C(F)(F)F)CC(F)C2)=O)CC1 76689,C(=O)(C1c2ccccc2C2CC1C2)NCC1(C)CC(NC(C=CC=CC)=O)C1 76690,Cc1ccc(-c2ccc(C3CCN(Cc4ccnc(Cl)c4Cl)CC3)cc2)c(F)c1 76691,c1(NCCOCCOC)nc(NC(C2CCCCC2)CO)c2c(ncn2C)c1 76692,CC(O)C(C)(C)C(=O)N1CCN(C(=O)CC(O)CC2CC2)CC1 76693,CC1(CNC(c2cc3occc3s2)=O)CCCN(C(C2C(F)(F)C23CC3)=O)C1 76694,c1(C(=O)OC)cc(Cl)cnc1NC(=O)CC1NCCC1O 76695,c1(OC)cc(N(C)C)ccc1C(=O)NCC(C)(C(C)C)NC(=O)CC(C)F 76696,c1(CC(=O)NCC#CCNC(C2CCC(C)C2)=O)cc(Cl)ccc1[N+](=O)[O-] 76697,N1(C(c2c(C)nc(O)nc2C)=O)CCC2(CCOC2)C(CNC(=O)CNC=O)C1 76698,C1(C2CCN(C(c3cnn(C(F)(F)F)c3)=O)C2)(NC(c2cc(OC)ns2)=O)CC1 76699,CC1(C)OC(=O)NC1C(=O)NCC1CC(NC(=O)COc2ccc(C#N)cc2)C1 76700,C1(C2CC2)(CNC(CC2C(C)(C)CCCC2)=O)CCN(C(C2SCCCS2)=O)C1 76701,c1(OC)ccc(C(=O)NC2CN(C(=O)CCCCN(C)C)CC2C)c2[nH]ncc12 76702,c1(C(=O)NCC(CNC(C2CCOC2)=O)OC)ccc(C)c(Cl)c1 76703,C12(NC(c3c(C)cc(=N)[nH]c3)=O)COCCC1CN(C(c1c(Cl)n[nH]c1C)=O)C2 76704,c1(C(N(C)C)C2CC2)cn(CCC(N2CCCC2C(N)=O)=O)nn1 76705,N1(C(C(CC)N(CC)CC)=O)CC(NC(=O)CC(CC)C2CC2)C(C)C1 76706,N1(C(C(CCC)NC(=O)CCCNC(N)=O)=O)CCOC(C)(C)C1C 76707,n1(CC)ncc([N+](=O)[O-])c1C(=O)NC1CCCC(NC(c2csc(C)n2)=O)C1 76708,CC1(C)CN(C(=O)C=CC2CCCCC2)C1COC.c12cn(nn1)CCNC2=O 76709,C(=O)(C1=NN(CC(C)C)C(=O)CC1)N1CC(N(C(C(CC=C)(C)N(C)C)=O)C)C1 76710,C12(NC(c3c[nH]c(=NC)o3)=O)CCCC(NC(c3cc(OCC)no3)=O)(C1)C2 76711,c1(C(=O)NC2CCC(NC(c3cc(C(C)=O)sc3)=O)C2)ccc2c(c1)ncn2C 76712,N1(C(C(C2CCC2)OCC)=O)CC2CCC1C2NC(c1nccnc1CC)=O 76713,c1(OC)ccnc(C(N2CC(NC(C3OCC4CCCC34)=O)C(SC)C2)=O)c1F 76714,C(C(C(F)(F)F)c1ccccc1)NC(c1cccc(OC2CCOCC2)n1)=O 76715,c1(C(CO)N(C(=O)CC2(CN)CCOCC2)C)ccc(F)cc1 76716,c1(N2C(CC)CN(C(=O)Cc3cccc(SC)c3)CC2)ncc(C#N)cc1Cl 76717,C1(CNC(c2cnc(C(C)OC)s2)=O)C2CN(C(=O)Cn3nnc(=N)[nH]3)CC12 76718,c1(NC(C(N2CCCCC2c2ccccn2)=O)=O)cccc(C2CC2)c1 76719,Cc1ccc2c(c1)CCN2C(c1ccc(OCc2nccn2C)cc1)=O 76720,c1(NC(c2n(CCCC)nnn2)C2(C)CCCO2)ccc(F)c(C(N)=O)c1 76721,Cc1ncoc1C(=O)NCC1CCCC1NC(=O)C(C)n1cncn1 76722,C=CCCN=C1NN2CCC(N1)CC=NC=C2.C1(C)(C)CC1(Cl)Cl 76723,Cc1c(Cl)ccc(C(=O)NCCC2(O)CN(C(=O)C(C)(C)C(=O)N(C)C)C2)c1N 76724,C1(C(N(CC)Cc2nc[nH]n2)=O)CN(C(=O)COc2ccccc2)CCC1O 76725,C1(NC(C2(CNC(C(CC)C)=O)CC2)=O)CC(=O)N(CC(=O)NC)C1 76726,C1(CNC(CCNS(CC)(=O)=O)=O)CCCC2(CCN(C(=O)C(C)OC)CC2)O1 76727,C1(C(=O)NC2(C3CN(C(c4[nH]cc(C(C)=O)c4)=O)C3)CC2)CCCC(C)(C)CC1 76728,C1(C(=O)NCC(C)C(=O)N(C)C(c2ncccn2)C)C(C)(C)C1(C)C 76729,C1(CN(C(COC(CC)C)=O)CC)CN(C(=O)CNc2cc(C)on2)CCO1 76730,c1(CNC(C(COCC)NC(=O)C=CC(C)CC)=O)ccc(F)cc1F 76731,c1(N(C(C(C)Cc2ccc(Cl)cc2)=O)C)ccc([N+](=O)[O-])nc1 76732,c1(CC)cc(C(=O)NCc2ccc(C(=O)NC(C)C(O)C(F)F)cn2)n(C)n1 76733,C#Cc1cc(F)c(C(=O)NCC(C)N(C(c2cc(C)c(F)cn2)=O)CC)c(F)c1 76734,C=C(C)CC(C(=O)NCC(=O)N(CCOC)C(C)C)OC 76735,c1(C(N2CC(OCC(=O)N(C)CC3(C)CCC3)C2)=O)cc(Cl)ccn1 76736,c1(-c2ccc(N(C(C)C)C(c3ccc(Cl)cc3F)=O)cc2)ccc2occc2n1 76737,N1(C(COCCOCCOC)=O)CC2C(CN(C(=O)C(C)CC#C)C)C2C1 76738,C1(C(N2CC(C(C)NC(=O)COc3cccc(F)c3)C2)=O)CCc2nc[nH]c2C1 76739,c1(C(c2n(CCC)nnn2)NCCCN2CCCCC2)ccnc(C)c1 76740,C(CC1CC1)(C(=O)NC1CN(c2ncco2)C1)NC(c1csc(CO)n1)=O 76741,C1(NC(C)=O)CC(CNC(=O)CCc2cc(F)cc(F)c2)C12CCC2 76742,CC(C)(C)CCCCC(=O)NC1CCCCN(C(C2C(Cl)(Cl)C23CC3)=O)C1 76743,C1(CCN(C(C(C)Cl)=O)C)CCCCN1C(=O)CN1C(=O)CNC1=O 76744,Cc1noc(Cl)c1CC(=O)NC1CN(CCCNC(=O)CC2(CO)CC2)CCO1 76745,C1(NC(c2c(COC)cco2)=O)CN(C(=O)CCc2nc(C)c(C)[nH]2)CC1SC 76746,C1(NC(C(C)C2CCC2)=O)CC2CCC(C1)N2C(=O)CCCN(C)C(C)C 76747,c1(OC(C)C(=O)N(CC(O)CN(C(=O)C=CC=C(Cl)Cl)C)C)cccc(N)c1 76748,C1(F)(CNC(CCOCC#C)=O)CCN(C(c2ccnnc2O)=O)C1 76749,c1(C(C)(F)F)ccc(CC2(c3nnnn3NCC3CCCO3)CCCSC2)nc1 76750,C1(NC(C(c2ccc(OC)cc2)C)=O)CCC2(CC1)CC2N 76751,C1(CC)CC(C(=O)NC2CCCC(CO)C2)CCN1C(=O)C(C(C)(C)C)OC 76752,c1(COC)oc2ccccc2c(=O)c1C.C12CN(CC1O)CCN1CCN2CC1 76753,N1(C(CNC(CC(C)C)Cc2ccccc2)=O)CC2OC(=O)N(C)C2C1 76754,c1(C(=O)NC(CCC(=O)NCC2C(C(=O)OC)C2)C)cnc(O)c(F)c1 76755,c1(C(=O)NCC(CC)NC(C=CC=CCCCCC)=O)ncc(F)cc1F 76756,c1(C(CC)Nc2cc(OC)ccc2OC)cc(C)cc(Br)c1OC 76757,CC1CCCN(C(c2ccnc(Cl)c2)=O)C1CNC(C1CC2CC1C1CC21)=O 76758,N1(C(C(C)CC2CCCC2)=O)CCCCC1C1(NC(C2CCCSC2)=O)CC1 76759,C1(C(=O)NCC#CC)CCN(C(=O)CCn2ccc(C)n2)C1 76760,C(=O)(C1=C(CC(C)C)N(CC)C(=S)NC1c1nccc(Cl)c1Cl)OCC 76761,CC1CC2CC2CC1C(=O)N(CCN(C)C(c1csc(=N)[nH]1)=O)C(C)C 76762,C(=O)(CCN(C)C(C1(CCN=[N+]=[N-])CC1)=O)NC(COCC=O)C.CO 76763,C=C(I)CC(=O)NCC1(NC(=O)CN2CCCCC2)CC1 76764,C(=O)(C1=NOC(C)(C)C1)NCCCC(C)NC(c1csc(C)c1C1CC1)=O 76765,C1(CCN(C(=O)CCCCc2cnc[nH]2)C)CCCCN1C(c1cncnc1)=O 76766,c1(C(C(=O)NCC(F)F)N(CC)Cc2ccncc2)ccc(C)c(OC)c1 76767,C1(CCOC)(C(=O)NCC2CCC2NC(=O)CC(=O)NCC2CC2)CCCC1 76768,c1(CC)cc(C(=O)NCC(C)(C)OCCNC(=O)C(C)CC2CCCC2)c(C)o1 76769,C1(C(=O)NCCCN(C(C(C)NS(CC)(=O)=O)=O)CCO)Cc2ccccc2S1 76770,N1(C(C(C)=C(C)C)=O)C(C(=O)NCc2ccc(O)nc2)CCC1C(C)C 76771,N1(C(C2CCN(S(C)(=O)=O)C2)=O)CCOCC(C)(CN(C(=O)C=C2CC2)CCO)C1 76772,Cc1ccc(F)cc1C(=O)NCC1(CNC(=O)CCNS(C)(=O)=O)CCCC1 76773,c1(C(=O)NCCN(C(C2(CC=C)CCOC2)=O)C)ccccc1CC 76774,N1(C(C(COC)OC)=O)CC2(CC(NC(c3cnnc(C)c3C)=O)CO2)C1 76775,CC1CC=C(C(=O)NC(C(=O)N2CCC(O)(CO)CC2)C(C)(C)C)CC1 76776,C(=O)(CCC[N+](=O)[O-])N1CC(N2CCN(C(C3C(=C)CC3)=O)CC2)C1 76777,C1(CNC(CC(CN(C)C)O)=O)C2CCCC1N(C(c1csc3nnsc13)=O)C2 76778,C(=O)(CCCCc1cnc[nH]1)NC(C)CC(C)NC(C1CCC(F)C1)=O 76779,C(=O)(C1=NNC(=O)CC1)N1CCC(C2C(NC(CC(CCC)C)=O)CCO2)CC1 76780,C(C(C)C(=O)NC(c1cn(C)nn1)C(=O)NCCC1(O)CCOC1)SC 76781,Cc1cccc(OC(C)C(=O)NCCCNC(C2(CC3CCC3)CCCC2)=O)c1 76782,C1(O)(C(=O)NCC)CCN(C(C2CCCN(c3ccc(Br)cc3)C2=O)=O)CC1 76783,N1(C(Cc2[nH]c(=NCCC(=O)O)sc2)=O)CCCC2(C1)CC(F)(F)C2 76784,CC(O)C(C)(C)C(=O)N(C)CC1CN(C(c2ccc(CN(C)C)cc2)=O)CCO1 76785,c1(C(N2CC3CCCC(C2)N3C(c2cnc(Cl)[nH]2)=O)=O)cc2c(s1)CCCCC2 76786,N1(C(COCCCOC)=O)CC2(CCN(C(=O)CN3CCCCCC3)CC2)CC1C 76787,C(C(=O)NOCC1CC1)N(C(=O)C=Cc1cc[nH]c1)CC#C 76788,c1(NC(C2C(C(=O)NC)C2)=O)cc(Br)cn2ccnc12 76789,N1(C(CC)=O)CCCCC1C(=O)NCCCCCNC(C1(C)CC1)=O 76790,C(=O)(C1CCCc2cn(C(C)C)nc21)N1CCN(C(C2(CC)CC2)=O)CC(O)C1 76791,c1(CC)cccc(Cl)c1Cl.N1(C(C(=O)Nc2ccccc2O)C2CC2)CCN(C)C(C)C1 76792,c1(-c2cc(C(N(C3CN(C(Cc4c(C)cns4)=O)C3)C)=O)on2)ccccc1F 76793,C(=O)(C(C)C(O)CC(C)C)NC(C(=O)NCC(COC)C)CC1CCOCC1 76794,Cc1nc2ccncc2cc1C(N1CCN(C(C2CCC(=O)NC2)=O)CC1)=O 76795,c1(N2CC(CNC(=O)NCCCCl)C(O)C2)ncnc2n[nH]cc12 76796,c1(C(=O)NCC(CC=C)NC(C2CC(Cl)(Cl)C2)=O)cnn2cccnc12 76797,N(C(=NCc1cc(-c2ccco2)on1)N1CCC(OC)C1)C1CCN(CCC)C1 76798,C1(NC(C(=C(C)C2CC2)F)=O)CC(C)N(C(=O)Cn2cncc2C)C1 76799,Cn1ncc2c(SCC(=O)NCc3cccc(Cl)c3)ncnc12 76800,c1(CNC(C2CCCC2NCC2CCC(F)(F)C2)=O)cc(Br)c(Br)s1 76801,C1(CCC)CCCN(N(Cc2cccc(C)c2)CC(F)F)C1 76802,C(=O)(C1=CC(O)C(NC(C2(C(N)=O)CCC2)=O)C1)Nc1c(CC)noc1 76803,N1(C(CC(C)CNC(c2ccc3c(c2)CC3)=O)=O)CCC2(C=CCO2)C1 76804,C1(C2N(C(c3c(C)noc3)=O)CCC2)CCCN(C(=O)CC(=O)N(C)C)C1 76805,N1(C(c2c(CC)con2)=O)CC2CCC1C(CNC(C13CC(OC)C1C3)=O)C2 76806,C#Cc1ccc(C(=O)NC2CCCC(CNC(c3cc(C)[nH]n3)=O)C2)c(OC)c1 76807,c1(C(N2CC3(CCCN3C(C3CC34CC(O)C4)=O)C2)=O)ccc2cnoc2c1 76808,c1(C(N(CC(C)N(C(c2c(CC)noc2)=O)C)C)=O)nc(C)c(C)nc1O 76809,N12CC3CC1CN3C2=O.c1(SCCCNS(C)(=O)=O)ccccc1 76810,N1(C(C2CN(C(C)=O)C2)=O)CCC(CNC(=O)CC2CC3(CC3)C2)C(O)C1 76811,C1(CC)CN(C(C2CCCCC2NC(C2C3CC(=O)CC23)=O)=O)C(C)CO1 76812,c1(C(N2C(C(=O)NC(C)C(=O)NCC(C)C)(CC)CCC2)=O)cn(C)c(=O)cn1 76813,C=CCCCCCCC(=O)NCc1nnn(C)c1C(=O)NCC(O)CN(C)C 76814,Cc1cc(C(N2CCC(CO)(NC(=O)Cc3cncnc3)CC2)=O)c(C)cc1Br 76815,C(=O)(C(O)CCCNC(=O)CC1CCCNC1=O)NCC1CCN(C(CC)=O)C1 76816,c1(C(N(CCC)CCNC(C2(F)CC2)=O)=O)cc(F)c(O)c(F)c1 76817,c1(C(=O)NC2CCC(N(C(c3c(C)snc3)=O)C)C2)ccn(C)c(=O)c1 76818,C1(N(CC(F)COCC2(N)CC2)C)CCC(C(=O)C(=O)OC(C)(C)C)O1.CO 76819,C1(O)(CN(C(c2cnc(C(C)C)[nH]2)=O)C)CCCN(C(C2CC23CC(O)C3)=O)C1 76820,C1(C(=O)NCCN(CCOC)C(c2ccc(C(F)F)o2)=O)CC2(C)CC1CO2 76821,CCCC(C(=O)NCC1CN(C(c2nc(Cl)sc2Cl)=O)CCO1)NC(N)=O 76822,c1(C(N2CCCC(NC(c3nccc(C)c3)=O)C2C)=O)cnc2c(F)cccn12 76823,C=CCCC(C)(c1nnnn1CC1CCOCC1)NCC1CC1(Br)Br 76824,N1(C(C(C(C)C)n2cnnc2)=O)CC(N(C)C(c2ccc(F)cn2)=O)C(C)(C)C1 76825,N1(C(C)CO)CC2C(C(=O)NCc3noc(-c4ccccc4)c3Br)C2C1 76826,Cc1cc(Br)ccc1CC(=O)NC1CN(C(=O)CCNC(N)=O)CC1C#N 76827,c1(C(N2CC(CCO)C2)=O)csc(C2CCCN2C(=O)CCBr)n1 76828,C1(CNC(c2cc(OC)no2)=O)CN(C(C2SCC=C2C)=O)CCCO1 76829,C1(CC(=O)NCCCN(C)C(C23CC(O)C2C3)=O)CCC=CCC1 76830,c1(NC)ccc(Cl)c(C(=O)NCC(C2CCCC2)NC(=O)CCSC2CC2)c1 76831,CCC(C)(COC)C(=O)NCC(C)N(C(=O)Cc1cccc(C(N)=O)c1)C 76832,c1(SCC(=O)NCC(C)(C)CNC(=O)CC2COCCOC2)cccc(Cl)c1 76833,C12(NC(c3cc(C)n(-c4cccc(F)c4)n3)=O)CCN(C(C3CCC3)=O)CC1C2 76834,c1(NC2CCN(C)C2)cc(NCc2cc[nH]n2)ncn1 76835,C(CCC(=O)N1CC(CC(F)C(=O)NCC(C)(C)C2CCC2)C1)C1C(C)C1 76836,C(=O)(CC1=NNC(=O)C1)NC1CC(CC)(CC)N(C(C2(F)CCOC2)=O)C1 76837,c1(C(C)NC(c2ccc(Cl)c(C)c2)c2n(C(CC)C)nnn2)ccc(F)c(Cl)c1 76838,C1(C(C)CC(=O)NCC(C)(C)C)CCCN(C(=O)OC(C)(C)C)C1 76839,C(CCC(=O)NC(C)CN(C(c1csc(N(C)CC(C)=O)n1)=O)C(C)C)OCC 76840,C#CC1(C(=O)NCC2CC(=C)C2)CN(C(=O)Cn2cnc(C(N)=O)n2)C1 76841,Cc1nc2c(C#N)cnn2c(O)c1CCC(=O)N1CC(SC(F)F)C1 76842,[N-]=[N+]=NC1CC(C(=O)NCCc2cccs2)N(C(=O)CC2CCC2)C1 76843,C(=O)(CC(C)CC(C)(C)C)N1C(CNC(CCC#CC)=O)CC(O)C1 76844,C(=O)(C1CCCc2scnc21)N(CC(C)(C)Cn1cc(CC(O)C(C)(C)C)nn1)C 76845,C1(OCC(=O)NCC(CC)N(C(=O)CC2CCN(C)CC2)C)CCN(C)CC1 76846,c1(C(CNCc2cccc(C)c2Br)O)cccc(S(C)(=O)=O)c1 76847,N1(C(CCOCCN(C)C)=O)CC2CC(C1)N(C(c1ccc(N(C)C)nn1)=O)C2 76848,C(=O)(N=c1cc2n([nH]1)CCOC2)NC1(O)CC2N(C(=O)OC(C)(C)C)C(CC2)C1 76849,c1(NC(C2CC(C)CN2C(=O)CCc2cccc(O)c2)=O)nc(Cl)nc(Cl)n1 76850,Cn1ccc(S(=O)(=O)N2CCC(NC3CCCC4CC34)CC2)c1 76851,C1(CC(=O)NC(c2cscn2)C)CC2(CC2)CN1C(c1cccc(F)c1N)=O 76852,c1(CNS(CCCOCCN(C)CC2CCCO2)(=O)=O)c(F)cccc1F 76853,CCCCCCOC(C)C(=O)NCCOC1CCN(C(=O)CNS(C)(=O)=O)C1 76854,c1(C(=O)NC2(CF)CCN(C(CCC(=O)OC)=O)C2)cc(C)cc(Br)c1F 76855,c1(NCC2(CC)CCCC2)ncccc1S(=O)(=O)NCCCC1CCCC1O 76856,C(CC)(C(C)(F)F)NC(CN(C(=O)CSC(F)F)CCC)=O 76857,CC1=NOC(C(N2CC(NC(=O)C(C)COc3ccccc3)C2)=O)C1 76858,N1(C(C=CCOCCOC)=O)CC2CC2(CNC(C2CCOC2C2CC2)=O)C1 76859,C1(NC(CN2C(C)CCC2)=O)COCCC1NC(c1cc(CO)[nH]n1)=O 76860,Cc1c(C(=O)NC23CCN(C(=O)Cn4cnnn4)CC2C3)oc2c(F)cccc12 76861,C1(C(=O)NC(C(C)C)CNC(=O)C(C)(C)N(C)C)Nc2ccccc2C1(C)C 76862,c1(OC(C)C(=O)NC(C)(C)CNC(=O)CS(C)(=O)=O)ccc(F)cc1Cl 76863,c1(C(=O)NCC2N(C(CC3CC(=O)C3)=O)CCCC2)ccc(Br)c(F)c1 76864,c1(CNCC(CC(C)C)NC(=O)NC(C)=O)ccc(O)c2ccccc12 76865,N1(C(Cc2nc(NC(c3ccnc(O)c3)=O)sc2)=O)CCCC(F)(CO)C1 76866,C1(CCC)CN(C(c2c(N)sc(C)c2C)=O)CCN1C(c1cnn2c1OCC2)=O 76867,N1(C(C(=Cc2cccs2)C)=O)CCC(C2CC2)C1CNC(c1ccoc1C)=O 76868,C1(C(N2CC3C(CO)C3C2)=O)C(O)CCN1C(=O)C(c1ccccc1)O 76869,Cc1nc2nccc(N(C(C)CNC(c3cc(F)cnc3O)=O)C)n2n1 76870,c1(C(=O)NC2C3N(C(C(C)C#N)=O)C(CC3)C2)nnn2c1C(=O)NCC2 76871,CCC(C#N)C(=O)NCC(C)C(=O)NCCc1cnco1 76872,n1(CC(=O)NC(c2nc(C(=O)NOC3CCCC3)co2)C)cc(C#N)cn1 76873,C12(C(=O)NCC3C=CC(NC(C4(OC)CCOC4)=O)C3)C3C4C1C1C2C3C41C 76874,c1(C(N2CC(C(C)NC(C(C=CC)O)=O)C2)=O)coc2cc(C)c(C)cc12 76875,N1(C(CC2(OCC)CCC2)=O)CC(C(=O)NC2(CO)CCCCCC2)C2(CC2)C1 76876,c1(C(C(N2CCCC(N(C(=O)CCCF)C)C2)=O)OC)ccc(Cl)c(Cl)c1 76877,N1(C(c2ncccc2Br)=O)CCC2CCN(C(C3(F)CC3)=O)C2C1 76878,Cc1ncccc1C(N1CCOCC1C(=O)N(C1CCN(C2CC2)C1)C)=O 76879,c1(-c2ccc(OC)cc2)ccc(NC(=O)Nc2cnccc2Br)cc1F 76880,CC(C)C(C)C(=O)NC(N)=O.N1(OC(=O)NC2CC2)CC1 76881,C1(F)(CNC(C(C)SC(C)C)=O)COCCN(C(c2snc3ccccc23)=O)C1 76882,C1(CC)(NC(=O)CC2CCN(C)C2)CC(C)(C)C1.C12CC(C1)CNC(=O)CO2 76883,N1(C(c2c(OCC)nccc2)=O)CCN(C(=O)C(C)n2ccnn2)C(CCO)C1 76884,CC1(CNC(=O)CCC2CC(NC(C3(O)CCC3)=O)C2)CC2CC2C1 76885,CCC(C(=O)NC1(C)CCN(C(=O)CCN2CCC(C)CC2)CC1)C(C)C 76886,C1(C)(C(NOC(CC)C)=O)CCCN1C(=O)C=CC(C)(C)SC 76887,CC(O)C(C(=O)NC(c1cnc(N(C)C(=O)OC(C)(C)C)o1)=O)N(C)C 76888,N1(C(CS(CC)=O)=O)CC=C(CC(=O)N2CCN3CCCC3C2C)CC1 76889,CC1CC(=O)NCC1C(N1CC2(CCN2C(c2nscc2Br)=O)C1)=O 76890,C(=O)(C(CCSC)NC(C)=O)N1CC(c2ccccc2)(CC)C1 76891,Cn1ccc2c(C3(C(=O)NC4CC(c5cc(CF)on5)C4)CC3)cccc12 76892,Cn1cncc(C(N2CCN(C(c3cncc4c3CCC4)=O)CC2CO)=O)c1=O 76893,c1(C(=O)NC(C2CN(C(C(F)OC)=O)C2)C)csc(CC(F)(F)F)n1 76894,c1(OC)csc(C(=O)NCCCC(C)NC(=O)CC2(C)CC2)c1 76895,C1(C)(CNC(c2ccc(CCC)[nH]2)=O)CCCN(C(C2CC3CCC(C2)O3)=O)C1 76896,C1(CC(=O)N(CC(C)C)CC(C)C)CN(C(=O)C(C)c2ccco2)CCO1 76897,CCC(C)C(C(=O)NC(CC(N)=O)C(=O)NCC(C1CC1)SC)N(C)C 76898,c1(CN(C(CC)CC)C)cn(Cc2ccccc2)nn1 76899,n1(CC)cc(C(N2CCCCC2C(C)NC(=O)CCCN(C)C(C)=O)=O)c(C)n1 76900,CC(C)CC(CC(C)(C)C)C(=O)NC(=O)C(c1ccn(C)c1)C 76901,c1(OCC)nc(Cl)ccc1C(=O)NC1CN(C(=O)C2=C(C)CCC2)CC1C 76902,Cc1cc(C)c(C(=O)NCCC(O)CNC(=O)Cc2ncccc2C)c(S)n1 76903,c1(NC(C)C(N2CCCC2CC2CCCCC2O)=O)ncccc1S(C)(=O)=O 76904,N1(C(c2nc(SC)sc2)=O)CCC2(CC2NC(=O)COc2ccsn2)C1 76905,c1(C(=O)NC2C3CN(C(CN4C(C)CC4)=O)CC32)cccc2c1CCC2=O 76906,N1(C(c2ccc(CC)s2)=O)CC(NC(=O)C(C)(O)C2CC2)C(SC)C1 76907,N1(C(C(=O)N(C(C)C(C)(C)O)C)=O)CC2CC(N)C(C2)C1 76908,CCCCC(CC)C(=O)N1CCCC1C1(NC(c2nncs2)=O)CC1 76909,N1(C(C2C(NC(=O)CCc3ccncc3)C=CCC2)=O)CCCC2(CCCO2)C1 76910,c1(C(=O)NCC2C3CN(C(c4cc(CC)oc4C)=O)CC32)cc2c([nH]1)CCC2 76911,C1(C(=O)NCC2(COC)CN(C(c3c[nH]ccc3=O)=O)C2)Cc2cccc(C)c2O1 76912,c1(C(=O)NCCC2CC(NC(C3C(C)CC3)=O)C2)cncc(N(C)C)c1 76913,N1(C(C(C(=O)OC)(C)F)=O)CC2CC(C(=O)Nc3cnc(N(C)C)nc3)CC2C1 76914,C(=O)(C(C)C(O)C(C)C)N1CCN(C(C(CCC)(C)C)=O)CC1CF 76915,C1(CNC(c2ccnn2CC2CCC2)=O)C2CN(C(C3C4CCCC34)=O)CC12 76916,C(=O)(C#CC1CCOCC1)NC1C(C(=O)NC(C(=O)NCC)C)OCC1 76917,N1(C(C(C(CC)CC)OC)=O)CC2OCCN(C(=O)CCCC3CCCO3)C2C1 76918,CCCCCCCc1cn(C(C)C(=O)NCC(=O)NC(CC)CC)nn1 76919,CN1CCN(N2CCCC2C2CCCO2)CC1NC(=O)OC(C)(C)C 76920,CC(C)CC(C(=O)N1CCN(C(c2ccc(F)o2)=O)C(CC(F)F)C1)N(C)C 76921,c1(CC)noc(C)c1C(=O)NC1CCN(C(C23CC(C)C2C3)=O)C1C 76922,O=C1CCN(CC2CCOCC2)C(=O)N1CCOCc1nc2ncccn2n1 76923,c1(OC)ccc(C(N2C3CN(C(C4CC4(C)C)=O)CC23)=O)c(Br)n1 76924,C=CCC(C)C(=O)NCC1CCN1C(=O)C(=Cc1ccccc1)C 76925,c1(NCC(=O)N(c2cccc(O)c2)CC)cccc(C(=O)NC)n1 76926,C(=O)(CCCCC(=O)NCC1(OC)CN(C(=O)C(c2ccccc2)SC)C1)NC 76927,c1(C(=O)NCC(CCNC(=O)CCc2nncs2)OC)cc(F)c(F)cc1O 76928,c1(OCCCC)ccc(C(C)Nc2ccc(I)cn2)cc1OC 76929,c1(C(=O)NC2CN(C(C3C(CC)CCO3)=O)CC2C)ccc(OC)c(OC)c1Cl 76930,c1(C(=O)NC2C(CNC(c3c[nH]c(C(F)(F)F)c3)=O)COC2)ccc(O)cn1 76931,c1(C(N2CCC(NC(c3cnc(Cl)s3)=O)C(F)C2)=O)ccc2nc[nH]c2c1F 76932,C1(O)(CCNC(C2(C(=O)OCC)CC2)=O)CCCN(C(=O)C(C)(C(C)C)OC)C1 76933,C1(C(=O)NCc2c(C(=O)NC3(CC(C)C)CC3)cco2)CC(=O)CCO1 76934,N1(C(c2c(C)c(Br)sc2)=O)CC2(CCC2NC(C2CC(C)C2)=O)C1 76935,C1(NC(CCC=CC)=O)CN(C(=O)C#CC2CCCCC2)C2(CCOC2)C1 76936,c1(C(N2C(C3CCCN(C(C(=O)N(C)C)=O)C3)CCCC2)=O)cc([N+](=O)[O-])n[nH]1 76937,c1(C(CC(=O)NC(c2cnccn2)C)NC(C2(F)CCCC2)=O)ccc(F)cc1 76938,c1(CC(=O)NCC23CC2CN(C(C2CCSC2)=O)C3)ccc(Cl)c([N+](=O)[O-])c1 76939,c1(C(C=CC(=O)ON(C(c2c(C)ncs2)c2ccccc2)C)=O)ccc(F)cc1 76940,C(=O)(CCCCCN(C(=O)CSCCC(C)C)C)N1CCC(C(C#C)C)CC1 76941,CN1CC(NC(=O)C(C)(CO)NC(C2CCCCN2C)=O)C(F)(F)C1 76942,CCC(C)(CCC(C)C)C(=O)N1CC2CC(C1)C2(C)C 76943,N1(C(CSCCCC)=O)CCCC(CC)(NC(=O)C(C)NC(=O)C(C)(C)C)C1 76944,c1(-c2cc(CNC(N3CC(C(=O)O)(COC)C3)=O)sc2)ccc(C(=O)O)cc1 76945,C1(CNC(=O)Cc2ccoc2)CCCN(C(c2ccccc2-n2cncn2)=O)C1 76946,C1(NC(c2c(OCC)oc(C)n2)=O)(CO)CCCN(C(c2cc(C)ns2)=O)C1 76947,c1(CC)nc(C)cc(=NC(C)CCN(C(=O)CNC(=O)CC(C)(C)C)C2CC2)[nH]1 76948,C1(C(N2CC(c3cn(C(C45CC(CO4)C5)C)nn3)C2)=O)CCC(=O)N1C1CC1 76949,C(=O)(CC(C)CC(C)C)NC1(C(=O)NCCC(CC)CO)CCC1 76950,c1(N(CC#C)C2CC2)nnc(CCc2ccccc2)n1Cc1ccccc1 76951,C1(NC(CC2(CSC)CC2)=O)CC(CO)N(C(c2nc(O)sc2C)=O)C1 76952,c1(C(=O)NCCCCN(C(C2C(OC)CCCC2)=O)C)cnc2cc(C)[nH]c2c1 76953,N1(C(C2CC(OC)C2)=O)CC(C2(NC(C3CC3Cl)=O)CC2)C1.C(C)(=O)O 76954,N1(C(CSCC(C)=O)=O)CCCC(C2CN(C(=O)C(c3cccnc3)C)C2)C1 76955,c1(CC(=O)NCC(CC)NC(c2cc3nccnc3[nH]2)=O)ccc2ncsc2c1 76956,c1(CC(=O)N(C2CCCN(C(CC=C)=O)C2)C)coc2cc(O)ccc12 76957,Cc1nnc(=NCC(CC(C)C)NC(=O)CC(C(F)F)n2cccn2)[nH]c1C 76958,c1(C(=O)NC2CC(N(C(c3ncn(C(C)C)n3)=O)C)C2)cncc2cnccc12 76959,C1(C(N2C(CNC(C(C)(C)C3CCCC3)=O)CC(O)C2)=O)CC2(C1)CC2(F)F 76960,C(=O)(C(C1=CCCCCC1)N1CC(OC)C(NC(=O)OC)C1)NCCC 76961,N1(C(CCCSC)=O)CCC(C(F)CNC(=O)CN2CC(=O)NC2=O)CC1 76962,C(C(C)(C)CC(=O)N1CCCC1C1CCCCN1C(C1CC12CC2)=O)OC(C)=O 76963,C(CC)(C(C)(F)F)NC(C(CC1CCC1)NC(COCCC=C)=O)=O 76964,c1(CC(=O)NCCN(C(=O)C(=Cc2ccc(C)cc2)C)CC)c(F)cccc1F 76965,C1(CNC(c2ccc(SC(F)F)cc2)=O)CN(C(=O)NCc2ccccc2)CCO1 76966,CCCCC(CNC(c1ccsc1C(F)(F)F)=O)NC(c1cnsc1C)=O 76967,CC(CN(C)C)CC(=O)NC1(C(=O)NC(C)CCc2cn[nH]c2)CCC1 76968,N1(C(Cc2c(OC)cccc2)=O)CC(OCc2ccccc2)CCC1C 76969,N1(C(C(CC)C)=O)CCC(CNC(C23CC2COC3(C)C)=O)(OC)CC1 76970,C(C(CC)(CC)C(N)=O)NC(c1ccc(CNC(C(CC)N(C)C)=O)s1)=O 76971,CCC(C(=O)NC1COCC1C(N1CCC(CC(C)C)CC1)=O)C(C)C 76972,c1(C(=O)NCC(c2ccc(O)cc2)NC(c2ccsc2)=O)ccn2nncc2c1 76973,N1(C(CCN(C)CC)=O)CCCCC1CCC(=O)N(C)Cc1cccnc1 76974,C12(C(N3C(CC(=O)NC)CC3)=O)CC(CCO1)N(C(c1cnn[nH]1)=O)C2 76975,c1(C(N2CCC(C)(CCNC(c3c(C)occ3)=O)C2)=O)cc(F)ccc1N 76976,C1(C(N2C(COC)COCC2)=O)CCOCCN1C(C1CC(F)CN1C)=O 76977,N1(C(C2(C)C(C)C2)=O)CC2(CCCN(C(C3C=CC(=O)N=N3)=O)C2)C1 76978,C1(CCC(=O)NCc2cn(CC#C)nc2)CCCN(C(c2cc(Cl)cn2C)=O)C1 76979,C1(NC(Cc2n(C)nnc2)=O)CC(CNC(=O)CC(C)(C)c2cccs2)C1(C)C 76980,C1(COC)(NC(=O)C(c2ccccc2)N(C)C)CN(C(=O)C(CSC)OC)C1 76981,Cc1noc(C(F)F)c1C(=O)NCCC1CCN(C(=O)C=Cc2cc[nH]n2)C1 76982,C(CC(C)(C)CC(=O)NCC(C1CCN(C(=O)CCCCCF)CC1)F)OC 76983,c1(C(C)=O)ccc(C(=O)NCCO)s1.C(C)(C)(CNC(=O)CNC=O)OCC 76984,c1(OC)cnc(C(=O)NC2CCC2NC(C2(C)CC3CC3C2)=O)c(F)c1 76985,S(=O)(=O)(c1ccc(NCCCc2ccccn2)cc1Br)N(C)CC1CCN(C)C1 76986,CCCCC(C(=O)NC1CCCN(C)C1=O)NC(c1cnnn1CC)=O 76987,C=CC(C)C(=O)NC(c1ccccc1)C(=O)NCc1nn[nH]c1C1CC1 76988,C1(C(N(CC(C)NC(c2cnc(Cl)c(Cl)c2)=O)C)=O)Cc2ccccc2C(=O)O1 76989,C12(NC(CCc3cn(C)nc3)=O)CCCC1N(c1cc(Cl)ncn1)CC2 76990,C(=O)(C#CC(=O)N(C)C)N1C(CNc2cnc(CC(C)C)[nH]2)CCC1 76991,c1(C(=O)Nc2nc3c(s2)CC(C)CC3)cncc(C2=CCNCC2)c1 76992,Cc1nc(=N)[nH]cc1C(N1CCC(CNC(c2ccc(F)o2)=O)C1(C)C)=O 76993,C(=O)(C1COc2cc(C)c(C)cc21)NCCC(C)NC(c1c(Cl)cn(CC)n1)=O 76994,C(C1CCCC1)=CC(=O)N(CCNC(C(n1ccc(Br)n1)C)=O)C 76995,c1(C(=O)NC2CCC(CCNC(CC=CC=C)=O)C2)cccc(-n2cccn2)c1 76996,CC1(C)CN(C(c2c[nH]c(Br)c2)=O)CC1NC(c1cccc(C(N)=O)c1)=O 76997,c1(CNC(CC2CCC(NC(CCNC(=O)OC)=O)CC2)=O)cccc(F)c1I 76998,c1(CC(=O)NCC2CCCN(C(C(CC)OC)=O)C2)ccc(S(C)(=O)=O)cc1 76999,C1(C)(NC(CC(CC)C2CC2)=O)CCCN(C(=O)CC(C)(C)O)C1 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77035,c1(C(N2C(CN(C(C(C)n3cncn3)=O)C)COCC2)=O)ncc2[nH]ncc2n1 77036,N1(C(c2cccc(C(C)=O)c2)=O)CCN(C(=O)CCC2CCC(=O)N2)CC(O)C1 77037,c1(N(C2CCCN(C(C3ON=C(C)C3)=O)C2)C)ncc2c(n1)COC2 77038,C1(C(N2C(C(=O)OC)C(C)CC2)=O)CC2CC1CN(C(=O)C(O)CC(C)(C)C)C2 77039,c1(C(N2CCC(CCNC(C3OCCN(C)C3)=O)C2)=O)ccc(N)c(Cl)n1 77040,Cc1cc2ccc1C(=O)N1CCC(C1)C(=O)N2.c1(CN(C)C)nccc(Cl)c1C 77041,CC(CC1CC1)C(N(C=O)CC1(CS(N)(=O)=O)CCC1)C1CC1 77042,N1(C(c2n(CC)ncc2Cl)=O)CC(NC(=O)CCCCN2CCCC2)C(C)(C)C1 77043,c1(C(N2CC(NC(c3cc4c(nn3)CCC4)=O)C2)=O)cc2ccccc2c(O)n1 77044,C(=O)(C1=NOC(C)C1)N1CC(O)(CNC(COCCCCCC)=O)C1 77045,c1(C(C)(C(=O)O)NC(C2CC(N(C)C)C2)=O)c(F)cc(Br)cc1F 77046,CCCCS(=O)(=O)CC(=O)NCC(C12CCC(CC1)C2)NC(=O)C(O)C(C)C 77047,C(=O)(C(F)(F)C(O)C1CC1)NC1CCC(CNC(=O)CC2(O)CCCC2)C1 77048,C1(NC(=O)C(c2ccc(Cl)cc2)O)CCCCC1NC(C1(CO)CCOCC1)=O 77049,C(=O)(C(O)C(C)(C)CC)NCCN(C(c1cnc(-c2ccoc2)[nH]c1=N)=O)CC 77050,N1(CC)CCCC2C1CCCN2Cc1ccc(-c2ccccc2C=O)s1 77051,C1(C(=O)NCc2ccc(C(N)=O)o2)(NC(C2(CC)CC2)=O)CC1(C)C 77052,C#CCC(C(=O)NCC1=CCCC1)NC(=O)Cc1cccnc1 77053,C(C(=O)NC1CC(CNC(C2CC2(F)F)=O)C1)(C(C)(C)C)NC(C)=O 77054,CCCCCC(=O)NCC=CCNC(=O)CN1CCN(CCS(C)(=O)=O)CC1 77055,C1(C(=O)OCC)CN(Cc2ccc(-n3cccn3)cc2)CC1(C)C(F)F 77056,Cc1cc(CC(=O)N(C)CC2(CNC(c3cc(CCO)on3)=O)CCC2)c(C)s1 77057,C(=O)(C1=NNC(=O)CC1)N1CCC(O)(CCNC(C(CC)=CC)=O)C1 77058,N1(C(C2CC(C(F)F)(OC)C2)=O)CCC2(CC1)CC(C)N(C(C1CCCS1)=O)C2 77059,N1(C(C=CC=CC)=O)CCCC2(CNC(=O)CCN3CCCC3)CCCC12 77060,C1(CC)C(C(=O)NCC(C)(CNC(=O)CC2CCC(=O)N2C)OC)CCN1C 77061,c1(CN2C(CNC(c3ccc(OC)c(I)c3)=O)CCC2)ccc2c(c1)OCCO2 77062,CC1CC(CCNC(c2nocc2Cl)=O)CCN1C(c1ccn(C2CC2)n1)=O 77063,C1(NC(C2(N(C)C)CC2)=O)CCCC1NC(=O)CCOCC(F)F 77064,C#CC(CC)(CC)NC(C1(C(C)C)CCN(C(C2CCSC2)=O)C1)=O 77065,C(=O)(C#CC1CCCCO1)NCC(n1cc(CN(CC)CC)nn1)C 77066,N1(C(C2(NC(c3cc(C)sc3)=O)CCSC2)=O)CCCC2(CC(O)C2)C1 77067,C1(C2(N)CCC2)(C(=O)NC(C(n2ncc(C)c2)C)C)CCC1 77068,n1(CC)nnc2c(NCC(C)CNC(=O)C(C)(C)N3CCCCC3)ncnc12 77069,CCCS(=O)(=O)NCC(=O)NC(C)C(C)NC(=O)C(C)Cn1ccnc1 77070,c1(C(N2CC(NC(Cc3c(C)[nH]nc3O)=O)C(F)C2)=O)n[nH]c2c(F)cccc12 77071,c1(NC2CCCN(CC)C2)[nH]c(=NC2CCCn3ncnc32)nc2sccc12 77072,C1(OC)CN(C(c2ccc(CC(C)C)s2)=O)C(C)(CNC(c2cccs2)=O)C1 77073,c1(NC2C(O)CN(Cc3cccc(F)c3Cl)C2)ncnc2c(F)cccc12 77074,CCS(=O)(=NC(=O)C1CCCCCN1C(=O)CN)c1ccc(C)cc1 77075,CCCCC(C)C(=O)N1CCN(C(C2CC(C)(C)C2C(F)(F)F)=O)CC1C 77076,O=C(CCCC(=O)c1cccs1)NCC1CCN1C(=O)CCC1CNC(=O)N1 77077,C1(NC(CN(C(C(CC=C)NC(C)=O)=O)C(C)C)=O)CC2CCCC2C1 77078,O=CN1CCOCC1C(=O)NC1CCCCN(C(=O)C2=NOCC2)C1 77079,C1(C(=O)NCC(C)C(C)(F)F)CC12CCN(C(C1COCC1C(N)=O)=O)C2 77080,n1(CC(=O)NC(CC)CN(C(=O)C(F)=C2CCC2)C)ccc2cc(F)ccc12 77081,C(CN(C)C)(C(=O)NC1CCC1N(C)C)NC(C1(OC)CCC1)=O 77082,CC(C)C(C(=O)N1CC(OC(=O)CN(S(C)(=O)=O)C)C1)NCc1cc(Cl)no1 77083,c1(CCC(N2CCC(N(CCC)C(C)=O)C2)=O)ccc(F)cc1F 77084,N1(C(c2c(N)n(C3CCCCC3)nc2)=O)CCCC2(COc3ccccc32)C1 77085,N1(C(C2N(CC)CC2)=O)CC2C(CNC(c3ccc(CN(C)C)cc3)=O)C2C1 77086,C1(NC(c2[nH]cc(C#N)c2)=O)CCCCCCC1NC(=O)CC1CNC(=O)O1 77087,N1(C(Cc2n(C)ncc2)=O)CCSCC1C(=O)NC1CC(O)C1O 77088,C1(CCNC(CCCNC(C(C)NC(=O)Cn2cnnn2)=O)=O)CC(F)(CO)C1 77089,N1(C(C(CSC)(C)C)=O)CC2CCN(C(c3[nH]nc4ncccc34)=O)C(C2)C1 77090,Cc1cc(C(=O)N(CCCNC(=O)CS(=O)(=O)C2CC2)C(C)C)c(O)cc1F 77091,c1(C(N2CCC(c3c(COC)c[nH]n3)C2)=O)cnccc1C#N 77092,c1(OC)cc[n+]([O-])c(C(=O)NCC2CN(C(c3ccnn3C3CC3)=O)CC2C)c1 77093,C1(CNC(C(CC)C)=O)CCC2CN(C(=O)C3=CCCO3)CCC2C1 77094,c1(CC(=O)NCCN(C(c2ccc(C)s2)=O)C)ccccc1C(C)C 77095,Cc1cncc(C(=O)NC(C2CCN(C(c3cc(=O)cc[nH]3)=O)C2)(C)C)c1 77096,C=CCCCC(C)(C)C(=O)NCC1CCC1NC(=O)C(=Cc1cccnc1)C 77097,c1(C(N2C(C)CCC(C)C2C)=O)ccc2cc(Cl)ccc2n1 77098,C12(C(=O)NCC3CC(O)(CNC(c4ccc(O)nn4)=O)C3)CCN(CC1)C2 77099,c1(C(N2CC(NC(C3(OC)CCCOC3)=O)C(OC)C2)=O)c(C)cc[nH]c1=N 77100,C1(CNC(C2(OC)CC2)=O)CC(C)(C)CN1C(=O)C(N1CC(C)CC(C)C1)=O 77101,N1(C(C(CC(=C)Cl)NC(=O)CC2CC3C=CC2C3)=O)C2CCCC1CC(=C)C2 77102,c1(C(C(=O)NCC=C)N(C)CC=CC(C)(C)C)ccc(-n2cccn2)cc1 77103,C1(C(=O)NCCc2c(C)nc[nH]2)C2CCC(C2)N1C(=O)C1=NNC(=O)C1 77104,N1(C(CC(C)(C)C)=O)CC2CCCC2(NC(c2ccc(N)cc2F)=O)C1 77105,Cc1cccc(C)c1CNC(=O)NC(C)COc1ccccc1Br 77106,N1(CC(O)C)CC23CCCC2(C1)C3.c1ccccc1OC(F)F 77107,c1(C(N2C(C(=O)Nc3c(C#C)nccn3)CC(OC)C2)=O)ccc(O)c(O)c1Cl 77108,n1(CC(N2C(CNC(CCS(=O)(=O)NC)=O)CCCC2)=O)nc2c(n1)CCCC2 77109,CC(C)(F)CCC(=O)NCC(CNC(c1ccnc(C(F)(F)F)n1)=O)CO 77110,c1(C(N2CCN(C(c3cc(C)ncn3)=O)CC2)=O)c2c(nn1C)CCC2 77111,C1(C(N2C(C)CN(C(c3cnnn3C)=O)CCC2)=O)COc2ccccc2C1 77112,CCN=c1ccc(C(N2CC(O)(CNC(=O)CCc3nnc(C)n3C)C2)=O)c[nH]1 77113,c1(CC)[nH]c(=N)sc1C(N1CCCCC1CN(C(=O)CCC1CCCCO1)C)=O 77114,Cc1cccc(C(=O)NCC2CCC(NC(=O)C(C)(C)Br)CC2)c1Cl 77115,C1(NC(CNC(C2CCCCC2)(C)CO)=O)CC2CCCC(C1)N2 77116,C1(C(=O)NC2CC(CCNC(c3ccn(CCC)n3)=O)C2)CCCN(C(C)=O)C1 77117,C12(CNC(c3cc(C)cc(N)c3)=O)CC(CCO1)N(C(=O)C(C)CC(C)(C)C)C2 77118,N1(C(c2cnc(C)[nH]2)=O)C(CNC(=O)CC2CC3C=CC2C3)CC2CCCC12 77119,Cc1cc(NCC2CCCO2)nc(C2CCN(C(=O)C(C)(O)C3CC3)CC2)n1 77120,N1(C(CSCC(N)=O)=O)CCC2CCC(NC(c3ccc(C(F)F)c(Cl)c3)=O)C12 77121,c1(CNC)cccc2ccnn12.Cc1cnc(N2CC(C(N)=O)(NC(=O)N)C2)nc1 77122,C1(COCC)(CNC(=O)C(=O)Nc2nccs2)CC12CCC2.C1(=O)C(C(C)C)N1 77123,C(=O)(C(F)(F)CCn1ccnn1)NCC(C)NC(C(c1c(OC)cccc1)O)=O 77124,N(C1CCCc2c1cnn2C)CC.c12nnnn1CCNC2(CO)C 77125,C(=O)(C(C)CCCOC)OC.n1(CC)cc(C(N2CCC(c3cn(C)nn3)C2)=O)cn1 77126,C(=O)(CCCCCCNC(C1CCOCC1)=O)N1C(C)(C)C(CO)C1 77127,N1(CCNC(C(C)OC)=O)CCCN(C(c2sc(Br)nc2C)=O)CC1 77128,C#CCCCC(=O)NC1CC(OCC(=O)NC(C)C(C)CO)C1 77129,CC1(C)Cc2nc(NC(c3cc(Cl)cc4c3CCC4)=O)sc2C(=O)N1 77130,C1(O)(C(=O)NC(CC)CNC(=O)C(C)(C)CC(F)F)CCc2ccccc2C1 77131,N1(Cc2nc(CC)sc2)CCC(O)C1C(=O)Nc1sccc1C(=O)OC 77132,N1(C(Cn2nnc(C)n2)=O)CC2(CC2)CC1CNC(C12CCC(CC1F)C2)=O 77133,C1(NC(C2(SCC)CC2)=O)CC2CC1CN(C(c1cncs1)=O)C2 77134,CC1CC=C(C(=O)N2CC3(CC(NC(c4ccccc4OCCF)=O)C3)C2)CC1 77135,Cc1cc(C(N2CCCC2CC(=O)N(CC(C)(C)N(C)C)C)=O)co1 77136,C#Cc1ccc(CC(N2CCCC2(C)CNC(C2(C)CC(F)C2)=O)=O)cc1 77137,C=CCCC(F)(F)C(=O)NC1CN(C(=O)C(C)N(CC(F)(F)F)C)CC1(C)C 77138,c1(C(=O)NC2C(CNC(C34CC(OC)C3C4)=O)CCC2)cc(S(C)(=O)=O)oc1C 77139,c1(OC)ccc(C2CCN(C(c3c(C)n[nH]c3C)C(=O)NC(C)(C)C)C2)cc1 77140,N1(C(C2C(CC)N(C(=O)C(F)F)CC2)=O)CCCN(C)CC1C 77141,CC(CC(C)(C)C)C(=O)N1CC2C(C(=O)NC3CN(C)CC3(F)F)C2C1 77142,N1(C(C(CCC)OC)=O)CCC(C2CC2)(CNC(c2cccc(F)c2CC)=O)C1 77143,C=CCCC(C)C(C(=O)NCC(C)NC(=O)C(=O)NC(C)(C)C)N(CC(F)F)C 77144,N1(C(c2cc(C#N)sc2)=O)CCC(CNC(=O)CC2CCCC2O)C(F)(F)C1 77145,C1(NC(CCc2cnc(C)o2)=O)COCCC1NC(=O)CCc1cnc[nH]1 77146,c1(C(N2CC(NC(=O)CCc3cnoc3)C3C2C3)=O)ccnc2[nH]c(O)nc12 77147,N1(C(C=C(CC)C)=O)CCC(C2CCN(C(=O)CCn3nc(C)cc3C)C2)C1 77148,c1(C(COC(C2C(C(=O)OCC)CC2)=O)F)ccc(F)cc1F 77149,N1(C(c2cnc(C(C)(C)C)[nH]2)=O)C2CCC1C(CNC(C1(C(N)=O)CC1)=O)C2 77150,CC1(C)CCC(C)(C(N2CC(CO)(NC(c3cncc4nc[nH]c34)=O)C2)=O)CC1 77151,c1(CCC(=O)NCC(C2CCOC2)O)ccc(Cl)c(F)c1 77152,C1(NC(CN(CC(C)(C)C)C)=O)CC2C1CCN2C(c1cnn(C)c1Cl)=O 77153,N1(C(C(COCC)(C)C)=O)CC(C)CN(C(=O)Cc2ccc(O)c(Cl)c2)C(C)C1 77154,c1(CC(=O)NC2COCC2CNC(C2(N(C)C)CCC2)=O)nnc(S)nc1O 77155,N1(C(CNC(C(CC)C)=O)=O)CCN(C(C2(C(C)C)COC2)=O)CC1CC(F)F 77156,c1(C(N(C2CC2)CC2N(C(C(CSC)C)=O)CCC2)=O)cnn2ccsc12 77157,N1(C(C2C(C(C)C)CCC2)=O)CCCN(C(=O)CCCCC#N)CC1CO 77158,c1(C(=O)NCC(C(C)C)NC(c2cccc3nn[nH]c23)=O)ccnc2[nH]cnc12 77159,C1(C(C(=O)OCc2ncccc2Br)OC)CCC(F)(F)C1 77160,C(=O)(C(C)(C)CCCC=C)NC(C(N1C(C#C)CC1)=O)COC 77161,C1(N(C(c2cnc(OCC)s2)=O)C)CCCC(NC(=O)CCc2cnccn2)C1 77162,Cc1c(F)ccc(C(=O)NC2(CNC(C3CCCCO3)=O)CCOC2)c1O 77163,CCC(C)CCCC(=O)NCC(N1CC(CO)C2(CC2)C1)=O 77164,N1(C(c2c(COC)noc2)=O)CCC(N=c2cc[nH]cc2C#N)CC1C 77165,N1(C(c2scc(OC)c2)=O)CC2CN(C(c3cc(C4CC4)on3)=O)CC2C1CO 77166,c1(NCC(=O)NC2CN(C(C=C(C)C(C)C)=O)C2)cccc(C#N)c1 77167,C1(CC(=O)N(C(CNC(C2COC(=O)N2C)=O)C2CC2)C)CCCCC1(C)C 77168,C1(CNC(C2CN(CCOC)C(=O)C2)=O)(CO)CCN(C(=O)CSC)CC1 77169,C=CC(C)C(C)C(=O)N1CC(OCCNC(c2ccc(N(C)CCC)nc2)=O)C1 77170,C1(C(N(C(c2ccco2)C)C)=O)COCCN(C(C2CC3C=CC2CC3)=O)C1 77171,C1(C)(CNC(C2CC(OCC)C2)=O)COCCN(C(=O)CNc2ccncc2)C1 77172,CCC(CC)CC(F)C(=O)NC1CC=C(C(=O)N(C2CCNC2=O)C)C1 77173,C1(CNC(COCCC)=O)CN(C(=O)C=Cc2cccc(O)c2)CC(C)(C)O1 77174,C(=O)(CCC(=O)C(C)(C)C)N1C(C(=O)NCCN(C(C)C)C(C)C)CNC(=O)C1 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77226,N1(C(C#CCNC(=O)CC2CC(C3CC3)C2)=O)CCc2sccc2C1 77227,C1(N(C(C(C)NC(CC)=O)=O)C)CCCN(C(c2cnn(C)c2COC)=O)C1 77228,C1(NC(c2ccc(C)o2)=O)(CNC(C2CCOCC2)=O)CC(F)(F)C1 77229,C1(CC)CN(C(c2ccc(Cl)nc2)=O)CCN1C(=O)CCc1cccc(OC)n1 77230,c1(CCCC)ccc(CC(=O)NC2CC2NC(=O)C(C)OCC2CC2)cc1 77231,C1(C)(CC)CCC(C(=O)NCC(C(=O)NCCCc2cccnc2)N(C)C)O1 77232,c1(NC(C2(C)CN(C(=O)NCC(=O)OCC)C2)=O)cc(F)cc(F)c1C#N 77233,C=CCC(C)C(C)(c1nnnn1C(C)C)NCC1CCC(F)(F)C1 77234,CC(C)(C)C(CNC(=O)Cn1ncnn1)C(=O)NC(CCO)C(C)(C)C 77235,N1(C(Cc2c(C)cccc2F)=O)CCN(C(C2(S(C)(=O)=O)CC2)=O)CC12CCC2 77236,C(=O)(CC(CC1CCCCC1)NC(=O)Nc1ccccc1)OC 77237,C1(F)(C(N2CC(OCCOC)C2)=O)CCCN(C(=O)CC2CCCSC2)C1 77238,Cc1cc2c(C(=O)NC(C3CCCCN3C(=O)Cc3cnc[nH]3)C)nccn2n1 77239,N1(C(C(CCC)C(C)C)=O)CCN(C(C2CCCCC2C(N)=O)=O)CC(C)(C)C1 77240,S(=O)(=O)(c1cccc(N2CCOC3(CCC3)CC2)n1)NC1CC(C)SC1 77241,N1(C(=O)Nc2scc(C(CC)(C)C)n2)CCc2cnn(C(=O)OC)c2C1 77242,N1(C(C(CCC)C)C(=O)NC2COC2)CCc2c(CCC)cccc2C1 77243,c1(C(=O)NCC(c2ccccc2)CN)cccn1Cc1ccncc1 77244,C1(C(=O)NCC2CN(C(CCN(C(C)=O)C)=O)C2)CCCC(C(F)(F)F)O1 77245,C(=O)(CCC(C)OCC)NC(C1N(C(C(C=C)O)=O)CCC1)(C)C 77246,C12(C(=O)NC3C(NC(=O)COCC(F)(F)F)CCC3)C3CCC(CC13)C2(F)F 77247,N1(C(CCC)=O)CCC(C(=O)NC2CC(C)(NC(C3CCCN3CC)=O)C2)CC1 77248,C#CCC(CC(=O)NC1(C(O)COC)CC1)NC(C1(CO)CCOC1)=O 77249,c1(C(C)=O)nc(C(=O)NC2CC(CCNC(c3cnn(C(C)C)n3)=O)C2)cs1 77250,c1(C(=O)NCC(C)CNC(c2ccc(C3CC3)s2)=O)ccc(C#N)c(Cl)c1 77251,N1(CCNC(CCN2CCN(C)CC2)=O)CC2CCC(C1)C2Cc1nnn(C)n1 77252,CC#CCCC(=O)N1CCC(N(C)C(c2cc(-c3ccccc3F)[nH]n2)=O)C1 77253,c1(OC)cc(C(=O)NCC2CCC2NC(=O)CN2CC(C)C2)cnc1OC 77254,C12(NC(c3ccc(CCC)[nH]3)=O)CC1CN(C(=O)C(CC)n1cccn1)C2 77255,C1(CNC(c2c(OC)cccn2)c2nnnn2C2CCC2)CC2CCC(C1)O2 77256,c1(C(=O)NC(CC)CN(C)C(C2(C(N)=O)CC2)=O)cn(C)c(=O)c2cncn12 77257,c1(OC)ncc(C)cc1NC(=O)C(=O)NC(Cc1nccn1C)C(F)F 77258,C1(CNC(CN(C2CCCC2O)C)=O)CCN(C(C2(C3CC3)CC2)=O)C1 77259,c1(C(=O)NC2(CNC(c3onc(OC)c3Br)=O)CC2)ccc2c(c1)CCC2 77260,N1(C(COCC)=O)CC2COCC(C1)C2NC(=O)CCC1CCC(=O)N1 77261,c1(NC(C2C(C)(C(=O)OCC)C2)=O)ccc(-n2cccc2)nc1 77262,C1(CNC(C2C(CNC(COCC(C)C)=O)C2)=O)CC=CCC1 77263,N1(C(C2(C)CC2)=O)CC2(CCN(C(C3C4CCC3(c3ccc(F)cc3)C4)=O)C2)C1 77264,C=Cc1ccc(C(N2CC(O)CC2C(=O)Nc2cnc(C)c(CC)c2)=O)cc1 77265,c1(CC)ccc(C)cc1C(=O)NCC(CNC(c1ccc(C)o1)=O)S(C)(=O)=O 77266,c1(C(N(CC(=O)N(C2CCC(C#N)C2)CC2CC2)C2CC2)=O)coc2c1COC2 77267,c1(C(=O)NCC2(C(N(CCCN=[N+]=[N-])C)=O)CC2)cncc(Cl)c1 77268,C(=O)(C(F)CC(C)(C)NC(=O)Cc1ccc(F)nc1)Nc1c(CC)ccc(F)c1 77269,c1(NC(C2CCN(Cc3c(Br)ccnc3Cl)C2)=O)cccc2nsnc12 77270,N1(C(C(C)CCN(C)C)=O)CCC2(CCC(NC(=O)Cc3nccn3C)CC2)C1 77271,c1(C(c2nnnn2CCCOC)NC(CC)CC#N)cc2c(cc1OC)CCC2 77272,C1(NC(Cc2n(C)ccc2)=O)CCN(C(=O)CCc2ncco2)CC12CCC2 77273,N1(C(C2C(CNC(=O)CC3CCOC3)OCC2)=O)CCN2C(=O)CCC2C1 77274,C#CCC(CC#C)C(=O)NCC1CCN(C(=O)CCc2cccc(F)c2)C(C)C1 77275,C1(C(=O)NCC2(C)CCCCCC2)(OC)CCC(C)(C)C1.C12CCN1C(=O)C2 77276,N#Cc1c[nH]cnc1=NC1CCCN(C(c2ccc3c(c2)CCCS3)=O)CC1 77277,C1(c2nnnn2C)(Oc2ccc(NC3CCN(OC)C3)cc2C)CC2COCC2C1 77278,c1(NC(c2c(C)nc(C)o2)=O)cnc2c(c1)CN(C(=O)CC#N)CC2 77279,CC1(C)C(CNC(=O)CCNC(=O)CO)CCN1C(=O)C(O)C1CC1 77280,C12(NC(c3c(OC)c(=O)cco3)=O)CCCC1CN(C(c1cc(=O)cc[nH]1)=O)C2 77281,CCC(C)C(=O)C(=O)N1CCC(F)(C(=O)NC2CC2c2ccn(C)n2)CC1 77282,N1(C(C2(Cl)C(C(C)=O)C2)=O)CCOC(c2cn(-c3cccc(C)n3)nn2)C1 77283,C12(NC(c3c(=N)[nH]cnc3)=O)CCN(C(=O)CCOC3CCC3)CC1C2 77284,C1(CC(=O)NCC(CC)NC(CCOCC#C)=O)CC(O)C1(C)C 77285,C1(C)(C(=O)OCC)CN(C(=O)C(C2CC(F)(F)C2)Oc2cc(CC)[nH]n2)C1 77286,CC(C)C(C)CC(=O)N(CC(O)CN(C(=O)Cc1nncs1)C)C 77287,O=S1(=O)CC2CN(c3cc(Nc4cc5c(s4)CCCC5)ncn3)CC2C1 77288,c1(C(=O)NCC2C(C)CN(C(=O)Cn3ncnn3)C2)csc2cc(Cl)cnc12 77289,CCCC(C(=O)N(CC(C)(C)NC(C1CC(SC)C1)=O)C)OCC 77290,c1(NC(=O)NCCc2ccc(CC)cc2)ccc(Br)c(Br)c1 77291,N1(C(CCC)=O)CCC(C(=O)NC2CC(F)(C(=O)OCC)C2)CC1 77292,c1(C(=O)NCC2C(N(C(=O)CCF)C3CC3)C2)cccc(Cl)c1N1CCOCC1 77293,c1(CC(=O)NCCCC(C)(C)NC(C(c2cccc(C)c2)C)=O)c(F)cccc1Cl 77294,N1(C(CCC=C(C)C)=O)CCCC(NC(=O)COc2cc(C)on2)C1C 77295,CS(=O)(=O)c1cnc(CCNC(=O)NC2COCC2C2CC2)nc1 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77313,Cc1ccc(Br)c(C(=O)NC2(C)CCN(C(c3c(C)cccc3O)=O)C2)c1 77314,c1(NC(C(C2(C)CC2)NC(CC2C(C)(C)C2)=O)=O)cnc2ccnn2c1 77315,C(=O)(C(C1CCOCC1)N1CCC(n2cc(C(N)=O)nn2)C1)NCC=C 77316,C1(C(=O)NCc2ccc(OC)cc2)CN(C(=O)COCC2CCC2)CCC1O 77317,c1(C(=O)NC2C(C(N(CC(F)(F)F)C)=O)C2)ccc2cnccc2n1 77318,C(=O)(C(F)CCC(C)(C)C)NC(CN(C)C)C(N1CCC(CO)C(C)(C)C1)=O 77319,S(=O)(=O)(c1ccc(=NCC2CCN2CC)[nH]c1)NCC1(CCC)CC1 77320,CC(CC(C)(C)O)NC(=O)C(Cc1ccccc1Br)NC(=O)C=Cc1cscn1 77321,C(CCCCC(=O)NC1CCCCCC1C(=O)NCCC(C(C)C)OC)OCC 77322,C(=O)(C1=CC2CC=CCC12)NCCOCCNC(c1nccs1)=O.C1(C)(CO)CC1 77323,Cc1c(C(=O)N(CCCNC(C2CC(C(C)(C)C)C2)=O)C(C)C)nnn1C(C)C 77324,CCC(CC(F)F)C(=O)NCC1(F)CN(C(C2(C3CCCCC3)CC2)=O)C1 77325,N1(C(C2C(C)(CC)C2)=O)Cc2nccn2CC(NC(=O)C(c2cnn(C)c2)C)C1 77326,Cc1cc(C(N2CC(F)CC2CN(C)C(C2CN3CCN2CC3)=O)=O)cnc1C 77327,C#Cc1ccc(C(=O)N(CCCNC(c2cc(C)n(CCO)n2)=O)CC)c(C)c1 77328,CN1CCC(C(C(=O)NCC2CCN2C(=O)OC(C)(C)C)N(C)CC2CC2)CC1 77329,N1(C(CSCCN(C)C)=O)CCCC(C2CCCN(c3nnc(C#N)s3)C2)C1 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77348,C1(COC)CC(CNC(c2nc(Cl)sc2C)=O)N(C(C2CCC(=O)NC2)=O)C1 77349,N1(CCNC(CCCOC)=O)CCC(NC(=O)CSc2ccccc2F)CC1 77350,c1(Sc2snc(-c3cccc(C)c3)n2)nc(=NCC(C)C(C)C)[nH]c2ccsc12 77351,N1(C(=O)NCC2CCCOC2)CCCC(Cc2cnnn2-c2ncccc2O)C1 77352,CC(C)CC(C)(C)C(=O)N1CCCC1CN(C)C(c1cncnc1C(C)C)=O 77353,C1(CNC(C2(CNC(C3CCC(CO)CC3)=O)CC=CC2)=O)CC2(C1)CC(O)C2 77354,C1(CCOC)(NC(=O)CC2CCC(=O)O2)CCN(C(=O)CC2CCSCC2)C1 77355,n1(CC)cc(NC(=O)CC2CCN(C(c3ncccc3F)=O)C2)ccc1=O 77356,c1(C(=O)NCC)cc(NC2CC2C(=O)Nc2cccc(OC3CC3)c2)cc(C)n1 77357,N#CC1CN(C(c2cccc3c2OCO3)=O)CCN1C(C1CC1C1CC1)=O 77358,C(C(C)(COC)C(=O)N(CCCN(C)C(c1ccnc(O)c1)=O)C)OC 77359,CCCC(C)(O)CC(=O)N1CC(OC)C(NC(=O)Cn2cc(C(F)(F)F)cn2)C1 77360,N1(C(=O)CSCc2cccc(Cl)c2)CC2CC(NC(C3(Cl)CC3)=O)C2C1 77361,c1(C(=O)NCCNC(CC(C)c2ccco2)=O)ccnc(-c2ccco2)c1 77362,N1(CC)CCCN(C(C2CCC(C)CC2)C(=O)NCCCF)CC1=O 77363,N1(C(c2c(CC)cns2)=O)CCN(C(=O)CS(C)(=O)=O)C(CCO)C1 77364,c1(C(N(C(C)CCNC(c2nnsc2C(F)F)=O)C)=O)nc2ncccn2n1 77365,C(=O)(C(C)(O)c1ccccc1)NCC(CC)NC(=O)Cc1csnn1 77366,c1(C(N2CC3(N(C(c4c(C)cc(F)cc4)=O)CC3)C2)=O)ccc(C)c(C)c1Cl 77367,c1(OC(C(=O)NC(C(C)NC(COCCCC#C)=O)C)(C)C)ccc(Cl)cc1C 77368,CN1C(=O)NC2(CCC(NC(=O)CCc3cnoc3)CC2)C1 77369,C(=O)(CC(C)CCCCC)NCCc1c(C(=O)NCCC=CC=C)c[nH]n1 77370,N1(C(C2CC(=C)C2)=O)CC(C)CCC1CNC(c1ccc(C(C)C)c(F)c1)=O 77371,C(=O)(C(O)C(C)(C)CC)NC1CC(C(=O)NCC(CCC)O)CC1O 77372,CN1Cc2ccc(C(=O)NC3CCCCC3N(C(=O)COCCF)C)cc2C1 77373,C1(CC(=O)NCCN(C(=O)C=C(C)C(F)F)CCOC)CNC(=O)C1 77374,O(P(C)(=O)CNC(=O)CC1(C)CCN1C(C12CCC(C1)C2)=O)CC 77375,c1(C(=O)NC2CCC(CNC(C3N(CCC)CCC3)=O)C2)ccc(F)c(O)c1 77376,c1(OCC(=O)NCC23C(CN(C(C(C)OCC=C)=O)C2)C3)cccc([N+](=O)[O-])c1 77377,CC(CNC(=O)CCC1CCCCN1C(=O)CCCC1CC1C)C(C)(C)C 77378,C1(CC)CCCCN1CCC12CC(C(=O)NCC=C(C)C)(C1)C2 77379,c1(OC)ccc(C(=O)NCCN(C(=O)CC(c2ccc(F)cc2)O)C)c(C)n1 77380,c1(C(N2CCCC(C3CCCN3C(=O)Cc3cnsc3)C2)=O)cccc(=S)n1O 77381,c1(C(=O)NC2C(NC(C(COC)N(C)C)=O)CCC2)ccn(C)c1C 77382,c1(CC)nnc(O)c(C(=O)NCC23CCCNC2CCC3)c1CC 77383,c1(C(N(CCNC(c2c(C)n(C(C)C)nn2)=O)CC2CC2)=O)cc(F)cnc1O 77384,C(=O)(C(C)(C)C(=O)OC)NCC(CC=C)NC(=O)CC1(C)CC1 77385,c1(CC)c(C(N2CCCC(NC(C3CC(C)(F)C3)=O)C2)=O)cnn1C(C)(C)C 77386,C1(CC=C)(C(=O)N(C(C)CC)C)CN(C(C2CCC(=O)C2)=O)C1 77387,C1(N(C(=O)CCCF)CC)CCCN(C(c2cn(C(C)C)nc2Br)=O)C1 77388,C1(C(=O)NC)CCN(C(=O)CCN(C(=O)CN2CCCC2C)C(C)C)C1 77389,C12(NC(c3cn(CC)nc3)=O)CCCC1N(C(c1c(C)cc(O)nc1C)=O)CC2 77390,N1(C(c2c(OC)scc2)=O)CCCCCC(NC(=O)CN2CCC(F)(F)C2)C1 77391,C1(NC(c2n(CC=C)nnn2)C2CCOCC2)CC(=O)N(CC(C)C)C1 77392,c1(C(N(CCN(C(C2C(CC)OCC2)=O)CC)CC)=O)ccn2cc(C)nc2c1 77393,c1(OC)ccccc1C(=O)NCC1(CCNC(C2(CO)CCCO2)=O)CC1 77394,CC(N=c1nc2scnc2c(NCCS(=O)(=O)C(F)F)[nH]1)c1cn(C)nn1 77395,c1(C(=O)NC(C)C2=CCN(C)CC2)cccc(P(C)(C)=O)c1 77396,C(=O)(CCCC(C)(C)C#N)N1C2(C(N(CC(CC)O)C)=O)CC(C1)C2 77397,C(C1(C)OCCc2ccccc21)NC(C1CN(C)CCO1)C 77398,N1(C(c2cc(C)on2)=O)CCCC(N(C(=O)CCCOc2ccccc2F)C)C1 77399,c12ccc(Cl)c(c1)N(C)C2=O.N1(C(C)C)CCCC(c2nc(C3CC3)no2)C1 77400,N1(C(C(CC)CO)=O)CCN(C(c2cccc(Cl)c2N)=O)CC1C(C)C 77401,CC(C)CCC(C(=O)NCC1(F)CC(CO)C1)NC(=O)CC=CC(C)(C)C 77402,C(=O)(C1=CC2C=CC(C1)C2)N1CC(C(=O)NC(C=C)C2CCC2)C(C(C)C)C1 77403,c1(C(N(CCC(C)=O)C)=O)ccc(-c2cn(CCCCCO)nn2)o1 77404,c1(C(=O)OC)cc(C(N2CC(NC(=O)CN=S(C)(C)=O)CC(F)C2)=O)cc(C)c1 77405,S(=O)(=O)(c1ccc2nc(N3CC4CC=CCC4C3)sc2c1)N1CC2C(C)(CC2)C1 77406,N1(C(C2(NC(c3c(C)n(C)nn3)=O)CC2C)=O)CCOCC(O)C1 77407,Cc1c(N)ccc(C(N2CCC(=CCNC(C3CCCC3(F)F)=O)CC2)=O)c1C 77408,Cc1nc(C(=O)N(C2CC(NC(C3(Cl)CC3(C)C)=O)C2)C)c(=O)[nH]c1C 77409,C1(CCC(N2CCC(CN(C)C(C3(F)CC3)=O)C2)=O)CC(C)(C)CO1 77410,N1(C(C(C(=O)OC)OC)=O)CCCC2(CNC(=O)CC(C)CC(C)C)CCCC12 77411,CC1(C)CC(NC2CNCCOC2)c2cc(F)ccc2O1 77412,c1(C(N2CCCC(NC(C3(C)CCC(OC)CC3)=O)C2)=O)cc(C)n(C)c(=O)c1 77413,CCCC(CC(=O)NCCCCOC(C)=O)NC(c1c[nH]nc1C(C)C)=O 77414,c1(C(=O)NC2(CNC(C(CC(C)C)(C)O)=O)CCC2)ccc2c(c1)C=CS2(=O)=O 77415,N1(C(C(C(C)C)NCOCC(F)(F)F)=O)CCOCC1(C)C 77416,c1(C(N(CCC)CCNC(=O)C(CC)C(F)(F)F)=O)ccc([N+](=O)[O-])c(C)c1 77417,c1(OC)ccccc1CN1CCC(C)(NC(=O)COc2ccc(CO)cc2)C1 77418,C12(NC(CCN(CCCO)C(C)=O)=O)CCC(C1)OC2C 77419,C1(NC(C(CC)C(C)C)=O)C2CCCN(c3cc(Cl)nc(C)n3)C2C1(C)C 77420,CC(O)C(C)(C)C(=O)N1CC2CC1(C(=O)NCCCn1cnnc1)C2 77421,c1(COC)ccc(C(=O)NC2CC(CNC(C3CCC(=O)C3)=O)C2)cc1F 77422,C1(CNC(c2ccc(C(C)O)cc2)=O)CCC(C)CN1C(=O)CCc1nncs1 77423,C=CC(C)(O)CC(=O)N(CCC(=O)N1CCC(O)C1CC)OC 77424,c1(C(=O)NCC=CCNC(C2CCC(C)O2)=O)c[nH]c2nc(Br)ccc12 77425,c1(C(N2C(C)CCC(NC(=O)C(=O)NCC3CC3)C2)=O)cc([N+](=O)[O-])ccn1 77426,c1(NC(C(N2C(CCC(=O)NC)CCCC2)=O)=O)cnc2[nH]cnc2c1 77427,C(=O)(C(O)CC(N)=O)NC1CC(CCNC(CCCOc2c(C)cccc2)=O)C1 77428,C1(NC(c2ccc(CO)cn2)=O)CCC12CN(C(c1ccc(C3CC3)cn1)=O)C2 77429,c1(C(=O)NC2(CF)CCN(C(CCC(=O)OC)=O)C2)coc2c(F)cc(F)cc12 77430,CCCS(=O)(=O)N1CCCC1C(C12CC(n3cc(CC4CC4)nn3)C1C2)OC 77431,c1(CNC(C2(CC)CCC2)=O)nc(CNC(C2CC(C(F)(F)F)C2)=O)cc(O)n1 77432,CCS(=O)(=O)c1ccccc1CC(=O)NCC1CC(NC(=O)OC(C)(C)C)C1 77433,C1(C(N(CCCCNC(CSCCC)=O)C)=O)CCC(=O)CC1C 77434,N1(C(C(CO)N(C)C)=O)CC2CC(C1)CN(C(c1n[nH]c3c1CCOC3)=O)C2 77435,C1(C)(CNC(COc2cccc(C)c2)=O)CN(C(=O)C(C)N(C)C)C(C)(C)C1 77436,n1(CCC)nccc1C(C(=O)NC(C)C)N(C)CCn1cncn1 77437,c1(C(=O)NCC(CC=C)NC(c2cc(C#N)c[nH]2)=O)nc2sccn2c1C 77438,N1(C(c2cc(COC)oc2C)=O)CC2(CC2)CC1CNC(C1(C)CC(OC)C1)=O 77439,N1(C(c2c(CC)nco2)=O)CCC2CCCN(C(=O)C=Cc3ccccc3)C2C1 77440,CC1CC(=O)NC(C(=O)NCC(O)CNC(=O)C(=O)NCCC(N)=O)C1 77441,c1(CNC(C2CCC(F)(F)C2)=O)cccnc1CNC(C1CCCOC1)=O 77442,CCCCS(=O)(=O)CC(=O)NC1CC1NC(c1cc(N2CCOCC2)cc(F)c1)=O 77443,CCC(C)(C)C(O)C(=O)NCC1CN(C(=O)COC2(C)CCCC2)CC1(C)C 77444,CN1CCn2nc(C(NC3CCc4ccc(CC(=O)O)cc43)=O)cc2S1(=O)=O 77445,c1(C(N(CC(CC)NC(C2CC2C(C)(F)F)=O)CC)=O)ncc(Br)cc1F 77446,CC1CC(CC(=O)NC(C)Cn2cnnc2)CN1C(c1ccnc(CO)c1)=O 77447,c1(C(=O)NCC2CC(NC(CCC=CC)=O)CC2O)cc2c(nc1O)CCC2 77448,c1(C(=O)NCCN(CCC)C(C2(C)CC2C)=O)ccc(-n2ccnc2)c(C)c1 77449,Cc1n[nH]c(=NCC2(C(C)C(c3ccco3)=O)CC2)o1 77450,C(=O)(C1OCCn2ccnc21)NC1C(NC(c2ccc3c(c2)CC3)=O)CCC1 77451,CCCCC(CNC(=O)CCC(C)SC)NC(C1(SCCC)CCC1)=O 77452,c1(-n2c(-c3scnc3Cl)nc(-c3ccc(O)cc3)n2)nc2ccccn2n1 77453,N=c1nc(CO)[nH]c(=NC2CCCC23CN(C(c2cn(C(C)(C)C)nn2)=O)C3)[nH]1 77454,C1(C)(C(N2C(C(N(C3CCC(F)(F)C3)C)=O)CCC2)=O)CCC2CC2C1 77455,C1(C(=O)NCCn2cc(CNC(C(C(C)C)C)=O)nn2)CCCCNC1=O 77456,Cc1cc(Cl)c(C(N2CCCN(C(c3n[nH]c4c3CCO4)=O)CC2)=O)cc1C 77457,C1(C)(CNC(C(C)OCCCC)=O)CCN(C(c2cc(N)cc(F)c2)=O)CC1 77458,C(=O)(CCC(C)(C)[N+](=O)[O-])NC1CCN(C(CNC(=O)OC)=O)CC1C(N)=O 77459,c1(C(=O)NC2(C)CN(C(c3ccc(CO)cc3)=O)C2)ccc(N)c(O)c1 77460,c1(NC(N2CCOC(CC3CC3)C2)=O)ccc(-c2nn[nH]n2)c(F)c1 77461,CCC(CC)C(c1nnnn1Cc1nnn(C)n1)NCCC1COCCCC1 77462,N1(C(C23CC(CCC)(C2)C3)=O)CCCCC(CNC(=O)C(C)n2cncn2)C1 77463,Cc1cc(C(N2CC(NC(c3cc(Cl)ccc3N)=O)CC(F)C2)=O)c(Cl)cc1F 77464,CCCC(CC)CC(=O)NC(C)CN(C(C1CC1CC)=O)CC 77465,C1(C(=O)NC(c2cccnc2)CO)(SC)CN(C(C2CC2Cl)=O)C1 77466,C(=O)(CCN)OC.C1(CC(=O)C(=O)OC(C)(C)C)OCCCOC1 77467,C1(CC(=O)C(=O)OC(C(=O)NOC(C)(C)C)C)CC(NC(=O)NCC)C1 77468,c1(NC(CCC(=O)OCCCC(C)=O)=O)ccc(C)c(OCCF)c1 77469,C1(CCC=C)(C(=O)NC(CCCC)c2ccccc2)CN(C(=O)C=CCO)C1 77470,c1(OCC)cc(C(=O)NC2(CNC(C3CCC3(C)C)=O)CC2)on1 77471,c1(NC)ccccc1NC(=O)C(CC1CC1)NC(c1cn(CCO)nn1)=O 77472,N1(C(Cn2cc(C(C)O)nn2)=O)CCC2CN(C(c3n[nH]c(=N)[nH]3)=O)CC2CC1 77473,CC(C(F)F)=CC(=O)NCC1(NC(=O)Cc2cnoc2)CC1 77474,c1(CNC(c2cnn(C)c2C)c2n(C(CC)C)nnn2)cc(F)ncc1C 77475,C(=O)(C(C)S(C)(=O)=O)N(C(CNC(C=C(CCC)C)=O)C)C 77476,c1(OC)ccc(CNC(=O)CC2CCCN2S(=O)(=O)Cc2ccccc2)cc1O 77477,CN1CCN(C(=O)C(C2CCCCC2)O)CC1C(=O)NCC1(C)NC(=O)NC1=O 77478,c1(OCC(=O)N(C)CC2CCCN2C(c2cc(C(F)F)on2)=O)ccccc1F 77479,N1(C(C=CCCC(C)C)=O)CCC(N(C(c2cscn2)=O)CC2CC2)CC1 77480,N1(C(CCCC=C)=O)CC(CN(C)C(c2ccc(CC(C)C)nc2)=O)C2(CC2)C1 77481,C(=O)(CCC(=O)NCC(=O)NCC1CCCCC1OC)NCCC 77482,C1(CC#C)(C(=O)NCC(C)(CC)NC(c2cncc(Cl)c2)=O)CC=CCC1 77483,c1(C(=O)NCC2(CNC(c3cc(CC)no3)=O)CC2)cc(C#N)c[nH]1 77484,c1(C(=O)NC(CNC(c2ccc(C)o2)=O)C2CCC2)cc(N)ccc1[N+](=O)[O-] 77485,C(=O)(CC(C)(C)CNC(=O)C1=C(C)CC1)N1C(CC(=O)NC)CC1 77486,c1(C(C(=O)NCCCOC(C)C)N(CC=C)C)cccc(Cl)c1 77487,CC1C(NC(C2CCCCCC2)=O)CCN1C(c1cccc(C2CCCC2)c1)=O 77488,N1(C(C(CCC)C)=O)CCC2(CC1)CCN(C(C1CC13CCOCC3)=O)C2 77489,N1(C(C(C2(C)CC2)NC(CN(C(COC)=O)C)=O)=O)CCC(CN=[N+]=[N-])C1 77490,CC(C)CC(C)C(=O)N1CCCC(F)(C(=O)NCCCc2cc[nH]n2)C1 77491,N1(C(CN2CCOCC2Cc2ccn(C)n2)=O)CC2CC1(C(=O)NOCCO)C2 77492,c1(C(N(C)CC2N(C(C(CN(C)C)O)=O)CCC2)=O)ccsc1C#N 77493,c1(C(=O)NC2C(CN(C(C3(CC)CCC3)=O)C)CCC2)c(C)nc(C)n1O 77494,C1(CNC(C(C)OCCC#C)=O)N(C(=O)CCC2CCCC2)CCC1(C)C 77495,c12ccc(c(O)c1)N(C(=O)CCC(C)N(C)C)CCN(CC)C(=O)C2.OC 77496,c1(C(=O)NCC(CN(C(C2CC2F)=O)CC)(C)C)ncccc1Br 77497,C1(NC(CN(C)C(N)=O)=O)(CNC(=O)CC2CCCOCC2)CC(F)(F)C1 77498,c1(OC(C)(C)C(=O)NCCC(=O)Cc2ccc(F)cc2)cc(F)cc(F)c1 77499,C1(CNC(COCCCOC)=O)CC2CCC(C1)N2C(=O)C(C)(C)C(C)C 77500,Cc1ccc(O)c(C(=O)N(CCCOCCNC(=O)CNC=O)C)c1 77501,c1(CC)nn(C)c(Cl)c1C(=O)NCCCC1(NC(c2cccc(C#N)c2)=O)CC1 77502,N1(C(c2c(C)n(C)nn2)=O)CC(CNC(c2ncc[nH]c2=O)=O)CC(C)(C)C1 77503,C1(NC(C2(CC=C)CCOC2)=O)CCN(C(=O)Cc2cccc(C)c2Cl)C(C)C1 77504,c1(C(=O)NC(C2CCCN2C(C2CC(F)(F)C2(C)C)=O)C)cc2n(n1)CCCO2 77505,NS(=O)(=O)c1ccc(C(=O)NC2CCCC23CN(C(c2cnns2)=O)C3)o1 77506,Cc1nn(CCO)cc1C(=O)NC(C)(CNC(=O)C(C)CC1CCCC1)C(C)C 77507,c1(C(=O)NCC2CCC(C)N(C(c3ccnc(O)c3)=O)C2)ccc(Cl)c(Cl)c1N 77508,n1(CC(=O)C(CCCNC(C2CCN(C(C)=O)CC2)=O)=O)ccc(C)cc1=O 77509,C1(NC(CC(C)(C)OC)=O)CCN(C(=O)C(F)OC(F)(F)F)CC1OC 77510,c1(C(N2CCCC(c3nc[nH]n3)C2)=O)nc(=O)c2c(Br)cccc2[nH]1 77511,C(=O)(CCC(=O)NCC1(C)CCN(C(=O)CC(CC)SC)C1)NCC 77512,C1(CNC(CSCC#C)=O)CN(C(c2cccc(F)c2CC)=O)CCC1(C)C 77513,c1(N2CCC(CCOC)(NC(c3cc(C#N)c[nH]3)=O)C2)ncnc(C)c1F 77514,N1(C(CN2CCCC(CC)C2)=O)CC=C(CNC(=O)CN2CCNC(=O)C2)CC1 77515,CCC(CNC(c1ncccc1F)=O)(CC)C(=O)NC1CC1CC 77516,N1(C(CC)=O)CCOC2(CCC(NC(c3cc(C#N)ccc3Cl)=O)CC2)C1 77517,CC1CN(C(C)CNC(=O)CCC(=O)Nc2ccc(F)cc2)CC(C)O1 77518,C1(CC(N2CCC(NC(C(C)OCC#C)=O)(CF)C2)=O)Cc2ccccc2N1 77519,N(C(=NCCF)NCC12CC(C1)C(C)(C)O2)C1C(C(C)C)C1 77520,c1(OC)cccc(OCCC(N2CC3(NC(c4ncoc4C)=O)CC2C3)=O)c1 77521,c1(N2CCC(CC=C)(NC(=O)CN3CCOCC3)C2)ncnc2c1CCC2 77522,N1(C(c2c(N)ccc(C)c2F)=O)CCCC12CCN(C(c1c(C)n[nH]c1C)=O)C2 77523,C1(C(N(CC(C)(C)NC(C2(CCCC)CC2)=O)C)=O)CC(=O)NC(C)C1 77524,c1(NC)ccc(CNCC2=CCCOC2)cc1[N+](=O)[O-] 77525,C(=O)C1CCCn2c(Br)cnc21.N1(C(=O)OC(C)(C)C)CCC1(C)C(=O)NC 77526,Cc1cc(N2CCN(C(C3CCCC4(CC4)C3)=O)CCC2C)n2ncc(C)c2n1 77527,C1(O)(CNC(COC2CCN(C)CC2)=O)CCCN(C(c2cnns2)=O)CC1 77528,N1(C(CC2(CN(CCC(=O)NC3CC3)C)CC2)=O)C2CCC1CC(CCF)C2 77529,C1(OC)CC(NC(=O)C2=C(Cl)CC2)C12CCN(C(=O)C(C)(C)C(F)F)CC2 77530,c1(CC(=O)N(CCCNC(c2nc(C)sc2C)=O)C(C)C)cc(F)ccc1Cl 77531,C(=O)(C(O)C(C)(C)c1ccccc1)NC(C)CCNC(=O)COCCF 77532,c1(OC)ccccc1C(C(=O)NCC1CCCO1)N(CCOCCO)C(C)C 77533,O=C(CC(=O)c1ccccc1)OCCCSCc1ccccc1 77534,C1(N(C(=O)Cn2ccsc2=N)C)CCCN(C(=O)CC2CCCCCO2)CC1 77535,C1(OC)CCCN(C(C2CC(O)CN2C(c2ncncc2N)=O)=O)CC1 77536,c1(SC)nc(O)nc(C)c1C(=O)NCC1CCN(C(=O)C(C)C(C)(C)C)C1 77537,C1(C(N(CC(=O)NCC(C)(C)C(F)F)C2CCC2)=O)CC2C=CC1CC2 77538,Cc1ccc(C(=O)NC(C)(C)CC2CCN(C(C3(O)CC3(C)C)=O)CC2)nc1 77539,n1(CC)cnc2[nH]c(=NCC3CCCC3)nc(N3CCCC(n4ccnn4)C3)c12 77540,N1(C(C2NC3CC2C3)=O)CCOC(Cn2cc(-c3cscn3)nn2)C1 77541,C1(NC(c2ccc(C(C)=O)cn2)=O)CCC(C)N(C(C2CCOC2)=O)C1 77542,C1(C(=O)NCCn2ncc(C)c2)CCCN(C(c2scnc2C(C)C)=O)C1 77543,N1(C(C2C(COC(=O)OC(C)(C)C)CCC2)=O)CC2CCCN2CC1COC 77544,C1(C(N2CCC(CF)(NC(c3cnco3)=O)C2)=O)(CC)CCNC1=O 77545,c12cccc(c1)S2.Cc1nc(C(=O)N(C)CCN(C(=O)C(C)C2CC2)C)cs1 77546,c1(NC(C(C)OC(CCC(C)NS(CC)(=O)=O)=O)=O)cccc([N+](=O)[O-])c1 77547,c1(OCCCC(=O)N(C(c2c(C)noc2C)C(F)(F)F)C(C)C)cc(Cl)cc(Cl)c1 77548,N1(C(=O)C2CC2)CCN(C(=O)NC2C#CCCCCC2)C(CCO)C1 77549,c1(C(=O)NCCCN2CCN(C(C3N(N=O)CCC3)=O)CC2)cc(O)ccc1F 77550,c1(C(=O)NCC2CCN(C(c3c(CC)nco3)=O)CC2)ccc2occ(C)c2c1 77551,C#CCC(C(=O)NOCCCOC)NC(C1CC1CC(C)C)=O 77552,c1(CNC2C(C(=O)NCCC#N)CCCC2)cc(O)c(O)c(O)c1 77553,C1(NC(c2scc(COC)c2)=O)C2CCN(C(c3c(CO)n[nH]c3C)=O)CCC12 77554,C12(NC(CN(C)C(N)=O)=O)CCC(CC1)N(C(C1CC13CC(O)C3)=O)C2 77555,c1(C(=O)NCC2C=CCN2C(=O)C=CBr)c[nH]c2ccc([N+](=O)[O-])cc12 77556,N1(C(c2c(C)nc3sccn32)=O)CCCC2(CCCN2C(c2ccnn2C)=O)C1 77557,C1(NC(CCCCOC)=O)CC2CCC1N2C(=O)C(C)Cc1cccc(Cl)c1 77558,C#CC1(OCC(=O)NCC2CCN(C(=O)C(CO)c3ccccc3)C2)COC1 77559,C(N=c1cccc(S(=O)(=O)NC2CCC=C2Br)[nH]1)C1CC(C)(C)OC1 77560,C=CC1(C(=O)NCC(F)(CC)CC)CCN(C(=O)CC(CC)CC)C1 77561,c1(CC(=O)NCC2CCN2C(c2cc(C(F)F)no2)=O)ccccc1Br 77562,c1(C(=O)NC2CCCCN(C(CCC=C)=O)C2)cc(S(N)(=O)=O)c(F)cc1OC 77563,C(=O)(C1=CS(=O)CCC1)N1CC(N(C)C(C2CC(=CCc3ccccc3)C2)=O)C1 77564,c1(C(N2CC(NC(=O)Cc3cccnc3Cl)CC(C)C2)=O)c[nH]c2ccccc12 77565,N1(C(c2cnc(OC)s2)=O)CCN(C(c2cnc3n2CCC3)=O)CC(C)(F)C1 77566,c1(CCC2(N(C)C)CCCC2C(=O)O)ccc(F)cc1F.c1(CC)c2cnn1[nH]2 77567,N1(C(c2c(CNC(CCc3ncn(C)c3)=O)c[nH]n2)=O)CCCC(N=[N+]=[N-])CC1 77568,N1(C(C2CCCCO2)=O)CC2CC(C(=O)NOC3CCCC3)(C2)C1 77569,C1(C(N(C(C)C)CCN(C)C(c2ccoc2Cl)=O)=O)CCn2c(O)nnc2C1 77570,C1(C(=O)NCC(C)(C)C2CCC2)C=CCN1C(=O)COCCN(C)C 77571,C1(CNC(c2n(CC)cnn2)=O)CCCCN1C(C1OCCOC1C(F)(F)F)=O 77572,c1(C(C)NC(=O)OC(C)(C)C)ccc(OC(F)F)nc1.C12CC(C)(C1)NC2=O 77573,C(=O)(C(C)N=c1[nH]c2ccccc2s1)NC1CC(CNC(CCCCC#C)=O)C1 77574,CC(C)(C)CCNC(N1C(C(=O)Nn2cc(C#N)cn2)COCC1)=O.C1CC1 77575,Cc1cc(C(O)C(C)NC(=O)Nc2cccc(-n3cnnn3)c2)ccc1F 77576,CN1CC(C(N2CC(F)(CNC(=O)COc3ccon3)C2)=O)CC1=O 77577,C1(CC(=O)N(C)CCN(C(=O)CN2CCC(CO)CC2)C)Cc2ccccc2O1 77578,N(C1CCC(NC(C2(CO)CCCC2)=O)c2ccccc21)C(c1c(C)[nH]cc1)=O 77579,C1(CNC(COCCC=C)=O)CCC2CN(C(=O)CC3CCSC3)CC12 77580,c1(C(=O)NCCCN(C(CC2(OC)CC2)=O)CCO)cc2cc(Cl)ccc2s1 77581,C1(C(N(CCCNC(CNS(CC)(=O)=O)=O)C)=O)CC(F)(F)C1(F)F 77582,Cc1ccc(OCC(=O)NCC2(C(N)=O)CN(C(=O)CSCC(C)C)C2)cc1 77583,C(N=c1[nH]cc(Br)c2ccc(Br)cc12)C1C(O)COC1 77584,c1(C(=O)NC(c2cccnc2)C(=O)NCc2[nH]nc(C(C)C)n2)ncncc1Cl 77585,C1(CNC(C(N2CCC(O)CC2)C)=O)CCCCC1NC(=O)C(O)C1CCC1 77586,Cc1cc2c(C(N3CC(NC(C4CC4(C)C)=O)C4(CCC4)C3)=O)nccn2n1 77587,N1(C(CCS(C)(=O)=O)=O)CC(C)(CNC(c2csc(C3CC3)n2)=O)CC1(C)C 77588,N1(C(=O)NC(c2ccc(C(C)C)cc2)C)CCCC(C#N)(C(=O)OC(C)(C)C)C1 77589,C(=O)(C#CC1(C)CC1)NC(CC)CNC(=O)CCC1CC1(Cl)Cl 77590,CCCC(O)CC(=O)NCC=CCNC(C1CC2CCC(C1)S2)=O 77591,C12(NCc3c(C(=O)OC)noc3)CCN(C(=O)Cc3ccccc3)CC1C2 77592,CC1CN(C(=O)C=CC(C)(C)C)CC(C)CN1C(c1nscc1N)=O 77593,c1(C(=O)NCC23CC(NC(C#CC(=O)N(C)C)=O)(C2)C3)nnc2ccccn12 77594,Cn1nc2c(c1C(N1CC(NC(C3CCOC3)=O)C(C(F)(F)F)C1)=O)CCC2 77595,C1(N(C(Cn2c(C)ncc2)=O)C)CN(C(C2CC(F)(CO)C2)=O)CC1O 77596,c1(CC)cc(Cl)ccc1C(=O)NC1CCC1CNC(c1ccccc1C)=O 77597,C1(CC=C)(C(=O)NC2CCCSCC2)CCN(C(C2CC(F)C(=O)N2)=O)C1 77598,C1(N(C(C(c2cnn(C)c2)OC)=O)C)CCC(NC(C2CC(C)(F)C2)=O)CC1 77599,c1(NCc2nn(CC)nc2C)cc2c(I)cnn2cn1 77600,C(=O)(C(F)(F)CC(C)C)N1CCN(C(Cc2c(SCC)cccc2)=O)C(CF)C1 77601,O=C(CCC(F)(F)F)NCC1C(O)C(O)CN1C(=O)C=CSCc1ccco1 77602,N1(C(C2(CC)CCCC2)=O)CCC(C)C(N(C(=O)CCC2(C)CC2)C)C1 77603,N#CC1(C(N2CC3CC3(CNC(=O)CCc3cnc(O)[nH]3)C2)=O)CC12CCC2 77604,c1(C(=O)OC)cc(C(=O)N(C(=O)C(=O)N(C)C2CC2)C(c2nccn2C)C)ns1 77605,c1(NC(C)=O)ccc(F)c(C(N2CCC(N(C(=O)CC3CC3(C)C)C)C2)=O)c1 77606,CC1=C(CNC(=O)C(C2CCN(C(=O)CC3CCC(=O)C3)CC2)C)CCC1 77607,c1(C(N2CC3CC(NC(C=CC=CC)=O)C3C2)=O)c(N)c(F)cc(F)c1F 77608,c1(C(=O)OC)cc(C(N2CCCC(C(F)(F)F)C2)C(=O)NCCCF)c(C)s1 77609,C=CC(CC)CC(=O)N1CCOCC1CN(C)C(c1cn(C(F)F)cn1)=O 77610,CC1(CNC(=O)CC2CC(O)CN2C(=O)COC2CC=CC2)CCCCCC1 77611,C1(N(C(c2sc(CC)c(C)c2)=O)C)CN(C(C23CCC(C2)C3)=O)CC12CC2 77612,c1(C(C)N(C(=O)NCCc2ccnc(Cl)c2)CC2CC2)cccc(F)c1 77613,CC(C)C(O)CCNC(=O)C(CCOCCO)NC(c1cc(=N)[nH][nH]1)=O 77614,c1(C(=O)N)c(C)cc(C)nc1S.n1(C2(C(N3CC(OC)C3)=O)CC2)ccc(C2CC2)n1 77615,C1(CC(=O)N(C)CC2CCN(C(=O)CS(N)(=O)=O)C2)CCC2(CCC2)O1 77616,CC1CC(NC(c2ccco2)=O)CN1C(C1CCCC(O)C1)=O 77617,c1(OC)ccc(CCC(=O)N2CC(NC(c3c(N)cnn3C)=O)C2)cc1F 77618,C1(NC(c2cc(CCC)no2)=O)CCN(CC2(CC(=O)NC)CC2)CC1 77619,c1(CCC(=O)OC(C2C(CCC(Br)(c3ccco3)OC)CC2)=O)csc(C(C)C)n1 77620,Cc1cc(C)c(C)c(C(=O)NCC2CCN(C(=O)C=CC=CCO)C23CC3)c1C 77621,c1(OC(C(=O)NCCCC(C)NC(C2(C=C)CCC2)=O)C)cccc(C)c1C 77622,C1(C(N(C(c2ccccc2)CNC(c2ccc(C(N)=O)s2)=O)C)=O)CC12CCC2 77623,C(=O)(CN=c1cc[nH]cc1)N1CC2C(CNC(c3c(C)scc3)=O)(C2)C1 77624,c1(C(N2CC(N(C)C)C(C)(C)C2)C(=O)NC)cc(Br)cnc1OC 77625,N1(C(C(C)Cc2ccc(F)cc2)=O)CC2CC(NC(=O)C3CC3)CC1C2 77626,N1(C(CSCCN(C)C)=O)Cc2ccccc2C1C(=O)N(C)C1CC1 77627,c1(CC)cc(C(=O)NC2CCN(C(=O)C(CC)CC)C2c2ccccc2)c(C)o1 77628,C1(C(N2CCC(C(=O)NCC3CC(OCC)C3)C2)=O)CCCC(C#N)C1 77629,C(=O)(C1=CCC2CCC1N2C(=O)C(C)(C)CC(F)F)NCC(C(C)C)(C)O 77630,CC(=O)CCC(=O)NCC(C(C)(C)C)NC(c1ccc(-c2ccco2)o1)=O 77631,C(CC(C(=O)NC(C)C(C)SC)NC(=O)CC1(O)CC1)SC 77632,C1(C)(CNC(c2cnn(CC)c2C)=O)CCCN(C(c2c(C#N)cnn2C)=O)C1 77633,Cn1nnc(CNC(=O)C(C)(C)C#N)c1C(N1CC(C)(C(F)(F)F)C1)=O 77634,N1(C(C(C#C)(C)C)=O)CCOC2(CCC(NC(=O)CCCCN(C)C)CC2)C1 77635,c1(C(=O)NCC=CCNC(C(Br)=C(C)C)=O)nn(C)c(=O)c2ccccc12 77636,c1(CCNC(=O)CCC2CCCC2)csc(Cc2nn[nH]n2)n1 77637,N1(CCC#C)CCC(C(=O)NC2CCCC(CNC(=O)C(COC)CC)C2)CC1 77638,CCC(C(=O)NCCCN(C)C(C1CC1[N+](=O)[O-])=O)OC1CCCCC1 77639,c1(NC)ccc(C(N2CCCC2C(C)NC(=O)C(C)SC)=O)cc1 77640,c1(CN2CC3C(C(=O)Nc4c(OC)cccc4Br)C3C2)cc(Br)cc(F)c1O 77641,CC1CN(C(c2c(Cl)ncn2C)C(=O)NCC2CCOC2)CCN(C)C1 77642,NC(=O)CCC(=O)NC1CCCC1NC(c1cccn1CCc1ccccc1)=O 77643,C1(C(=O)NC2(CSC)CCC2)CCCCN1C(=O)Cn1cccc1 77644,C12SC3C=CC1CC3CN(C(=O)OC(C)(C)C)CC(C(C)C(F)(F)F)CN2 77645,C1(CNC(C2CCN(CCC#C)CC2)=O)CC2CCC1N(C(=O)C(C)C1CC1)C2 77646,N1(C(CCCCCNC(c2n[nH]c(CC)c2C)=O)=O)Cc2ccncc2C1 77647,c1(NC(C(N2CCC3(C=CCO3)C2)C)=O)nc2ccc(F)cc2s1 77648,N#Cc1ccncc1N1CCN(C(=O)CCc2cccs2)CC1 77649,c1(C(N(C2C(C)CCN(C(c3cc(C)[nH]n3)=O)C2)C)=O)cnc(O)c([N+](=O)[O-])c1 77650,c1(-n2cc(C(=O)NC(C3CN(C(=O)Cn4cncn4)C3)C)nn2)ccccc1Br 77651,c1(CC(=O)NCCNC(C(c2cc(C)cc(F)c2)C)=O)ccccc1S(C)=O 77652,C(=O)(CCCCC(F)(F)F)N1CC(N(C(COC(CC)(C)C)=O)C)C2(C1)CC2 77653,C1(C(=O)NCC(O)CC(F)(F)F)CCN(C(=O)C2CCCOCC2)O1 77654,C#Cc1cncc(CNC(c2ncc(OC)cc2F)=O)c1 77655,C(c1cscn1)=CC(=O)NC1CC1CNC(c1coc(C2CCC2)n1)=O 77656,C(=O)(C1=CCN(C(=O)CN2C(=O)CCCC2=O)C1)Nc1c(CC)cccn1 77657,N1(C(c2cc(Br)ccc2C)C(=O)NCCC)CC2CCC(C1)C2C#N 77658,C1(C)(NC(c2cc(-c3ccc(C)o3)[nH]n2)=O)CCN(C(=O)C2=CC(C)CC2)CC1 77659,c1(C(=O)NCCC2CCCN2C(=O)CCC=CBr)cnc2c(c1)CCOC2 77660,CC(Cc1cccc(F)c1)CC(=O)NC(CO)C(C)NC(=O)CSC(C)(C)C 77661,C1(C)(C(N(CC(C)(C)NC(C2C(C(=O)OC)CC2)=O)C)=O)CCOC1 77662,CC1CN(C(=O)CCOCCN(C(=O)C(c2ccn(C)n2)C)C)CC1C 77663,c1(CN(C2(C)CCCC2)Cc2ccccc2)cc2ccccc2nc1O 77664,c1(C(=O)NCCn2cc(C(CC)N(C)C)nn2)cc(C)c2nc(C)nn2c1 77665,c1(C(=O)NC2(CCNC(C(COC)N(C)C)=O)CCC2)cn2cnnc2cn1 77666,Cc1cc(=NC(=O)C(=O)NC2CC3CN(C(=O)CCc4nccs4)CC3C2)[nH]o1 77667,Cc1cc(=NCc2nc3ncccn3n2)[nH]c(N(C)Cc2cc(C)on2)n1 77668,N1(C(c2cc(C(C)C)[nH]n2)=O)CC2CCCC(C1)C2C(=O)NCc1cc(C)on1 77669,C1(C)(NC(C(n2c(C)ccn2)C)=O)CCCN(C(=O)C2=COCCO2)C1 77670,Cc1ccc2c(c1)C(C(=O)N1CCN(C(c3cc(=O)cc[nH]3)=O)CC1C(C)C)C2 77671,c1(OC)ncc(Br)c(=NC(CNC(C2COCCO2)=O)C(C)C)[nH]1 77672,N1(C(CC2CC(C)C2)=O)CCC(CO)CC1CNC(=O)CCn1cccnc1=O 77673,N1(C(c2cn(C)nn2)=O)CCN(C(=O)C=CC2CC2)C(c2ccnn2C)C1 77674,N(C1CC2(CCCC2)c2ccccc21)C(C(CC)n1cc(C2CCCC2)nn1)=O 77675,c1(C(N(CCNC(c2cccc(N)c2O)=O)C2CC2)=O)cnn2c1CC(F)(F)C2 77676,c1(CC)nc(NC2(CNC(=O)C(C)(C)CF)CC2)c2ccsc2n1 77677,C1(CNC(C2ON=C(C)C2)=O)(CNC(c2csc(C)c2)=O)CCCCC1 77678,C1(C(N(C2(C)CCCC2)C)=O)CN(C(C2CC(C3CC3)C2)=O)CCO1 77679,C1(NC(c2cc(F)c(OC)c(Br)c2)=O)C(C#N)CCC12CCOCC2 77680,n1(CCOC)nc(C(=O)NC(CNC(=O)CC2(O)CCCC2)C2CC2)ccc1=O 77681,N1(C(c2ccc(Cl)o2)=O)CC2(CCCC2)C1C(N1CCC2C(O)CC12)=O 77682,C(C(C)(C)CCNC(c1csc(CO)n1)=O)NC(Cc1c(C)ncs1)=O 77683,c1(OC)cccc(CC(N2CCC(N(CCO)C(c3c[nH]ccc3=O)=O)C2)=O)n1 77684,C1(CNC(c2c(OC)nsc2)=O)CC2CCC1N(C(C1CCC3CC3CC1)=O)C2 77685,N12CCCC(C3CN(C3)C(=O)C3(CC3)C1=O)C2.C1(COCC)C2CCCCC12 77686,c1(CC(=O)NCC(CC)N(C(c2c(CC)c[nH]n2)=O)C)cncc(C)c1 77687,CCCC(C)C(=O)NCc1cc(C(=O)NC(C2CCOC2)CO)ccn1 77688,C12(CC(=O)N(C)CC3(C)CC3)CCC1CN(C(C1(C3(O)CCC3)CC1)=O)C2 77689,CC(C)C(C(=O)NCCn1cc(C2(O)CCOC2)nn1)n1cc(Br)cn1 77690,C(C(CNC(c1n[nH]c2c1CCC2)=O)S(C)(=O)=O)NC(C1OCC(C)(C)C1)=O 77691,N1(C(Cc2cn(C)nc2)=O)CCC2(NC(=O)CC(F)(F)C(F)F)CCCCC12 77692,N1(C(c2occ(C(C)=O)c2)=O)CCC(C2CCN(C(=O)C(C)N3CCC3)CC2)C1 77693,C12(C(=O)NC(C3CCN(C(=O)CC4CCOCC4)CC3)(C)C)CCOC(C)(C1)C2 77694,c1(C(N2CCC(NC(c3c(C)nn[nH]3)=O)(CF)C2)=O)cc(Cl)cc(Cl)c1F 77695,C(=O)(C(O)CC(F)F)N1CCCC(NC(=O)C=CCCc2ccccc2)C1 77696,C1(NC(=O)Cn2cnnn2)(CNC(C2CC3(C2)CC(O)C3)=O)CC2CCC1CC2 77697,C1(C2CN(C(C3CCN3Cc3ccccc3)=O)C2)(NC(=O)CC2CCCO2)CC1 77698,c1(C(N2CC(OCCNC(CNS(CC)(=O)=O)=O)C2)=O)nnc(C)s1 77699,c1(C(N2C(CNC(CCCOC(C)C)=O)CC(O)C2)=O)nccn2ccnc12 77700,n1(C(C)C)ncc(C(=O)NC2CC(CNC(=O)C(C)c3cccs3)C2)c1N 77701,c1(C(C)=O)cn(C)nc1C(=O)NC(c1ccc(C)cc1)CNC(c1cnsc1)=O 77702,Cc1ccc(C(C)NC(C2(C)CCN(C(=O)CCn3ccc(C)n3)C2)=O)cc1 77703,N1(C(N(c2nc(C)n(C)n2)CC)=O)CC(c2noc(C(F)(F)F)n2)OC(C)C1 77704,CC(C)(F)C(C)(F)C(=O)NCC1(O)CC(CNC(c2cc(O)nc(Cl)c2)=O)C1 77705,c1(CCC)n[nH]cc1C(=O)NC(COC)C(=O)N(CCC(C)(C)O)C 77706,n1(CCC)c(CNC(Cc2ccc(Cl)cc2)C(C)(C)C)nc2cc(NC)ccc12 77707,c1(-n2cc(C3C(OC)CN(C(c4cnncc4N)=O)C3)nn2)ccc(C)c(F)c1 77708,c1(CNC(CCC2CCC(NC(C3CCC(CC)O3)=O)C2)=O)cc(C)nc(O)c1 77709,N1(C(C(C)(C)C2CCN(C(C3CN(c4ncco4)C3)=O)C2)=O)CCC(C)(CO)C1 77710,c1(C(N(C2CN(C(C(C)CF)=O)CC2(C)C)C)=O)c2ccccc2nn1C 77711,c1(C(N2C3CC(CNC(C4C(=C)CC4)=O)CC2CC3)=O)c[nH]c2ccc(F)cc12 77712,N1(C(C(C(C)SC)O)=O)CCC(C)(CNC(C2CC(OC(F)F)C2)=O)CC1 77713,c1(CC(=O)NC2C3CN(C(C4CCCOC4)=O)CC23)c[nH]c2cnccc12 77714,Cc1cc(C)n(C(C)CC(=O)NC2C=CCN(C(=O)CSc3cn[nH]c3)C2)n1 77715,Cn1nc([N+](=O)[O-])cc1C(=O)NCC1C2CC2CN1C(C1CCS(=O)(=O)CC1)=O 77716,C1(N(C(=O)CCn2cc(C3CCCCO3)nn2)C)CNC(=O)C12CC2 77717,S(=O)(=O)(c1ccc(F)c(C(=O)NC2CCC(NCc3ccoc3)C2)c1)N(C)C 77718,c1(CC(=O)OC)cccc(C(=O)NCCCNC(=O)C(c2ccc(Cl)s2)C)c1 77719,C(=O)(CC(CC(C)C)NC(=O)C(F)(F)CCCC)NCC(CC#C)(C)C 77720,Cc1cc(C)n(CCNC(=O)C(CC2CC2)NC(=O)COC2CCOC2)n1 77721,c1(C(N2CCCN(C(CCC(=C)Br)=O)CC2)=O)cc(OC)c(OC)cc1F 77722,Cc1cnc(C(=O)NCC(O)CN(C)C(c2nocc2C(C)(C)C)=O)c(F)c1 77723,N1(C(C(=O)NC(C)C)=O)CC2CCN(C(c3ccn4nccc4c3)=O)CC2C1 77724,N1(C(CSCCC)=O)CCCC(C2CCN(C(=O)C(C)N(C)C)CC2)CC1 77725,c1(CN(C(=O)NCCCN(C(CCC)=O)CCO)C)conc1C1CC1 77726,C1(CNC(c2c(SC)snn2)=O)CC2(CO1)CN(C(C1CC=CC1)=O)C2 77727,N1(c2cnc(C(C)=O)c(C)n2)CCCC1C1CCCCN1C(=O)C(C)CO 77728,C1(CC(=O)NC(C)CCNC(=O)COCCN(C)C)CCC12CCC2 77729,Cc1ncnc(C)c1OCC(=O)NC1CCC(NC(C2CS(=O)(=O)CCO2)=O)C1 77730,N1(C(C2CCC(=C)CC2)=O)CCCC(C)(C)C1C(N1CC(CN=[N+]=[N-])C1)=O 77731,O=C1NC(C2CCOC2)C(=O)N1CC1CC2CCC1CC2 77732,c1(OC)oc(C)nc1C(=O)NC(C)CC(C)NC(c1c[nH]nc1C(C)(C)C)=O 77733,CCC(C)(C#N)C(=O)N(C)CC=CC(N1CCC(C)CC1C)=O 77734,C1(C2CN(C(=O)Cc3ccc(C#N)s3)C2)(NC(C2(c3ccn(C)n3)CC2)=O)CC1 77735,Cn1cc(Cl)c(C(=O)NC2CC(CCNC(=O)Cc3ccc(C4CC4)cc3)C2)n1 77736,C1(CC(=O)NCC2C(CNC(C(C)CC3CCC3)=O)C2(F)F)CC(O)C12CCC2 77737,C1(CNC(C(=O)NCc2nccc(-c3ccccc3)n2)=O)CNCCC1(F)F 77738,Cc1ccc(C(C)NC(C23CC(C(N4CCCNCC4)=O)(C2)C3)=O)nc1 77739,N1(C(COCC)=O)CCC(C(F)F)(CNC(c2cncnc2)=O)C1 77740,Cc1[nH]nc(Cl)c1C(=O)NC1CCC(NC(=O)CC(O)c2ccccc2)CC1 77741,c1(C(N(C2CN(C(c3ccc(OC)nc3F)=O)C2)C)=O)c[nH]c2nc(F)ccc12 77742,C(=O)(CCCC(C)CC)N1C(C)CC(CC(N2CC(C(=O)OC)C2)=O)C1 77743,N(C(=NCCCCC)N1Cc2cnn(CCO)c2C1)C(C#C)(COC)CC 77744,CCCCC(C(=O)NC1CCC1CC(=O)OC)NC(c1cn(C)cc1C)=O 77745,N1(C(C(C)c2cc[nH]n2)=O)CCCC12CCN(C(=O)CC(C)(C)N(C)C)CC2 77746,n1(CC)nc(C)c(C(=O)N)c1C.c1(N(C(COC(=N)O)C)C)ncnc(Cl)c1C(C)C 77747,c1(C(=O)OCC)cn(C)nc1C(N1CC(NC(=O)CN2CCC2C)C(F)C1)=O 77748,CCC(C)(C)CC(=O)NCC1CN(C(=O)COc2ccc(F)c(CO)c2)CC1O 77749,c1(CC(=O)NCC(C2CC2)NC(=O)CCn2ccnc2)ccc(Cl)nc1F 77750,c1(C(=O)NCC(C)N(C(=O)C(C)CC(F)F)CC)ccnc2[nH]c(C)nc12 77751,Cc1cc(C(=O)NCC(CNC(=O)CC#N)CO)n(C(C)(C)C)n1 77752,n1(CC)ccnc1CC(=O)NC(CNC(C)=O)C(=O)NC(COC)COC 77753,c1(C(=O)NC(C2CCN(C(C(C)OCC)=O)CC2)C(C)C)csc2nnsc12 77754,c1(CCCN(CCCNC(=O)C(C)OCCC(C)C)C(C)C)ccccc1 77755,n1(CCC)ccnc1C(F)(F)C(=O)N(CC(C)NC(=O)CC(C)C1CCCC1)C 77756,CCC(C)CC(C)NC(C(=O)O)c1cccs1 77757,C1(N(C(C(C2N(C(c3cnc(OCC)s3)=O)CCC2)(C)C)=O)C)COCC1(C)C 77758,CCCCC(O)C(=O)NCCC1CCCN(C(c2ccc(C)c(OC)c2)=O)CC1 77759,N1(C(C2CCC(=C)CC2)=O)C(C(=O)NCCCCc2ncc[nH]2)CCC12CC2 77760,CCS(=O)(=O)CC(=O)N1CCN(C(C2CN(Cc3ccc(C)nc3C)C2)=O)CC1 77761,c1(C(=O)NCC(N(C(c2cn(CC=C)nn2)=O)C)C2CC2)cnc(C)c(N)c1 77762,c1(C(=O)OC)cccc(CNc2ccc(C(C)NC(C3CC3)OC)cc2)n1 77763,N1(C(=O)OC(C)(C)C)CCC2CC1CN(Cc1ccnn1-c1ccccc1)C2 77764,c1(-c2onc(CNC(=O)NC3CCCC=C3Br)n2)cccc(F)c1 77765,N1(C(C(c2cccs2)SC)=O)CCN(C(c2cnn(CC3CC3)c2)=O)CC(O)C1 77766,C1(CNC(c2nc(C(C)=O)sc2)=O)C2CN(C(=O)CC=C(C)C)CC12 77767,n1(C(C)C)ccc2c(C(=O)NS(=O)(=O)CCC3CC3C3CC3)cccc12 77768,CC1CN(C(=O)CCC2(C)CC2)CC2(CCN(C(C3CCCN3C)=O)CC2)O1 77769,c1(C(N(C)CC2N(C(C(CC#C)O)=O)CCC2)=O)cc(C)nc(C)c1 77770,N1(C(c2c(C)nsc2)=O)CCCCC1CCCNC(C1CC1C#N)=O 77771,S(=O)(=O)(c1nc(C)cs1)NC(c1cc(OC)c(F)cc1)C 77772,N1(C(CC=CC)=O)CCCC2CCN(C(C3CC4(CSC4)C3)=O)CC12 77773,N1(C(CCC2N(C(C3CCSCC3)=O)CCC2)=O)CC(CO)C2(CC2)C1 77774,N(C(=NCC(=C)C)NCc1ccc(C)cc1OC)C(c1ccc(Cl)cc1)C#C 77775,C(CC(C(=O)NC1CC(=O)N(C)C1)NC(=O)C(CC1CCC1)OC)OC 77776,c1(C(C)C)c(C(=O)N(CC(C)NC(=O)CC2COC(=O)N2)C)cnc2ncnn12 77777,C1(C(=O)OCC)COCCN1C(C1(C)CCN1C(c1cnccc1Cl)=O)=O 77778,Cc1cc(C(=O)NCC2CCCC(NC(C3CC3F)=O)C2)cc(S(C)(=O)=O)c1F 77779,CC1(C)CC(C(=O)NCC2(O)CCCN(C(c3cc(F)ccc3F)=O)CC2)=NO1 77780,CCCC(CCC)C(=O)N1CCOCC1CCNC(=O)CSCCN(C)C 77781,CCC(C)C(O)CC(=O)NCCC1(NC(C2CC(F)(CF)C2)=O)CCCC1 77782,C1(c2n(CC)nnn2)(NC2(C3CC3)CCCCCCC2)CC2(CCOCC2)C1 77783,C(C)(CCN=c1[nH]cnc2cc(C3CC3)nn12)NC(c1c(C)nn[nH]1)=O 77784,c1(C(=O)NCC(=C)CCNC(=O)CSc2ccncc2)[nH]nc(C(F)(F)F)c1C 77785,C(C(C)(C)C(=O)NCCc1cn(C)cn1)NC(C1CCC(C)C1)=O 77786,N1(C(CCC2CCN(C(CC3C(C)OCC3)=O)CC2)=O)CC2CCC2(C)C1 77787,C(c1cscn1)=CC(=O)NCCSCC(=O)N(CC#C)Cc1ccco1 77788,Cc1[nH]c(=N)sc1C(=O)NC1CCCC1N1CCN(C(=O)CC(C)(C)O)CC1 77789,N1(C(CC(N2C(=O)CCC2=O)C)=O)CCC(C)(CNC(c2ccoc2Br)=O)CC1 77790,N1(C(C2CC(OC)C2)=O)CC2CC(O)C1C2NC(c1cccnc1N)=O 77791,Cc1ncc(C(=O)NCc2nc(C3CC3)no2)o1.C12(CCC1)C(=O)N2 77792,N12CC(CCC1(C)C)C(=O)NC1(CCC1)C2=O.C(C(C)CC(C)C)OCC 77793,c1(C(C)NC(=O)C(C)(C2CC2)N(C)C(c2cn(C)cn2)=O)cccc(O)c1 77794,c1(CC)nnc2n1CCCC2C(=O)N1CCN(C(c2cccn2C)=O)C(CO)C1 77795,C1(n2cc(-c3cccc(C)c3)nn2)CON(C(=O)C2CC(n3cc(CO)nn3)CO2)C1 77796,c1(CC)ncc(C(=O)NC2(C)CC(NC(C3CN(c4nncs4)C3)=O)C2)s1 77797,C(=O)(N1CCC(C(=O)NC2CC2C(=O)NCN=[N+]=[N-])O1)C1N(C(C)C)CCC1 77798,C1(NC(C=CC(=O)OCC)=O)CC12CCN(C(C1(n3ccnc3)CCCC1)=O)C2 77799,c1(CC(=O)NC2CCN(C(C3C(CCOC)C3)=O)C2C)ccc(Cl)cc1F 77800,CC(CCC(F)(F)F)NC(C1C2CCC1(c1ccco1)C2)=O 77801,C1(NC(CCCSC)=O)(CO)CCN(C(=O)CC2CC(F)C2)CC1 77802,Cc1nc(O)sc1C(=O)NC(CNC(=O)C=Cc1ccncn1)CO 77803,N1(C(C2C(=C)C2)=O)CCC2(CCCN(C(=O)CC3(CO)CCCC3)C2)C1 77804,C1(CC(C(=O)NC(C)CC)N(C)CC2(OC)CCCC2)COC(C)(C)O1 77805,c1(C(=O)OC)ccc(CC(=O)NC2(CO)CN(C(=O)C(C)C(C)O)C2)c(N)c1 77806,C1(C(=O)Nc2cccc(CC)c2F)CC(C)(C)CCN1C(=O)C(C)c1cc[nH]n1 77807,c1(CC(=O)NCC2CC(NC(=O)Cc3cnc(C4CC4)[nH]3)C2)cncc(F)c1 77808,N1(C(Cc2cc(C(C)C)no2)=O)CC(NC(=O)Cc2ccn(C)n2)CC12CCC2 77809,Cc1cc2c(cc1C)C(NC(=O)C(C1CCCCC1)O)CCCO2 77810,c1(C(=O)NC(C2(O)CN(C(c3cc(F)ccc3N)=O)C2)C)ccc2occc2n1 77811,c1(CNCCC(C)CC(C)(C)C)cc2nc(Cl)ccc2s1 77812,N1(C(CC2(OC)CN(C(C34CCCCC3C4)=O)C2)=O)CCC2(CC1)CSC2 77813,C(=O)(C(O)CCCNC(=O)CCc1cccnc1)NC(CCC)c1nn[nH]n1 77814,C=C=CC(C)C(=O)N1CC(C)C1C(=O)Nc1cnc(OC)nc1 77815,C1(C(=O)NC2(CC)CN(C(C3CCN(C)C3)=O)C2)OCCN(C)C1=O 77816,C1(CNC(c2csc(C)c2C)=O)CN(C(C2CCOC2)=O)CC(C)(C)C1 77817,C1(NC(C2(C=C)CCC2)=O)CC(O)CN(C(c2ccc(OC)c(C)c2)=O)C1 77818,c1(C(=O)NCCCN(C(CNS(CCOCC)(=O)=O)=O)C)ccc(C)cc1CC 77819,C1(NC(C2CC=CCN2C(=O)Cn2cccnc2=O)=O)CC12CCCCC2 77820,c1(C(N(C2CCN(C(CCCOC(C)C)=O)C2)C)=O)nccc(Br)c1O 77821,c1(OC)cc(C(N2CCCC(O)(CCNC(=O)C(C)CO)C2)=O)c(N)c(C)c1 77822,c1(NC(C2CCCN(Cc3ncccc3O)C2)=O)cccnc1O 77823,N1(C(c2ccn(CCOC)n2)=O)CCC(C)(CNC(c2cn(C(C)C)nn2)=O)C1 77824,N1(C(Cn2ncc(CC)c2)=O)CC=C(CNC(C2CCN(C(N)=O)CC2)=O)CC1 77825,C1(CNC(CCC)=O)CN(C(=O)C(O)C2=CCCCC2)C2CCCC2O1 77826,C(=O)(C(F)CC(C)(C)NC(=O)C(C)c1ccco1)Nc1cccc(C#C)c1 77827,C1(CCC=C)(C(=O)NCc2cnn(C)c2)CN(C(C2CCO2)=O)C1 77828,Cc1[nH]c2ccccc2c1C(=O)NCC(C)N(C)C(C1CCC(C)(C)C1)=O 77829,c1(CNC(C2CC2F)=O)cccc2c1CN(C(c1cc(O)ncc1F)=O)C2 77830,c1(C(N(C)CC2COC(C)(C)O2)=O)ccc(Cl)cc1N=[N+]=[N-] 77831,C1(C#N)(C(N(CCNC(CC(C)C)=O)C2CC2)=O)CCCO1 77832,C=CCCCCC(=O)NC(C)CCCCNC(C1CCCN1c1cnccn1)=O 77833,NC1CC2(CC(CNC(C3(O)CCCNCC3)=O)C2)C1 77834,C1(C)(CNC(Cn2nnc(C(C)(C)C)n2)=O)CN(C(=O)CC2CC(F)C2)CC1C 77835,C(=O)(C1=C(Cl)CCC1)N1C(NC(=O)CCCn2cncn2)CC1.C12CN1C2 77836,Cc1cc(C(N2CC(CNC(C3COC3)=O)CC2C)=O)c2nc(C)n(C)c2n1 77837,CCC(C)(O)C(=O)NC(CNC(=O)CCc1ccc(Br)cc1)C1CCC1 77838,c1(COC)ccsc1C(N1CCC(NC(c2ccc(C(C)(C)C)[nH]2)=O)C1)=O 77839,c1(C(N(CC(CC)NC(=O)C#CC2(C)CC2)C)=O)c(SC)cccc1F 77840,c1(NC(C2C(C)(C(=O)OCC)C2)=O)ccc(Br)cc1Br 77841,C(=O)(CC(C)CC(=O)NCC1(NC(c2ccc(Br)cc2C)=O)CCOC1)OC 77842,c1(-c2cn(C3CC(C(=O)NCCC(C(C)C)O)C3)nn2)cc(Cl)c(F)cc1F 77843,CC1CC(C)(C)CN1C(=O)COC1(C)CN(C(=O)C=Cc2cc[nH]n2)C1 77844,c1(CC(=O)NCCC2CCC(NC(CC(C=C)C)=O)C2)cn2cccc(C)c2n1 77845,Cc1cc(N2Cc3nn(C)c(N)c3C2)nc(=NCCn2ncc(Br)n2)[nH]1 77846,C(=O)(CCC(F)(F)C(F)(F)F)NCC1CN(C(c2c(C)cc(O)nn2)=O)C1 77847,N1(C(c2cc(SC)oc2)=O)CC(C2CCN(C(C3CCOC(C)(C)C3)=O)CC2)C1 77848,C(CC(=O)NC(C)COCCOC(C)=O)N(CC(=O)NC)CCC 77849,C1(C(NOC(C)(C)CO)=O)CC1C1CN(C(C2CCCCCC2)=O)C1 77850,CC(CC(=O)NCCCC1CCCN1C(=O)CCN1CCCC1)P(C)(C)=O 77851,C(CC(C)(C)CC(=O)NCC(CNC(=O)C1=CCCC1C)CO)OC 77852,c1(CNC(C(N2CCC(C#C)C2)c2cccc(SC)c2)=O)ccc(F)cc1F 77853,N1(C(c2ncc(OCC)nc2)=O)CCC2(NC(=O)CCc3c[nH]c(=N)[nH]3)CC2C1 77854,C(C(N=[N+]=[N-])C(=O)NCc1nc(C(=O)NOC)co1)OCC 77855,C#CCC(CC(=O)N(C)CC1(N(C)C)CCC1)NC(=O)CC(C)C(F)F 77856,C#CC1(CNC(=O)CC2CCC(NC(C3CC4(CCO3)CC4)=O)C2)CCOCC1 77857,c1(CC)cc(N)c(C(=O)NC2CCCCN(C(=O)C(F)(F)CC(C)C)C2)c(F)c1 77858,C1(NC(c2cc(O)ncc2F)=O)CC2CCC1CN2C(C1CCCC1)=O 77859,N1(C(CCN(CCC)C)=O)CCC(CF)(NC(=O)CNc2ccccn2)C1 77860,C1(C(N(C2CCCCC2(C)C)Cc2cnn(C)c2N)=O)CCC2(CCC2)C1 77861,Cn1nc(CC(=O)NC2CC(F)(CNC(c3cc[nH]n3)=O)C2)cc1C(F)(F)F 77862,C(=O)(C(C)(C)C)N1CC(CNC(C(C)=C(C)C)=O)C1.C1(=O)CCN1 77863,C12(C)CCCC1NC2=O.N1(C(C(=O)N(C(C)C)C2CC2)C)CCC(N(C)C)C1 77864,C1(C(C(=O)NCCC=C=C)C)CCN(C(c2noc(C)c2C)=O)CC1 77865,c1(CC)nnc(CNC(C2COCC2NC(=O)C=CC(=O)N(C)C)=O)o1 77866,C1(C(N2CCN(C(CSCCCC)=O)CC2CF)=O)COC2CCCCC12 77867,c1(C(=O)NCCCN(C)C2CC2)coc(CNC(C2CCC(=O)C2)=O)n1 77868,c1(NCCC(=O)NC(C2(C)CCC2)C)ncnc2sccc12 77869,c1(C(N2CCC(N(C(C3COC(=O)O3)=O)CCO)CC2)=O)cc2c(Cl)cncc2s1 77870,CN1CCC2(CCN(C(=O)COCCNC(c3ccc([N+](=O)[O-])o3)=O)C2)C1 77871,C1(NC(C2C(CC)C2)=O)CC(CCNC(c2csnn2)=O)C1 77872,N1(C(=O)Cc2ccccc2)CCC(F)(C(=O)Nc2cnc(-c3ccccc3)s2)C1 77873,c1(C(N2CCC(N(C(=O)C(c3ccc(C)s3)C)CCC)C2)=O)nc(CC)oc1C 77874,Cc1cc(N)cnc1C(=O)NCC1CCN(C(C2CCC3CC3C2)=O)C1(C)C 77875,C(=O)(CC(CC)C(C)(C)C)NCc1cn(C(c2cccnc2)C(N2CC(=C)C2)=O)o1 77876,C(=O)(C(C)(C)C(=O)N(CC(O)CNC(C1CCNC1=O)=O)C)N(C)C 77877,N1(C(c2c(OC)nccc2)=O)CC(NC(=O)CCc2ccn(C)n2)CC12CCC2 77878,C(C)(CN=c1[nH]c(N2C3CCC2COC3)nc(=N)[nH]1)N1CCCC(C)C1 77879,c1(CC)nc(C)cc(=NC(CNC(=O)C(F)C(C)C)C2CC2c2ccccc2)[nH]1 77880,C1(CCCNC(Cc2cc(C)no2)=O)CCCCN1C(c1c[nH]nc1C)=O 77881,c1(C(=O)NC2C(CNC(c3c(CCC)onc3C)=O)CC2)cc(F)c(Cl)cc1Cl 77882,C1(CCCC)(C(N2CCC(CNC(N)=O)C2)=O)CCC(=O)CC1 77883,c12cccc(c1)CN1CCCCC1CN(C)C2=O.C1(CC(=O)NC)CC(=O)N1 77884,c1(CC(C)C(=O)N(C)CCOCCNC(C2CCC(=O)N2)=O)cccc(F)c1 77885,C1(F)(CNC(C(CC)F)=O)CCN(C(=O)CCCc2csc(C)n2)C1 77886,N1(C(CC(CN(C)C)O)=O)CC(C)(C)CC1CNC(c1cc(O)nc(O)c1)=O 77887,c1(NC2C(CC)C2)ncccc1S(=O)(=O)NCc1nc2ncccn2n1 77888,C(CCCC(C)(C)NC(C1CCN(C)C1=O)=O)NC(C(C)NC(=O)C1CC1)=O 77889,c1(C(N2CCCCCC(NC(C(COC)C)=O)C2)=O)ccc(OC)c([N+](=O)[O-])c1 77890,c1(C(N(C(CNC(C(CC=C)C)=O)C)C)=O)c[nH]c2cccc(Cl)c12 77891,CC1(C)CNCCC1N1CCN(Cc2cc(Cl)ncc2Cl)CC1 77892,c1(C(N2CC(CNC(c3cc(CCO)on3)=O)OCC2)=O)cc(Cl)c(O)c(Cl)c1 77893,C1(O)(CNC(C(C(C)C)F)=O)CCCN(C(c2ccc(C(F)F)cc2F)=O)CC1 77894,CCC(CC)C(C)(F)C(=O)NCC(C)(C)C1(O)CNC1 77895,c1(C(N(C)CC2OCCN(C(C3C(OCC)C3)=O)C2)=O)cc(C)cc2c1CCC2 77896,N1(C(=O)OC(C)(C)C)CC2CC2(C(=O)NC2CCN(Cc3cccnc3)CC2)C1 77897,c1(C(N2C3C(NC(=O)C=CC4CCC4)CC(C3)C2)=O)ccc2ccncc2n1 77898,c1(N2CCN(C(=O)Nc3cc(C)ncc3Cl)CC2)cccc2nsnc12 77899,C=C(C)C(C)(C)C(=O)N(C1CCCN(C(c2cnc(S)nc2)=O)CC1)C 77900,N1(C(C=CC=CCCCCC)=O)CC2C(CNC(C3CCC(=O)N3C)=O)C2C1 77901,N1(C(C2CCN(CC)C2)=O)CCOC(CCCNC(=O)CSC2CC2)C1 77902,N1(C(CCc2c(C)noc2Cl)=O)CCC2(CCN(C(=O)CCn3ccnc3)C2)C1 77903,N1(C(c2c(C)ncnc2)=O)CC2CCC(C1)C2NC(C1(C)CC2CCC(C1)S2)=O 77904,c1(NC(c2n(CCC)nnn2)C(C)COC)ccc2c(c1)OC(F)(F)O2 77905,c1(CC#N)cccc(C(=O)NC2CC(C(=O)NCC3NC(=O)NC3=O)C2)c1 77906,N1(C(c2cc(C)on2)=O)CCCC(O)(CN(C)C(c2ccc(C(C)C)nc2)=O)C1 77907,C(=O)(C(C(=O)c1ccccc1)NC(=O)OC(C)(C)C)OCC1(CCCC)CC1 77908,C(=O)(C1=CC2C=CC1C2)NC(C1CCCN1C(c1cc2ccccn2n1)=O)C 77909,c1(OCC(=O)NCCN(C(c2[nH]c(C)cc2C)=O)CC)ccc(Cl)nc1 77910,C(=O)(CC(O)CC(C)C)NC(C(=O)NC(CC(=O)OC)C)COC(C)C 77911,c1(C(N(CC(C)C)CCC)=O)cccc(CNC(=O)CSCC(=O)OC)n1 77912,CCC(C)C(O)C(C)C(=O)NCCCCCC(=O)NCC(F)(F)Cl 77913,CCC(CC(F)(F)F)NC(=O)CC(C)N(C(=O)Cc1cncnc1)C 77914,c1(CNC(CN(C)C(C2CC=CCC2)=O)=O)cccc(F)c1O 77915,C(=O)(C(C)CC(C)CC)N1CCC(OCC(=O)NCC(=C)CC)C1 77916,CC1CC2(CCN(C(=O)C(N3CCCC(N4CCC4)C3)=O)C2)CO1 77917,Cc1cc(O)c(Cl)cc1C(=O)NCCCCNC(=O)C(C)CC1CCC1 77918,N1(C(CC)=O)CCc2nn(C)cc2C1.C1(N2C(=O)C2CCCl)Cc2nccn2C1 77919,C1(CNC(C23OC(C)C(CC2)C3)=O)CC2(CO1)CN(C(C1CC(O)C1)=O)C2 77920,C#CC1CCN1C(C1CC(N(C(=O)CC2(C(=O)N(C)CC)CC2)C)C1)=O 77921,c1(SC)sccc1C(N1CCCC1CNC(c1ncoc1C(F)(F)F)=O)=O 77922,c1(C(=O)NCCn2c(C)nnn2)ccc2c(c1)CCN2Cc1ccco1 77923,C1(CC)CC(SCC)CCO1.C12(CCOCC1)CC(=O)OC2=O 77924,c1(CC(N2CCCC(NC(C(CC)O)=O)C2)=O)ccc(Cl)c(Cl)c1 77925,C=C(C)C1CN(C(=O)CCNC(C2CC2(C)C(C)C)=O)CCO1 77926,N1(C(c2cccc(C(C)C)c2N)=O)CCC2(CC(NC(C3CC3(C)C)=O)C2)C1 77927,CCCCCC(CC)C(=O)NCC1CN(C(C23CC(C2)C3)=O)CCCO1 77928,c1(C(C(=O)NCC(=C)C)N(CCCCO)C)ccn(-c2cnn(C)c2)c1 77929,Cc1n[nH]cc1C(=O)NC1(C(=O)NCC2(F)CCOC2)CSC1 77930,N1(C(C2(CCC=C)CN(C(=O)C(COC)CC)C2)=O)CCOC(C)C1C 77931,N1(C(CCC#C)=O)CCC(C=C)(C(=O)NCCCS(C)(=O)=O)CC1 77932,c1(CNC(C2C(NC(CC3(OCC)CCC3)=O)CC2)=O)cc(C)c(C)cn1 77933,C1(NC(CC(C)OC)=O)CN(C(=O)CCCc2cnccn2)CC12CCC2 77934,C1(C(=O)OC)CCC2(CC1)CC(S(=O)(=O)N1CC(NC(C)=O)C(C)(C)C1)C2 77935,CC1(C)CCC(NC(=O)C=C2CC2)C(CNC(=O)CSc2nncn2C(C)C)C1 77936,C1(CC)(CC)CC(O)CN1C(C1CC(CNC(c2c[nH]c(=S)cn2)=O)C1)=O 77937,N1(C(CC2(CNC(C3C(C(C)C)OCC3)=O)CC2)=O)CCC(N=[N+]=[N-])C1 77938,C1(CC)CN(C(=O)C(CCOC)OC)CCN1C(c1ccc(O)c(Br)c1)=O 77939,C1(NC(C(CO)NC(C(CCC)NC(N)=O)=O)=O)CCCC(O)CC1 77940,C1(C(C)C)CCC(C(=O)NC2COCC2NC(=O)CC2COCCO2)CC1 77941,C1(C(=O)NCC2(CO)CCCN(C(C=C(C)Cl)=O)C2)C(C)(C)CCCC1(C)C 77942,c1(C(=O)NC2C(CNC(c3cnc(O)s3)=O)CCC2)ccncc1Br 77943,c1(SC)cc(N2CCC(C(=O)Nc3ccccc3CCO)C(F)C2)nc(C)n1 77944,S(=O)(=O)(c1cccc(=NCC2(C)CC3CC3C2)[nH]1)N(C(C)(C)C)C 77945,Cc1cc(Cl)ncc1CC(=O)NC(C1CCCCC1)CNC(=O)C1=COCC1 77946,N1(C(CC(=O)NC2CC2)=O)CC2CC(C(N3CC4CCC(CC4)C3)=O)CC2C1 77947,C1(OC)Cc2ccccc2C1NC(=O)NCC1(CO)CCOCC1 77948,N1(C(C=NOC)=O)CCN(c2ccccc2CNC(C2CCC2OC)=O)CC1 77949,c1(C(N2C3CN(C)C(C3)C2)=O)cccc2[nH]nc(C3=COCC3)c12 77950,C(=O)(C(C)(C)C1=CCN(C(=O)C2=CC3(CCOC3)C2)C1)N(C)CC1CCCS1 77951,C=CCC(CC=C)C(=O)NCC(CNC(=O)CCc1c(C)nc(O)nc1O)OC 77952,C#CC1C(C(=O)NCC2C=CC(NC(c3cnc(C4CC4)s3)=O)C2)C1(C)C 77953,c1(C(C)C)n[nH]c(=NC2CC23CC(NC(=O)C(C)(C)S(=O)(=O)C2CC2)C3)o1 77954,c1(OC)cc(Br)ccc1CNC(N1CC(C(CO)C(=O)Nc2ccncc2)C1)=O 77955,C(=O)(C(CO)NC(=O)C(CC1CC1)NC(c1cc(C(C)=O)on1)=O)OC 77956,N1(C(C(C)CS(C)(=O)=O)=O)CCN(C(c2ccc3cnsc3c2)=O)CC12CCC2 77957,Cc1cc(C(=O)NCC=CCNC(c2cc(C)n(C)c2)=O)cnc1C(F)F 77958,C1(CC(N2CCCC2CF)=O)CN(C(n2cc(-c3ccccc3F)nn2)=O)CCO1 77959,c1(C(N2CC3CN(C(COCCCCC)=O)C3CC2)=O)cnn2cc[nH]c(=O)c12 77960,c1(C(N2CC3(C(NC(c4cnc[nH]4)=O)CC3)C2)=O)noc2ncccc12 77961,Cc1cc(=NC(=O)C(=O)N(CC(N2CCCC2)C)CC)[nH]n1-c1ccc(Cl)cc1Cl 77962,CS(=O)(=O)CCCCN(C1CCC12CCNCC2)C(=O)C(N)Cc1cscn1 77963,C1(CNC(Cc2c(C)nsc2)=O)C(C)CCCN1C(=O)Cn1nccn1 77964,C1(C(=O)NCCC2CCCC2)CN(C(c2n[nH]c3c2COC3)=O)CC1C1CC1 77965,c1(-n2ccc(C)n2)ccccc1NC(=O)NCC(C1CCCCC1)C 77966,N1(C(C=C(C)CNC(=O)CC2CCC(C)CO2)=O)CCC2=C(CCCC2)C1 77967,CC1(C)CCN(C(=O)C(F)C2CCCC2)CC1NC(c1cc(C2CCC2)no1)=O 77968,C#CCCCC(C)C(=O)NC1CC(OCC(=O)NCC(=O)N(C)C)C1 77969,c1(C(N2CC(C(=O)NC)OCC2)=O)c[nH]c2c(F)cc(OC)cc2c1=O 77970,C1(C(=O)NC(CNC(C2COC(=O)N2C)=O)CO)(CC)CNC(=O)C1 77971,c1(NC(COC)COC)cc(=NC2CCC(CS(N)(=O)=O)C2)[nH]c(C(F)(F)F)n1 77972,C1(CNC(C(C)OCC)=O)(Cn2cc(C3(O)CCOC3)nn2)CC12CCC2 77973,C1(NC(C)=O)CC(C)CN(C(=O)CC(C)F)C1 77974,c1(C(C)C)c(C(c2nnnn2C)NCC(c2ccccc2)CO)cccc1F 77975,S(=O)(=O)(c1ccc(=NCc2cnn(C)c2Br)[nH]c1)NCCc1ncc(C)cn1 77976,C(=O)(C1=NOC(C)(C)C1)N1C(CC(=O)Oc2c(CC)ccc(F)c2)C2CCCC21 77977,C1(NC(c2ccc(F)c(CO)c2)=O)CCS(=O)(=O)C12CN(C(C1C=CCC1)=O)C2 77978,N1(C(c2ccc(CC)cn2)=O)CCC(O)C(C(N2CC3CC(CO)C3C2)=O)C1 77979,CC1CCC(NC(=O)CCCC2CCCC2)CN1C(=O)Cc1cc(F)ccc1O 77980,c1(OC)ccc(CC(=O)NC(C)C(C)NC(c2csnn2)=O)c(Cl)c1 77981,N1(C(c2coc(Nc3ncccn3)n2)=O)CCc2c(Br)cccc2C1 77982,C(C1=CCCOC1)N(C(=O)CC1CCC(NC(c2cnc(C3CC3)o2)=O)CC1)C 77983,N1(C(C2N(CC)CCC2)=O)CCC2CCCC12C(=O)NC(C)C(C)SC 77984,C(CCN(C(=O)Cn1nnc(C2CC2)n1)C)(C(C)C)NC(c1n(CC)nnc1)=O 77985,C(C)(C)(CC(F)C(=O)N1CCC(OCCOC)C1)NC(c1c(CC)ocn1)=O 77986,N1(C(=O)OC(C)(C)C)CC2CCC1(NCC=C1CCOC1)C2 77987,c1(C(N2CC(CNC(C3(CC#C)CCC3)=O)C2)=O)nccc(C)c1N 77988,c1(OC(C)C(=O)NCCCCN(C(=O)CC2COC(=O)C2)C)cc(Cl)cc(Cl)c1 77989,n1(CC(=O)N(CCC)CCN2CCC2C)cc(-c2ccnn2CC)nn1 77990,CC(C)(F)CCC(=O)NCC1CCCC1C(N1CCC(CC(N)=O)CC1)=O 77991,c1(C(=O)NCC2(O)CCN(C(C(C=C)(C)CC)=O)C2)cnc2c(c1)CCCC2 77992,c1(C(=O)NC2C(C)CN(C(=O)CC3SC(=N)NC3=O)C2)nc2ccccc2[nH]1 77993,N1(C(CN(CCC)C)=O)CCC2(CC1)CN(C(c1ccnnc1NC1CC1)=O)C2 77994,c1(C(=O)NCC(C)(C(C)C)NC(C2N(CC)CCC2)=O)ccc2ncnn2c1 77995,C1(C(=O)NCC(C)CC2CCCC2)CC=CCC1NC(=O)CC1CCCC(=O)C1 77996,c1(C(C(=O)NCC(C2CC2)NC(C(C)OCCN(C)C)=O)=O)cccn1C 77997,C1(NC(C(CCC)N(C)C)=O)CC12CCC(NC(=O)COCCOC)CC2 77998,n1(CC=C)cc(C(=O)NCCN(CCC(=O)NCC2CCCO2)C)cn1 77999,C#CCC(C)(C)C(=O)NCc1ncccc1C(=O)Nc1ccc(C(C)C)cc1 78000,O=C(C1=Cc2ccc(Cl)cc2OC1)NCC(C1CC1)NC(c1cscn1)=O 78001,n1(CC(N2CCC(CCCC)C2)=O)ccc2ccc(F)cc12 78002,c1(C(=O)Nc2ccc(OC(F)F)nc2)cc2c(o1)=CCC(c1sccc1CO)=CC=2 78003,C(=O)(CCC(C)CC)N1CC(CCNC(C2CC(=C)C2)=O)OCC1 78004,N1(C(COC)=O)CCN(C(C2CCC(NC(=O)CSCc3cscn3)C2)=O)CC1 78005,c1(C(N(CC(O)CN(C(=O)C(C)(C)O)C)C)=O)cnn(C)c1C(F)(F)F 78006,C(Cc1cccs1)(CC(=O)Nc1cnccc1C(C)C)NC(c1c(C)ccs1)=O 78007,CCC(CCCC(=O)N1CC2(CNC(=O)C2)C1)NC(=O)C=CC(C)(C)C 78008,N1(C(C=CCN(C)CC)=O)CCC2CN(C(c3c(Cl)cccc3Cl)=O)CCC2C1 78009,CC(C)(CC(=O)NC1(C2CCN(C(=O)C(F)CC3CC3)C2)CC1)C(F)F 78010,C1(O)(CN(C(=O)Nc2c(-n3cc(C=CC)nn3)cccc2)C)CCC(F)(F)CC1 78011,C1(CC)CCCC1(C)C(N1CC(NC(=O)CSc2ccccc2OC)C1)=O 78012,c1(C(N(CC(C)NC(C(C(CC)O)(C)C)=O)C)=O)nc(=N)[nH]c2ccccc12 78013,C1(C(=O)NCc2cc(Br)ccn2)CC12CCN(C(c1ccc(Br)cc1F)=O)C2 78014,C(C(C(=O)N1CC(OC(C)=O)C1)NC(C1C=C(C)CS1)=O)OC 78015,N#Cc1cncc(C(N2CC(NC(=O)C(O)Cc3cnn[nH]3)C(O)C2)=O)c1 78016,Cc1ncnc(C)c1OCC(N1CC2C(NC(c3cccc(F)c3O)=O)C2C1)=O 78017,C1(C(=O)NC23CN(C(CN(C4CCC4)C)=O)C(C2)C3)CC2(CCCCC2)C1 78018,c1(C(=O)NC(C)C(CO)NC(C2CCCCN2C2CCCC2)=O)ccc[n+]([O-])c1 78019,c1(C(=O)NCC(C2CC2)NC(=O)CN2CCCCCC2)cc2c(Cl)cncc2o1 78020,C(=O)(C1=CC2C=CC1C2)N1CC2C(CC(=O)N(CCCO)C)(CC2)C1 78021,N1(C(C2CCC(NC(Cc3c(C)nc[nH]3)=O)C2)=O)CCN(CC2CCCC2)CC1 78022,Cc1cccc2c(C(=O)NC3CC4CCC(C3)N4C(=O)C=CCO)csc12 78023,c1(OC)cc(=O)n(C)cc1C(=O)NCCOC1CN(C(=O)C2=CCSC2)C1 78024,N1(C(CCc2cc(C)on2)=O)CCC(NC(c2conc2C2CC2)=O)C(O)C1 78025,C1(C(N2CCCCC(NC(c3c(C)c(N)n(C)n3)=O)C2)=O)CC2C=CCC(C1)C2 78026,N1(C(CCC)=O)CC=CC(C(N2CCC(OCCF)C2)=O)C1 78027,c1(C(=O)NC(C2(CNC(CC3CC(=C)C3)=O)CC2)C)sc2ccccc2c1Cl 78028,n1(CCC)ccnc1CN(C(=O)NCC(C)(O)C1(C)CC1)CC 78029,c12ccccc1C2.c1(C(COC)NC(=O)Nc2c[nH]nc2Cl)ccccc1F 78030,c1(C(=O)NCCC(C)N(C)C(C2C=CCC2)=O)c[nH]nc1-c1ccccc1 78031,n1(CCC=C)c(N2CCC(CF)C2)nnc1Cc1cccs1 78032,c1(-n2ncc(C)c2)ccc(CNC(N2CCOC(C)(C3CC3)C2)=O)cc1F 78033,N#Cc1cnccc1CN1CC(NC(C2Cc3ccccc3O2)=O)C(F)(F)C1 78034,N1(C(C(N2CCCOCC2)C2CCC(CCSC)O2)=O)CCSCC1C(N)=O 78035,CC(C)CC(C)CNC(=O)CCN(CCCO)C(C1CCCC(C)C1)=O 78036,C1(N(C(C=C(C)C(F)F)=O)C)CN(C(=O)C(CCN(C)C)N(C)C)CCC1O 78037,CCC(=O)CCC(=O)NC(C)CCCC(=O)NCc1nccn1C 78038,N1(C(C2CCCCCCC2)=O)CC2CCN(C(C3CC4CC3CN4)=O)CC12 78039,c1(C(N2C(CNC(C(C)Cc3ccccc3)=O)CCC2)=O)nc[nH]c2ncnc1-2 78040,O=C(CC1=CCOCC1)NC1CCC1NC(c1ccc(C2CC2)cn1)=O 78041,c1(C(=O)NCC2CCC(NC(CCSC)=O)C2)ccc(N(C)C)c([N+](=O)[O-])c1 78042,C1(CNC(C2(C(C)(C)OC)CC2)=O)CN(C(c2cc(C)c(C)o2)=O)CC1C 78043,Cc1noc(C)c1C=CC(=O)NCC1CC(NC(=O)CN2CCOCC2)C(O)C1 78044,C1(C)(C(=O)OC)CCCN1C(C1(C)CN(C(c2cc(Br)ccn2)=O)C1)=O 78045,c1(C(N2C(CNC(c3n(CC)ncn3)=O)CC(O)C2)=O)cc(Cl)c(Cl)cc1O 78046,C1(C)(CNC(CCOC(C)=O)=O)CCN(C(=O)C=Cc2cnn(C)c2C)CC1 78047,Cc1ccc(C(N2CCOC(C(C)NC(c3ccc(C(F)F)o3)=O)C2)=O)c(N)c1 78048,c1(C(N2C(CNC(C3CC(=C)C3)=O)CCC2)=O)ccc2c(=N)[nH][nH]c2c1 78049,c1(C(N2C(C(=O)NC3CC3(F)F)CC3CC32)=O)ccc(O)cc1O 78050,N1(C(C)=O)CCC2(CC1)CC(NC(=O)C(C)CS(C)(=O)=O)C2 78051,c1(C(C(=O)NCCSC)N(C)Cc2ccnc(Br)c2)noc2ccc(Br)cc12 78052,C(=O)(C1=Cc2ccccc2C1)N1CCC(CNC(C(CO)N(C)C)=O)C1 78053,C1(CC)CN(C(=O)C(N2CCCC2)C2CC2)CCC1NC(c1ccncc1)=O 78054,N1(C(CCC(=O)N(CC)CC)=O)CCC(NC(=O)C(C)(C)CO)C(C)(C)C1 78055,C(CC1c2ccccc2CCN1C(=O)Cn1ccnn1)NC(c1c(C)c[nH]n1)=O 78056,O=C(C#CC1CC(F)(F)C1)N1CCCC(F)C1 78057,C(C)(C)(CCCNC(=O)C(CNC(C)=O)Sc1cccc(Cl)c1)NC(COC)=O 78058,CC1CCCCC1(CNC(=O)CCC1CCCCO1)NC(=O)C1=CCCOC1 78059,c1(C(=O)NC(CC)CNC(=O)C(C)(C)F)ncc(OC)cc1F 78060,N1(C(C(CC)n2cncn2)=O)CC(F)(F)CC1CNC(c1ncccc1C)=O 78061,C#CCC(C)(C)C(=O)N(C1C2CN(C(c3ccc(C(F)F)nc3)=O)CC12)C 78062,Cc1ccncc1C(=O)NC1(CCNC(c2occc2Cl)=O)CC1 78063,C1(CNC(=O)CN2CC=CC2)CCCCCN1C(=O)CC1COCCO1 78064,C(=O)(C(C)(C)CN(C)C)NCc1c(C(=O)NCCN(C(C)C)C)occ1 78065,C(=O)(CCC(C)SC)N(C(CNC(C1(C=C)CCC1)=O)Cc1ccccc1)C 78066,N1(C(c2cnc(Cl)cn2)=O)CCC2CN(C(c3cccc4sccc34)=O)CC2C1 78067,c12cccc3c1CN(CC3)C2.C1(c2noc(C3CCCC3)n2)(CC)CCCC1O 78068,N1(C(=O)C(Cl)=CCl)CC(NC(C2(c3cccnc3)CC2)=O)C(F)C1 78069,N1(C(c2cc(C)c(C)nc2)=O)CCCC(NC(=O)C(O)CCC(C)C)CCC1 78070,N1(C(CCC)=O)CCCC1C(=O)NC(CNC(=O)COc1ccccc1)C1CC1 78071,N1(C(C(N)=O)=O)CC23CCCCC2(C1)CN(C(c1cc2c(Cl)cccn2n1)=O)C3 78072,C1(COCCOC)CN(C(C2CCCN(c3ccc(Br)cn3)C2)=O)CCO1 78073,n1(CCC)nc(C)cc1C(=O)NC1CCCCC1NC(c1n[nH]c(C)c1C)=O 78074,C1(C(=O)NC2C=CC(CNC(CSC(C)(C)C)=O)C2)C2CC(F)(F)CC12 78075,Cn1ncc2c(NCC3CSC3)nc(N3CCOC(C4CCOC4)C3)nc12 78076,C1(NC(C=C(C)C(C)(C)C)=O)C(C)CCN(c2ccnc(C3CC3)n2)C1C 78077,N1(C(CCCCC)=O)CCN(C(c2ccn(CCC(F)(F)F)n2)=O)C(C)C1C 78078,C#Cc1ccc(CCCC(N2CCC(O)C(NC(=O)CC(C)OC)C2)=O)cc1 78079,c1(C(N(CC(=O)NCC2CCCC(O)C2)CC2CC2)=O)cc2ccccn2n1 78080,CCN=C(NCc1noc(-c2ccccc2)n1)NC(c1cccs1)C 78081,C1(C(=O)NCCCC(O)CO)CCN(C(=O)Nc2ccccc2)CC1 78082,C(=O)(C1=CC(C)CC1)NCCC(C)NC(c1c(C)occ1C(F)(F)F)=O 78083,C(=O)(C(F)C(C)C(F)(F)F)NC1CN(C(c2cccc(C)c2C)=O)C(C)C1 78084,C1(CNC(C2C(C)C(=O)C2)=O)CCCN(C(=O)C(c2cscn2)N(C)C)C1 78085,C#Cc1ccc(Cl)c(C(=O)NC2CCCN(C(C3CCC(C(N)=O)C3)=O)C2C)c1 78086,C1(C(N2CCN(C(C3(O)CCSC3)=O)CC23CCC3)=O)CCCCC12OCCO2 78087,CN1CC(CC(=O)NOc2ccc(N)c(Cl)c2)CCC1C(F)(F)F 78088,C(=O)(C1=C(C)OCCS1)NC1C(OC)CN(C(=O)CN2CCC(C)(C)C2)C1 78089,C=CC(C)N=C(NC1CC(OCc2ccccc2)C1)N1CCC(C2CCOC2)CC1 78090,C(=O)(CC1COCc2ccccc21)N1CC(F)(CNC(C2(C)ON=C(C)C2)=O)C1 78091,C12(C(=O)NC3C(NC(C(C)C4CCOC4)=O)CCOC3)C3C4C1C1C2C3C41C 78092,C1(O)(CNC(C(CC=C)c2ccccc2)=O)CCCN(C(=O)C(=O)NC(C)C)C1 78093,N1(C(c2cnn(C3CCOCC3)c2)=O)CC2(C1)CN(C(C1(Cl)CC1)=O)CCO2 78094,c1(C(N2CCC(O)(CCNC(CC(C=C)C)=O)C2)=O)cc(F)c(C(F)F)cc1F 78095,C1(NC(c2coc(Cl)c2)=O)C2CC3CN(C(c4ccc5n[nH]cc5c4)=O)C1C3C2 78096,CCC(CC(=O)NC(CNC(c1csc(-c2ccc(Cl)cc2)c1)=O)CO)C(C)C 78097,c1(N2CC(C)OC(C)C2)nc(Nc2ccc3c(c2)C(C)CO3)[nH]c2ncnc1-2 78098,c1(N(C2(CCO)CCC2)C)ncccc1S(=O)(=O)NCc1n(CC)ccn1 78099,C#Cc1cn(C)nc1C(=O)N(C1CN(C(=O)CC2CS(=O)(=O)C2)C1)C 78100,CC1CC(C(=O)Nc2cc(C3CCCNC3)no2)C(C)O1 78101,C12(CC(=O)NCCC(CC)C)CCC1CN(C(c1cc(CO)on1)=O)C2 78102,N1(C(C2Cc3ccccc3C2)=O)CC2(CCCCN2C(C2CCCS2)=O)C1 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78120,c1(NC(C(CCNC(=O)OC(C)(C)C)N(C)C)=O)ccc(-n2cccc2)c(F)c1 78121,c1(C(=O)NCC(CN(C(C2(C#C)CCOCC2)=O)C)O)ccc(C)c2c1CCC2 78122,C(=O)(CC(CNC(=O)Cc1cccnc1F)OC)NCc1cc(C(=O)OC)no1 78123,C1(CCNC(=O)Cc2ccccc2)CCCCN1C(C1CC=CCO1)=O 78124,c1(C(=O)NC2CC(OC)CN(C(c3coc(C)c3)=O)C2)c(F)c(F)cc(F)c1F 78125,c1(C(=O)NCCCc2cccc(N(C)C)c2)cc(S(C)(=O)=O)ccc1N 78126,C1(NC(c2c(C)nc(Br)s2)=O)CCC12CN(C(c1cnsc1)=O)C2 78127,CCCCC(CC)C(=O)NCCC1(O)CCN(C(c2ccc([N+](=O)[O-])cn2)=O)C1 78128,Cc1cc(CCC(N2CCC(C(C)(C)NC(=O)C(F)=CC3CC3)C2)=O)no1 78129,N1(C(c2cc(CC)[nH]n2)=O)CCC(C(C)(C)C)(CNC(C2C(F)(F)C23CC3)=O)C1 78130,c1(C(N(C(C)C(=O)NCC(O)C2(Cl)CC2)C2CC2)=O)c[nH]nc1C(F)F 78131,c1(C(CC(=O)Nc2ccc(N(c3ccccn3)C)nc2)N)ccc(C#N)cc1 78132,c1(C(=O)NC2C(SC)CN(C(c3cccc(F)c3N)=O)C2)ccc(F)c(C)c1C 78133,CCCC(CCC)=CC(=O)NC1(CNC(C2CNC(=O)C2)=O)CCC1 78134,c1(C(C)NC(N2CCC3(C(C(=O)OC)C3)CC2)=O)cn(C)c2cc(Cl)ccc12 78135,c1(C(C(=O)NCCCN(C(c2ccncc2)=O)CC)(C)C)cccc(OC)c1 78136,C1(NC(c2n[nH]c(C)c2Cl)=O)CN(C(C2(C3CCC3)CC2)=O)CCC1CO 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78154,c1(C(N2CCC(NC(c3c(C)ncnc3)=O)C2C)=O)cc(C)c2[nH]cnc2c1 78155,c1(OC)ccc2c(c1)OC(C(=O)OC(=O)COC1CCCC(C)C1)C2 78156,C(=O)(CCCN=[N+]=[N-])NCC12CC(NC(C(C)NC(CC)=O)=O)(C1)C2 78157,N1(C(C)=O)CC(CNC(c2ccnn2CC2CC2)=O)CC(C)(C)C1 78158,C(=O)(N=c1[nH]onc1-c1cccnc1)NC1C(COCCOCCOCCOC)C1 78159,c1(NCC2CC(C)C2)[nH]c(=NCCCC2CCCN(C)C2)nc2scnc12 78160,C1(C)(C(=O)NC(C(C(=O)NC(c2c(C)cccc2)C)C)C)CC2CCC1C2 78161,Cc1c(Cl)ccc2c1CN(C(C1CC13CCC3)C(=O)NC1CCOC1)CC2 78162,c1(C(Cn2cccn2)NC(c2cnc(C(C)(F)F)s2)=O)ccc(Cl)cc1 78163,C1(CNC(CCC=C)=O)CCN(C(C2(C3CCCO3)CCCC2)=O)C1(C)C 78164,c1(C(c2nnnn2C2CCC2)NCC(COC)OC)c(C)c2ccccc2n1C 78165,c1(C(N2CCCC(C)(CNC(C3=C(C)CC3)=O)C2)=O)cnc2cc[nH]c2c1 78166,c1(CN(C(C(=O)Nc2c(C)n(C3CCOC3)nc2)=O)C)cccc(Cl)c1Cl 78167,C1(C(=O)NC2CC(F)(CNC(C3(C(=O)NC)CCC3)=O)C2)Cc2ccccc2C1 78168,CC(CN(C(=O)C(C)N(C(c1ncccc1Cl)=O)C1CC1)C)C(F)(F)F 78169,c1(NC2C(F)CN(Cc3cccc(C(F)(F)F)n3)CC2)ncc2sccc2n1 78170,N1(C(c2cnc(C)[nH]2)C(=O)NCCCC)CCC(c2nncs2)CC1 78171,C(=O)(N1CCCc2nncn21)C1CC(NC(CC2COCC(C)O2)=O)C(O)C1 78172,C#CCCC(C(=O)N(C)Cc1ccoc1)NC(=O)CCOCC(C)(C)C 78173,c1(OC)cccc(CC(=O)N(C2CCN(C(=O)CCc3c(C)c[nH]c3C)C2)C)c1 78174,C(=O)(CCC(=O)NC1(C(N2CCC(NC(N)=O)CC2)=O)CCCC1C)NC 78175,CCCCCC(C)(C)C(=O)N1CCCC(C2(NC(c3cn(CC)nn3)=O)CC2)C1 78176,C1(CNC(CCC)=O)CCCCC1NC(=O)C=CCN1CCCC1 78177,N1(C(C(CCOCC)N)=O)CCC2(CC1)C(=O)Nc1cc(Br)ccc12 78178,c1(C(=O)NCC2(C)CCC(NC(c3cn[nH]c3)=O)C2)ccc(N)c(Cl)c1 78179,C(=O)(C#CC1(C)CC1)N(C(C)Cc1ccc(NC(=O)CO)cc1)C 78180,c1(OC)c(C(=O)N(C(C)CNC(=O)CNc2ncccn2)C)cccc1C(F)F 78181,N1(C(=O)CCc2nccs2)CCC(CCC(N2CCCC2CCO)=O)CC1 78182,C1(NC(C2(CCCC)CC2)=O)CCN(C(=O)CN2CCC(C)C2)CC(C)(C)C1 78183,N1(CC(C)O)CCN(C(c2cc(CNC(C34CCC(CC3)C4)=O)cs2)=O)CC1 78184,c1(NC(C2CC3(CC(NS(=O)(=O)CCBr)C3)C2)=O)cccc([N+](=O)[O-])c1F 78185,c1(C(=O)NC(=O)NC(CNC(=O)CC2(CC3CC3)CCC2)C2CCC2)cc(O)cs1 78186,N1(C(c2c(CC)nn(C)c2)C(=O)NC(C)CC)CC(N=[N+]=[N-])CCC1(C)C 78187,c1(OC)ccc(S(C)(=O)=O)cc1C(=O)NC1CN(Cc2cn[nH]c2)CCC1(F)F 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78206,C(=O)(C(C)CC(N)=O)N1CCC(NC(c2c(C)nsc2C)=O)C1 78207,C(=O)(CCCC(C)(C)C)N1CCCN(C(C2N(CC)CCCC2)=O)CC1 78208,CCCC(CC(C)C)C(=O)NC1CCC(C(=O)NC2CC3CC(OC)C3C2)C1 78209,c1(N(CCOCC)C)nc(-c2cccc([N+](=O)[O-])c2)nc(=NC(C)CCO)[nH]1 78210,N#Cc1ccc(F)cc1C(N1CC2C(C1)N2C(C1CCC2(CC1)CC2)=O)=O 78211,C(=O)(CC(O)CNC(=O)C(c1ccccc1)O)N(CCC)CCC 78212,O=S(=O)(CCO)c1ccc(CNCC2CN(c3ncccn3)CCO2)cc1 78213,C1(C)(CNC(c2nccc(CC)c2)=O)CCCN(C(C2CCC3(CC2)CC3)=O)C1 78214,S(=O)(=O)(CCC(=O)N1CCC12CN(C(C1(C)CCOC1)=O)C2)N(C)C 78215,CCCCC(O)C(C)C(=O)NCc1ccc(C(N2CCC(c3ccco3)C2)=O)o1 78216,N1(C(C2(C=C)CCN(C(c3ccn4cncc4c3)=O)C2)=O)CC(=O)N(C)C(C)C1 78217,N1(C(C2CC(C)OC2C)=O)CCC(C2CC2)(CNC(=O)CSC(F)(F)F)C1 78218,c1(SCC)cc(C(N2CC=CC(NC(=O)C(C)N(C)C)C2)=O)ccn1 78219,Cc1ccc(-c2ccc(N3CCCC3)nc2)cc1NC1CC(C)OC(C)C1 78220,C1(CNC(C(C)N(CC(F)(F)F)C)=O)(CNC(C2(CCF)CC2)=O)CC12CCC2 78221,c1(C(=O)NCC2N(C(CCc3c(C)noc3C)=O)CCC2)c(Cl)ccc(Cl)c1O 78222,N1(C(c2cn(C)nn2)=O)CC2(CC(NC(=O)C(F)C3CC3)CO2)C1 78223,C(=O)(C1CCCc2ncc(C)n21)NC1(CNC(c2cnc(C)o2)=O)CCOCC1 78224,c1(COC)nnc(N2CCCC(C(C)(F)F)C2)n1CCC(=O)OC(C)(C)C 78225,Cc1ncc(C(=O)NC2CCC2NC(c2cnnc(O)c2)=O)cc1C#N 78226,c1(CC(C)C(=O)NC(C2CCN(C(C3C(C)C3C)=O)CC2)C)ccc(F)cc1 78227,CCCC(C)(O)CC(=O)N1CCC(CNC(c2cnncc2C(F)(F)F)=O)CC1 78228,C1(C(=O)NCC(C)NC(C2(COC)CCCCO2)=O)CCn2ncnc2C1 78229,c1(NC(c2cc(Br)nn2C(C)C)c2n(CCCOC)nnn2)cc(Cl)cnc1C 78230,N1(C(c2c(N)cc(F)cc2)=O)CCC2(CCC(NC(c3cnc[nH]3)=O)C2)CC1 78231,c1(OC)cnnc(C(=O)N(CCN(C(=O)C(=O)Cc2ccc(O)cc2)C)C(C)C)c1 78232,N1(C(c2ccnc(C)n2)=O)CCC2(CCCN(C(c3ccnc(Br)c3F)=O)C2)C1 78233,C1(NC(COC)=O)CS(=O)(=O)CC1NC(c1ccc(N)c(CC(C)C)c1)=O 78234,S(=O)(=O)(c1ccc(F)cc1)NCCOC.C1(C(=O)NCC(=O)OCCN)CCCCS1 78235,N1(C(C(C(C)C)NC(CC(=O)OCC)=O)=O)CC(=O)N(C)C(C)C1 78236,N1(C(CC2N(C(Cn3c(C)cc(C)n3)=O)CCCC2)=O)CCCC2(CC1)CC2 78237,n1(-c2ccc(CCCN3CC(CO)OCCC3)cc2)nnc2ccccc12 78238,c1(CN(CC(C)(C)CO)CCC)ccc(OC)c(CC2CC2)c1 78239,CN1CC(CNC(C2(C)CCN(C(C3CC(=O)CCO3)=O)C2)=O)CC1=O 78240,C(=O)(C(C)(CC)CCCCC)N1CCC(OCCNC(C(CC=C)(C)C)=O)C1 78241,CC1CCOCC1C(N1CC(CO)C1)=O.C1C(=O)N1C 78242,Cc1ccsc1C(=O)NCCCCc1cn(Cc2nc(C(=O)O)cs2)nn1 78243,c1(OC)ccc(Br)nc1NC(c1ccc(NC(c2ccccc2SC)=O)cn1)=O 78244,C1(CNC(CCN(C(C)=O)C)=O)CN(C(=O)CN(C2CCCC2)C)CC12CCC2 78245,c1(C(C)C)noc(C(C)NC(=O)CC2CCN(C(C3CNC(=O)N3)=O)C2)n1 78246,c1(C(=O)NC(C2CCCN2C(=O)COC2(C)CCC2)C)ccc(F)cc1F 78247,C1(CCC)CN(C(=O)C(CCOC)OC)CC1C(=O)NCC(C)C(C)O 78248,C1(C2CCN(C(C3CC34CC4(F)F)=O)CC2)(NC(c2c(OC)n(C)nc2)=O)CC1 78249,c1(-c2c(NC(C)CNC(=O)Nc3ccc(Cl)nc3)cnn2C)ccc(F)cc1F 78250,c1(CC)oncc1C(N1CCC(CNC(C2CC(C)(F)C2)=O)C1)=O 78251,c1(C(=O)NC2C(CNC(C(C)(F)F)=O)C2)cnc2cc(Br)ccn12 78252,C(=O)(C1CCCn2cnnc21)NC(CCNC(C(F)=C(C)C)=O)C 78253,N1(C(c2[nH]cc(C(=O)OC)c2)=O)CC2(CCC2)CC1CNC(C1CNC(=O)N1)=O 78254,c1(SC)cc(=NC(=O)NC2CCN(Cc3cccc4ccccc34)CC2)[nH]n1C 78255,N1(C(C2CC(CCNC(=O)Cn3ccccc3=O)C2)=O)Cc2c[nH]nc2C1 78256,CC1CS(=O)CCN1C(C1CN(C(C2CNC(=O)N2)=O)CCN1C)=O 78257,c1(C(=O)NC2CCC(NC(C3(CC=C)CC3)=O)CC2)cc(F)c2c(c1)CCC2 78258,Cc1cn(CC(=O)N(CCCCN(C(=O)C(C)C(F)(F)F)C)C)c2ccccc12 78259,C1(NC(c2n(CCC)ccc2)=O)CCOCC1C(N1CCC1(C)C)=O 78260,N1(C(C2OCCN(C)C2)=O)CC(C2CC2C(=O)NCc2ccc(Cl)o2)C1 78261,c1(C(=O)OC)cc(CCC(=O)N2CC(NC(c3cnc(CC(C)C)s3)=O)C2)c[nH]1 78262,N1(C(CC(C)C)=O)CCC2(CCC(NC(=O)C(N)=O)C2)C1 78263,C=C1CCC(C(=O)NC(CN(C)C)C(=O)NC2(CCOC)CC2)CC1 78264,CCC(C)(CNC(=O)CSC)NC(=O)Cc1ccccc1.c1(C(=O)N)cc(C)no1 78265,C(c1ccc([N+](=O)[O-])cc1)=C(C)C(=O)NCCN(C(=O)CCCC(N)=O)C(C)C 78266,Cc1cc(C#N)cc(NC(=O)CCC2CC(F)C2)n1 78267,N1(C(=O)CC2CCN(C(c3ccnn3CCF)=O)CC2)CC2(CCNC2=O)C1 78268,c1(NC(C)=O)ccc(C)nc1C(=O)NC(C)CNc1cccc(C)c1C 78269,c1(C(N2CCCC(N(C(C(C#C)(C)C)=O)C)C2)=O)c(F)ccc(C(=O)OC)c1C 78270,c1(NC(N2CC(N3CCN(C(CC(=O)OC)=O)CC3)C2)=O)cc(S(N)(=O)=O)co1 78271,N1(C(CC=C(C)C)=O)CC(O)(C2CCN(C(C3(C)CC(C(C)C)=NO3)=O)CC2)C1 78272,N(C(=NCC1CCCS1)NCc1cccnn1)C(C1CCCO1)C 78273,C1(CNC(CCC=CC)=O)C2CCC(C2)N1C(c1ccc(F)c(F)c1)=O 78274,N1(CC(N2C(C(C)NC(c3cnc(C)[nH]3)=O)CCC2)=O)CCC(C(F)(F)F)CC1 78275,N1(C(c2[nH]cc(C)c(=O)c2)=O)CCC2(CCN(C(=O)C(C)CC(N)=O)C2)C1 78276,c1(CS(N)(=O)=O)cc(C(N2CCC2C2CC2)=O)n[nH]1.n12cc(nn1)C1(CCC1)C2 78277,C1(NC(C2(O)CC(C)(C)C2)=O)CN(C(C2CC23CCOC3)=O)C2CCCCC12 78278,C1(C#N)(CNC(C2(CNC(=O)NC3C(OCC)COCC3)CC2)=O)CC12CCC2 78279,CC(C)N(O)C(=O)C(=O)N1CC(C)(C)OCC1CNC(=O)C(C)n1ccnc1 78280,C1(NC(=O)CN2CC3CC3C2)CCCC(NC(C2CCC(F)(F)C2)=O)C1 78281,C1(NC(c2cc(C3CC3)cc(F)c2)=O)CCN(C(c2cccc[n+]2[O-])=O)C12CC2 78282,c1(CN(C2CC3CNC2C3)Cc2nccc(C)c2)ccc2c(c1)OCC2 78283,CS(=O)(=O)c1cccc(-c2ccc3nc(C(=O)N=c4[nH][nH]cc4Br)cn3c2)c1 78284,c1(OC)cc(CN2CC(C(=O)O)C(NC(=O)C=C(C)C)C2)c(OC)cc1Cl 78285,c1(C(=O)NC2C=CC(CNC(C3ON=C(CC)C3)=O)C2)cc(F)c(Cl)cc1F 78286,C1(NC(c2cccc(Cl)c2F)=O)CN(c2ncnc3sccc23)C2CCCCC12 78287,N1(C(C2(CCC)CC2)=O)CCC(CNC(c2cn(C3CC3)cn2)=O)C(O)C1 78288,c1(C(N2CC(C)(NC(CCCC)=O)C2)=O)cnn(-c2ccncc2)c1C 78289,c1(SC(C)C(N2CC(NC(C3CCS(=O)CC3)=O)C(C)C2)=O)ccc(F)c(F)c1 78290,N1(C(CC2C(C)(C)C2(C)C)=O)CC2CN(C(C3(C#N)CCCCC3)=O)CCC12 78291,CC(C)(C)C(=O)NCC(=O)NC1CCC(NC(c2ccccc2)=O)C1 78292,CC1OCCC1(C)C(=O)NC1CN(C(=O)Cn2cc(C(F)(F)F)cn2)C1 78293,C1(NC(CC=C(C)C)=O)CC2CN(C(=O)C(C)(C)COC(C)C)CC2C1 78294,N1(C(C(C(CC)C)N(C)C)=O)CC(C(N2CCCC3(C2)N=N3)=O)C2(CCC2)C1 78295,N1(C(C2C=C(C)CS2)=O)CC(C2CC2C(=O)N(C)CCO)C1 78296,N(C1CCCn2ccnc21)C(CCCC(CC)NC(CC(=C=C)C)=O)=O 78297,c1(C(=O)NCC2C(NC(=O)COc3cncc(Cl)n3)C2)cnc2n1CCC2 78298,n1(CCOC)cc(NC(C2CN(C)C(=O)CN2)=O)ccc1=O 78299,N1(C(c2c(CC)nns2)=O)CCCC(C(C)NC(=O)C(C)(C)C2CCOCC2)C1 78300,c1(CC(=O)NC(CNC(C(CC#C)O)=O)CO)ccc([N+](=O)[O-])cc1 78301,c1(C(N2CC3CN(C(COCC)=O)CC3C2)=O)cc(Br)c2c(c1)OCCO2 78302,N1(C(CC(C=C)(C)C)=O)CC(C)CN(C(c2c(F)cc(OC)cc2Cl)=O)CC1C 78303,c1(NC(C2N(C(C=CC=CCC)=O)CC(O)CC2)=O)cncc([N+](=O)[O-])c1 78304,Cc1ccc(N(C(=O)CCC2NC(=O)NC2=O)C)cc1C 78305,c1(C(C(=O)NCC2CC(F)(CNC(C34CC(OC)(C3)C4)=O)C2)O)ccc(F)cc1 78306,c1(C(=O)NCC(CC)NC(c2cn(C(C)(C)C)nn2)=O)c[nH]c(C)c1 78307,C1(CNC(CN(C)C(c2ocnc2C(F)F)=O)=O)CC(O)C12CCC2 78308,C1(O)(C(C)NC(C(CC#C)C)=O)CCN(C(c2ccnn2CCF)=O)CC1 78309,C(=O)(C1CCc2ccc(Cl)nc21)NC1CN(C(C(N)=O)=O)CC1CCO 78310,CC(C)(C)CC(F)C(=O)NC1CN(C(C2CN3CCC2(C)CC3)=O)CC1O 78311,c1(C2C(C)C2)ccc(C(=O)N(C)CCN(C)C(c2csc(Cl)n2)=O)o1 78312,c1(NC(C2CCCN(C(c3cc(O)cc(Cl)c3)=O)C2)=O)cccc([N+](=O)[O-])c1Br 78313,C1(CN(C(CN(C(C2OCC(C)(C)C2)=O)C2CC2)=O)C2CC2)CC2CCCC2C1 78314,CC1=C(C(=O)N2CCC(CO)(NC(=O)CCc3cc(C)cc(C)c3)C2)SCCO1 78315,Cc1ncc(C(=O)N(C2CN(C(c3nn(C)cc3Br)=O)CC23CC3)C)cc1N 78316,CC1(C)CC(C(F)(F)F)(C(=O)NC2CN(C(C3(n4cncn4)CC3)=O)CC2O)C1 78317,C1(=CC(=O)NC(C2N(C(c3c(C)oc(Cl)n3)=O)CCCC2)C)CN2CCC1CC2 78318,Cc1ncc(C(=O)NCC2CCN2C(C2CC23CCCC3)=O)cc1CC(C)C 78319,C1(C(=O)NC(C)CCN(C)C)COC(CNC(=O)COCCN(C)C)C1 78320,n1(C(C)C)cc(Br)c(C(=O)NCC23CC(CN2C(=O)C(C)C#N)C3)n1 78321,c1(N2CCC(C)(CNC(c3cnc(Br)s3)=O)CC2)ccncc1[N+](=O)[O-] 78322,CC1(C)CC(NC(C2CCCS2(=O)=O)=O)CN1C(c1csc2nnsc12)=O 78323,CCCC(C(=O)N(C(CC)C1CC1)C)NC(=O)C(F)COC 78324,CC(C(=O)N(CCCCNC(=O)C1=NOCC1)C1CC1)C(C)(C)c1ccccc1 78325,CCCCC(CNC(=O)C(C)=C1CC1)NC(c1ccccc1OC1CCCC1)=O 78326,CCCC(C)(CCC)C(=O)NC(C1CN(C(=O)Cc2ccc(C)nc2)CCO1)C 78327,N1(C(c2noc(C)c2[N+](=O)[O-])=O)CCCCC(C2CN(C(C3(F)CC3)=O)C2)C1 78328,C(CC(CC)C(=O)N(CC(=O)N(CC(C)(C)O)C(C)C)CCOCCOC)=CC 78329,N1(C(Cc2ccc(C(=O)OC)nc2)=O)CCCC(NC(=O)C(F)C(C)(C)O)C1C 78330,c1(C(=O)OCCn2ncc(C)c2)csc2ccc(F)cc12 78331,c1(OC)ccc2c(c1)C(N(C)C(c1cc(C)c(Cl)s1)C(=O)NCCC#N)CC2 78332,N1(C(CCN(C(=O)CC2C(CC)C2(F)F)CC=C)=O)CCCC(C)C1CCO 78333,Cc1ccc(C(N2CCCCC2C(=O)NCC2=NOC(C)C2)=O)nc1C 78334,c1(C(C(F)(F)F)NC(=O)NCc2cn(C(C)C)nn2)ccc(F)c(Cl)c1 78335,C12(C(N)=O)CCCC1(C(=O)NC1CCCC1NC(=O)Cc1nnc(O)s1)C2 78336,C1(C(=O)NC2CCC2)COCCC12CN(C(c1ccnc(Cl)n1)=O)C2 78337,N1(C(c2cc(CC)ncn2)=O)CCCC(O)(CCNC(c2ccc(Cl)o2)=O)C1 78338,c1(C(=O)NCC2N(C(c3cnc(=N)[nH]c3)=O)CCC2)ccn2nnnc2c1 78339,N1(C(C(C)=C2CCC2)=O)CCC(CC(N)=O)(NC(=O)CCn2cncn2)CC1 78340,C(=O)(C1CCCc2sccc21)NCC(C(C)C)NC(c1nc(CC)oc1)=O 78341,C1(OC)CCC(C(N2CC(F)CC2CC(=O)NCC(C2CCCC2)O)=O)CC1 78342,c1(C(=O)NCC(n2ccnc2)C)cn(C2CCOC2)nn1 78343,C(CC(=O)NC1CC1CN(C)C)N(C(=O)C(C)n1cncn1)CC=C 78344,c1(OC)ccc(C(C)(C)C(=O)NC(C2CN(C(=O)C(O)CN(C)C)C2)C)cc1 78345,c1(C(N2CCCC(CC)C2)C(=O)NCC(=C)C)csc([N+](=O)[O-])c1 78346,c1(C(=O)NCCOCCCNC(COC)=O)cnn(C)c1C(C)(F)F 78347,C(=O)(C(C)(C)CCCF)NCC1C(C)CCN1C(c1cccc(N)n1)=O 78348,C(=O)(C1CCCn2cnnc21)NCC(CO)NC(c1ccc(OCOC)cc1)=O 78349,c1(C(=O)NCCCC(C)NC(C(COC)C)=O)cc(C2(C)CC2)ccc1F 78350,c1(CNC(C(=O)Nc2ccc(OC)c(C)n2)=O)c(C)cc(Br)cc1C 78351,CC1(C)C2CCC(C2)C1C(N1CC(NC(C2CC(O)C2)=O)C1)=O 78352,c1(NS(C)(=O)=O)cc(C(F)(F)F)ccc1C(COC(C(COCC)O)=O)=O 78353,c1(OC)ccn2cc(C(N3CC=CC3CNC(c3cc(Cl)c[nH]3)=O)=O)nc2c1 78354,c1(C(N2CCC(NC(c3cn(CC=C)nn3)=O)C(C)C2)=O)c(N)cc(F)cc1Cl 78355,CC(C)C1=NOC(C(=O)NCC2CCN2C(C2CCC3CC3CC2)=O)C1 78356,C1(NC(c2cnn(C)n2)=O)CCCCC12CCCN(c1nc(C3CC3)ns1)C2 78357,c1(C(N2C3C(NC(=O)C(F)n4ccnc4)C(C3)C2)=O)ccc(Cl)c([N+](=O)[O-])c1 78358,c1(C(=O)NC2CCC(CNC(C3C(C)(C)C3(F)F)=O)C2)cc(F)ccc1F 78359,c1(N(CC)CC)cncc(NCc2csc(-c3ccccc3OC)n2)c1 78360,C(=O)(C1=CNC2=NCCCC2=C1)N(CC(CO)(CO)NC(CSC(C)C)=O)C 78361,CC1CCC(CNc2ccccc2)CN1 78362,N1(C(c2cc(Cl)nc(Cl)c2)=O)CC2CC(C1)N(C(c1coc(O)n1)=O)C2 78363,C1(NC(c2ccc(C)cn2)=O)CCN(CC(=O)NCc2ccco2)CC1C 78364,C1(CNC(C(COC)(C)O)=O)CC2CCC1N(C(c1cnn3c1OCC3)=O)C2 78365,c1(CN(c2ccccc2C(C)C)C(C(C)OCCOC)=O)cccc(C#N)c1 78366,C(=O)(C(F)(F)C(C)(C)O)NCC(=C)CCNC(=O)C(c1ccccc1)F 78367,N1(C(CCSC)=O)CCC2(NC(=O)CCCCC(C)C)CCCCCC12 78368,C1(NC(CCC(C)OC)=O)CN(C(c2cnc(O)c(Cl)c2)=O)CCC1(C)C 78369,Cn1cc(C2CC2NC(=O)CCCn2cc(CCC3CCCCC3)nn2)cn1 78370,C1(CC)CCN(C(=O)C(=O)NCC2(C(=O)NCCC(=O)NC)CC2)C1CC 78371,c1(C(=O)NC2C(NC(c3sccc3C3CC3)=O)CC2)cn2c(n1)CCC2 78372,C#Cc1ccc(C(=O)NCC(C)(C)C(=O)NCC2(COC)CCCC2)cc1 78373,c1(C(=O)NCC2(C)CCN(C(c3c(C(C)C)cco3)=O)C2)ccc(N)c(Cl)c1O 78374,C(=O)(C(F)(CNC(C1(C)CCC(=O)C1)=O)C(C)C)N(C(C)C)CC 78375,N1(CCN(C(c2c(C)cccn2)=O)C)CC2CCC(C1)O2 78376,C1(NC(CC(COC)C)=O)CCN(CCOc2ccc(Cl)cc2)CC1C 78377,c1(C(N2CC(CNC(C3C(=C)C3)=O)CC23CCC3)=O)csc2cccc(F)c12 78378,CC(C)CCCC(C)CNC(=O)C(F)CC1CN(C(C2CC2[N+](=O)[O-])=O)C1 78379,c1(OC)cccc(CNC(=O)OC(C)(C)C)c1C.C12CCCN(C1)C(=O)C(=O)N2 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78398,N1(C(CCc2ncc(C)[nH]2)=O)CCC2CN(C(=O)C#CC3(C)CCCO3)CC2C1 78399,c1(C(N2CC(C(C(N3CC(C4CC4)(COC)C3)=O)OC)C2)=O)ccc(C)c(C#N)c1 78400,c1(C(=O)OC)cc(NC(=O)NC(C2CCCC2O)C)c2c(c1)CCC2 78401,CC1CCC(NC(=O)C=C2CCCC2)CN1C(c1cc(Br)n(C)c1)=O 78402,c1(C(CNC(=O)NC(CC)C(F)F)CC)ccc(F)c(F)c1 78403,N1(C(c2ccc(NC=O)cc2)=O)CC2CN(C(=O)C(=O)c3ccco3)C2C1 78404,N1(C(c2cc(C3(C)CC3)n[nH]2)=O)CC(CN(C(=O)CO)C2CC2)C(C(F)(F)F)C1 78405,c1(CC)nc(NC2(CO)CCCN(C(c3sccc3OC)=O)C2)cc(C)n1 78406,c1(OC)cc(C(N2CCCC(SC)CC2)C(=O)NC2CCC2)ccc1S(C)(=O)=O 78407,C1(OCC)CCCN(C(=O)CCC2(CN)CCCCC2)C1 78408,C1(CC=C)(NC(=O)CCN2CCCC2)CCN(C(C2(CSC)CCC2)=O)C1 78409,C1(CNC(=O)C=CCN2CCCC2)(NC(C2COC(=O)N2)=O)CCOC1 78410,CC1CCN(C(=O)Nc2coc(Oc3ccccc3)n2)CC1Nc1ccccn1 78411,CC(C)CCCC(C)C(=O)N1CCC(C(C)NC(C2(C)COC(=O)N2)=O)C1 78412,CCC(C)(C(=O)NC)NC(C(=O)Sc1ccc(F)cc1)C1CC1C(=O)OC(C)(C)C 78413,c1(N2C(CNC(C(C)C)=O)CC(F)C2)cc(-c2cccs2)ncn1 78414,c1(C(=O)NCC2CC(OC)CN2C(c2cscc2OC)=O)cc2cnccc2o1 78415,c1(C(=O)OCC)cc(NC(C2CCCN(Cc3cncs3)C2)=O)ccn1 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78554,CCC(CC(C)C)C(=O)NCC1C2CC1N(C(c1nc(Cl)cc(N)c1Cl)=O)C2 78555,c1(NC(N2CCCC(CCCO)C2)=O)cccc(-c2ccc[nH]2)c1 78556,c1(CC)cc(C(=O)NCCC2CC(NC(C3CN(C(C)C)C3)=O)C2)oc1CC 78557,C(=O)(CCC1=CCCCC1)NC1CN(C(c2c(N)nc(C(F)(F)F)cc2)=O)C1 78558,CC1=NOC(CNC(=O)C(C)(C2CC2)N(C(=O)CN=[N+]=[N-])C)C1 78559,c1(C(=O)NCC(CC=C)NC(=O)Cc2cccnc2C)ccc([N+](=O)[O-])cc1O 78560,C1(C)(C(=O)NC(c2cn(Cc3cnc(C)nc3)nn2)C)Cc2ccccc2C1 78561,CCCC(CC)CCC(=O)NC1CC2(C(=O)NC(C)(CO)CO)COC1C2 78562,C12(NC(=O)OC(C)(C)C)CCCC1CCN2C(c1ccc(F)c(N)c1F)=O 78563,C(CNC(=O)CCC(C)N(C)C)(CC(F)(F)F)NC(Cn1c(C)nnn1)=O 78564,C1(C(=O)OCC)CC(C(N2CCC2(C)NC(CCC)=O)=O)C1(C)C 78565,C(C(CN=c1[nH]cnc(Cl)c1[N+](=O)[O-])C(F)(F)F)C(N(CCN(C)C(N)=O)C)=O 78566,C1(C(CC)CC)CCN(C(c2ncccc2Cl)C)CC1 78567,C(CCC(=O)NCC1=NOC2CCCC12)(C(C)C)NC(c1nc(C)oc1C)=O 78568,N1(C(C(C)(C)C2CCC2)=O)CCOC2(CCN(C(C3CC(=O)N(O)C3)=O)CC2)C1 78569,c1(C=O)ncc([N+](=O)[O-])cc1C.C(=O)(CCCN1CCCC1)N1C2CCN1C2.CO 78570,C1(C(=O)NC(CC)C(F)(F)F)CN(C(c2ccncc2F)=O)CC12CCC2 78571,CC1C(C(=O)NC2CC(F)C2)C(C(=O)O)C1(C)C 78572,c1(C(=O)NC2CC(C(=O)NCCCn3c(C)nnc3)OCC2)c(F)cccc1F 78573,C1(O)(CNC(c2cccc[n+]2[O-])=O)CCCN(C(=O)C(Cl)=CCl)CC1 78574,c1(OCC(N2C(Cn3cc(CCS(C)(=O)=O)nn3)CCC2)=O)ccc(F)c(F)c1 78575,c1(C(=O)NCC(C)N(C)C(c2cc(C3CCC3)no2)=O)cn(CC2CC2)nn1 78576,Cc1cc(C(N2CCC(NC(=O)CCc3ccsc3)C(C)C2)=O)ncc1N 78577,N1(C(Cc2c(C)noc2C)=O)CC2CC1CN2C(=O)C(CC(F)(F)F)N(C)C 78578,C(C)(C(=O)NC1CC(OCC(=O)NCCc2ccncc2)C1)(C1(C)CC1)OC 78579,N1(C(C(c2cccc(C)c2)=O)=O)CC2(CCCC2NC(C2CCC(C)O2)=O)C1 78580,c1(SC)ccc(C(=O)N(CC(O)CNC(=O)CSc2ccccn2)C)s1 78581,CCC(CNC(=O)CCCN(C(=O)C(C)NC(C)(C)CC)C)CO 78582,CC1(C)CC(C(=O)NCC2CC2(F)F)CN1C(=O)CCc1cccc(O)n1 78583,N1(C(CCN(C(C2CCC(C)(C)OC2)=O)CC)=O)CC(S(N)(=O)=O)C1 78584,c1(C(C(=O)NC(C)C)N(C(CC)C#N)C)csc(C(F)(F)F)n1 78585,c1(C(N2C(C(C)NC(CN3CC(C)(OC)C3)=O)CCC2)=O)ccc(N(C)C)cn1 78586,Cc1ccc(CN2CCCC2CCC(=O)N(C)Cc2ccccc2)c(Cl)c1 78587,c1(NCC2(CNC(=O)CSC(F)F)CC2)nc2c(cc1Cl)C(=O)OC2 78588,C1(NC(C(C)OCCN(C)C)=O)CCN(C(=O)C2=CCCCCC2)CC12CCC2 78589,c1(CC)nc(O)c(C(N2CCC3CN(C(C45CCCC4C5)=O)CC23)=O)cc1C 78590,C1(N(C(C(=O)N(CCN(C(C=C(COC)C)=O)C)C)C)C)CCCOC1 78591,C=CCCCCC(=O)N(C)CC1(C)CCCC1NC(c1ccc(C)s1)=O 78592,C1(OCC(=O)N(C)CC2(NC(CN(C(=O)OC(C)(C)C)CC)=O)CC2)CCCCC1 78593,N1(C(Cc2ccn(C(C)C)n2)=O)CCCN(C(=O)CO)C(C)C1 78594,c1(OC)ccn2c(C(=O)NCCN(C(c3c(C)nsc3C)=O)C3CC3)cnc2c1 78595,CN=C(NCCc1noc(C)n1)NCC(=O)N(C)CCc1ccccc1 78596,N12CC3C(C3C1)C2=O.C1(N(C)CC)CC(C(=O)NC(C)Cn2cncn2)C1 78597,C1(C(=O)NCC2C(C)CN(C(c3cc(O)n(C)n3)=O)C2)CN2CCCN1CC2 78598,C(=O)(C(COC)CC(C)C)N(C(C(COC)NC(C1CCC(OC)CC1)=O)=O)CC 78599,C=CC1(CO)CCN(C(=O)C(CCC)NC(=O)CSCC(N)=O)C1 78600,C1(NC(c2cc(C(F)F)ccn2)=O)CC2(CCCCN2C(C2(CO)CC2)=O)C1 78601,C(=O)(CC(O)C(=O)OC(C)(C)C)OC(C)(C)C.C123CC(C1)C(CO2)CN3 78602,S(=O)(=O)(c1cccc(=NCc2cn(C)nn2)[nH]1)NC(c1ccn(C)n1)CO 78603,N1(C(C)=O)CC(O)CC1C(=O)NCC1CCN(C(C2(C)CSC2)=O)C1 78604,C(=O)(CCCCCCCCCO)N(CC(CC)NC(C1(F)CCCCC1)=O)C 78605,Cc1ccccc1C=CC(=O)NC(C(=O)NCC12CCN(CC1)C2)c1cccs1 78606,c1(SC)cccc(C(N2CC(O)CC2C(=O)NC2CN(c3ncco3)C2)=O)c1 78607,c1(C(=O)NCC(Cn2cc(CN(C)CCO)nn2)OC)cc(C(=O)O)oc1C 78608,N1(C(c2n(C)nc(CC)c2Cl)=O)CCCC2(C1)CN(C(=O)C(C)Br)CCO2 78609,n1(CC)cnc2c(NCCc3nc(=N)[nH][nH]3)nc(N(C)CC3CCOC3C)nc12 78610,C1(N(C(C(C)OCC)=O)C)CCCN(C(=O)CCc2nc(CC)no2)CC1 78611,c1(C(=O)NCC(C)CN(C)C(C2CNC(=O)N2C)=O)coc2c(F)cc(F)cc12 78612,O=C(C1CCc2c(Br)cccc21)N1CC(N2CCN(C(=O)C3=CCC3)CC2)C1 78613,C1(C(=O)NCC2(OCC)CN(C(=O)C(C)=CCO)C2)CCNC(=O)C1 78614,c1(OC)ccc(=NC(=O)C23CC2CN(C(c2cc(Br)ncc2F)=O)C3)[nH]n1 78615,n1(CC(=O)N(C2CN(C(c3cnn(C)n3)=O)CC2(C)C)C)nc(Cl)ccc1=O 78616,N1(C(C(C)C2CCC2)=O)CCC(F)(CNC(=O)C(c2cc(Cl)cc(Cl)c2)=O)CC1 78617,N1(C(C)=O)CC2CC1C2CNC(C1(COC)CC1(F)F)=O 78618,c1(C(=O)NC(C)CCNC(=O)CC(C)(C)C)c(O)cnc2cc(F)ccc12 78619,N1(C(C(C)C2CCCO2)=O)CC2(NC(c3ccc(Br)cc3N)=O)CCC1CC2 78620,C1(CNC(=O)C(=O)NC2CC2)CCC2CN(C(c3ccc(O)cc3)=O)CCC2C1 78621,C1(NC(C(C)(C)SC)=O)CC12CCN(C(=O)Cc1ccoc1C)CC2 78622,C(c1cn(C)nn1)=C(C(=O)NCCN(C(c1cc(C)no1)=O)CC1CC1)F 78623,C(=O)(C(C)N(C(C1CCC1C)=O)C1CC1)NCCN(C(C)C)CC 78624,c1(C(N(CC(CNC(c2n(C(C)C)ccc2)=O)C)C)=O)[nH]ncc1C#N 78625,CCCCS(=O)(=O)NCC(=O)N(C)CC1CCCCN1C(=O)CCCCSC.O 78626,c1(C(=O)NC2CN(C(C3(OCC)CCOCC3)=O)CC2C)ccccc1N=[N+]=[N-] 78627,c1(C(=O)NC(CCCNC(c2nnc(C)s2)=O)C)cccc(CO)c1C 78628,CC(C)CCN=C(NCCc1cnn(CC(F)(F)F)c1)NCc1ccc(Cl)nc1 78629,c1(C(C(N2CC(NC(C3(OC)CCCC3)=O)C2)=O)N(C)C)c(F)cccc1F 78630,N1(C(Cc2ccc(OC)nc2)=O)CCC2C(C1)NC(=O)CN2C(C1CC1F)=O 78631,N1(C(C(CC)(F)F)=O)Cc2occ(C(N3CC(CO)CC3CO)=O)c2C1 78632,Cc1cc(C)n(CCNC(=O)CC(N)Cc2ccc(F)cc2)n1 78633,Cc1sc(Br)nc1C(=O)NCC1(C)CCN(C(C2CC(F)(F)C2)=O)C1 78634,c1(C(C(=O)NC2C(OC)CN(C(C3CN(C)C3)=O)C2)O)ccc(Cl)cc1Cl 78635,Cc1cc(C)c2c(=NC(=O)NC(c3ccnc(Cl)c3)C)[nH]sc2n1 78636,Cc1nc2ccc(S(=O)(=O)NCC3(C)CC=CCO3)cc2o1 78637,Nc1ccc(Br)c(F)c1C(=O)NC(c1ccccc1)Cn1cncn1 78638,N1(C(c2cn(CC)nn2)=O)CC2CCC2(CNC(c2oncc2C)=O)C1 78639,c1(CC(=O)NCC2N(C(C(CC)C(C)C)=O)CC2)ccccc1[N+](=O)[O-] 78640,C1(N(C(C(CC)F)=O)C)CN(C(c2ccc(C(=O)NC(C)C)cc2)=O)CC1(C)C 78641,C1(=CC(=O)NCC2C3CN(C(c4c(C)nsc4N)=O)CC32)CCCCC1(C)C 78642,N1(C(c2cc(CC)on2)=O)CC(NC(c2sc3cncn3c2C)=O)C(C2CC2)C1 78643,C(CCCCCC(=O)N1CC2CCC2(CNC(=O)C(O)C(C)(C)C)C1)SC 78644,C(=O)(CC(C)(C)C(F)F)NCCCC(CCC)NC(C1CC1C(=O)OCC)=O 78645,c1(C(=O)NCC(C)CNC(=O)CCCC(C)(C)C)n[nH]c2c1CCCCC2 78646,Cc1cc(C(=O)NCC(C)(C2CC2)NC(c2ccn(C)n2)=O)sc1C 78647,C(CC(F)F)(C(=O)N1CCC2C(O)CC12)NC(=O)CCN1CCOC1=O 78648,c1(NC(c2occ(C(C)=O)c2)=O)ccc(NC(C2(O)CCCCCC2)=O)cc1C 78649,C1(N=c2[nH]nc(C(F)F)s2)(NC(C2(C)CCC(C)(C(=O)OC(C)(C)C)C2)=O)CC1 78650,C(=O)(N=c1cc(C)n(C)[nH]1)C1OCCC(NC(CCCOCC=C)=O)C1 78651,N1(C(CCNC(COC)=O)=O)CCCC1(C(=O)NC1(C(=O)N(C)OC)CC1)CC 78652,c1(OCCOC)ccc(C(=O)NC2CCC(NC(=O)C(C)C(C)C)CC2)cc1 78653,C1(C(=O)NCC2CN(C(CN(CC)CC)=O)C2)CCc2cncn2C1 78654,N1(C(COCC(C)C)=O)CC2C3CCC(C2C1)N(C(c1ncccc1CO)=O)C3 78655,Cc1cccc(C(=O)NCC(=O)NCCCN(C(c2nn(C)cc2Cl)=O)C2CC2)c1 78656,C1(NC(c2n(CCOC)nnn2)CCC2(C)CC2)CCc2ncccc2C1 78657,c1(CC)ccc(CNC(=O)C(CCSC)NC(=O)C2=CCSC2)cc1 78658,Cc1nsc(N)c1C(N1CSCC1C(=O)NCCSCCO)=O 78659,CCCC(C)C(=O)N1CC=CC1(C(=O)NC1CC(C)(C)C1)COC 78660,C(=O)(C1=NOC2COCC12)NC(CCC(=O)NC1(C#C)CCC(C)CC1)(C)C 78661,Cc1nn(C)c(C)c1CC(N1CC(NC(c2cc(C(C)(C)C)n[nH]2)=O)C(C)C1)=O 78662,N#CC1CCCC(C(=O)NC2CC(C(=O)NC3CCOC3)C2)C1 78663,c1(N(CCN(OC)C)C)cc(NCC(C)CC(C)O)nc(C(C)C)n1 78664,CC1CC=C(C(=O)NC2COCC2NC(c2cccc3nccn23)=O)CC1 78665,C1(C)(Cc2cn(-c3n(C)nnc3)nn2)CCN(Cc2csc(C#N)c2)CC1 78666,CC1(C)CCCC(C(=O)NCCC2CN(C(c3cncc(CO)c3)=O)C2)O1 78667,c1(OC)cc(C)c(Cl)cc1CN(CCCN=[N+]=[N-])C(=O)CN1C(C)CCCC1C 78668,CC1=C(C(=O)NCC2(NC(=O)CC3CCCN3C(C)C)CCOCC2)CCC1 78669,Cc1c(C(=O)N(CCC(C(C)C)NC(C2CSC2)=O)C)[nH]c2c1CCCC2 78670,c1(C(CC(=O)O)NC(C2NCCN(CC)C2)=O)cccc(-c2cscn2)c1 78671,N1(C(c2nc(CC)sc2)=O)CC2CC1CN2C1CCN(Cc2ccccc2)C1=O 78672,C=CC1(CC(=O)NC(C)C(C)NC(=O)CC2CSC2)CCCCC1 78673,C1(NC(C(CCOC)OC)=O)CCN(C(=O)Cn2nnnc2C(C)C)C(C)C1 78674,N1(C(c2cc(OC)n[nH]2)=O)CCC2CN(C(=O)CC3CCC=CCC3)CC2CC1 78675,N1(C(COC(C)C)=O)CCC(C)(C)C(NC(=O)COCC2(F)CC2)C1 78676,C1(C(=O)N(CCCN(C)C(c2cnn(CCOC)c2C)=O)C)(CC)CCNC1=O 78677,c1(C(=O)NC2CN(C(c3c(CC)cccc3)=O)CC2F)c(C)nn(CCO)c1C 78678,Cn1cnc(CCNC(=O)CC2(CNC(=O)COCC3CC3)CC2)n1 78679,CCC(C(=O)N1CC(COC)(NC(=O)C(C2CCOCC2)C)C1)OC1CCCC1 78680,N1(C(C2CC(=O)NCC2)=O)CC=C(C(=O)NC2CC3CCCCC23)CC1 78681,CC1(C)COCCC1C(N1CCC(CC(N)=O)(NC(C2(CO)CCC2)=O)CC1)=O 78682,C(CCC(F)(F)F)N(C(c1scc(C(C)=O)n1)=O)C 78683,C(=O)(CC(CC)C(C)(C)C)NCC(CC=C)NC(=O)CNS(=O)(=O)C1CC1 78684,c1(C(N(CC(C)NC(c2cc3ccnn3cn2)=O)C)=O)c(F)ccc(N)c1F 78685,c1(-n2c(CC3(CO)CCCC3)nc(-c3ccncc3)n2)cccc2nc[nH]c12 78686,C(=O)(CC(C)(C)CNC(=O)Nc1cc(C(C)(C)C)ccn1)OCC 78687,C1(C(=O)NC(C(NOCC(=C)Cl)=O)c2ccnn2C)CC2(CCC2O)C1 78688,CC(CCCC(=O)NCC#CC#CCO)NC(C1(CCN(C)C)CC1)=O 78689,c1(C(C(=O)NCCCC)N(C)Cc2ccncc2)ccc(OC)cc1Br 78690,c1(C(=O)NC2(CNC(C3CCC4CCCCN34)=O)CC2)ccc2n[nH]cc2c1F 78691,c1(CNC(CCNC(CCC(=O)OC)=O)=O)ccc(C)c(F)c1 78692,C#CC1(O)CCN(C(C)C(=O)NC(C)CCCCNC(C2CCC(F)C2)=O)CC1 78693,CCCCCCCC(=O)NC(C(=O)NCC12CCN(CC1)CC2)C(C)(C)C 78694,C1(C(=O)NCCCCCN(C(C2CC(C(C)C)C2)=O)C(C)C)CCCS1(=O)=O 78695,c1(C(=O)NCC(n2cncn2)C)ccn(CCNC(=O)CCCc2ncco2)c1 78696,C1(C(N2CC(CC(CNC(C(n3cc(Cl)cn3)C)=O)(C)C)C2)=O)CCC2(CC2)C1 78697,N1(C(c2cc(C)c(Br)o2)=O)CC(NC(c2snnc2C)=O)CC(F)C1 78698,C(=O)(CCS(N)(=O)=O)NCC(N1CCC(C)(CO)C1)=O.C1CN1CCO 78699,c1(CN2CCCC(CNC(c3cccc(OC)c3)=O)C2)cc([N+](=O)[O-])ccc1Cl 78700,C1(NC(=O)CC2COCC2O)C2CN(C(=O)CCCc3ccccn3)CC12 78701,C1(NC(=O)COCC2CC2)CC2CCC1(C(=O)NCC1(F)CCC1)C2 78702,C1(N2C(=O)C2)CCN(C(C2CCOC2C(F)(F)F)=O)C1.C(C(C)C)SC 78703,C1(C(=O)NC2C=CC(CC=CC(N3CC(c4nc(C)on4)C3)=O)C2)CCCN1C=O 78704,C1(CNC(CC2C(C)CCO2)=O)CCCCCN1C(c1csc(=N)[nH]1)=O 78705,N1(C(Cc2c(C)occ2)=O)CCOC(CCNC(=O)CC2COCCOC2)C1 78706,Cc1ccc(F)c(C(=O)NC(C2(O)CCN(C(=O)CCC3(O)CCC3)C2)C)c1F 78707,C1(C)(C(=O)NC(C2CCOCC2)CC)CCN(C(c2cc(CO)[nH]n2)=O)CC1 78708,C12(NC(c3snnc3C3CC3)=O)CCCC1CN(C(=O)Cc1ccsn1)C2 78709,C1(C(N2CCC(CCNC(=O)Cc3ccc(O)cc3)CC2)=O)CCC2(CCC2)C1 78710,c1(C(N2CC(CC)N(C(C3CC4CC4C3)=O)CC2)=O)ccc2nccn2n1 78711,C1(NC(C(COC)OC)=O)CS(=O)(=O)C12CCN(C(c1ccoc1Cl)=O)CC2 78712,N1(C(c2cc(CSCC)on2)=O)CC2C(NC(C3CCCC(C(C)C)O3)=O)C2C1 78713,CCC(CC)(C(C)C)NC(C1CCC1NC(c1cc(CO)on1)=O)=O 78714,c1(C(C)NC(CONC(Cc2scc(C)c2)=O)=O)ccc(F)cc1 78715,N1(C(c2c(C)[nH]cc2)=O)CC2C3CCC(C2C1)N(C(C1CC(C)CO1)=O)C3 78716,C1(CC)CC(N=c2[nH]c3c(c(=NCC(F)C4CCCCC4)[nH]2)SCC3)C1 78717,c1(OC)cc(F)c(C(N2CC(O)C(O)C2CNC(=O)C(O)CSC)=O)cc1OC 78718,C1(C(=O)NC2CN(C(C(C)OCCOC)=O)C2)CC2(CCCCC2)S1(=O)=O 78719,c1(C(=O)NC(C)CCNC(C2(C)CCCOC2)=O)cc2c(nn1)CCCC2 78720,N1(C(=O)CN2CCCC2)CCC(O)C(N=c2ccnc(Br)[nH]2)C1 78721,c1(C(=O)NC(CC(C)NC(c2ccc(C3CC3)cc2)=O)C)nnc(O)cc1O 78722,c12ccc(cc1)-c1nc(c(C)s1)C(=O)N1CCCC21.N1(CC)CCC(Br)CC1 78723,c1(C(=O)OCC)cc([N+](=O)[O-])cc(CNC2CCCN(C(C)(C)C)C2)c1O 78724,C1(NC(COc2cccc(OCC)c2)=O)CCN(C(=O)CC2CC2)CC12CCC2 78725,c1(C(=O)NC2CC(C)N(C(=O)C#CC(C)(C)C)C2)cc2n(n1)CCCO2 78726,N#CC1(C(N2CC(NC(=O)C(N)=O)C(n3cccn3)C2)=O)CCSCC1 78727,Cc1onc(C2CCCCC2)c1C(=O)NCC1(NC(=O)CC(F)(F)F)CC1 78728,Cc1ccc(F)c(C(=O)NCC2(C)CC(NC(c3cnc4n3CCS4)=O)C2)c1F 78729,N1(C(C2(CC(C)C)CC2)=O)CC(C(=O)NCC2C3COCC23)C(C)(C)C1 78730,CC(C)(CC=CC(=O)NC1CCCC1n1cccn1)NC(=O)CC1CCSC1 78731,c1(C(=O)NCC2C3CCOCC23)cccc2cc(Cl)ccc12 78732,C1(CC)CNC(=O)CN1C(C1CC(NC(C2CCCCNC2=O)=O)C1)=O 78733,C1(N(C(c2nn(C)nc2Br)C(=O)NCC(F)F)C)CS(=O)(=O)C12CCOCC2 78734,C1(C(=O)NC2CCC(CNC(CCC3C(C)(C)C3)=O)C2)CCc2n[nH]cc2C1 78735,c1(C(N(CC(CC)NC(C2(CF)CC(F)(F)C2)=O)C)=O)cnc(S)n1C 78736,N#CC1(CNC(C2CCN2C(C2CC2(Cl)Cl)=O)=O)CCC1 78737,CCCC(O)C(=O)NCCCN(C(C1C2CC2C2CC12)=O)Cc1ccccc1 78738,N(C1CCCn2ncnc21)C(C(CCCN(C(=O)COCCCN=[N+]=[N-])C)O)=O 78739,c1(SCC(=O)NCC2CCCN2C(c2ncccc2Cl)=O)ccsc1[N+](=O)[O-] 78740,CC(CNC(C1(CCCF)CC1)=O)CC(=O)Nc1cccc(O)c1 78741,CN=c1[nH]c(=NCc2cncc(C)c2)[nH]c(=NC2CCN(c3cnccn3)C2)[nH]1 78742,Cc1cnc(C(=O)NCC2(CNC(=O)C(c3ccn(C)c3)C)CC2)cn1 78743,C(C(F)(F)C(=O)N1CC1)OC.c1(COCC(C)NC(=O)C2CC2)ccccc1.CO 78744,N1(C(c2ccccc2[N+](=O)[O-])=O)CC2CCN(C(C3CC3(Cl)Cl)=O)CC2C1 78745,C1(CNC(C=CSC)=O)CCC(C)(C)CN1C(c1sc(C)nc1C)=O 78746,C1(COC)CCCN1N(C)C(C)C1CCN(CC(F)(F)F)C1 78747,C1(NC(CS(=O)(=O)NCC)=O)(CNC(c2ccccc2)=O)Cc2ccccc2C1 78748,C12(C(N3CCC(OCCNC(CCCOCC=C)=O)C3)=O)CCCC1CC(=O)C2 78749,c1(CNC2C(C(=O)NCc3ccc(C)cc3C)C2)cc(F)c(F)cc1O 78750,c1(C(N2C(CNC(C(CC)C)=O)CC(C)(C)C2)=O)ccc(S(N)(=O)=O)cc1F 78751,c1(OC)ccc(CNC(=NCC2CCCOC2)NCC2CCOC2)c(OC)c1 78752,CC1CCNCC1NC(=O)C(=O)NC(c1cccc(F)c1)c1ccccn1 78753,N1(C(C(C=C)C)=O)CCC2(C=C(C(=O)N3CCOCC3C3CC3)C2)C1 78754,c1(C(C(N2CC(COC)(NC(c3nccnc3N)=O)C2)=O)O)ccc(F)c(Cl)c1 78755,C(CC(C)(C)CNC(=O)C(=O)NCc1ncc(C)o1)OC 78756,C(=O)(CC(C)C(C)(C)NC(C1CC(=O)OC1(C)C)=O)NC(CC)C(F)(F)F 78757,CC1CC2(CCCC2)CN1C(C1CCC(C2CC2)N1C(C1CCCN1C1CC1)=O)=O 78758,CC1CC(NC(=O)CCc2ccsc2Br)CCS1(=O)=O 78759,N1(C(C(C)(C)c2ccccn2)=O)CCN(C(=O)C(C)(C)C2CCOCC2)CC1 78760,C(CS(=O)(=O)c1ccc(COC(C2(C3CCCO3)CC2)=O)cc1)OC 78761,C(C(C)C(F)C(=O)NCC1CN2CCC1C2)NC(c1c(C)cnn1C)=O 78762,C(=O)(C(C)(C)NC(=O)C=Cc1ccco1)N(CCCCO)C 78763,c1(NC(C2(C)C(C)CN(C(C(CC=C)C)=O)C2)=O)ccccc1C(=C)C 78764,C(=O)(CCCCC(C)=O)N1C(C)CC(CC(N2CC(C(CC)C)C2)=O)C1 78765,N1(C(C=C(C)C2CC2)=O)CCCC(N=[N+]=[N-])C1.C12CC(C1)OCC(=O)N2 78766,c1(C(=O)NCC(CNC(=O)CCOC(C)C)OC)c(C)cc(Cl)cc1C 78767,C(CCC(=O)N1CC(CC2CCCC2)C1)N(C(C(C)=C(C)C)=O)C 78768,CC1CN(C(c2ocnc2C2CC2)=O)CC(C)C1NC(=O)Cn1ccnn1 78769,c1(NC)ccc(C(=O)NCC2CCCN2C(c2snnc2C2CC2)=O)nc1 78770,Cc1ncc(C(C)NC(c2cn(CCNC(=O)CC34CCCC3C4)cn2)=O)s1 78771,c1(C(=O)NC(c2cc(N)n(-c3ccccc3)n2)C)cc(OCC(F)F)ccn1 78772,CCC(C)C(=O)NCC(=O)N(CCC(C)NC(=O)Cc1cc(C)no1)C 78773,N1(C(c2c(CC)c[nH]c2)=O)CC(N=[N+]=[N-])CC1C(=O)N(C)CC1CCCCO1 78774,Cc1cc(C(=O)N(C2CCN(C(=O)C(C)CN(C)C)CC2)C)cc(N)c1Cl 78775,N1(CC(C)(C)NC(C(C)=C(C)C)=O)CCN(C(=O)C(C)(C)N(C)C)CC1 78776,N1(C(C2C(C(=C)C)OCC2)=O)CC(C(=O)NCCOCC(C)(C)C)CC(C)(C)C1 78777,c1(N(C)Cc2nnc(C)s2)nc(N2CCn3nncc3C2)c2c(n1)CSC2 78778,C1(NC(CC2N(C(c3c(OC)cnnc3)=O)CC(O)C2)=O)CCN(C)CC1C#N 78779,N1(C(CNC(CCC(C)C)=O)=O)CC2CCCC1(CNC(=O)Cc1cnoc1)C2 78780,C1(F)(C(N2CCOCC(CNC(c3cnccc3Cl)=O)C2)=O)CC12CCCCC2 78781,CC1(C)CC(NC(=O)C=Cc2cncs2)CN(C(=O)COC(F)(F)F)C1 78782,Cc1cnc(CC(=O)NCCOCCCNC(=O)CN2CCC2C)[nH]1 78783,Cc1cc(C(N2CCC(C)(CNC(c3nc(Cl)sc3Cl)=O)CC2)=O)c(Br)cc1F 78784,c1(C(=O)NC2CC3CN(C(CSC(C)C)=O)C(C2)C3)nc2cc(O)ccc2[nH]1 78785,C1(CCC)COCCN1C(=O)CC(C1CC1)NC(C1OC2CCC1C2)=O 78786,N1(C(C2C(C=C)OCCC2)=O)CC2OCCN(C(c3oc(CC)nc3C)=O)C2C1 78787,Cc1csc2cc(C(N3CCCC(NC(c4csc5nccn45)=O)C3)=O)[nH]c12 78788,CC1(C)CN(C(c2c[nH]c(C(F)(F)F)c2)=O)CCN(C(=O)C(C)(C)C#N)C1 78789,c1(CC2C(NCc3scc(N(N=CCC)C(C)C)c3)C2)ccc2c(c1)CC(C)O2 78790,C#Cc1cccc(C(N2CCN(C(c3c[nH]nc3CC)=O)CC2)=O)c1 78791,c1(C(=O)NC23CC(NC(C4C(C)(CC)C4)=O)(C2)C3)cnc2ncc(Cl)cn12 78792,C12CC(F)CN(C1)C2.N1(C(c2c(SC)cccc2)=O)CCC(CO)C(O)C1 78793,c1(C(N(CCCNC(c2c(OC)cco2)=O)C(C)C)=O)ncc(N)cc1C 78794,c1(OCC)cc(CNCCS(N)(=O)=O)ccc1OC(C1CC1N)=O 78795,C1(O)(CNC(C2(CCC)CC2)=O)CCCN(C(C23CCC(C)(C2)OC3)=O)C1 78796,C(=O)(CCCC(F)(F)F)N1CCNCC1.C(C(=O)NCC(F)F)SCC#C 78797,N1(C(CC2CCC(C)CO2)=O)CC(NC(c2nccc(C(F)F)n2)=O)CC(F)C1 78798,CCC(O)C(C)C(=O)N1CCC(CO)(NC(c2nn(C)cc2SC)=O)CC1 78799,c1(C(N(C(C)CNC(=O)Cn2[nH]cnc2=N)C)=O)ccnc(Cl)c1Cl 78800,c1(SC)cc(=NC(=O)C(C)C(C)NC(=O)C(C)OC(C)=O)[nH]n1C 78801,CC1(C)C2CCC(C(=O)NC3CCCC(NC(=O)C(C)(O)C4CC4)C3)C1C2 78802,C1(c2ncc(C(=O)OC)s2)CN(N2CCCC3(COCCO3)C2)C1 78803,Cc1ncc2n1CC(C(N1CCCC(C)(C)C1CO)=O)CC2 78804,C(=O)(CCCCC(F)(F)F)NCCCN(C)C(c1nccc2ncncc12)=O 78805,CC1CCCCC1(CNC(C1C2(CC2)C12CC2)=O)NC(=O)CN1CCSCC1 78806,C1(C(N(C)CC2CC(O)C(O)C2)=O)COCCN(C(c2n[nH]cc2[N+](=O)[O-])=O)C1 78807,c1(C(=O)NC23CCN(C(c4c(CC)non4)=O)CC2C3)ccc2nc(C)cn2c1 78808,CC1=CCC(C(=O)NCC(C)(C)NC(C2CCCN(C(=O)OC(C)C)C2)=O)CC1 78809,N1Cc2ccc(Cl)nc2C1.Cc1nccn1CCC(=O)N(CCO)CCN(C)C 78810,N1(C(C2C(=C)C2C(=O)OC)=O)CC2CN(C(c3cnn4ccsc34)=O)CC(C1)O2 78811,C1(C(N2CC(OCCNC(CCCO)=O)C2)=O)CC2(C1)CC2(F)F.CC 78812,c1(Cn2cc(C(C)N(C(=O)C(O)c3ccsc3)C)nn2)cccc(Cl)c1Cl 78813,C(=O)(C(CNC(=O)NCSC(C)(C)C)Cc1ccc(OC(F)(F)F)cc1)NC 78814,Cc1c(N)cc(C(N2CCC(C)(NC(=O)C(C)C(C)O)CC2)=O)cc1N 78815,Cc1cc(NC(c2ccccc2O)=O)sc1C(=O)NC1CONC1=O 78816,C1(CC)CN(C(=O)C(c2ccccc2)C)CCC1NC(C1(F)CC2(CCC2)C1)=O 78817,C(=O)(C(O)CCN(C)C)NC(C1CCCCC1)C(=O)NC(C)COC(F)(F)F 78818,C1(C(=O)O)CN(C(c2ccccc2OCF)=O)CCN1Cc1ccccc1 78819,C(c1ccc(Br)cc1)=CCC(=O)NCC(CNC(C(C)O)=O)CO 78820,N1(C(C(CCCC)O)=O)CC2CCCC2(CNC(c2ncc(F)c(OC)n2)=O)C1 78821,C1(NC(c2c(CC)n(C)nn2)=O)CCCCCC1NC(=O)CCCn1ccnn1 78822,N1(C(CCCC#C)=O)CCCC(C(=O)NC(c2ccccc2F)CC)CC1 78823,c1(C(C(C)OC(=O)C(CC(F)F)NC(=O)OC(C)(C)C)=O)c[nH]c2ccccc12 78824,C(C)(CCCNC(=O)NC1CC(N2CCN(C)CC2)C1)(OC)OC 78825,C1(CO)(CNC(c2cc(I)cs2)c2nnnn2C)CCCO1 78826,CC(C)C(N=[N+]=[N-])C(=O)NC1CC(C(=O)NC(C)(C)CO)C12CCC2 78827,C1(NC(C(C)(C)C#N)=O)CC2(C1)CN(C(=O)CC1(C(F)F)CC1)C2 78828,C1(C(N2C3CN(C(c4nnc(O)cc4O)=O)C(C3)C2)=O)CC2CCC(C1)S2(=O)=O 78829,Cc1ncc(NC(C2CCN2C(c2cc(Br)cnc2F)=O)=O)c(C)n1 78830,C1(O)(CN(C(c2ccc(COC)s2)=O)C)CCN(C(=O)C2=COCC2)CC1 78831,C1(C(N2CCC(CCCNC(c3cscn3)=O)CC2)=O)CC1C1CC(F)(F)C1 78832,C(=O)(C(F)C(C)CNC(=O)C(C)OCC=C)NCCSCC#C 78833,c1(C(C)C)ccc(C(N2CC(NC(=O)CC(C)c3cccnc3)C(O)C2)=O)nc1 78834,N1(C(c2c(C)snn2)=O)CC2ON=C(CNC(=O)CNC(c3ccco3)=O)C2C1 78835,c1(NC(c2n(CC(=C)C)nnn2)c2cnc(C(C)(C)C)[nH]2)cc(C)cnc1OC 78836,C1(C(=O)Nc2cnoc2)CCN(C(C2CC2c2ccccc2)=O)CC1O 78837,C1(C(=O)NC(c2nc(=O)o[nH]2)C)CC2(CCN1C(C1CC(=O)C1(C)C)=O)CC2 78838,Cc1nn(C)c(C(=O)NC(C)CCC2CCCC2)c1I 78839,C1(C(C)C)CN(C(=O)Cc2cn[nH]c2)CCN1C(c1cc(Cl)n(C)n1)=O 78840,c1(C2(C)NC(=O)N(CC(CCC)C)C2=O)c[nH]c2ncccc12 78841,c1(CN2C(C(=O)Nc3cnn(C(F)F)c3)CC3CC32)cc(Cl)c(Cl)c(Cl)c1 78842,N1(C(C(CC)C2CCOCC2)=O)CCN(C(C2(C)COC2)=O)C(C)C1 78843,c1(-c2ccc(CCCC)s2)n[nH]c2cccc(C(=O)Nc3cc(O)ncc3C)c12 78844,CCC1=NOC(C(=O)NC(C2CCCN2C(=O)C2CC2)(C)C)C1 78845,Cc1cc(C(=O)NC(C)CC(C)NC(c2ccc(N(C)C)cc2)=O)ncn1 78846,N1(C(C2CCC(F)(F)C2)C(=O)NCC(C)C)CCN(c2cnccn2)CC1C 78847,CC(C)CCC(C(=O)O)NC(=O)CCCCCCn1cc(CCC#N)nn1 78848,O=C(O)CC(C(=O)NC1CCC(c2nc[nH]n2)CC1)C1CC1 78849,C(=O)(CCCCN=[N+]=[N-])NC1(C(NOCCN(C)C2CC2)=O)CC=CC1 78850,O=C1CCC2(CCCN(C(c3cnn(C4CC4)c3Cl)=O)C2)CN1 78851,c1(SCC(=O)NCC(=C)CCNC(=O)CC2(OC)COC2)cccc(Cl)c1.C(C)=O 78852,C1(C(N2CC(CCCCNC(=O)CCc3ncc[nH]3)C2)=O)Cc2ccccc2O1 78853,CC1CN(C(C23CC(CC(F)F)(C2)C3)=O)C(C)CN1C(c1cc(Cl)c(Cl)[nH]1)=O 78854,C12CN(CCC1C)C(=O)C1C(Cl)(C1)N(CCC(F)(F)F)C(=O)C2.C(C)(=O)OC.CO 78855,C12(CC(=O)NCCC(C)N(C(=O)Cc3ccccc3F)C)CCC(CC1)C2 78856,C(C(N=[N+]=[N-])C(=O)NCC1CCCN(C(=O)CCN2CCN(C)CC2)C1)OCC 78857,c1(CN(C)CC2CCN(C(c3ccn(C4CC4)n3)=O)C2)cccc(F)c1 78858,Cc1cc(C)c(C(=O)NC2C=CCCC2)cc1O 78859,C1(OC)(OC)CC(C2CCN(c3nnc(-c4ncccc4F)n3C3CC3)C2)C1 78860,c1(C(N2CCCC2)=O)ccc(-c2nc(N(CCC)C)no2)cc1 78861,Cn1[nH]cnc1=NC(=O)NC1CN(c2ccc(C(F)(F)F)cc2Br)C1 78862,C1(CNC(CCCCC=CC)=O)CN(C(=O)C=C(Cl)Cl)CCC12CCC2 78863,N1(C(c2c(C)n(C3CC3)cc2)=O)CCC(C2CCN(C(=O)CSS(C)(=O)=O)C2)C1 78864,O=C(CC1CCCc2ccccc21)N1CCC2CN(CC3CC34CC4)CC2CC1 78865,C1(NC(c2c(CC)nc[nH]2)=O)CN(C(C2CC2(Cl)Cl)=O)CC1S(C)(=O)=O 78866,C12(C(N(CC(CC)O)CC)=O)COCC1CN(C(=O)CCc1ccncc1)C2 78867,C1(C(N2CC(NC(c3ccc(-c4ccco4)s3)=O)C2)=O)CC2CC1C1C2C1(F)F 78868,N1(C(COC)=O)CCN(C(C2CCCC2(F)F)=O)CC(C)(C)C1 78869,N1(C(C=CC(c2cn(C)nc2)=O)=O)CC(F)(c2nn[nH]n2)C2(CC2)C1 78870,c1(C(C)C)cccc(C(=O)N(CC(C)(C)NC(c2cc(C3(C)CC3)on2)=O)C)c1 78871,CC1CC(C)CN(C(=O)C(N2CCCC2c2ccccc2)=O)C1 78872,CN(C)NC(=O)CCC(=O)NC1CC2(C(=O)NC3CC3(C)C(F)F)COC1C2 78873,N1(C(c2[nH]cc(C)c2C)=O)CCN(C(=O)NC(c2ccccc2)=O)C2CC12 78874,N1(C(C(C2CC2)OC)C(=O)NC2CCOCC2)CCn2c(C(F)(F)F)nnc2C1 78875,C1(CNC(C2CCC(C)O2)=O)C2CN(C(=O)CCNC(N)=O)CC12 78876,C1(CNC(C(C)NC(C)=O)=O)CC2COCC2N1C(c1cncn1C(C)C)=O 78877,c1(C(=O)NC2CN(C(C(C)CN(C)C)=O)CC2C2CC2)cc2cc(F)ccc2[nH]1 78878,N1(C(C2(CC)CCC2)=O)CCC2(CCN(c3ccc(C#N)nc3)C2)C1 78879,c1(C(N(CC2N(C(COCCC)=O)CCC2)CC)=O)cc(S(=O)(=O)NC)cs1 78880,N1(C(C2(C(=O)OCC)C=CCC2)=O)CCN(C(=O)CN(c2ncccn2)C)CC1 78881,N1(C(c2c(C)cco2)=O)CC2CC2(CNC(c2sccc2-n2cccc2)=O)C1 78882,c1(NCCCOC(=N)O)nccc(N2CCCC(OC3CCOCC3)C2)n1 78883,C1(NC(=O)CC2CCSCC2)C2CC3CN(C(c4ccc(O)cn4)=O)C1C3C2 78884,n1(CC(=O)NCCC(C)NC(C2CC2(Cl)Cl)=O)c(O)nc2ccccc12 78885,CCCCC(F)C(=O)N1CCCC1C=CC(N1CCC(CN=[N+]=[N-])C1)=O 78886,C=C(Br)CC(C)(C)C(=O)NC1CN(C(c2cc[nH]c2C2CC2)=O)CCC1C 78887,CC1(CNC(c2cscn2)=O)CCN(C(C2(C)CCCNC2)=O)C1 78888,c1(CC)cc(CC(=O)N(CCC(=O)N(CC(C)OC)CC(C)C)C)on1 78889,C1(NC(C(CC=C)C)=O)(CNC(c2cc(C)nc(OC)n2)=O)CCCCC1C 78890,C(=O)(CC(C)CC(F)(F)F)NC1CCC(C)N(C(C2(O)CCCC(C)(C)C2)=O)C1 78891,C(CC(C)C(=O)NCCC(O)CNC(C1(CCN2CCCCC2)CC1)=O)=CC 78892,S(=O)(=O)(c1ccccc1F)C(N1C(C)CC(c2ccc(C)cc2)C1)=O 78893,C1(NC(C=CCC)=O)CC(OC)C12CCN(C(C1CCC=CCCC1)=O)CC2 78894,c1(C(=O)NCC(CNC(C2C(C#N)C2)=O)CO)ccc(OCC2CC2)nc1 78895,C1(NC(Cc2n(C)nnc2)=O)CCCCCC1NC(C1CCCCS1)=O 78896,c1(OCC)ccc(Br)cc1CN1CCC(NC(c2cc(CC)[nH]n2)=O)C(O)C1 78897,N1(C(C2(CNC(C3C(CC(C)(C)C)C3)=O)CC=CC2)=O)CC2(CCCC2)C1 78898,C1(NC(C(CCSC)OC)=O)CN(C(=O)C2CC2)CC2(CC2)C1 78899,C12(NC(C(C)CC(N)=O)=O)CCC(CNC(c3cccnc3O)=O)(CC1)OC2 78900,c1(C(=O)NCCCCCNC(C2C(C=C)C2)=O)cc(=NS(C)(=O)=O)cc[nH]1 78901,c1(CC)c[nH]nc1C(=O)NC(Cn1cccn1)C(=O)NC(CO)C1(O)CC1 78902,Cc1ncccc1C(N1CC(NC(=O)COC2CCN(C)CC2)C(C(F)F)C1)=O 78903,c1(C(=O)NC2(CC=C)CN(C(c3ccccc3CC)=O)C2)nc(=O)n(C)[nH]1 78904,C(CCC(C)C(=O)NC(C)C(C)(C)C(=O)NCc1cc(C)sc1C)OC 78905,c1(OCC)ncc(C(=O)NCC2CCN(C(C3CC(O)CN3C)=O)C2)cc1Cl 78906,N1(C(CCN(CCC)C)=O)CC2CC(NC(=O)C=Cc3ccncn3)CC1C2 78907,C1(CSCC(=O)NC(=O)Nc2c(C)csc2)CCCC2(CC2)C1 78908,N1(C(Cn2ncc(C)c2)=O)CC2CCC(NC(=O)CCS(C)=O)CC1C2 78909,c1(C(=O)OC)ccc2[nH]c(=NCC3CCN(C(=O)CNC(N)=O)C3)sc2c1 78910,C1(CC)(CC)CC(NC(=O)Cc2nocc2C)CN1C(c1ncn2c1CCC2)=O 78911,c1(OC)cncc(C(=O)NCC2CC2NC(C2CC(n3cnnc3)C2)=O)c1 78912,n1(CC(=O)NCC2N(C(C(CO)N(C)C)=O)CCC2)nnc2ccccc12 78913,CC1CNc2ccc(C(=O)N(C(C)CCNC(=O)C=CC(C)(C)C)C)cc21 78914,CC(=O)CCCC(C)C(=O)NC1(C(N2CCCC2CC(C)O)=O)CC(O)C1 78915,c1(C(N2C(C)C(NC(c3n[nH]c4c3COC4)=O)CC2)=O)cccc(F)c1F 78916,N1(C(CSc2n(C)cnn2)=O)CC(NC(=O)CCSC2CCC2)CC1CO 78917,c1(C(=O)NC(C2CCN(C(=O)C(C)OCCN(C)C)C2)C)cccnn1 78918,C1(C(C(=O)NCC(C)N(C)C)(C)C)CCCN(C(=O)CC(=O)NC2CC2)C1 78919,C1(CNC(c2cn(C)nc2)=O)CCC2(CO1)CC(NC(=O)C=Cc1ccco1)C2 78920,CC1CCc2nc(N3CCC(CO)C3)[nH]c(=NCc3ccc(S(N)(=O)=O)s3)c2C1 78921,N1(C(C2COCCN2C(=O)C(F)F)=O)Cc2cccc(O)c2C1 78922,C=CCC(CNC(=O)C(CC)CC=CC)C(=O)NCc1scnc1C 78923,C1(NC(CCC(C)NC(=O)CN2CCC(F)CC2)=O)CCC(O)C(O)C1 78924,C1(C(=O)NC(C(=O)OC)Cc2cn(C(C)C)nn2)CCn2cncc2C1 78925,Cc1cnccc1C(C)C(=O)NC1CCCCC1NC(c1ncn(C)c1C)=O 78926,C1(NC(CS(CC)(=O)=O)=O)CN(C(=O)Cc2conc2C)Cc2ccnn2C1 78927,c1(OC)ccc2c(N3CCCN(C(c4cc(C)ccc4Cl)=O)CC3)ncnc2c1 78928,CC1(C(=O)NC2CC2NC(C2(CC3CC3)CCOCC2)=O)CCCCO1 78929,c1(CC(N2C(C)(CNC(=O)C3=NOCC3)CCC2)=O)cc(F)cc(F)c1 78930,CC1(C)Oc2ccsc2C(N=c2ccnc(N3Cc4ccc(OC)cc4C3)[nH]2)C1 78931,c1(C(=O)NC2C3CN(C(C(CCOC)C)=O)C2C3)c(Br)c(C2CC2)nn1C 78932,c1(CC)c(C(=O)N(C2CCCN(C(=O)CC(C)(C)OC)C2)CCF)cccc1F 78933,C(=O)(C#CC1CCC1)NC1CC(C)N(C(c2nc(=O)n(C)[nH]2)=O)C1 78934,N1(CCOCC)CCN(C(=O)C(C)(F)NC(=O)OC(C)(C)C)CC1 78935,C1(CCCNC(C2CC(OC)C2)=O)CCN(C(=O)Cc2nnc(C)o2)CC1 78936,Cc1cnc(C(=O)NCC2(F)CC(NC(C3CC3C(F)F)=O)C2)nc1 78937,C(=O)(CC(C)(C)CN(C)C)NCCCC(=O)NC1(COC)CCOC1 78938,Cc1ccc(CNC(C2CCC(NC(c3ccccc3O)=O)C2)=O)c(C)c1 78939,N1(C(C)=O)CC2(CC2)CC1C(=O)Nc1ccc(SCCCO)cc1 78940,C1(N(C(c2c(CC)c[nH]n2)=O)C)CCN(C(c2cn(C)nn2)=O)CC12CC2 78941,CS(=O)(=O)c1ccc(F)c(C(N2CCCN(C(=O)C3=CCCC3)C(CO)C2)=O)c1 78942,C1(C)(C(=O)NCCC(CNC(C(CC)(C)CC)=O)(C)C)CCCNS1(=O)=O 78943,c1(C(=O)NCCN(C(c2ccnc(O)c2)=O)CC2CC2)c(F)ccc2[nH]ccc12 78944,CN1CCOC(C(=O)NCC2CN(C(=O)CCc3ncc[nH]3)CC2(F)F)C1=O 78945,c1(CC(=O)NC2CN(C(=O)CC3CCCCC3O)C2)ccc(O)cc1Cl 78946,C1(C)(CNC(CSCCC)=O)CCCN(C(C2C3C4CCC(C4)C23)=O)C1 78947,c1(NC(c2c(NCc3c(C)c(Cl)ccc3)cnc(Cl)c2)=O)c(Br)ccc(F)c1F 78948,CC1(CNC(=O)CC(C)(C)NC(C2(C)CCC(=O)NC2)=O)CC2(CCC2)C1 78949,c1(COC)ncc(C(=O)NC2CN(C(=O)CNC=O)CC2OC)c(O)n1 78950,N1(C(c2ncn(C)n2)=O)CCCC(NC(=O)Cn2cnc([N+](=O)[O-])n2)C(F)C1 78951,C(CCC)(C(=O)N1CC(O)(C(C)NC(=O)COCc2nc(C)no2)C1)=CCC 78952,Nc1cc(Cl)ncc1C(=O)NC1CC2CCC1(CNC(=O)Cn1ncnn1)C2 78953,C1(CN(C)C(c2nncs2)=O)COCCN1C(c1c[nH]nc1C1CCOC1)=O 78954,CC(CS(C)(=O)=O)C(=O)NC1CC(CNC(c2ccc(-c3cc[nH]n3)s2)=O)C1 78955,Cc1[nH]nc2c1C(NC(=O)N(C)C(c1ccco1)C1CCCO1)CCC2 78956,c1(C(N2CC(C)(NC(C(C)OC3CCCC3)=O)C2)=O)ccnc(CC(F)(F)F)n1 78957,O=C(C1=CS(=O)CCC1)NC1CC2CC1N(C(c1cncc3[nH]ccc13)=O)C2 78958,N1(C(c2ccc(C)o2)=O)CCc2nc(C(=O)N)cn2CC1.N1(CC)CCCCC1=O 78959,CC1(O)CCN(C(C2CCCCC2NC(C2CCCC(C#N)C2)=O)=O)CC1O 78960,C1(C(=O)NCC(CC)C#N)CC2CCCC2N1C(=O)C=CCN1CCC1 78961,C1(C#N)(C(N2CCC(C3N(C(c4c(C)n[nH]c4)=O)CCC3)C2)=O)CC2C=CC1C2 78962,c1(OC)cc(N)c(Cl)cc1C(=O)NC(CCN(C)C(c1ccon1)=O)C(C)C 78963,N1(C(C(COC)C)=O)CCC(O)CC1C(=O)NC1C2C=CC(C2)C1CO 78964,c1(C(=O)NC(C(=O)N(CCOCCOC)C)CO)ccc(=O)n(C)c1 78965,C(=O)(C1=CCCCCC1)NC(C(=O)NCC(C)O)CN(C)C 78966,C1(C)(C(N2C(CNC(c3ccc(CC)[nH]3)=O)CC2)=O)CCCCCC1 78967,C(c1ccc(C2CC2C)o1)=CC(=O)NC1CCC(CNC(C(CC)OCC)=O)C1 78968,Cc1cc(C(N2CCC(O)(CNC(c3coc(C(C)C)n3)=O)CC2)=O)cc(O)c1 78969,c1(C(=O)NC2C=CC(CC(=O)NCCCN(C)C)C2)cc(O)cc(F)c1 78970,C1(C=C)(NC(CCN(C(=O)CCN2CCOC2=O)CC=C)=O)CCCCC1 78971,N1(C(C(N(C(Cc2nc(C)sc2)=O)C)C2CC2)=O)CC(CO)C1(C)C 78972,C1(NC(C2C(C)(CO)C2)=O)C=CCC(C(=O)NCc2ncoc2C2CCC2)C1 78973,N1(C(C2(C)CCCCO2)=O)CCOCC(NC(c2c[nH]nc2-c2cccs2)=O)C1 78974,n1(C(C)C)ncc2c(NCCCCC#N)[nH]c(=NCC(C)=C3CC3)nc12 78975,C#CC1(C(N2CCC(N(C)CC)C2)=O)CCN(C(C2CN(C3CCC3)C2)=O)C1 78976,Cc1onc(Br)c1C(N1CCC(C(C)NC(c2cccnc2O)=O)C1)=O 78977,CC(C)C(F)(CNC(C1(C)CCCC1O)=O)C(=O)NC12CC1COC2(C)C 78978,c1(OC)ccc(C(=O)N(C2CN(C(c3c(C)cccc3Cl)=O)CC2F)C)c(F)n1 78979,C(CC(O)CC(=O)NC1CC(NC(=O)CC(C)O)C1)SC 78980,c1(N(CC(CC)(C)OC)C)ncnc(NCc2cc(Cl)cc(Cl)n2)c1C 78981,C1(NC(C2C3CN(C(c4cn(CC)nc4C)=O)CC32)=O)CC2(CCC2)C1OC 78982,CC(C)C(CCNC(=O)CCC1CCCCO1)NC(C1(C)CCCO1)=O 78983,CCCN=C(NCc1cc(C)cc(Cl)c1)N1CCN(c2ccccc2F)C(=O)C1 78984,CC(C)(C(=O)NCC(C)(C)NC(=O)CC(F)F)C1CCCCC1 78985,c1(C(N(CCCNC(C(C)OC)=O)C)=O)ccc(N(C)C)c([N+](=O)[O-])c1 78986,c1(OC)cccc(C(N2CCC2(C)C(=O)NCC2CCN(C)CC2)=O)c1O 78987,n1(-c2ccc(C(=O)OC3CC(OCC)C3(C)C)cc2)nc(C)ccc1=O 78988,C(=O)(C1=CCCCC1)NCC(CNC(=O)CC1CC12CC2)O 78989,C1(CNC(C(C)OC)=O)CN(C(c2cncc(C(=O)N(C)C)c2)=O)CC(C)(C)O1 78990,N1(C(C(C(CC)O)C)=O)CC2CCC(C1)N2C(=O)CN(C)S(N)(=O)=O.C(COC)S 78991,C1(C(=O)NC(C)Cc2ccco2)CN(C(=O)C(F)CC(C)(C)C)CC1C1CC1 78992,CC(CC1CC1)C(C(=O)NC1CCC1)N1CCC(C)(Cc2ccccc2)CC1 78993,CCC(C)(O)C(=O)NN1CCCC1C(=O)N(CCC1CCCC1C(=O)O)CC 78994,N1(C(c2cc(OC)no2)=O)CC(NC(c2ccc(CCC#N)cc2)=O)C(C)(C)C1 78995,C(=O)(CC(C)n1cccn1)NCC(C)N(C(COCCSC)=O)C 78996,c1(C(=O)NCCCCCN(C(C2C(C(C)C)C2)=O)C)cc2cccc(Cl)c2s1 78997,c1(CC(N2C(CNC(CC(C)(C)O)=O)CCCC2)=O)c(Cl)cccc1Cl 78998,CC(CNC(C12CC1CCN2C(C1CC1C(F)(F)F)=O)=O)C(F)(F)F 78999,N1(C(c2c(C)onc2)=O)CCC2(CCC2)C(NC(C2CC3CC2C3)=O)C1 79000,C1(NC(=O)CSc2nncs2)CC2CC1N(C(c1ccc(O)nc1Cl)=O)C2 79001,CC1(C)CCCN(C(c2ccc(C#N)o2)=O)C1CNC(=O)Cc1cncnc1O 79002,c1(C(=O)NCCN(C)C(c2ccc(C(F)(F)F)c(F)c2)=O)cc2cn[nH]c2cn1 79003,C(CC(F)F)(C(=O)NC1CCCC1C(N)=O)NC(C(CC=C)NC(C)=O)=O 79004,C1(C#N)(C(N2CC(CNC(c3ccc(COC)cc3)=O)C2)=O)C(C#N)C1(C)C 79005,C(C(CNC(C1(CO)CCCO1)=O)C(F)(F)F)NC(C=C1CCN(C)CC1)=O 79006,c1(C(N(C2CCN(C(c3sc(C)nc3C)=O)C2)CC)=O)cccc(C(C)(F)F)c1 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79060,c1(N2CCC(CC)(NC(c3cc4c(s3)CCC4)=O)CC2)nccc(S(C)(=O)=O)n1 79061,n1(CCC(=O)N(CC(C)NC(CC(=O)OCC)=O)C)c(C)csc1=O 79062,CON=Cc1ccc(-c2ccc(OC(F)(F)F)cc2)cc1 79063,N1(C(C=CC(C)NC(C(CC(C)C)C(C)C)=O)=O)CCc2ccc(C#N)cc21 79064,N1(C(C(=O)NCCCC)c2csnn2)CCCC(c2nn(C)cc2C(N)=O)C1 79065,C1(C2(C(N(CCOC(C)=O)C)=O)CC2)CCCN1C(=O)CCn1ccnc1 79066,C(C(CC)CCCCCC)c1n(CCCCCCCC)nc(CO)n1 79067,c1(C(=O)NC(C(C)NC(=O)CC(O)CN(C)C)(C)C)ccc(N)c(Cl)n1 79068,C1(NC(CNC(C(CC)CC)=O)=O)CN(C(C2CCC2OC)=O)CC12CCC2 79069,N1(C(C23CN(C(c4ccc(O)nc4)=O)C(C2)CO3)=O)CCN2C(=O)NCC2C1 79070,c1(NC(c2cncc(-c3cncc(C#CC)c3)n2)=O)nc2ccc(C)cc2[nH]1 79071,C1(N)CCCCC1OC.C(C(C)(C)CN(C(=O)COC)C)NC(C=CC)=O 79072,N1(C(CN2C(=O)CNC2=O)=O)C2CCC1CC(NC(C1(F)CCOC1)=O)C2 79073,C(C)(CC(=O)NC12CC(NC(=O)C(C)CC3CC3)(C1)C2)SC 79074,C(=O)(CCCCCCN=[N+]=[N-])N(C1CCN(C(C2CC2C2CC2)=O)C1)CC 79075,CC1CN(C(c2c[nH]nc2-c2cccc(F)c2)=O)CCN1C(=O)C(C)(C)C#N 79076,Cc1nc(O)c(C(=O)NCC(N2CCCCC2)c2cccs2)c(C)c1[N+](=O)[O-] 79077,C(=O)(C(O)C(F)(F)F)N(CCOCCCN(C(=O)CCc1ccccc1Cl)C)C 79078,C(CCC)(C(=O)NCc1ncc(C)s1)NC(C(C=C)C)=O 79079,N1(C(C(C2CCOCC2)C)=O)CC=C(C(=O)Nc2c(O)cccc2Cl)CC1 79080,CC(C)(C)C(C(=O)NCC1(NC(=O)Cc2ccoc2)CCCC1)C(O)C(F)(F)F 79081,N1(CCCNC)CC(NC(=O)COC)CCC1C 79082,c1(N2CCC(C)C(CO)C2)ncnc2cc(F)c(F)cc12 79083,C1(C)(C(N2CC(COC)(CNC(C3(F)CC3C)=O)C2)=O)CC2CC2C1 79084,N1(CCC)CCCC(C(N2CCCC2C(C)NC(=O)CC(C)(F)F)=O)C1 79085,CCC(CN=c1nc2c(cnn2C)c(N(C)Cc2cccc(OC)c2Cl)[nH]1)OC 79086,C(=O)(CC(C(N)=O)SC)NC(C1CCCC1)CNC(CCCOCC=CC)=O 79087,c1(C(=O)NCC(O)CNC(C2COCCC2(F)F)=O)ccc2ccnn2c1 79088,N1(C(C2C(C=C)CC2)=O)CCC2CN(C(c3cccc4cc[nH]c34)=O)CC2C1 79089,N1(C(C(CC=C)CC)=O)CC(C2CN(C(=O)Cc3ccc(O)nc3)C2)C1 79090,Cc1cc(C(=O)NC(C2CCOC2)CNC(C23CC4CC2C3C4O)=O)cc(N)c1 79091,c1(CN2CCN(C(c3c(C)nsc3)=O)C(C)C2)ccccc1[N+](=O)[O-] 79092,c1(CC)ccc(NC(C2CCCN2C(C2CCCN2C2CC2)=O)=O)cn1 79093,CC(C)C(CNC(C1CCN1C)=O)C(=O)N1CCC1c1ccccc1 79094,O=S(=O)(c1cccc(O)n1)N1CCN(c2ccc(F)nc2)CC1 79095,Cc1ocnc1CC(N1CC(C(C)NC(=O)C=CC2CCCO2)C1)=O 79096,C1(NC(CCCCOC)=O)CC2CCC1N(C(=O)CNC(c1nc(C)no1)=O)C2 79097,CCC(CC(=O)NCC1(C)CCC(NC(c2ccc(CO)o2)=O)C1)CC(F)(F)F 79098,c1(C(=O)NC2C(C)CCN(C(=O)C=CBr)C2)nccc2ncccc12 79099,N1(C(CC)=O)CCC(NC(=O)CCCc2cc(C)no2)C(O)C1 79100,C(=O)(C1SCCc2sccc21)NCC1(C)CCCN1C(=O)CCn1cncn1 79101,c1(OC(C(=O)NC2(C)CCN(C(c3c(CC)nns3)=O)C2)F)ccc(Cl)c(F)c1 79102,C(=O)(CCCCCC(C)O)NC1C2CN(C(c3nn(CC)c(C4CC4)c3)=O)C1C2 79103,c1(C(=O)NCC(CC)NC(=O)Cc2cccc(C)c2Cl)ccc2c(c1)nnn2C 79104,Cc1occc1S(C)(=O)=NC(=O)C1(C)CS(=O)(=O)C1 79105,c1(C(CNC2CCC(COC)C2)O)c(F)cccc1Cl 79106,C(=O)(CC1=CCCCC1)N1CC2(CN(C(C(CC)OC3CCCCC3)=O)C2)C1 79107,N1(C(C(C)SC(C)C)=O)CCOCC(C(=O)N(C)CCc2cccc(Cl)c2)C1 79108,c1(CCC)cc(C(=O)NC2CC(CNC(C3CC34CCC4)=O)CC2O)nn1C 79109,c1(C(=O)NCC2(CN(C(C(CC)SC)=O)C)CC2)cnn(CCO)c1C 79110,Cc1ncc([N+](=O)[O-])n1CC(=O)NCCCCC(CO)NC(c1n[nH]cc1Cl)=O 79111,c1(OCC)cccc2c1CNC2=O 79112,Cc1ccc(S(=O)(=O)NC2CCOCC2CSc2ccccc2)cc1[N+](=O)[O-] 79113,N1(C(C2CCC(C)(F)CC2)=O)CCN(C(=O)C=CCO)CC2CCCCC12 79114,C12CCN(CCC1(F)F)CC2.Cc1ccc(C(=O)N(C)C)c(F)c1F 79115,C1(NC(C(C2CN(C(=O)CN(CC(C)(C)C)C)C2)OC)=O)CCC2CCC1C2 79116,N1(C(c2c(OC(C)C)cncc2)=O)CC2CC(NC(=O)C(F)=CCCF)CC1C2 79117,CC(C)CCCC(=O)N1CC2(CNC(=O)C(O)Cn3cncn3)CC1CO2 79118,N1(C(C2C(CC(C)(C)C)C2)=O)CC=CCC1C(=O)NCC1=CCCC1 79119,c1(C(N2CC(CC)C(NC(=O)C(c3ccccc3)O)C2)=O)cc(C)cc(O)c1 79120,N1(C(C2C(=C)C2)=O)CCC2(COC(CNC(c3sc4cncn4c3C)=O)C2)C1 79121,c1(NCCNC(c2ccsc2)=O)ccc(S(=O)(=O)NC2CCSC(C)C2)c(Br)c1 79122,C1(C(=O)NC2CCN(C(CSCCC(C)C)=O)C2C)CCC2CC1CO2 79123,N1(C(CCCC)=O)CCN(C(C2C(C)C2C)=O)CC1c1cc(F)cc(F)c1 79124,C1(C(=O)NCC(C(C)(C)C)(C)O)CC2(CCN(C(C3(C)CNC(=O)C3)=O)C2)C1 79125,Cc1oc(CNC(C2CCCC(F)C2)=O)nc1C(=O)N(C1CSC1)C 79126,c1(C(=O)NCC2CC(NC(C3C(C)(CC)C3)=O)C2)cnc(C)n1C(F)F 79127,C1(C(=O)NCC(C)OCC#C)(CO)CCN(C(c2cccn2CCC)=O)C1 79128,C1(NC(C(C)OCC)=O)CN(C)CC12CC2.C1=CCNC1=O 79129,c1(SCC)cccc(C(=O)N(C)CC2CCN(C(C3NC(=O)OC3C)=O)CC2)c1 79130,N1(C(CCC(=O)NC)=O)CCn2nc(CNC(=O)CC(O)C3CCCC3)cc2C1 79131,c1(C(=O)NCCNC(C(C=C=C)C)=O)cc(Br)ccc1N1CCCC1 79132,c1(-c2scc(CC(=O)N(c3ccc(Cl)cn3)C)n2)ccccc1Cl 79133,N1(C(CCn2c(C)ncc2)=O)CCCCCCC1C(=O)N(C)CC1CCOC1C 79134,N1(C(c2c(CC)c[nH]n2)=O)CCC(C)(CNC(C2(CC)CCCCO2)=O)CC1 79135,c1(C(=O)NCC2C=CC(NC(C3(C#N)CC3)=O)C2)cnc(CC(F)(F)F)c(Cl)c1 79136,C1(NC(C(C2CCC2)NC(C=C(C)C)=O)=O)CC(F)(F)C1(C)C 79137,C1(C(N(CC(O)CNC(c2cscc2Cl)=O)C)=O)Cc2nccnc2C1 79138,C1(N(C(N(CC(N2C(CC)CC2)=O)C)=O)C2CC2)CCCCC(=O)C1 79139,c1(C(=O)OC)ccc(C(=O)NCCN(C(c2cnns2)=O)C(C)C)cc1Cl 79140,N1(C(c2[nH]cc(C)c2)=O)CCN(C(c2ccnc(C(C)C)n2)=O)C2CCCCC12 79141,C(=O)(CC(C(F)(F)F)NC(=O)C(F)=CC1CC1)NC(CC)COC 79142,C12(CC(N3C(CCNC(CCC)=O)CCC3)=O)COC(C)(C1)C2 79143,C(C1=CCN(C(=O)Cc2ccc(O)cn2)CC1)NC(c1c(C(C)C)n(C)nc1)=O 79144,CC1CCCN(C(=O)CCCCCN(C)C)C1CNC(=O)CCC1CCC1 79145,n1(CC(CC)O)cc(C(=O)NCC#CCNC(=O)C(C2CCCC2)OC)nn1 79146,c1(C(=O)NCCCCNC(C2C3CCC2(c2cncs2)C3)=O)cccc(Cl)c1F 79147,CC(C)CCCCCC(=O)N(CC(O)CNC(=O)C=CC1CCOC1)C 79148,CCC(C)(C)C(O)C(=O)NCC1(O)CCCN(C(=O)CN2CCCNC2=O)CC1 79149,C=CCCC(CC(C)C)C(=O)N(CCCCCNC(C1CC12CC(C)(C)C2)=O)C 79150,N1(C(COCCCC#C)=O)CCC2(CCCCN(C(=O)C#CC(=O)N(C)C)C2)C1 79151,CC1CCN(C(=O)COC2CC=CC2)CC1N(C)C(C1CCOCC1(C)C)=O 79152,C1(CC)(NC(c2ccc(C#N)s2)=O)CCN(C(=O)CCC2CCC(C)O2)CC1 79153,C(c1ccccn1)=C(C)C(=O)NC(C1CCCC1)CNC(C1(C#N)CC=CC1)=O 79154,C(CO)(CCCCNC(=O)C(F)CC1CCCC1)NC(C(c1ccccc1)C)=O 79155,C(c1cccnc1)=C(C)C(N1CCC(=CCNC(=O)CC2(C)CC2(F)F)CC1)=O 79156,CC1COC(CO)CN1C(=O)CCN(C(=O)CCc1cccs1)CCO 79157,C1(C)(NC(CN2C(C)CCCC2)=O)CCCN(C(=O)CC2CC3CC3C2)C1 79158,Cc1ccc(N2CCC(C(=O)NCC(F)Cc3ccccc3)C2=O)cc1 79159,c1(CCC)coc(=NCC2(S(=O)(=O)N(C)C)CC2)[nH]1 79160,C1(NC(c2ccn(C(C)C)c2C)=O)CN(C(c2cn(CC)nn2)=O)C(C)(CC)C1 79161,c1(C(N(CC(C)C(=O)N(C2CCOC2)C2CC2)C)=O)cnn(C)c1Cl 79162,c1(C(=O)NC2(C(F)F)CC2)cnn(-c2ccccc2)c1I 79163,n1(CC(=O)NC(C2CCCN(C(c3cncnc3)=O)C2)C)cc(Br)c(=N)[nH]1 79164,c1(CC(N2CC(C(Cn3cc(C(C)OCC)nn3)F)C2)=O)ccc(O)cc1 79165,c1(NC(C(=O)NCC(C)O)=O)ccc(-c2ncn(C(C)C)n2)cc1 79166,Cc1nc[nH]c1CC(=O)NC1(CNC(c2ccn(CCC(F)(F)F)n2)=O)CCCC1 79167,c1(CC(N2CC(NC(C(C(CC)O)C)=O)C2)=O)ccc2cccnc2c1 79168,c1(C(N(C)CC2(CNC(C(C)OCCCC)=O)CC2)=O)nnn2c1CCCC2 79169,C#Cc1ccc(C(=O)N(CCNC(c2cnn(C)c2N)=O)CC)c(C)c1 79170,C1(C(=O)NCC2(CNC(c3c(C)cncc3)=O)CCCC2)CC2(C1)CC(C)(C)C2 79171,N1(C(c2scc(C)c2)=O)CC2(CCC2)CC1CNC(C1COCCN1C)=O 79172,C(=O)(CCCCCC#N)NCC(C)NC(c1cccc(CCCN)c1)=O 79173,N1(C(c2c(SC)nn(C)c2)=O)CC2CC3CC2C1C3NC(c1ncoc1C)=O 79174,N1(C(CC=C=C)=O)CCC2CN(C(=O)CCSc3ccc(Cl)cc3)CCC2C1 79175,c1(C(=O)NC(CCOC)C(=O)NCCCC(=O)NC)ccc(Cl)c(F)c1 79176,C(CC(=O)NC(c1ccc(C)nc1)C)(C(F)(F)F)NC(C=CCC)=O 79177,CC(C)(CNC(=O)C(F)CC1CN(C(=O)CC(C2CC2)C2CC2)C1)C(F)(F)F 79178,CC(CCC(=O)NCCC1(NC(=O)CSCc2ncc[nH]2)CCC1)N(C)C 79179,C(N=c1[nH]c(=NCc2ccc(Cl)cc2C)[nH]c2c1CCC2)C1C(CC)CCCC1 79180,N1(C(C)CNC(c2cccc(Cl)c2-n2cccn2)=O)C(=O)c2ccccc2C1=O 79181,C1(N(C(CCOCC#C)=O)C)CCCCN(C(=O)CCC2CCCCO2)C1 79182,N1(CCN(C(N(C(c2ccco2)C)C)=O)CCN)CC2CCCCC2C1 79183,C12(NC(Cc3c(Cl)cn(C)n3)=O)CCCC1N(C(c1cc(F)cnc1O)=O)CC2 79184,C1(NC(CCOCCOC)=O)(CF)CCN(C(=O)CN2CCOC2=O)C1 79185,N1(C(c2c(OC)csc2)=O)CC2=C(C1)CN(C(C1(C(F)(F)F)CC3CC3C1)=O)C2 79186,CCCC(C)CC(=O)NCc1cc(C2CCN(C(c3ccno3)=O)CC2)no1 79187,c1(C(N2CCN(C(C3CCS3(=O)=O)=O)C3C2C3)=O)cc2nc(=O)ccn2[nH]1 79188,N1(C(C2CN(CCC)C(=O)C2)=O)C2CCCC1CC(NC(c1cscc1C)=O)C2 79189,Cn1c(C(=O)NC2CCCC(CNC(C3CC4(CC4)C3)=O)C2)cnc1S 79190,c1(C(C)=O)ccc(C(N2CC(NC(=O)C(C)NS(=O)(=O)CC)CC2C)=O)cc1C 79191,C(C(F)(F)C(=O)NCC1(C)CCCC1NC(=O)CC1COCCN1C)N(C)C 79192,C1(NC(c2cc(COC)on2)=O)CN(C(C2CCOC2C)=O)CCC12CCC2 79193,c12cn3cccc(c3n1)[nH]c2=O.N1(CC)CCC(C)C(CO)C1 79194,c1(C(=O)NCC2(NC(C(CC)SC)=O)CCC2)cc(NC)nc(Cl)c1 79195,C1(C)(CNC(C=C(C)C(C)(C)C)=O)CCN(C(=O)CCc2ccc(C)s2)C1 79196,c1(C(=O)NC(C2CCOC2)CNC(c2c(CC)ncs2)=O)c(C)nnn1CC 79197,N1(C(C(COC)OC)=O)CCC2(NC(=O)CCc3ccccc3OC)CC2C1 79198,CC(C)(CC(=O)NCC(CO)NC(=O)C(c1c(F)cccc1F)(F)F)C(F)F 79199,CC(C)(O)CC(=O)N(CCC(=O)NC1CCCC(O)C1)CC1CC1 79200,N1(C(CCCN(C(CC(=O)OCC)=O)C)=O)CC(C#N)C2(CCC2)C1 79201,C1(NC(C(c2cccc(F)c2)C)=O)CC(NC(c2cc(C(N)=O)c[nH]2)=O)C(O)C1 79202,C1(NC(C2C(CNC(CC3(N(C)C)CCC3)=O)CCC2)=O)COCC1N=[N+]=[N-] 79203,N1(C(CCC(C)SC)=O)CCCC(NC(=O)C=Cc2cnn(C)c2)CC1 79204,C1(CC)(CC)CC(NC(C2CCCC2CNC(=O)CC(=O)OC)=O)C1 79205,c1(C(N2CC(c3cccc(OC)c3)(F)C2)=O)cccc2c1NC(C)CC(=O)N2 79206,c1(C(=O)NC2C(CNC(C3=C(N)C(O)=CCC3)=O)CC2)ccc2ncnn2c1 79207,C1(NC(C=CC(C)C)=O)CN(C(C2CC2C2CC2)=O)CC1c1cccc(F)c1 79208,Cn1cc(S(=O)(=O)Nc2ccc(N3CC(O)C3)cc2)c2cccc(Br)c12 79209,c1(C(=O)NC(CC)CNC(=O)COCCC(C)C)ccc(O)nc1Cl 79210,C(CN(C(=O)CC(C)Cc1cccc(F)c1)CC)(C(C)(C)C)NC(CSCC=C)=O 79211,N1(C(c2n[nH]c(=N)[nH]2)=O)CC2CC(NC(=O)CCc3cccs3)CC2C1 79212,N1(C(Cc2c(C)n(C)nc2)=O)CC(NC(=O)C=CC(C)C)CC(F)C1 79213,CON1CCC(C(=O)NCC2CCCC2C(=O)N(CC(=O)N(C)C)C)CC1 79214,CC1CC(=O)CCC1C(=O)NC(C(=O)NCCC(=O)N(C)C1CC1)C1CCC1 79215,N1(C(=O)CCCCCl)CC2(C1)CN(Cc1c(Cl)ccnc1Br)C2 79216,N1(C(C(CCC)Cl)=O)C2CCC(C2)C1C(N1CCCC(C)C1)=O 79217,C(=O)(C(C(C)C(C)(C)C)N(CC(C)C#N)C)NCCCC 79218,C1(NC(CC(C)C(F)F)=O)CC2CC(C1)N(C(c1ccc(N)cc1)=O)C2 79219,C(=O)(C#CC(=O)N(C)C)NC1CC(NC(c2c(CC)occ2)=O)C1 79220,Cc1nccc(C(N2CCC(O)(CNC(c3cc(Cl)cs3)=O)CC2)=O)c1C 79221,c12cn(nn1)CC(=O)NC2(C)C.c1(C(=O)OC(C)(C)C)csc(Cl)c1 79222,CC1(CC(N2CC3CC2C3NC(C2CCCOCC2)=O)=O)CCCCC1 79223,Cc1nc(C)n(O)c1C(=O)NCC(CNC(=O)Cn1ccc([N+](=O)[O-])n1)CO 79224,N1(C(C(N2CCOC2=O)C)=O)C2CCC1CN(C(c1cncn1C)=O)CC2 79225,C1(C(=O)NCC2(F)CCN(C(C(C=C)O)=O)C2)(OC)CCCCCC1 79226,C(=O)(CCC(F)(F)F)N1C(C)(CC(=O)NC(C(=O)OCCCC)C)CC1 79227,N1(C(C2CCN(C(CCC)=O)CC2)=O)CCCC2(NC(C3CCC3)=O)CC2C1 79228,C1(NC(C2CC(F)(F)C2)=O)CC2CC(C1)N(C(=O)CCc1ccc(Cl)c(F)c1)C2 79229,CC1(C(=O)NCC2(F)CC(NC(c3cn(C4CC4)cn3)=O)C2)CC2C=CC1C2 79230,c1(C(=O)NCC2C(NC(COCCC)=O)CCC2)ccn2c1CCCC2 79231,C12(CNC(c3cnc4nccn4c3)=O)CN(C(=O)CCC(F)F)CC1CCO2 79232,c1(OC(C)C)ccc(C(=O)NCC2CC(C)(C)CN2C(=O)C(C)N(C)C)c(Cl)c1 79233,c1(SCC(=O)NCC2CC2C(=O)NCc2nc[nH]n2)ccccn1 79234,C1(C(=O)OC)CC(O)CN1C(C1CCN1C(c1ccc(F)cn1)=O)=O 79235,c1(C(C(=O)NCC(C)NC(C2(CC#C)CCCOC2)=O)OC)c(F)cccc1F 79236,CCC(C)(C)CC(=O)NC1CCCC1.C(=O)(CCS(C)=O)N1CCCC1 79237,c1(C(N2C(CNC(=O)Cc3ccns3)CCC2)=O)cc(C(F)F)cc(Cl)c1 79238,Cc1cc(-c2ccnc(C(=O)NC(c3cccc([N+](=O)[O-])c3)C)c2)cc(O)c1F 79239,CC#CCCCC(=O)NC(c1ccccc1F)CNC(=O)C(C)c1cc[nH]n1 79240,Cc1nn(C)c(=O)c(C(=O)NCC2C3CC2N(C(C2(C)CCC(=O)N2)=O)C3)c1C 79241,C(=O)(C(O)CC(F)(F)F)NCC(CC)NC(=O)COc1ccccc1 79242,c1(CNC(COC(CC)C)=O)nc(CNC(=O)C(O)CSC)cc(O)n1 79243,C1(NC(c2ccnc(C3CC3)n2)=O)C2CC1N(C(C1CC3CCC1O3)=O)C2 79244,C1(C(N(CCCNC(=O)C2=CCCCC2)CCO)=O)CCCC2CCCN12 79245,c1(CCCC)cc(C(=O)NC2CCCCC2NC(c2n[nH]c(C)n2)=O)c(C)o1 79246,C1(CCOC)CN(C(C2COC(C)(C)CO2)=O)CCN1C(=O)CC(C)(C)C 79247,N1(C(c2n(CC)nnc2)=O)CC(NC(=O)C2=CCCC(C)(C)C2)CC12CCOC2 79248,N1(C(c2c(O)ccc(C)c2)=O)CCCC(C)(C)C1CNC(C1CCNC(=O)C1)=O 79249,c1(C(=O)NCCN(C(C2C(C)(C(C)C)C2)=O)C)ccc2c(=N)[nH]cnc2c1 79250,c1(C(C(N2CCC(N(C(=O)CC3CC3)CCO)C2)=O)O)ccc(Cl)c(Cl)c1 79251,c1(CC(=O)NC2C3CCC2N(C(c2cccnn2)=O)C3)n[nH]c2c1CCCC2 79252,C12(C(=O)NCC3N(C(=O)CCCc4ncco4)CC(F)C3)CC1COC21CCC1 79253,c1(C(=O)NCC2(CNC(CCCOC)=O)CCC2)cccc(C(=O)OC)n1 79254,Cc1c(C(=O)NC2CCC2NC(c2ccn(CC(F)F)n2)=O)ccn1CC1CC1 79255,c1(C2(C(CCCCCn3cc(C4CCCC4)nn3)=O)CC2)ccc2c(c1)OCCO2 79256,c1(CC)cc(C(=O)NC2(C(N3CCC(n4cncn4)C3)=O)CSC2)nn1C 79257,c1(CC)c(C(N2CC(NC(C3C4CC4C4CC34)=O)C2)=O)oc2ccccc12 79258,C1(C(=O)NCc2cc(C)no2)(NC(=O)COc2ccsn2)CCCC1C 79259,C1(NC(c2cc(Cl)cc(F)c2F)=O)CN(C(C2(O)CCOC2)=O)CC2(CC2)C1 79260,c1(C(=O)NCC2CN(C(CCNC(=O)NC)=O)C3C2C3)ccnc2c1nnn2C 79261,N1(C(C(C)(N(C)C(C2CC(=O)CC(=O)N2)=O)C2CC2)=O)CC2(CCC(=O)N2)C1 79262,N1(C(C(CC)COC)=O)Cc2ccc(C(C)NC(C3CCCCCC3)=O)cc2C1 79263,c1(C(=O)NCC2C3CN(C(C(CC(N)=O)O)=O)CC32)cccc2nc(O)[nH]c12 79264,Cc1ccc(O)cc1C(N1CCC12CN(C(=O)C1=NOC(C3(O)COC3)C1)C2)=O 79265,N1(C(CN(C)C(N)=O)=O)C2CCCC1CC(CNC(C1(O)CCC1)=O)C2 79266,C1(O)(CNC(c2c(C)oc(C3CC3)n2)=O)CCCN(C(=O)CCC2CCOC2)C1 79267,C(C)(C)(CC(=O)N(C1CCCN(C(c2ccc(F)cc2)=O)C1)C1CCCCC1)OC 79268,N1(C(C(CCC)n2cc(COC)nn2)=O)CCCC(NC(c2c[nH]nc2C)=O)C1 79269,C1(NC(CC=CCC)=O)CCC2(CCCN(C(c3cnc4n3CCC4)=O)C2)C1 79270,c1(OC)ccc(CN(C)CC2(Cc3ccncc3C)CC2)cc1Br 79271,c1(CN2CC(CNC(C3C(C)(C)C3)=O)SCC2)ncc(Br)cc1[N+](=O)[O-] 79272,C12(NC(c3cncc(NC)c3)=O)CCCC1(F)CN(C(=O)Cc1coc(C)n1)C2 79273,c1(C(=O)NC2CN(C(CCC(=O)OC)=O)CC(O)C2)cccn2cnnc12 79274,C#CC1(C(=O)NCC2(C)CCCOC2)CN(C(c2nnsc2C)=O)C1 79275,O=[N+]([O-])c1cc(Cl)c(F)c(S(=O)(=O)OCCCOCC2CCC2)c1 79276,CN1C(=O)CN(C(C2CCCCN(C(c3cc(C#N)ccc3N)=O)C2)=O)CC1=O 79277,N1(C(C2N(C)CC2)=O)CCC(C(=O)NC2CC2c2ccco2)C1(C)C 79278,c1(CC)cnoc1C(=O)NCC1CC(CNC(=O)CCSC(F)(F)F)CO1 79279,N1(C(C(N2C(C)CCC(CO)C2)=O)=O)CC2(C=C(C(=O)O)CO2)C1 79280,C1(C(=O)NOCCCF)(COC)C=CCN1C(c1c[nH]c(C(N)=O)c1)=O 79281,CC(C)(C(=O)NCC1(O)CCN(C(c2ccccc2O)=O)CC1)C(N)=O 79282,c1(CCC(=O)NC2CN(C(C=C(C)Cl)=O)C2)c(C)nc(-c2ccccc2)nc1O 79283,N(C)(S(=O)(=O)N1CCC(C(N2CCNCC2)=O)CC1)C(CC)COC 79284,C(CC(C)C)(C(=O)NC1(C)CCN(C(=O)Cc2ccc(C(C)=O)cc2)C1)OC 79285,C(=O)(CCCC(c1ccccc1)NC(c1cc(C(C)(F)F)on1)=O)OC 79286,CC1OCCC1CNC(=O)NC1(CO)CC1c1ccccc1 79287,C(=O)(CCCN(C)N=O)N1CCC(C)C1CNC(=O)COCC1CCC1 79288,C1(CC)C(NC(=O)Cc2ccccc2O)CCCN1C(=O)CC1CCC(=O)N1 79289,c1(SCC(N2CCCC2Cn2cc(C(=O)O)cn2)=O)ccccc1Cl 79290,c1(C(=O)NC2CCC(NC(C(CC)(C)O)=O)CC2)c(Cl)cncc1Cl 79291,C1(NC(=O)COCc2nccn2C)CCOCC1.C12CCN(C1)C(=O)COC2C 79292,C1(C(=O)NCCC(C)NC(c2cccc(C(N)=O)n2)=O)CC2C(C1)C2(C)C 79293,c1(CC)nc(=N)[nH]c(=NC2CC3CC(C2)N(C(C2CC(=O)N(C(C)C)C2)=O)C3)[nH]1 79294,C1(CNC(c2ccccc2OCc2cccs2)=O)CC2(C1)CC21CC1 79295,C12(COC)CC(NC(=O)CN3C(=O)CNC3=O)(CN1C(=O)C(C)C(C)(C)C)C2 79296,CC1=C(C(=O)NCC2CCCCC2NC(=O)C(N)=O)C(C)n2ncnc2N1C 79297,c1(OC(C(=O)NCC(C(C)C)NC(c2cn(CC=C)nc2)=O)C)cccc(F)c1 79298,N1(C(CCNC(=O)C=CCl)=O)CCC2(CC(NC(C3CCCCC3(F)F)=O)C2)C1 79299,C(=O)(CCC(C)(C)F)NC(C1CCN(C(c2ccn(C)n2)=O)C1)C 79300,N(C(=NCCCN1CCOCC1)NC1COC2CC1C2)CC1(O)CCSC1 79301,c1(N2C3CN(C(c4ccc5nc[nH]c5c4)=O)CC2C3)ncnc2cccc(F)c12 79302,C(N=c1[nH]c(=NCCOCCC2CC2)[nH]c2c1CCCC2)c1c(F)ccc(F)c1 79303,C=CCC(C(=O)NC(CCC)C(O)C(=O)N(C(CC)CC)CCO)C(C)C 79304,c1(C(N2CCCC2)CNC(N(C)Cc2c[nH]c(=N)s2)=O)cccnc1Cl 79305,C(N=c1ccnc(NC(CC)CO)[nH]1)C1(C=C)CCC1 79306,C1(NC(C(CC)C(C)C)=O)CCOC2(CCC2)C1 79307,N1(C(c2c(C)cco2)=O)CCCC(C(C)NC(=O)C2=CCCC2)C1 79308,c1(C(=O)NC2CN(C(COCC)=O)C(C)C2)ccc([N+](=O)[O-])cc1 79309,C1(NC(c2c(COC)ncs2)=O)CCN(C(c2oncc2C)=O)C(C2CC2)C1 79310,C1(C(=O)NCC2(F)CC(CO)C2)CCN(C(=O)c2cc(O)ncn2)O1 79311,C1(C2CN(C(=O)CCCCNC(=O)C3CC3)C2)(NC(c2cc(Cl)ns2)=O)CC1 79312,C1(C(=O)NC(C2CCN(C(c3ccncc3N)=O)CC2)C)Cc2ccncc2C1 79313,N1(C(CC2ON=C(C)C2)=O)CC(NC(c2c(N)cccc2Cl)=O)CC(F)C1 79314,CC1CN2CCC1NCc1cc(no1)C2=O.c1(C(N(C)C)=O)csc(C2CC2)n1 79315,CCN=c1cc(C(N2CC3OCC(NC(=O)CN(C)C4CC4)C3C2)=O)cc[nH]1 79316,c1(NC(c2nnnn2CC2CC2)(COC(C)=O)C)cnc2c(c1)COCC2 79317,C1(CCN)(NCC(C2CC3CCC2C3)NC(=O)O)CCOCC1.S 79318,CC(Cn1cccn1)C(=O)NCC1C(CNC(=O)C(F)CC2CCOC2)C1(F)F 79319,Cc1cn2cc(C(N3CCCC3CNC(C3(C)CCCN3C)=O)=O)cc(F)c2n1 79320,CC(CC(C)(F)F)C(=O)N(CCCCCNC(c1cc2n(n1)CC(F)C2)=O)C 79321,C1(C(N2CCCC(C(=O)NCC3N(CC)CCC3)C2)=O)CCCCC(C)O1 79322,S(=O)(=O)(C1CC2(CC2C(=O)O)C1)Nc1ccc(SC(CC)(C)C)cc1 79323,C=C(C)CCC(=O)N1CCC(C(C)(C)NC(c2c[nH]cc2-c2ccc(C)s2)=O)C1 79324,c1(C(NOC(CC)CC)=O)cc(CNC(=O)C=CC(F)(F)F)c[nH]1 79325,c1(C(=O)NCC2(OC)CCN(C(C3CC34CC4)=O)C2)nncc2c1CCCC2 79326,N1(c2nc(CC)on2)CCC2(CC1)CC2C(N1CCC2OCC2C1)=O 79327,c1(OC)cc(CO)ccc1C(=O)NC1C2CC1N(C(=O)C(=Cc1ccco1)C)C2 79328,Cc1cc(OCCCC(=O)N(CC(C)(O)C2CCC2)C)ccc1Cl 79329,N1(C(C(F)=CC)=O)CCCCC2(C1)CN(C(=O)CCn1ccnc1C(C)C)C2 79330,c1(C(=O)OC)cc(NC(=O)C(C2CCOC2)NC(=O)OC(C)(C)C)c(C)o1 79331,Cc1cc(CCNC(=O)CN2CCC(N(C)C(C3CCCCCC3)=O)C2)c(C)s1 79332,N1(C(Cc2c(OC)nccc2)=O)CCCC(C)(NC(=O)CC2CCCN2C)C1 79333,N1(C(C2C(=O)OCC2)=O)CCC2(CCCCN(C(c3ccc(O)nc3)=O)C2)C1 79334,c1(OC)ccc(C(N2CCN(C(C3CCCSS3)=O)C(C)C2)=O)cc1C 79335,C1(CNC(C2(C=C)CC2)=O)CCCCN1C(C1(C(F)F)CC(=C)C1)=O 79336,C1(C(=O)NC2(CCCNC(CCCCN(C)C)=O)CC2)CCC2CC2CC1 79337,c1(N2CCC(c3nnc(C)o3)CC2)nc2cc[nH]c2c(=NCC2(C)CSC2)[nH]1 79338,N1(C(=O)CC23CCC(CC2)CC3)C2CCCC1CC(NC(C1CCCCS1)=O)C2 79339,c1(C(=O)OC)c(OC)cc(NC(=O)CCSC2CC(=O)N(C3CC3)C2)cc1Br 79340,C(C1CN(C(=O)COCCO)Cc2ccccc21)NC(CC(C)(C)O)=O 79341,C1(CC(=O)NC2CCCCC2NC(C2(CC3CC3)CC2)=O)(COC)CCOCC1 79342,c1(CC(N2CC(NC(CC(C)c3ccccc3)=O)C2)=O)ccc(SC2CC2)cc1 79343,C1(CC=C)(C(N2CC(OCC(=O)NCCCF)C2)=O)CC=CC1 79344,N1(C(C2CC(=O)NC2)=O)CC(CNC(c2cccc(Cl)c2Cl)=O)C2(CCC2)C1 79345,C(=O)(C(O)C(C)(C)CC)NC1C(NC(c2cc(CC)[nH]n2)=O)C1 79346,CCC(O)C(C)(C)C(=O)N1CCC(C(F)C(=O)N(C2CC3(CCC3)C2)C)C1 79347,Cc1cccc(OCC(N2CCC(C)(c3cn(C4CCOC4)nn3)C2)=O)n1 79348,c1(CC(N2CC3C(CNC(C4C(C)C4)=O)C3C2)=O)cc2ccccc2s1 79349,C1(=O)C(F)(F)CCn2cc(nn2)CC2CN1C2.N1CCCCC1.C1(C=O)CC1(Cl)Cl 79350,c1(NC(C(C)C)CNC(C2CCCNS2(=O)=O)=O)ncnn2cccc12 79351,Cn1cc(NC(=O)Cn2cc(Cl)c(C(F)(F)F)n2)ccc1=O 79352,C1(NC(C(COCC)C)=O)C2CC3C1C3C2C(=O)NC1CCC(N(C)C)C1 79353,C(=O)(CCCCC(=O)NC(c1ccccc1)c1nccn1C)NC 79354,C(CC(=O)N=c1cc2ccccn2[nH]1)N(C(=O)Cn1nccn1)CC1CC1 79355,Cc1ccc2c(C(=O)N(C)CC3(O)CN(C(c4ccnc(O)c4)=O)C3)c[nH]c2c1 79356,CC(CC(C)(C)C)NC(c1[nH]ccc1CNC(=O)CCC1CCCCC1)=O 79357,c1(C(=O)NC2(CC=C)CCN(C(=O)CCC(C)C#N)C2)cccc2ccncc12 79358,C#CCC(O)C(=O)NC(c1cn(C)nn1)C(=O)N(C)Cc1conc1CC 79359,c1(C(C(=O)NC(CN(C(C=CSC)=O)C)C)O)ccc([N+](=O)[O-])cc1 79360,C(=O)(C1CCCc2nc[nH]c21)NCC1CC(OC)CN1C(C1CCC1(F)F)=O 79361,Cc1nn2cccnc2c1C(=O)NCCCCNC(=O)COC1CCCCC1C 79362,Cn1ncc(C(=O)NCC2(NC(C3CCC(F)CC3)=O)CCC2)c1Cl 79363,C(=O)(C(C)C(F)(F)F)N1CCC(NC(c2cc(OC)c(Cl)s2)=O)C1 79364,N1(C(Cc2c(C)cnn2C)=O)CCC(NC(=O)CC(=O)Nc2nccs2)C(F)C1 79365,Cc1cc(O)cc(C)c1C(=O)NC1CCCC(NC(=O)Cn2cnccc2=O)C1 79366,Cc1cncc(CCC(=O)N(CC(C)CNC(=O)Cn2nnc(C3CC3)n2)C)c1 79367,C1(C(=O)NCC)Cc2c([nH]c3ccccc23)CN1Cc1ccnc2ccccc12 79368,Cc1cc(CCC(=O)NC(C(=O)NCC2CC2(Cl)Cl)C2(O)CCC2)n[nH]1 79369,S(=O)(=O)(c1cc(C(N2CCCN(C(=O)C=CCO)C(C)C2)=O)cc(C)c1C)NC 79370,CCCCC(O)C(=O)NCC(CC(F)(F)F)NC(c1cc(Cl)ccc1C(F)F)=O 79371,C1(C(=O)NCC2N(C(C(C)Cc3cnc[nH]3)=O)CC(O)C2)CC(C)(C)CCO1 79372,c1(C(=O)NC2CCC(NC(C3CCC(C)C3)=O)CC2)cnn2c1N(C)CC2 79373,C12(NC(c3cc[nH]c3)=O)CN(C(=O)CSC3CC3)CC1CS(=O)(=O)C2 79374,C(=O)(CC(C)c1cnn(C)c1)N(C(C)CNC(=O)CCOC1CC1)C 79375,c1(C(=O)NC2CC(C)N(C(c3cc4oc(Cl)cc4[nH]3)=O)C2)cn2ccccc2n1 79376,C(=O)(CCC(=O)C(C)(C)C)N1CC(C(=O)NCCc2ncn(C)n2)CC(C)(C)C1 79377,C(=O)(C(CCC1CCC1)NC(=O)CCC=C(C)C)NC(CC)C1CC1 79378,c1(NC)ccnc2ccccc12.c1(CC)cc2nc(n1)N2 79379,N1(C(c2cc(C)n(C)c2)=O)CC(NC(c2conc2C(C)(C)C)=O)CCC1C 79380,C1(CC)CN(C(C2CCOCC2(C)C)=O)CCN1C(=O)C=CSc1ccccc1 79381,C(=O)(C1=CC2C=CC(C1)C2)NCC1CCCC(NC(c2c(C)cccc2)=O)C1 79382,C=CC1CN(C(c2cn(C)ccc2=O)=O)CC1NC(c1conc1C(C)C)=O 79383,c1(C(N(C2CCCCN(C(=O)C=CS(C)=O)C2)C)=O)noc2ccc(F)cc12 79384,C1(C(=O)NC2CC(CNC(c3ccccc3C(N)=O)=O)C2)(OC)CCCC(C)C1 79385,N1(C(c2n(CCCC)ncc2)=O)CC2CC(NC(c3cnoc3C)=O)CC1C2 79386,C1(NC(=O)C2CC2)C2CC3CN(C(c4cnc5sccc5c4)=O)C1C3C2.c1cc[nH]n1 79387,N1(C(CC2CC(CC)OCC2)=O)CCCN(C(c2cnsn2)=O)CCC1 79388,C(C1c2ccsc2CCN1C(=O)C(O)CC1CCCCC1)NC(CCC=C=C)=O 79389,c1(OC)ccc(S(=O)(=O)N(C)C)cc1C(=O)O.c1(C(C(=O)O)N)cscn1 79390,Cc1cc(C(=O)NC23CC2CN(C(c2cc(-c4cccs4)on2)=O)C3)nc(Cl)c1 79391,C1(CN(C(CSCC(C)C)=O)C)CN(C(=O)CC2COCCN2C)CCO1 79392,N1(C(CC)=O)CCC(C(=O)N(C)CC2CN(C(C3(CCF)CCC3)=O)C2)C1 79393,CC1(CNC(=O)CC2CCCC(C3CC3)O2)CCCN1C(=O)CS(N)(=O)=O 79394,Cn1nnc2cc(C(=O)NC3(C)CC(NC(c4cnn[nH]4)=O)C3)ccc12 79395,C1(NC(Cc2ccc(C)cc2)=O)CCN(C(=O)C=CC(=O)NC2CC2)CC1CO 79396,C(=O)(CC1CCc2ccccc21)N(C1CN(C(=O)C(F)F)CC1(C)C)C 79397,C1(CCNC(C(CC)CO)=O)CN(c2nc(C(C)C)cc(C)n2)CCS1(=O)=O 79398,C(C(=O)NCCNC(=O)Cc1ccnc(Br)c1)(C(C)(C)C)N(C)C 79399,c1(C(N2C(C(C)NC(=O)C(C)(Cl)Cl)CCC2)=O)ccc2ccoc2c1 79400,CCC(C#N)(CC)C(=O)NCn1cc(C(=O)NCC2CC(C(C)C)C2)nn1 79401,c1(C(=O)NC2CN(C(C(C)NC(CC)(C)C)=O)C2)n[nH]c(C)c1Cl 79402,c1(N2CCC(C=C)CC2)nc2ccc(S(=O)(=O)NC3CCCC(CC)C3)cc2s1 79403,C1(CNC(C2(CC)CCCC2)=O)CCCCC1C(=O)NCc1ccc[n+]([O-])c1 79404,N1(C(c2c(Cl)cc(C)nc2)=O)C2CCCC1CN(C(=O)CC1COC(=O)N1)C2 79405,c1(C(N2CCN(C(C(C)OC)=O)CC3(C2)CC3)=O)cc2c(O)ccc(F)c2[nH]1 79406,c1(C(=O)NC(C)CN2CCCC2)c(I)ccc(Cl)c1Cl 79407,c1(C(C)C)n[nH]c(=NC2CCNCC2)o1.C(=O)C(C)C(C)S(C)(=O)=O 79408,C1(C(=O)NCC2(F)CCN(C(C(F)=C(C)C)=O)CC2)CC(C)(C)OC(C)(C)C1 79409,C1(C(N2CCC(N(C(=O)Cn3nnc(C4CC4)n3)C)CC2)=O)OC2CCC1CC2 79410,c1(C(=O)OC)ccn(CC(=O)NCCN(CC(C)O)C(c2cnccn2)=O)n1 79411,N(C(=NCc1ccc(OC(F)F)cc1)NCC12CC(CCO1)C2)Cc1c(C)ocn1 79412,c1(C(=O)NC(CCOC)CNC(=O)CC2(NC(C)=O)CC2)ccnc(C)c1N 79413,C1(C(N2CC(CCC)C(CO)C2)=O)CCCCC1(C)NC(=O)C(=O)N(C)C 79414,N1(C(CC(C)=C(C)C)=O)CC(C)(C)CC1CNC(=O)CCc1cccnc1F 79415,Cc1cc(C(=O)NCC2CCC(CNC(=O)CC(C)C3CC3)CC2)cn1C 79416,C1(C(=O)Nc2cc(O)n[nH]2)CCCC12CCN(Cc1cscn1)C2 79417,Cc1cc(=NC(CCO)C2CCSCC2)[nH]c(=NCc2cccc(CO)c2)[nH]1 79418,C1(NC(CNC(CC)=O)=O)(CF)CCN(C(=O)C=C2CCC2)C1 79419,c1(C(=O)NC(CNC(c2c(CC)ccs2)=O)C2CCC2)ccc(F)c(C)c1F 79420,C=CC(C)(CC)C(=O)NC(CC(=O)Nc1cnc(N(C)C)nc1)C1CC1 79421,N1(C(c2cn(CCC)nc2)=O)CCC2(C)CN(C(=O)CC3CNC(=O)O3)CC12 79422,C1(N(C(C(C2CCCC2)OCC)=O)C)CCCCC1NC(c1ccc(C)nn1)=O 79423,Cc1c(-c2cnc(F)c(C(=O)Nc3cnccc3C(N)=O)c2)cccc1[N+](=O)[O-] 79424,c1(C(=O)NCCCNC(C(CC2CCCCC2)OC)=O)c([N+](=O)[O-])c(C)nn1C 79425,n1(CC(=O)NC(C)CCNC(C2CC2(C)Br)=O)nc(C(C)(C)C)cc1N 79426,c1(CC)cccc(CC)c1C(=O)NC1CCN(Cc2cnc(Cl)s2)CC1F 79427,c1(CC(=O)NCC(n2cc(C3(CO)CCN(C)CC3)nn2)C)c(F)cncc1Cl 79428,c1(C(=O)NC2C(CC)N(C(c3ncc(F)cn3)=O)CC2)cc(=O)cc(Cl)[nH]1 79429,C=C(C)CCCC(=O)N(C)CC1CCCN1C(=O)C(N1CCOCC1)C 79430,N1(C(CSCCC)=O)CC(CO)C2(C1)CN(C(=O)C(O)CN1CCOCC1)C2 79431,N1(c2cc(NCc3cnc(C(C)(C)C)[nH]3)nc(C)n2)CC2CCCCC2(CO)C1 79432,c1(C(=O)NC2CCC(CCNC(C3(CC(C)C)CC3)=O)C2)cnn2ccsc12 79433,Cc1cc(C(N2CCC(CNC(=O)CN3CCCC3=O)C(C)C2)=O)c(N)c(Cl)c1 79434,c1(OC)cccc(N(C(=O)COC(C)(C)CNC(c2nc(C)oc2C)=O)C)c1 79435,C(CC(O)C(=O)N(CCCCNC(=O)CCC(C)OC)C)SC 79436,Cc1c(CC(=O)N(CC(=O)NOC2CCOC2)C2CC(C#N)C2)cco1 79437,C(=O)(CS(=O)C(F)(F)F)NCCC(C(C)C)NC(c1cnc2ccoc2c1)=O 79438,c1(C(C)CC(=O)NCC(O)CN(C)C(c2ncn(C)n2)=O)ccc(Br)cc1 79439,N1(C(c2cccc(N(C)C)c2)=O)CCN(C(C2CC(C)(F)C2)=O)C2COCC12 79440,N1(C(=O)NCC2(CC)CC2)CCN(C(C)C(=O)NC)C(=O)C1 79441,C12(CNC(CNC(=O)OCC=C)=O)CCC1CN(C(=O)CC1CC(F)(F)C1)C2 79442,c1(NC(C2(O)CCN(Cc3ccccc3SC(F)(F)F)C2)=O)ccccc1I 79443,N1(C(C(=O)Nc2cnc(N3CCOCC3)nc2)=O)CCC(C2CCOC2)CC1 79444,N1(C(c2n[nH]c(C)c2O)=O)C2CCC1C(C)C(NC(c1ccc(CF)cc1)=O)C2 79445,c1(CC(=O)NC(CC)CNC(=O)C(C)n2cnnn2)ccc(C)c(C)c1 79446,N1(C(CSCC(C)=O)=O)CCCC1COC(F)(F)F 79447,c1(CNC(C2(NC(C3SCCS3)=O)C(C)C2)=O)ccc(Cl)cc1 79448,C1(C(=O)NCCC(=C)CNC(=O)CC2=CCOCC2)C2CC3CC(C2)CC1C3 79449,C(=O)(C(F)CCC(C)(C)C)NC(C)C(CO)NC(=O)C1=NOC2(CCC2)C1 79450,C(CCCN=C(NCC1CCC(C)O1)NCC(C)(C)C)N(C(C)C)C 79451,c1(CC)nc(C)[nH]c1C(N1CCOC(CN(C(=O)Cc2cnccc2Cl)C)C1)=O 79452,C1(C(=O)NCC2C(NC(c3cc(OC)no3)=O)CCC2)CCC(C)(O)CC1 79453,N1(C(CC2(OC)CC2)=O)CC(CCNC(c2cnoc2SC(F)F)=O)OC(C)C1 79454,c1(CN2CCC(CC(=O)NC(c3ccccc3)CO)C2)c(F)ccc(O)c1F 79455,Cc1nc(Br)cnc1NC(C1CCCN(C(c2cnnn2C)=O)CC1)=O 79456,C1(C(=O)NC(c2ccc(OC)nc2)CC(N)=O)CCCCCC1(F)F 79457,C[Si]1(C)CC(C(=O)O)N(C(C2CCCN2N=O)=O)C1 79458,N1(C(c2c(C)nc[nH]2)=O)CCC(F)(F)C(CNC(=O)Cc2ccnc(Br)c2)C1 79459,N1(C(CN(CCCCCC)C)=O)CCOC(C(N(C2(CC)CCC2)C2CC2)=O)C1 79460,C(=O)(CCCCSC)NCC1(OC)CN(C(=O)COC2CCOCC2)C1 79461,C(=O)(C1Cc2ccccc21)NC1CC(CNC(c2ccnc(C)c2N)=O)OCC1 79462,C1(CNC(N2CCC(O)C2c2ccc(Br)cc2)=O)CC(F)(F)C(=O)N1 79463,C1(NC(CSC)=O)CCCN(C(=O)CC2(O)CCC2)CC1 79464,C1(NC(c2cnccc2Cl)=O)CCCC12CN(C(c1cn[nH]c1)=O)C2 79465,C1(OC)(CNC(=O)CS(=O)(=O)N2CCOCC2)CCN(C(=O)C2=CCCC2)CC1 79466,N1(C(C(C)OC)=O)CCCC(C)(NC(C23CC(C(=O)OCC(F)(F)F)(C2)C3)=O)C1 79467,Nc1ccc(C(N2CCCC(O)(CCNC(=O)C=CC3CCCO3)C2)=O)c(Cl)c1 79468,N1(CCC)CCCCC1C(N1CC2CC2(CNC(=O)CSC(F)F)C1)=O 79469,N1(C(CC2C(=O)NC(=N)S2)=O)CC2CC(CNC(=O)Cc3cc(C4CC4)no3)C2C1 79470,c1(COC(C)=O)cccc(-c2cnc(CNC(c3cc(O)ncn3)=O)nc2)c1 79471,C(c1cc(Cl)cc(Cl)c1)=CC(N1CCCCC(CNC(c2cccnc2)=O)C1)=O 79472,C1(C(=O)NC2C3CN(C(CSCC)=O)CC32)CC2(CCC2)CCO1 79473,N1(C(C2(C#C)CC2)=O)CC(OC)C(C(=O)NCC2(OCC)CN(C)C2)C1 79474,C(C)(c1ccc(OC)cc1)=CC(N1CC(F)(CNC(CSCCOC)=O)C1)=O 79475,N1(C(c2ccc(C)c(NS(C)(=O)=O)c2)=O)CCN(C(=O)CC(F)F)C(C)C1C 79476,c1(OC)cc(C(N2CCC3(CC2)CC3NC(=O)C(O)C(C)C)=O)cc2ccoc12 79477,C#CC1(C(=O)NCc2ccco2)CN(C(=O)CN2CCOCC2=O)C1 79478,Cc1cnc(N2CCC(NC(C3CN(C)C(=O)N3)=O)C2C)nc1 79479,c1(C(N2CCC(c3ccccc3)(COC)C2)C(=O)NCC)cn2ccccc2n1 79480,Cc1cc(Cl)c(C(N2CCC(NC(c3c[nH]c(C(N)=O)c3)=O)C(F)C2)=O)cc1C 79481,c1(-n2c(CC3CCCCC3)nc(C(C)C)n2)cccc2c1CCCC2 79482,c1(OC)cccc(-c2nc(CCC3CCOCC3)n(CC3CC3)n2)c1 79483,n1(CC)cnc2c(NCC3(SC)CC3)[nH]c(=NCc3n[nH]c4c3COCC4)nc12 79484,CC1CCCC2(CC2)CN1C(C1(CC(=O)NC2CC2)CCCC1)=O 79485,C(=O)(N1CC(O)CCO1)NC(C)CS(C)(=O)=O 79486,N(C(=NC)N1CCC(NC(c2cccs2)=O)C1)CC1N(CC)CCC1 79487,N1(C(C(CC)(C)O)=O)CCC2(CCN(C(c3cc(COC)[nH]n3)=O)CC2)C1 79488,CCCCCCCCN(C)C(C1CCCC1CNC(c1ccc(C(C)=O)o1)=O)=O 79489,Cc1ccc(C(=O)NCC(CO)NC(C2(CC(F)(F)F)CC2)=O)nc1 79490,C(C)(C(=O)N1CC(CCNC(=O)C(O)C2CC2)C1)(C1CC1)OC 79491,C(=O)(CCCN=[N+]=[N-])N(C1CCN(C(C2CCCC(=O)N2C)=O)CC1)C 79492,Cc1ccc(C=CC(=O)NC2CCCC(NC(=O)C(C)C(C)C)C2)o1 79493,C1(C(=O)NC(C)CNC(N)=O)CC2(CCN(C(C3CCC4(CCC4)C3)=O)C2)C1 79494,c1(C(=O)NCC2C(C)CN(C(c3ccc(F)s3)=O)C2)csc2nnsc12 79495,C1(NC(C(C2CCOCC2)C)=O)CCCC(NC(=O)Cc2csc(S)n2)CC1 79496,C1(O)(CCNc2ccc(C(=O)OCC)cn2)CCCN(C(c2n[nH]cc2F)=O)C1 79497,c1(N(CC(=O)NCCC)C)nc(=NC2CCCC2)[nH]c2ncn(CC)c12 79498,N1(C(Cc2cc(COC)on2)=O)CC2CCN(C(=O)CSC(C)(C)C)CCC2C1 79499,N1(C(=O)Cc2cccnc2Cl)CC2CCCC(C1)N2C(C1CCC(C(N)=O)O1)=O 79500,NS(=O)(=O)c1cccc(C(=O)NC2CCCC2CNC(=O)CCc2cnc[nH]2)c1 79501,c1(C(=O)NC2CC3CN(C(C(F)OC)=O)C2C3)ccc2c(c1)NC(=O)CN2 79502,c1(C(=O)NC2CCCN(Cc3c(C)ccnc3)C2)cc2cc(Cl)ccc2[nH]1 79503,c1(C(N(CCC(C)NC(c2c(CC)con2)=O)C)=O)csc2ccc(F)cc12 79504,N1(C(C(CC)(CO)OC)=O)C2CCC(C(=O)NCC3CCC3(F)F)C1CC2 79505,c1(CC)cc(C(N2CCCC2(C)CNC(=O)C=CCOC)=O)c2c(c1)CCO2 79506,CC(C)(CO)C(=O)NC1CCN(C(c2cnc(C(F)(F)F)o2)=O)C1 79507,CC1(C)C(NC(=O)C(O)CC2CCOCC2)CCN1C(C1CCS(=O)(=O)CC1)=O 79508,N1(C(CN2C(C)CCC2)=O)CCCC(O)(CN(C)C(c2cccnc2CO)=O)C1 79509,CC1OC2(CNC(=O)COC3CCCCC3)CC1(NC(=O)Cc1ccn(C)n1)C2 79510,c1(CC(=O)NCCCN(CCCOCC(=O)OC)C)ccc(C)c(C)c1 79511,N1(C(C2CCCCC2CO)=O)CC2CCC1CN2C(=O)CCCC1CCOCC1 79512,N1(C(c2c(C)[nH]nc2C(F)F)=O)CCC(NC(=O)OC(C)(C)C)CC(C)(C)C1 79513,C1(C(N2C(CN(C)C)COCC2)=O)CCN(C(=O)C=CC2CC2)C1(C)C 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79566,c1(C(N2C(C)(CNC(C3(CCF)CCC3)=O)CCC2)=O)ccn2nccc2c1 79567,C1(CCC)CN(C(c2cn(C)nn2)=O)CCN1C(c1cc(CC2CC2)on1)=O 79568,c1(CN(C(C(Cc2cc[nH]n2)NC(c2cc(CC)sn2)=O)=O)C)cc(C)ccn1 79569,C1(C(C)(C)O)CCCCCN1C(=O)CNC(c1cncnc1)=O 79570,C1(NC(C2(C(=O)NC)CC2)=O)CCN(C(=O)C(c2ccncc2)C)CC1C 79571,Cc1cc(C)c2c(C)c(C(=O)NCC3CCC3NC(=O)C=CC3CC3)[nH]c2c1 79572,Cc1nc(CC2CC2)sc1C(N1CCC(CNC(=O)C(C)Cn2ccnc2)C1)=O 79573,N1(C(c2ccc(C(=O)OC)s2)=O)CC(NC(c2cccc(O)n2)=O)CC2(CC2)C1 79574,c1(CNc2cc(-c3cn(C4CC(CO)C4)nn3)cc(Cl)c2)ccc2c(c1)OCC2 79575,C(=O)(C(F)CC(C)(C)C)NCC(C(=O)NCCc1cc(C)ns1)N(C)C 79576,C(CN=c1[nH]c(N2CCOC(CC(C)C)C2)nc2c1CC(C)CC2)NC(=O)NC 79577,Cc1cc(Cl)ccc1OC(C)C(=O)NCC(F)CNC(C1(CC(F)(F)F)CC1)=O 79578,c1(C(N2C(C(=O)Nc3ccn4ncnc4c3)CC2)=O)ccc2cccc(F)c2n1 79579,c1(SCC(=O)NCC(c2ccccc2)NC(C=C(COC)C)=O)ccc(C)cc1 79580,C1(C(C)C)NCC12CCN(C(c1ncccc1N)=O)CC2 79581,C1(C(N(CC(CC)NC(C2CC(F)(CO)C2)=O)C)=O)CCCN(C(N)=O)C1 79582,c1(C(=O)NC2C(C(N(CC)CC3CCCO3)=O)CCC2)cc(C)cc(O)c1 79583,CCC(CC(=O)NC1COCC1N1CCN(C(=O)C=C(C)Cl)CC1)c1cn[nH]c1 79584,Cc1noc(C)c1CC(C)C(=O)NC1(CCNC(c2[nH]nnc2C(F)F)=O)CC1 79585,c1(C(=O)NC2(C)CN(C(C(C)NC(CC)=O)=O)C2)cc2ccc(C)cn2c1 79586,Cc1cc(O)c(C(=O)NCCOCCCNC(=O)C(C)NC(N)=O)cc1F 79587,C1(CC)CCC(C(=O)NCC(C(=O)N(CCC(=O)NC)C)N(C)C)O1 79588,S(=O)(=O)(c1ccc(Br)cc1N1CCC(CC(F)(F)F)C1)N(C)Cc1ccc(Cl)s1 79589,C1(CNC(CC(C)NC(N)=O)=O)CC2(CC2)CN1C(=O)Cc1cccc(N)c1N 79590,c1(C(=O)NC2C(NC(c3ncc(C)cc3F)=O)C2)cc2sc(C)cc2n1CC1CC1 79591,C(=O)(C1=CCS(=O)(=O)C1)N1CC(NC(c2ccncc2)=O)C(CO)CC1 79592,c1(C(=O)NCC2(O)CCN(C(CCCOCCC)=O)C2)c(F)cc(F)c(F)c1F 79593,C1(C(C)NC(=O)NCc2cc(C(N)=O)ccn2)CN(C)CCN1C 79594,C1(NC(c2ncn(CC)c2)=O)CC1C1CCCN(C(c2cc3n(n2)CCC3)=O)C1 79595,Cc1[nH]nc2ccc(C(N3CCC(CNC(=O)C4=CCCS4)C3)=O)c(Cl)c12 79596,n1(CC)nnc2c1CCC(C(N1CCN(C(=O)CCc3nccs3)CC1)=O)C2 79597,c1(C(=O)NCCc2cnc(NC(c3c(C)c(Cl)ccc3)=O)s2)cc(F)c(F)cc1O 79598,N1(C(COc2cccc(C)c2)=O)CC=C(CNC(C2(O)CC(C)(C)C2)=O)CC1 79599,N1(C(CCCC#CC)=O)CCC(C2(NC(c3cnc(N(C)C)c(Cl)c3)=O)CC2)C1 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79617,N1(C(C2COC2)=O)CCC2CCN(C(=O)CCc3cc[nH]n3)C2C1 79618,C1(CNC(C2(N(C)C)CCCC2)=O)CC(C(=O)NCC2CC(O)C(O)C2)=NO1 79619,c1(C(=O)O)cc([N+](=O)[O-])cnc1NCc1cn(CC2CC2)nn1 79620,c1(CC)ncc(C(=O)NCCC2CCCCN2C(C2CN(C)CCO2)=O)c(O)n1 79621,C1(NC(C(CCC)(C)C)=O)CN(C(=O)Cc2cnc(C)o2)C2(CCCCC2)C1 79622,C1(NC(C(CC=C)C)=O)CN(C(C23C(=O)C4CCC2C3C4)=O)CC1C1CC1 79623,C1(C(=O)NC(c2cnsc2)C)CCC(C(C)C)N1C(=O)COC1CCCC1 79624,C(=O)(CCC(C)(C)OC)NC(CC#C)C(=O)N(C)CCOCCOC 79625,c1(N(CCNC(c2c(CC)nc(C)[nH]2)=O)C(C)=O)cc(OC)nc(OC)n1 79626,N1(C(C2C(C)=C2)=O)CC2(CCOCC2)CC1CNC(c1cc2oc(Cl)cc2[nH]1)=O 79627,C1(NC(CC(COC)(C)O)=O)CN(C(=O)C=C2SCC(=O)N2C)C2(CCCC2)C1 79628,C1(C)(C)C(C)CC(=O)N1CCCO.C(C)(CCCC)CN(C(C=CCC)=O)C 79629,N1(C(C(CC)(F)F)=O)CCC(CNC(C2(C)CCCOC2)=O)C(C2CC2)C1 79630,Cc1cc(C)nc(-c2cccc(NC(=O)C(N3CCC(C)C(CO)C3)=O)c2)n1 79631,c1(C(=O)NC(CC(C)NC(CNC(C(CC)C)=O)=O)C)sc(C2CC2)nc1C 79632,N1(C(CCN(C2CCCCC2)C)=O)CC=CC1CNC(c1cscc1C)=O 79633,c1(C(=O)NC2CCCN(C(C(C=C=C)C)=O)C2)ccc2c(c1)NC(=O)CC2 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79651,N1(C(C2(OC)CC2)=O)CCC2CCC(C1)N2C(c1cc(Cl)cc(Cl)c1[N+](=O)[O-])=O 79652,CCCCC(O)C(=O)NCC(CC(=O)N1CCC(C(C)C#N)CC1)C1CCC1 79653,N1(CC)C(C)CN(C(=O)CN(C(C2CC2(F)Cl)=O)CC2CC2)CC1C 79654,N1(C(C=CCC)=O)CC2CCC(C1)N2C(c1nccn1C(C)C)=O 79655,Cc1ccc(C(=O)NCCC(C)N(C)C(C2CCS(=O)(=O)N2)=O)c(Cl)c1 79656,c1(N2CCC3(C(COC)C3)CC2)nc(=NCc2ncccc2C)[nH]c2c1COC2 79657,CCCCCC(O)C(=O)N1CCN(C(c2n[nH]c(C)c2[N+](=O)[O-])=O)CC(C)C1 79658,c1(NC(C2(C)CCOCC2)c2n(CCCC)nnn2)cccc(S(C)=O)c1 79659,S(=O)(=O)(c1cc(F)cc(Br)c1)N1C(C(=O)Nc2cnsc2)CCC1 79660,O(C1CCCc2ccccc21)CC(N1CC(NC(=O)C=CCF)C(C(F)F)C1)=O 79661,c1(C(=O)NC2(COC)CN(C(C3C(CC)CCCC3)=O)C2)ccc(O)cc1F 79662,C1(CNC(C2N(C)CC2)=O)C(C2CC2)CCN1C(C1C(C)(C)C1(C)C)=O 79663,C(=O)(CC(O)CC(C)C)NC(CC#C)(C)C(=O)N1CC(CC(F)F)C1 79664,c1(-n2ccc(CN(c3cnn(Cc4ccccc4)c3)C)n2)ccccc1F 79665,C1(NC(C)=O)CN(C(C2(C(=O)OCC)CCO2)=O)C2CCCCC12 79666,C1(NC(=O)CC2(OCc3ccccc3)CC2)CSCCN1C(C1CC=CCC1)=O 79667,C(N=c1[nH]c2c(c(=NCc3cccc(C(F)F)c3)[nH]1)CCC2)c1c(CC)nns1 79668,C(CCN=c1[nH]c2c(c(=NCC3CC4C(C3)C4(F)F)[nH]1)CSC2)OCCO 79669,C#CC1(NC(C2(NC(=O)C(CC)OCC)CCN(C)C2)=O)CC2CCCC12 79670,C1(NC(CN(c2ccncc2)C)=O)CN(C(C2CCOC2C2CC2)=O)CC12CC2 79671,CCC(CC)C(F)C(=O)NCC(CNC(c1cccc2ccoc12)=O)CO 79672,C1(CC)CN(C(C2(NC(=O)C(C3CC3)SC)CCN(C)C2)=O)CCO1 79673,CCC(CNC(=O)C(O)CCCNC(C1CCC(=O)CC1)=O)(CC)C(N)=O 79674,CCCCC(CC(=O)N1CCC=CC1CO)NC(C1(N2CCCC2)CC1)=O 79675,c1(C(N(C)CC2(CNC(=O)Cn3ncccc3=O)CC2)=O)cc2scnc2[nH]1 79676,c1(C(N(C(C)C)CCNC(c2cnn(C3CC3)c2Cl)=O)=O)cc(F)c(F)cc1Cl 79677,C1(CN(C(c2c(CC)ocn2)=O)C)CCCCN1C(c1ccn(C(F)F)n1)=O 79678,C1(NC(=O)CC23CCCC2C3)COCCN(C(c2cn(CC3CC3)nn2)=O)C1 79679,N1(CC(=O)NCc2c(CNC(C3C(CC)OCC3)=O)nco2)CCC(C)(C)CC1 79680,C(=O)(CC(F)(F)F)NC(C)C(=O)NCCCN(C(C1(OC)CC1)=O)C1CC1 79681,CN1CCC(CC(=O)N2CC3(NC(c4csc(Cl)n4)=O)CC2C3)c2ccccc21 79682,c1(C23CC(C(N(CCC)CCNC(C4CCN4CC)=O)=O)(C2)C3)ccc(F)cc1 79683,C1(F)(CNC(c2cnc(S)[nH]2)=O)CCC(CNC(=O)C(O)C2CCC2)CC1 79684,C(CCF)(C(=O)N1CC(F)(CF)C1)NC(CN1C(C)CCC1)=O 79685,c1(OC)cc(N)c(C(N2CC(NC(c3cnn(C)n3)=O)C2)=O)c(F)c1 79686,c1(NC(C)=O)ccc(C(=O)NC2CC(CNC(C3C(C)CC3C)=O)C2)cc1 79687,c1(C(=O)NC(C2CCCC2)CNC(CCSCC(N)=O)=O)cc2cccnc2[nH]1 79688,C1(NCCC2(C3CCN(C(=O)OC(C)(C)C)C3)CC2)CC(=O)N(CC(F)(F)F)C1 79689,C(c1ccc(C(F)F)o1)=CC(=O)NCCC(C)NC(c1cc(Cl)c[nH]1)=O 79690,C1(NC(c2c(C)ncn2O)=O)CCOC2(CCN(C(c3cnc(O)s3)=O)CC2)C1 79691,C=CCCC(C(=O)N1CCCC(C(=O)NC)C1)NC(C1CCCSC1)=O 79692,c1(CNC(C2CCSC2)=O)ccc2c(c1)CN(C(C1CCCC(CF)C1)=O)C2 79693,C=CCC(C(=O)N(C1(NC(c2ccc(-n3cccn3)nc2)=O)CC1)C)C(C)C 79694,C(=O)(CC(C)(C(F)(F)F)N(C)C)OC(c1ccc(F)nc1)C 79695,c1(CC(=O)Nc2cc(Br)ccc2OC(F)(F)F)c[nH]c2cc(Cl)ccc12 79696,O=S(=O)(c1ccc(Br)c(Cl)c1)N1CC2(CN(Cc3cnc4ccccn34)C2)C1 79697,c1(CNC(c2n(C)nnn2)C2CC(C)(C)C2)cncc(C(C)(F)F)c1 79698,c1(CC(=O)N(CCN(C(CC=C=C)=O)CC)CC)c(OCC)cccc1Cl 79699,N1(C(C=CC=CCC)=O)CC(CNC(c2cc3ccsc3s2)=O)C2(CCC2)C1 79700,C(C(CC(=O)N(C1CCOC1)C)NC(=O)Cc1cc[nH]n1)OC 79701,N(C1CN(C(=O)CC2CC3CC3C2)CCc2ccccc21)C(=O)C=CC(F)(F)F 79702,c1(OC)ccc(CC2CCN(C(c3ccccc3)=O)CC2)cc1C(F)(F)F 79703,c1(C(=O)ONC(=O)N(C(CC)COCC2CCCC2)C)cccc2ncoc12 79704,C12(NC(CCOCC#C)=O)CCCC1N(C(c1cc(C(N)=O)ccc1C)=O)CC2 79705,C1(CC(=O)NCCC2CC(C(=O)NC(C(C)C)C3CC3)C2)COCC1O 79706,c1(C(N(CCNC(CCN(CCCCC)C)=O)C(C)C)=O)nccn1C 79707,C1(COC)(NC(=O)C=CCN2CCOCC2)CCN(C(=O)CS(N)(=O)=O)C1 79708,C1(CNC(C2(C3CC3)CCC2)=O)CC(NC(C2(CCOC)CC2)=O)C(O)C1.OC 79709,C1(CNC(=O)CC2CCC3CC23)(NC(=O)CSc2cccc(O)c2)CCOCC1 79710,CCC(C)C(C(=O)N1CCCCC1CCO)NC(c1cncn1C)=O 79711,c1(OC)cnc(NC(C2C3CCC(C3)C2CNC(=O)OC(C)(C)C)=O)c(F)c1 79712,C1(NC(C2CNC(=O)O2)=O)C2CC1N(C(C13CCCCC1C3)=O)C2 79713,C(=O)(C(C)CC(C)(C)C)NC12C(NC(C(C(CC)O)C)=O)CC(CC1)C2 79714,c1(CCNCC2C(c3ccc(C(=O)OC)cc3)C2)ccc(F)cc1Cl 79715,N1(C(C(CCC)NC(c2ccc(C#C)cc2)=O)=O)CC(C)(C)CCC1C 79716,C1(C(N(CCNC(c2cn(CC(F)(F)F)nn2)=O)C2CC2)=O)CCC2(CCC2)O1 79717,C12(C(=O)NCC3N(C(CC4C(CC)C4)=O)CC(F)C3)CCCN(CCC1)C2 79718,C1(NC(C2CC(=O)NC2)=O)CCCCN(C(c2cccnc2Cl)=O)C1 79719,Cc1ccncc1C(C)NC(c1nc(CNC(c2cc(C)c(C)[nH]2)=O)oc1C)=O 79720,N1(C(=O)NCCOCCCC)CCC(CC#N)C(F)(F)CC1 79721,c1(C(=O)NC2CN(C(Cc3ccn(CC)n3)=O)CC(C)C2)ccc(Cl)c(C)c1Cl 79722,C(=O)(C1=Cc2ccccc2C1)NCCOCCNC(CCC(C)OCC)=O 79723,c1(C(N2CCN(C(c3c(C)nsc3)=O)CC2C#N)=O)ccc(Cl)c2[nH]ccc12 79724,Cc1n[nH]cc1C(=O)NC(C)CCN(C(=O)CC1(O)CCOC1)C 79725,C1(C(N(C2CCN(C(C(CN(C)C)(C)C)=O)C2)C)=O)CC2CCC(C1)N2C 79726,c1(CNC(C2C3CN(C(C(C)Cc4ccco4)=O)CC32)=O)cc(F)ccc1[N+](=O)[O-] 79727,c1(C(=O)NC(CNC(c2c(Cl)ccc(OC)n2)=O)CO)cccc2c1CCO2 79728,c1(CNc2c(CC(=O)Nc3c(CC)scc3)cccc2)ccc(Br)cc1[N+](=O)[O-] 79729,C1(NC(C(C)(C)n2cc(Cl)cn2)=O)CCC(O)CN(C(C2CC2(F)F)=O)C1 79730,C1(S(N)(=O)=O)(C(=O)NCC2N(C(c3cc(OC)ncc3)=O)CC(O)C2)CCC1 79731,C(=O)(C(C(=O)N1CC(O)(C(C)NC(=O)CCCCC(C)=O)C1)C(C)(C)C)OCC 79732,Cc1cc(C(=O)NCC(O)CNC(=O)C(C)CS(C)(=O)=O)c2occc2c1 79733,c1(C(=O)NCC(C)(C2CCC2)NC(COCCC=C)=O)c(C)ncn1O 79734,c1(CC)nc(C(N2CCC2NC(C2CC(c3cccnc3)C2)=O)=O)c(C)o1 79735,c1(SC)cc(C(=O)Nc2cccnn2)co1 79736,N1(C(c2c(CC)nc[nH]2)=O)CCN(C(c2c[nH]cc2Br)=O)C2(CC2)C1 79737,C1(NC(CCOCCOC)=O)CS(=O)(=O)CC1NC(c1cc(OC)ns1)=O 79738,C(=O)(CCC(C)(C)F)NC(C1OCCN(C(c2nc(C)n(C)n2)=O)C1)C 79739,N1(C(C(C)SCC)=O)CC2(CC(NC(c3ccc(SC)o3)=O)CO2)C1 79740,c1(C(=O)NC2CCCN(C(CSCC#C)=O)C2C)ccc2c(c1)N(C)C(=O)CO2 79741,C1(C(N(C(CNC(=O)C2=CC(C)(C)C2)C2CC2)C)=O)CCCN2CCCCC12 79742,Cc1cc(C(=O)NCCC(C)NC(=O)C(F)Oc2ccc(Cl)c(F)c2)cc(O)c1 79743,c1(C(=O)NCC(C(C)C)NC(C2CCCOCC2)=O)n[nH]c2c1CN(C)CC2 79744,CCC(CC(=O)NC1CC=C(C(=O)NCC2CC3(CCC3O)C2)C1)C(F)F 79745,N1(C(C(CC)(C)F)=O)CCC(C2CCN(C(c3cc(C)cc(C)c3N)=O)C2)CC1 79746,N1(CCC)CC(C(=O)NCCCCN(C(=O)CC2CC2(Cl)Cl)C)CC1=O 79747,c1(C(=O)NC2C(NC(C3(C)CC3)=O)COC2)ccnc(OC2CCOC2)c1 79748,N1(C(C)CNC(C2CCCCO2)=O)CCN(C(c2ccncc2Cl)=O)CC1 79749,C1(C(=O)NC2C(C)CN(C(c3ccn(C4CC4)n3)=O)C2)CCCC(C)(C)C1 79750,N(C(=NCCCCl)NCC(Cc1ccccc1F)CO)CCN1CC(=O)NCC1 79751,C1(NC(C2(CC)CCC2)=O)CN(C(c2ccc(=N)[nH]n2)=O)CC1C 79752,n1(CCC)ccc(=NC(=O)C2(F)CCCN(C(C34CCC(C3)C4(C)C)=O)C2)[nH]1 79753,c1(COC(C(=O)N(C(C)CN(C)C(c2sccc2F)=O)C)C)ccc(Cl)cc1 79754,N(C(=NCC1(C)CCCC(=O)N1)N(C)Cc1ccc[nH]1)C(CC)C 79755,C=C(C)C1CN(C(=O)C(=O)NCCN(C(=O)C(C)OCCOC)CC2CC2)CCO1 79756,N1(C(C(CCCCCC)C)=O)CCC2(CC1)COC(CNC(C1CCCS1)=O)C2 79757,c1(C(N(CCC[Si](C)(C)C)C)=O)ccn2ncc(Br)c2c1 79758,c1(OC)cnncc1C(=O)N(C)CC1CCN(C(C2CCN(C)C2)=O)C1 79759,C1(NC(C2CC(O)(CC#C)C2)=O)CN(C(c2cn(C)nc2C)=O)CC2CCCC12 79760,c1(SC)ccc(C)c(NC(=O)NCC2(O)CCS(=O)(=O)C2)c1 79761,C#Cc1ccc(CC(N2CCC(CC(=O)NCCCOCC(C)C)C2)=O)cc1 79762,CCCCCCCCCC(O)CC(=O)N1C2CC1CN(C(=O)C(O)C(C)CC)C2 79763,C(C(=O)N(CCOCCO)CC1CC1)(C1CC1)OC.C1(=O)C(C)ON1 79764,CC1(c2cccc(F)c2)CCN(CC(c2ccccn2)N2CCCC2)C1.C12CC1OC2 79765,C1(C(N2C(CC(=O)NCc3cnc(CC)s3)CCCC2)=O)C2C3CCC(C3)C12 79766,C=C(C)CCC(C)N=c1[nH]c(=NCc2ccc(N)cc2)c2ccc(C)cc2[nH]1 79767,c1(C(=O)NC(C2CCOC2)C)cc2occc2[nH]1 79768,c1(-c2ncc(C(=O)NCC(CO)NC(c3cccs3)=O)s2)ccccc1Cl 79769,C(=O)(CCCC1CC1)N(C(C)(C)CNC(=O)COCCCF)C 79770,c1(C(=O)NCCCNC(C(=CC2CCC(C)CC2)C)=O)ccc(Cl)c2occc12 79771,C(=O)(C(C)(C)C(=O)NCc1nc(C(=O)NOCC(F)F)c(C)o1)NC 79772,N1(C(CC(C)C2CC2)=O)C2CCC1CC(N(C(=O)C(C)(C)C1CCC1)C)C2 79773,N1(C(c2c[nH]nc2C2CC2)=O)CCN(C(C2(C3CCC3)CC2)=O)C2CCCC12 79774,CC1CCC(CC(N2CCCC(CN(C)C(c3nnn(C)n3)=O)C2)=O)CC1 79775,C1(NC(c2cc(C)cc(Cl)c2)=O)CS(=O)(=O)C2CN(C(C3CSC3)=O)CC12 79776,N1(C(COC2(C)CCC2)=O)CCC(C2(NC(=O)Cc3ccc(F)cc3)CC2)CC1 79777,c1(NC(C2CCC(C#C)C2)=O)ccc(F)cc1Cl.C1(=O)CCO1 79778,Cc1cnc(NC(C2CN(C(=O)C(Cl)(Cl)Cl)CCC2O)=O)c(C)c1 79779,C1(C(=O)NCCN(CCC)C(c2ccc(C)c(C)n2)=O)(CC)CCC(O)CC1 79780,CC1CN(C(C2CCC(C)(C)N(C(=O)C(C)(O)C3CCC3)C2)=O)Cc2c[nH]nc21 79781,N1(C(CC(CC)O)=O)CCN(C(c2ocnc2C(F)F)=O)CCC1C 79782,c1(CCCC(=O)NCC(C)CN(C(=O)CN2CCC2)C)ccc(F)cc1 79783,c1(OCCOC)ccc(C(=O)N(C)CCNC(c2ccsc2C)=O)cn1 79784,C1(O)(CCNC(c2cccc(CS(C)=O)c2)=O)CCN(C(C2CCCC2)=O)CC1 79785,CCCC(C(=O)NCc1ncccc1C(=O)N(c1cnn(C)c1)CC)NC(N)=O 79786,C(=O)(CC(C(F)(F)F)NC(C12CCC(CC1)C2)=O)N(c1cnc(C2CC2)nc1)C 79787,N1(C(CCN(CC#C)C(c2ccn(CC)c2C)=O)=O)CCOC2COCC12 79788,Cc1ncc(Cl)c(-c2nc(C3CC3c3cncn3C)no2)n1 79789,C1(C(=O)NCCN(C(=O)CC2CC(=O)C2)CC)CC(n2cnnc2)C1 79790,N1(C(C(=O)NCCNC(C)=O)=O)CCN(C(c2coc(O)n2)=O)CC1 79791,c1(C=O)cccc2c1cnn2C.C12CN(CC1(F)F)N(CC)C2.C1(C)(CO)CC1 79792,N1(C(C(CCOC)C)=O)CCC(NC(C2CCN2C)=O)C12CC2 79793,N1(C(C2(SC)CC2)=O)CCCCC12CC(NC(C1CSC(C)=N1)=O)C2 79794,C1(C(=O)NC2CCN(CC)C2)CCN(C(=O)c2cccn2C2CC2)O1 79795,C12(NC(COCCOC)=O)CC(C)(C1)OC21CN(C(c2cc(C)c(C)cc2C)=O)C1 79796,C1(CNC(CCCCN(C(C)C)C)=O)CCC2(CCN(C(=O)C3CC3)CC2)CO1 79797,C1(C)(C(=O)NC(C)CCO)CCN1C(=O)COc1ccccc1 79798,CCCC(C(=O)NC1(c2ccsc2)CC1)NC(c1cscc1OC)=O 79799,C1(OCCNC(C2CC(OCC)C2)=O)CCN(C(=O)C(C)=C2CCC2)CC1 79800,c1(CNC(C=CC2N(C(C(CC)CN(C)C)=O)CCC2)=O)ccc(F)cc1F 79801,C1(NC(CNC(=O)OC)=O)CCOC12CCN(C(c1cc(=O)n(C)o1)=O)CC2 79802,Cn1cccc1-c1cn(CCCC(=O)NCC(O)Cn2cccn2)nn1 79803,Cc1nnc2cc(NCC3CCCC(CNC(C4(NC(N)=O)CC4)=O)C3)ncn12 79804,N1(C(C(CC)O)=O)CCC(n2cc(NC(=O)CSc3nc[nH]n3)nn2)CC1 79805,CCC(F)(F)C(C)(C)C(=O)N1CC2CCC1CN(C(c1[nH]nnc1C)=O)C2 79806,N1(C(COC(C)=O)=O)CCC2C1CCCN2C(=O)C=Cc1ccccc1[N+](=O)[O-] 79807,C12(N3CCN(c4c(C#N)ccnc4)CC3)COCC1CN(C(=O)CCC(N)=O)C2 79808,c1(C(C(=O)Nc2ccccc2)N(C(C(=O)NCC)CC)C)cc(C)nn1CC 79809,c1(C(=O)NCCCC(=O)NC(CC(=O)OCC)C)cccc(C)c1O 79810,c1(C(N2CCC(C(C)(C)C)(CNC(CC3(OC)CC3)=O)C2)=O)cc(C)nc(C)c1 79811,C1(CNC(c2c(C)cc(CC)o2)=O)CN(C(c2scnc2Cl)=O)C2CCCC2O1 79812,C(CCCCC(=O)NC(C)C(C(C)C)NC(C1CCSCC1)=O)OC 79813,O=C(CC1COCc2ccccc21)NCCC1CCN(C(=O)Cn2cnnc2)C1 79814,c1(C(=O)NCC2(COC)CN(C(C3C(C)(CC)C3)=O)C2)c(C)nc(C)n1O 79815,c1(C(=O)NCC2C(NC(=O)Cn3cncn3)C2)c[nH]cc1C1CC1 79816,C1(C)(CC)CCCN(C(C2(CNC(c3cnc(C4CC4)o3)=O)CC2)=O)CC1 79817,C1(CNC(=O)C(=O)NCc2cccc(OC3CCCC3)n2)CCC=CCCC1 79818,C1(NC(=O)COC(c2ccc(-n3cc(Br)cn3)nn2)=O)C2CCCOC12 79819,C1(OC(C2(CNC(COC(CC)(C)C)=O)CC2)=O)CCCC(CO)C1 79820,Nc1ccnc(C(=O)NCC2CCC2NC(c2scnc2C(F)(F)F)=O)c1 79821,C=C(C)CCCN=c1c(Br)ccc(I)c2ccccc12 79822,C1(C(N2C(C3CCN(C(CC=C)=O)C3)CCCC2)=O)CCC(=C(F)F)CC1 79823,C1(NC(C2C(CNC(c3c(CC)oc(C)c3)=O)CCC2)=O)CC2CC1C(O)C2O 79824,C1(CNC(C(CCCC)O)=O)CCC12CCN(C(c1cnc(C)[nH]1)=O)CC2 79825,N1(C(C=CC2N(C)CCC2)=O)CCN(C(c2cc[nH]c(=N)c2)=O)CC1CC(F)F 79826,C1(CC(=O)N(CC(=O)N(C)Cc2ncc[nH]2)C2CC2)CC1C1CC1 79827,C1(NC(CC(C)c2ccco2)=O)CN(C(c2cn(C)nc2O)=O)CCC12CCC2 79828,CC1CN(C(c2cn(C)c(=O)n2C)=O)CCC1NC(C1(CO)CCCC1)=O 79829,C12(CCC1)CCN2.C1(CC(=O)OC)CN(C(=O)CSc2nc[nH]n2)C1 79830,CCC(O)C(C)C(=O)N(C1CCN(C(C2CC(CN(C)C)C2)=O)CC1)CCOC 79831,C1(NC(C2CC2(F)Cl)=O)CC2CC1CC2C(=O)NC1(CF)CC1 79832,CC(O)C(C(=O)NCCC1CCCN(C(c2csc(Cl)n2)=O)C1)N(C)C 79833,C1(NC(C(CC=CC)C)=O)CC12CCN(C(c1cc(C#N)cn1C)=O)CC2 79834,c1(CCC)ncc(C(=O)NC2CCC(NC(=O)CSc3nncn3C(C)C)C2)s1 79835,C(=O)(C#CC1CCOC1)N1CCCC(N(C(Cc2nc(C)c(C)s2)=O)CCO)C1 79836,C12(NC(COCCOC)=O)CCCCCC1N(C(C1CCCCC(C)(C)C1)=O)CC2 79837,c1(NC(C(C(C)C)NC(=O)Cc2ccns2)=O)ccc(F)cc1CO 79838,c1(C(=O)NCC(C)N(C(c2ccc(N)c(O)c2)=O)CC)ccc2c(C)[nH]nc2c1 79839,C1(C(N(C)CC2(O)CCN(C(Cn3c(C)csc3=O)=O)C2)=O)C2CCC(F)(F)C12 79840,c1(CNC(=O)NC2CC(C(N)=O)OCC2)cc(O)cc(Br)c1 79841,CC1COc2ccc(C(=O)NC3CCC3NC(=O)CCCc3ccsc3)cc21 79842,c1(CC)cc(C(F)F)c(C(=O)NCC2(F)CC(NC(=O)CC3(CC)CC3)C2)cn1 79843,C1(CNC(C2C(=C)C2)=O)(CO)CN(C(=O)C(C)C2CCCC2)C1 79844,C1(CC(N2CC(O)(CN(C(=O)C(C)(C)C3CCOC3)C)C2)=O)OC(C)(C)OC1=O 79845,C(=O)(C(C)C(O)CC(C)C)NCC(C)(C)OCC(=O)NCC1CC(OC)C1(C)C 79846,C(=O)(C1=C(C)OCCS1)N1C(CCNC(=O)CC(C)CN(C)C)CC(OC)C1 79847,C1(C(=O)NC(CNC(CNS(CCCOC)(=O)=O)=O)CC)CC2(C1)CC21CCC1 79848,C1(CC=C)(NC(=O)CC2CCCC2C)CCCN(C(c2cc(O)ccc2O)=O)C1 79849,n1(CCOC)cc(C(=O)NCCN(C2CCCCC2)C(C2CCCCC2)=O)cn1 79850,C1(CCC)COCCN1C(=O)C(C)C(C)NC(=O)C=C(C)C 79851,C1(NC(c2ncc(F)cn2)=O)CN(C(C2CN3CCC2CC3)=O)CC12CCCC2 79852,C1(CNC(CC(C)C)=O)CN(C(C2CCN(C)CC2)=O)CC(C(F)(F)F)O1 79853,C1(SCC(=O)NC2(C(=O)NC(C(=O)OC)CO)CC2)COC(=O)N1C 79854,C1(NC(=O)NCC(C2CCCO2)O)CC12CCS(=O)(=O)CC2 79855,N1(C(C(C)C2CC2)=O)CCCC12CCN(C(C1CCOC1)=O)C2 79856,C1(NC(Cc2ccc(C)nc2)=O)CC2CC(C1)N(C(=O)CCc1ccco1)C2 79857,c1(C(=O)N(C2(C=C)CC2)C2CC2)noc2c1CCC2 79858,C1(NC(C(COC)(C)C)=O)CCC2(CCCN(C(=O)C(C)(C)N=[N+]=[N-])C2)C1 79859,N1(C(CCCCCC)=O)CCN(C(=O)Cc2cccc(C#N)c2)C(C)CC1C 79860,Cc1[nH]nc2cc(C(N3CCOCC(NC(=O)C(C)C4=CCCC4)C3)=O)ccc12 79861,C1(CNC(C2CC2F)=O)COCCN1C(c1cccc(CC2CCCO2)c1)=O 79862,c1(C(=O)NC(C(CCC)O)CO)cc2[nH]nnc2cc1OC 79863,C1(C(N(C(CCSC)C)C)=O)CC(=O)CN1C(c1cc[nH]c1C)=O 79864,N1(C(CN2CC(C)C2)=O)CCCC(n2cc(CNC(C3CC3(C)C)=O)nn2)C1 79865,CCCCCCC(O)CCC(=O)NC1(C)CCCN(C(=O)CC2OCCO2)C1 79866,N1(S(CCC)(=O)=O)CC2CN(C(c3cc4n(n3)CCC4)=O)CC2C1 79867,C(=O)(C1SCc2cccnc21)NCC1(O)CCN(C(c2nccc(N)c2)=O)C1 79868,C1(NC(=O)OC(C)(C)C)CCN(CCc2nc(-c3ccccc3Cl)no2)CC1 79869,CN=c1ccc(C(=O)NCCCN(CCO)C(c2csc(CO)n2)=O)c[nH]1 79870,C(=O)(C(C)S(=O)Cc1nnnn1CC(C)C)N(c1ccccc1OC)CC 79871,N1(C(C(CCO)N(C)C)=O)CC(C2CCN(C(C3CC3(C)C)=O)CC2)C1 79872,N(C(=NCc1cc(C)on1)N(C)Cc1cccc(Cl)c1)CC(=O)NCC 79873,CC1(NC(c2cc(-c3ccoc3)[nH]n2)=O)CCCN(C(=O)CC2CCC(=O)N2)C1 79874,CCS(=O)(=O)CC(=O)NCC1C(C(=O)Nc2ccc(O)c(C(N)=O)c2)C1(C)C 79875,Cc1cnc(N2CCC(CNC(=O)C(C)C(C)(C)C)C2)nc1S(C)(=O)=O 79876,c1(C(=O)NC2CN(Cc3ccc(Br)nc3)CC2F)ccnc(Cl)c1Cl 79877,c1(C(=O)NCC(CC=C)NC(=O)Cc2cc(C)cc(C)c2)cc(OC)ccc1C 79878,C(=O)(C1=CCCS1)N1C(C)CCC1.C1(CC(=O)N(C)C)(C(=O)OC)CC1 79879,c1(C(=O)NCCC(C)NC(CCc2c(C)cccc2)=O)c(C)cc(O)nc1C 79880,Cc1cc(F)ccc1N(C(c1csc(-c2cnn(CC3OCCO3)c2)n1)=O)CCBr 79881,N1(C(CNC(=O)OCC=C)=O)CCC(NC(=O)CC(C)(C)CC)C(C)C1 79882,C1(C(N(CCOCCOC)C)=O)CCCC1CNC(C1CS(=O)(=O)C1)=O 79883,C1(C(=O)NC(C)CC2CN(C(c3cc(Cl)ccc3F)=O)C2)Cc2ccccc2N1 79884,c1(C(N2C(C(=O)NC3C(CC=C)COC3)C3CC3C2)=O)ccc(C#N)cn1 79885,C12(CNC(Cc3c(C)cccc3F)=O)CCCC(CN1C(c1ccn(C)c1)=O)C2 79886,C(=O)(C(F)CCC(C)(C)C)N1CCN(C(CCCC#C)=O)C(CCO)C1 79887,C=CC1(C(=O)NC(C2CCCCC2)CNC(=O)Cc2n[nH]c(C)n2)CCCC1 79888,C1(CC(=O)NCc2cc(C)ncn2)CCCN(C(c2cc(C3CC3)on2)=O)CC1 79889,c1(C(=O)NCCOC2CN(C(C(C(=O)OC)C)=O)C2)ccc2nccn2n1 79890,c1(C(=O)NC2CC(NC(C3COCC(C)(C)O3)=O)C2)c[nH]c2c(C#N)cccc12 79891,C(=O)(C(C(C)C)n1cnnc1)NC1C(NC(CC(OCC)OCC)=O)CC1 79892,N(C1CCCc2c(C)cc(C)cc21)CC(CCC)CO 79893,c1(C(N2CC(C)C(NC(=O)Cc3cccc(O)c3)C2)=O)cc2cccc(Br)c2[nH]1 79894,C1(C)(CC)C=C(C(=O)NC(C)CC2CN(C(=O)C(O)Cc3ccccc3)C2)C1 79895,C1(OCC)CC(C(=O)NC)N(C(c2cnc(C)s2)C(=O)NC2CCCC2)C1 79896,Cc1ncncc1C(=O)NC1CN(C(c2occc2CN(C)C)=O)CC1F 79897,C(CC1=CCN(C(C2CC23CC(C)(C)C3)=O)CC1)NC(CCCC(=C)C)=O 79898,N1(C(C(C)CC(F)F)=O)C2CCC1CN(C(C1(O)CCCC1)=O)C2 79899,c1(C(C)C)ccc2cc(C(=O)NC(C3COC(C)(C)O3)C3CC3)[nH]c2c1 79900,c1(C(=O)NCC2N(C(C3CCCC(OC)C3)=O)CCC2C)cccn(C)c1=O 79901,CCC(CC)C(C(=O)N1CCCC1C(C)NC(c1nncn1CC)=O)OC 79902,C1(NC(c2ccc(CC)[nH]2)=O)CCCC(N(C(=O)CCCc2cccnc2)C)C1 79903,n1(CC(C)C)cc(NC(c2ccn(C)n2)c2nnnn2Cc2cccs2)cn1 79904,c1(NC(C2C(NC(=O)COCCc3cc[nH]n3)CCC2)=O)cccc(F)c1F 79905,c1(N(C)C)ccncc1CNC(C1CCCC1NC(=O)CC(C)(C)N(C)C)=O 79906,C1(C(C)C)CCc2[nH]nc(C(=O)NC3(CNC(=O)C(O)CCN(C)C)CC3)c2C1 79907,CC1(C)CN(C(c2csc(C(F)F)n2)=O)C(CNC(C2(Cl)CC23CCC3)=O)CO1 79908,C(C(CO)(CO)NC(C1CCN1S(C)(=O)=O)=O)N(C(c1nc(CC)sc1)=O)C 79909,C12(NC(COCCSC)=O)CCCC1CN(C(=O)C(=O)NCC1CC1)C2 79910,N1(C(C(C)(C)n2cncn2)=O)CCC(C(=O)N2CCCC2C2CCOC2)=C(F)C1 79911,N1(C(CSC)=O)CC2CCC2(CCNC(=O)C(C)(C)Nc2ccccn2)C1 79912,N1(C(=O)C=Cc2ccncn2)CCN(C(C2(O)CC2)=O)CC(O)C1 79913,C(=O)(CC(C)CNC(C1(C2CCCN2C(c2nc[nH]n2)=O)CC1)=O)OC 79914,C1(C(NOCCCCC)=O)CC(C)CN1C(=O)C(=O)NOC 79915,Nc1cc2[nH]cnc2cc1C(N1CCC(NC(=O)Cc2csc3cncn23)C1)=O 79916,C(C(O)CC(=O)NCCC1(C)CCOCC1)NC(C(C)OCC=C)=O 79917,C(=O)(C(C)(O)CCC)NC(CN(C(c1c(CC)nccc1)=O)C)CC 79918,C1(C(=O)NC2C(C#N)CCCC2)CN(C(c2cc3ncccc3[nH]2)=O)CCC1(F)F 79919,C(=O)(C1=CS(=O)CCC1)N1CCC(NC(c2cn(C(F)(F)CO)nn2)=O)C1 79920,N1(C(c2c(C(C)C)con2)=O)CC(CCNC(C2CC(=C3CC3)C2)=O)OC(C)C1 79921,C12(NC(C(N)=O)=O)CCCC1N(C(c1cnc(-c3cccnc3)s1)=O)CCC2 79922,C(=O)(C1CCc2cc(Br)ccc21)NCCn1cc(C2CCCN(C)C2)nn1 79923,Cc1scc(C(N2CC3C(CNC(c4ccoc4C4CC4)=O)C3C2)=O)c1N 79924,c1(NC(CCn2cc(C(CCC)CC)nn2)=O)ccc(=N)[nH]n1 79925,c1(C(C(c2n(CCCC)nnn2)NCc2csc(C)c2C)(C)C)cccc(F)c1 79926,Cc1cc(C(N2CCC3(CC3C(=O)Nc3cccc(Cl)c3O)C2)=O)ccc1O 79927,C(C(=O)NN1CCCC1C(N1C(C)CCC1C)=O)c1c(C)n[nH]c1 79928,C(=O)(C1CCCc2ccccc21)NC(C1N(C(Cc2cnc(C)[nH]2)=O)CCC1)C 79929,c1(C(N2CC(O)(C(C)NC(C3CCCN3C)=O)C2)=O)ccccc1Br 79930,C1(NC(C(Br)=C(C)C)=O)CC2CCC1N(C(C1(O)CCC(C)CC1)=O)C2 79931,c1(C(N(C)Cc2c3ccccc3nn2C)=O)cc([N+](=O)[O-])c2nsnc2c1 79932,Cc1cc(CNC(C2(C)C=CCN2C(=O)CS(C)(=O)=O)=O)ccc1F 79933,N1(C(C2CCCC(C)(C)C2)=O)Cc2nccn2CC(NC(c2ccns2)=O)C1 79934,c1(OC)cc(Br)c(C(=O)NC2CC2CNC(=O)CC(F)F)cc1F 79935,N1(C(c2ccn3cncc3c2)=O)CCCC2(CCCN2C(=O)CCCCCO)C1 79936,C1(NC(C2CC=C(C)CC2)=O)CCN(C(c2ccncc2Cl)=O)C(C)C1 79937,c1(C(=O)NCCCC(C)NC(C2(OC)CCOC2)=O)cccc2cc(F)ccc12 79938,N1(C(C(C)=C(CC)C)=O)CC(F)CC1CNC(=O)COc1ccccc1Cl 79939,CC(C)C(C)(C)C(=O)NCCCNC(C1(C(F)(F)F)CC(O)C1)=O 79940,c1(C2C(C(N3CC(c4cn(CC(C(=O)OC)O)nn4)C3)=O)C2)ccccc1F 79941,CC1CCN(C(C2CC(=O)N(O)C2)=O)CCN1C(c1cc(-c2ccco2)[nH]n1)=O 79942,c1(SCC(N2CCC(OCC(=O)NC3CC4CC3C4)C2)=O)nc2ccccc2[nH]1 79943,c1(C(=O)NCCN(C(CCc2onc(C(C)OC)n2)=O)C)cnncc1O 79944,C1(NC(C(C)OCCCC)=O)CC2CN(C(=O)CNC3(CO)CCCC3)CC12 79945,Cn1nc(Br)c2c(NC3CC(=C4CC4)C3)ncnc12 79946,c1(CC=C)ncccc1NC(=O)NC1CCN(C2CC2)C1=O 79947,N1(C(=O)NCC(CC2CC(F)(F)C2)OC)CCC2(CC1)OCCO2 79948,N1(C(CCc2onc(C)n2)=O)CC2(C1)C(NC(=O)CC(C)C(F)F)CCS2(=O)=O 79949,c1(C(CC)NC(=O)C(c2ccccc2OC)O)ccc(OC)c(Cl)c1 79950,n1(CCC(=O)NCC2CCN2C(c2cnns2)=O)c(S)nc2ccccc2c1=O 79951,c1(C(=O)NCc2cc(C)c(C(N3CC(F)C(F)C3)=O)o2)cc2ccncc2[nH]1 79952,O=C(C1=CC2CCC(C1)C2)N1CCC2(CC1)CN(C(c1ncccc1F)=O)C2 79953,c1(C(C(N2CCCN(C(CC(C=C)(C)C)=O)CC2)=O)O)cccc([N+](=O)[O-])c1 79954,CC(O)C(C(N)=O)NC(=O)COC1CCN(C(=O)CCC2CCOCC2)C1 79955,C1(C(N(C)CC2CN(C(c3cc(CN(C)C)ncc3)=O)C2)=O)CC2C(C1)C2(F)F 79956,C1(C(N2CC(CC)C(NC(=O)COCCN(C)C)C2)=O)CC2C(C1)C2(C)C 79957,O=S(=O)(c1cccnc1NCCCN1CCC(O)CC1)NCCC1CC1(F)F 79958,c1(SCC(=O)NC(CCN(C(C(CC)F)=O)C)C)ccc(F)c(F)c1 79959,Cc1cc(C(N2CC(NC(=O)CC3(C)CCCC3)C3(CC3)C2)=O)nc(O)n1 79960,N1(C(C2N(C)C(=O)C(F)C2)=O)CCS(=O)(=O)CC1C1CC1 79961,c1(OC)ccccc1C1CC1NC(c1n[nH]cc1NC(c1ncc(Br)cn1)=O)=O 79962,C1(NC(C2ON=C(C)C2)=O)CCCCC1NC(C1(C(N)=O)CCC1)=O 79963,Cc1nc2ncnn2c(C)c1C(=O)N(CC(C)(C)NC(=O)CC1CC(F)(F)C1)C 79964,C(c1cccc(Cl)c1)=CC(=O)NC(CC)CNC(C1CC=CCC1C)=O 79965,N1(c2ccnc(C(=O)OC)n2)CCC(C)(NC(=O)CSC2CC2)CC1 79966,c1(N2C3CC(CNC(C4CCS(=O)(=O)N4)=O)CC2CC3)nc2ccc(Br)cc2s1 79967,N(C1CCOc2c(C)ccc(C)c21)C(=O)NC(CC#C)C 79968,CC(c1ccsc1)=CC(=O)NCC1CC(NC(=O)C(C2CCCCC2)F)C1 79969,C1(NC(CN2CCN(C(C(C)CO)=O)CC2)=O)CCCC2(CCC2)C1 79970,N1(C(c2n(C)ncc2Cl)=O)CCCCC2C1CCCN2C(=O)CC1CNC(=O)C1 79971,O=NN1CCCC1C(=O)NCCC1CCN(C(C2CC(CF)C2)=O)CC1 79972,n1(CC)nc(C)c(C(N2CCCC(N(C(=O)CC3(C#N)CCC3)C)C2)=O)c1Cl 79973,c1(NCc2c(C)nc(CC)o2)nccc(=NCC2(OC)CCCC2)[nH]1 79974,c1(C(=O)NCC(CO)NC(C(CC)OC)=O)ccc(N2CCOCC2)cc1 79975,Cc1c(C(=O)NCC2(NC(=O)CCSCC(N)=O)CCCC2)c(C(F)F)nn1C 79976,C#Cc1ccc(C(N2CC3CC3(C(=O)NCC3CC(SC)C3)C2)=O)c(C)c1 79977,N1(C(C2CC(=O)NC2)=O)CCCC(C2(NC(c3c(F)cc(F)cc3Cl)=O)CC2)C1 79978,CC1CC(NC(=O)Cc2nc(C3CC3)no2)C(=O)N1c1cnn(C)c1 79979,n1(C(C)C)cc(C(=O)NC(C)(CNC(C2CC=CC2)=O)C(C)C)c(Br)n1 79980,c1(CC(N2C3CC(NC(c4cc(Br)co4)=O)(C3)C2)=O)ccc2c(c1)OCO2 79981,c1(-c2nc(C(=O)NC(c3cccc(Br)c3)C(C)C)on2)cccc(OCC#N)c1 79982,CC(C)S(=O)(=O)CC(=O)N(CC(O)CNC(=O)CNC(c1cccc(O)c1)=O)C 79983,Cc1ccc(C(C)C)c(OC(C)C(N2CC(C)CC2CO)=O)c1 79984,CCC(C)C(O)C(=O)NCc1nc(CNC(c2ncccc2F)=O)cc(O)n1 79985,CCC(C)(CO)C(=O)NCC#CC(=O)NC1CCCCC1 79986,c1(-c2nc(CS(=O)(=O)NC)n(-c3ccc(OC)nc3)n2)cccn2ccnc12 79987,Cc1cnc(C(N2CCC(C(=O)NCCC3CCCCCC3)C(C)C2)=O)c(F)c1 79988,N1(C(c2cnc(CC)o2)=O)CCC(F)(C(=O)Nc2ccc(F)c(C)c2)CC1 79989,CCC(CC(F)F)C(=O)NC1CC(NC(C2NC(=O)CC2C(F)(F)F)=O)C1 79990,c1(C(=O)NC23CC(NC(CC4CC(C)OC4)=O)(C2)C3)cccc2ccn(C)c12 79991,CC(C)CC(O)C(C)C(=O)N(CCCCNC(c1cc2occc2n1C)=O)C 79992,N1(C(c2ccc(C)cc2)=O)CCC(C(N2CCC(OC3CCC3)CC2)=O)CC1C 79993,c1(C(=O)NC2CCC(NC(C3C(OC)CC3)=O)C2)nc(C(F)(F)F)cn1C 79994,c1(C(c2n(CCCCCC)nnn2)NCC2CC(CF)C2)cnn(CC)c1CC 79995,Cc1cc(C(N2CCN(C(C3CCCC(=O)O3)=O)C(CF)C2)=O)nc(O)n1 79996,c1(CNC(CC2(NC(Cn3c(C)nnn3)=O)CCC2)=O)cc(Cl)ccc1F 79997,C(CN1C(=O)Cc2ccccc21)NC(=O)NC1CCCC12CCNCC2 79998,C#Cc1cncc(C(=O)NCC2C3CN(C(c4cnc(OC(C)=O)s4)=O)CC23)c1 79999,N1(C(CC(=C)Br)=O)CC(NC(=O)CCCN(C)C(C)=O)CC1C 80000,C(=O)(C(O)C(C)(C)CC)N1CC(CCNC(=O)CN2CCC(C)(O)C2)(OC)C1 80001,C(CCCCCC(=O)NCC1CC(C)N(C(c2ncc(F)cn2)=O)C1)SC 80002,c1(C(=O)NC2CC3CC2N(C(=O)CC2CC2(Cl)Cl)C3)cc2n(n1)CCCCO2 80003,C1(NC(C)=O)CCN(C(=NCCCC2CCCCO2)NCc2cccs2)C1 80004,c1(CN(CCNC(=O)C(=O)Nc2ccc(Cl)cc2)C2CC2)ccccc1C#N 80005,C1(N(C(CCCOCCC)=O)C)CC2CCC(C1)N2C(c1occc1CC)=O 80006,C(CCCC(=O)NCCC(C)NC(c1n[nH]c(C2CC2)c1Br)=O)OCCC=C 80007,O=C(C#CC1CCCOC1)NC1(CNC(c2ccnc(S)c2)=O)CCOC1 80008,c1(OC(C)C)cc(N2CC3C(C2)N3C(=O)CCc2ccc(F)nc2)ncn1 80009,CN1CCN(CCC(=O)NCC2C=CCN2C(C2CC(O)C2)=O)CC1 80010,C1(F)(CNC(c2ncc(C)s2)=O)CCCN(C(C2(C(F)(F)F)CC2)=O)C1 80011,S(=O)(=O)(c1ccc(N2CC(C)c3ccccc3C2)nc1)NC1C(C=C)COC1 80012,c1(C(=O)NC2CCN(C(C(CCC)C#N)=O)C2)cnn2c(Br)cccc12 80013,C1(F)(C(N2CCC(c3cnc(Cl)s3)C2)=O)CS(=O)(=O)CC12CCC2 80014,C12CCN(C13CC3)C(=O)CNC2=O.C(C(C)CC(=O)NCc1ccco1)OC 80015,c1(C(N2CC3(C2)CN(C(C2(CF)CC2(F)F)=O)C3)=O)ccc([N+](=O)[O-])cc1 80016,c1(C(=O)NCC23C(CN(C(C(C(=C)Cl)(C)C)=O)C2)C3)cccc2c1ncn2C 80017,C1(C(=O)NC2CN(C(C(C)NS(CC)(=O)=O)=O)C2)(SC)CC(C(F)F)C1 80018,c1(NCC2CCCCN(C(C(c3ccc(C)s3)C)=O)C2)nc(Cl)nc2sccc12 80019,Cc1c(NCCCOCCC(C)C)ncnc1N1CCC(C)(F)C1 80020,c1(C(C)NCC=CC2(C)CCOCC2)cc2ccccc2[nH]1 80021,c1(C(=O)NC2CCCC(NC(CC(C=C)(C)C)=O)C2)cc2ccccc2nc1C 80022,c1(C(=O)NCC2N(C(C(C=C)(C)CC)=O)CC2)cc2ccc(OC)cc2[nH]1 80023,O=C(CCCCc1ccc(F)cc1)NCCC1CN(C(C2C3CC3C3CC23)=O)C1 80024,C1(NC(C2C(C(C)O)C2)=O)CCCN(C(c2cncn(C)c2=O)=O)CC1 80025,C1(NC(=O)CCc2ccccn2)CCN(C(c2cc(O)nc(Cl)c2)=O)CC1CO 80026,c1(C(=O)NC(CNC(C2C(C)C2)=O)C)nc(C2CC2)ncc1Br 80027,c1(CC(C)C)ncc(C(=O)NC2CC(CCNC(C3CC3C3CC3)=O)C2)s1 80028,c1(NC(c2c(Cl)ccc(Cl)c2O)=O)cc(Cl)cc2nc[nH]c12 80029,C1(C(C)C)C(NC(=O)CCC2CCOC2)CCN1C(=O)CCCN(C)C 80030,c1(C(N2CCN(C(C(CC)C)=O)C(C)C2)=O)oc2ccccc2c1CO 80031,n1(CC)cc(Br)c(C(=O)NC(C)CC(C)NC(c2scnc2Cl)=O)n1 80032,N1(C(CN(C(C)C)C)=O)CC(NC(c2ncn3c2CCC3)=O)C(C2CC2)C1 80033,C1(NC(C(c2cc(N)ccc2F)N(CCC)CCC)=O)CCC2CCC1O2 80034,N1(C(c2n(CC)ncc2)=O)CCCCC(N(C(=O)COCc2ccccc2)C)C1 80035,C1(C(=O)NC2CC(n3cc(C(C)(C)C4CC4)nn3)C2)CCC(C2CC2)C1 80036,C(C)(C)(CN(C(=O)C(C1(C)CC1)NC(=O)C(=O)NCC(F)F)C)OC 80037,c1(OCCOC)cncc(C(=O)NC2CCC(NC(C3CC=CC3)=O)C2)c1 80038,N1(C(CC2(COC)CC2)=O)CCOC2CN(C(C3CCSCC3)=O)CC12 80039,N1(C(c2cnc(OC)nc2)=O)C(CNC(c2cc(Br)c[nH]2)=O)CC2COCC12 80040,c1(C(N2C(CCNC(CCOCCOC)=O)CSCC2)=O)cnc2ccoc2c1 80041,c1(C(=O)OC)sc(NC(C2C(O)CCN2C(c2nccn2C)=O)=O)c(C#N)c1C 80042,CC(C)CCC(=O)C(=O)N1CCOC(C(=O)NCC(C)(C)CC(C)O)C1 80043,C1(C(N2C(CCCC)CCC2)=O)CC(C)CN(C(c2cc(C)cc(Cl)c2)=O)C1 80044,C=CC(C)(CC)C(=O)NC1CCN(C(c2c(C)ccnc2OCC)=O)C1 80045,C12(C(=O)OC)CCC(COCCN(CC(F)F)C)(CC1)CO2 80046,N1(C(C(C)(C)NC(=O)OC)=O)CCN(C(C)CNC(=O)Cn2ccnc2C)CC1 80047,C#CCCC(O)C(=O)N1CC(C2(NC(=O)Cc3ccc(CO)cc3)CC2)C1 80048,Cc1c[nH]c(-c2ncccn2)nc1=Nc1ccc(Cl)cc1N1CCOCC1 80049,C(=O)(CC(CC(C)C)NC(=O)COCC1CCC1)N1C(CC)C(O)CC1 80050,CCCCCCC(C)CC(=O)NC1COCC1CNC(C1(O)CCCCCC1)=O 80051,N1(C(C2(OC)CC(CF)C2)=O)CCC(C)(NC(C2(C#N)CCCO2)=O)C1 80052,CC(C(C)C(=O)N(C1CCNCC1)C1COC1)Nc1cc(C(F)(F)F)ncn1 80053,Cc1ccc(OC)c(CN2CC3(CC3C(F)(F)F)C2)c1F 80054,C(CCOCCO)(C(=O)N(C(C)CO)C)NC(Cc1c(C)scc1)=O 80055,CCCN=C(NCc1nnnn1C1CC1)NC(c1ccnn1C)COC 80056,C1(C(N(C2CC(=C)C2)C)=O)CCCCC1NC(=O)CCOCC(F)F 80057,c1(CC(=O)NC(C(C)C)CNC(=O)CC2CCNC2=O)ccc(F)cc1Cl 80058,N1(C(C2COC3(CCC3)C2)=O)CCC2(CCCN2C(=O)COC(F)(F)F)C1 80059,n1(C(C)C#N)cccc(NC(=O)C(C)C(N)C2CC2)c1=O 80060,C=Cn1ncc(C(=O)NCC2CCCN2C(=O)CCc2ccc(C)o2)c1N 80061,CC1(CO)CC1(Cl)Cl.C1(=O)CCCn2cc(nn2)N1C(CN1CCCC1)C1CC1 80062,N1(C(C2CC(OCC)C2)=O)CCCOC(CNC(=O)CCCCC2CCSS2)C1 80063,N1(C(C(C)NC(=O)NC)=O)Cc2ccnn2CC(NC(c2cnoc2C)=O)C1 80064,c1(C(=O)NCC(CNC(C2CC(C(C)=O)C2(C)C)=O)F)ccc(F)cc1F 80065,N1(C(c2cc(C)c(Br)cc2)=O)CC(CNC(c2cnoc2C)=O)C2(CCC2)C1 80066,C1(C)(C(=O)NCc2c(C(=O)NC(c3nnc(C)o3)C)occ2)CCNC1=O 80067,N1(c2n(CCOC)c(-c3cnn(C)c3Cl)nn2)CCOC2(CCOC2C)C1 80068,C1(OC)(CO)CCC(c2ccccc2)CC1.C(CCC(=O)OCC)NC(=O)NC 80069,Cn1nc(C(C)(C)C)cc1C(N1CC(F)CC1CNC(=O)C(F)(F)C1CC1)=O 80070,C(=O)(C(C)(C)CCN(C)C)NCCN(C(C(CSC)O)=O)C 80071,C(=O)(C1=CCCN(C(C2CC2OC(=O)C2CC2)=O)C1)N1C(C)CC1(C)C 80072,c1(NC(C=C2CCN(Cc3ccc(OC)cc3O)CC2)=O)nc(Cl)c(C)c(Cl)n1 80073,C1(CC(=O)N(C)CC2(CNC(=O)CC3CCCO3)CC2)Cc2ccccc2NC1=O 80074,Cc1ncnc(C)c1C(=O)N(CC(C)N(C(=O)C(CC(C)C)n1ccnc1)C)C 80075,Cc1cc(C(=O)NC2CC(CC(=O)Nc3nccnc3Cl)C2)ncc1[N+](=O)[O-] 80076,CC1CCN(C(=O)C(C)CC(N)=O)C(CNC(=O)Cc2cccc(O)c2)C1 80077,N1(C(C2C(C)C2)=O)CC2CC2(NC(c2coc(Cc3ccccc3)n2)=O)C1 80078,C1(OCC)CCN(C(=NCCNS(C)(=O)=O)NCC(Cl)C(F)(F)F)CC1C 80079,n1(C(C(=O)NCC2CCN(C(C(C=C)O)=O)CC2)C)nc([N+](=O)[O-])cc1C 80080,N1(C(c2cn(C)nc2)=O)CCCC2CCN(C(c3cc(C(N)=O)cs3)=O)CC12 80081,C1(NC(C(N2CC(OCCCCC)C2)=O)=O)CCCC(CN=[N+]=[N-])C1 80082,NS(=O)(=O)CCCC(=O)NC1COC2(C1)CN(C(C1(Cc3cnn[nH]3)CCC1)=O)C2 80083,C1(NC(CNC(CC(C)C)=O)=O)CC2CC1CC2C(N1CC(C)C(O)C1)=O 80084,Cc1cc(-n2cc(C3CCN3C3(CC4COC(=O)N4)CC3)nn2)ccc1Cl 80085,C1(C(=O)NCC2C(NC(c3cc(OC)no3)=O)CCC2)CCCC(=O)O1 80086,C(=O)(C(CC1CCCC1)NC(c1ccncn1)=O)NC(C(=O)N(CC)CC)C 80087,C1(O)(CN(C(CCC(C)SC)=O)C)CCCN(C(=O)C(F)=CC2CC2)C1 80088,N1(C(CC(=O)N(C)C)=O)CCCC1C1CCCN1C(C1CC2(C1)CC(F)(F)C2)=O 80089,N1(C(c2ccc(Cl)cn2)=O)CCN(C(c2ccc([N+](=O)[O-])o2)=O)C(CC(F)F)C1 80090,N1(C(c2cnn(CC(F)F)c2C)C(=O)NCCOC)CCC(OC)C(C)C1 80091,c1(C(=O)Nc2n(CC)ncc2)cc([N+](=O)[O-])ccc1SCC1CC1CC(=O)NC 80092,N1(C(c2nnn(CC)c2C)=O)CC2(CNC(C3(COC)CCOC3)=O)CC1CO2 80093,Cc1cc(NC(c2nncn2C2CCCCC2)=O)ccc1OC(F)(F)F 80094,c1(C(=O)NC(C2CCCO2)CC)ccc(CNC(C2CC(C)(O)C2)=O)o1 80095,CC(CC1CCCCC1)N=c1ccnc(NC2CC3CNC2C3)[nH]1 80096,N1(C(CC(C=C)CC)=O)CCC(CNC(=O)C2=CCCC2(C)C)C(F)(F)CC1 80097,N(C1CCC(NC(C2CC3CC2C3)=O)c2ccccc21)C(CSC(C)C)=O 80098,C1(C(N(CCCOCCN(C)C(C2(C)COC2)=O)C)=O)CNC(=O)C1 80099,c1(-c2cn(C3C(C=C)OCCC3)nn2)cccc2cnccc12.N12CC3C(C3C1)C2 80100,c1(C(N(c2ccccc2F)C(CN2C(C)CSCC2)=O)=O)cc(Cl)ncc1Br 80101,CC(C)C(CNC(=O)CN1CCCCCC1)C(=O)NCc1ccc(CO)cc1 80102,c1(CC)cccc(CC(N2CCCC2(C)CNC(=O)Cc2cnn(C)c2)=O)c1 80103,C1(NC(CC2C(C)CCO2)=O)(CO)CCCN(C(=O)CCC(F)(F)F)C1 80104,CN(C)NC(=O)CCC(=O)NCC(CC1CCCC1)C(=O)N1CCC(C)(F)C1 80105,C1(CCC(=O)NCC(C)(CO)NC(C)=O)CCCCC1N.C(C)(C)(C)OC(=O)OC 80106,C1(C)(CCNC(C2(N(C)C(c3nc(Cl)cs3)=O)CC2)=O)CCOCC1 80107,c1(C(=O)NCC2C3CN(C(C(C)OC4CCCC4)=O)CC32)nnn2ccccc12 80108,C1(C(=O)NC(c2n(CC)ncn2)C)CCOCC1NC(=O)C(C)=NOCC#N 80109,N1(C(CC=C(C)C)=O)CCC(CCNC(=O)C=Cc2cscn2)CC1C 80110,Cc1ccc(C)c(CC(=O)NC2CC(C)N(C(C3CCC(N(C)C)CC3)=O)C2)c1 80111,CCCC(F)C(=O)NCC(C1CCN(C(c2ccc(C)cn2)=O)CC1)O 80112,n1(C(CC)C)nnnc1C(c1sccc1Cl)NCC1CC2(CC2)C1 80113,S(=O)(=O)(c1ccc(C(=O)N(C)CCNC(=O)CC2CCC(OC)CC2)o1)NC 80114,Cc1ccc2nc(C(N3CCCCC(NC(c4ccc(Cl)o4)=O)C3)=O)c(N)n2c1 80115,N1(C(c2cncc(OC(C)C)c2)=O)CC(C)(C)CCC1CNC(C1CCSC1)=O 80116,N1(C(CC2CC(NC(CCCOCC)=O)C2)=O)CCOCC(O)C1 80117,N1(C(C(C)=C2CC2)=O)CCC2(CC1)CN(C(c1cccc(C#N)c1C)=O)C2 80118,c1(C(c2nn[nH]n2)CNC(CNC(C)(C)CO)=O)ccccc1F 80119,O=C(C1CCCc2n[nH]cc21)NCC1CCN1C(=O)CCc1ccc(Cl)c(F)c1 80120,c1(C(=O)NC(CCCC)CNC(=O)CN2CCCCC2)cncc2nc[nH]c12 80121,NS(=O)(=O)c1n[nH]cc1C(N1CCCC(NC(=O)CC2CCCCC2O)CC1)=O 80122,Cc1cnc2cc(C(N3CCOCC3CNC(=O)CCc3cnoc3)=O)ccn12 80123,C(=O)(C1=CC2(CN(C(=O)C(C(CC)CC)OC)C2)OC1)N(CCC#C)CC 80124,C(=O)(C(CNC(=O)C(OC)OC)C(C)C)Nc1c(CC)noc1C 80125,C1(C(=O)NCc2cc(COC)n[nH]2)CCCN(C(=O)COCCC(C)C)C1 80126,c1(C2(C)CSC2)cn(CC2CCN(C(C3CN(C4CCCC4)C3)=O)C2)nn1 80127,Cc1cc(C#N)ccc1NC(C1CCN(c2ncc(Br)cn2)C1)=O 80128,C12(C(N(CCN(C)C(c3cnc(O)s3)=O)C)=O)CCC(CC1)C2(C)C 80129,c1(C2OCCN(C(C(CCNC(CC(C)C)=O)F)=O)C2)ccc2ccccc2c1 80130,C1(C(=O)NC)CCC2(CCN(C(C3CC(F)(F)C3)=O)CC2)O1 80131,Cc1cccc(NC(=O)Nc2ccc(C(=O)NC(c3cccnc3)C)cc2)c1 80132,c1(NC(C(NNC(=O)C2CC(OC)C23CCC3)=O)=O)cccc2c(O)nccc12 80133,CC1(C)OCCC1C(=O)NC1CCC(NC(C2CC(C)(C(C)(C)C)C2)=O)CC1 80134,C(CCCCCNC(C1(C)CCCCC1)=O)NC(C(C)Cc1ccncc1)=O 80135,c1(CC)ccc(F)c(C(N2CC(C)(NC(c3ccnc(C(C)C)n3)=O)C2)=O)c1 80136,C(=O)(C1=CC2(CCN(C(=O)CN3CCOC3=O)C2)C1)NC(C)CO 80137,C(=O)(CC(CC)C(C)(C)C)NCCN(CCCCCC)C(=O)C(O)CC1CC1 80138,C(C(=O)NCC1(NC(=O)CCc2nccs2)CCC1)(C1CCCO1)SCC 80139,C=CC(C)(C)CC(=O)NCCN(C1CCCC1)C(=O)COCC1(F)CC1 80140,c1(C(=O)NC2CCC(CNC(C3(SCC)CC3)=O)C2)cncc2c[nH]nc12 80141,C1(NC(C(C(C)C)O)=O)C2CC1CN(C(c1cc(C#N)c[nH]1)=O)C2 80142,N1(C(C(c2cccnc2)NC(C2CC(C)=C(C)CC2)=O)=O)CC2CCCC(C2)C1 80143,N1(C(C(C(C)C)SC)=O)CCCC2(C1)CN(C(c1cccc(O)c1Cl)=O)CCO2 80144,C12(C(N(C3CCN(C(c4n[nH]c(C)c4Cl)=O)C3)C)=O)CCCN(CC1)C2 80145,CC1(CNC(c2cc(N)ccc2O)=O)CCCN(C(c2c(F)cccc2Cl)=O)C1 80146,CC1(C)CN(C(c2ccc3sncc3c2)=O)C(CNC(=O)C=CCO)CO1 80147,c1(C(=O)NCC(C)(C2CC2)NC(=O)CCCC#N)cc2cncn2c(O)n1 80148,c1(C(N(C2CCN(C(CC(C=C)C)=O)C2)CC)=O)cc2nc(Cl)ccc2s1 80149,c1(NC(Cc2cn(C(CC=C)CC)nn2)C(=O)OC)nccc(CC#N)n1 80150,C1(NC(CC(CC)C)=O)CCOC12CCN(C(=O)C(C)OC)CC2 80151,C1(NC(c2cc(COC)on2)=O)CC1C1CCN(C(=O)Cc2sccc2C)CC1 80152,c1(C(CO)NC(NNC(c2cccc(OC)c2)=O)=O)ccc(S(C)(=O)=O)cc1 80153,c1(CN2CC(CCCCNC(C3CC(CC)C3)=O)C2)c[nH]c2ccc([N+](=O)[O-])cc12 80154,C1(C(=O)NCCCN(C(c2cncc(N(C)C)n2)=O)CC)CCCCC1C1CC1 80155,N1(C(CC(CC)NC(=O)CCN2CCOCC2)=O)CCC(O)C(CO)C1 80156,Cc1nc(C(C)C)ccc1C(=O)NC1CN(C(=O)CN2CCC(C)CC2)CC1F 80157,C(=O)(C(C)(C)CS(N)(=O)=O)NC1CC(C)(C)N(C(=O)CC(F)(F)F)C1 80158,Cc1ccc(O)c(C(N2CCC(C(F)C(=O)NCC=Cc3cccnc3)C2)=O)c1 80159,c1(OC)ccc(C(=O)NCC2CC(NC(C3(n4cncn4)CC3)=O)CCO2)cc1 80160,C1(COC)COCCN(C(=O)CC(C)NC(c2cc(Br)cs2)=O)C1 80161,C(=O)(C1CCc2cc(C)ccc21)N(CCCNC(C1(COC)CCCO1)=O)C1CC1 80162,C12(CNC(C(C)NC(CC)(C)C)=O)CC(CCO1)C2.C12(CCC1)CCOC2=O 80163,c1(CC(=O)NCCCOCCN(C(=O)C(c2cncn2C)O)C)c[nH]ccc1=N 80164,O(NC(=O)C(CCF)NC(c1cccc(O)c1F)=O)C(C(C)C)CO 80165,c1(C(=O)NC2CCCN(C(CC3(C=C)CCC3)=O)CC2)cc(C)cc(OC)c1C 80166,N1(C(c2[nH]cc(C)c2)=O)CCC2(C1)CN(C(=O)CCCNS(C)(=O)=O)C2 80167,c1(OC)ccc(C(=O)NC(C2(O)CN(C(C3CCCSS3)=O)C2)C)cn1 80168,c1(C(N2C3C(N(C(C(CC)SC)=O)C)CC(C3)C2)=O)ccn2ncccc12 80169,Cc1nc(N2CCCCC(CNC(=O)CC(C)C)C2)c2c[nH]nc2n1 80170,CC(N=c1cc[nH]cc1S(=O)(=O)NCCc1cncn1C)c1ccccn1 80171,c1(C(N(CCN(C(C2(C(=O)NC)CC2)=O)C)C(C)C)=O)c(C)cc(Br)cc1C 80172,c1(C(=O)NC2CCC(CCNC(c3cscc3F)=O)C2)cn2c(n1)SCC2 80173,C(C(=O)N(C1CCCCC1N(C(=O)CN1CC=CC1)C)C)(C(C)C)N(CC)CC 80174,N1(C(c2cc(CC)nn2C)=O)CC(NC(C2CCC(CC)CC2)=O)CC12CCC2 80175,N1(C(C2C(CC)NCC2)=O)CCC(N)c2c(Br)cccc21 80176,CC(C)C(C)CC(=O)NCC1CC(O)(CNC(c2cc(Br)sn2)=O)C1 80177,N1(C(c2ccc(Br)c(F)c2)=O)CC2(CCC(N3CCc4ccc(Cl)cc43)CC2)C1 80178,c1(CC(CC(=O)OC)NC(C)=O)ccc2c(c1)CCO2.C12CN(C1)S(=O)(=O)C2 80179,C1(NC(CC(C)NC(N)=O)=O)CCSC12CN(C(c1cccc(C(N)=O)n1)=O)C2 80180,c1(C(=O)NC23C(CN(C(C=CC)=O)C2)CCCC3)cc2ccc(F)cc2nc1C 80181,N1(C(c2cccc(N3CCCC3=O)c2)=O)CC2CCC(C1)N2C(C1CCC1F)=O 80182,CC1CCN(C(=O)CN(c2ncccn2)C(=O)NC2CC2)CC1C(F)(F)F 80183,C1(C(=O)NCCc2cccnc2O)CC2CC1CC2O 80184,n1(CC)ncc([N+](=O)[O-])c1C(=O)NCC(C)CNC(c1ncn(C(C)(C)C)n1)=O 80185,c1(C(=O)NCC(C2CCCC2)NC(c2cc(CCO)on2)=O)n[nH]c(C2CC2)n1 80186,N1(C(CC2(OC)CCCC2)=O)CCC(NC(=O)Cc2cncn2C2CC2)C1C 80187,c1(C(N(C2CCCCN(C(CC)=O)C2)C)=O)cc2cc(OC)ccc2o1 80188,n1(C(C)C(N2CC=CC(NC(=O)CCC3CCOC3)C2)=O)cnc2ccccc12 80189,c1(NC(c2c(OC)ccs2)=O)ccc2c(C(N3CCOCC3(C)C)=O)ncn2c1 80190,C1(C(=O)NCCCN(C(C(C)=C(C)C)=O)C2CC2)CC12CCS(=O)(=O)CC2 80191,c1(N(C2CNCC2(F)F)C(c2cn(C(C)(C)C)nc2)=O)ncnc2cnccc12 80192,N1(C(c2c(C(C)C)cnn2C)=O)CC2(CCN(C(=O)CSCC(N)=O)C2)C1 80193,c1(CC(C)OC)nc(C2CCCC2O)n(-c2ccncc2C)n1 80194,C#CC1(C(=O)NC2CCC(C)(CC)CC2)CCN(C(=O)C(O)C(F)(F)F)CC1 80195,C1(C(=O)NC(C=C)C)(COC)C=CCN1C(=O)CC1CCCC(=O)C1 80196,N1(C(Cc2cnc(C)s2)=O)CCC(CNC(c2c[nH]nc2C)=O)C(C)C1 80197,C1(NC(C2CCn3nccc3C2)=O)CCC2(CCNC2)C1 80198,c1(C(C(C)N(c2cn(C)cc(Br)c2=O)CCC)=O)nc2c(s1)CCCC2 80199,c1(C(=O)NCC(C)CNC(C2CC2c2ccco2)=O)coc2c1NC(=O)CCC2 80200,C(=O)(C1Cc2c(Cl)cccc21)NCCCOCCCNC(C1N(C)CCOC1)=O 80201,N1(CC(C)NC(CNC(=O)OCC)=O)CCN(C(C2CCOC2CC)=O)CC1 80202,c1(NC(CC2(C)CN(C(C3CCCCCC3)=O)C2)=O)ccc(O)cc1O 80203,C1(CCOC)(NC(=O)CCC2CCC2)CCN(C(=O)C2=NOC(C)C2)CC1 80204,C1(CCSCC(=O)Nc2cccc(NC(C)=O)c2)CCC=CCCC1 80205,C12(C(N3CCC(N(C(=O)C(C)N(C)C)CCC)C3)=O)CCC(O)(CC1)CC2 80206,c1(C(N2CCCC(F)(C(=O)NCCC(O)C3CCC3)C2)=O)cc2occc2[nH]1 80207,CC(C)(C)C=CCNC(=O)NCCNC(=O)C(=O)NC1CC1 80208,c1(CC)cnc(O)c(C(=O)NC(C)(CNC(C2CC2(Cl)Cl)=O)C2CCC2)c1 80209,S(=O)(=O)(c1ccc(Cl)s1)N1CCN(C(Cn2ccc(C(=O)OC)n2)=O)CC1 80210,C1(NC(C(CSC)O)=O)CCN(C(=O)Cc2c(F)cncc2Cl)CC(O)C1 80211,C=CCC(CC=C)C(=O)N1CCC(F)(F)C(CNC(c2cncn2C2CC2)=O)C1 80212,c1(C(N2C(CC(C)O)CCCC2)=O)cccc2c1COC2 80213,c1(C(=O)NC2CN(C(c3c(Cl)ccc(OC)c3)=O)CC2C)cc(F)c(N)cc1F 80214,C1(NC(C2C(CC)C2)=O)CCCC1(C)CNC(=O)CCSc1ccccc1F 80215,CCCCS(=O)(=O)CC(=O)NC1(CC)CCN(C(=O)C(C)=C2CCCC2)CC1 80216,c1(C(=O)NCC(C2CCOC2)NC(Cc2n(C)ccn2)=O)ncccc1F 80217,c1(C(N2CCC(C)(N(C)CC)C2)=O)cnc(O)c2ccccc12 80218,c1(S)nnnn1C.c1(SCCC(=O)N(CC(CC)OC)CC)nc(C2CC2)ns1 80219,N1(C(CC(CC)(F)F)=O)CCC2CCN(C(C3C(C=C(C)C)C3(C)C)=O)C2C1 80220,C1(CNCC(CN(C(=O)OC)C)O)CC2CCCC2C1 80221,CCCCCC(=O)NCCOCCCN(C)C(c1cnc(C(C)C)[nH]1)=O 80222,C(=O)(CCN(OC)C(=O)CC(C)C1CCCO1)NCc1cccc(OC)n1 80223,C1(NC(CSCC(N)=O)=O)(CNC(C2CC2F)=O)CC2CCC1CC2 80224,C1(CNC(C)=O)CCN(N2CCC(CCc3nc(C)no3)CC2)CC1 80225,C1(F)(CNC(Cc2ncc(CC)[nH]2)=O)CC(N=c2[nH]nc(C3CC3)s2)C1 80226,C=CCC(CC)C(=O)N(CC(C)NC(C1(C)COC1)=O)C 80227,N1(C(c2cn(C3CC3)nn2)C(=O)NCCSC)CCc2ccc(Br)cc2C1C 80228,N1(C(c2c(CC)nc(C)o2)=O)CC(C(=O)N(CCCO)C2CC2)C(C)(C)C1 80229,c1(NC(C(=O)NCCc2cc(C)oc2C)=O)ccc(S(C)(=O)=O)cc1 80230,C1(NC(C(=O)NCC)=O)CCCC(CNC(=O)C(C2CCCCCC2)O)C1 80231,c1(C(N2CCC(C)C2)=O)ccc(CNC(c2cc(O)n(C)n2)=O)cn1 80232,C1(C(N(C2CCCN(C(=O)C=Cc3cnc[nH]3)C2)C)=O)OCCOC1(C)C 80233,C1(NC(=O)OC(C)(C)C)CCCC12CCN(C(c1cc[nH]c(=N)c1O)=O)C2 80234,C1(CC(N)=O)(NC(=O)Cc2ccccn2)CCN(C(C2CCCN2C=O)=O)CC1 80235,N#Cc1ccc(C(=O)NCC2C=CC(NC(C3CCC4(CC4)C3)=O)C2)cc1 80236,n1(CC(=O)NCC(C(C)C)NC(C2CN(C)CCO2)=O)cc2ccccc2n1 80237,c1(OCCN2CCCC(C(=O)NC3CC(C)(NC(C)=O)C3)C2)c(C)cc(C)cc1C 80238,C1(COC)(NC(=O)COC2CC=CC2)CCN(C(=O)C(O)C2CC2)C1 80239,C(CC(=O)Nn1cnn(CC(=O)OC)c1=O)N(C(=O)C(C)CCCC)CC#C 80240,Cc1ncc(C(N2CC(C)CNC(C)C2)=O)c(Cl)c1Cl 80241,CC(C)(N=[N+]=[N-])C(=O)NCC(C)(O)CNC(=O)CP(C)(C)=O 80242,CC1(C(=O)NC2C3CN(C(=O)CC4CC4(Cl)Cl)CC23)CC2(C1)CC(F)(F)C2 80243,c1(C(c2nnnn2CC(F)F)NC(c2ncnn2C)C)ccc(C#N)s1 80244,c1(OC)cccc(NC(C2(CNC(c3ncnn3C(C)C)=O)CCCO2)=O)c1 80245,C1(C(N2CCN(C(CSC(C)C)=O)CC2)=O)CCc2n[nH]cc2C1 80246,c1(C(=O)NC2C(C)(C)CN(C(C3CCCC3O)=O)CC2)cc2cc(O)ccc2[nH]1 80247,C1(C(=O)NCCCCC)CN(C(C2CC2(C)C(F)F)=O)CC1C(C)C 80248,C1(CNC(C(CC#C)C)=O)CN(C(=O)COc2c(C)occc2=O)CC12CC2 80249,n1(CC(=O)NC(CNC(C(=Cc2cccc(Cl)c2)C)=O)C)cc(S(C)(=O)=O)cn1 80250,CC1=NNC(=O)C1CC(N1C(C(=O)NCc2nnc(C)o2)CCC1C1CC1)=O 80251,Cc1ccc(C(=O)NC(c2cccnc2)C(=O)NC2CC3OCCCC23)c(O)c1 80252,C(=O)(CCCCCN=[N+]=[N-])N1CC(C)C(CNC(C2(C(F)(F)F)CCO2)=O)C1 80253,c1(C(=O)NC2CC(CNC(CN(C)CC)=O)OCC2)sc(Cl)c(Cl)c1OC 80254,C1(NC(c2cc(N(C)C)ccn2)=O)CN(C(=O)C(O)c2ccsc2)CC2(CC2)C1 80255,c1(OC)cccc(CNC(C2(CC)CN(C(C3CCOC(C)C3)=O)C2)=O)n1 80256,N1(C(C(N2CC(Cc3c(C)noc3C)C2)=O)=O)CCOC(C)(C)C1 80257,c1ccc2nc(C3CCCCC3)c(N3CCC4CNCC4C3)nc2c1 80258,c1(C(=O)NC(C)CNC(C2C(C)(C)C2(F)F)=O)ncn2cc(Br)sc12 80259,C1(C(N2C(CCCNC(c3cn(CC=C)nc3)=O)CCC2)=O)COCCC1(F)F 80260,CCC(CC)CCCC(=O)N1CC(C(N2CC3CC=CCC3C2)=O)(CC)C1 80261,C12(C(=O)NCc3cc(C)on3)CCCC1CCN2C(c1cn(C)cc1C)=O 80262,c1(C(=O)NCCN(C(CCC(=C)C)=O)CCC)ccc(OC)c(OC)c1C 80263,CCC(C)(O)CCNC(C1CCN1C(=O)C=CCOC)=O 80264,N1(C(Cc2c(Cl)cn(C)n2)=O)CCC(NC(c2cnc(N(C)C)nc2)=O)C12CC2 80265,N1(C(c2[nH]cc(OC)c(=O)c2)=O)CCC2C1CCCN2C(=O)Cc1cn[nH]c1 80266,C1(C(=O)NC(C2CCOC2)(C)C)CC2CN(C(=O)C=Cc3ccncc3)CC2C1 80267,C1(C(=O)NC(=O)COCc2ccccc2)CCC(F)CC1.C1(=O)CCOCCN1 80268,C(C)(CO)(CS(C)(=O)=O)OC(=O)NCC(OCOC)C 80269,N1(C(c2cnc(OC)s2)=O)CCC2CCCC12C(=O)NCC1CC2CCCC2C1 80270,c1(C(N(CCNC)C)=O)cc2c(s1)CCOC21CCN(C(=O)OC(C)(C)C)CC1 80271,c1(C(=O)NCC(CNC(c2c(C)c(N)ccc2)=O)O)ccccc1S(C)=O 80272,C1(C(C)C)OCCC1C(=O)NCC(C)(C)CN(C(=O)CC1CN(C)C1)C 80273,c1(OC)cc(C(N2CC3C(C2)N3C(C2(C)CCCC2)=O)=O)cc(C(F)(F)F)n1 80274,Cc1cc(Cl)ncc1S(=O)(=O)NC1CCC(C(=O)Nc2ccc(Br)cc2O)OC1 80275,CC(C)CC(C)(O)C(=O)N1CCN(CC(=O)NCCCOCC(F)F)CC1 80276,C1(C(=O)NCC(CNC(C(C)(CO)OC)=O)(C)O)CC2(C1)CC(CO)C2 80277,C(C1c2ccccc2CCN1C(c1cnsn1)=O)NC(c1cccc(OC)n1)=O 80278,Cc1noc(NC(C2C3CN(C(=O)CCCN4CCCC4)CC23)=O)c1C 80279,C1(NC(CCN(C(C2(C(=O)OCC)CC2)=O)C(C)C2CC2)=O)CCCCC1 80280,C1(C(N(C2CCN(C(c3c(CC)[nH]cc3)=O)CC2)C)=O)COc2ccccc2O1 80281,N1(C(c2c(OC)c(Br)ccc2)=O)CCC2CN(C3CC3)CC12.c12ccc(cc1)OC2 80282,N1(CCN(C(CN(C2CCC2)CC)=O)C)CCN(C(c2c(C)n[nH]c2C)=O)CC1 80283,C(=O)(C1=NN(C)C(=O)CC1)N1CCCCCC(NC(c2nccc(CC)c2)=O)C1 80284,N1(C(c2c(C)n(C)cc2)=O)CC(CC(=O)NCc2cnc[nH]2)CC1(C)C 80285,C1(NC(c2nc(Cl)cs2)=O)CN(C(C2CS(=O)(=O)C2)=O)CC2CCCC12 80286,N1(C(CCS(=O)(=O)N(CCOC)C)=O)Cc2ccccc2CC1CC(=O)O 80287,N1(C(C(C)N(C)C)=O)CCC(C)C(CNC(c2cc(O)nn2C)=O)C1 80288,Cc1nc(Cl)ccc1CC(N1CCN(C(=O)Cn2cnnc2O)CC1C)=O 80289,CC1CCCCC1C(=O)NCC(C)(C)CCNC(=O)Cn1ncnn1 80290,CS(=O)CCC(=O)N1CCCC(CCNC(C2(c3ccc(Cl)nc3)CC2)=O)C1 80291,CN1CC(O)(CN(C(=O)C(Cc2cc[nH]n2)NC(=O)CCC2(C)CC2)C)C1 80292,N1(C(C2C(C)(C)C2)=O)CCCC2(CC(NC(=O)Cn3ncc4ncccc34)C2)C1 80293,C1(C(=O)OC)(C(=O)NCC(C)NC(=O)CCC2CC2(Cl)Cl)CC2(CCC2)C1 80294,c1(NC)ncccc1C(=O)NC1CC(C)N(C(=O)CCc2nc(C)c(C)o2)C1 80295,C(=O)(C(O)C(F)(F)F)NC(CN(C)C(c1ccc(C(C)(C)C)s1)=O)(CO)CO 80296,CN=c1[nH]cc(C(=O)NCC2CCC(C(=O)NCCC3(O)CCOC3)C2)o1 80297,c1(C(=O)NCC2(NC(C3CCCCS3)=O)CCC2)ccnc2nccnc12 80298,Cc1nc(C=CC(=O)NCC2(CNC(=O)CC3(CO)CC3)CC2(F)F)cs1 80299,N1(C(CC2(OC)CN(C(=O)Cc3cc(C)cs3)C2)=O)CCCOC(C(C)C)C1 80300,c1(C(N(C(CNC(CSCCC)=O)C)C)=O)cccnc1O 80301,CC(C)C(C(C)NC(c1cncc(C2CC2)c1)=O)NC(=O)C(F)(F)CO 80302,C=CCCCC(C(=O)N1CCSC(C)CC1)NC(=O)Cc1cccnc1O 80303,c1(N2CCC3(C(F)(F)C3)C2)[nH]c(=NC2CCC(C3CC3)CC2)nc2sccc12 80304,c1(C(=O)NC2(C)CN(C(=O)C3=CSCS3)C2)ccc2c(=O)cc[nH]c2c1 80305,Cc1csc2c(NC3CCC(NC(=O)CCCC(=O)NC(C)C)CC3)ncnc12 80306,c1(C(N2CC(NC(c3cncc(C(F)(F)F)n3)=O)(CO)C2)=O)ccnc(Cl)c1F 80307,c1(CC)cccc(C(=O)NC2CC2NC(=O)CS(=O)(=O)N2CCOCC2)c1.N1CCCC1 80308,c1(C(N2CC(CC)C(NC(C)=O)C2)=O)ccc(OC)cc1OC(F)F 80309,C1(C(C)C)C(NC(C2(C)CC2C(F)(F)F)=O)CCN1C(C1C2CC3C(C2)C13)=O 80310,N1(C(c2[nH]cc(C)c2C)=O)CCC2CN(C(C3CN(C)CC(C)O3)=O)CC2C1 80311,N1(C(COC(C)=O)=O)Cc2ccccc2C1CNC(C1CCC1(F)F)=O 80312,c1(N2CCCC(CC=C)(NC(=O)COc3ccon3)C2)ncnc2ccccc12 80313,C1(C(=O)NC(CCCOC(=O)NCC2CN(CC)C2)=O)C2CCC3C(C2)CC13 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80782,C(N=C(NC1CC1)N1CCC2=C(COC2=O)C1)C1CN(C)C(C)(C)C1 80783,CC(CCC(=O)NC1CN(C(C2CC2Br)=O)C1)N(C)C 80784,CC1(CNC(=O)CCCC#N)CCN(C(=O)COCC2CCCO2)CC1 80785,C1(C(=O)NCCNC2CCCCC2)CCCC(Nc2cn[nH]c2)C1 80786,CC(O)(CC(F)F)C(=O)NCc1ccc(C(=O)NC2CCCC2)cc1 80787,C1(NC(=O)CCc2ccon2)CN(C(C2CC3(CCC3)CO2)=O)C2(CCC2)C1 80788,c1(C(N(C(CC(=O)OCC)CC(C)C)C2CC2)=O)cccc2nc(C(C)C)[nH]c12 80789,C12(NC(C(C)NC(N)=O)=O)CCCN(C(c3cc(C(F)F)on3)=O)CC1C2 80790,c1(C(N2C(C)CC(NC(c3cccc(COC)c3)=O)C2)=O)cnn2c1CCCC2 80791,N1(C(C(=O)NCc2ccc(C)o2)C)C(C)CCCC1C 80792,S(=O)(=O)(c1cccc(C(=O)OC(C)(C)C)c1)N(C1CCCCCC1O)C 80793,C1(CNC(C2C(=C)C2)=O)CCCN(C(=O)CCn2ccnc2C)CC1 80794,c1(N(C2CCN(C(C3C(C#C)C3)=O)C2)CCO)ccc2c(n1)CCC2=O 80795,C1(CC=C)(NC(c2cnc(C)o2)=O)CCCN(c2cc(C)nc(SC)n2)C1 80796,N1(C(C2N(C(C)C)CCC2)=O)CC(CO)C2(C1)CN(C(=O)C(F)F)C2 80797,CCC(CCCC(=O)N1CCCC1CN(C)C)NC(C1CC(O)C(F)C1)=O 80798,Cc1oc(C(C)C)cc1C(=O)NC1CCOCC1NC(=O)CCc1cc[nH]n1 80799,C1(CNC(C(C)OCCCC)=O)COCCN1C(=O)C(O)CCc1ccccc1 80800,C(=O)(C(CC)C(=O)N1CC=C(CNC(=O)CN2CCCC2CO)CC1)OC 80801,N1(C(c2nnn(CC)c2C)=O)CCC(C(F)(F)F)C(NC(=O)C(C)C2CCC2)C1 80802,C1(C(N2CC(CN(C(=O)COCC3(F)CC3)C)OCC2)=O)Cc2cscc2C1 80803,c1(C(=O)OC)cc(NC(Cc2ccccc2OC(C)C)C(C)C)ccc1C 80804,N1(C(C(C(C)C)n2cncn2)=O)CCC(CO)(NC(=O)CCCCC#N)CC1 80805,C(CC(F)(F)Cn1cc(CC(O)COC)nn1)NC(c1c(CC)con1)=O 80806,N1(C(c2c(C)nn(C)c2)=O)CCN(C(c2cc(C(C)C)ccc2F)=O)C(CF)C1 80807,c1(OC)ccc(Br)c(OC)c1NC(C1CC(=O)N(C)C1c1ccccc1)=O 80808,C1(CNC(NC2C(c3c(C)n(C)nc3)N(C)C(=O)C2)=NC)CCCCCC1(F)F 80809,Cc1nn(C2CCC2)cc1C(N1CC2CC1C2NC(=O)Cc1ccnn1C)=O 80810,Cc1cccc(C)c1C(N1CC(NC(c2cc3sccc3[nH]2)=O)C2(CC2)C1)=O 80811,C1(C(N2CCC(CCC)(CO)C2)=O)CC(C)CN(C(c2cccs2)=O)C1 80812,C1(C(N(C)CC2(CO)CC2)=O)COC2(C1)CN(C(=O)CC1CCC(C)(C)C1)C2 80813,C1(NC(=O)CNc2ccccn2)CCSC12CN(C(=O)C1=C(Cl)CC1)C2 80814,c1(C(C(N2CC(C#N)(CC)C2)=O)C)ccc(F)c(F)c1 80815,C1(C(=O)NC(C)Cn2cnnc2)CC2(CCN1C(C1CCCC3(CC3)C1)=O)CC2 80816,c1(OC)cnc2c(c1)C(NS(=O)(=O)CCOC1CC1(F)F)CCC2 80817,C(C1=COCCC1)(c1n(-c2c(COC)cccc2)nnn1)NCC1(COC)CC1 80818,CC#CCCCC(=O)N(C)CCOCCCN(C)C(C12CCCC1(C(N)=O)C2)=O 80819,c1(CNCC2(NC(c3c(Br)ccnc3Cl)=O)COC2)c[nH]c2cccnc12 80820,C1(NC(c2c(CC)nns2)=O)CCC(C)N(C(C2(CSC)CCC2)=O)C1 80821,CCC(CN(C)C)CC(=O)NC1C2CC1N(C(=O)CNS(C)(=O)=O)C2 80822,C1(CNC(C(C)C2CCCC2)=O)C2CN(CCOc3cccc(Cl)c3)CC12 80823,c1(C(=O)NC2C(NC(c3c(C)nc(Br)o3)=O)CC2)cnc2ccccn12 80824,C1(CNC(c2cc(C)c(Cl)cn2)=O)C(C2CC2)CCN1C(=O)CCc1cnco1 80825,C1(CC(N2CC(C(C(=O)NC(C3CCCCC3)COC)OC)C2)=O)CCCN(C)C1 80826,C1(C(N2CC(C(N)=O)(CNC(=O)CC3CCC(=O)N3)C2)=O)CC2C=CC1O2 80827,C1(N(C(C(C)OC)=O)C)CCC(NC(=O)CCN(c2ccncc2)C)CC1 80828,N1(C(C(C)=CC)=O)CCC2CN(C(=O)CCN3CCCCC3=O)CC2C1 80829,N1(c2nnc(-c3c(C)sc(O)n3)n2CC(C)C)CCC2(CC1)CNC(=O)O2 80830,C1(CC(=O)NC2CC(CNC(CSCCN(C)C)=O)C2)CCCC2CCCCC12 80831,C1(NC(C=CCOC)=O)C=CC(CC(=O)NC(Cc2cnc[nH]2)CO)C1 80832,C1(C(=O)NC(C2(O)CN(C(c3cc(N(C)C)ccn3)=O)C2)C)CC(C2CC2)=NO1 80833,C(=O)(CCCC(C)C)NC(C(=O)NCCSC)CCCCO.C1(N)CC1 80834,C(=O)(C(C)C(F)(F)F)N(C)CC1N(C(Cn2cc(C(C)O)nn2)=O)CCC1 80835,C(=O)(C1=CC(C)(CC)C1)N1CC(OC)(CNC(c2cc(Br)oc2C)=O)C1 80836,N1(C(C(C=C=C)C)=O)CCOC2(C1)CN(C(=O)C(C)(C)COC)C2 80837,CC(C)CC(C)(O)C(=O)NC(CC(=O)NC1CC(N(C)C)C1)C(F)(F)F 80838,c1(C(C)=O)cccc(OCC(=O)NC(CNC(C2C3CCCC23)=O)C(C)C)c1 80839,C(=O)(C1CCc2cc(F)ccc21)NC(C)CN(C)C(c1cc(O)cc(=O)o1)=O 80840,c1(NC(=O)C(N2CCC(N3CCCC3)C2)=O)cc(N2CCOCC2)nc(Cl)c1 80841,C1(NC(C23C(CN(C(C(N4CCOCC4)C)=O)C2)C3)=O)CCCCCCC1O 80842,Cc1c(Br)cc(S(=O)(=O)N2CCCN(Cc3ccccc3)C(C)C2)c(C)c1C(=O)O 80843,c1(C(N(C2(CC(=O)NCC(O)CC(F)(F)F)CC2)C)=O)cccn2nccc12 80844,N1(C(CNC(=O)OC)=O)CCC(NC(c2ncc3[nH]ncc3n2)=O)C2(CCC2)C1 80845,CC(C)(CC(F)C(=O)NC1(c2nc[nH]n2)CC1)NC(c1cccc[n+]1[O-])=O 80846,N1(C(c2c(OC)ncc(Br)c2)C(=O)NC2CCOC2)CCCC2C(O)CC12 80847,Cc1nn(C)c(C(=O)NCCCN(C)C(C2CCCCN2C)=O)c1Br 80848,N1(C(C(C)OCCC(C)C)=O)CCC(C(C)C(=O)NCC2(C)CCCO2)CC1 80849,C12(C(=O)NCCCN(OC)C)CCCC1CCN2C(C1CCOCC1)=O 80850,N1(C(c2n(COC)ncc2)=O)CCC(NC(=O)C(N2CCN(C)CC2)C)C12CC2 80851,CC1(C)CC(C(=O)NCC2(C)CC2(F)F)CN1C(c1ccc(C#N)cn1)=O 80852,N1(C(C=C(CC)CC)=O)CCC(NC(=O)CC2CC2(C)C)C12CCC2 80853,c1(OCC(=O)NC2C(NC(c3c(CC)c[nH]n3)=O)C2)nn(C)cc1[N+](=O)[O-] 80854,C1(CC(=O)N(CC(C)NC(=O)CCc2ccc(C)s2)CC)(CC)CCOCC1 80855,C#CCC(CC#C)C(=O)N1CCCCC1CN(C)C(c1cnn2c1OCCC2)=O 80856,C(=O)(C1=NNC(=O)C1)N1C(CNC(=O)CC2C=CCC2)CC1 80857,Cn1ccnc1C(F)(F)C(=O)NC1CCN(C(=O)Cc2cnc[nH]2)C1 80858,c1(OCC)cnc(N2CC3C(CNC(=O)C(C)CCN(C)C)C3C2)nc1C 80859,C(c1cccnc1)=C(C)C(=O)NC(C)CC(C)NC(=O)Cc1ncc(C)s1 80860,Cc1ccc(C(=O)NNC(=O)c2cn(CCNC(=O)OC(C)(C)C)nn2)cn1 80861,C(=O)(C(C)(C)C(C)NC(c1cn(C2CC2)cn1)=O)NCC(N1CCCC1)C 80862,c1(NC(c2n(CCCSCC)nnn2)CC2CC2(Cl)Cl)cn(CCF)nc1C 80863,C(=O)(CC(C(F)F)NC(c1cccc(OC)c1)=O)NC(CC)(C)CO 80864,N1(c2n(CC3CCC(C)C3)c(C(C)(C)CC#N)nn2)CCn2nnnc2C1 80865,C1(NC(c2cc(C)c(C)o2)=O)CC2CC(C1)N(C(=O)CCc1cn(C)nn1)C2 80866,C1(NC(Cc2c(C)cc(F)cc2)=O)C2COCC1CN(C(=O)CC1CC(F)C1)C2 80867,C1(C(=O)NCC2C3CN(C(COC(C)=O)=O)CC32)CCC2CC1CO2 80868,n1(CC(C)NC(=O)C(CN(C)C)N(C)C)cc(-c2cnc(C3CC3)o2)nn1 80869,CC1CN(C(=O)C(c2ccccc2)O)CC1CNC(=O)Cc1ccccc1F 80870,c1(C(N2CC(CCNC(=O)CC(C)(F)F)(OC)C2)=O)cc(S(C)(=O)=O)cnc1O 80871,C(=O)(CCN=c1[nH]ccs1)NC1CC(NC(C(CC)Cc2ccccc2C)=O)C1 80872,c1(C(N2C(CNC(Cn3c(C)ncc3)=O)COCC2)=O)cc(O)c2ccoc2c1 80873,c1(C(=O)NCC(C)NC(c2cc(F)n[nH]2)=O)ccnc2c1nnn2C 80874,C1(C(=O)NCCCN(C(=O)CCc2ccoc2)CC)CCn2ncnc2C1 80875,C1(C(=O)Nc2cccc(C)c2)CC2(CCN1C(=O)CNC=O)CC2 80876,N1(C(Cc2n(C)ncc2Cl)=O)CC(CNC(C2CCCC(=O)N2)=O)C2(CCC2)C1 80877,CCCCC(C(=O)N1CC2CN(C(c3ccc(CO)cn3)=O)CC2(C)C1)C(C)C 80878,c1(OC)ccc(O)cc1C(N1CC(OC)CC1CCNC(=O)CC12CC(C1)C2)=O 80879,N1(C(C(C2CC2)OC)=O)CC(O)CC1CNC(C)=O 80880,c1(C(=O)NC)ccc(CC(=O)NC2C=CCN(C(=O)CSCC#N)C2)cc1 80881,C#Cc1cccc(CC(=O)NCCC2CCN(C(C3CC34CCSCC4)=O)C2)c1 80882,N1(C(C2CC2(F)F)=O)CCN(C(C23CC(CN2C2CC2)C3)=O)C2CCCCC2C1 80883,O=C(N=c1c(Cl)c[nH]cc1I)c1cc2nc(-c3ccsc3CO)ccc2[nH]1 80884,c1(OC)cc(Cl)c(Br)cc1NC(c1ccc(-c2csc(C)n2)cc1)=O 80885,c1(CN(C2CCN(c3ccc(C)cc3)CC2)CCC)c(C)n[nH]c1C 80886,C1(C(=O)NCC(C)NC(C=C(C)c2ccsc2)=O)CC2(CCC(F)(F)CC2)CO1 80887,Cc1csc(=O)n1CCC(=O)NCC1(CNC(C2CS(=O)(=O)C2)=O)CCCCC1 80888,C(CCC(C)(C)SC)NC(C1(COC)CN(C(=O)CSC(F)(F)F)C1)=O 80889,c1(C(=O)NC(CC(C)C)(C)CNC(=O)CC2CCC2)cnc2n1CCCC2 80890,Cc1cc(C(=O)NC2CN(C(=O)CC(C)c3ccncc3)CCC2F)cc(F)c1 80891,C1(NC(c2scc(C(C)(C)C)c2)=O)CCN(C(C2(C3CC3)CC2)=O)CC1CO 80892,C(=O)(C(CNC(=O)C(F)=C(C)C)(CC)CC)NCCC(CC=C)(C)C 80893,N1(C(C=CCOC)=O)CCCC(C(=O)NC(C)C(N)=O)C1 80894,c1(COC)cccc2sc(NC(C3CCC(C#N)C3)=O)nc12 80895,c1(SCC(=O)NCC2(CNC(CCCOC)=O)CCC2)cc(C)ccc1C 80896,c1(C(N(C(C)CCO)C)=O)ccc(C2COCCN2C(C2CC2C(F)F)=O)n1C 80897,c1(C(=O)NC(CCNC(C(CC#C)C2CC2)=O)C(C)C)c[nH]c2c(F)cccc12 80898,C12(COC)CN(C(=O)CCC3CCCC3)C(CNC(=O)C=CC=C(Cl)Cl)(C1)C2 80899,C(=O)(C(C)(C)C(=O)NN1Cc2ccccc2C(=O)N1)OC 80900,C1(NC(Cc2cnc(C)[nH]2)=O)CC(C)N(C(=O)C(C2CCCO2)C2CC2)C1 80901,CCCC(C)(C)C(=O)NCC1(F)CCN(C(c2noc(C3CC3)c2C)=O)C1 80902,C12(CNC(C3C(C)(C)CO3)=O)CC1CN(C(c1cnc(CC3CC3)s1)=O)C2 80903,C1(C(=O)OC)CCC(Cn2cc(CNC(c3cn(C)nc3Cl)=O)nn2)CC1 80904,CC1(C(N2CCOC(CNC(=O)Cn3cc(C4CC4)cn3)C2)=O)CC2CC2C1 80905,CCCC(CNC(=O)C(CC)C(C)C)C(=O)N(CC)OCC 80906,Cc1ccc(-c2cncc(F)c2)c2nc(C(=O)Nc3cnc4[nH]cnc4c3)cn12 80907,N1(C(CNC(C2C(C)=CCS2)=O)=O)CC2CCCCCC2C1 80908,Cc1ccc(CC(N2CCCC2(CO)CNC(C2CCC(=O)O2)=O)=O)cc1Cl 80909,c1(COC)nn(C)c(Cl)c1C(N1CCCCC(CNC(=O)C(C)=CC(C)(C)C)C1)=O 80910,c1(C(N2CCCC(NC(COC(CC)(C)C)=O)C2C)=O)cnc(S(C)(=O)=O)s1 80911,c1(C(=O)NCC2CN(C(CNC(C(CC)C)=O)=O)CC2C)cc(C)c(F)c(C)c1 80912,CC1CN(C(=O)COC2CCCC(C)C2)CC1NC(=O)C(N1CCCCCC1)C 80913,c1(NC(C(CC=CC)NC(C2CCCN2C=O)=O)=O)cnc(C)nc1C 80914,C1(CC=C)(NC(C2CC2c2cnc[nH]2)=O)CCN(C(c2cnn[nH]2)=O)C1 80915,N1(C(C(C)SCC)=O)CC(CO)C2(C1)CN(C(=O)C(c1cnn(C)c1)O)C2 80916,N1(C(Cc2c(C)cccn2)=O)CC2CCC1C(NC(c1cc(N)ccc1F)=O)C2 80917,C1(NC(C2(NC(CC3(C)CC3)=O)CCSC2)=O)CC2(CCOC2)C1 80918,Cc1noc(C)c1CSCC(=O)N(CC(C)NC(C1(O)CCOCC1)=O)C 80919,C=CCCC(C(=O)NCc1c(F)cccc1F)NC(=O)C(C)CC(=O)OC 80920,C(=O)(CCCC(=O)N1CC(C2CC2)(C(=O)NC2(C)CCSC2)C1)OC 80921,C12(NC(=O)C(C3CCCO3)C3CC3)CC(NC(C3CC4CC4C3)=O)(C1)C2 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81061,c1(C(=O)NC(C)(C)CN2CCCCC2=O)cnn2cc(F)cc(F)c12 81062,C1(NC(c2c(SC)cccc2)=O)CN(C(C2(C)CCCCO2)=O)CC1S(C)(=O)=O 81063,c1(OCC(N2CCC(OCCNC(C(CC)F)=O)C2)=O)ccc(Cl)cc1F 81064,C(CC(C)(C)CC(=O)N1CC(N(C(=O)CSC2CC2)C)C(F)C1)OC 81065,N1(C(CS(CC)(=O)=O)=O)CCN(C(=O)CCn2cc[nH]c(=O)c2=O)CC(O)C1 81066,C12(C(N3CCC(SC)CC3)=O)CCN(C(=O)CCC=C(C)C)CCC1C2 81067,C1(NC(c2ccc(C3CC3)s2)=O)CCCC12CN(C(=O)COCC1CCOC1)C2 81068,c1(C(=O)NC(CNC(CC(CCC)O)=O)C2CCC2)c(F)cc(F)c(O)c1F 81069,C1(NC(C(C)CF)=O)CN(C(c2cc[nH]n2)=O)C2(CCOCC2)C1 81070,c1(C(N(CC(O)CN(C)C(C2CC3(CC3)C2)=O)C)=O)c[nH]nc1-c1ccccc1 81071,Cc1cccc(Cn2nc(-c3ccc(C(C)C)cc3)nc2-c2ccsc2CO)c1 81072,c1(C(N(CCCNC(C2C(OCC)C2)=O)C)=O)cc(C2CCCCC2)no1 81073,O(NC(=O)C(c1cccnc1)NC(=O)Cc1cn[nH]c1)CC1(C)CC1 81074,c1(C(N2CC(COCC)OCC2)C(=O)NCCC#N)ccc(C#N)c(C)c1 81075,CCCCCCCCC(=O)N1CC2(CC(NC(C3(C)C(C)(C)C3(C)C)=O)CO2)C1 81076,C1(C(=O)NC2(C)CC(C(N(CCOCC)C)=O)C2)CC(C)(C)CO1 81077,C=CCC(C(=O)N(C(C)CCNC(=O)C=CC(C)(C)C)C)OC 81078,CC1(C)CC(CC(=O)NCCCCC(CO)NC(=O)CSc2nc[nH]n2)CCO1 81079,Nc1cc(C(=O)NCC2CN(C(c3cccs3)=O)CC2C(F)(F)F)ncc1Cl 81080,C=CC(C)(C)CC(=O)NCC1CN(C(=O)C(C)=C(C)CC)CCC1C 81081,C(=O)(C1=CCCC1(C)C)N1CCC(C(CNC(c2ccc(C#C)cn2)=O)F)CC1 81082,c1(C(=O)OC)ccccc1CC(C)(CO)n1cc(-c2cc[nH]c(=N)c2)nn1 81083,N1(C(C)C(=O)NC(C(=O)NCCc2cocn2)C2CCOC2)CCNC1=O 81084,N1(CC(CN(C)C)NC(=O)Nc2nc(SC)c(C)s2)CCc2ccccc21 81085,c1(C(=O)NC2CN(C(c3[nH]nc(OC)c3Cl)=O)C2)cccc2sncc12 81086,C(=O)(CC(F)(F)C(C)C)NC1CC(CNC(c2c(C)noc2)=O)C1 81087,N1(C(CC2ON=C(CC)C2)=O)CCN(C(c2cnc(C(C)(C)C)o2)=O)C(CO)C1 81088,C1(C#N)(CNC(C2CC(C(=O)NCCCSC)C2)=O)CC12CCC2 81089,C1(C(=O)Oc2n[nH]cc2C(=O)NC)C2CN(C(=O)Cn3cc(C4CCC4)nn3)CC12 81090,N(C(=NCC1CCOC1)N1CCC(CN2CCOCC2)C1)Cc1c(Br)scc1 81091,C(=O)(C1CCCn2nccc21)NCC1(OC)CN(C(=O)CCc2c[nH]c(=N)[nH]2)C1 81092,Cc1cc(CN2CC(Cc3ccccn3)CC(F)(F)C2)c(Br)cc1F 81093,c1(C(N(c2ncc(SC)cn2)C2CCNCC2F)=O)cc([N+](=O)[O-])c(F)cc1F 81094,C#Cc1c[nH]nc1C(N1CC2CC2(NC(C2CCC(=O)N2)=O)C1)=O 81095,N1(C(c2c(C)n(C)nc2)=O)CC2CCCC2(NC(C2CC=CC(O)C2)=O)C1 81096,c1(CC(N2CC(O)(C3CCCN3C(=O)C=CBr)C2)=O)cccc2ccoc12 81097,CC(CC(=O)NCCCCCNC(C1(O)COC1)=O)c1cccnc1 81098,C#CC1(O)CCCN(C(=O)C(C)(C)CNC(=O)CC2NC(=O)NC2=O)C1 81099,n1(CC)cnnc1CC(=O)NC(C)CC(C)NC(c1ncsc1NS(C)(=O)=O)=O 81100,C1(OC)CN(c2cc(C(C)=O)ncn2)CCC1Oc1ccccc1 81101,C1(OCC(=O)NCC2(CC(=O)N(C)CC3C=CCS3)CC2)CCCOC1 81102,N1(C(CCCNC(C)=O)=O)CC2=C(C1)CN(C(=O)CCOc1cccc(Cl)c1)C2 81103,C1(C(=O)Nc2nccnc2Cl)CC12CCN(C(c1ccc(CCO)cc1)=O)CC2 81104,N1(C(CCOCC)=O)CCCC2(CNC(=O)Cc3cc(F)ccc3F)CC12 81105,CC(C)C(C)(Cc1ccccc1)C(=O)NC1CC1NC(C1CCC(F)(F)CC1)=O 81106,C(=O)(C(C)CCCC(C)=O)NC(CC#C)(C)C(=O)NCCC1(O)CCCCC1 81107,N1(CC(N2CC(F)(CNC(=O)Cc3cc(CO)on3)C2)=O)CCNC(=O)C1 81108,C12(C(N3CC(OC(N(C)C)=O)C3)=O)C(NC(=O)CN3CCOC3=O)C3CC1C2C3 81109,c1(CC)nc(=N)[nH]cc1C(=O)NC1CCC1NC(=O)CSCc1ccccc1Cl 81110,c1(COC)nc(NCC2(OCCO)CCOC2)cc(=NC2CCC(=O)NC2C)[nH]1 81111,N1(C(C(N2CC3C(N)CC(CCC3)C2)=O)=O)CC(F)(F)C2(CCOCC2)C1 81112,C1(CNC(c2scnc2C(F)F)=O)CCCCN(C(=O)CC2CCOCC2)C1 81113,C1(NC(C(C)C2CC2)=O)C2CCC1N(C(c1cccc(-c3nnco3)c1)=O)C2 81114,CC12CN(C(=O)C3=CC4(CCOC4)C3)CC1(C)CN(C(=O)COC(F)(F)F)C2 81115,c1(C(N2CCCCC(NC(=O)C=CCBr)C2)=O)cc(I)ccc1[N+](=O)[O-] 81116,C(=O)(CS(=O)(=O)C1CC1)N1C(CNC(c2cccc3c2CCC3)=O)CCCC1 81117,Cc1nn(C)c(C(=O)O)c1S(=O)(=O)N1CCC2(CC1)CC2(F)F 81118,C(CCF)(C(=O)N(C(C)COC)C)NC(COCCC=C)=O 81119,C12(C(N3CCC(NC(=O)C=C4CCCC4)C3)=O)CCOCC1C2 81120,N1(C(C(C)CO)=O)CC2(C1)CN(C(c1c[nH]ccc1=O)=O)CC2CO 81121,N1(C(C(COCC)N=[N+]=[N-])=O)CCCC2(CCN(C(=O)C=CCF)CC2)C1 81122,C1(C(=O)OC)CCCC(C(=O)NC(C2CCN(C(CC=CCOC)=O)C2)(C)C)C1 81123,CCCC(CCO)N=c1[nH]c(=NCC2CCN(C(=O)OCC)C2)[nH]c2c1COCC2 81124,C1(NC(c2cc(=O)cc[nH]2)=O)CC(NC(C2(N3CCCC3)CCC2)=O)C12CCC2 81125,C(CC(C)C(C)(C)C)NC(c1cc(C#N)n(C)c1)c1n(CCC)nnn1 81126,C1(NC(CC2(C)CCN(C(=O)C(F)C3CCC3)C2)=O)C(O)C2CCOC12 81127,C1(C)(C(=O)NC(c2cncnc2)C)CCCN(Cc2c(C(F)F)nn(C)c2Cl)C1 81128,C1(N(C(C(COC)C)=O)C)CC2CCC(C1)N2C(c1ncccc1C)=O 81129,c1(C(N2CC3ON=C(CNC(C(C)SCC)=O)C3C2)=O)ccc2scc(C)c2c1 81130,c1(C(=O)NC(CN(C(C=CC)=O)C)CC)cc(Br)c2[nH]nnc2c1 81131,N1(C(CC2CCC(C)CO2)=O)CCC2(CC(C(=O)NCC3CCCC(=O)N3)C2)C1 81132,c1(C(=O)NCC2C(OCC)CN(C(=O)C(C)(C)C)C2)cc(C)c(C)cc1N 81133,C1(N(c2nnc(C(F)F)s2)C)CCCN(C(=O)C(C)(C)CC2CCOCC2)C1 81134,N(C1CCc2cc(CNC(C3(Cl)CC3(F)F)=O)ccc21)C(c1cccc(C)n1)=O 81135,N(C1CC2(CCN(C(=O)CC#N)CC2)Oc2ccccc21)C(C(CCC)C)=O 81136,N1(C(=O)CC2CC2)CCCC1C1CCCN1C(C1CC1c1ccccc1)=O 81137,N1(C(C2CCCC(=O)O2)=O)CCCC2(CCCN2C(C23CSC(C2)C3)=O)C1 81138,C(=O)(CC(C)(O)CCC)NC(CC#CC)C(=O)NC1CC(C)N(C)CC1C 81139,N(C1CCSc2ccc(Cl)cc21)C(C1COCCN(C(C2CN(C)C2)=O)C1)=O 81140,Fc1cc(-c2ncc(CN3CCCC(CN4CCOCC4)C3)s2)cc(Br)c1 81141,N1(C(C(CC)N(CC)CC)=O)CCCN(C(c2cc(F)cc(Cl)c2N)=O)C(C)C1 81142,c1(C(N(C(CNC(Cc2c(C)ccc(C)c2)=O)C)C)=O)cc(F)c(Cl)cc1F 81143,C1(CNC(COCCCC#C)=O)CN(C(C2CC(Cl)(Cl)C2)=O)CCC12CCC2 81144,C1(CC=C)(NC(C2CC2C(C)C)=O)CCCN(C(=O)C(C)(C)n2cnc(C)c2)C1 81145,c1(OC)cc(C)c(Cl)cc1CNC(=O)CN1CCC(OCCN(C)C)C1 81146,N1(C(c2cnc(C)[nH]c2=N)=O)CC2(CCN(C(=O)CSc3n[nH]c(C)n3)CC2)C1 81147,c1(NC2C(OC)CN(C)C2)nc(C)cc(=NCC2CC2c2ccc(C)cc2)[nH]1 81148,N1(CCO)CCc2nncn2CC1.c1(C(C)NCCNC(=O)N)nc[nH]c2ncnc1-2 81149,C1(C2CCC(=O)NC2)(C(=O)NC2C(NC(C(C)(C)C#N)=O)CCC2)CCC1 81150,c1(C(=O)NC2CN(C(c3c(C)cco3)=O)C(C)(C)C2)c[nH]c2ccccc2c1=N 81151,C(C(=O)NC(C1CCCC1)CO)(C(C)(C)O)NC(c1c(C)nc(C)s1)=O 81152,c1(SCCC(N2CC(CNC(c3c(CC)non3)=O)(OC)C2)=O)ccccc1Cl 81153,c1(C(=O)NCC2CN(C(c3c(CC)nco3)=O)C2)ccncc1I 81154,n1(C)cc(C(C)(C)C)cn1.C1(NC=O)CCC(CCNC(C2(C3CC3)CCC2)=O)C1 81155,CCCCCC(C(=O)NC1CC2C(NC(C3CC(OC)C3)=O)C2C1)C(C)C 81156,S(=O)(=O)(c1ccccc1Cl)N1CCCC(CNC(c2cnc(Cl)nc2)=O)C1 81157,N1C(=NCCCOC)NCC(C)N(C)C2CC12.c1(CC)ccccc1 81158,CCCCCCC(CC)(CC)C(=O)NCC(C)(O)CNC(C1CC(=C2CC2)C1)=O 81159,C1(NC(N2CCC(c3ccccc3)C(F)(F)C2)=O)COc2ccccc2C1 81160,Cc1oc(C(=O)NC2CC2NC(=O)CCc2ccc(C(C)C)cc2)cc1Br 81161,Nc1c(F)ccc(Cl)c1C(N1CCC(CCNC(C23CCC2C3)=O)CC1)=O 81162,N1(C(C#CC(C)(C)C)=O)CCCC12CCN(C(C1(CCF)CC1)=O)CC2 81163,c1(N2CCC(C(=O)NC3CC(C(F)(F)F)C3)C2)ncc2scc(Br)c2n1 81164,N1(C(CC(C)C)=O)CCC(F)(CNC(C2(n3cnnn3)CCCCC2)=O)CC1 81165,CC1CC(C)CN(C(=O)CN2CCCCC2)C1.C(=O)(CCc1ccon1)NC(C)C 81166,c1(C(=O)OC)ccc(C(=O)NC2CN(C(=O)Cc3cc(C)no3)C2)cc1C 81167,c1(C(=O)NC2C(NC(C=COCC)=O)COC2)ccc2nc(C)n(C)c2c1 81168,Cc1c(Cl)cccc1S(=O)(=O)NC1C2CN(Cc3ccc(Br)[nH]3)CC12 81169,c1(C(=O)NC(CC)CNC(=O)C(c2nccn2C)OC)cc(Cl)ccc1OC 81170,C1(NC(=O)C(c2ccc(F)cc2)CO)CN(C(c2ccnnc2)=O)CC1C(F)F 81171,CC1(C)CCC(CNC(=O)CC2CCCNC2=O)N(C(=O)C=Cc2cnc[nH]2)C1 81172,c1(C(=O)NCC2CN(C(=O)C(F)Cc3ccccc3)CC2O)cc(O)ncc1F 81173,c1(CC)nnc2n1CC(Nc1cc(CC)ncn1)CC2 81174,N1(C(C(C)OCC=C)=O)CC(CO)C2(C1)CN(C(=O)CCCC1CCOCC1)C2 81175,C=CC(C)CN=C(NC(c1ccc(Br)cc1)C)NC1CCS(=O)(=O)C1 81176,C(C(C(C)C(C)C)NC(=O)C=CCCC=C(C)C)NC(C1(CCOC)CCC1)=O 81177,C#Cc1cccc(CNC2(c3nnnn3C(C)C)CN(C)CC2C)c1 81178,CCCC(C)(CC)C(=O)NCC1CN(C(c2cnn3c2N(C)CC3)=O)CCO1 81179,CC#CCCCC(=O)OC.c1(CNC2=NCC3CCN(N2)C3)noc2c1CCC2 81180,C1(CNC(C(C)Cc2ccncc2)=O)CCCCN1C(=O)COC1CCCOC1 81181,O=C1CCC(C(F)C(=O)NC2CC(F)(CNC(=O)COC3CCCC3)C2)CC1 81182,N1(C(CSc2cccc(C)c2)=O)CC2CC(NC(c3cccn3C3CC3)=O)C1C2 81183,c1(C(=O)NC2C(C(=O)NCCOCCC#C)OCC2)cnc(S)nc1 81184,N1(C(COCC#C)=O)CCC2C(CCCN2C(C2Cc3nnc(C)n3C2)=O)C1 81185,C1(C(C)(C)C)(CNC(C2(C)C=CCCC2)=O)CCN(C(=O)C=CCF)C1 81186,C1(NC(c2cc3ccccc3[nH]2)=O)CC2(CCCCN2C(=O)CCC2CC2)C1 81187,CCC(CNC(c1cn[nH]c1)=O)(CC)NC(=O)CCCn1ccnc1C 81188,N1(C(c2onc(CC)c2C)=O)CCC(NC(=O)C=Cc2cocn2)C2(CCC2)C1 81189,c1(C(=O)NCC(CNC(C(N2CCOCC2)C)=O)C)n[nH]c2c1COCC2 81190,c1(C(=O)NC2C3(CN(C(CC(COC)(C)O)=O)C3)CC2)ccc2ncc(C)n2c1 81191,N1(C(C)=O)CCOC(C(=O)NC(C)CCNC(=O)COCc2ccc(C)cc2)C1 81192,c1(CCC)cc(CC)ccc1F.C12CCCC1CNC(=O)C2 81193,Cc1cc(F)c(C(=O)NCCCN(C(=O)CC2CC(F)(F)C2)C2CC2)cc1F 81194,O=C1CCc2c(C(=O)NCCCCNC(c3cc4ccncc4s3)=O)cccc21 81195,C1(N(C(=O)Cn2nnc(C)n2)CC#C)CCN(C(=O)C(C)C(C)C)CC1 81196,C1(C)(CCNC(Cn2c(C)ncc2)=O)CCN(C(=O)Cc2cocn2)C1 81197,CCC(C)CC(C(=O)N1CC2CC=CC1C2)NC(c1cn(C)nc1OC)=O 81198,c1(OC(C(=O)NS(CCCC)(=O)=O)C)cccc2ccccc12 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81758,c1(OC)cnc(C(C(=O)NC2CCCC2)N(CC(F)F)CCCO)cc1Br 81759,N1(C(C2(C)COC2)=O)CCC(O)(CNC(=O)C(O)Cc2c(F)cccc2Cl)CC1 81760,Cc1nncc(C(=O)NC(c2cn(CC3CC3)nn2)C2CC(F)(F)C2)c1C 81761,C1(C(N2CCC(C(N(CCN(CC)CC)C)=O)C2)=O)CC2CCCC2C1 81762,Cc1ccc(C(=O)NCCC(C)NC(c2cn(C3CC3)cn2)=O)c(F)c1Cl 81763,C1(C(N2CCCCC2)=O)C2CC1N(C(C13CCCCC1C3)=O)C2 81764,C1(C(=O)NCCCC(CCC)NC(C2(CF)COC2)=O)CCC2(CCC2)CO1 81765,Cc1cnsc1C(N1CC(F)(CNC(C2CC2c2ccccn2)=O)C1)=O 81766,N1(C(c2cc(OC)ns2)=O)CC2(NC(c3nc(C)ccc3O)=O)CCCC2(F)C1 81767,O(N(CC)C(=O)CN=c1ccnc(Nc2nc(C(N)=O)co2)[nH]1)CC 81768,Cc1cncc(C(=O)NCCC2CSCCN2C(C2CCC(C(N)=O)O2)=O)c1 81769,C(=O)(C(O)CCC(F)(F)F)NC(CNC(CN(CC)CC)=O)(C)C 81770,c1(NC(CC2CC3(CN(Cc4ccc(OC)cn4)C3)C2)=O)noc2c1CCCC2 81771,N1(CCC(=O)NCCC2CN(C(CSCCOC)=O)C2)CCOC1=O 81772,Cc1cc(C(N2CCC(c3cn(C4CC4)nn3)C2)=O)ncc1C(F)(F)F 81773,C1(CNC(CCC=C)(C)c2nnnn2CC)CC2(CCC2O)C1 81774,c1(C(N2CCN(C(c3c(C)ccc(F)c3N)=O)CC2)=O)ccc2c(c1)CC(C)O2 81775,c1(C(N2CCN(CC(C)(C)NC(C(C)OC)=O)CC2)=O)nccc(Cl)c1C 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81917,CC1(CNCC(=O)NC(c2cccc(CO)c2)C2CCCCC2)CCCCO1 81918,C(=O)(CC(C)(C)N(C(=O)Cc1cccnc1C)C)N(CCCC(=O)NC)C 81919,C1(NC(C2CCC(c3ccccc3)C2)=O)CCN(C(c2cnccc2Cl)=O)CC1 81920,C1(NC(c2nccc(C)n2)=O)CC2(CCN(C(C3COC(C)(C)C3)=O)C2)C1 81921,N1(C2N(C(C(C)c3cc[nH]n3)=O)CC2)CCC(C)C(C(F)(F)F)C1 81922,C1(C(=O)NC(c2ccccc2-n2cccn2)C)CC2(CC2)CN1C(=O)C(=O)C(C)C 81923,N(C1CN(C(=O)CC(C)(C)OC)CCc2ccccc21)C(CSCCOC)=O 81924,N1(C(c2cnc(CC)[nH]2)=O)CC(CNC(=O)C(c2cncnc2)C)C(C)C1 81925,c1(C(C(=O)NC(CC)(C)C)N(C)Cc2cc(C)on2)ccc2c(c1Cl)OCO2 81926,c1(OC)c(C(N2CC(C(C)NC(=O)C#CC3CC3)C2)=O)ccc2c1CCC2 81927,c1(OC)cccc(C=CC(=O)NCC(C)OC)c1OC(C)=O 81928,c1(C(=O)NC2(C(N(CCC(C)C)CC(C)C)=O)CC2C)cccn(C)c1=O 81929,C(=O)(C(C)(C)CCNC(C1(F)CCCN(C)C1)=O)N1CC(OCC)C1 81930,C1(NC(C(C)N(CC(F)(F)F)C)=O)CC(C)CN(C(c2cc(Cl)c[nH]2)=O)C1 81931,c1(C(=O)NCCCN(C(C)=O)C)cnc2ccccn2c1=O 81932,C1(CNC(c2c(N)nccn2)=O)CN(C(C2COCCC2(F)F)=O)CCCO1 81933,c1(OC)ccc(C(N2CCC(NC(=O)C=Cc3ccn(C)c3)CC2C)=O)cc1F 81934,C1(N(C)C)C(COC)C1(F)F.C12CC(C1)CC(=O)N(CC(C)O)CCNC(=O)C2.CS 81935,c1(COC)cccc(C(=O)NCC#CCNC(=O)CSc2ccccn2)c1 81936,c1(C(=O)NCC2C(NC(C=C(CC)C)=O)CC2)cnn(CCCC)c1C 81937,c1(C(N2CCCC(C)(NC(=O)C=CC3CCOCC3)C2)=O)cnc2sccc2c1 81938,C1(NC(C2(c3cc(C)no3)CC2)=O)CCC(C)N(C(=O)C(C(C)C)C2CCC2)C1 81939,CC(C(C)C(=O)N1CC(C)(F)C1)NC(c1ccc[nH]1)=O 81940,C(c1cncnc1O)=CC(=O)N(C1CCCC(NC(c2n[nH]c(C)c2Cl)=O)C1)C 81941,c1(C(=O)NCCC(C)(C)NC(C2CC2F)=O)cc(F)c(Br)cc1F 81942,N#CCCCCCC(=O)N1CCN(C(=O)CCF)C(CCO)C1 81943,CC(C)(C(=O)N1CCC(O)(CCNC(C23CC(CCO2)C3)=O)CC1)C(N)=O 81944,CCC(C)(CCC(C)C)C(=O)N1CCCC(CNC(=O)C(C)(C)COC(C)C)CC1 81945,N1(C(Cc2ccc(SC)[nH]2)=O)CCOC2(CCC(NC(c3ccsn3)=O)CC2)C1 81946,C1(NC(C=C(C)C)=O)CN(C(=O)C(N2CCNC2=O)C)Cc2nccn2C1 81947,C#Cc1cccc(C(=O)NCCC(C)(C)NC(=O)COCc2ccccc2)c1C 81948,c1(CN(C(=O)CC=CCNC(C2CC2C(=O)N(C)C)=O)CC)cncn1C 81949,N1(CC(C)(C)NC(C2N(CC)CCC2)=O)CCN(C(=O)Cc2scnc2C)CC1 81950,c1(C(c2nnnn2C)NC(Cc2c(C)noc2C)C)ccc(Cl)cc1F 81951,CC(F)(C(=O)N(CCNC(C1CCCOC1)=O)C1CC1)c1ccon1 81952,C(=O)(C(C(C)O)N(C)C)NCC1N(C(c2ccc(C(C)=O)s2)=O)CC=C1 81953,Cc1ncnc(O)c1C(=O)N(C)CCC1CCCCN1C(=O)CCF 81954,S(=O)(=O)(c1cccs1)NC(CN(CCCNC(C1(O)CCN(C(C)=O)C1)=O)C)=O 81955,C1(CCC)CN(C(=O)CC2CCS(=O)(=O)C2)CCN1C(=O)CN1C(=O)CCC1=O 81956,N1(C(C2(CC#C)CC=CCC2)=O)CCC2(CCCCN(C(=O)CNC=O)C2)C1 81957,Cn1cc(C(=O)NCC(N2CCN(C3CC(F)(F)C3)CC2)=O)c(-c2nn[nH]n2)c1 81958,Cc1noc(C)c1C(C)C(=O)NCC(CNC(=O)Cc1cccnc1)CO 81959,c1(CC)nn(C)c(C(=O)NCCN(C(=O)C(CC)C(C)O)C2CC2)c1Cl 81960,C=CC(C)(C)C(=O)NCC12CC(CN1C(=O)C(C)NS(=O)(=O)CCCC)C2 81961,c1(C(=O)NCC2CN(C(C=C3CCN(C)C3)=O)C(C)(C)C2)csc(S(C)(=O)=O)c1 81962,C(=O)(CC1=CCCCC1)NC1C(C(N2CC(C(C)(C)C)OCC2)=O)OCC1 81963,C1(NC(C2(C)CC2)=O)CC2CCC1CC2NC(C1CCC(CC#N)CC1)=O 81964,S(=O)(=O)(CCCC)NCC(N1CCC(CCNC(C2(C=C)CCC2)=O)C1)=O 81965,C1(C)(CCNC(COC2CN(C(C)=O)C2)=O)CC1(Cl)Cl 81966,N1(C(Cc2n(C)cnc2)=O)CCOCC(CNC(C2(C3CCCO3)CCC2)=O)C1 81967,Cc1noc(Cl)c1CC(=O)NCCCN(C)C(c1c[nH]c(=N)s1)=O 81968,c1(N2CC(SC)C(N(C)C)C2)ncc(C)cc1S(=O)(=O)NC1(CO)CC=CC1 81969,Cc1oc(C2CC2)nc1C(N1CC2C(N(C(=O)CNS(=O)(=O)C3CC3)C)C2C1)=O 81970,c1(-n2c(COc3ccccc3)nc(COC)n2)ccc(F)cc1C(=O)O 81971,c1(C(N(CCNC(c2ccnc(CO)c2)=O)CC2CC2)=O)cccc(O)n1 81972,c1(C(N2CC(C)C(NC(=O)C(c3ccc(F)cc3)(C)F)C2)=O)cccc(Cl)c1N 81973,C1(CC)CN(C(=O)C(F)(F)C(C)O)CCC1N=c1nc[nH]n2c(Br)ccc12 81974,c1(C(N2CCC(N(C(CCC(C)C)=O)CCO)C2)=O)ccc([N+](=O)[O-])cc1 81975,N1(C(c2cc(C)[nH]c2)=O)CC2CCC(C(=O)NCC3=NOC4CCCC34)(C2)C1 81976,CCCC(C(=O)NC(C(=O)NC1CCCCC1N(C)C)C1CCCC1)OC 81977,C1(C(=O)NCCCC(C)NC(c2scc(C)c2Cl)=O)CCC(=O)C(C)C1 81978,N1(C(c2cc(Br)n3c2CCC3)=O)CCCC2C1CCCN2C(=O)CO 81979,c1(C2(C(N3CCC(C(C)(C)N)C3)=O)CCC2)ccc(Cl)c(Br)c1 81980,C1(CC)CCCCCCN1C(=O)CC1CCCN(C(C2CN(C(C)=O)C2)=O)C1 81981,c1(C(N2CCC(NC(C3C(C)C3)=O)CC(O)C2)=O)cccc2nc(C(F)F)[nH]c12 81982,C1(OC)(CNC(C2CC(=O)N(C(C)C)C2)=O)CCN(C(C2CCSCC2)=O)C1 81983,C1(NC(=O)Cn2nnc(C3CC3)n2)CCN(C(=O)Cc2cnc[nH]2)CC1O 81984,C=CCC(CC(=O)N1CCC(CC)(NC(=O)CCCOCC)CC1)NC(C)=O 81985,c1(OCC(N2CC(C(N(CCCCN(C)C)C)=O)C2)=O)cnn(C)c1 81986,Cc1cccc(CC(=O)NCCCCN(C)C(c2c(Cl)nsc2Cl)=O)c1 81987,CON(C)C(=O)CNC(c1c(C(C)C)cnn1C)c1nnnn1CC1CCCO1 81988,N1(C(c2c(C)scc2)=O)CCCC(O)(CNC(=O)C(C)OCC2CC2)C1 81989,Fc1ccc(CNC(c2cc(I)cs2)c2nnnn2C2CCC2)cc1OC1CC1 81990,Cc1ccc(=NCCC(=O)NCC(C)NC(c2cc3n(n2)CCN(C)C3)=O)[nH]c1 81991,n1(COC)ccc(C(=O)NCC2COCC2NC(c2cnoc2C)=O)n1 81992,c1(C(CNC(C(CC)NC(C)=O)=O)NC(=O)CCC2CC2)cccc(C)c1 81993,C(C(=O)NCC(O)CC(=O)NCC(O)C(N)=O)(C(C)(C)C)N(C)C 81994,C(=O)(CCCC(C)CC)NCC1CN(C(c2c(C)cc(CC)o2)=O)CC12CC2 81995,C(CC(C)C(=O)NCC1CN(C(C2(CO)CC(C)(C)C2)=O)C1)=CC 81996,Nc1c(F)cc(-c2ccc(-c3nccn3C3C4CNCC34)c(F)c2)cc1F 81997,c1(N(CCC(=O)N(C)C)C(=O)C=CCN2CCCC2)cnc(O)cc1C 81998,C1(CN(C(CCCSC)=O)C)CCN(C(=O)CCSc2ccccc2Cl)CC1C 81999,C1(C(=O)NCCCCC(C)NC(C2C(C)OCCC2)=O)CCCC2C1C2(F)F 82000,O(NC(=O)C(C1(O)CCCCC1)NC(=O)CCC(C)C)C(C=C)C 82001,c1(OC)ccc(F)c(C(=O)NCCC2CCCCN2C(C2CCC(O)C2)=O)c1Cl 82002,C1(CC(=O)NCC(C)(C)OCCNC(C(C)=C(CC)C)=O)CCCNC(=O)C1 82003,c1(CNC(=O)NC2C(c3ccc(C)o3)C2)cccnc1N1CCCC1 82004,n1(CC)c(C)cc(C(N2CCCC(C)(CNC(=O)C(O)CC(F)F)C2)=O)c1C 82005,c1(NC(=O)NC2(CCCC)CC2)cccc(CO)n1 82006,C12(C(=O)NC3CC4(C(C(=O)NCc5cc(C)n(C)n5)C4)C3)CCC(CC1F)C2 82007,C1(CC(N2CC(COC)(NC(=O)C(Br)=C(C)C)C2)=O)CCOCC1(C)C 82008,N1(C(c2cc(CC)n(CCO)n2)=O)CCN(C(c2ccsc2Cl)=O)C(CC)C1 82009,Cc1cccc2c1ccn2CC(=O)N(C1CN(C(=O)C(F)C(F)(F)F)CC1O)C 82010,N1(C(=O)Cc2cnsc2)CCN(C(C2C3CNC(=O)C23)=O)C(c2ccccn2)C1 82011,Cc1c(C(=O)NC2CCC2CNC(=O)CCS(C)(=O)=O)sc2cncn12 82012,c1(OC)ccnc(C(=O)NC(C)CCNC(=O)C=Cc2ccnn2C)c1N 82013,CCC(CCC(=O)NC1CC(OC)CN(C(c2ccc(F)c(OC)c2)=O)C1)OC 82014,c1(C(=O)NCC(CNC(c2cc(C)cs2)=O)OC)cc(O)n(C)n1 82015,N1(C(c2c(COC)cccc2)=O)CCN(Cc2cc(C)sc2C)C2CC12 82016,N12CC(F)(F)CC1C2.c1(NCc2c(C(OC)OC)cncc2)cccc(Br)c1C 82017,CC1CCC(C)(C=CC(=O)NC2CC3(CCN(C(c4cnc[nH]4)=O)C3)C2)C1(C)C 82018,c1(C(=O)NC)cc(Cl)ccc1NC(C)C(=O)OC(c1ccc(C(C)(C)C)cc1)C 82019,c1(CC)cccc(C(N2CC(O)(C(C)NC(=O)C(O)C(C)C)C2)=O)c1N 82020,c1(CN(c2c(F)cnc(OC)n2)C2CC23CCNCC3)ccc(F)c(Cl)c1F 82021,c1(CCC(=O)NC23CCN(C(c4ccoc4)=O)CCC2C3)cnc2ncccn12 82022,C1(CNC(c2n(C=C)ncc2)=O)CN(C(C2(C#N)CC3CC3C2)=O)CCN1C 82023,C(CCCC(C)(C)C(=O)NNC(=O)CC1CCC(O)C1)CNC(CC(C)(C)C)=O 82024,c1(CNC(C(C2CCOC2)NC(C(F)=CCC)=O)=O)ncnn1C 82025,C12(NC(CC)=O)CCC(C(N3CCNC(=O)C3C(C)C)=O)(CC1)C2 82026,C(=O)(CC(O)C1CCCC1)N1C(CNC(=O)Cc2csc(Br)c2)CC1 82027,c1(NC(c2ccc(C)cc2)CNC(C2(Cl)C(C(C)=O)C2)=O)nc[nH]c2ncnc1-2 82028,N1(C(=O)NC(c2ccccc2)=O)CCN(C(c2occc2Cl)=O)C2CC12 82029,C1(CC(=O)N(C)CC2CN(C(=O)C(C)(C)n3cccn3)C2)(OC)CCCCC1 82030,N(C(=NCCCc1ccc(Cl)c(Cl)c1)NCCCCl)Cc1c(C)cccn1 82031,N1(Cc2c(-c3c(C)cccc3)n[nH]c2)CC(=O)N(C)CC1C(=O)O 82032,CC(C)(C)CCCC(=O)NC1(C)CCCN(C(=O)CC2(O)CCC2)C1 82033,N1(C(C(OC)OC)=O)CC(=O)NCC1C(=O)NCCOCCCF 82034,c1(C(N2CC3CN(C(C(CCC)O)=O)CC32)=O)ccc2cnn(C)c2c1 82035,c1(C(=O)NC2COCCC2NC(C2CCCCO2)=O)ccc2c(c1O)CCC2 82036,C1(NC(CCC=C)=O)CC(C)CN(C(C2CC3(CCC3)CO2)=O)C1 82037,C(=O)(C1CCCc2nn[nH]c21)N(C)CC1CCN(C(CCNC(=O)NC)=O)C1 82038,N1(C(CCSC)=O)CC2C(CNC(=O)Cc3scnc3C)C2C1 82039,Cc1c(F)ccc(C(N2CCOC(CNC(C3(C)C=CCC3)=O)C2)=O)c1Cl 82040,N1(C(C2(NC(C(C(C)C)C(C)C)=O)CCN(C)C2)=O)CC2CCC(C1)C2C#N 82041,N1(C(CC=CCC)=O)CCN(C(c2scnc2C)=O)C2(CCC2)C1 82042,c1(N(C)C)ccc(C(=O)NC2CCC2NC(c2ccncc2F)=O)cc1[N+](=O)[O-] 82043,O=C(NNc1nc[nH]n1)c1ccc2n[nH]cc2n1 82044,C1(NC(c2cnc(CC(C)C)[nH]2)=O)CCSC12CN(C(=O)CCc1nc[nH]n1)C2 82045,C1(C(N2CCCC(OC)C2)=O)COCCN(C2CCCC(C)C2)C1 82046,c1(CC)ccc(CCCC(=O)NC2CCN(C(C3CC34CCC4)=O)C2)cc1 82047,c1(N2CC3C(NC(C(CC)CCOC)=O)C3C2)c(Br)cccc1[N+](=O)[O-] 82048,c1(C(N(CC(C)(C)NC(CC2CC(OC)C2)=O)C)=O)csc(C(F)(F)F)n1 82049,n1(CC(=O)NC2C(C)N(C(=O)CC(C)c3ccncc3)CC2)nc(O)ccc1=O 82050,C(N=c1[nH]c(C)ncc1F)C1C(NC(C=CCC)=O)C2(CC1)CCC2 82051,N1(C(Cc2cnc(C)o2)=O)CCCC2(CCC(NC(C3(C)CC(F)(F)C3)=O)C2)C1 82052,C1(C(=O)NC2CC(C(=O)NC(C(C)C)C)C2)(CF)CCOCC1 82053,Cc1cc(N)ccc1C(N1CCC(O)(CCNC(c2ccnc(CO)c2)=O)C1)=O 82054,c1(C(N2CCCC(Nc3cc(C)nc(C)n3)C2)=O)cc(C)c(F)cc1F 82055,C1(C(N2CC(CNC(=O)Cn3cncn3)C2)=O)CC(O)CN1c1ccncn1 82056,N1(C(C2CCC(CNC(CC(C)F)=O)C2)=O)CCOC2(CCCC2)C1 82057,C1(N(C(C2CC(CC)(CC)C2)=O)C)CCCC(NC(=O)C=Cc2nccs2)C1 82058,C(=O)(CC(C)(C)CC(=O)NCC(C)NC(C1CCC1(F)F)=O)OCC 82059,c1(C(N2CC(NCCNC(=O)OC(C)(C)C)CC2C)C(=O)NC)nc(C)n(C)n1 82060,N1(C(c2c(OC)ccc(C)n2)=O)C(CNC(=O)C(C2CC2)OC)CC2COCC12 82061,N1(C(C(n2cc(C)nc2)(C)C)=O)CCCCC1CCNC(C1CC2(C1)CC2F)=O 82062,N1(C(C2C(C)CCO2)=O)CCOC2CCN(C(c3ccc(N)cc3O)=O)CC12 82063,CC(CC(F)F)C(=O)NCC1CCCCN1C(=O)CCCNC(N)=O 82064,N1(C(c2scc(C)c2)C(=O)NCCCF)CCN(Cc2ccccc2)C(=O)C1 82065,c1(OC)cc(F)c(S(N)(=O)=O)cc1C(N1CCC(n2cc(C(N)=O)nn2)CC1)=O 82066,n1(CCOC)cccc(C(N2CCOC(C3CCCCC3)C2)=O)c1=O 82067,C1(CC#C)CCN(C(C2CCC(NC(=O)CCC3CC3C)CC2)=O)CC1 82068,C1(C(=O)NC2(CF)CN(C(C3C(C)CCC3)=O)C2)COCCN1C=O 82069,N1(C(C2N(Cc3ccc(C#N)s3)C3C(C2)C3)=O)CC2CCC(C1)O2 82070,c1(N(C2CCN(C(c3cccc(C4(C)CC4)c3)=O)C2)CCO)ncc(Br)cc1C#N 82071,C12(C(=O)NC3(C)CC(NC(C(C)Cc4ccncc4)=O)C3)CCC(C1)OC2 82072,N1(C(C2(CCC=C)CN(C(C3C4C5CCC(C5)C34)=O)C2)=O)CC(O)C(C)(C)C1 82073,C(=O)(C(C(C)C)NC(=O)CC(C)F)NC(C(=O)NCC)CO 82074,c1(C(=O)NCC(c2ccccc2)NC(=O)CCC2CC2)cnn2c1OCC(O)C2 82075,C1(C(=O)NCC(CNC(=O)CCc2ccc(Cl)cc2)F)NC(=O)C2CCC12 82076,N1(C(c2cnc(OCC)nc2)=O)CC2CC(NC(C3C4CCC3CC4)=O)C2C1 82077,c1(C(C(=O)NC(C)C(CO)NC(c2ccc(CO)o2)=O)O)ccc(F)cc1 82078,c1(C(=O)NCC(C)=CC(=O)NC(C)CC2CCCCO2)cc(F)n(C)n1 82079,C1(CC(=O)NCCC(CCC)O)C2CCC(C2)N1C(C1CC(=O)C1)=O 82080,C(=O)(CCCCCN(C(=O)C(F)C(C)(C)O)C)N(CCC#C)CCO 82081,N1(C(C(C=C)(C)CC)=O)CCC(N(C(=O)CCOc2ccccc2)C)C2(CC2)C1 82082,Cn1cc(C(=O)NCCC2CCN(C(=O)C(C3CCCO3)C3CC3)CC2)nc1O 82083,C1(OC(c2cncc(OC(C)(C)C)n2)=O)CCC=CCCC1 82084,C(c1cccc(Cl)c1)=CC(N1CC(NC(c2ccc(OCC)nc2)=O)C(O)C1)=O 82085,C1(NC(C2CCCC3(CCC3)C2)=O)CN(C(C2CC(F)(F)C2)=O)C2CCCCC12 82086,N1(C(Cc2ccc(OC)cc2C#N)=O)CC(NC(=O)C(F)(F)F)CC12CCOC2 82087,c1(CC(=O)NC2CCCC(CNC(COC(CC)C)=O)C2)ccc(C#N)nc1 82088,CC1CCOCC1C(=O)NCC1(C(=O)NC2CC(=O)N(O)C2)CCCCC1 82089,c1(CC(N2CC(CC)N(C(=O)C(C)C(C)C)CC2)=O)cnn2c1CCCC2 82090,O=S(=O)(c1ccc(Br)cc1NCCCCCCSC)NCC1(c2ccon2)CC1 82091,c1(CC(C)NC(C2CCCC2)C)ccc2c(c1)CCCC2 82092,C1(CNCC2CC=CCC2)CCCN(CCc2ccccc2)C1 82093,C1(C(=O)NCC(CNC(c2ccc(C(=O)OC)cn2)=O)O)C(F)(F)C12CCC2 82094,c1(C(=O)OC)ccc(C(=O)NC(CNC(=O)CC(C)C2CC2)C(C)C)o1 82095,C1(C(N2CCC(O)(CNC(COCC(C)(C)C)=O)C2)=O)CC2(CCCC2)CO1 82096,c12cccc(c1)C2.C(=O)(CC(C)(O)c1cn(CC(=O)O)nn1)N(CCCSC)C 82097,c1(C(=O)NCc2ccc(C(C)NC(CC(C)SC)=O)cc2)ccc2nn[nH]c2n1 82098,N1(C(c2cc(C)no2)=O)CC(C)N(C(=O)CN(C(=O)C(C)C)C)C(C)C1 82099,C(N=c1cccc(S(=O)(=O)NC2CCCc3occc32)[nH]1)C1C(C)(C)CCO1 82100,c1(-c2ccn(C)n2)cc(C(=O)Nc2cc(Cl)nc(Cl)c2)cc2cc[nH]c12 82101,Cc1cc(C(=O)NCc2n[nH]cc2C(=O)N(C)Cc2cnn(C)c2C)c(C)nn1 82102,CC1CCN(C(=O)Cn2[nH]cnc2=N)CCN1C(c1ccn2nccc2n1)=O 82103,N1(C(C(COC)N(C)C)=O)CC2CC3CC2C1C3NC(=O)CCN1CCCCC1 82104,c1(NC2C(C(=O)OCC)CNCC2)ccc(-n2cccc2)c(Cl)c1 82105,c1(NC(CC)=O)nc(C)c(C(=O)NC2CC(C)(C)C2)s1 82106,C(=O)(CCC(=O)NCC1(C(=O)NCc2ccn(C)n2)CC1)NCCC 82107,c1(OC)cc(C)c(Br)cc1NC(=O)C(C1CC1)(OC)OC 82108,c1(NC(C2C(C(=O)Nc3cc(C(C)(C)C)[nH]c3)C2)=O)c(O)cccc1Cl 82109,c1(C(=O)NC(C(=O)NC2(CO)CC(C)C2)c2cccs2)cc(C#N)cs1 82110,CC(CC1CCC1)N=c1[nH]c(=NC2CCn3c(O)nc(C)c3C2)[nH]c2ccsc12 82111,c1(C(=O)NCC2C(CNC(C34CCCCC3C4)=O)C2(F)F)ccc(F)cc1F 82112,N1(C(CC2CC(C)(C)OCC2)=O)CC2(CCN(C(=O)CC3COC(C)(C)C3)C2)C1 82113,C1(NC(CC2CC(COC)C2)=O)CCN(C(c2c[nH]c(C(=O)OC)c2)=O)C(C)C1 82114,Cc1ccc2nc(C(N3CCN(C(=O)CC4(CO)CC4)C(CF)C3)=O)cn2c1 82115,C1(CNC(Cc2ccc(SCC)cc2)=O)CCCCN(C(C2OCCCO2)=O)C1 82116,CC1(C)C=C(C(=O)Nc2nc(CC(=O)Nc3cncc(Cl)c3Br)cs2)C1 82117,C1(CNC(c2c(C)cnn2C(C)C)=O)CN(C(=O)CCCC2CC2C)CC1(F)F 82118,c1(C(=O)NCCN(C(C2CCC(C)O2)=O)CC)ccc(N)c(C(F)(F)F)c1 82119,C1(C)(OC)CCC(NC(C2CC(NC(=O)CC3CC(C)(C)CO3)C2)=O)CC1 82120,COn1cnc(C)c1C(=O)NCc1nc(C)c(C(=O)NCC2C=CCC2)o1 82121,CC1(NC(=O)Cc2csc(S)n2)CCCN(C(C2CCCC2(F)F)=O)C1 82122,N1(C(C(C)OCCOC)=O)CC(CNC(=O)CC(N2CCC(C)CC2)=O)C(O)C1 82123,C(c1cnn(C)c1)=C(C(=O)NC(CCOC)CNC(c1cncn1C(C)C)=O)C 82124,C(CNC(=O)Cc1cccs1)(CC(=O)NCCC1CC(F)C1)OC 82125,n1(C(C(=O)N)C)cc(C2(N(C)C)CCC2)nn1.CC(C)N(C(N)=O)C(C)C 82126,C1(OC)CC2CCC1CC2C(=O)NC1CN(C(=O)C(C)Cc2ccc(F)cc2)C1 82127,c1(C(CF)NC(=O)NCC2(C(C)C)CC2)cccc(OCC#N)c1 82128,c1(C(N2CC3CCN(C(C4ON=C(C)C4)=O)CC32)=O)cnc2ccc(F)cc2c1 82129,C1(CNC(C2(OC)CCCCC2)=O)CC2CN(C(C3CCN(OC)CC3)=O)CC12 82130,c1(CC(=O)NCC2(NC(c3c(C)nn(C)c3)=O)CC2)ccc(F)c(Cl)c1F 82131,C123CCC(CC1)N2C3=O.c1(C(=O)NC(C2CC(CC)C2)=O)c[nH]nc1OC 82132,c1(NC(CC2(C)CCN(C(C=C)=O)C2)=O)cc(Cl)c(N=[N+]=[N-])cc1C(=O)OC 82133,C(=O)(C(CO)C(F)(F)F)NCC(C1(O)CCCCC1)(C)C 82134,c1(C(N2C(CC(=O)NCCCc3cc[nH]n3)COCC2)=O)occ2c1CCC2 82135,C1(CNC(CN(C)C2CC2)=O)CN(C(=O)CC2NC(=O)NC2=O)CCC1(C)C 82136,C1(C(C)NC(=O)C(C)(C)C2CCCC2)CN(C(C2COCCO2)=O)CCO1 82137,Cn1cc(C(N2CCN(C(=O)COC3(C)CCCC3)C(C3CC3)C2)=O)ccc1=O 82138,C12C=CCCN1C2=O.C=C1CCC1C(=O)NC1CC1C(=O)OC(C)(C)C 82139,C1(CC(N2C(CCN(C)C(C3CCCS3)=O)CCCC2)=O)CCC2(CC1)CC2 82140,c1(CC)nc(N2CCC(NC(=O)CSCCN(C)C)C(F)C2)c(C)c(Cl)n1 82141,Cc1sncc1C(=O)NCC(C)C(=O)NCCNS(N)(=O)=O 82142,c1(C(=O)NC(C2CN(C(=O)COC(C)(C)C)CCO2)C)noc2cc(F)ccc12 82143,C1(C)(C(N(C2CCCN(C(C3(C#N)CCCC3)=O)CC2)C)=O)CCC(=O)NC1 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82284,N1(C(c2c(C)cn(C)c2)=O)CCC(CO)(CNC(c2cnc(S)[nH]2)=O)CC1 82285,CCCCCC(O)C(C)C(=O)NCCC1(CNC(c2ccnn2CCC)=O)CC1 82286,Cc1cc(C(=O)C(=O)NC2CC2NC(=O)C=CC2CC2)ccc1F 82287,C1(NC(C(=O)NCCC(N)=O)=O)CC(F)(CNC(c2csc(C(F)(F)F)n2)=O)C1 82288,C1(CNC(=O)CCC2CCCO2)CC(NC(c2cc(CO)on2)=O)C(O)C1 82289,c1(NC(C23C(CN(C(c4c(C)cc[nH]4)=O)C2)C3)=O)cccc2c(O)nnc(O)c12 82290,c1(C(=O)NC2(CF)CCN(C(c3ncc(CC)nc3)=O)C2)cc2ccncc2s1 82291,N1(C(CN(C)C2CC2)=O)CCOC2(C1)CN(C(C1(C)CCC1)=O)C2 82292,C1(NC(c2c(C(C)C)n[nH]c2)=O)CC2(C1)CC(NC(C1CCCC(C)O1)=O)C2 82293,C(CN=c1[nH]c(=NCc2ccc(SC)o2)[nH]c2c1COCC2)(c1ccsc1)OC 82294,CON(CCO)C(=O)C1CCCCCN1C(c1csc(C#N)c1)=O 82295,C1(CNC(C(C)CF)=O)CN(C(c2cc(C(F)F)on2)=O)CCC12CCC2 82296,C1(C)(C(=O)OC)CN(C(c2ccc(O)nc2Cl)=O)CC1(F)F 82297,CC(C)C(C(=O)NC1CCN(C(c2cc(C(N)=O)co2)=O)C1C)n1cncn1 82298,C(c1cccc(F)c1)=CC(N1CC(NC(c2cnc(O)s2)=O)C(O)C1)=O 82299,c1(OC)ccc(C(C)CC(=O)NCC(O)CNC(=O)C(C)O)cc1 82300,C(c1cc[nH]c1)=CC(=O)NCC=CC(=O)NCC1CC1Cl 82301,C1(NC(C(CSC)OC)=O)COCCC1NC(C1CC(C)(C)C1)=O 82302,C#Cc1ccc(Br)c(C(=O)NC2CCC(C)(C)CC2CNC(=O)C=CC)c1 82303,C1(C(=O)NC(CC(C)NC(C2COC(=O)O2)=O)C)CN2CCN1CC2C 82304,c1(N(C2CCN(C(c3ccc(C)c(F)n3)=O)C2)C)ccc2c(n1)CCC2=O 82305,C1(C)(CC)CCCN(C(=O)CC(C)NC(c2csnc2C)=O)CC1 82306,C(C)(N=c1[nH]c(Cl)ncc1C1CC1)C1N(C(Cc2nnn(CC(C)C)n2)=O)CCC1 82307,Cc1cc2cc(NC(C3CCC(F)(F)CO3)=O)ccc2n(C)c1=O 82308,C1(N(C)C(c2cc(S(N)(=O)=O)co2)=O)COC2(CCN(C(=O)C(C)(F)F)CC2)C1 82309,C1(N(C(=O)Cc2ccnnc2O)C)CCCCN(C(=O)C=C2CCOCC2)C1 82310,c1(NCCCCOCC)cc(C)c(S(=O)(=O)N2CCCCC(C)(C)C2)cn1 82311,C1(C(N2CCN(c3cccc(OC)n3)CC2)=O)Cc2ccccc2CN1C 82312,C12(NC(=O)Nc3scc(-c4cc(SC)cc(F)c4)n3)CC3CC(CC1C3)C2 82313,O(C=CC(=O)NCC(C)N(C)C(c1ccn(CC)n1)=O)CC 82314,C1(NC(C2(CC)CCC2)=O)CC2CC(NC(=O)C(C)(O)Cc3ccccc3)CC2C1 82315,Cc1ccc(F)cc1C(=O)N(CCC(=O)NCC(CNC(N)=O)ON)C 82316,C1(F)(C(=O)NCC(C)(CO)NC(C(CSC)OC)=O)CCCCCC1 82317,C1(NC(CCCOC)=O)CCC(NC(c2cccc(OC(C)C#N)c2)=O)CC1 82318,C(CCCC(=O)NC1CC(=O)N(C(C)C)C1)NC(COCCSC)=O 82319,CC(O)C(C(N)=O)NC(C1C2CC1N(C(=O)CN1CC(=O)NC1=O)C2)=O 82320,C1(C(=O)NCC2CCC2NC(C2(CC3CC3)CCC2)=O)CCC2(CC1)OCCO2 82321,CC(C)CC(C(=O)N1CCCC(O)(CO)C1)NC(=O)CN(C)C(=O)C1CC1 82322,N1(C(C(F)OC)=O)CC(O)(CNC(=O)CCCC2CC2)C1 82323,c1(N(CC)CC)cccc(N=[N+]=[N-])c1.C1(C=O)CCN(C(C2CCCO2)=O)C1 82324,C12(NC(c3ccc(C#N)o3)=O)CCN(C(c3nocc3Cl)=O)CC1C2 82325,Cc1c(C(N2CCN(C)CC2CNC(=O)C(O)C(C)(C)C)=O)cccc1CO 82326,C(=O)(CC(C)C(F)(F)F)NCCC(C)NC(=O)CSCc1ncc[nH]1 82327,C1(CNC(Cc2cnn(C)n2)=O)CCCC(NC(c2coc(CO)c2)=O)C1 82328,C1(NC(c2cc(NC)nc(Cl)c2)=O)CN(C(C2CC3C=CC2C3)=O)CC(C)(C)C1 82329,N1(C(CC(C)SC)=O)CC(CNC(=O)C=CCCc2ccccc2)C(O)C1 82330,c1(OCC(N2CC3C(NC(COCCC)=O)C3C2)=O)cc(Cl)ccc1C(C)C 82331,n1(CCN(C)C)cc(C(=O)NCC2(NC(C3C4COCC34)=O)CCOC2)nn1 82332,CCC(C)CCC(=O)N(C(CC)CC(=O)N1CC(F)(F)C1C1CC1)C 82333,N1(C(CC(C=C)C)=O)CC2(C(=O)N(C(C)CC(N)=O)C)CC1CCO2 82334,c1(OC)ccccc1CC(N1CCC(NC(=O)CCN2CCNC(=O)C2)C1C)=O 82335,N1(C(CCc2ncc(C)[nH]2)=O)CCCC(NC(=O)CCC2OCCO2)C1C 82336,Cc1cc(C#N)ccc1C(=O)NC(C(=O)NCc1c[nH]nc1C(C)C)C1CC1 82337,CC(C)(CCCF)C(=O)NC1CCCCC1CC(=O)NCC1(C)CC2(CCC2)C1 82338,N1(C(CS(=O)(=O)NC)=O)CCC2C(C1)NC(=O)CN2C(c1cc(C2CC2)no1)=O 82339,c1(CN(C)C(=O)NC2COC3(CCOC3)C2)nc2ccccc2[nH]1 82340,C(C(C(=O)NC1(C(F)(F)F)CCC1)C(C)(C)C)NC(CCC(C)(C)N(C)C)=O 82341,c1(OC)cc(C(N2CCOCC2CNC(C2C=CC=CC=C2)=O)=O)ccc1C 82342,C1(N=[N+]=[N-])(C(=O)Nc2c(C)cccc2F)CCN(C(c2csc(C)c2C)=O)C1 82343,C(=O)(C1CCCc2nncn21)N(C(COC)OC)CC(OC)OC.c12ccc(o1)OC2.OC 82344,C12(CNC(C=CC(C)(C)C)=O)CC(NC(c3cc(O)nc(O)n3)=O)(CCO1)C2 82345,N1(C(c2c(C)nc(C)[nH]2)=O)CC(N(C)C(C2CCCSC2)=O)C(C)(C)C1 82346,CCC1=C(C(=O)N2CCC(n3cc(-c4cc(F)ccc4OC)nn3)C2)CCCO1 82347,N1(C(C(CCCC)F)=O)CCC2(C1)CN(C(c1ccc(CCC(N)=O)cc1)=O)C2 82348,c1(COC)ccnc(C(=O)NC(C)(CNC(c2cc(C)c(C)s2)=O)C2CCC2)c1 82349,C=CCC(C)C(=O)N(CCCNC(c1ccc(OC)cn1)=O)C(C)C 82350,C(=O)(C(CCC)NC(=O)CC1CCCOC1)NC(CC=CC)CO 82351,CC1(C)CN(C2CCN(C3CCC3)C2=O)CCC1NC(=O)CCC1CC1 82352,C1(CN(C)C(c2cc(CO)n(C)n2)=O)CCN(C(=O)COCC2CCOC2)CC1 82353,CCC(CNC(=O)CCCc1nc(C(C)C)no1)(CC)NC(c1nc(O)sc1C)=O 82354,CC#CCC(C(=O)N1CC(c2ccccc2)C1)NC(C1CC2CCC2C1)=O 82355,C1(CC(=O)NCC(CSC)OC)CCN(C(c2nc[nH]n2)=O)CC1 82356,C1(C(=O)NCCC(O)CNC(=O)C(C2CC2)C2CC2)CCCS1(=O)=O 82357,CCC(CSC)N=c1[nH]c2c(c(=NCc3cccc4sccc34)[nH]1)CSC2 82358,N1(C(C(C)N(CCC)C(c2cc(Cl)no2)=O)=O)CCCCCC1C 82359,N1(C(C(C)OC)=O)CCN(C(=O)CSc2cccs2)C(C2CCCC2)C1 82360,C(=O)(CC(F)(F)CC(=O)N1CCCC1(C)CNC(C1CCC(C)CC1)=O)OC 82361,C1(CCNC(c2nn(C)c(C(N)=O)c2)=O)CN(C(=O)C(C)(C)C)CCS1(=O)=O 82362,c1(C(CC)(C2CC2)NCC(C)(C)N2CCCC2)nnnn1CCOCC1CC1 82363,Cc1cccc(C(=O)NCC2(F)CCC(NC(=O)C(c3ccccc3Cl)C)C2)n1 82364,C12(NC(=O)CCc3ncccn3)CCCN(C(c3cncc(F)c3)=O)CC1C2 82365,Cc1nccc(C(=O)NC(C)CC(C)NC(=O)C(C)Sc2ccccn2)c1C 82366,C1(NC(COCCOC)=O)CN(C(=O)C(c2cccc(Cl)c2F)(C)C)CC12CC2 82367,N1(C(c2c(CC)n(C)cc2)=O)CCC(C)(NC(c2cccc(OC)c2N)=O)CC1 82368,N#CC1(C(N2CCC(O)(c3nc(C4CC4)no3)C2)=O)CC12CCCC2 82369,N1(C(c2c(C#N)scc2)=O)CCC2(CCN(C(C3CCCCC(F)(F)C3)=O)C2)C1 82370,n1(-c2ccc(COC)cc2)ncc2ccc(NC(c3ccc(F)cc3F)C)cc12 82371,C1(C(N(C)Cc2ccon2)=O)C2CC1N(C(c1csc(F)c1)=O)C2 82372,Cc1cc(Br)c(S(=O)(=O)NCC2(CO)CC23CCOCC3)cc1Br 82373,c1(NC(CCC(C)NC(Cc2c(C)con2)=O)=O)cnc(F)cc1C 82374,CCCC(C(=O)NC1(CO)CCN(C(c2ccc(OC)c(C)c2)=O)C1)S(N)(=O)=O 82375,CC(CC(=O)NCCc1ncnn1C)C(C)(C)NC(=O)C=CC1CC1 82376,N1(C(c2n(CC)cc(Cl)c2)=O)CCC(CNC(=O)COCC2CCCOC2)C1(C)C 82377,C(C(C)(C)CNC(=O)C(C1CC1)NC(c1ccc(Cl)s1)=O)SC 82378,C1(C(=O)NCCN(C(=O)C=CBr)CC(C)O)CN(C)CCN(C)C1 82379,Cc1c(C(=O)NCC(C)(C)NC(C2CCCS2)=O)ccc(F)c1F 82380,C12(NC(=O)CC3CCC=CCC3)CCN(C(c3cnn(C(F)F)c3)=O)CC1C2 82381,C1(C(N(C)CC2N(C(C3(C)ON=C(C)C3)=O)CCC2)=O)CCCC12CCC2 82382,c1(NC(CC)CNC(c2cc(O)n(C)n2)=O)nc2c(cc1C#N)COCC2 82383,C(N=c1[nH]c(=NCCCCOCC(C)C)[nH]c2c1SCC2)C1C(C=C)C1 82384,Cc1cnc(C(=O)NCC2CCN(C(=O)C=CC3CCCC3)CC2)cc1C#N 82385,c1(N(C(=O)NC(CC)C#N)C)ccc(Cl)c(Cl)c1.C12CC(C1)O2 82386,c1(C(=O)NC2(C)CC(NC(COCCOCC)=O)C2)cnc2[nH]c(=N)sc2c1 82387,C#CC1(NC(c2ncnc(C)c2C#N)=O)CCCC(C)(C)C1 82388,C12CCCCN1N1CCCC1CC2.CP(C)(=O)COCC1CC(OC)C1.CC=O 82389,C1(C(N2CC(CCCCNC(c3cc(C(C)C)[nH]n3)=O)C2)=O)COCC(C)O1 82390,C1(CC(C)NC(C2CCS2(=O)=O)=O)CCN(C(=O)CCc2cccs2)CC1 82391,Cc1ccc(F)cc1CNC(C1(C#N)CC1(C)C)=O 82392,C1(CCCC)CN(C(=O)CCNC(N)=O)CCN1C(=O)C=C(C)c1cccnc1 82393,c1(OC)ccc(C)c(C(=O)NC2CC2NC(=O)CC2CCC(OC(C)C)CC2)c1 82394,Cc1nonc1CC(=O)N(CCCn1cc(C(O)C2CC2)nn1)Cc1ccccc1 82395,c1(C(=O)NC(C(C)NC(Cc2c(C)scc2)=O)C)cccc(-c2nc(O)n[nH]2)c1 82396,Cc1cc(C(=O)NCC2(O)CCN(C(c3c[nH]cc(C)c3=O)=O)CC2)ccc1Cl 82397,N(C1CCCn2nccc21)C(c1c(CNC(c2nc(C)c(C)s2)=O)ccs1)=O 82398,CC1(C)CN(C(=O)C2=COCCC2)CCN(C(=O)C(C)(C)c2ccns2)C1 82399,c1(NCC=CCNC(c2c(C)nc(-n3cccc3)s2)=O)ncccc1[N+](=O)[O-] 82400,c1(C(=O)NC2(C)CCN(C(COCCCC)=O)C2)cc(C#N)c(N)cc1O 82401,S(=O)(=O)(c1ccccc1N=[N+]=[N-])NC1CN(C(C)=O)C1 82402,c1(C(=O)NCC23C(CN(C(CC4(C)OCCO4)=O)C2)C3)cc2cc(Cl)ccn2n1 82403,C(=O)(CC(C)n1cccn1)NC1CC(CCNC(CSC)=O)C1 82404,c1(SC(C(=O)NCCC(C)NC(=O)C(C)(C)N(C)C)C)nc2ccccc2[nH]1 82405,c1(C(=O)NC2CCCCN(C(C(CCC)OC)=O)C2)coc(=O)c2ccccc12 82406,C(=O)(CCCCCN(C)C(C1CC1[N+](=O)[O-])=O)N1CC(CCC#C)C1 82407,N1(C(c2cnsc2)=O)CCC2(CCCN(C(C3CC34CC(O)C4)=O)C2)C1 82408,c1(C(N2CCC(O)(C(C)NC(c3cccc(O)n3)=O)C2)=O)occ2c1CCC2 82409,CC(C(C)(C)C(=O)N1CCC1C1CCCC1)NC(=O)CC1C=CCC1 82410,C1(NC(CNS(CCCC)(=O)=O)=O)CCN(C(c2ccc(O)nn2)=O)CC1CC 82411,N1(C(CCC(C)OC)=O)CCC2CCC(C1)N2CC1CC1(C)C 82412,C(=O)(C1=CCC(C)(C)CC1)NC(C1CN(C(c2cnncc2O)=O)CCO1)C 82413,c1(CCNC(C2CN(C(C3C(c4n(C)cnc4)C3)=O)C2)=O)cccc2c1OCCN2 82414,N1(C(C2C(NC(Cc3n(C)ncc3)=O)CCO2)=O)CCCC1(CO)CO 82415,c1(C(=O)NCCNC(=O)NCCc2csc(C3CCCN3)n2)ccccc1 82416,CCCCCCCCC(C)C(=O)N1CC=C(CCNC(C2CCCSC2)=O)CC1 82417,C(CC(F)F)(C(=O)N1CC=CCO1)NC(c1ccc(CC#N)cc1)=O 82418,C(=O)(N1OC2CCC1CC2)C1C(c2c(C)occ2)C1.c1(CN)cccc(O)c1F 82419,c1(N2CC(O)(CCNC(c3cncn(C)c3=O)=O)C2)nc(O)c2c[nH]nc2n1 82420,N1(C(CC2N(C)CCC2)=O)CCOC(CC(=O)NCC2(C(=O)OC)CCC2)CC1 82421,C1(C(=O)NC2(CC3CC3)CC2)CCN(C(=O)C=C(C2CC2)C2CC2)CCO1 82422,CC1(C)CC(C)(C(N2CC3(C2)CC3(F)F)=O)CN1C(=O)CCCC1CCC1 82423,C(=O)(C1SCCc2ccccc21)N1CCN(C(C=C=C(C)C)=O)C(CCO)C1 82424,C(C)(CC(C)C(F)F)NC(CCCCNC(C1(CC)CC(C)(C)C1)=O)=O 82425,c1(CC(=O)NCCCCNC(CCC(=C)Br)=O)c(F)cccc1C#N 82426,Cc1ccc2[nH]c(C(N3CCCC(N(c4ncnc(=N)[nH]4)CCO)C3)=O)cc2c1C 82427,CCCC(CC(=O)NCCCCCCO)NC(=O)C=Cc1cncs1 82428,N1(C(C2C(CC)N(C(=O)C(C)OCC3CC3)CC2)=O)CCC(C)CC1C 82429,N1(C(c2ccc(CC)o2)=O)C(CNC(=O)COCc2ccnn2C)CC2CC12 82430,C1(NC(C23CC(C)(C2)C3)=O)COC2(CCN(C(c3cc(Cl)c(F)cc3N)=O)C2)C1 82431,N1(C(CCC(=O)N(C)C)=O)CCN(C(C2CCC(C(C)(C)O)CC2)=O)CC(O)C1 82432,Cc1ccc(N2CCC(NC(C3(F)CCCCC3)=O)C(O)C2)c([N+](=O)[O-])c1 82433,Cc1ccc(C=CC(=O)NCC2CN(C(=O)CCC3COC(C)(C)O3)C2)c(C)c1 82434,C(C(C)NC(=O)C(C)(C)n1cc(Cl)cn1)(C(C)C)NC(Cn1ccc(C)n1)=O 82435,c1(OC)nccc(C(=O)NCC(C)N(C(=O)CC(O)C(C)C)C)c1F 82436,C1(C(N2CC3(CC3)C2)=O)CCCN1C(C1CC(O)CN1)=O 82437,NC(C(=O)NNC(=O)c1ncon1)c1c(F)cccc1Cl 82438,c1(-c2n(C)ncn2)ccccc1CNC(=O)Nc1ccc(F)nc1 82439,c1(C(=O)NC2CC(C(=O)O)CN(C(C(CC(N)=O)O)=O)C2)n[nH]c2c1CCSC2 82440,O=C1NCC2(CO1)CN(C(c1ccc(Br)c(Cl)c1Cl)=O)C2 82441,N1(C(=O)CCc2ccco2)CCC(C2CN(C(c3cccc4nncn34)=O)C2)C1 82442,C1(NC(CCC#C)=O)CN(C(=O)CSc2nnc(-c3ccccn3)o2)CC1C 82443,c1(CC)ccc(C(=O)N(C2CCN(C(C3CCCC(CF)C3)=O)C2)C)cn1 82444,n1(C(CC)C)ncc(C(=O)NCC(CC(C)C)NC(=O)C=Cc2cnc[nH]2)c1C 82445,C(CO)(CCC(C)C)NC(CC(C)(C)N(C(CSCC#C)=O)C)=O 82446,C(=O)(C1=CC(c2ccccc2)NC(=O)N1)N(CC(=O)O)Cc1cnccn1 82447,C(c1cn(C)cn1)=CC(=O)NC1CCN(C(c2nc(CC)oc2)=O)C1 82448,C1(NC(C)=O)CCCN(C(C2CC(O)(CNC(c3ccn(C(C)C)n3)=O)C2)=O)C1 82449,CC1(c2cn(C3CCC(C(=O)NCCC4(O)CCCC4)C3)nn2)CCOC1 82450,Cc1cc(Cl)cc(C(=O)NCC(C)N(C)C(c2ccc(F)c(Cl)c2)=O)c1N 82451,C1(=CC(N2CC(O)(CN(C(=O)CCCn3cncn3)C)C2)=O)CCCCCC1(F)F 82452,C1(NC(C=CCN(CC)CC)=O)CC2CN(C(=O)CS(N)(=O)=O)CCN2C1=O 82453,c1(C(=O)OC(c2ccc(Br)s2)C)ccc(C2CCCC2)c(F)c1 82454,c1(CC(N2CC(C3N(c4ncc(C)c(C)n4)CCC3)C2)=O)ccn2cncc2c1 82455,N1(CC(C)NC(C2CCCN2C(=O)Cn2nccn2)=O)CCCC1=O 82456,N1(C(C(c2c(C)cccc2Br)NC(C(COCC)C)=O)=O)CCCCCC1CC 82457,C1(c2onc(-c3cc(C)nn3C3CC3)n2)C2CN(C(=O)C(=O)CC)CC12 82458,C12(CNC(C(C)SC)=O)CN(C(=O)Cn3ncn4cccc4c3=O)CC1CCO2 82459,c1(C(N2CC3(CC(NC(=O)Cc4c[nH]nc4O)C3)C2)=O)cnn2c1OCC(O)C2 82460,Cc1cccn2cc(C(=O)NC3CC3NC(=O)CC(C)(C(F)F)N(C)C)cc12 82461,O=C1CC2(CCN(c3ccncc3S(=O)(=O)NC3CN4CCC3CC4)C2)C(=O)N1 82462,C1(CNC(C2(OC)CCSC2)=O)CCC(CN(C)C(c2ccoc2)=O)CC1 82463,N1(C(=O)C=CCN2CCOCC2)CC2(CNC(=O)CC3CC34CC4)CC1CO2 82464,C1(N(C(Cc2cccc(OCC)n2)=O)C)CCN(C(=O)C(C)(C)CC)CC12CC2 82465,C1(C(=O)NC(C2(C)CC2)CO)COC2(C1)CN(C(=O)C=C1CCC1)C2 82466,C(C(C)(O)C(F)(F)F)NC(C1(F)CCN(C(COCCCOC)=O)C1)=O 82467,CC1COCCC1N=c1[nH]c2c(c(=NCCCN3CCCCCC3=O)[nH]1)COC2 82468,C(=O)(C(C)(C)CNC1CCS1)N1C(CNC(C(C)NC(=O)C(C)(C)C)=O)CCC1 82469,C12(NC(Cc3c(C)n[nH]c3)=O)CN(C(=O)C(C)(C)CN(C)C)CC1CS(=O)(=O)C2 82470,C1(CN(C(c2ccc(C)n2C)=O)C)CN(C(C2CCCCC2O)=O)CC12CC2 82471,c1(OC)cc(C(=O)N(CCC(=O)O)C(C)(C)C)cc([N+](=O)[O-])c1O.C(CS)N 82472,c1(C(N(CCN(C(C)C)C(c2cnn(C3CCOC3)n2)=O)C)=O)cnnn1C 82473,C=CCC(CC(=O)N(CC(C)C(C)(C)C)C)NC(c1cnccc1OC)=O 82474,Cc1[nH]nc2ccc(C(=O)NCC(C)CN(C(=O)C(C)(C)CO)C)cc12 82475,C1(C(CC2(N(C)C)CCCC2)=O)CN(CC)CCS1(=O)=O.c1(CC=O)cccs1 82476,c1(CN(C(C(c2ccccc2)C)=O)C)cnn2c1CN(C(=O)CCS(C)=O)CC2 82477,C1(NC(c2cscn2)=O)CN(C(=O)COc2cccc(SC(F)F)c2)CC1O 82478,CC(=Cn1ccnn1)C(=O)N1CCCC(NC(c2coc3c2CSC3)=O)C1C 82479,c1(C(=O)NC2C(NC(c3c(C)nncc3)=O)COC2)cc2ccccc2[nH]1 82480,N1(CC)CCCC(NC(=O)CC2CCN2C(C2CCCN2C(=O)OC)=O)C1 82481,C(C1CN(C(=O)CC(O)CN(C)C)CC1C(N1CCOC(C#N)C1)=O)=CC 82482,C1(C(=O)OCC)CC2C(CC1C(=O)NC1(C(C)(C)O)CCOC1)C2(F)F 82483,CCCC(O)CC(=O)N(C)CC1(O)CCN(C(=O)CC2CSCCO2)CC1 82484,C1(C(N2C(CN(C(c3n(CC)ncc3C)=O)C)CCCC2)=O)COCCN1C=O 82485,c1(C(=O)NCC2OCCN(C(C3(C#C)CCC3)=O)C2)cc(O)ncc1Br 82486,N1(C(C2N(CC#C)CCC2)=O)CC(NC(c2cc(N)cnc2C)=O)C(C)(C)C1 82487,c1(C(=O)NC(CCCNC(CC(CC)CC)=O)(C)C)ccn2ncccc12 82488,C1(CNC(=O)C(O)C2CCC2)CCCN1c1nccs1 82489,N1(C(COCC(=O)NC)=O)CC(C2CCCN(C(C3(C)CCC(=O)NC3)=O)C2)C1 82490,C1(CC)CN(C(=O)CCC=C(C)C)CC1NC(c1cn(C(C)C)nc1C)=O 82491,C1(N(C(C(c2scc(C)n2)C)=O)C)CCCCC1N(C)C(c1ccc(O)cn1)=O 82492,C(=O)(C1Cc2ccccc21)NC1C=CCN(C(CC2CCN(C)CC2)=O)C1 82493,Cc1nc(NCc2cncc(Br)c2)cc(=NCC(C)N2CCCCC2)[nH]1 82494,C(=O)(C1=CC2(CCOC2)C1)NCc1occ(C(N2C(C(C)(C)O)CCC2)=O)n1 82495,C1(NC(CCCC=C)=O)CN(C(=O)CCCc2ccc(F)cc2)CC1C=C 82496,C1(NC(CC(C)O)=O)CCC(C(=O)Nc2cccc(CS(N)(=O)=O)c2)OC1 82497,c1(OC(COC)C)cc([N+](=O)[O-])ccc1SCC(=O)NCc1ccccc1 82498,C1(CNC(C2CCOC2c2ccc(F)cc2)=O)CCC(C(F)F)CC1 82499,C(=O)(CCC(=O)N1CCCCC1CNC(=O)CC1CCCO1)N(CC)CC 82500,c1(C(=O)NC2C(NC(C3C(CCOC)C3)=O)CC2)cc([N+](=O)[O-])c(C)s1 82501,N1(C(C(C)N(C(=O)C(F)=CC2CC2)C2CC2)=O)CCCC(C2CC2)CC1 82502,C1(NC(c2cn(C(C)(C)C)nc2)=O)CCC(O)CN(C(C2CCCN2C=O)=O)C1 82503,Cc1cc(Br)c(S(N)(=O)=O)cc1C(N1CCC(CO)C(C2CC2)C1)=O 82504,c1(C(N2CCC3CC23C)C(=O)NC(CC)(C)C)ccc(F)cn1 82505,C1(C(=O)NOCCN2CCCC2=O)(NC(C=CC(=O)N(C)C)=O)CC(F)C1 82506,C(C(C)(C)C(=O)NC(C)CCNC(=O)CN1C(=O)CNC1=O)SC 82507,C1(OC)CN(C(c2ccn(C)c2C)=O)CC1NC(C1CC2CC1C2)=O 82508,c1(C(N2CCC(C(F)C(N)=O)CC2)C(=O)NCCOC)cccc(CO)n1 82509,c1(C(N(CCNC(C(CC(C)C)NC(C)=O)=O)C2CC2)=O)ccn(C)c(=O)c1O 82510,Cn1c(C(=O)NCCC2CN(C(C3CCCCC3C(F)(F)F)=O)C2)cccc1=O 82511,C1(CC(=O)NCC(N(C(CCOCC)=O)C)C2CC2)CCCN1C(C)C 82512,c1(CC(=O)NC2CN(C(c3c(C)nc(C4CC4)o3)=O)C(C)C2)nc([N+](=O)[O-])n[nH]1 82513,C(c1cncs1)=CC(=O)N(CCC(=O)NCC(C)(C)OCC)C1CC1 82514,CC1CN(C(=O)CC2CC2)CC1NC(C1(c2cccs2)CC1)=O 82515,N1(C(c2c(Br)cn(C)n2)=O)CCOC2(CCN(C(C3CC4(CC4)C3)=O)CC2)C1 82516,C(=O)(C#CC1(C)CC1)NC1CCN(C(C(CC)COC)=O)C1 82517,c1(CC(N2CC(F)CC(NC(=O)C3=CCSC3)C2)=O)cncc2ccccc12 82518,Cc1cc(CC(=O)N(CCCCN(C(=O)CCOC2CCC2)C)C)cc(C)c1 82519,C1(NC(=O)NCC2CCCCO2)CCCN(c2ncccn2)C1 82520,C1(C)(NC(C=C)COC)CCCC1CNC(=O)OC(C)(C)C 82521,CC1CN(C(=O)CCCC2CC2)CC1NC(=O)CC1CC(=O)NC1=O 82522,n1(CC(N2CC(NC(C(COC)(C)OC)=O)C(O)C2)=O)cc(P(C)(C)=O)cn1 82523,C(C(C)(C)C1=CCCC1)NC(CONC(c1ccc(COC2CCN(C)C2)o1)=O)=O 82524,C(=O)(CP(=O)(C(C)C)C(C)C)N1C2C(NC(c3c(C)cnn3C)=O)CC(C2)C1 82525,Cc1cc(C(=O)NC(C)CCNC(=O)CC2CCC(C)(C)CO2)n2nccc2n1 82526,C12(NC(c3nc(C)sc3)=O)CC1CN(C(c1cccnc1SC(C)C)=O)C2 82527,n1(C(C)C)ncc2c(N3CCC(NC(c4csc(S)n4)=O)C3(C)C)nc(Cl)nc12 82528,c1(SC)cc(C(=O)NC2COCC2NC(c2cc(C(C)C)oc2C)=O)c(C)o1 82529,N1(C(C(c2ccccc2)NC(CCCCC=CC)=O)=O)CCOC(C)(C)CC1 82530,N1(C(C(C)Cc2ccc(Cl)cc2)=O)CC(NC(C23CC4CC2C3C4)=O)CC(C)C1 82531,CC(CC(N)=O)N=c1[nH]c(N2CCOCC2)nc(=NCc2cc(Cl)c(F)cc2F)[nH]1 82532,N1(C(CC(=O)NC)=O)CCOC2(CCN(C(=O)CCc3cccnc3Cl)CC2)C1 82533,N1(Cc2c(C)ccnc2)CCC(NC(c2cccnc2C(F)F)=O)CC(C)(C)C1 82534,N1(C(C(C)=C2CCCC2)=O)CCCC(O)(CNC(=O)C=Cc2cn(C)cn2)C1 82535,C1(CNC(C(C)(C)C2CC2)=O)CCC12CN(C(=O)C1=COCC1)C2 82536,N1(C(C=C(C)C(C)C)=O)CCC2CN(C(=O)CCN3CCCC3)CCC12 82537,N1(C(c2cn(C)nc2)=O)CCN(C(C2CC23CCCCCC3)=O)C2(CC2)C1 82538,n1(CC)ncc(Br)c1C(=O)NCC1CC1CNC(=O)C(C)N1CC(C)C1 82539,N1(C(C2C(C)C2)=O)CCOC2(CCN(C(C3CCC4(CC3)CC4(F)F)=O)CC2)C1 82540,c1(CC(=O)NC2(c3cn(CCCCCCO)nn3)CCC2)cccc(C(F)F)c1 82541,Cc1ccc(C(N2CCN(C(=O)CC3CCCN3C)CC2)=O)cc1Br 82542,n1(C(C)CC(=O)N(C)CCOCCN(C2CCCCO2)C)cnc2ccccc12 82543,c1(C(=O)NC2CC(F)(CNC(C3CC(OC)(OC)C3)=O)C2)nc[nH]c2nccc1-2 82544,C1(O)(CC(=O)NCC(COC)(C)SC)CCN(C(c2ccc(OC)nc2)=O)CC1 82545,N1(C(c2n(CC)ncn2)=O)CCCOC(CNC(C2(OC)CCS(=O)(=O)C2)=O)C1 82546,C(C(C)(O)CC(=O)N(CC(=O)NCC#CC(F)(F)F)C(C)C)OC 82547,N1(C(c2c(C)nn[nH]2)=O)CC2C=CC1C(C(=O)NC(c1ncc(F)cn1)C)C2 82548,CC(O)C(=O)NC1CC(N(C(=O)COc2ccsn2)C)C1 82549,C(=O)(C(O)CC[S+](C)C)N(c1ccccc1)C(C)CN(C(=O)C=CC(=O)N(C)C)C 82550,C(=O)(C(C)(C)C)N(C1CN(C(=O)C(C)OCCOC)C1)CC 82551,C(=O)(C(Cc1ccco1)C(=O)NC1CC(NC(=O)Cc2cc(C)n(C)n2)C1)OC 82552,N1(C(C(C)=CC2CC2)=O)CCC(C)(C)C(NC(=O)CCC2CCCN2C)C1 82553,CC(Cc1ccccc1)C(C1CCCCC1)OC(c1cnn(-c2nccs2)c1)=O 82554,c1(NCCC(C(C)C)OCC)ncccc1S(=O)(=O)N(C)CCSC 82555,C1(NC(c2n(CCC)ncc2)=O)CCC2CN(c3ncc(C)c(C)n3)CCC2C1 82556,c1(OC)cn(CC(=O)NC2CC2NC(=O)CCCC(N)=O)c(C)cc1=O 82557,C1(OC)CC(C(=O)N(C)Cc2cnc(C)s2)N(C(=O)CCn2ccnn2)C1 82558,C(=O)(C1=CCC(F)(F)CC1)NCC(C(C)C)NC(c1cccc(O)n1)=O 82559,N1(C(C(Cc2c(C)cccc2)C)=O)CC2CCN(C(C3CCC3)=O)C2C1 82560,N1(C(=O)C(C2CC(F)(F)C2)O)CCOCC(CNC(C2(CO)CC2)=O)C1 82561,N1(C(C(CC(CC)C)C)=O)CC2CCCC(NC(=O)CSc3nccs3)C2C1 82562,N(S(=O)(=O)N1CCCC1C)(C1CCCCC1)Oc1c(CC)cccc1 82563,c1(C(=O)NCC(CC)NC(c2cnc(O)nc2O)=O)ncc(Cl)cc1Cl 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82758,c1(C(=O)NCC2C(NC(C3(C)CC3(F)F)=O)CC2)cnc(Cl)c(N)c1 82759,N1(C(Cc2scc(C)n2)=O)CCOCC1c1cccs1 82760,Cc1nn(C)c2c(NCC3COCC3O)nc(=NCCCC3CCCCC3)[nH]c12 82761,CC1CN(c2cc(CNC3CCNCC3C)ccn2)CCO1 82762,c1(C(=O)NCC(CNC(CCOCC#C)=O)(C)O)cc(C)n(CCO)n1 82763,C12(NC(C3C(=C)CC3)=O)CCC(C1)N(C(c1ccnc(-c3ccco3)c1)=O)C2 82764,N1(C(C2N(C(C3CNC(=O)O3)=O)CCC2O)=O)CCC2(CC1)N=N2 82765,Cc1nc(CC(=O)NC(C(=O)NCC2CCCSC2)c2cccs2)n[nH]1 82766,N1(CCSC)CCN(CC2CCCN(C(C)C(C)(C)C)C2)CC1 82767,C1(N(C(C2N(C(C)=O)CCC2)=O)C)CN(C(c2cnccn2)=O)CCC1C 82768,c1(CC)cc([N+](=O)[O-])ccc1C(N1CCCC1CNC(=O)C(C)OCC(C)C)=O 82769,CCCC(C)(C)CC(=O)N1CC2CC(NC(=O)CCC3CCOCC3)CC1C2 82770,C1(NC(c2ccnnc2O)=O)C=CCN(C(c2ccc(CF)cc2)=O)C1 82771,C1(C#N)(C(=O)NC2CCCN(C(CN(CCC#C)C)=O)C2)CCOCC1 82772,C(=O)(CCCCCCCCCO)N(C1CN(C(C2CC3CC2CC3(F)F)=O)C1)C 82773,N1(C(C(C)SC)=O)CCCCC1C(=O)NCC1CC1(C)C 82774,C#Cc1ccc(C(=O)NC2(C)CCCC2NC(C2C3COCC23)=O)nc1 82775,S(=O)(=O)(c1cccnc1)N(CC(N1CCOC(CNC(=O)C(C)(C)C)C1)=O)C 82776,CN1CC(NC(C2CN(C(=O)Cc3cccc(O)n3)CCS2)=O)CC1CO 82777,C1(NC(C(C2CCC(C)CC2)CC)=O)CCCN(C(=O)CN2CCCCC2)CC1 82778,N1(C(CN(C)CC)=O)C2CCC1CN(C(=O)C(C)Cc1cnc[nH]1)C2 82779,CC1=NNC(=O)C1CC(=O)NC(CO)C(C)NC(=O)CCCn1c(C)csc1=O 82780,C12(C(CNC(=O)CC3CCCC3C)NC(CC=C(C)C)=O)CCC(CC1)C2 82781,C1(=CC(=O)NC2CCCC(NC(=O)Cc3ccoc3)C2)CN2CCC1CC2 82782,C(CC(=O)Nc1cc(O)cc(F)c1)(C(F)F)NC(c1n(CC)nc(C)c1)=O 82783,C1(NC(c2ccc(OCC)cc2)=O)CCC12CCN(C(c1scnc1Cl)=O)CC2 82784,C=CC(C)(CC)C(=O)N1CCCC(CNC(c2ccnc(CC)c2)=O)CC1 82785,c1(CNC(=O)CC(O)C2CC2)ccc(-c2cn(-c3ncc(Br)s3)nn2)cc1 82786,C(=O)(C1CCCc2ccccc21)NCC(=C)CCNC(=O)CC1CCC(=O)NC1 82787,c1(C(C)NC(CCn2cc(COC)nn2)=O)cccc(C(C)(C)C)c1 82788,C(=O)(CC(C(F)F)NC(c1cccc(=O)o1)=O)N(CCn1ncc(C)c1)C 82789,C1(NC(C(C)(c2ccccc2)OC)=O)CCN(C(=O)CCOC(C)=O)CC1C 82790,C12(CNC(C3(CC#C)CCOC3)=O)CC(CO1)N(C(c1cc3n(n1)CCC3)=O)C2 82791,C=C1CC(C(N2CC(N3CCCC3)C2)=O)(CNC(=O)CC2(C)CC2)C1 82792,C1(CC(=O)NC2CCC(NC(c3cc(CO)ccn3)=O)CC2)C=CS(=O)(=O)C1 82793,c1(OC)ccc(C(=O)NC2CC(F)(CNC(C3(C4CC4)CC3)=O)C2)s1 82794,C1(C)(C(N2C(C=C)CC2)=O)CCN(C(C2CCCCC2C(=O)OC)=O)CC1 82795,O(N=C1CCCCCC1)CC(=O)NCC(CNC(C(C)OCCC=C)=O)F 82796,N1(C(C2(CC)CC2(F)F)=O)CCN(C(c2cc(-c3ccccn3)no2)=O)CC1 82797,N1(C(C(c2ccc(OC)c(F)c2)C)=O)CCN(C(=O)CCc2cn[nH]c2)C(C)C1C 82798,C(=O)(CCCS(C)(=O)=O)NC(C1CCCN(C(c2cccc(C)c2N)=O)C1)C 82799,CC(C)S(=O)(=O)CC(=O)NC1(CNC(=O)C(=O)Nc2ncc[nH]2)CCCCC1C 82800,N1(C(C2(COC)CCOC2)=O)CCCC(CCNC(c2cc(OC)cs2)=O)CC1 82801,Cc1onc(CO)c1C(=O)N(CC(C)NC(c1ccc(C(C)(C)C)nc1)=O)C 82802,C1(CCOC)CN(C(c2csc(-c3ccncc3)n2)=O)CCN1C(=O)C(N)=O 82803,N1(C(C2C(OC)(OC)CC2)=O)CCC(F)(CNC(c2cnn(C(F)F)c2)=O)C1 82804,c1(C(=O)NCCCCCNC(c2ccc[n+]([O-])c2)=O)ncc(F)cc1F 82805,Cc1nccc(C(N2CCCCC2CCC(=O)N(C2(C)CC2)C)=O)n1 82806,C(C)(C(=O)NC1CC(F)(CNC(C2(N(C)C)CCCOC2)=O)C1)(C(C)C)OC 82807,C1(C(=O)NC2C(C)CN(c3nnc(C#N)s3)CC2)CN2CCN1C(C)C2 82808,C1(CNC(c2c(CCC)n[nH]c2)=O)CC2CCC1N2C(=O)CC1(O)CCCCC1 82809,c1(C(=O)NCCNC(C(COC(C)(C)C)N(C)C)=O)cc(Br)ccc1O 82810,C(c1cn(C)cn1)=CC(=O)NC(CCOC)CNC(=O)CSCCC(F)(F)F 82811,c1(CC(=O)NCC(CNC(CC2C(C)C2(F)F)=O)(C)C)cc(Cl)sc1Cl 82812,C1(COC(CCC(=C)C)=O)CCCN(C(c2cc(NC(C)=O)cnc2C)=O)CC1 82813,N1(C(CNS(N(C)C)(=O)=O)=O)CCN(C(=O)C2=CCCS2)CC(CO)C1 82814,S(=O)(=O)(c1cc(C(F)(F)F)ccc1NCCc1cc2ccccc2o1)NC(C)C 82815,c1(CNC(CCC2(C)CCN(C(C3C(C)(C)C3)=O)C2)=O)ccnc(C#N)c1 82816,C(CCC(C)CO)NC(CC1(OCC)CCC1)=O 82817,C=C1CC(C(=O)Nc2cc(C(=O)OC)no2)N(C(=O)Cc2ccc(Br)cc2)C1 82818,Cc1nnc2n1CC(C(N1CCOCC(NC(=O)Cc3ccoc3)C1)=O)CC2 82819,Cc1cc(NC(=O)CCF)ccc1NC(c1cnn(C2CC2)c1C1CC1)=O 82820,C(=O)(C1COc2ccc(Cl)cc21)N1CC(NC(C(C)(C)C2CC2)=O)C(C(F)F)C1 82821,C1(CC(=O)N(CC(c2nn[nH]n2)C)C2CC2)CCCN1C(=O)CCc1ccoc1 82822,n1(CC)nccc1C=CC(=O)NCC(C1CC1)N(C)C(c1snnc1C)=O 82823,c1(C(N(CC(C2CC(F)(F)C2)O)C)=O)ccc(N)c(Cl)c1 82824,c1(C(=O)NC2CC2C(=O)Nc2ncc(F)cc2Br)cc(Cl)c(Cl)cc1F 82825,C(=O)(CC(F)(F)C(F)F)N1C(CNC(=O)C(c2ccc(Cl)nc2)C2CC2)CCC1 82826,N1(C(c2ccc(OCC)cc2)=O)CCN(C(=O)C=C2CCC2)C(CSC)C1 82827,Cc1nc(-c2cccs2)sc1C(N1CCCC1C(C)(C)NC(=O)COCCF)=O 82828,CC(C)C(O)C(=O)N1CC(C(F)Cn2cc(Cn3cccc3)nn2)C1 82829,c1(CCCC(N2CC3C(C(N4CCC(C)CC4)=O)(C3)C2)=O)cc(F)ccc1F 82830,c1(C(N2C(CN(C(C3(CC(C)C)CC3)=O)C)COCC2)=O)nccc2cc[nH]c12 82831,c1(C(N(C)CC2C(C)OCC2)=O)c(CNC(C2SCCS2)=O)nnn1C 82832,C1(CCOCC)CN(C2=CC(=O)N(c3ccc(Cl)cc3)C2=S)CCN1CCCO 82833,C1(C(=O)NC(C2CCCCC2)CNC(=O)C2=CCCC2)CCC(F)(F)CC1 82834,c1(CC)ccc(CNC(=O)CCC(C)NC(C2CCOC2C(C)C)=O)cc1 82835,CC1(C(N2CC(F)CC2CNC(=O)COc2ccc(F)nc2)=O)CCCCC1 82836,CC1CC=C(C(=O)NCc2cc(C(=O)NCC(C)C(C)(F)F)n[nH]2)CC1 82837,c1(CC)ccc(F)cc1C(=O)NC(C(C)NC(=O)CN1CCS(=O)CC1)C(C)C 82838,C1(NC(CCC(=O)OCC)=O)CCCC12CCN(C(C1CCC1(C)C)=O)CC2 82839,Nc1cc([N+](=O)[O-])ccc1C(N1CCCCC(NC(c2c[nH]c(Br)c2)=O)C1)=O 82840,N1(C(c2nn(CC)c(C3CC3)c2)=O)CC(CO)C2(C1)CN(C(=O)C(O)C(F)(F)F)C2 82841,c1(N2CCSCC(C)C2)nc2ccsc2c(=NCC2(C)CS(=O)(=O)C2)[nH]1 82842,C1(CC)CN(C(c2ccnc(F)c2F)=O)CCN1C(=O)Cc1ccccc1OC 82843,c1(N2CC(C)C(NC(=O)CC3CC(F)C3)CC2)ccc(Br)cc1[N+](=O)[O-] 82844,N1(C(c2ccncc2N(C)C(C)C)C(=O)NC)CC2CC(OC)C(C2)C1 82845,N1(C(c2nn(C)c(=O)cc2)=O)C2CCC1CN(C(c1ncc(Cl)c(N)c1Cl)=O)C2 82846,N1(C(c2nc(OCC)oc2)=O)CCCC(CN(C(c2nc(Cl)cs2)=O)CC)C1 82847,c1(CC(=O)NCC(C2CCOC2)NC(CC2(OC)CCCC2)=O)ccncc1F 82848,CC1CN(C(c2ccc(Cl)cc2)C(=O)NCC2CCCCC2)CCO1 82849,c1(CN(C(C(=O)NC(CC)C(=O)NC)=O)C)ccc(C(N)=O)cc1F 82850,C1(NC(Cc2n(C)nnc2)=O)C2CC(O)C1N(C(c1ccc(C(F)(F)F)s1)=O)C2 82851,Cc1cc(=NCC2CCCC(C)CC2)[nH]c(=NCCc2cccc(N)c2)[nH]1 82852,CCCC(CC)CCC(=O)NC1CCC(NC(c2sccc2OC)=O)CC1 82853,N1(C(C(C)OCC2CC2)=O)CCC(NC(=O)CCC2CCOCC2)C(CO)C1 82854,CC1(C)CC(CNC(C2CC23CC(F)(F)C3)=O)CN1C(=O)CCP(C)(C)=O 82855,c1(C(=O)NCC2(C(N)=O)CN(C(=O)CCC(N)=O)C2)cnc(O)c2cccnc12 82856,Cc1cc(C)c(C(=O)NC(C)(C)C(C)NC(=O)CN(c2ccncc2)C)c(C)c1 82857,C1(CC(=O)NCc2[nH]nnc2C)(OC)CN(C(=O)C(c2cnn(C)c2)=O)C1 82858,CC1CCCC(CCNC(C2CCOCC2NC(=O)CC2(C#N)CC2)=O)C1 82859,c1(C(=O)NC(C(=O)N(CCNC(c2c(C)occ2)=O)C2CC2)C)cccc(Cl)c1 82860,C1(C(=O)NCc2cncc(C)c2)CCN(C(=O)COCCN(C)C)CC1(C)C 82861,C1(C(=O)N(C(C)C(C)C)C)(OC)CCN(c2cc(O)nc(=N)[nH]2)CC1 82862,C(=O)(C(C(C)=Cc1ccccc1)N1CC(OC)C(F)C1)NCCOCC 82863,CCC(CC(=O)NC(C)CCN(C)C(c1ncoc1-c1cnn(C)c1)=O)C(C)C 82864,c1(CC)ccccc1C(=O)NCC1C2CC2CN1C(C1C2CC3C(C2)C13)=O 82865,c1(NC(c2cnc(OC)s2)c2nnnn2C)ccc(CCC(C)C)cc1 82866,N(C(=NCCN(CC(F)(F)F)C(C)C)NCCN1CCCC1)C1CCC(C)CC1 82867,C1(CNC(CCN(C(=O)CCOC2COC2)C)=O)(CO)CCCO1 82868,C1(CNC(C2(CC=C)CCC2)=O)CCCC1C(=O)Nc1c[nH]nc1OC 82869,C1(C)(NC(C2CN(CC)C(=O)C2)=O)CCN(C(C2CC(CC(C)(C)C)C2)=O)CC1 82870,N1(C2CCN(CC)C2=O)CC(NC(c2ccn(-c3ccncc3)n2)=O)C(C)(C)C1 82871,c1(C(=O)NCC2C=CC(NC(c3cc(CCC)on3)=O)C2)ccc(C(N)=O)cn1 82872,C12(C(=O)NC3C(NC(=O)Cn4cnc(Br)n4)C3)CC(C1)C(C(F)(F)F)O2 82873,C=CC(O)C(=O)N(CCNC(=O)CN1CCC(C)C1)CC 82874,c1(N2CCN(CC)C(C)(C)C2)nc(N(CC(F)(F)Br)C)c2ncn(CC)c2n1 82875,c1(C(=O)NCC2(C)CCCN2C(c2ncccc2Br)=O)n[nH]c2c1COC2 82876,C1(NC(c2ccc(F)cc2Cl)=O)COCC1C1CC1 82877,C1(NC(c2c(CC)nco2)=O)CCC2CCN(C(C3(C)CC(C)C3)=O)C1C2 82878,c1(CC)nccc(=NCCNC(=O)CC2COCCN2C(=O)OC(C)(C)C)[nH]1 82879,c1(C(C)CC(=O)NCCC2CN(C(C3(O)CCSCC3)=O)C2)c(F)cccc1F 82880,C(=O)(C1=Cc2ccccc2C1)N1CCC(C(C)NC(C2C3CC3C3CC23)=O)CC1 82881,N1(C(C(C2CCC2)OCC)=O)CC2(CCCCN2C(c2ccnc(S)c2)=O)C1 82882,CC(C)(C)CC(F)C(=O)N1CCC(NC(c2cc3cnccc3[nH]2)=O)C(F)C1 82883,CCCC(C(=O)N1CCC(C)N(C(c2cc(C)c(F)cc2F)=O)CC1)S(N)(=O)=O 82884,N1(C(C)=O)CCN(CCN(C(=O)C(F)OC(F)(F)F)C)CC1.c12ccc(cc1)[nH]2 82885,Cc1coc(C)c1CNC(=O)C(=O)NCC1CCCC1CC(C)C 82886,Cc1cc(=NC(=O)NC(CO)C(O)c2cccnc2)[nH]n1C(C)C 82887,Nc1sc2ccccc2c1C(N1C2CCCC1CN(C(=O)COCCCF)C2)=O 82888,CCC(CC(C)C)C(=O)NC1CC(F)(CNC(c2cc3ccccc3o2)=O)C1 82889,CCC(CC)(C(=O)N1CCC(NC(=O)CCC(C)(C)F)C(C)C1)OC 82890,c1(OC)cc(C)cnc1C(=O)N(C)CC1C2CN(C(C3CC3C)=O)CC12 82891,c1(C(=O)NCCN(C(c2ncoc2C(C)C)=O)CC)cnc(CC(C)C)cn1 82892,CCCC(O)(CCC)CC(=O)N1CCCC(CNC(=O)C(COC)COC)CC1 82893,C1(C(N(C(C(=O)NC2CN(CC)C(=O)C2)C2CC2)C)=O)CN(C)CCN1C 82894,CC1CN(C(=O)C2=CCC(NC(=O)CCC(F)(F)F)C2)C(C)C1C 82895,Cc1cccc(C)c1C(c1nnnn1CC(F)F)NCC1(C)CC=CC1 82896,Cc1nc(-c2ncccn2)ncc1C(N1CC(O)(CCNC(=O)CCF)C1)=O 82897,c1(OC)ccc2[nH]nc(C(=O)NCC(C)NC(C3(c4cc[nH]n4)CC3)=O)c2c1.CN 82898,C(=O)(C(F)C(=O)NCC(CC)NC(=O)CCCc1cc(C)no1)OCC 82899,CCC(C(=O)NC1CC(C)(C(=O)NCc2cccs2)C1)OC 82900,C(CCCC1CC1)(c1nnnn1CCOC)NC1(CCOC)CC1 82901,CCS(=O)(=O)C=CC(=O)NCC1CC2CCC(C1)N2C(=O)CCC=C(C)C 82902,C12(C(N3CC(CCNC(Cc4c(C)n[nH]c4)=O)C(C)C3)=O)CCC(CC1)CC2 82903,c1(CNC(=O)Nc2cn(C(C(=O)OC)(C)C)nc2)ccc(C)n1C 82904,C1(CN(C(c2[nH]cc(C(=O)OC)c2)=O)C)CCCCN1C(C1CC1C)=O 82905,C1(NC(=O)C=Cc2cnccn2)CS(=O)(=O)CC1NC(c1cc(Cl)ccn1)=O 82906,C1(CCNC(CN2C(C)CC2)=O)CSCCN1C(=O)CSCC(N)=O 82907,C1(C(=O)NCC2C(C(N3CCC(C(C)C#N)CC3)=O)C2)CC12CCOCC2 82908,Cn1cnc2nc(=NCc3nncs3)[nH]c(NCC3C4CCCCCC34)c12 82909,C=C(Cl)C(C)(C)C(=O)N1CC(NC(=O)CCc2cccc(OC)c2)C2(CC2)C1 82910,CC(C)CC(C(=O)N1CCCC(C)(NC(c2cn3ccnc3cn2)=O)C1)C(C)C 82911,C12(C(=O)Nc3cccc(Cn4ccnc4)c3)CCCC1C2(F)F 82912,C(=O)(N=c1[nH]onc1C1CC1)Nc1ccc(C(N(C(C)CO)CCC)=O)cc1 82913,C(CCCCCNC(c1ccc[n+]([O-])c1)=O)NC(c1ccsc1)=O 82914,C1(CNC(C2C(CC)CCC2)=O)CC(OC)CN1c1cc(C(=O)NC)ncn1 82915,C1(N(C(C(C)N=[N+]=[N-])=O)C)CCCN(C(=O)C(c2cncnc2)C)CC1 82916,C12(NC(c3c(Cl)ccc(C#C)c3)=O)COCCC1CN(C(=O)CC(C)(C)C)C2 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82987,C(=O)(C(F)(F)C(O)CC)N(CC(CC)NC(=O)Cc1sc(C)nc1C)C 82988,C12(CNC(Cc3c(OC)cccc3Cl)=O)CCCC1CN(C(c1nc[nH]n1)=O)C2 82989,N1(C(C=CCN(CC)CC)=O)CC2CC(C1)CN(C(C1CCCCN1C)=O)C2 82990,Cc1cc(N)c(C(=O)NC(CO)C(C)NC(C2C3CC4C(C3)C24)=O)c(F)c1 82991,C(=O)(C1CCCc2cncn21)NC(C(C)C)CCNC(c1c(O)cccc1Cl)=O 82992,c1(C(=O)NCC(C)N(C(=O)C(C)SC(C)(C)C)CC)sc(CNC(C)=O)cc1C 82993,c1(C(=O)NCC(CC=C)NC(C2CS(=O)(=O)C2)=O)cnc2c(F)cc(C)cc2c1 82994,CCCC(C(=O)N1CC(N2CC(F)C2)C1)NC(=O)C(C)c1cccs1 82995,C1(CNC(CCOCCCNC(C2C(C(N)=O)CCC2)=O)=O)NC(=O)NC1=O 82996,C(=O)(CS(=O)CC)NC1(CC=C)CN(C(=O)CCCNS(C)(=O)=O)C1 82997,C#Cc1cc(C(=O)NCC(C)CNC(c2ccc(Cl)nc2O)=O)ccc1C 82998,CC(=O)CCCC(C)C(=O)N1CCSCC1C(N1CC(C)(C)C1)=O 82999,C1(C(=O)NC(C(C)NC(CNS(CCCOC)(=O)=O)=O)CO)CC12CC(F)(F)C2 83000,C1(N(C(=O)CC2CCCOC2)C)CCCN(C(=O)C(O)C2CCCC2)CC1 83001,c1(NN(C(=O)C=CC2CCCCC2)CC2CCN2CC(=O)C(C)=O)cccc(N)c1 83002,Cc1cc(C#N)ccc1C(=O)NC1CC2(C1)CC2C(=O)NC12CCC(C1)OC2C 83003,C1(C(N2CC(C(=O)OCC)C2)=O)COC2(C1)CN(C(=O)C(C)(C)NC(C)=O)C2 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83092,C1(C#N)(CN2CC(NS(NC)(=O)=O)C(c3nc(C4CC4)no3)C2)C(C#N)C1(C)C 83093,CCC(C)C(C(=O)NCC(C)(C)CNC(=O)Cc1ccccc1Cl)NC(=O)OC 83094,N(C1CCc2c(Br)ccc(Cl)c21)C(C1C2(C(=O)O)CC(C)(C2)O1)=O 83095,C1(C(=O)NC2(CC=C)CCN(C(=O)Cc3cnns3)C2)CCC=CCCC1 83096,C1(C(N(CC(NOCC(C)C)=O)C(C)C)=O)CC2(CCC2=O)C1 83097,c1(C(=O)NCC2(C(C)NC(C)=O)CC2)ccc(C#N)c(F)c1Br 83098,C1(NC(c2c(NC)snc2C)=O)CCC2CCN(C(c3cc(C(N)=O)c[nH]3)=O)C12 83099,C1(C(N2C(C(=O)NCC3CN(CC(C)C)C3)CC(F)C2)=O)NC(=O)OC1(C)C 83100,c1(C(=O)NC2C(C)CN(C(=O)C(C)(C)C3CCOC3)C2)cn2ccsc2n1 83101,C1(C(N2C(C)CC(CNC(c3c(CC)csc3)=O)C2)=O)CC2CCC(C1)C2=O 83102,N1(C(CNC(CNC(c2n(C)ccc2)=O)=O)=O)CC2(CCC2)CC1CO 83103,O=C(N=S1(=O)NC(=O)c2ccccc21)C1COCCC1C 83104,C1(NC(c2cccc(O)n2)=O)COCCC1C(=O)NN1CC(CC2CC2)C1 83105,C=CC1CN(c2cc(C)nc(N3CCCC(CCO)CC3)n2)CCO1 83106,N1(C(CC)=O)CC2CCN(Cc3cn(-c4coc5ccccc45)nn3)C2C1 83107,C(=O)(C1=C(c2cnn(C)c2)N(C)C(=S)NC1c1cnc(-c2ccccn2)s1)OCC 83108,N1(C(C(C)N)=O)CC(C)(C)C1C1CC1.N(C)CC 83109,CC(CC(=O)NCCN(C(=O)Cc1nnc(O)s1)C)P(C)(C)=O 83110,c1(CC(=O)NCC23CC(NC(=O)C(F)CC4CCCC4)(C2)C3)c(F)cccc1F 83111,CCCCCCCCCC(=O)NCCN(CCC)C(c1cc(C)cc(C)c1N)=O 83112,C(=O)(C(O)CCCC)N(CC(=O)NCC1CC(CC)C1)C(C)C 83113,C1(C(=O)NCCCSc2ccccc2)CCCN(CCC2CCCCO2)C1 83114,N1(C(CCc2c(C)cccn2)=O)CC2OCCN(Cc3ccccc3)C2C1 83115,N1(C(C(CCC)(C)CC)=O)CCCC(C2CCN(c3nc(C4CC4)ns3)CC2)C1 83116,C=CC1(C(=O)NCCN(CC(C)C)C)CCN(C(C2CCCCC(=O)N2)=O)C1 83117,C(CCC(O)C(=O)N(C)C)NC(c1cccc(OC)c1)=O 83118,C(=O)(CCCCCCN=[N+]=[N-])N1C2C(NC(C(CC)O)=O)C(C2)C1 83119,N1(C(CCc2nnc(C)o2)=O)CCC(C)C(NC(=O)CCCCF)C1 83120,C1(C=C)(C(=O)NC2C(C#C)CCC2)CCN(C(=O)CC2COCCO2)CC1 83121,CC1(C)CCC(CN2CC3CNS(=O)(=O)C3C2)c2ccccc21 83122,C1(NC(C(CC#C)C2CC2)=O)CCN(C(=O)C=Cc2cnccn2)CC1(C)C 83123,c1(C(=O)OC)ccc(F)c(NC(C2CC(F)CN2C(=O)CN2CCCCC2)=O)c1 83124,N1(C(C2(C)N(C(c3cc(C(C)C)no3)=O)CCC2)=O)CC(O)CC(O)C1 83125,c1(NC(=O)NC(c2ccc(C#N)cc2)CC(=O)OCC)nc(Cl)c(Cl)nc1Cl.O 83126,c1(N(CCOC)CC2CCCNC2)nnc(-c2cncc(Cl)c2)n1CCOC 83127,C1(NC(COCCC)=O)(COC)CCN(C(C2CCN(OC)CC2)=O)CC1 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83145,Cc1cccn2cc(CC(N3CCN(CCNC(=O)C(C)C)CC3)=O)nc12 83146,N1(C(CC(C)F)=O)CC2CCC(CNC(=O)C(F)C3CCOC3)C2C1 83147,C(CN=C(NCC1(OC)CCS(=O)(=O)C1)NC1CCCC1)CCC(=O)NC 83148,c1(C(=O)NCCCC(C)NC(C2CCC(CC)O2)=O)snc(C)c1N 83149,CC1CCC(NC(=O)C(C)N2CCCC2)CN1C(=O)CC1CCCCO1 83150,c1(C(N2C(CNC(c3cc(CC(C)C)on3)=O)CCC2)=O)cc2n(n1)CC(F)C2 83151,CCCC(C)(C)CC(=O)N1CCC(C(C)(COC)NC(=O)C(O)C(C)(C)C)C1 83152,c1(C(=O)NCC2(F)CN(C(C3CCC(COC)C3)=O)C2)ccc2nnn(C)c2c1 83153,C(=O)(C1CCCn2ccnc21)NCC1N(C(c2cccc(OC)n2)=O)C2C(C1)C2 83154,N1(S(c2c(N)ncc(Cl)c2)(=O)=O)CCCC12CCS(=O)(=O)CC2 83155,C1(CNC(c2onc(C)n2)=O)CC2(CCN(C(c3[nH]c(C)c(C)c3C)=O)C2)CO1 83156,N1(C(C(C=C=C)C)=O)CC2(CC(C(=O)NCCc3cc(OC)no3)CO2)C1 83157,n1(CCC(=O)NC2C=CCN(c3c(C)cnc(C)n3)C2)cc([N+](=O)[O-])nc1C 83158,CCC(C)CCCC(=O)N(CCNC(c1ccc(C#N)cn1)=O)C(C)C 83159,c1(C(=O)NC(C)CCC(=O)Nc2ccccc2Br)ccc(C(=O)O)cc1F 83160,c1(C(C(N2CC(NC(C3CCOCC3)=O)C3(C2)CC3)=O)O)cc(F)c(F)c(F)c1 83161,N1(C(CNC(=O)NC2CCCCCCC2)=O)CCC(C(F)(F)F)C(CO)C1 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83179,Cc1c(CNC(=O)C(C[Si](C)(C)C)NC(=O)OC(C)(C)C)cnc(Cl)c1Br 83180,c1(NC)cnncc1C(=O)NCCn1cnc(C(N2CCC(N(C)C)C2C)=O)c1 83181,CC1CCCC1(C)C(=O)NC1CCC(NC(C2(Cc3cnn[nH]3)CCC2)=O)CC1 83182,c1(OC)cccc(Cl)c1C(=O)NC(C)CC(C)NC(c1cnoc1C1CC1)=O 83183,C1(C(N2C(C)CN(C(c3ccncc3Cl)=O)CC2)=O)CCC2C(C1)C2(F)F 83184,c1(C(CC)C(=O)N(CCNC(=O)C=CC(C)C)C(C)C)ccc(OC)cc1 83185,c1(C(C)NC(C2CC(n3cc(-c4cnccn4)nn3)C2)=O)ccc2c(c1)CCO2 83186,C(CCCCC(=O)NCC(O)C(F)(F)F)NC(c1c(C)cncn1)=O 83187,N1(C(c2cc(COC)[nH]n2)=O)CCOCC(C(N2CCSC(C(C)C)C2)=O)C1 83188,C(CC(C)C)(C(=O)NCC(c1ccccc1)NC(c1ccn(CC#N)n1)=O)OC 83189,C(=O)(C(CNC(C1(O)CCOC1)=O)C(C)(C)C)NCCC(CC)(C)C 83190,c1(C(=O)NCC=CCNC(C2CC(CC)C2)=O)ccncc1Br 83191,CCC(O)CC(=O)N1CC2C(NC(c3cc(-c4ccc(F)cc4)no3)=O)C2C1 83192,C1(C(N(C(C(=O)OC)C)C)=O)(NC(C2CC2(F)F)=O)CCN(C)C1 83193,c1(C(=O)NC2C(NC(c3c(C)cccc3)=O)CC2)ncc(F)cc1F 83194,C1(C(N2CCC(NC(C)=O)C2)=O)CCCN(C(c2ncccc2N)=O)CC1 83195,c1(C(c2n(CC)nnn2)NCCOC2CCOC2)ccc(Br)cc1Cl 83196,c1(C(N(CC(=O)NCC(C2CC2)NC(C2CCCC2)=O)C)=O)ocnc1C(F)(F)F 83197,N(C(=NCCC1CCCCC1C)NCc1cccc(C(C)(F)F)c1)CC(C)C 83198,N(C(=NCCCCc1cn[nH]c1)N1CCC(C2CCOC2)C1)CC(O)CF 83199,C(=O)(C(O)CNC(c1cnsc1)=O)NC(COC)COC 83200,Cc1nc[nH]c1CC(O)C(=O)N(C)CC1(CNC(c2cn(C3CC3)cn2)=O)CC1 83201,N1(C(C(n2c(C)ncc2)C)=O)CC2(CC(CC(N3CC(O)CC3(C)C)=O)C2)C1 83202,N1(C(c2ccc(-c3ccc(OC)cc3)o2)C(=O)NCC=C)CC(CO)C2(CC2)C1 83203,C12(NC(CCCNC(c3cc(C)n(C)c3)=O)=O)CCCCC1OCC2 83204,C1(N(C(CCCN(C(c2c(CC)n[nH]c2)=O)C)=O)CC)CCCC(O)C1 83205,N1(C(c2ccc(SCC)cc2)=O)CCCC(CCNC(=O)C=CSC)CC1 83206,C1(C(=O)NC(C#C)CC(C)(C)C)CN(C(C2(O)CCC2)=O)CC(C)(C)C1 83207,C(N1CCN(Cc2cc(Cl)ccc2[N+](=O)[O-])C(C)(C)C1=O)n1nc(C)c(Br)c1C 83208,Cc1c(NC(C23CC(C(=O)NC4CCCN(CC5CC5)C4)(C2)C3)=O)cnn1C 83209,C(=O)(CCCN(C(=O)COc1ccsn1)C)NCCN(CCOC)C 83210,N(C(=NCC1CC(C(F)(F)F)C1)N(C)C)CCOCC=C 83211,Cc1cc2n(n1)CCN(C(=O)C(Cc1cc[nH]n1)NC(=O)CSC(F)(F)F)C2 83212,c1(C(N2CC(NC(C(C)OCC=C)=O)C(C)C2)=O)cccc2c1OC(C)(C)C2 83213,Cc1cc(CC(=O)NCC2CCCCN2C(=O)CCc2cccnc2)ccc1Cl 83214,CP(C)(=O)c1ccc(C(N2CCCC2CNC(=O)CSC(F)(F)F)=O)nc1 83215,N1(C(c2cc(C)ns2)=O)CC2CCC(NC(=O)C(C)S(C)(=O)=O)(C2)C1 83216,N1(C(CCC(=O)NC)=O)CCCC2(NC(=O)Cc3nncn3C)CC2C1 83217,c1(NCC(O)CC2CCCO2)ccc2nc(Cl)ccc2c1 83218,c1(C(=O)NCCCCCCNC(C(N)=O)=O)cccc2c1OCC(=O)N2 83219,c1(NC(c2cn(C3CN(C(c4ccn(C)n4)=O)C3)nn2)=O)[nH]cnc1C#N 83220,C1(C(=O)NCC(CNC(c2cccc(F)c2)=O)O)CC2(C1)CC2(F)F 83221,c1(SC)nc2ncnc(NC(CNC(=O)CNN3CCCCCC3)CO)c2s1 83222,c1(C(N(C(C)C)CCNC(C2CCC3(CCC3)O2)=O)=O)ccnc2c1CCC2 83223,c1(C(=O)NC(C2CCN(C(c3cccc(C(=O)NC)c3)=O)C2)C)cc(Cl)nnc1O 83224,C=C=C(C)CC(=O)N(C1CCN(C(=O)CN(C)C(=O)OC)C1)CC 83225,C1(C)(CNC(CC2(CSC)CC2)=O)CCC(NC(=O)C(=CC2CCCCC2)F)C1 83226,CC(C)(CNC(=O)CCCn1ccnc1)CC(=O)NC(C1CCOC1)(C)C 83227,c1(C(N2CCC3CCC(C2)N3C2CC2)C(=O)NC)csc2ccccc2c1=O 83228,c1(C(C(=O)NC)N(C)CC2CCCO2)cc(Br)c(F)cc1F 83229,C=CC1(O)CCN(C(=O)CNC(=O)CNC(c2nn(C)cc2C)=O)C1 83230,c1(C(N2C(CCC)COCC2)C(=O)NCCC)ccc(C)c(C#N)c1 83231,N1(C(c2cc(F)cc(Br)c2)=O)CCC2C1CCN2C(c1ccsc1)=O 83232,Cn1cc(C(N2CC=CC2(C)C(N2CCCCC2CC(N)=O)=O)=O)ncc1=O 83233,c1(C(N2CCCC(NC(C(C)c3cccs3)=O)C2C)=O)ccc(F)c(F)c1F 83234,c1(CN2CCCC(C(=O)NCc3ncc(Cl)cn3)CC2)cc(Cl)c(Cl)cc1Cl 83235,N1(C(C2C(C)(C(F)F)C2)=O)CC2CC(C1)C2NC(=O)CCCC1CCCC1 83236,c1(C(=O)NCC2N(C)CCN(C(C3CCCCS3)=O)C2)cc2c(nn1)CCOC2 83237,C(CC(F)F)(C(=O)N(C)CCC1CCCC1)NC(C1C(OC(C)=O)C1)=O 83238,c1(C(N2CCCC(CNC(c3c(C(C)=O)ccs3)=O)C2)=O)ccc(C)c(O)n1 83239,C1(NC(C=CC(C)NC(C2CS(=O)(=O)C2)=O)=O)CCCC(O)CC1 83240,Cc1ccc(CN(C(=O)CCOCCCNC(=O)Cc2conc2C)C)cn1 83241,c1(CC(=O)NC)ccc(C(=O)NC2C=CC(CNC(C3(F)CC3)=O)C2)cc1 83242,C=CCC(CNC(=O)CC1CCCCCC1)C(=O)NC(C)COCC 83243,c1(C(=O)NCc2cccc(C#C)c2)cc(F)c(F)cc1F 83244,c1(C(=O)NC2CC3(C2)CC3Nc2nccc(CO)n2)ncc(F)cc1F 83245,C1(CC=C)(NC(=O)CN=[N+]=[N-])CN(C(=O)CCN(C)CCO)C1 83246,c1(C(N2CC(C3(NC(=O)Cc4ccc(Cl)s4)CC3)C2)=O)cc2c(=O)[nH]ccn2c1 83247,C1(NC(C2(C)CCOCC2)=O)CC(CO)C(O)C1O.C12CN(C1)C(=O)CO2 83248,C(CCN=c1[nH]c2c(c(=NCCC(N)=O)[nH]1)CCC2)NC(c1cccs1)=O 83249,N1(C(c2ccc(C#N)s2)=O)CCCC12CCCN(C(=O)C=C1CCCCC1)C2 83250,Cc1ccc(CNC2CCN(C(c3ccc(C4CC4)cn3)=O)CC2C)c(O)n1 83251,c1(CN2CCN(C(c3cccnc3C)C(=O)NC)CC2)cnc2ccsc2c1 83252,c1(CC)cc(NC2CCCC(NC(c3coc(CC4CC4)n3)=O)C2)ncn1 83253,N1(C(CCC(CC)NC(C(CC)=CCCC)=O)=O)CCC2(CCCO2)C1 83254,N1(C(c2cc(C)ncc2C)=O)CCC2(COC(CNC(c3nc(Cl)cs3)=O)C2)C1 83255,c1(C(N(CCN(C(CC(=O)OC)=O)C)C)=O)cccc2c3c([nH]c12)CCCC3 83256,c1(C(N2CCC(NC(C(=Cc3ccccn3)C)=O)C2)=O)ccc2c(c1)C(=O)NC2 83257,c1(C(N2CC(C)N(C(C3C=CCC3)=O)CC2)=O)cccc2c1CCCCC2 83258,C12(CCNC(C=CC(C)(C)C)=O)CCC1CN(C(c1cc(O)ccc1Cl)=O)C2 83259,C#Cc1ccc(C(=O)NCCC(C)N(C)C(c2cc3scnc3[nH]2)=O)c(C)c1 83260,c1(CNC(=O)OCC(CO)C(O)c2cccnc2)cc[nH]c1NC1CCCCO1 83261,C1(CN(C(CC2C(C)C2)=O)C)COCCN1C(c1ccc(N(C)C)cn1)=O 83262,C(C)(C(F)(F)C(F)(F)F)=CC(N1C2(CN(C(C3CCC(=C)CC3)=O)C2)CC1)=O 83263,C1(C(=O)NCC(N2CCN(C(c3ncn(C)n3)=O)CC2)CO)CCCCN1N=O 83264,C1(C(=O)NC(CC(=O)OCC)C)CCCCCCN1C(=O)C(O)CN1CCCC1 83265,c1(NC(c2n(CC=C)nnn2)(C)C(C)SC)nc2c(n1C)CCCC2 83266,c1(C(C)=O)cnc(N2CCNC(C)C2)nc1C.C1(C=O)CC1C 83267,C1(C(F)F)(OC)CC(C(=O)NCCN(C(=O)CCCNS(C)(=O)=O)C2CC2)C1 83268,C(=O)(CCCC(F)(F)CO)NC(CNC(c1n(CC)ccn1)=O)(CC)CC 83269,Cn1cc(CCC(=O)NCC2CCC(NC(=O)CC3CCCOC3)C2)cn1 83270,c1(NC(C2(CNCc3c(C)ncc(Cl)c3)CC2)=O)ncc(C#N)cc1I 83271,c1(CC)c(C(=O)NC(C2CCN(C(=O)CCCCSC)C2)(C)C)cnn1C 83272,C(CCC(C)C(=O)NCC(C)(C)CCNC(c1sccc1OC)=O)OC 83273,N1(C(c2nc(COC)sc2)=O)CCC2(CCCC2NC(c2[nH]c(C)nc2C)=O)C1 83274,C#CCCCCC(=O)NC(C)(CNC(c1cn(C2CCOC2)cn1)=O)C1CCC1 83275,C1(C(N2CCC(O)(CNC(CN3CC(C)C3)=O)C2)=O)CCCC12CCOCC2 83276,C1(OC)CN(C(c2csc(-c3cccs3)n2)=O)CC1NC(=O)CNc1nccs1 83277,C(Cc1ccco1)(C(=O)N1CCCC1CC1CC1)NC(c1ccns1)=O 83278,C1(C(=O)NCC2=C(C)CCC2)CC2CCC(C1)N2C(c1c[nH][nH]c1=N)=O 83279,Cc1oc(C(=O)NC2CCN(C(=O)CCc3cccc(O)c3)C2C)cc1Br 83280,C1(CC)CC(O)CN1C(=O)CC1CC(NC(=O)CC2OCCC2C)C1 83281,C(=O)(C(C)C(=O)NCC1(CC(=O)NC(c2cncs2)C)CC1)OC 83282,N1(C(CCCC)=O)CC2(COC(CNC(C3(F)C(C)(C)C3(C)C)=O)C2)C1 83283,C1(C(F)(F)F)(NC(CC(C)(C)CNC(=O)CC2CC23CC3)=O)CCCCC1 83284,c1(OC)cc(C(N2CC(F)CC2CN(C(=O)C(c2cnn(C)c2)C)C)=O)n(C)n1 83285,c1(C(=O)NCC2=CCN(C(=O)Cc3ccccc3F)CC2)cc(Cl)ncc1F 83286,c1(CC(C)C)ccccc1C(F)(F)F.C1CC(F)Cn2cc(nn2)SCC(=O)N1 83287,C(=O)(CC1=CCCC1)NCC(C)N(C(=O)Cc1ccc(C(C)(C)C)cc1)C 83288,c1(C(=O)NC2CN(C(CC(CC)SC)=O)CC(O)C2)cncc2sccc12 83289,c1(OC)cc(C)c(S(=O)(=O)N2CCN3CCCC3C2)cc1Cl 83290,c1(NC(COC(C(c2ccccc2)N(CC)CC)=O)=O)cccc(F)c1C 83291,CC(C)CC(C(=O)N1CCCC1CCNC(=O)CC1CCC(=O)NC1=O)N(C)C 83292,C1(CNC(C(CCC)(C)CCC)=O)CC2(CCOCC2)CN1C(c1cnns1)=O 83293,N1(C(C2(N(C(c3ncc(NCC)nc3)=O)C3CC3)CCC2)=O)CCC(O)C(F)(F)C1 83294,N1(C(C=C(C)C)=O)CC2CC(NC(c3cc(C)on3)=O)C2C1 83295,C12(CCNC(C3ON=C(C)C3)=O)CCC(C1)N(C(c1cc(O)cc(Cl)c1)=O)C2 83296,N1(C(C2CCC(=O)N2)=O)CC2CC(NC(c3cc(C(F)F)[nH]n3)=O)C2C1 83297,c1(C(N(C)CC2CCN(C(COCCCC#C)=O)CC2)=O)ccc(CO)c(Cl)c1 83298,N1(C(CCS(C)(=O)=O)=O)CCC(NC(C2CC(C)(F)C2)=O)C(F)(F)CC1 83299,C1(C(C)(C)C#N)CCN(C(c2cc(Cc3cccs3)ccn2)=O)CC1 83300,Cn1cnc2ncnc(N3CC(F)(F)CC3C(=O)Nc3c(F)cc(F)cc3F)c12 83301,CN=c1[nH]c(=NCc2cc(Br)ccc2C)[nH]c(=NCCSC2CC2)[nH]1 83302,c1(CC)nn(C)cc1C(C)NC(=O)Nc1cccc(OC2CC2)c1 83303,c1(COCCCC(=O)Oc2cc(F)cc(F)c2)c(F)cccc1Br 83304,C1(C(N2C(C3(C(=O)NC(c4ccc(O)cc4)C)CC3)CCC2)=O)CC1C1CCC1 83305,C1(O)(CN(C)C(C2CCC(F)(F)C2)=O)CCCN(C(c2ccc(C3CC3)o2)=O)C1 83306,C1(NC(C(CC)c2ccccc2)=O)CC(F)(F)CC1NC(c1ccc(Cl)cc1)=O 83307,c1(CNC(=O)NC2CCC2C(F)(F)F)cccc([N+](=O)[O-])c1F 83308,C1(CC(=O)NC2CCN(C(CCCCC#C)=O)CC2O)CCCC2(CCC2)O1 83309,C(=O)(CC(C(=O)NCC1CC(NC(c2coc(Cl)c2)=O)C1)N(C)C)OC 83310,S(=O)(=O)(c1ccc(Br)cn1)N(C1CCNCCC1C)c1ccc(SC)cc1 83311,C1(C(=O)NC(CC)C(=O)N(C)CC2COC(=O)N2)CCCCC(=O)C1 83312,CCCC(CCCNC(=O)CC(C)Cc1cccc(F)c1)NC(C1OCCO1)=O 83313,C#CCCCC(C)C(=O)NC1CC12CCN(C(c1ccccc1C(C)=O)=O)CC2 83314,CC1(C)CC(C)(C(=O)NCCCC(F)(F)F)CN1C(C1CCC(=O)NC1)=O 83315,Cc1ccc2c(C(N3CCCC(NC(=O)C(C)(C)C(C)(F)F)CC3)=O)n[nH]c2c1 83316,C1(NC(c2c(C)nn[nH]2)=O)CCCCC12CCN(C(=O)C(C)(C)C(F)(F)F)C2 83317,C1(C2CCN(C(C3CCCC3C)=O)C2)(NC(C2CC(C)=C(C)CC2)=O)CC1 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83404,c1(C(CNC(C2CC2C2CC2)=O)NC(COCC)=O)cccc(Cl)c1 83405,c1(OC)nccc(C(=O)NCC2C=CCN2C(=O)C(N2C(=O)CCC2=O)C)c1F 83406,C(C(CNC(=O)CCCCC1CC1)S(C)(=O)=O)NC(c1cc(C)no1)=O 83407,c1(N)ccnc(C(F)(F)F)c1.c1(C(N(C)CCN2CCOC2=O)=O)ccc(C2CC2)o1 83408,C1(C(=O)Nn2cc(-c3nc(C4CCCO4)no3)nn2)CCCC1C(F)F 83409,C(CNC(=O)C(C)n1ccnc1)(CC(=O)NCC(C)C(C)O)OC 83410,c1(C(N(CCN(C(C2C(CC)CCC2)=O)C)C(C)C)=O)cc(=O)n2nccc2[nH]1 83411,CC(C)(CNC(c1ocnc1C1CC1)=O)CCNC(=O)C=CCOc1ccccc1 83412,CC1(CN=c2[nH]nc(C3CC3)o2)CCN(C(C2CSCCS2)=O)CC1 83413,C(=O)(CCS(C)(=O)=O)NC12CC(NC(CCc3c(OCC)cccc3)=O)(C1)C2 83414,C(C1COCc2ccccc21)NC(c1ccc(OCC(C)C)cc1)=O 83415,CC(C)CS(=O)(=O)CC(=O)NCC1CC2(CO1)CN(C(=O)C(C)S(C)(=O)=O)C2 83416,N1(C(CCSCC)=O)CCN(C(=O)CCc2ccc(OC)cc2)C(CC)C1 83417,C1(NC(C2(C(N(C(C)C)C)=O)CC2)=O)CCCC1NC(=O)C1=CCC1 83418,c1(C(=O)NCC(CC)NC(c2c(C)coc2C2CC2)=O)cccc(OC2CC2)c1 83419,CC1(C)C(NC(c2nccc3ccsc23)=O)C2CCCN(c3cncc(Cl)n3)C12 83420,C1(C(N2CC(O)(CNC(c3cn(C4CC4)cn3)=O)C2)=O)(COC)CC1(F)F 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83438,c1(C(=O)OC)ccc(Br)c(NC(=O)NCc2ocnc2C(C)(C)C)c1 83439,c1(CCC(N2CCC(Cn3cc(CC(C(C)C)O)nn3)C2)=O)ccc(F)cc1F 83440,C(=O)(C(F)C(C)CNC(=O)CCN1CCCC1=O)NCC(CC)CC 83441,C1(COCC)CCCN1C(C1CCC(n2cc(C(C)(C)CC)nn2)C1)=O 83442,c1(OC)cccc2c(C(=O)NCC3CN(C(c4n[nH]cc4OC)=O)C3)c(C)[nH]c12 83443,CC1CC(CNC(c2cncs2)=O)CN1C(c1cc(C2CC2)nn1C)=O 83444,c1(C(=O)NCCC2(NC(CC(CCC)(C)C)=O)CC2)ncc(F)c2ccccc12 83445,CC1(CC(F)(F)F)CN(NC2CC(Nc3cn(Cc4ccccc4)cn3)C2)C1 83446,Cc1cc(Br)cc(C)c1CN1CCN(C(c2ccc(O)cc2CO)=O)C(CO)C1 83447,N1(c2nnn(C)n2)CCCC(C2CC2NC(c2cccs2)=O)C1 83448,N1(C(C(CNC(c2c(CC)ncnc2)=O)O)=O)CCN2CCCCC1C2 83449,c1(C(N(C2CC(NC(C3(CC#C)CCCC3)=O)C2)C)=O)ccccc1C1CCC1 83450,C1(C(N(C(CCC)C)CC)=O)CN(C(c2cnn(CCC)c2)=O)CC12CCC2 83451,c1(OC)ccc(CC(=O)NC(C)C(C(C)C)NC(C)C)cc1[N+](=O)[O-] 83452,N1(C(c2c(C)ncn2C)=O)CC(C)C(NC(c2ccc3ncnn3c2)=O)C(C)C1 83453,C#CCCCC(C)C(=O)NC1(CNC(=O)Cc2nocc2CC)CCCCCC1 83454,N1(C(C(C(=O)OCC)C2CC2)=O)CCOC2(C1)CN(C(C1CCCCO1)=O)C2 83455,C#CC1CCC(CN2CC(C)CC(C(=O)NCc3c(C)cccc3F)C2)CC1 83456,C1(NC(=O)CC2C3COCC23)CCC12CCCCC2 83457,N1(CCNC(=O)C=C(C2CC2)C2CC2)CCN(C(=O)CC2COC(=O)N2)CC1 83458,CC1(CNC(C2(F)CN(C(=O)Cc3cscn3)C2)=O)NC(=O)NC1=O 83459,c1(C(=O)NCCn2cc(C(N(C)Cc3nnc(O)o3)=O)nc2)cccnc1S 83460,N1(C(=O)OC(C)(C)C)CCC(C(N2CC(N3CCN(C(N)=O)CC3)C2)=O)(CF)CC1 83461,c1(C(N2CCCC(N(C(C3C(C)CC=CC3)=O)C)C2)=O)cc2scc(Cl)c2[nH]1 83462,C#Cc1cccc(SCc2nc(NC(C)=O)ns2)c1 83463,C1(CCCCNC(CCOCC)=O)CCN(C(=O)C(O)CC2CCOCC2)CC1 83464,C#CCC(CC(F)F)C(=O)NCCOC1CCN(C(=O)C2=C(Cl)CCC(C)C2)C1 83465,c1(CCC)cc(C(=O)NCCN(C(=O)CCCn2cccn2)CCOC)nn1C 83466,Cc1c(CCC(=O)NC(C)CC2CN(C(=O)C(CCO)N(C)C)C2)cnn1C 83467,c1(C(=O)NC2CN(C(CCCCC#C)=O)CC(O)C2)cncc2n[nH]cc12 83468,C1(NC(c2ccccc2Cl)=O)C2CCC(C2)C1C(=O)NC1CC(O)C(O)C1 83469,c1(CC(=O)N(CC(C)(C)NC(C(C)O)=O)C)cnnn1C 83470,c1(NC2CCN(CCOC)C2)cc(Br)ccc1S(=O)(=O)NCc1ccc(Cl)nc1 83471,CCC(CC(=O)N(C)CCOCCNC(c1ccc(COC)s1)=O)OC 83472,C1(C(=O)NCCN(C(C2CCCC23CCC3)=O)CC)CN(C)CC(C)O1 83473,c1(C(N2C(CCCNC(C3(C)CC4CC4C3)=O)CCC2)=O)ccc(Cl)c(Cl)c1N 83474,c1(C(=O)NCCN(CCC)C(C2(C)CCCCO2)=O)cc(C(F)(F)F)nn1CC 83475,CC1CCCCN1C(C1(CNC(=O)C(C)OC2CCCC2)CC=CC1)=O 83476,Cn1cccc(C(=O)NC2CCC(C(N3CCC(O)CC3C3CC3)=O)C2)c1=O 83477,C(C(CC1CC1)C(=O)NCC1C2CCCCC12)NC(c1ccc(CC)o1)=O 83478,c1(C(=O)NC2C(CNC(Cn3nnc(=N)[nH]3)=O)CCC2)cccn2nccc12 83479,CC1CCN(Cc2ccc(Cl)cc2Cl)CC1NC(c1cnn(C(F)F)c1)=O 83480,CCCC(CNC(C1CCCCCN1C)=O)C(=O)N(C1CCCCC1CC)C 83481,N=c1[nH]cc2c(c1C(N1CC3(CCN3C(C3C=CCC3)=O)C1)=O)CCC2 83482,N1(C(CCCC(C)O)=O)CCCC12CCN(C(c1cc(Cl)c(Cl)[nH]1)=O)C2 83483,C1(CC(N2CC3CSCC(C3)C2)=O)C2CCC(C2)N1C(C1(CO)CCCC1)=O 83484,C12(C(=O)NC3CCCN(C(C(F)OC(C)=O)=O)C3)CCCCC(OC(C)C)(C1)C2 83485,CCCCCC(C)(C)C(=O)NCC(C)NC(c1nnn(C(C)(C)C)n1)=O 83486,c1(C(=O)NC2C3CN(C(c4cc(C)c(C)nn4)=O)CC32)cccc2nsnc12 83487,N1(C(C2CCN(CC)C2)=O)CCCC2(CCCN2C(C23CC4CC2C3C4)=O)C1 83488,c1(NC(C2N(C(c3c(C)ccs3)=O)CC(F)(F)C2)=O)ccc2c(c1)C(=O)N(C)C2 83489,C=CCCCC=CC(=O)NCCC1(NC(=O)C(O)Cc2cnc[nH]2)CCCC1 83490,C12(C(=O)NCC3CCN(C(C=CC(C)=O)=O)C3(C)C)CCOC1CCOC2 83491,C(=O)(C(C(C)(C)O)NC(=O)C(C)c1ccco1)NCc1c(COC)noc1 83492,N1(C(C(CC=CC)C)=O)CCc2cc(CNC(c3ccco3)=O)ccc2C1 83493,c1(CNC(CC=C)=O)cc(C(=O)NC(C)C(C)COC)n[nH]1 83494,c1(CC(N2CC(F)(C(=O)NCC3COCC(C)O3)C2)=O)cccc2ccoc12 83495,N1(C(CNS(N)(=O)=O)=O)CCOCC(CNC(c2ccc(-c3ccco3)o2)=O)C1 83496,C(=O)(CCCCC(C)(C)C)N(c1ccc(C2CC2)nc1C)CC.c1(=O)c(=O)n1CC 83497,CN1C(=O)CN(CC(N2CC(CNC(c3ccco3)=O)C(O)C2)=O)C1=O 83498,N1(CC(=O)NC(C2(O)CCN(C(C3(C=C)CC3)=O)C2)C)OC(C)(C)CC1=O 83499,C(=O)(CC(C)C(=O)NC(C)(C)CCNC(=O)COCC=Cc1ccccc1)OC 83500,N1(C(C(C)C(F)F)=O)CCN(C(C2(C#N)CCSCC2)=O)CC1CF 83501,N1(C(C2C3CN(C(C4N(C)CC(O)CC4)=O)CC32)=O)CCC12CCOCC2 83502,N1(C(c2ccc(CC(=O)Nc3ccc(C)cc3)o2)C)CCC12CC(C(N)=O)C2 83503,C=C1CC(C(=O)N(c2cccc(SCCC)c2)C2CC2)N(CCOC)C1 83504,CC(C)S(=O)(=O)C(C)C(=O)NCC(C)(C)NC(=O)Cn1cc([N+](=O)[O-])ccc1=O 83505,c1(NCCCSCC)oc(C)nc1C(=O)NC1CCCCC1 83506,C#CC1CN(C(C2(NC(=O)C=Cc3cocn3)CCSC2)=O)CCO1 83507,C1(C)(C(N(C)OC2CCCC2)=O)CCCN1C(C1COC(=O)N1)=O 83508,C1(CC(=O)N(C2CCN(C(=O)CC3(O)CCC3)C2)C)CC2(CCC2)C1 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83526,CCCC(CCC)C(=O)NCC(c1ccccc1CC)NC(c1c[nH]nc1C)=O 83527,Cc1cnc(CC(=O)N(C(CNC(=O)CCCN2CCCCC2)C2CC2)C)s1 83528,N1(C(CCOCC(C)C)=O)CC(NC(C2C3CCCCCC23)=O)CC(F)C1 83529,CC(C)CCCCN(C(=O)C(n1cc(-c2cnc(C3CC3)s2)nn1)C)C 83530,C1(C(=O)NCC(CC)(CC)NC(=O)Cc2ccc(C)c(O)c2)CC12CCSCC2 83531,C(=O)(C(C)(CCC)CCCCCC)NCCOCCOCCNC(C(CC=C)C)=O 83532,N1(C(C)(C)C)CC2(CNCC(F)(F)F)CC(F)(C1)C2.N12CCC(C(O)C1)C2 83533,Nc1ccc(F)c(CNC(=O)NCCCn2nccn2)c1 83534,C1(C(=O)NC2CC(NC(c3ncn(C)n3)=O)CC2O)CCc2ncncc2C1 83535,c1(C(=O)NC2C(NC(=O)Cc3cncn3C3CC3)C2)cc2ccccn2n1 83536,Cc1ccccc1OCC(=O)NC1CC(C(=O)NCC(C)CO)C1 83537,C1(C)(CNC(COC(CC)C)=O)CCCN(C(c2cc(C(C)(C)C)n[nH]2)=O)C1 83538,N1(C(C(=O)NCCCCC)=O)CCCC(C2(NC(=O)CC)CC2)C1 83539,O=C(CCCCc1cccs1)N1CCC1.C1(c2ccc(F)cc2)(CCCC(=O)N)CCCCC1 83540,N1(CC)CCCC(N=c2[nH]c(=NCCc3cc(CC)no3)c3cccc(F)c3[nH]2)C1 83541,C(=O)(C(=O)N=S(C)(C)=O)N1CCC(C)(NC(C2C(=C)CC2)=O)C1 83542,C1(C(N2C(C(=O)OC)C=CC2)=O)CN(C(c2cc(OC)no2)=O)CC1C 83543,C=C(Cl)CCC(=O)NC(C)CN(C(=O)CCC1CCCC1O)C 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83562,C1(C2CN(C(=O)COc3cccc(Cl)c3Cl)C2)(NC(c2nc(C)nn2C)=O)CC1 83563,C1(CC=C)(C(=O)NC(C(C)C)c2ncc[nH]2)CCCN1C(c1ccncn1)=O 83564,c1(C(N(C2CN(C(c3ncncc3Cl)=O)C2)C)=O)cc([N+](=O)[O-])n[nH]1 83565,CC1CC(C(=O)NC(C)(C)CN(C(=O)COc2ccc(CO)cc2)C)C(=O)O1 83566,C#CCCCCCC(=O)N1CCCCCC1C(=O)NC(CCCCC)C1CC1 83567,c1(C(C(=O)NCc2cccs2)N(C2CCCSC2)CCOC)ccc(F)cc1C 83568,C(=O)(C#CC1CCC1)N1CCC(CNC(CSc2n(C(C)(C)C)cnn2)=O)C1 83569,C(=O)(C1=NNC(C(F)(F)F)C1)N(CC(C)NC(CCC(=O)c1ccc(C)s1)=O)C 83570,N1(C(CCC(C)OC)=O)C2CCC1CC(N(C(=O)CCc1cc(C)no1)C)C2 83571,Cc1noc(N)c1C(=O)NCc1cc(C(=O)NCc2ccccc2Cl)n(C)n1 83572,C1(NC(C(CCCNC(C)=O)C)=O)CCSC12CN(c1cc(C)nc(C)n1)C2 83573,c1(C(N2C(C)CCC(NC(CCCC(=C)C)=O)C2)=O)cc(=O)c2ccncc2o1 83574,C1(OC)CN(C(c2ccc(C(C)C)cc2)=O)CC1NC(c1scnc1C)=O 83575,c1(OCC)ccc(C)nc1C(=O)NC(C)CN(C)C(c1[nH]ccc1CN(C)C)=O 83576,N#CC1CN(C(C2CCCN2Cc2cccc(O)c2OC(F)(F)F)=O)CCO1 83577,C(=O)(C1=CC2CCCCCCC12)NCCC(C)N(C(=O)Cc1cccc(F)c1)C 83578,N1(C(C(C2CCCCC2)C)=O)C2CCC1C(F)C(NC(c1cc(Cl)n[nH]1)=O)C2 83579,C(C(=O)C(N)C(C)C)N(C)Cc1ccc(SC)cc1 83580,c1(C(=O)NCCc2cc(CC)no2)cc(F)c(F)cc1OC 83581,c1(CNC(c2n(C)cnc2Br)c2nnnn2CC(F)F)cccn2ccnc12 83582,c1(C(=O)NC2(CNC(C(c3ccccc3)OC)=O)CCOC2)cccc(C)c1Cl 83583,Cc1occc1CNC(C1C=CCN1C(=O)COc1ccccn1)=O 83584,Cc1nc(C)c(C(N2CC3(COC(CNC(C4CN(C)C4)=O)C3)C2)=O)c(C)n1 83585,CC1CN2CC1(C)C(=O)NC(CCN1CCC1CC)CCS(=O)CC2=O 83586,C=CC1OCCC1C(=O)NC1CC(O)C1CC(N1CC(N(C)CC)C1)=O 83587,N1(C(c2c(C#C)c[nH]n2)=O)C2CCC1CN(C(c1ncn3c1CCC3)=O)C2 83588,C1(C(=O)NC2(c3noc(C)n3)CC2)(OC)CCN(C(C2CNC(=O)C2)=O)C1 83589,C(=O)(C1CCOc2ccccc21)NC(CNc1c(C#N)nccn1)C1CC1 83590,c1(C(=O)NC2(C)CN(C(C3CCCN(C)C3)=O)C2)cnn2ccn(C)c12 83591,c1(OC)cc(C)cc(C(=O)NC2(C)CC(NC(C34CC3CNC4=O)=O)C2)c1N 83592,N1(C(CC2(OC)CCC2)=O)CC(C)CN(C(c2cncc(C)c2Cl)=O)CC1C 83593,C(=O)(C(F)(F)CCn1ccnn1)N(CCN(C(CCC#C)=O)C)C 83594,N1(C(c2cc(OCC)ncc2)=O)CC2(CCCC2NC(C2COC(=O)C2)=O)C1 83595,C1(C2CCC2)(CNC(C(C)(C)OCC)=O)CCN(C(c2cc(CO)on2)=O)CC1 83596,c1(C(N2CC(NC(c3n(C)cc(Cl)c3)=O)C(F)C2)=O)ccc2sncc2c1 83597,C(CC(CC)C(=O)N1CC(O)(C(C)(C)CNC(=O)COC(F)F)C1)=CC 83598,C1(NC(c2ccc(CNC(=O)C(F)F)nc2)=O)CC2(C1)CC(O)C2 83599,N1(C(CCC(CC)NC(=O)Cc2cccs2)=O)CCN2C(=O)NCC2C1 83600,C(c1ccc(O)cc1)=CC(=O)N(CCCNC(c1csc(C(C)C)n1)=O)CC 83601,Cc1cc(C)c(C#N)c(NC(CNC(c2c[nH]cc(C)c2=O)=O)CO)n1 83602,c1(C(=O)NC(CNC(C2CC3(CC3)C2)=O)C2CC2)cccc2c[nH]nc12 83603,C1(CNC(c2c(CC)cccc2)=O)CC(C(=O)N2CC(N=[N+]=[N-])C2)=NO1 83604,N1(C(C2C(C=C)C2)=O)CCOC2(CCN(C(C3CN4CCC3CC4)=O)CC2)C1 83605,N1(C(c2c(CNC(C3C(C)CC3)=O)nccc2)=O)CCn2nccc21 83606,c1(OC)nc(C(=O)NCCCC(C)(C)NC(=O)CN2CCC2C)sc1C 83607,C(C1CCCO1)=CC(=O)NCC1CCN1C(=O)CC1(C2CC2)CCC1 83608,C1(OC(C)C)CCN(N2CCn3c(C4CCCC4)nnc3C2)C1 83609,Cc1cc([N+](=O)[O-])cn(CC(=O)NCc2ccc(CO)cc2F)c1=O 83610,c1(C(=O)NC(C2CCCOC2)C(N2C(CC(=O)NC)CC2)=O)ccc(C(=O)O)cc1 83611,N#Cc1cccnc1NC(C12CC(C(N3CCC(O)C(F)C3)=O)(C1)C2)=O 83612,c1(CN2CCCC(C(C)NC(c3ccsc3)=O)C2)ccc2cc(F)ccc2n1 83613,c1(OC)cccc(C(=O)NCC2CCN(C(=O)CCC3CCC3)CC2)c1 83614,C(=O)(C1CCCc2nncn21)N(CCC)CCNC(=O)Cc1ccnc(O)c1 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83687,N1(C(CSC)=O)C(C(=O)NCC(C)S(C)(=O)=O)CCC12CC2 83688,O=C(C1=CCN(C(=O)CCc2ccncc2)C1)NCc1cc[nH]n1 83689,C1(C(=O)NCc2c(CC)nccn2)CN(C(C2(CC3CC3)CCC2)=O)CC12CC2 83690,C1(CNC(CCC=C=C)=O)C2CCC(C2)N1C(c1cc(-c2ccc(Cl)s2)on1)=O 83691,n1(CCOC)cc(C(=O)N(C2CC(SC)C2)CCCO)nn1 83692,Cc1cccc(-c2noc(C(N3CCN(C(=O)OC(C)(C)C)CC3=O)C)n2)c1C 83693,N1(C(c2n(C)c3c(c2)ccs3)=O)CCC2(CCC(NC(c3ccns3)=O)C2)CC1 83694,Cc1nc(N)cnc1C(=O)NCC1CCN(C(=O)COC2CCCOC2)CC1 83695,c1(C2C(C(=O)NC3C=CC(CNC(C(CC)=CC)=O)C3)C2)cccc(Cl)c1 83696,C1(C(=O)NC2(CNC(CN(C3CCC3)C)=O)CCC2)COCCN1C=O 83697,CC(C)S(=O)(=O)CC(=O)NC1CC(CNC(C2CCCN2S(C)(=O)=O)=O)C(O)C1 83698,Cc1ncc(C(=O)NC2CC2CNC(c2cccc(C(C)(F)F)c2)=O)c(C)n1 83699,C1(CNC(c2ncncc2Cl)=O)CN(C(=O)C(F)(F)CC2CCCO2)CCC1(F)F 83700,Cc1cc(S(N)(=O)=O)sc1C(N1CCC(C2(NC(=O)C(=O)N(C)C)CC2)C1)=O 83701,C(C(=O)N1CCC(CNC(C2(C(=O)N(C)C)CC2)=O)C1)(C(C)C)SC 83702,c1(OCC(=O)NC2CC(NC(c3n[nH]cc3Br)=O)C2)ccc(Cl)cc1 83703,C(C(C(=O)NCCC1CC(C)C1)C(C)(C)C)NC(CC1C(C)=NNC1=O)=O 83704,C1(NC(CCCOC)=O)COCCC1NC(=O)C(CC1CCCC1)OC 83705,n1(CC)c(NC(=O)NC2CCC(c3nc(C)no3)C2)nc2c1CCCC2 83706,CC1CN(C(c2cocn2)=O)CC1CNC(C12CSC(C1)C2)=O 83707,C(C(O)C(F)(F)F)N(C(=O)C(C)CN(C)Cc1ccccc1)CC(=O)OC 83708,c1(OC)cc(NC(C2CCCCN2C(=O)CCC2CC(F)(F)C2)C)ncn1 83709,c1(CN(C(=O)NC(CCC=C)C2CC2)CC)cccc(F)c1N1CCCC1 83710,N1(C(CSCC#C)=O)CCN(C(c2ccccc2C)=O)C(CF)C1 83711,C(=O)(C#CC1(C(F)(F)F)CC1)N1CC(C(C)NC(c2c(CC)noc2)=O)OCC1 83712,Cc1ccc(F)c(C(=O)NCC2CCC(C(=O)NCC(C)(C)O)C2)c1 83713,C1(NC(c2coc(Cl)n2)=O)CC2CCC1(CNC(C1CC1CF)=O)C2 83714,N1(C(c2ocnc2COC(C)(C)C)=O)CCC(F)(F)C(CC2CCOC2)C1 83715,CC(C)C(C)CC(=O)N1CC2CC(C1)C2NC(C1COCC(C)(C)O1)=O 83716,N1(C(=O)C=CCOc2ccccc2)CC2CC(C1)N2C(=O)Cn1cccc1 83717,C1(CNC(C(CC)F)=O)CCN(C(=O)Cc2ccc(C3CCC3)cc2)CC1(F)F 83718,c1(CC(N2CC(NC(CC(C(=C)C)O)=O)C(O)C2)=O)c[nH]c2cccc(Cl)c12 83719,c1(C(=O)NCC2(O)CN(Cc3cccc(Cl)c3)C2)cccn2nccc12 83720,C1(C(N(CC(C)NC(=O)CCCSC)CC)=O)CC(=O)N(C2CC2)C1 83721,Cc1ncnc(N2CCCC(NC(c3cc(=O)n(C)cn3)=O)C2C)c1Br 83722,C(CC(C(=O)NC(C1CCOC1)CO)NC(c1sc(C)cc1C)=O)OC 83723,C(=O)(C1CSc2ccccc21)NC1CC(NC(C=C(CC)CC)=O)C1 83724,C(=O)(C(N=[N+]=[N-])C(C)C)NCC1(C(=O)NCc2ncc(C)nc2)CC1 83725,C1(C(=O)NCCC(C)N(C(=O)CC2CCC(=O)C2C)C)CCC(C#N)CC1 83726,CCC(CC)C(C)C(=O)N1CCCC(CC(=O)NCC2(C)CCC(=O)N2)CC1 83727,Cc1csc2cc(C(=O)NCC3CN(C(=O)COCC(C)C)CC(C)(C)O3)[nH]c12 83728,C1(COC)(NC(=O)C=CS(C)(=O)=O)CCN(C(=O)C=Cc2cscn2)CC1 83729,CC(C)C(O)CNC(=O)CCOCCNC(=O)CCc1nccs1 83730,Cc1cc(N2CCC(N(C)C(c3cncs3)=O)CC2)c(C#N)cn1 83731,c1(CCCNCc2ncc(-c3ccccn3)o2)ccc2c(c1)OCCO2 83732,Cc1noc(C(=O)NCC(F)CNC(C2CN(c3nnnn3C)C2)=O)c1C 83733,C(=O)(C#CC1CCOC1)NC1CCC(C)(CNC(CCS(=O)(=O)N(C)C)=O)CC1 83734,C#CC1(C(N2CC(C)(CSC)C2)=O)CN(C(=O)CN2C(=O)CNC2=O)C1 83735,C1(NC(c2c(OC)n[nH]c2)=O)CCN(C(=O)CC(C)F)CCC1(F)F 83736,C(CC(=O)N1CCCCC1C(C)(C)O)(C(C)C)NC(c1cc(C)on1)=O 83737,C(C(C)C)(C(C(=O)NCC(F)F)N1CCC(n2cnc(C#N)n2)CC1)OC 83738,C1(NC(C2CC(=O)NC(=O)C2)=O)CN(C(=O)CCCN2CCCC2)C2CCCC12 83739,C(=O)(C(C)CC(C)(F)F)NCCN(CCC)C(c1cc(C)c(C#N)cn1)=O 83740,CC(c1ccccc1)=CC(=O)NC(C)(CO)C(=O)NCC1(O)CCCC1C 83741,C1(C(N2CCCC(CNC(c3c(C(C)C)[nH]cc3)=O)C2)=O)CCS(=O)(=O)N1C 83742,N1(C(C)C)CC(C(=O)NCC(O)CNC(c2occc2Cl)=O)CCC1=O 83743,CC(C)CN=c1[nH]c(N2CCN3C(=O)CCC3C2)nc2c1CCCCC2 83744,C1(C(C)C)C(C(=O)NCC2CC=CC2)CCN1C(=O)CCc1nc(=N)[nH][nH]1 83745,N1(C(C(C=CC)O)=O)CCCN(C(c2ccc(NC(=O)NC)cc2Cl)=O)CC1 83746,CCC(C)C(C)C(=O)NC1(C)CCN(C(=O)C(C2CC2)N(C)C)C1 83747,N1(C(Cc2ccc(SC)cc2)=O)CCC(NC(=O)CCCCCF)CC1C 83748,C1(C(=O)NCc2cn(C(C)C)nn2)(NC(C(C)C)=O)CCCC1 83749,C1(NC(CCc2c[nH]c(=N)[nH]2)=O)CC2CC1CC2NC(=O)CN1CC=CC1 83750,c1(C(N(C2CCN(C(C(C)OCC)=O)C2)C)=O)onc(C)c1-c1ccc(O)cc1 83751,C1(C(=O)NCC(C)(C)OCCNC(C2(COC)COC2)=O)CCC(=O)N1C 83752,S(=O)(=O)(c1ccc(F)cc1)N1CCCC(C(=O)NCC(C(CC)C)CO)C1 83753,C(CC(=O)N(C1CCC(CO)CC1)C)(C(C)(C)C)NC(C1C2CN(C)CC21)=O 83754,C1(C(N(C2CCN(C(=O)Cn3nnc(C)n3)C2)CC)=O)CN2CCN1CC2C 83755,C1(NC(=O)CN2CCCC2)COC2(CCCN(C(=O)COC3CCOCC3)C2)C1 83756,C1(NC(=O)Cn2cc(CO)nn2)CCCCN(C(c2ccc(F)nc2)=O)C1 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83775,C#CC1CN(C(=O)CCC2CCN(C(c3snnc3CC)=O)C2)CCN1C 83776,c1(C(c2n(C)nnn2)Nc2ccc(F)cc2)ccc(-c2cn[nH]c2)cc1 83777,Cc1nn(Cc2cn(CCC(N3CCC(N4CCCC4)C3)=O)nn2)c(C)c1C 83778,C(CCC(=O)NCC(C)(F)CNC(=O)C(C)c1ccco1)C1C(C)C1 83779,CCCCC(O)CC(=O)NC(CC(F)F)C(=O)N(C1CCCCC1O)C 83780,C1(CC(=O)NC(C)Cc2cnc[nH]2)CCCN(C(=O)CC2CSC2)CC1 83781,CC1(C)CC(CC(=O)NOCc2cccnc2)CN1C(=O)Cn1cnnc1O 83782,c1(C(c2n(CC(=C)C)nnn2)NC2CC2CC)ccc(OCC)cc1F 83783,C12(C(=O)NCC3C(CNC(C4(C)COC4)=O)C3)CCC(C(F)F)(CC1)C2 83784,CN1CCN(C(=O)CC2C=CCC2)CC1CNC(c1ncccc1Br)=O 83785,N1(C(C(C)=C2CC2)=O)CCC2CCN(C(C3(C#N)CCC3)=O)CC2C1 83786,C1(C(CN)O)CCN(CCc2nnc(-c3ccccc3F)s2)CC1 83787,c1cc(=NC2CC3CCC2N(Cc2cncnc2)C3)[nH]c(OCC2CCC2)n1 83788,c1(OC)ccc(F)cc1CCC(=O)NC1(CCNC(=O)CCSC)CC1 83789,N1(C(c2c(C)sc(Cl)n2)=O)CCC2(CCCN2c2ncnn3cccc23)CC1 83790,C12(CNC(C=CCCC)=O)CCCC1CCN2C(=O)CCOc1ccccc1 83791,C1(CC#C)CCN(CC(O)CCC2CC2)C1 83792,c1(CC(N2CC3C(NC(C(F)=CCC)=O)(CC3)C2)=O)coc2ccc(C)cc12 83793,CCCCCC(C)(CC)C(=O)NCC1(F)CCN(C(c2ccc(C)cc2)=O)C1 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83828,C1(C(N2C(CNC(c3cnns3)=O)CC3CC32)=O)CCc2ncccc2C1 83829,C12(C(=O)NCC#CCNC(c3n(C)ncc3C(F)F)=O)CCCCC1NC(=O)C2 83830,CCC(O)C(C)(C)C(=O)NCC1(CNC(=O)C=CC(=O)N(C)C)CCCC1 83831,C(=O)(CC(C(F)(F)F)C1CCOCC1)N1CC(CC(CC)O)C1 83832,n1(CC(=O)NC2C(NC(C(CC)OCC)=O)CCC2)ncn2nccc2c1=O 83833,CCC(CC(F)(F)F)C(=O)NC1(CCNC(=O)COCc2nc[nH]n2)CC1 83834,c1(C(=O)NC2C(F)CCN(C(C3ON=C(C)C3)=O)C2)c(C)ccc2c1CCCN2 83835,c1(C(N2CCC2c2ccccc2)=O)cc2cccc(-c3ccc(CO)s3)c2[nH]1 83836,N1(C(c2ccc(C#C)c(C)c2)=O)CCC2CCC(C1)N2C(=O)Cn1ccnc1C 83837,N=c1nc(Cl)cc(C(=O)NCC(O)CNC(c2nncn2C2CC2)=O)[nH]1 83838,c1(CC(=O)NC2C(CNC(=O)Cc3cccs3)CCCC2)cc2ccccc2[nH]1 83839,N(C(=NCCOC(=O)NCSc1ccccc1)NC1CC1)CC(c1n(C)ncc1)O 83840,c1(C(N2C(C)CC2C(=O)NOC2CCCCC2)=O)ccc(N)cn1 83841,C(=O)(C(O)Cn1cncn1)NC(C)CN(C1CCCCC1)C 83842,c1(C(OCOC)C)cc(F)c(CNCc2cc(C)c(C)s2)cc1Br 83843,c1(C(C)C)cccc(C(N2CCOCC2CNC(C2CC3CC3C2)=O)=O)n1 83844,C(=O)(C#CC1CCOC1)NCC(C(=O)NC(CC#C)CC(F)F)(C)CC 83845,CC1C(C(=O)NCC=CCO)CCN1C(=O)Cc1ccccn1 83846,Cc1cc(=NCC23CC(NC(c4ncc(Cl)cc4Cl)=O)(C2)C(C)O3)c(C#N)c[nH]1 83847,N1(C(c2c(OC)nc(Cl)cc2)=O)CCCc2nc(Br)ccc21 83848,C1(NC(=O)CSCc2ccccc2O)CC12CCN(C(=O)C(O)C(F)(F)F)CC2 83849,C(=O)(C1=CC=CN2CCS(=O)(=O)N=C12)N1C(C2(NC(COCC)=O)CC2)CCC1 83850,N1(C(c2nn(C)cc2Br)C(=O)NCC(=C)C)CC(S(C)(=O)=O)CCC1C 83851,c1(C(=O)NC2C3CC(NC(Cc4cc(C)sc4C)=O)CC32)ccnc(C)c1N 83852,[N-]=[N+]=Nc1cccc(C(=O)NCC2CCCC2NC(=O)CCc2cc(Cl)cs2)c1 83853,c1(C(N(CC(C)NC(c2c(C(C)C)cnn2C)=O)C)=O)cc2ccccc2s1 83854,c1(C(=O)NCc2cc(C(N(C(C)CO)CC)=O)sc2)cc2n(n1)CCC2 83855,CC(C)CC(C)CC(=O)N1CCN(CCOc2cc(O)ccc2OC(F)F)CC1 83856,C1(NC(CN(C(C(CCCOC)C)=O)C)=O)CC1C1CCCCC1 83857,C(N=c1cc(Cl)nc(C2CC2)[nH]1)C1OCCN(C(C2CCC(C)(C)OC2)=O)C1 83858,N1(C(c2c(COC)ncs2)=O)CCC(CNC(c2ncc(Cl)n2C)=O)C(C)C1 83859,C1(CC)CN(C(c2c(Cl)noc2C)=O)CC1NC(=O)Cc1ccccc1 83860,C1(N(C)C(C2CCC3(CC3)C2)=O)CN(C(C2CC2c2cnn(C)c2)=O)CCC1O 83861,Cc1ccccc1C=CC(N1CCC(C)(CNC(C2C3CCCOC23)=O)C1)=O 83862,c1(CNC(C2CCN(C(C=CC(=O)OCC)=O)CC2)=O)cc(F)c(F)cc1F 83863,c1(OC)cccc(C(=O)NCCCC(C)(C)NC(C2CCN(C)C(=O)C2)=O)c1N 83864,C(CCCN=c1[nH]c(Cl)nc2c1SCC2)NC(C(CCCC)O)=O 83865,Cn1nc(C(=O)NC2CC2NC(c2ncsc2C(F)(F)F)=O)ccc1=O 83866,Cc1cc(C)c(C(N2CC=CC(NC(=O)CCCc3ccncc3)C2)=O)c(N)c1 83867,N1(C(C#CCNC(=O)CSc2nc[nH]n2)=O)CCn2ncnc2C1 83868,c1(CNC(C(CNC(CCC=C(C)C)=O)O)=O)cccc(C#N)c1 83869,n1(CC(=O)NCCC2CC=CCC2)cncc1C(=O)O 83870,c1(OCC(=O)NC2CC(NC(C3CC(CF)C3)=O)C2)ccccc1Br 83871,N1(C(c2cc(C)[nH]n2)=O)CC2CC(C1)N(C(C1CCC(C)(C)O1)=O)C2 83872,CCCC(C)(O)CC(=O)NC(C)(CC)CCNC(C1CCCC(O)C1)=O 83873,N1(C(C2CC(C)=C(C)CC2)=O)CC(CNC(=O)C=CC2CCCC2)CC12CCC2 83874,C#CCC(C)(C(=O)NC(C(O)CO)C1CC1)NC(=O)Cc1cc[nH]n1 83875,N1(C(C2(C(=O)NC)CC2)=O)CC(CNC(=O)CSC(C)C)C1 83876,c1(C(N(CC(C)SC)CC)=O)nc(OC)ccc1C.C12CCN(C1)C(=O)C(=O)N2 83877,Cc1cc(NCCC2CCC(NC(C3(C)CCCOC3)=O)C2)ccc1[N+](=O)[O-] 83878,c1(C(N2CCC(SC(F)(F)F)CC2)C(=O)NCCCCCC)cc(C)nnc1C 83879,Cc1ccc(C2CC2C(=O)NCC2(NC(=O)CC(C)C(C)C)CCC2)c(Cl)n1 83880,Cc1c(C(=O)NC2CC2NC(=O)CC2CCCO2)cccc1C#N 83881,N1(C(c2c(F)ccc(C)c2)=O)CCCN(C(c2cc(Cl)cs2)=O)CC1C 83882,Cc1cnc2c(C(N3CC(CNC(=O)CC4=CCOCC4)CC3C)=O)cccn12 83883,C1(CNC(CC2(N(C(C(COC)(C)O)=O)C)CC2)=O)CC(C(N)=O)=NO1 83884,N1(C(CNC(CC)=O)=O)C2CCC(C2)C1CNC(c1c(F)cccc1F)=O 83885,c1(C(=O)NC2CC(NC(c3cc(Cl)c(Cl)cn3)=O)C2)cnc2cc(Cl)ccn12 83886,C12(C(N3CCCC(NC(C=C(CC)C)=O)(CO)C3)=O)CCC(C#N)(CC1)CC2 83887,CC(CC(=O)NC1CS(=O)C1)N(C(=O)CCc1ccn(C)n1)C 83888,c1(NC(C(=O)NC2CCC(CCC(C)C)C2)=O)ccc(Br)cc1O 83889,Cc1ccc(C)c(C(=O)NCCCNC(c2cnc(-c3ccc(F)cc3)s2)=O)n1 83890,O=C(N1CC(NC(C2(O)CC2)=O)CO1)C1CCCCN1C1CC1 83891,C(=O)(C(CCC)C(C)C)NCC1N(C(CCCOCC=C)=O)CCCC1C 83892,C(=O)(CC(C)(C)OC(C)(C)C)NCC1C(CNC(C(N2CCSCC2)C)=O)C1 83893,C1(C(=O)NOCC(C)C)(CCOCC)CCN(C(c2cnn(C)c2)=O)CC1 83894,C(=O)(C(C)(C)C(C)(F)F)N(C(C(N1CCCC(C#C)C1)=O)C)CC 83895,C(=O)(CCCCC(F)F)N1C(CCNC(C2CCN(C)C2=O)=O)CCC1 83896,c1(C(N(CCN(C(C2CC(CC(C)(C)C)C2)=O)CC)CC)=O)ccc(Br)nc1N 83897,C1(C(N2CC(OC)CC(NC(CCC#C)=O)C2)=O)CC(C(C)(C)C)=NO1 83898,c1(C(=O)NCC(CC=C)NC(=O)C(O)CN(C)C)ccc(Cl)cc1C 83899,c1(C(=O)NCC(C)NC(C2CC3CC2C3)=O)ccc(OC(F)F)cc1 83900,N1(C(c2c(C)n(C)nn2)=O)CCN(C(c2ccnn2C)=O)CC1c1cccnc1 83901,CC(C(=O)NC1C2CC1N(C(C1CCCCC1C(F)(F)F)=O)C2)C(C)(C)C 83902,CC1(C)CCCC(CC(N2CC(CCO)(NC(C3CCCOC3)=O)C2)=O)C1 83903,C=CCC(C)(C)CC(=O)N1C(C)C2CC1C2NC(c1cnc(O)n1C)=O 83904,C1(CN(C(=O)C=CC(C)(C)C)C)CCN(C(=O)CSc2nncn2C)CC1 83905,CN1CCN(CCC(=O)NC(C)(C)CN2CCN(C(C3CCOC3)=O)CC2)CC1 83906,c1(C(=O)NCC2C(C)CN(C(c3cccc(Cl)c3)=O)C2)cc2cnn(C)c2s1 83907,CC(CC(=O)NC1CCCC(NC(c2ccn(C)c(=O)c2)=O)C1)CC(F)(F)F 83908,N1(C(CC(C(C)C)O)=O)CCC2(CCCCN(C(c3cn(C)c(=O)cn3)=O)C2)C1 83909,C(C)(CNC(=O)C(C)C(C)(F)F)(CC(C)C)NC(CCNC(C(C)C)=O)=O 83910,c1(C(c2ccccc2)CC)n[nH]c(=NC(=O)N(C)Cc2ccc(C)nc2)s1 83911,c1(CN(C(=O)NCc2cccc(C)c2)C2CC2)ccc([N+](=O)[O-])cc1 83912,C=CCC(CC(=O)NC(C)C(CC)CC)NC(=O)Cc1ccc(C)s1 83913,c1(C(C(=O)NCCOC)N(CC(C(=O)OCC)(F)F)C)sc(C)c(C)c1C 83914,C(=O)(C1CCCc2nncn21)N1CC(CNC(C(CCC(C)C)NC(C)=O)=O)C1 83915,C1(NC(Cc2cc(C)sc2)=O)CN(C(=O)C(C)C2CCC2)CCC12CCOCC2 83916,C1(NC(CCC(=O)NC(C(C)NC(C)=O)(C)C)=O)CC1C1CCCCC1 83917,c1(C(N(C2C3CN(C(c4c(C)ncnc4)=O)CC32)C)=O)ccc2nn[nH]c2c1 83918,CC1(C)CCCCC1=CC(N1CC(CNC(C2C3CCCOC23)=O)C(O)C1)=O 83919,N1(C(CC)CC)CC(C(N2CC(O)(CNc3ncc(C(F)F)cn3)C2)=O)CC1=O 83920,C1(O)(C(=O)NCC2CC(NC(c3cc(OC)nn3C)=O)C2)CC2(CCOCC2)C1 83921,C1(NC(=O)COc2ccsn2)CCN(C(=O)CCC2CCOCC2)CC1O 83922,Cc1noc2cc(C(N3CC(CCNC(=O)CN(C)CCO)C(C)C3)=O)ccc12 83923,CCCC(CC(C)C)C(=O)N1CCOCC(C(=O)N(CC)Cc2occc2C)C1 83924,c1(C(=O)NCc2cccc(CNC(CCCSC)=O)c2)c(C)cc(C)cc1N 83925,CC1CCN(C(c2cnc(Cl)cn2)=O)CCN1C(=O)CC1CCC=CCC1 83926,N1(C(C2N(CC)C(=O)CC2)=O)CCCC2(CCN(C(=O)CN3CCC(C)C3)C2)C1 83927,C(CC(C(C)C)NC(c1nccnc1C(N)=O)=O)NC(C(C)=C(C)C)=O 83928,CC(C)CC(CNC(=O)CC1(C)CC1)NC(c1ccc(C2CC2)o1)=O 83929,c1(OCCCCC)ccc(-c2nc(C(C)OC)nn2-c2ccnn2C)cc1OC 83930,C(C)(CO)(C(=O)N1CCOC(C(=O)Nc2nccs2)C1)NC(=O)OC(C)(C)C 83931,CC(C)(C)[Si](C)(C)OC1CCN(C2CC(c3cccs3)C2)C1 83932,N1(CC(N2CCC(O)(CN(C)C(c3cn(C)nn3)=O)C2)=O)CCCCCC1=O 83933,c1(N(C)Cc2ccc(CC)cc2)[nH]c(=NCC(CC)C(C)(F)F)nc2scnc12 83934,c1(C(=O)NCCN(C(=O)C(C)C2CCOC2)CCOC)cc(C(C)C)no1 83935,C(=O)(C(C)C(C)(C)C)NC(C1CCCN(C(COc2c(C)cccc2)=O)C1)C 83936,N1(C(C(C)OC)=O)CC2CCC(C1)C2C(N1CCCC1c1ccccc1)=O 83937,c1(C(N(CC(CNC(C(c2cccc(C)c2)=O)=O)O)C)=O)cc2sccc2n1C 83938,Cc1cc(C(=O)NCC2C3CCC(C3)N2C(=O)CCc2cnn(C)c2)c(C)cn1 83939,C(=O)(C(C)(C)CC(F)F)NC1(CF)CCN(C(c2cnn(C)c2C(C)(F)F)=O)C1 83940,C(C(N=c1nc(C2CC2)[nH]s1)C1CCC1)NC(C(C)N(c1ccccc1)C)=O 83941,C#CCCN=C(NCC(c1cccc(F)c1)OC)NCC1(OC)CCS(=O)(=O)C1 83942,C1(CNC(Cn2ccc(C)n2)=O)CC2CN(C(=O)C(c3ccc(F)cc3)O)CC12 83943,N1(C(C(CSC)C)=O)Cc2n[nH]cc2C1C(=O)NCC1CCCCCC1 83944,c1(C(N2CC(CNC(C3CCC(CC)C3)=O)C2)=O)cc(CC)c(=O)n(C)c1 83945,c1(C(N(CCCNC(C(CCC)O)=O)CC2CCCC2)=O)c[nH]ccc1=O 83946,c1(CCC(N2CCC(n3cc(C(COC)OC)nn3)C2)=O)cccc(N(C)C)c1 83947,c1(CN2CCC(O)(Cc3ccccc3)C2)noc2c1COCC2 83948,CCC(C)CC(=O)NCC(C1CCC1)NC(CC)C1(Cc2n[nH]cc2C)CC1 83949,N1(C(C2C(=C)C2C(=O)OC)=O)CCN(C(C23CCOC(C)(C2)C3)=O)C(C)C1 83950,c1(C(=O)NCC(CN(C(c2cc(C)no2)=O)C)O)ccc(N)c(C)c1C 83951,O=C(C1=CCCOC1)N1CCN(C(=O)CC2CSC2)C(C2CC2)C1 83952,c1(NC(CC2(C=C)CN(C(=O)C(C)CSC)C2)=O)ccc(F)c(CC)c1 83953,N1(C(c2n[nH]c(C)c2[N+](=O)[O-])=O)CCc2ccc(N=[N+]=[N-])cc2C1 83954,N1(C(c2c(CC)nn[nH]2)=O)CCC(CF)(NC(=O)CCCN(C)C)C1 83955,CC1CN(C(C2(C#N)CCCC2)=O)CCC1N(C(=O)C1=NOCC1)C 83956,N1(C(CCCC)=O)CCN(C(C2CC2c2ccc(Cl)c(F)c2)=O)CC1CC 83957,c1(OC)ccc(C(C)=CC(=O)NC2(CF)CCN(C(C3(F)CCC3)=O)C2)cc1 83958,C(C)(c1ccc(F)cc1)=CC(=O)NCC1CCN(C(C(C(CC)O)C)=O)C12CC2 83959,c1(C(=O)NCC2C(NC(C(c3ccccc3F)OC)=O)C2)cc(C#N)[nH]c1C 83960,N1(C(CCOCCC)=O)CC(NC(=O)Cc2cc(F)c(N)cc2F)CC2(CC2)C1 83961,C1(CCNC(C(CC)C)=O)CN(C(c2cc(Br)cn2C(C)C)=O)CCO1 83962,CC(O)C(C(=O)N1CCC(CCNC(=O)C(c2ccccc2F)O)CC1)N(C)C 83963,C(=O)(CCOCCNC(=O)CCC1CC(C)C1)N(CC)CC1CCC1 83964,N1(C(c2nc(C)oc2C)=O)CC(C)(C)CC1CNC(=O)C=CC1CCCN1C 83965,CC(CC(=O)NCC(C)(C)C(F)F)C(C)(C)NC(=O)CN=[N+]=[N-] 83966,c1(OC)cc(C(N2CC(C)(NC(c3cnns3)=O)C2)=O)c(F)cn1 83967,C(CNC(=O)Cc1ccccc1OC(F)F)(C(C)(C)C)NC(C(C)C#N)=O 83968,N1(Cc2cnn(Cc3ccc(CC)cc3)n2)CCOCC(COCC)C1 83969,N1(C(CC(CC)CC)=O)CCC(C2CC2)(CNC(=O)C(c2cn(C)nc2C)O)C1 83970,C1(NC(c2cc(C)c(C3CC3)cc2)=O)CCCC12CN(C(=O)C(O)C(F)(F)F)C2 83971,Cc1nn2ccccc2c1C(=O)NCC1(CCNC(C2(C)CC=CCC2)=O)CC1 83972,N1(C(COCC)=O)CCC2(CCC2NC(=O)C=Cc2ccc(F)c(F)c2)CC1 83973,N1(C(C=C(CC)C)=O)CCC2(CC1)CCN(C(=O)C(C)(C)CF)C2 83974,c1(C(=O)NC(C2N(C(COCC#C)=O)CCC2)(C)C)ccc2c(c1)CCNC2=O 83975,CC1CC(NC(=O)CNS(N)(=O)=O)CN(C(=O)CCn2ccc(O)nc2=O)C1 83976,C1(NC(CC=CC=C)=O)C2CCCN(C(C3CC4OC3C3CC43)=O)C2C1(C)C 83977,C1(NCc2ccc(OC)c(C(F)(F)F)c2)C2CCCC(F)(F)C12 83978,n1(CCCC(=O)NCC2(C)CC(NC(=O)Cc3n[nH]c(=N)s3)C2)ccccc1=O 83979,c1(C(=O)NC2C(CN(C(c3c(C)ncn3O)=O)C)CCC2)cc([N+](=O)[O-])c[nH]1 83980,C1(C(=O)Nc2ccc(C(C)(C)C#N)cc2)CC2C(C1)C2(F)F 83981,c1(CNC(C(CC)F)=O)cccc(NC(=O)CC(C)CN(S(=O)(=O)CCC)C)c1 83982,c1(-c2cncc(C(=O)NC3CCCC(NC(C)=O)C3)n2)ccc2c(c1)NCCO2 83983,N1(C(C2OCC(C)C2)=O)CCC2(CCN(C(c3ccc4cc[nH]c4n3)=O)C2)C1 83984,c1(C(=O)NC(CC)CN(C(C2CCC(CCO)CC2)=O)CC)cnc(O)c(F)c1 83985,Cc1cc(O)ccc1NC(c1c[nH]nc1CCNC(=O)C(C)(C)N=[N+]=[N-])=O 83986,C1(NC(C2(C)ON=C(C)C2)=O)CC2(CCN(C(c3sc(C)nc3C)=O)C2)C1 83987,N1(C(c2c(C)ccc(OC)c2)=O)CCCCC(CNC(c2cnsc2)=O)CC1 83988,C1(C(N(CCC#C)CC)=O)CCCC(NC(c2ccnc(O)c2)=O)CC1 83989,C1(CC#C)(NC(=O)N)CCCCC1.C12(O)CC(C1)C(=O)NC2.C1(C)CC1(C)C 83990,CCC(CC)C(C)C(=O)NCCC(=O)N(C1CCC1)CCN(C)C 83991,C1(N(C(CN(C)Cc2ccccc2)=O)C(N)=O)CCCN(C(=O)C(N)=O)C1 83992,C12(NC(C3CC(C(=O)OC)C3)=O)CCCC1(F)CN(C(c1coc(C)n1)=O)C2 83993,C(=O)(C(C)CC(F)(F)F)NCC(CCCC)NC(=O)Cn1ccc([N+](=O)[O-])n1 83994,C1(N(C(Cc2cc(C)no2)=O)C)CCCN(C(=O)C2=CCCS2)C1 83995,C=CC1(CC(=O)NC2(CC)CCOC2)CN(C(C2CCN(CC3CC3)C2)=O)C1 83996,N1(C(C=CSC)=O)CCn2nc(C)c(CNC(=O)C(C)C(C)(C)C)c2C1 83997,c1(-c2c(C(N3CC(CNC(=O)CC4COC(=O)C4)C3)=O)cno2)ccccc1F 83998,c1(N(CCCN(C(C(C)OCCCC)=O)C)C)nc(Cl)nc2cc(C)sc12 83999,C12(C(=O)NC(CN(C(C)C)C)C)CC1CN(C(=O)Cn1c(O)nnc1O)C2 84000,Cn1cc(C(=O)NC2CCCC(CC(N3CCCC(CF)C3)=O)C2)n(C)c1=O 84001,c1(CC(N2C(C)(CNC(C=CCCC)=O)CCC2)=O)cccc(F)c1O 84002,C1(NC(=O)CSc2nnc(S)s2)(CO)CCCN(C(c2ccncn2)=O)C1 84003,N1(C(C(C)(C)c2ccno2)=O)CC(NC(c2cc3occc3s2)=O)CC2(CC2)C1 84004,c1(CCC(N2C3CN(C(c4ccc(OCC)nn4)=O)CC32)=O)cc(F)ccc1Br 84005,C1(CCNC(c2ccc(SC)s2)=O)CCCCN1C(=O)C=CC(=O)NC1CC1 84006,C1(NC(=O)NCC(C2CCOCC2)OC)CC(C)(C)C12CC2 84007,c1(C(c2nnnn2CCC)NC2(C)CC(=C)C2)ccc(N(C)CC)nc1OC 84008,N1(C(CC2CCN(C)C2)=O)CCC2(CCN(C(C3CC4CC4C3)=O)CC2)C1 84009,c1(C(N2CCC(C(C)NC(c3cc(C)cc(Cl)n3)=O)C2)=O)ccc(C)c(C#N)c1 84010,n1(CC(=O)NCC(CNC(C(COCC)C)=O)(C)OC)nc(C)n(C)c1=O 84011,N1(C(c2c(C)cc(F)s2)=O)CCC2(C1)CN(C(=O)C(C(C)C)n1cccc1)C2 84012,C1(CN(C(COCCC#C)=O)C)COCCN1C(c1ccc(C(F)F)cn1)=O 84013,C(N=c1[nH]c(N(C)Cc2cc(Br)ccc2F)nc(=N)[nH]1)C1C(C)CCC1 84014,N1(CC)CCC(NC(C2CCCN(C(=O)CCOCC(F)F)C2)=O)CC1C 84015,C1(CC)CCN(C(c2cscc2OC)=O)C1C(=O)NCc1sc(C)nc1C 84016,N1(C(c2c(Cl)ccc(C)c2)=O)CC2CC(C1)N(C(C1CC1F)=O)C2 84017,N1(C(c2cc(C)cc(C)n2)=O)CCC2(CC1)CC2(C)C(=O)NC(CO)C(N)=O 84018,Cc1nc2ccc(C(N3CC4CN(Cc5nccnc5Cl)C4C3)=O)cc2o1 84019,c1(OC)ccc(OC)c(CC(=O)NCC2CCN(C(c3occc3C)=O)CC2)c1 84020,c1(C(N2CC3CCC(C2)N3C(=O)Cc2ccnc(O)c2)=O)cccc2nsnc12 84021,c1(C(N2CCCC(CNC(c3nc(C(C)OC)oc3)=O)C2)=O)ccc(Cl)cc1N 84022,CCCC(C(=O)OC)C(=O)N(CCCNC(=O)C(C(C)C)n1ccnc1)C1CC1 84023,CCCCC(O)CCC(=O)N1CCC(NC(=O)Cc2cc(OC)no2)C(C)C1 84024,C1(C(=O)NCC(c2cccc(C)c2)NC(=O)C(Cl)=CCl)CCn2cncc2C1 84025,C1(C(=O)NC(C#CC#C)(C)C)CC(C)CCN1C(C1CC1C#N)=O 84026,Cc1nc(C)c(C(=O)NC(C)CCCNC(=O)Cc2ccc(Cl)s2)[nH]1 84027,c1(CN(C(=O)CC2(C)CC2(F)Cl)C)ccc(CNC(C2(C)CC2(F)F)=O)cc1 84028,C(=O)(C(C)CC(N)=O)NCC(CCCC)NC(=O)C(=Cc1ccncc1)C 84029,c1(C(=O)NCCN(C(CC2(C(=C)F)CCC2)=O)C(C)C)c(OC)cnnc1OC 84030,CC(CC(=O)N1CCCCC1c1ncccc1C(=O)O)CC(=O)c1ccc(Br)cc1 84031,N1(C(c2cc(C3CC3)no2)=O)CCC2(CCCN2C(=O)C2=CCCO2)C1 84032,CC1C(NC(c2nnc(O)nc2O)=O)C(C)CCN1C(=O)C=CC1CCCC1 84033,c1(OCC)ccc(NC(c2sc(Br)c(C)c2C)c2nnnn2C(C)CC)cc1Br 84034,c1(C(N2C(C)(COC)CC(NC(=O)C(OC)OC)C2)=O)n[nH]c2cc(Cl)ccc12 84035,CC1CC(CO)CN(C(=O)CCCCCNC(C2CCC(N(C)C)C2)=O)C1 84036,Cn1cc2c(n1)CCC(C(=O)NCCC1(NC(c3ccc(Cl)c(O)c3)=O)CC1)C2 84037,C=C(CCN(C(C)C)Cc1ccccc1CS(C)(=O)=O)C(=O)OC 84038,C1(C(N2CCCC2CNC(=O)CCCOC2CCOCC2)=O)(OCC)CCCC1 84039,N1(C(c2nn(C)c(Cl)c2)=O)CCC(c2ccccc2)(NC(=O)C2=CCCS2)CC1 84040,C(=O)(CCCCCNC(C(C1CCN(CCOC)CC1)N(C)C1CC1)=O)OCC 84041,N1(C(C2C(=C)CC2)=O)CCOC(CN(C(=O)CN2C(=O)CCC2=O)C)C1 84042,C1(C(N2CC3CC3(CO)C2)=O)(NC(CN(CCOC)C)=O)CCN(C)C1 84043,c1(C(N(CCN(C)C)CC2C3COCC23)=O)sccc1F 84044,c1(CNC(N2CCCN(C(C(C)(C)OCC)=O)CC2)=O)c(F)ccc(F)c1OC 84045,c1(C2(C(N(CCC(C)NC(=O)CC3(CO)CC3)C)=O)CC2)ccc(F)c(F)c1 84046,Cc1cccc(C(c2ccccc2)NC(=O)C(F)(F)c2ccncc2)c1 84047,c1(C(C)=O)c(CCC(=O)NCCCCNC(c2nc[nH]n2)=O)c[nH]c1C 84048,C(=O)(C(C)(C)CCC#N)NCCC1CN(C(Cc2ccc(C#C)cc2)=O)CC1C 84049,CN1CCCC(CCC(=O)N2CC(CCNC(=O)CC3(N(C)C)CCCC3)C2)C1 84050,C12(CCN(C)C1)C(=O)N2.C1(CNC(C2CC(C)(CC)C2)=O)CC(=O)N(C)C1 84051,N1(S(CC)(=O)=O)CCCC(C(=O)N(CCC(C)NC(=O)CS(N)(=O)=O)C)C1 84052,CCC(C)(C(=O)NCC1(O)CC(CNC(=O)CCOC)C1)C(N)=O 84053,c1(C(N2C3CC(CNC(CC(C)(C)C4CC4)=O)C(C3)C2)=O)cc2c[nH]cnc-2n1 84054,C(=O)(CC1CCCc2oc(C)nc21)NCC1(OC)CN(C(COCC=C)=O)C1 84055,C1(CNC(C=CCC)=O)(CNC(=O)C=CC(CC)=CC)CC2CCCC2C1 84056,C1(NC(CCNC(C)=O)=O)CCN(C(=O)CC2=CCCCC2)CC12CCC2 84057,c1(CNC(C(C2CCN(C(CC(C)(C)OC)=O)C2)F)=O)cc(F)ccc1C 84058,c1(NC23C(CN(C(C4CCC(C)CC4)=O)C2)CCC3)nc(Cl)nc2cnn(C)c12 84059,C1(C(N2CCCC(CCNC(CNC(C)=O)=O)C2)=O)CC(c2ccccn2)=NO1 84060,C(=O)(CCCS(C)(=O)=O)NC(CNC(C=CC(c1ccc(C)cc1)=O)=O)(C)C 84061,C1(NC(C(C(C)C)OCC(C)C)=O)CCCCCN(C(c2nnc(C)s2)=O)C1 84062,c1(C(=O)NCC2(F)CC(CNC(c3cnc(SC)s3)=O)C2)cn(C)nc1C(C)C 84063,Cc1ccc(C(=O)NC(CCN(C(=O)CC2(CO)CC2)C)C(C)(C)C)c(C)n1 84064,c1(-c2c(C)onc2)ccc2c(C(N3CCNC(=O)C3C)=O)cnn2c1 84065,C1(CC(=O)NCc2ns[nH]c2=O)COCCN1C(C1CCOC1=O)=O 84066,C#Cc1cc(C(=O)N(C(C)CC(=O)NC(C#C)CCC)C)ccc1C 84067,C1(C)(CNC(CC(C=C)C)=O)CN(C(C2CC(S(C)(=O)=O)C2)=O)CCO1 84068,c1(C(=O)NCC(C)N(C(C2C(C(F)F)C2(C)C)=O)CC)cccc2[nH]nc(O)c12 84069,C1(OC)CN(C)C(C)(C(N2CC(CO)(NC(=O)CC(C)(F)F)C2)=O)C1 84070,C1(CC(=O)N(CC(CC)NC(=O)CCn2ccnn2)CC)CCCOCC1 84071,Cc1cc(O)c(C(=O)NC2(CO)CCCN(C(c3c[nH]c(Br)c3)=O)C2)nn1 84072,c1(OC)ccc(C(C)CNC(c2ccnc(-n3ccnc3)c2)=O)cc1OC 84073,C#Cc1cccc(OCC(=O)NCC2CCN2C(=O)CCC(=O)OC)c1 84074,N1(C(COC(CC)C)=O)CCC2(CNC(c3ccnc(F)c3)=O)CCCCC12 84075,C(CCN=c1ccn2c(Br)cnc2[nH]1)N(C(C(C=CC)O)=O)c1ccccc1 84076,C1(NC(c2ccc(CC)s2)=O)CCC(F)(CNC(c2cccn2C2CC2)=O)C1 84077,C12(C(N3CC(C#N)(COC)C3)=O)CCC(CN(C(C3C=CCC3)=O)C1)C2 84078,CC(O)(CC(O)CNC(C1(O)CCS(=O)(=O)CC1)=O)C(F)F 84079,c1(C(N(C2CCCN(C(c3cc(Cl)cnn3)=O)C2)CC)=O)nccc2[nH]ccc12 84080,C1(C(=O)NCCC=C=C)CCC(O)CN1C(c1c[nH]nc1C)=O 84081,c1(OC)ccc2c(C(=O)NC3CCCN(C(=O)C(C)CC4CC4)CC3)c[nH]c2c1 84082,C1(C(N(CCN(C(C(CCCC)CC)=O)C)C)=O)CCC(F)(F)CC1(C)C 84083,c1(C(N2CC(C)C(NC(=O)CC3CC=CCC3)C2)=O)cc(F)cc2cnccc12 84084,c1(NC(C)=O)cc(-c2ccnc(CC(N3CCC(C#N)C3)=O)c2)ccn1 84085,C1(CN(C(C(n2cc(-c3ccc(OC)nc3)nn2)C)=O)C)CC(C)CC(C)C1 84086,N1(C(c2n(CC)ncc2Cl)=O)CC(CNC(=O)C(C)C2CC2)CC(C)(C)C1 84087,C12(NC(C3CC3(F)F)=O)CCCCC1CN(C(c1ccc(Br)c(F)c1)=O)C2 84088,C=CCCC(C(=O)NC1CC12CCOCC2)NC(C1CN(C(C)C)C1)=O.O 84089,CCCCC(C)(F)C(=O)N1CCC2C(C1)CN2C(c1ccc(OC(C)C)nc1)=O 84090,N1(C(C2(NC(C(C)(C)OC(C)=O)=O)CC2)=O)CC(S(C)(=N)=O)C1 84091,N1(C(C(C)OC2COC2)=O)CCC(NC(c2cnn[nH]2)=O)C(C(N)=O)C1 84092,C1(CCN)(OC)CCCN(C(C2(C3(c4ccccc4)NC(=O)NC3=O)CC2)=O)C1 84093,c1(C(=O)NCC2C(NC(=O)COCC(F)(F)F)C2)n[nH]c(C2CC2)c1Br 84094,c1(C(=O)NC2C(NC(CSCCC(C)C)=O)CC2)n[nH]cc1-c1ccncc1 84095,N1(C(C2CCCC(=O)N2)=O)CCN2CCN(C(=O)C(O)C3CCC3)CC2C1 84096,N1(C(c2ccc(P(C)(C)=O)cc2)=O)CCC2CN(C(=O)COC(F)F)CCC2C1 84097,N1(C(C2C(NC(C3C(C(=O)OC)C=C3)=O)CCO2)=O)CCN(C)CC1C 84098,N(C(=NCCCC(=O)N1CCCC1)NCC12CCCC1CCO2)CC(C)C 84099,c1(C(=O)NC(CNC(c2ccc(=N)[nH]c2)=O)C2CC2)ccc2cnnn2c1 84100,C(=O)(CC(C)NC(=O)CC1CC=CCC1)NCCOCCOCC 84101,Cc1nn(Cc2nc(C3CC3)nn2-c2ccc(C(=O)O)nc2)c2ncccc12 84102,N1(c2nc(C3(NC(=O)CCc4cn(CCO)nn4)CC3)on2)CCCCCC1 84103,c1(CC(C(=O)NC2CC(N(C(=O)CCF)C)C2)OC)ccc(C)cc1 84104,Cc1cc(NC(C2(NC(=O)CN(C)C)CCCCC2)=O)ccc1O 84105,C1(CC)(CC)CN(C(C23CCC(OC)(CC2)CC3)=O)CC(C)O1 84106,C(C(=O)N1CC(NC(c2cc(O)n(C)n2)=O)CC1(C)C)(C(C)(C)C)NC(C)=O 84107,C(C)(C)(CCCC(=O)N1CCC1C1CCCC1)NC(C1CCN(C)C(=O)C1)=O 84108,N1(Cc2c(F)ccc(N)c2)CC2(CCCCN2CCC2CCCCCO2)C1 84109,CCC(CC)CCC(=O)N(C)CCN(C(C)C(=O)Nc1ccc(F)cc1OC)C 84110,Cc1ccc(C(=O)NC2CCC(NCc3cc(C(=O)O)ccc3F)C2)cc1Cl 84111,N1(C(=O)Nc2n(C)ncc2N=S(C)(C)=O)CCC2(CC1)CCS(=O)(=O)CC2 84112,N1(C(c2c(C)c[nH]c2)=O)CCc2cc(C(=O)NCC(N)=O)cnc2C1 84113,C1(CC)(CC)CC(NC(c2cc(O)nc(C)n2)=O)CN1C(=O)C(C)N1CCCC1 84114,N1(C(C#CC2(C)CC2)=O)CCC2CCN(C(=O)C3=CCOC3)C2C1 84115,N1(C(C)C)CCCC(CCNC(C2CCCCN2C(=O)COC(C)(C)C)=O)C1 84116,C=CCC(CC=C)C(=O)NCC(C(C)C(C)C)NC(c1ccc(CO)s1)=O 84117,CC(CC(=O)N1CCCN(CCNC(C23COCC(C2)C3)=O)CC1)CC(C)(C)C 84118,C=CC(C)(C)CC(=O)NCCCN(C(C1CC(O)CN1c1ccncn1)=O)CC 84119,C(=O)(CCCN(C)N=O)NCCC1OCCN(C(CC2C(C)CCCC2)=O)C1 84120,c1(C(N2C3CN(C(C4N(CC)CCCC4)=O)C(C3)C2)=O)oc2ccccc2c1C 84121,C1(C(N(C2(C(=O)NCc3nccc(C)c3)CC2)C)=O)C2CCC(C2)C1C 84122,C(C)(CNC(C1(c2ccn(C)n2)CC1)=O)(C(C)C)NC(c1c(CC)ccs1)=O 84123,N1(C(=O)CC2CSCCO2)CCC2CC2(C(=O)N2OC3CCC2C3)CC1 84124,CC1=CCC=CC1C(N1CC2C(NC(=O)CC(C)O)C2C1)=O 84125,S(=O)(=O)(C1(CNC(N2CCC(Cc3cccc(Cl)c3)C2)=O)CC1)N(C)C 84126,N1(C(C(C)n2cccn2)=O)CCC(CNC(C2C3CCC23)=O)CC1 84127,N1(C(CCn2ncc(C)c2)=O)CCCC2(CC(NC(=O)CCC(C)N(C)C)C2)C1 84128,N1(c2nc(OC)c(F)c(C)n2)CCCC2(CCN(C(=O)C(C)(C)SC)C2)C1 84129,C1(C(NOCCCCCC)=O)CCCN(C(=O)Cc2cnccc2C)C1 84130,N1(C(C(CC)OCC)=O)CCN(C(c2cnc(O)nc2O)=O)CCC1C 84131,C(=O)(C(C)(C)C(N)=O)N(CCC(C)NC(c1cnn(C(C)C)n1)=O)C 84132,N1(C(c2c(C)cc(C)s2)=O)CCC(F)(CNC(=O)C(S(C)(=O)=O)C2CC2)CC1 84133,n1(C(C)(C)C)cnc(C(N(C2CCC(NC(=O)C(=O)N(C)C)C2)CCN)=O)c1 84134,C=CCC(CC(C)C)C(=O)N1CC(C(N2CCOCC2C=C)=O)C(C(C)C)C1 84135,c1(OC)ccc(CN2CCCC(NC(c3cccnc3OC)=O)C2)cc1F 84136,N1(C(C(=O)NCC2CC(C)OCC2)=O)CCc2ccccc2C(F)(F)C1 84137,CN1CC(CCNC(=O)N(CC2CCCC2)CC2CCCO2)CC1=O 84138,c1(C(N(CCNC(C2CC3CCC3C2)=O)CC2CC2)=O)cc(F)cc2nc[nH]c12 84139,c1(C(N2C(CNC(CCC=CCC=C)=O)COCC2)=O)cc(F)cc(C)c1N 84140,Cc1cc(C(C)NC(C2CCN(C(c3ccnnc3)=O)C2)=O)on1 84141,CCCC(CNC(c1ncn2c1CCC2)=O)C(=O)NC1CC2(CC(OC)C2)C1 84142,C(=O)(CCC(C)(C)[N+](=O)[O-])N(C(C)C(=O)NCCc1ccns1)C1CC1 84143,C(=O)(CCCCC(=O)N1CCC1CNC(=O)C(O)C(F)(F)c1ccccc1)OC 84144,CN1CCC(=CC(N2CC3C(CNC(=O)CCC4(C)CC4)C3C2)=O)CC1 84145,Cc1csc2ncc(C(=O)NC3CN(C(=O)CSCC(N)=O)CCC3C)n12 84146,c1(CC)ccc(C(C(=O)NC2CC2)NC(=O)CN(CCOC)C2CC2)nc1 84147,C(CC(O)C(=O)NCCC(C(=O)NC(C)C)OC(CO)C(=O)N(C)C)SC 84148,c1(CCC(=O)NC(C2(O)CN(C(C3(CC=C)CC3)=O)C2)C)ccc(Cl)cc1 84149,C(=O)(CC(C)C(C)(C)NC(=O)C1=CCCOC1)Nc1ccc(CC)cc1C 84150,C(CN=C(NC(C)C)N1CCC(O)(c2ccc(F)cc2)C1)=CCC 84151,N1(C(C2CC2CF)=O)CC2CCC(C1)N2C(c1cc(-c2ccccn2)[nH]n1)=O 84152,c1(C(N2CCCC2c2cccc(Cl)c2)=O)cc(Cl)c(F)cc1[N+](=O)[O-] 84153,c1(CC(=O)NC2CCN(C(c3c(C)ncnc3)=O)C2)cnn2c1OCCC2 84154,N1(C(C2CCCC(CC)C2)=O)CC2=C(C1)CN(C(c1cc(F)cc(Cl)c1)=O)C2 84155,c1(OC(C(=O)NCCN(C(=O)C(O)C(C)C)CCC)C)cccc(C(C)=O)c1 84156,CC(C(F)(F)C(F)(F)F)C(N1CCCN(C(=O)OC(C)(C)C)CC1C(=O)O)=O 84157,C(=O)(C(Cc1ccco1)NC(=O)CCC1CCCOC1)N(CC=C)C 84158,N1(C(CN(C(CCOC)=O)C)=O)CCN(C(=O)CCCCCSC)CC1CCO 84159,c1(CC)cc(C(=O)N(C2CCN(C(=O)Cc3cn(C)nc3C)CC2)C)c(C)o1 84160,c1(C(=O)NCC2CC(NC(c3ccnc(O)c3)=O)CC2O)cccc2c1CCC2 84161,C(CC(CNC(C1(C)CC(F)C1)=O)NC(=O)COCCF)OC 84162,c1(CC(N2CC3CC(CNC(C4(C)CC4)=O)C3C2)=O)ccc2ncsc2c1 84163,N1(C(=O)CN2CCN(CCF)CC2)CCC2OCCN(C(=O)C(=O)NC3CC3)C2C1 84164,C1(CC(=O)N(C2CCN(C(=O)C(C)CC3CC3)C2)CC#C)CSCCO1 84165,C12(CNC(C(C)c3ccsc3)=O)CCCC(CN1C(=O)C=Cc1cncs1)C2 84166,C1(C(=O)NC2CN(C(c3cc(SC)oc3C)=O)CC2C)(OC)CCOCC1 84167,S(=O)(=O)(C1CC1(F)F)NC(C1C2(C)CNC1C2)=O 84168,c1(CNC(C2CCN2C(c2cnc[nH]2)=O)=O)ccc(N)cc1.c1(S)ccccc1O 84169,c1(C(=O)NCC(CNC(C(C)OCC=C)=O)CO)cc(F)ccc1NS(C)(=O)=O 84170,C1(CNC(N(C2CCCN(C)C2)C)=O)CCCN2CCCCC12 84171,CC(C)CCCCC(=O)NC1(C)CC(NC(c2cnn(-c3ccccn3)c2)=O)C1 84172,c1(CN(C(C)C(=O)NCCC(C(=O)OC)OC)CCC)c(C(=O)O)nnn1C 84173,C(=O)(CC(CC(C)C)NC(C1CCOC1)=O)N1CC(c2onc(C)n2)C1 84174,C1(C(N(CC(C)O)CC(F)F)=O)CCCCC1CNC(C1CCCC(=O)N1)=O 84175,N1(C(CN2CCN(C(C(C)n3ccnn3)=O)CC2)=O)CC2CCCCC2C1C 84176,C(C)(CNC(c1c[nH]nc1C(F)F)=O)(C(C)C)NC(C(CO)OC)=O 84177,C1(N(C)C)CCC(C(=O)NC2C3CC2N(C(C2(C)CC=CC2)=O)C3)CC1 84178,c1(C(N2C3CCC2COC3)C(=O)NC)cnc2ccc(F)cc2c1 84179,N(C(=NCCF)N(C)Cc1ccccc1Br)C1CN(C(C)C)C(=O)C1 84180,C1(n2cc(C(C)(C)F)nn2)CCCCC1C(=O)NC1CC(c2ccccc2Cl)C1 84181,c1(OC)c(C(=O)NC2CCC(CNC(C3(C)CCOC(C)C3)=O)C2)c(C)nn1C 84182,C1(O)(C(N2CCN(CCN(C)C)CC2)=O)COC(C)(C)C1 84183,CCC(COC)(CC)C(=O)N1CCC(C(=O)N(C2CCOC2)C)O1 84184,N1(C(c2c[nH]c(=NC)s2)=O)CCC2(CC1)CC2C(N1CCCOCC1)=O 84185,c1(C(=O)NC2(CNC(=O)C(O)C3CCC3)CCOC2)cc2ccccc2cn1 84186,Cc1c(C(N2CCC(C(C)NC(c3cnc(N(C)C)nc3)=O)CC2)=O)nnn1C 84187,C1(COC)(NC(=O)CN)CCN(C(=O)CCC2(C)N=N2)C1.n1(C2CCC2)cccn1 84188,C1(C(=O)NCC(CNC(c2cc(C)ns2)=O)CO)CCC(=O)NC1 84189,C(=O)(C(C)(C)C(N)=O)N(C)CCNC(c1cnc(Cl)n1C)=O 84190,N1(c2nnc(CCC)s2)CC2C3CCC(C2C1)N(C(C1(CC2CC2)CC1)=O)C3 84191,CC(=O)CC(C)(C)C(=O)NCC1CC(C(=O)NCC(C)CC2CCC2)C1 84192,C1(C(N(CCCC=C)CC)=O)CCC(C2CC2)N1C(=O)C=Cc1cc[nH]n1 84193,c1(C(=O)NCC2(F)CN(C(C3C(CCC)CCC3)=O)C2)ccncc1F 84194,c1(C(=O)NCC2(NC(=O)C(C3CCOCC3)F)CCCC2)cnc2n1CCCC2 84195,C1(C(N2CC(C3(NC(C4C(C)OCC4)=O)CC3)C2)=O)CCC2(CCC2)OC1 84196,c1(C(N2CC=CC(NC(CC3COCC(C)O3)=O)C2)=O)cccc(F)c1F 84197,C(CCCCNC(=O)CCCF)NC(C(C)c1cccs1)=O 84198,C1(C(=O)NCC2(CCC)CC2)CCCCN(C(=O)C(C)(CO)OC)C1 84199,C(=O)(C1=CCOCC1)NC(C1(O)CCN(C(=O)CC2SC(=N)NC2=O)C1)C 84200,n1(C2C(C(N3CC(N4CCOC4=O)C3)=O)C2)cc(-c2cccs2)nn1 84201,c1(CC)ocnc1C(=O)NCC1(O)CC(NC(=O)CCOCCOC)C1 84202,Cc1ccc(C(N2CCCOC(CNC(=O)C(C)NC=O)C2)=O)c2c1CCC2 84203,N1(C(C)CN2CCC(c3noc(C(F)F)n3)CC2)CCN(C)CC1 84204,c1(NC(C(C(C)C)SC)=O)ccc(NC(=O)C(C2CCC2)N(C)C)cc1C 84205,C(=O)(C(C(C)(C)C)C1CCCCC1)N(C)CCNC(c1cn(C)[nH]c1=N)=O 84206,CC1CN(C(C2(c3ccccc3F)CC2)=O)CCN1C(c1ccc(O)nc1Cl)=O 84207,CCCC(C)C(=O)NC1CCCN(C(C2(C#N)CCC2)=O)C1 84208,Cc1cc(F)c(CNC2(CC(=O)Nc3csc(C)c3C)CCC2)cc1Br 84209,CCC(CNC(=O)C(c1cncnc1)C)(CC)C(=O)NCC(O)C1(Cl)CC1 84210,Cc1scc(C(=O)NC(C2(O)CCN(C(=O)CC3CCOCC3)C2)C)c1C 84211,CC1(C)COC(CCC(=O)NCCN(C(=O)CCOCC(F)F)C2CC2)C1 84212,c1(C(N2C3CC(NC(=O)C=Cc4cscn4)C3CC2)=O)cc(F)cc2nc[nH]c12 84213,Cc1cc2[nH]c(C(=O)NCC3(F)CCN(C(C4(CC5CCC5)CC4)=O)C3)cc2o1 84214,C(CC(C(=O)N(C)Cc1nnnn1C)NC(C1CC(OC)C1)=O)OC 84215,C12(CC(=O)NCC(COC)NC(=O)Cc3cnnn3C)CCCC1C2 84216,N#Cc1ccc(CC(=O)NCCOC2CCN(c3ncc(F)cn3)C2)cc1 84217,CC(O)C(C)(C)CNC(=O)C(F)CC1CN(C(c2cnsc2)=O)C1 84218,Cc1cc(C(=O)NCC2(F)CN(C(=O)CCCCC(C)(C)C)C2)cc2c1CCC2 84219,C1(CC(=O)NCC(C)N(C)C)CCCCN1C(C1CCCCO1)=O 84220,C1(NC(C=C(CC)C)=O)C2CC3CN(C(c4ccc(F)c(Br)c4)=O)C1C3C2 84221,c1(C(=O)NC(C2CCCCC2)CNC(C2CCC(O)C2)=O)cn2ncccc2n1 84222,C(CC1CC1)(CC1CC1)NC(CC)C 84223,C1(C)(CNC(CC(C)C)=O)CN(Cc2cccc(CO)c2)CCO1 84224,c1(C(CC)C(=O)N(C)CCN(C)C(C2CNC(=O)C2)=O)cccc(Cl)c1 84225,c1(C(=O)NCC2N(C(CNC(CSC)=O)=O)CCC2)cc(C(C)C)ccn1 84226,CCC(CC1CCCC1)C(=O)NCC(C)NC(C1CC(C)(F)C1)=O 84227,C(=O)(C1=CC(C)(C)C1)NCC(CNC(c1ccc(N2N=CCC2=O)cc1)C)(C)O 84228,c1(C(N2CC(CNC(C(C=C)OC)=O)C(OCC)C2)=O)cccc2ccoc12 84229,C1(C(=O)NCc2ncccc2C)(CC)CCCN(C(c2cnn(C3CC3)c2)=O)C1 84230,N1(C2N(c3scc(OC)c3O)C=C(c3csc(C)c3C)N=N2)CCC(F)(F)C(C)C1 84231,c1(N(CCNC(c2ccc3ocnc3c2)=O)CC)nc(O)c2c[nH]nc2n1 84232,c1(CC(=O)N(CC(O)CN(C)C(c2ccc(F)s2)=O)C)cnccc1C(F)(F)F 84233,CN1C(=O)CCC1CC(=O)NC1CC2C(NC(C3CCCC(=O)C3)=O)C2C1 84234,C1(CNC(C(CC)Sc2cccs2)=O)CC2(CC(NC(=O)Cn3cnnn3)C2)C1 84235,C1(NC(CCN(C)C)=O)CCC2(C1)CN(C(c1cc3cn[nH]c3cn1)=O)C2 84236,N1(C(CC=CC=C)=O)CC2CCC2(CCNC(=O)CCc2csc(=N)[nH]2)C1 84237,N1(C(=O)CC2CC2)CCC2(CCCN(C(c3cccnn3)=O)C2)C1 84238,CC1CCC(C)(CNC(c2c(CNC(=O)C(F)(F)C3CC3)nnn2C)=O)CC1 84239,C1(C(NOCC#C)=O)C2CN(C(=O)C(CO)OC)CC12 84240,N1(C(Cc2ccc(OCC)cc2)=O)CCN(C(=O)CNC2CCSC2)CC1CO 84241,c1(CC(=O)NC2CCC(C(=O)NC(C(C)C)CO)C2)cccc(OC(F)(F)F)c1 84242,C(=O)(CCCCCNC(=O)CC1CCOC1(C)C)NC(CC(=O)OC)(C)C 84243,C1(C(N2CCC(O)(CN(C(C(CC)SC)=O)C)CC2)=O)CCc2cnc(C)n2C1 84244,C(=O)(CC(CC)C(F)F)N(C1CC(C(N2C(CCC)C=CC2)=O)C1)CC 84245,C(=O)(CCCCC(C)(C)C)N1C2CC(C(=O)NC(c3ccn(C)n3)C)(OC2)C1 84246,C(=O)(CCCCCCBr)N1CCC(C(C(=O)OC)c2cccs2)CC1 84247,C(CC(C)CCNC(c1c(Br)n[nH]c1C)=O)NC(C(C)=C(C)C)=O 84248,C=CCC(C)(C(=O)NC1CCN(C(C2CCN(OC)CC2)=O)CC1CC)N(C)C 84249,c1(C(N2C(C(N3C(C)CCCC3)=O)C3CCC2C3)=O)ccc(S(N)(=O)=O)cc1 84250,c1(C(N2CC(OCCNC(C(Br)=C(C)C)=O)C2)=O)nc(C)oc1C 84251,C1(NC(c2c(CC)non2)=O)CCCC(N(C(=O)CCc2ccccc2C)C)C1 84252,c1(OC)ccccc1.C1(NC(CS)=O)CCCC1NC(=O)CN1CC(C)(OC)C1 84253,c1(C(N2C(CO)CC(NC(C(C=C)O)=O)C2)=O)ccc2c(c1C)CCC2 84254,c1(C(N2CC3(C(C(=O)Nc4onc(C)c4C#N)C3)C2)=O)cccc([N+](=O)[O-])c1I 84255,Cc1cc(C)nc(C(=O)NCC2(C(C)(C)O)CN(C(C3C(C)(C)C3(F)F)=O)C2)n1 84256,c1(C(=O)NCC(Cn2cc(-c3n(CC)ncc3)nn2)OC)ccc(F)cn1 84257,C1(CNC(C(CC)(C)CC)=O)CC12CCN(C(=O)CS(=O)(=O)N(C)C)CC2 84258,Cc1cc(Cl)cc(C(N2CCCC(NC(c3c[nH]nc3C)=O)CC2)=O)c1C 84259,CC(C)C(CNC(c1nnnn1C(C)(C)C)c1ccnn1CC1CC1)C(C)C 84260,C1(C(C)(C)NC(C(N2CCC(OCC)CC2)=O)=O)CCc2ccccc2O1 84261,N1(C(=O)Cc2nc[nH]n2)CCC(C2(O)CCN(C(=O)C(O)C3CCC3)CC2)CC1 84262,N1(C(CC=CC)=O)CCCC1CN(C)C(c1cscc1CC)=O 84263,Cc1ncc(C#N)cc1NC(=O)C(CCC1CCC1)NC(=O)CC1CCOC1 84264,CC1C(=O)CCC1CC(=O)OCC1(c2cccs2)COC1 84265,C12(C(=O)NCCCC)C(NC(=O)CC3(O)CCOC3)C3CC1C2C3 84266,N1(CCC)C(=O)CCC1C(=O)NC1(C)CCN(C(C2CCN(C)C2)=O)C1 84267,N1(C(=O)Cn2cnnc2O)CCN(C(c2n[nH]cc2[N+](=O)[O-])=O)CC1CCO 84268,c1(C(=O)NCCC2(CNC(COC(C)=O)=O)CC2)ccc2nnn(O)c2c1 84269,CS(=O)(=O)CC(=O)N1CCCC1CCCNC(c1cncn1C1CC1)=O 84270,CCC(O)C(F)(F)C(=O)NC1CCN(C(c2cscc2C(F)F)=O)C1 84271,c1(C(=O)NCC(CNC(c2ccc(C3C(C)C3)o2)=O)F)cc(Cl)nnc1O 84272,c1(C(=O)NC2C(NC(=O)Cc3cc[nH]c3)CCCC2)cnc(O)c2ccccc12 84273,C(=O)(C1=CC2CCCCCC12)NCC1(O)CC2N(C(CC(=O)OCC)=O)C(CC2)C1 84274,c1(SC)nc(C(F)F)cc(=NC2CCCCN(C(C3CCCN3C(C)=O)=O)C2)[nH]1 84275,C12CCC(=O)N(C1)C2.C1(COC(C(N)=O)=O)CCCN1C(c1ccccc1)=O 84276,c1(C(CC)NC(N2CCCC2c2ccc(C)s2)=O)c(OC)cccc1F 84277,Cc1ccc(-c2c[nH]cc2C(=O)NCC2CC2NC(C2CC(N(C)C)C2)=O)s1 84278,C1(C(N(C)CC2CCCN2C(=O)CC(O)c2ccccc2)=O)CC2OC1C1CC21 84279,C1(C(=O)NCCN(C(c2ccc(F)cc2O)=O)CC)COC2(CCC2)C1 84280,c1(NC)cnncc1C(=O)N(C)CC=CC(=O)NCC(C)(C)C1(O)CCC1 84281,c1(C(C)NC(C2(NC(=O)C=Cc3ccc[nH]3)CC2(C)C)=O)cc(F)cc(F)c1 84282,CCC(C)CC(C(=O)N1CCC12CC(O)C2)NC(C1CCC(O)CN1C)=O 84283,CN1CCC(NC(=O)CCN(C(c2ncc(F)cc2F)=O)C2CC2)C(C#N)C1 84284,c1(CC)nc(C(C(=O)NC(c2ccccc2)C)N(c2ccccc2)CC)n[nH]1 84285,c1(CN(C2CCS(=O)(=O)C2)C(C2C(c3cn(C)nc3)OCC2)=O)ccccc1Br 84286,N1(c2c(OC)cncn2)CCCC(C)(C(=O)NC(c2cccs2)C)C1 84287,c1(C(=O)NCCN(C(=O)CC2OCCCC2(C)C)CC)cc2occc2s1 84288,Cc1cc(C(=O)NC2CN(C(c3csc(C)c3)=O)CCC2CO)nc(C)c1 84289,CCCCCS(=O)(=O)CC(=O)N1CC2CCN(C(=O)Cc3ccccc3)CC2C1 84290,Cc1cc(=NCCCCNC(=O)C(c2ccccc2C)C)[nH]c(Cl)n1 84291,c1(C(=O)NC2CN(C(c3c(C)cc(C)o3)=O)CC2C)ccc2c(c1)NCCC2 84292,N1(C(CCS(CC)=O)=O)CCOC2(CCCCC2NC(=O)CCC2CCCC2)C1 84293,c1(SCCC)cccc(NC(=O)NC2CCCC2C(F)(F)F)c1 84294,C1(NC(Cc2cc(C)on2)=O)C2CCC1N(C(=O)COCc1nccn1C)C2 84295,c1(C(=O)NC2CCC(NC(C(C)CS(C)(=O)=O)=O)CC2)cc2ccnc(Cl)c2[nH]1 84296,C(=O)(C(C(C)(C)C)OC)N1CC(NC(CC(CC)SC)=O)(CO)C1 84297,N1(C(C(C)SCCCC)=O)CC(NC(c2ccc(OC(F)(F)F)cc2)=O)C(C)C1 84298,CC(CC(=O)NCC1CC1C(=O)NC(C)(C)C(C)(C)C)CC(C)(C)C 84299,c1(CC)cccc(CC(N2CC(NC(C3(CO)CC3(F)F)=O)CC2CO)=O)c1 84300,N1(c2nnc(Cc3cccc(C)c3)n2CC(C)C(F)(F)F)CC(C)C(O)C(C)C1 84301,Cn1cnc(C=CC(=O)NC2CCCC2NC(C2(N(C)C)CCC2)=O)c1 84302,C(=O)(CCC(=O)NN(C)C)NC(CSCC)C(=O)NCCn1ccnc1C 84303,C(C1=CCN(C(=O)COC)CC1)NC(CNS(CC)(=O)=O)=O 84304,CC1CCCCC1(CNC(=O)CC1CCC(=O)NC1)NC(=O)CCn1cncn1 84305,c1(CC(N2CC(CNC(CCCOC(C)=O)=O)C2)=O)ccc2c[nH]nc2c1 84306,C(C)(CO)(C(=O)N1CCC(OC2CC2)CC1)NC(C1C(C)C1C)=O 84307,C(=O)(C(C)(C)C(C)C)NC(CC)CN(C(=O)CSc1nc[nH]n1)C 84308,CCC(F)(F)CC(=O)NC1CC=CCC1C(=O)N(C1CC(C)CC(C)C1)C 84309,N1(C(C=CC=CC)=O)CCCC2C1CCCCN2C(c1cncn(C)c1=O)=O 84310,c1(CC)ccc(C(=O)NCC2(NC(c3cc(F)cnc3O)=O)CCCC2)cc1F 84311,c1(C(=O)NC2(C(=O)NCC(COC)(F)F)CC2)ncccc1O 84312,N1(CC(N2CCC(C(C(=O)NC(COC)(C)COC)F)C2)=O)CCC(=O)CC1 84313,c1(C(=O)NCC2C(CNC(c3c(OC)cccc3F)=O)C2)nc(C)c(C)nc1O 84314,CC1CCC(CC(=O)NC2(C(=O)NCC3(CO)CCCCC3)CCCCC2)CC1 84315,CCC(CC)(CN=c1[nH]nc(C(C)C)o1)NC(c1nocc1C)=O 84316,CCC(CNC(C1C2CN(C(=O)C#CC(C)C)CC12)=O)CC(C)C 84317,N1(C(=O)NCc2occc2C(=O)NOC2CCOCC2)CC(O)C(O)C12CCC2 84318,Cc1ccc2c(c1)CC(C(=O)NC(CNC(c1ccc(C(F)F)cc1)=O)CO)S2 84319,CCCCC(F)C(=O)NC1(C(=O)N(C)CC2(O)CCC2)CCN(C)C1 84320,N1(C(C(CN(C)C)O)=O)CCC2(C(N3CC(c4ccccc4)C(O)C3)=O)CC2C1 84321,N1(C(C2C(OC)(OC)CC2)=O)CCC2CCC(NC(=O)CC3(CO)CCC3)C1C2 84322,N1(C(c2c(Cl)cn(CCC)n2)=O)CCN(C(c2ccccc2)=O)CC(CO)C1 84323,CC1CN(C(=O)C(=O)NCC2CC2)CCCN1C(c1ccc2scnc2c1)=O 84324,c1(C2N(CCc3ccc(C(F)(F)F)cc3)CC2)ccc2c(c1)OCCO2 84325,Cc1ncn(C)c1C(N1CCC(C)C1CNC(c1c[nH]c(C(F)(F)F)c1)=O)=O 84326,N1(C(c2c(C)cnn2C)=O)CCC2CCC(C1)N2C(=O)CCC1CC(F)(F)C1 84327,Cc1cc(C(=O)Nc2ccc(-c3nnc(CCN)o3)cc2)c(C)o1 84328,C(=O)(C(CCOC)NC(=O)CC1CCC2CC12)N(CCCCC)C 84329,c1(OCCC)cccc(CN2CCC(C(=O)N(CC(C)O)CCN(C)C)CC2)c1 84330,C1(O)(C(N2C(C)CC(NC(=O)Cn3cc[n+](C)c3)CC2)=O)CCCC(C)(C)C1 84331,C(=O)(CC(C(C)C)NC(c1cnc(Cl)n1C)=O)NCC(C(=O)OC)(F)F 84332,CC1(C)OCCC1C(=O)NCC1CCN(C(c2cnc(S)[nH]2)=O)C1 84333,N1(C(CC(=C)Br)=O)CCN(C(=O)Cc2ccc(F)cc2)C2CCCCC12 84334,c1(C2(OC)CC2)cccc(C(N2CC(N(C(=O)C(=O)Nc3ncc[nH]3)C)C2)=O)c1 84335,C1(C(=O)NCCC2OCC(C)(C)C2)CC12CCN(C(=O)Cn1ccnc1O)CC2 84336,C(c1c(F)cccc1F)=CC(=O)NCC1(O)CCN(C(COCC#C)=O)C1 84337,C(=O)(C(C)(C(F)F)NC(=O)OC(C)(C)C)NCCCCN(C(C(CC=C)C)=O)C 84338,C1(NC(=O)Cn2ccccc2=O)CC(NC(=O)C(F)F)C12CCC2 84339,C(=O)(C#CC1CCOC1)N(CC(CN(C(c1c(F)ccc(C(C)C)c1)=O)C)O)C 84340,c1(CNC(=O)CC2C3CN(C(=O)CCc4cccnc4)CC23)cnc2n1CCC2 84341,CCC(C)(CO)C(=O)NCC(C1CCCC1)NC(c1ccccc1NC(C)C)=O 84342,Cc1cc(N2CCCC2)ccc1NC1CCCC(OC(C)C)C1 84343,c1(C(=O)NC2CC(CCNC(C(n3cc(Br)cn3)C)=O)C2)cc(C(N)=O)on1 84344,C12(CNC(C(C=C)(C)C)=O)CCCC1CCN2C(=O)CC1(O)CCC1 84345,c1(C(NNC(=O)N(C2CC(=O)N(C)C2=O)C)=O)cc(I)ccc1I 84346,C1(NC(CC=C)=O)CCN(C(c2ccc(-c3cc[nH]n3)cc2)=O)CCC1(F)F 84347,C(=O)(C(F)(CNC(C1CCCCO1)=O)C(C)C)NCc1n(CCC)ccn1 84348,N1(C(c2c(CCC)occ2)=O)CCCC(C(C)NC(c2snc(C)c2N)=O)C1 84349,N1(C(c2ccc(CC)o2)=O)CC(OC)CC1(C)CNC(c1cn(C)cn1)=O 84350,c1(C(c2nnc(N3CCCC(C(C4CC5(CC5)C4)C)C3)n2C)O)ccc(F)cc1 84351,CCCC(F)C(=O)NCC1CCCN1C(=O)NC.C12(COC)CCCN1C2=O 84352,N1(C(c2c(N)c(-c3ccccc3)ncc2)=O)CC(=O)NC2CCCCC12 84353,N1(CC(N2CC(C)(NC(c3c(C)n(C4CC4)nc3)=O)C2)=O)CCC(=O)NC1=O 84354,C12CCCN1NC(=O)C=CC(=O)N(C(C)(C)C)C2=O.c1(C(C)C)c[nH]nc1CC(O)=O 84355,c1(CC)ccc(C(C2CCN2C(=O)CCc2ccccc2C(=O)O)=O)cc1 84356,C(=O)(C(F)(F)C(F)F)NCC1N(C(C2CCCCCCC2)=O)CCCCC1 84357,C=CC(F)(F)C(=O)NC(CN(C)C(c1cnn(C2CCCCC2)c1)=O)CC 84358,C12(CNC(c3c(C)onc3)=O)CCCN(C(c3cc4n(n3)CCC4)=O)C1C2 84359,c1(C(N)=O)nc(Br)cnc1NC(C1CCCN(C(=O)CCc2ccoc2)C1)=O 84360,C1(NC(CN(CCC)C)=O)CC(C(=O)Nc2cc(C)ccc2CO)C12CCC2 84361,C1(CNC(c2cc(CC)no2)=O)(NC(c2cc(CCCO)on2)=O)CCCCC1 84362,c1(C(=O)NC2C(CNC(CCSCC)=O)C2)sc(-c2ccc(C)cc2)nc1C 84363,N1(C(C2C(C)(C)C2C#N)=O)CC2(C=C(C(=O)NC3CN4CCC3CC4)CO2)C1 84364,Cc1ncc(Cc2ccccc2)cc1C(F)(F)F.N1(CC)CC(OC(F)(F)F)C1 84365,C1(CC(N2C3C(CNC(c4cnc5sccn45)=O)C(C3)C2)=O)CC(O)C12CCC2 84366,C12(c3nc(-c4c(CCC)n(CC)nn4)on3)CCCCC1OCC2 84367,n1(CCNC2CC2)nnnc1C1(N(C)CCOC)CCC1CSCC 84368,Cc1nnc2cc(NC3CCCC34CN(C(=O)C(C)(C)NS(C)(=O)=O)C4)ncn12 84369,CC1(O)CCN(CC(=O)NC2CCCCC2CNC(=O)CNC=O)C1 84370,Cc1cccc(C(N2CC(C(=O)NC(C)CCCO)CCC2C)=O)c1C 84371,c1(OC)c(C(=O)NCC(F)CNC(c2c[nH]nc2[N+](=O)[O-])=O)cccc1F 84372,N1(C(CSCC=C)=O)CC(N(C)C(c2nnc(O)cc2C)=O)C(C)(C)C1 84373,C1(C(N(C(C(C)SC)C)C)=O)CN(C(C2(CCF)CCC2)=O)CCN1C 84374,C1(C(=O)NC(c2ncnn2C)CC)CC12CCN(C(C1(C)CC1)=O)C2 84375,CC1CN(C(c2ccccc2O)=O)CC1CNC(c1nnn(C)n1)=O 84376,N1(C(c2cc(C)ncc2)C(=O)NC2COC2)CC(C(F)(F)F)OC(C)C1 84377,C=C(Cl)CC(C(=O)N(CC(C)CCC)C)NC(c1ccc(=O)n(C)c1)=O 84378,C(=O)(C(O)CC(F)(F)F)NCC(CCOC)NC(c1c(F)ccc(F)c1Cl)=O 84379,c1(C(N(C2CCCN(C(C3CC34CCC4)=O)C2)CCO)=O)cc2n(c1)CCSC2 84380,Cc1ncccc1C(N1CCCCC1C(=O)NCC(O)CC1CCCC1)=O 84381,C1(NC(C(CC)OC)=O)CN(C(=O)CCCN2C(=O)CN(C)C2=O)CC12CCC2 84382,C1(CC(=O)NC(C2N(C(C=CC(C)C)=O)CCC2)(C)C)CCC(=O)NC1 84383,C1(C#N)(C(N(CC(CN(C(C2(CC#C)CC2)=O)C)O)C)=O)CC12CCCC2 84384,C1(NC(c2c(CC)csc2)=O)CCCN(C(c2cnc(O)c(C)c2)=O)C1C 84385,c1(CC(N2CCC(NC(C(C)OCC3CC3)=O)C2)=O)csc(Br)c1 84386,C1(NC(c2nn[nH]c2Cl)=O)CCCCC1NC(=O)C(F)CC1CCC1 84387,c1(C(N2CC(CNC(C3(COCC)CC3)=O)(OC)C2)=O)cn(C)c(O)n1 84388,N(C1CCCc2occc21)C(c1cnc(O)cc1C)c1n(CC)nnn1 84389,c1(C(=O)NCC2C(NC(c3ccc(Cl)c(F)c3)=O)C2)cccc2[nH]ncc12 84390,c1(C(N2CCCC(NC(c3csc(Cl)n3)=O)C2)=O)ccc([N+](=O)[O-])cc1Cl 84391,c1(C(=O)NCC2CCN(C(C(CC)C)=O)C2)ccc2c(c1)COC2=O 84392,CC(C)CCC(C(=O)NC1CNC(=O)C1)NC(=O)Cc1cc[nH]c1 84393,CC1CCC(c2cn(CCCCC(=O)NCCC3COCCO3)nn2)CC1 84394,N1(C(C(C(=C)Cl)(C)C)=O)CCC2CC(C1)CN(C(=O)C(C)(C)c1ccn(C)n1)C2 84395,c1(OC)cc(NC(C2(C)CCCC2C(=O)NC(C)(C)C)=O)cc(O)c1 84396,c1(C(=O)NC(CC=C)CNC(=O)C(C2CCC2)C2CCC2)cc2n(n1)CCO2 84397,N1(C(C2N(C(C)=O)CCCC2)=O)C(C)CC2CN(C(=O)CCc3cnn[nH]3)CC12 84398,C1(F)(CNC(Cc2n(C)ncc2)=O)CCC(NC(=O)COCC2CCOCC2)C1 84399,C(CC1CCC1)(C(=O)N1CC(O)(CN(C)C(c2cnns2)=O)C1)OC 84400,c1(C(N2CCCC(CNC(C(=O)N(C)C)=O)CC2)=O)cnc(C(F)(F)F)c(C#N)c1 84401,C1(NC(C(c2cnn(C)c2)C)=O)CCOC12CCN(C(C1CN(C)C1)=O)CC2 84402,N1(C(C2(NC(C3CC=CCO3)=O)C(C)(C)C2)=O)CC2CCC=CC12 84403,N1(C(C=Cc2cnc(C(C)(C)C)s2)=O)CC2CC(NC(c3cccs3)=O)C(C2)C1 84404,C1(CC(=O)NC(c2onc(C)n2)CO)COCCN1C(c1cc(O)cs1)=O 84405,CC1CC(C(=O)N(C2(C(=O)NC3(C)CCCC3C)CC2)C)CC(=O)N1 84406,c1(CNC(c2ncn(CC)n2)=O)cccc(NC(=O)Cc2csc(Cl)c2)c1 84407,N1(C(CCc2onc(CCC)n2)=O)CCN(C(C)=O)CC1.N12CC(C1)OC2=O 84408,c1(C(C(=O)NC2CC2)N(CC(C)(C)C)CCC#N)cccc(S(N)(=O)=O)c1 84409,CCCC(C(O)C(=O)N1CC2(CCN2C)C1)NC(=O)C(CC)(CC)OC 84410,C1(NC(c2csnn2)=O)CC2CC(C1)N(C(=O)C=CSCSc1ccco1)C2 84411,C1(C(C)=O)Cc2ccc(F)cc2C1.C(C)(CNC(C=CCC)=O)(CO)CCS.N 84412,C1(NC(C(CC)=CC)=O)CCC(n2cc(C3(O)CCOCC3)nn2)CC1 84413,C1(C)(CC(=O)OC)CCN(C(c2ccn(C)c2)C(=O)NC2COC2)C1 84414,C(c1cccc(F)c1Cl)=CC(=O)NCCC(C)NC(c1c(C)c[nH]n1)=O 84415,c1(C(=O)NC2(CO)CCCN(C(CCC(=O)NC)=O)C2)ccc2c(n1)CCC2=O 84416,Cc1cocc1C(=O)NC(C)CNC(C1CCCCC1)=O 84417,c1(CC)cnc(C(=O)NCC(O)CNC(C2CCN(c3nncs3)CC2)=O)cn1 84418,c1(-c2cc(C)ncc2)cccc(S(=O)(=O)Nc2cc3ccccc3n2C)c1 84419,C1(S(C)(=O)=O)(C(N2CC(C)C(N(C)C(c3c[nH]ccc3=N)=O)CC2)=O)CC(O)C1 84420,Cc1ccnc2ccc(C(=O)NCC(C3CC3)NC(=O)C(O)CCCC(C)C)cc12 84421,c1(C(=O)NC2CCN(C(C(CC)C)=O)C2(C)C)c(F)cccc1[N+](=O)[O-] 84422,c1(C(=O)NCC2CCN(C(C3CC=C(C)CC3)=O)CC2)cc(F)ccc1F 84423,CC1(C)C2CCC1(COC(C1CC3CCCN(C1)C3)=O)CC2 84424,c1(C(N2CCC(CCO)CC2)=O)ccc(C2=CCOCC2)c2cc[nH]c12 84425,CC1(C)CCCC(C(=O)NCC(CO)NC(C2(C)COC(=O)OC2)=O)CC1 84426,N1(C(CC2CC(=C)C2)=O)CCOC(CCNC(C2CC2c2ccnn2C)=O)C1 84427,S(=O)(=O)(c1cncc(F)c1)N1CCC(OCCO)C1 84428,C1(C2CCN(C(=O)C=C(C)C(F)F)CC2)(NC(C2CN(CC)C(=O)C2)=O)CC1 84429,N1(CC(C)NCC(Cc2ccccc2)CN)CCCCC1 84430,c1(NC(CCCN(CCC)CCC)=O)cc(C(=O)OC)cc(CC)c1 84431,C1(C(=O)NCCN(C(=O)C(C(C)(C)C)n2ccnn2)CC)CCc2nncn2C1 84432,CC(C)(C)CCCCCC(=O)NC1CC(NC(=O)C2=NNC(=O)CC2)C1 84433,C1(NC(C(CC#C)(C)C)=O)CC2CCCC(C1)N2C(=O)C(C(C)(C)C)OC 84434,N1(C(C(CC=C)(C)O)=O)CC(C(=O)NC2CCC(C3CC3)C2)CCC1(C)C 84435,C#Cc1cc(F)ccc1C(=O)NCCN(C)CC 84436,c1(CC(=O)NC2CC(C)CN(C(c3nn[nH]c3Cl)=O)C2)cc(S(N)(=O)=O)cn1C 84437,C1(NC(c2ccc(C#N)[nH]2)=O)CN(C(=O)CCc2cccc(O)n2)CC1C1CC1 84438,CCC(C)(C#N)C(=O)NCC(CC(C)C)NC(c1nc(Br)c(C)s1)=O 84439,c1(C(=O)NC(C(CO)NC(CCCC(CC)C)=O)C)cc2ccoc2cc1F 84440,N1(C(C2CC=C(C)CC2)=O)CCCC(C(N2CCOCC2C)=O)CC1 84441,C1(C(=O)NC(CCN(C(C2=CCN(C)C2)=O)C)C(C)(C)C)CCn2cnnc2C1 84442,C(C)(CCN=c1ncc(C(F)F)c[nH]1)NC(C(C1(OC)CCCCC1)(F)F)=O 84443,c1(C(=O)NC(C2CCN(C(CCN(CCC)C)=O)C2)C)c(C(C)C)n[nH]c1C 84444,c1(C(N(CC(C)NC(=O)C=Cc2ccccc2Cl)C)=O)cccn(C)c1=O 84445,c1(C(=O)NC(C(C)C)CNC(=O)CCC2CC2(F)F)ccnc(C(C)(C)C)c1 84446,CC12CN(C(=NCc3ccc(Cl)cc3)NCC3CCCO3)CCC1C2(F)F 84447,c1(C(N(C(CCCN(CC)CC)C)C)=O)nc2c(s1)CCC2 84448,N1(C(c2c(CCC)cccc2)=O)CCC2(CCC(NC(=O)C(C)N3CCC3)C2)C1 84449,C(=O)(CC(C)CNC(C1CCC(=O)CC1)=O)NCc1n(CC)cnn1 84450,C1(CC(=O)NC2C(CNC(c3ccc(C(C)(C)C)[nH]3)=O)CC2)CCCOCC1 84451,c1(C(=O)NCC(CCC)OC)cccc(Cl)c1C(F)(F)F 84452,CC1CCN(C(C2CC2F)=O)CC1CNC(c1cnn(CC2CC2)c1)=O 84453,C12(C(=O)OC)CCN(CC1)C2=O.C1(C(CCC)C)CCCC1OC 84454,Cn1ncc(C(=O)NC(CNCC2CCOC2c2ccnn2C)C(C)(C)C)cc1=O 84455,N1(C(c2n[nH]c(C)c2C)C(=O)NCCOC)CCCC2(C1)NC(=O)N(C)C2=O 84456,CC(C)CC(=O)NCC=CCC(=O)N(C(C)(CO)C1CCC1)C1CC1 84457,c1(SCCC(N2CCC(C(=O)NCC(C)O)(OC)CC2)=O)ccc([N+](=O)[O-])cc1 84458,c1(CCC)ccc2oc(C(=O)NCCC(CSC)OC)c(C)c2c1 84459,N1(C(c2ccnc(OC)n2)=O)CCN(C(c2cn(C)nc2Cl)=O)C(C2CCC2)C1 84460,N1(CC(=O)N(CC(CC)NC(=O)Cc2nc(C)sc2C)C)CCC(C)CC1 84461,c1(CC)c(C(N2CCC(CF)(NC(=O)CCC3(C)CC3)C2)=O)cnc2ncnn12 84462,C(C(CC(C)(C)C)NC(=O)C(N1CCC(C)(C2CCCO2)C1)=O)OC 84463,S(=O)(=O)(c1csc(-c2ccc(F)cc2)n1)N(C(CCSCC)C)C 84464,N1(C(Cn2nnc(C)n2)=O)CCOCC(C(=O)Nc2cc(N3CCCC3)ncn2)C1 84465,c1(C(=O)NCC(CNC(COC2(C)CCC2)=O)CO)ccc([N+](=O)[O-])s1 84466,N1(C(CCC#C)=O)CCCC(O)(CNC(C23CC(CN2C2CC2)C3)=O)C1 84467,c1(C(N2CC3C(CNC(C4(COC)CCC4)=O)(C3)C2)=O)ccc2nccnc2c1 84468,C12(C(N(C3CCC3)C)=O)CCCC1CCN2C(=O)Cc1cccnc1 84469,c1(C(N2CCN(C(C3C(=C)C3)=O)C3C2COC3)=O)cc(OC)cc2c1CCCC2 84470,c1(C(=O)NCCCNC(C2(F)CC2)=O)ccc(Cc2nc[nH]n2)cc1 84471,c1(C(=O)NCC(C)(O)CO)[nH]nc2ncccc12 84472,Cc1noc2cc(N3CCC4(CN(C(=O)CO)CCO4)C3)nc(Cl)c12 84473,C(=O)(C1=CNC2=NCCC2=C1)NC(CNC(c1ccc(COC)o1)=O)C(C)(C)C 84474,S(=O)(=O)(CCCCCl)CNCc1ccc(NC(CCSC)=O)nc1 84475,C1(C(N(CCCNC(C2C(C)C2C)=O)C)=O)CC12CC(F)(F)C2 84476,C(CC(=O)NOCC(C)(C)C)OC(CNC(C(C1CCCC1)OC)=O)(C)C 84477,CCC(C)CC(=O)NCC1CC(NC(C2(C(=O)OC(C)(C)C)CC2)=O)C1 84478,C1(OC)COc2c(C(=O)NC34CC(NC(=O)Cc5ccc(Cl)s5)(C3)C4)cnn2C1 84479,C1(NC(C(n2ccc(C(=O)OC)n2)N2CCC(OC)C2)=O)CCC(F)(F)CC1 84480,N1(C(C2C(=C)C2)=O)CCN(C(c2ccc(-n3cncn3)c(N)c2)=O)CC(C)(F)C1 84481,C1(NC(C2C(NC(C(C)N(C)C)=O)C=CCC2)=O)CCCC2(CC1)CC2 84482,c1(C(=O)NC2CN(C(c3c(CC)nco3)=O)CC(C)C2)ccc2nncn2c1 84483,CCCC(C)CC(=O)NCCC1CCCCN1C(=O)C=CSC 84484,c1(C(=O)NC2CC2C(=O)Nc2ccc(OC(F)F)cc2F)ccc([N+](=O)[O-])cn1 84485,C1(NC(C(C)OCCC=C)=O)CCCC1NC(c1cc(CC(C)C)on1)=O 84486,C1(N2CCC(COC)C2)C(C)OCC12CCN(C(c1cc(Br)ccc1Br)=O)CC2 84487,C(=O)(C(C(C)CC1CCCC1)N(c1ccc(Cl)nc1C)C)NCCCSCC 84488,N1(C(C2C(=C)C2)=O)CC(C(N2CCC(CC(=O)OC)C2)=O)CC(C)(C)C1 84489,N1(C(C(C)OCC)=O)CCN(C(c2cccc(OCC(F)(F)F)n2)=O)CC1C 84490,C(=O)(C1SCCc2sccc21)NC1CC(C)(NC(=O)C(O)CC(F)F)C1 84491,C(=O)(C(CC)C(F)(F)F)NCC(CCCC)NC(=O)C1=CCCC1 84492,CN1CCC(N2CC(NC(=O)NCCC3CC(CSC4CC4)C3)C2)CC1 84493,C(=O)(C(C)(C)C(C)C)NCC1CC(NC(c2c(C(=O)OC)c(C)[nH]n2)=O)C1 84494,CC1CCN(CC(=O)NCCNC(=O)NCc2cc(C(n3ccnc3)C)cs2)C1 84495,C1(COC)CN(C(=O)C(C)(C)N2CCCCC2)CCN1C(=O)Cc1ncoc1C 84496,c1(C(=O)NC(CC=C)CNC(=O)CN2CC=CC2)cnn(-c2ccncc2)c1C 84497,C1(CCCNC(=O)COCC2CCOC2)CN(C(C23CC(F)(C2)C3)=O)CCO1 84498,C(=O)(C1=C(Cl)CCOC1)N1CCC(O)(C(C)NC(=O)C(F)(F)c2ccccn2)C1 84499,c1(C(=O)OC)ccc(S(=O)(=O)N)c(Br)c1.C(C(O)C(N)=O)CCOC 84500,N1(C(CNC(CCC)=O)=O)CC(N(C(=O)C(C)Cc2ccccn2)C)C2(CC2)C1 84501,C1(NC(c2cc(C)no2)=O)COCCC1NC(=O)CCc1cc(Br)cs1 84502,Cc1onc(Cl)c1C(=O)NCCC(C)NC(c1c(C(F)(F)F)n[nH]c1C)=O 84503,N1(C(C2N(C)CC2)=O)CC2(CCC(NC(C3CC(O)C(F)C3)=O)CC2)C1 84504,C(c1ccc(Cl)cc1Cl)=CC(=O)NCCCCCCNC(C(CC)(C)CO)=O 84505,N1(C(CCSCCCC)=O)CCC2CN(C(=O)C(C3CCC3)OC)CC12 84506,N1(C(c2cc(CCCCC)[nH]n2)=O)CCCC2(CCN(C(C)COC)C2)C1 84507,C1(CNC(=O)C=CCF)CCCN(C(=O)CNS(=O)(=O)C2CC2)CC1 84508,c1(N2CCN(C(C=C(C)C(=O)O)=O)C(C(F)(F)F)C2)ncnc2[nH]c(C)nc12 84509,N1(C(=O)OC(C)(C)C)Cc2ccc(C(N3COC(C(N)=O)C3)=O)cc2C1 84510,c1(NC(C2C(NC(CC=C)=O)CCCC2)=O)ccc(C)c(CC)c1 84511,c1(OC)ccc(NC(c2c(NC)cnn2C2CCCC2)=O)cc1OCCN(C)C 84512,c1(NCC(C2CCCC2)NC(c2ccc(OC)nc2)=O)c([N+](=O)[O-])cnn1C 84513,Cc1ccc(C(=O)NCC(C)NC(c2c(C)noc2N)=O)cc1[N+](=O)[O-] 84514,Cc1cc(Br)ccc1CC(N1CCC(C)(C(N2CCCC(C(=O)OC)C2)=O)C1)=O 84515,N1(C(c2c(C)ncnc2C)=O)CCN(C(c2cc3ccccc3s2)=O)CC(O)C1 84516,C1(C)(CNC(COC(CC)C)=O)CCCN(c2nnc(C(C)(C)OC)s2)C1 84517,C(=O)(C1=CC2(CN(C(=O)C(C)(C)CC#N)C2)OC1)N(C(CC)COC)C 84518,C1(C(N(CCCF)CC)=O)CC12CCN(C(=O)C(C)C(=O)OC)CC2 84519,Cc1ccc(C23CC2CN(C(=O)NCCc2noc(C)n2)C3)cc1 84520,Cc1cncnc1C(=O)NC1(CNC(=O)C(C)Oc2ccccn2)CC(F)(F)C1 84521,C1(C(N(CCCCNC(C(CC=C)(C)CC)=O)C)=O)CCC2(CC1)CC2(F)F 84522,Cc1cccc(F)c1CC(=O)NC1C2CC1(C)CN2C(C1C2CCCCCC12)=O 84523,c1(C(N2CC(CC(C)NC(=O)Cc3ccns3)C2)=O)cc(Cl)cn1C 84524,N1(CCC)CC(NC(=O)CN(C(c2nnn(C)c2C)=O)C(C)C)CC1=O 84525,c1(C(N2C(C)CC(NC(C=CCN(C)CC)=O)C2)=O)ncc([N+](=O)[O-])cc1C 84526,CC1=C(C(=O)N(CC(O)CNC(=O)Cc2c[nH]nc2O)C)SCCO1 84527,NS(=O)(=O)c1cccc(C(=O)NCCNC(=O)CCSCc2ccccc2)c1 84528,Cc1cc(F)sc1C(=O)NC1(CNC(c2cc(C(F)(F)F)[nH]c2C)=O)CCCC1 84529,C(=O)(CC1C(=O)Nc2cc(Cl)ccc21)NCC1(NC(C)=O)CCOC1.C1C(=O)N1 84530,C=CCC(CC=C)C(=O)NC1CN(C(=O)Cn2cnc(=N)[nH]2)C2CCCC12 84531,CC(C)C1=NOC(C(=O)N(CC(=O)NCC2CCC(=O)O2)C)C1 84532,CN=c1[nH]cc(C(=O)NCC2CCC(C(=O)NC(C(C)C)C3CC3)C2)o1 84533,c1(N(C(C(C)N(C(=O)CCN(CCCN(C)C)C)CCN(C)C)=O)C)ccccc1 84534,c1(CN2C(CCC(=O)NC(C(=O)OC)C3CC3)CCC2)ccc(C#N)s1 84535,c1(C(=O)OC)ccc(N2CCCC2CCCNC(=O)C(C)SC(F)(F)F)nc1 84536,c1(COCC(=O)NCCN(C)C(C2CN(C3CCCCC3)C2)=O)ccncc1 84537,c1(COC)cc(C(=O)NCC2C(C)CCN2C(c2ccc[nH]2)=O)c(C)o1 84538,C1(CC)CCN(C(=O)C(CC)N(C)C)C1CNC(c1ncncc1Cl)=O 84539,C1(NC(C2(C(C)C)CCN(C(c3c(C)cc(C)s3)=O)C2)=O)C=CC(C)(C)CC1 84540,C12(C(=O)NCCCCCNC(C3CC34CCOC4)=O)CCN(CC1)CC2 84541,N1(C(C(CC)SC)=O)Cc2nccn2CC(NC(=O)C(F)(F)CO)C1 84542,CC1(CC(=O)NCC2CC2CC(=O)NC2(CO)CCOC2)CCOCC1 84543,C1(C(C)NC(c2c(CC)cns2)=O)CCCN(C(c2n[nH]cc2Cl)=O)C1 84544,Cn1ncc2c1CCN(S(=O)(=O)c1c[nH]c(C(=O)O)c1)C2C(=O)NS(C)(=O)=O 84545,C=CC(C)CC(=O)NC1COCC1NC(=O)C(C)=C1CC1 84546,N1(C(CSSC)=O)CC2(CCC(CNC(=O)CNC(=O)CCC(C)C)O2)C1 84547,N1(C(c2nc(C(C)C)oc2)=O)CC(O)CC1(C)C(=O)NOCCOCCOC 84548,C#CCC(C)(C)C(=O)NCC1CCN(C(=O)CCOCCOC)C12CC2 84549,C1(C(=O)NC2CCN(C(Cn3nc(C)c(Br)c3)=O)C2)CCC2C(C1)C2(F)F 84550,CCC(C)CCCCC(=O)N1CC(NC(=O)C=Cc2cnccn2)C2(CCC2)C1 84551,C(=O)(C1c2c[nH]nc2CN1C(c1cnc(C)c(C#N)c1)=O)NC1CCC(CC)C1 84552,c1(C(=O)OCC(=O)Nc2cccc(CNC(C=CC)=O)c2)nnc2ccccn12 84553,C(=O)(CCCCC(F)(F)F)NC1CCCC(NC(COC(CC)C)=O)C1 84554,C1(c2n(CC(=O)OC(C)(C)C)nnn2)(NC2CC=CCC2)CC2CSCC2C1 84555,C(C1c2ccccc2CN1C(C1C2COCC12)=O)NC(C(NOC)=O)=O 84556,N1(C(Cc2c(C)ccs2)=O)CC2CC(NC(C3CCC(C)(C)O3)=O)CC1C2 84557,N1(C(c2ccc(F)cc2Cl)=O)CCC(N=c2[nH]nc(CO)s2)(CO)CC1 84558,Cc1cc(C(=O)N(C(C)(C)CC(=O)NC2CCCC2(C)O)C)nc(O)c1 84559,C1(C(=O)NCC2(C(C)NC(Cc3c(C)ocn3)=O)CC2)CC2C=CC1CC2 84560,C1(CNC(C2CC(N(C)CC)C2)=O)CN(C(C2CCCCCCC2)=O)CCN1C 84561,N1(C(c2c(OC)c(C)ccc2)=O)Cc2ccnn2CC(NC(=O)CCCCF)C1 84562,c1(C(N(C2CCN(C(=O)COCc3nnc(C)s3)C2)CC)=O)cccc2sncc12 84563,c1(CNC(=NCC2N(CC)CCC2)NC2C3(CC3)C23CC3)ccc(F)cc1C 84564,N1(C(c2cc(SC)oc2)=O)CC2CCCC2C1C(=O)Nc1cccc(Cl)c1 84565,C=CCC(C)(C)C(=O)N1C2CCC(C2)C1C(=O)NC1COC2(CCC2)C1 84566,c1(OC(C(=O)NC2CC(CNC(c3c(C)cns3)=O)C2)C)ccc(Cl)cc1 84567,C1(O)(Cn2cc(CC(C)C)nn2)CCN(C(=O)CCC(F)F)C1 84568,C1(CNC(C2(NC(=O)CC3(C(F)(F)F)CC3)CCCCC2)=O)CN2CCC1CC2 84569,N1(C(c2c(F)ccc(OC)n2)=O)CCC2CCN(C(=O)CNC=O)CC2C1 84570,c1(C(=O)NC2C(NC(=O)C=Cc3cnccn3)CCCC2)c(Cl)cccc1Cl 84571,N1(C(C2CN(C(C3C(COC)CC3)=O)CC2C(C)C)=O)CCC(C2CC2)C1 84572,C(CC(C)(C)C(=O)NCC(CO)NC(C1(F)CCN(C(C)(C)C)C1)=O)OC 84573,c1(C(N(CCCCNC(CC(CC)OC)=O)C)=O)cc2cccc(Cl)c2[nH]1 84574,c1(C(=O)NCc2ccc(C(C)NC(COCC)=O)cc2)nnn2c1CCCCC2 84575,C(=O)(C1CCCc2nc[nH]c21)NCCCOCCCNC(CNS(N)(=O)=O)=O 84576,N1(C(C2CC(NC(CCCOCCC)=O)C2(C)C)=O)CC2(C1)CC(C)(C)C2 84577,C(=O)(CCN=[N+]=[N-])N(CCC(=O)NC(c1nc(=O)o[nH]1)C)CC1CC1 84578,CC(N=c1[nH]c2c(c(=NCc3ccn(C)n3)[nH]1)CCCC2)c1ccc(O)nc1 84579,C1(C2C(CC(=O)NC(=O)C(F)C3CCCC3)C2)CCC2CCC12 84580,Cc1cc(C(N2CC(NC(c3cc(C4CCC4)nn3C)=O)C2)=O)ncc1C(N)=O 84581,C1(C(N(CC#CC)C)=O)CC2(CC2)CN1C(C1CC12CCC2)=O 84582,c1(C(=O)Nc2c(C)cc(NC(C3CCCOC3)=O)cc2)ccnc2c1cnn2C 84583,C1(C(C(=O)NC(C)C)N(CC(C)C)Cc2ccnn2C)CCCOCC1 84584,C(C(C)(C)CCNC(C1COCCN1C)=O)NC(C=CC(CC)=CC)=O 84585,C1(C(=O)NCCCNC(c2c(F)ccc(C(C)C)c2)=O)Cc2cc(Cl)ccc2O1 84586,S(=O)(=O)(c1cc(Br)c(C)cc1F)N1CCCC(CN(CCC)C)C1 84587,Cc1ccc2c(C(=O)N(CCC(C)NC(=O)C(C)C(C)(C)C)C)coc2c1 84588,N1(C(C(CCOC)C)=O)CC2(CCCC2NC(=O)CC2(OC)CCOCC2)C1 84589,N1(C(c2c(C)nc(Br)s2)=O)CCC2C(CCN2C(c2cc(Cl)cc(Cl)c2Cl)=O)C1 84590,CCCC(CCC)C(=O)NC1CN(C(=O)Cc2cc[nH]n2)C1 84591,C1(N(C(c2cnc(CCCC)[nH]2)=O)C)CCCCN(C(c2cc(C#N)no2)=O)C1 84592,C(C(C(C)(C)C)NC(C1CCCCCC1)=O)NC(C(c1ccncc1Cl)C)=O 84593,C1(NC(CC(C)OC)=O)C2CC1CN(C(c1nc(C(F)(F)F)oc1C)=O)C2 84594,N1(C(C2N(C)CCOC2)=O)CCC2(CC1)CCN(C(=O)CCCC(F)(F)F)C2 84595,C1(NC(CCOCC)=O)CC(C)(NC(c2cnc[nH]2)=O)C1 84596,C1(CNC(c2ncccn2)=O)CCCCN(C(=O)CCOCC2CCC2)C1 84597,N1(C(C(CC)(C)C)=O)CCC(O)(C(C)CNC(c2cc(C)c(C)nn2)=O)CC1 84598,C1(CC(C(=O)NC2CC2)N(CCC)Cc2ccc(O)cc2)CCOC(C)(C)C1 84599,C12(CNC(C(CC)N(C)C)=O)CC(C1)C(NC(=O)C1=COCCO1)CO2 84600,c1(CC)cc(=NC(=O)CC2CN(C(=O)CC(O)C(C)C)CC2C)[nH]n1C 84601,N1(C(COCc2n(C)c(S)nn2)=O)CC(CNC(=O)C(C)(C)C#N)CC12CCC2 84602,Cc1cccnc1CC(=O)NC1CCN(C(=O)Cc2ccc(Cl)cc2)CC1 84603,c1(C(=O)NCC(CC)NC(=O)CCCCCSC)c(C)cccc1O 84604,C1(C(=O)NCCN2CC(Cn3ccnc3)C2)COC(C2CC2)C1 84605,C1(CC(N2CC(O)(CC)C2)=O)CN(C(=O)C(C)NC(N)=O)CCO1 84606,C(C(C)CC(=O)N(C(C)C(C)(C)O)C)NC(c1c(C)nco1)=O 84607,C1(C(N2CC(CNC(=O)C(F)(F)CC3CCCO3)C2)=O)CCc2[nH]nc(O)c2C1 84608,Cc1nc(CC(=O)NC(c2cccnc2)C(=O)NCCCC(=O)N(C)C)cs1 84609,CC1CC(C)N(C(=O)CNC(C2(C#N)CC3(CC3)C2)=O)CCN1C(c1cscn1)=O 84610,C(=O)(C(O)CC(F)(F)F)N1C(COC)(CNC(c2ccc(O)nc2Cl)=O)CCC1 84611,Cc1nc(N(C)C)sc1C(=O)NCCN(C(=O)C(O)CF)C(C)C 84612,C1(C)(CNC(c2cn(C)nc2C(F)F)c2n(C(C)C)nnn2)CC2CC2C1 84613,C12(NC(C(C)=C3CC3)=O)CCCC1N(C(c1cnn3c1OCC3)=O)CCC2 84614,C12(NC(CCC)=O)CC1CN(C(c1cnn(Cc3ccccc3)c1F)=O)C2 84615,C1(NC(CC(CCC)(C)O)=O)CCC2CCN(C(c3cc(C)nn3C)=O)C1C2 84616,C1(c2nccn2C)(OC)CCN(C(=O)C(=Cc2cccnc2)NC)C1 84617,CC(C)CN(CC(O)C1CC1)C(C)C 84618,C1(CN(C(COCCCOC)=O)C)CN(C(C2C3CC4C(C3=O)C24)=O)CC12CC2 84619,N1(C(C(C)Cn2ccnc2)=O)Cc2cccn2CC(C(N2CCOCC2)=O)C1 84620,CC1CC(CNC(=O)CCOCC(F)F)CN1C(=O)CCN1CCCC1=O 84621,C1(C(=O)NCC(C)CN(C)C(c2ccc(F)cc2F)=O)Cc2ccccc2C1 84622,C12(NC(c3cn(CC(N)=O)nn3)=O)CCCC1(F)CN(C(C1CCC1)=O)C2 84623,CC1CC2(CC(C(=O)NOCC(=O)NCC(O)C3CC3)C2)C1 84624,n1(CC(=O)N(C(CNC(COCCSC)=O)C)C)ccc(=O)c([N+](=O)[O-])c1 84625,C1(NC(CC(C)(C)C#N)=O)CCCCCN(C(=O)C2=CCCC2(C)C)C1 84626,N1(C(C(CC)OCC)=O)CCN(C(=O)C=Cc2c(C)coc2C)C(CC)C1 84627,c1(CN(C(c2csc(Cl)c2)C(=O)NC2CCOC2)CC)ccc(F)cc1 84628,c1(C(C)=O)cc(N(C2CCCCC2C)S(C)(=O)=O)ccc1F 84629,C(C(F)(F)C(=O)NC1CCOCC1C(=O)NCCC(C)(O)C1CC1)OC 84630,C1(C(N(OC)C)=O)CCCCCN1C(C1CC1C1CC1)=O 84631,c1(NC)ccc([N+](=O)[O-])cc1C(=O)NCCC1CN(C(=O)CC2(C)CC2(F)F)C1 84632,Cc1nn(CC(=O)NCCN(CCOCCO)C(C2(O)CC(F)(F)C2)=O)c(=O)o1 84633,C1(NC(c2cccc(C)c2)=O)CC2CCC(C1)N2C(C1(CF)CC2(CCC2)C1)=O 84634,c1(CN2C3CN(C(C4N(C)CCC4)=O)C(C3)C2)ccc(F)c([N+](=O)[O-])c1 84635,C1(C)(CNC(C2C(C)C2)=O)CCN(C(C2CC23CC(O)C3)=O)C1 84636,C1(C(=O)NCCCN(C(Cc2cccc(SC)c2)=O)C)CCCC(C)(C)C1 84637,c1(C(N2CC3C(C(=O)NCCCC(=O)OC)(CC3)C2)=O)c(F)cc(Br)cc1Br 84638,c1(CC(=O)NC2(CNC(C(COC)C)=O)CCCCC2)c(F)cccc1F 84639,C(CC(=O)NC1CCC(c2nncn2C)CC1)(C(F)(F)F)OCC 84640,C1(NC(c2ccn(CC(C)C)n2)=O)(CO)CCCN(c2ccc(C#N)nc2)C1 84641,Cc1ccc(CCNC(c2cccc(F)c2C)c2nnnn2C)cc1Cl 84642,CC1(C)CCCC(CC(=O)NCC2(C)CCCC2NC(=O)Cn2cccn2)C1 84643,N1(CCN2CCC(CC(=O)N(CC(=O)OC(C)(C)C)CCO)C2)CCNC(=O)C1 84644,C(=O)(CCCC(F)(F)F)N1CC(C)C(C)(C(=O)NC2CCn3ccnc3C2)C1 84645,C1(NCCN(C(CC)C)CC)CCC(C)(C)C1.C(C)(C)(C)OC=O 84646,c1(C(=O)NC(c2ccc(F)cc2)CC)cc(C)c2sccc2c1 84647,C1(NC(c2c(C)cc(SC)o2)=O)CC(C)CN(C(c2cn(C)cn2)=O)C1 84648,N1(C(c2nc(OCC)oc2)=O)CCC(NC(C2CC(=O)N2)=O)C(C)(C)C1 84649,C1(C(N2CC(C(C)NC(C3=C(C)CC3)=O)C2)=O)CC2CC1CC2=O 84650,c1(C(N2CCC(n3cncn3)C2)C(=O)NCC(=C)C)cc(F)ccc1Br 84651,C(Cn1cncn1)(C(=O)NC1C2CCCC12)NC(C1CC(=C)C1)=O 84652,c1(OC)cc(C)cc(C)c1C(C)NC(c1ccc(C)c(C)c1)C 84653,N1(C(c2c(CC)onc2C)=O)CCC(NC(=O)C=CC2CCCC2)C(C)C1 84654,c1(C(=O)NCC2C3CN(C(Cc4c(C)n(C)nc4)=O)C2C3)n[nH]c2c1CCCC2 84655,C=CC1(C(=O)NC2CCC(C(=O)NCC3CC3(C)C)C2)CCCC1 84656,C1(C2N(C(C3(CCC=C)CC3)=O)CCC2)CCN(C(=O)CC(C)CC)CC1 84657,C=CC1OCCCC1C(=O)N(C)CCOCCN(C)C(c1ccc(F)cc1N)=O 84658,C1(C(N2C(CC#C)CCCC2)=O)CCN(C(=O)CN(C)C(=O)OC)CCO1 84659,C1(N(C(c2ccn(CC)n2)=O)C)C2CN(C(C3(O)CCOCC3)=O)CC12 84660,C(=O)(C1=CCS(=O)(=O)C1)NCCCNC(C12OC(C)C(C1)C2)=O 84661,CCCC(C(=O)NCC(C)(C)C(=O)NCC1OCCC1C)N(C)C 84662,C(CN=C(NCC1(CO)CC2CC2C1)N1CCC1)N(C1CC1)CC 84663,c1(N(C(=O)C(C)OC2CCCC2)CCN(CC)CC)ncc([N+](=O)[O-])c(C)n1 84664,C#Cc1cc(F)cnc1NC(C1CN(C(c2cncc(F)c2)=O)CCC1O)=O 84665,N1(C(c2c(OC)nsc2OC)=O)CCC(C)C(NC(C2SCCCS2)=O)C1 84666,C1(CNC(C(COC)C)=O)CN(C(=O)C(c2ccc(C)s2)C)CCC12CCC2 84667,c1(C(=O)NCCC(C)N(C(=O)CC2(C)CCCCC2)C)cc(Br)cn1C 84668,CCC(C)CC(=O)NCC1(NC(=O)CSCC(N2CCOCC2)=O)CCCC1 84669,C1(F)(C(N(CCCCC=C)C)=O)CCN(C(C2SCC=C2C)=O)CC1 84670,Cc1cc(C(=O)Nc2ccnn2-c2ccccc2Cl)c(C)[nH]1 84671,C(=O)(C1SCCc2sccc21)NCCN1CCN(C(C(CC)SC)=O)CC1 84672,C1(CNC(C=CSC)=O)CCN(C(=O)NC2CCCC2c2nnc(S)n2C)CC1 84673,C1(C2CCN(C)CC2)(C(=O)NC2CCCC(CNC(COC(CC)C)=O)C2)CC1 84674,N1(C(c2ccc(N)c(F)c2)=O)CC2(CCCC2NC(C2CCCC23CC3)=O)C1 84675,Cc1c(NCC#CCOCCCCCN2CCCC2)ncnc1N1CCCC1 84676,N1(C(Cc2ccc(OC)cc2)=O)CC2CC1CN2C(c1cnc(SC)nc1)=O 84677,c1(C(N2CC(CCNC(=O)Cc3ccccc3Cl)OCC2)=O)cnc(O)cc1O 84678,c1(C(N2CCCC(N(C(=O)C(F)C3CC3)CCF)C2)=O)cc(Cl)cc(Cl)c1 84679,c1(C(N(C)CC2(O)CN(C(=O)COc3ccon3)C2)=O)c(F)cccc1[N+](=O)[O-] 84680,C1(C(=O)NC(C(C)NC(c2cc(C(F)(F)F)cs2)=O)(C)C)CCCN(CCF)C1 84681,C1(CC)C(NC(C2CC2c2cccs2)=O)CCN1C(=O)CCOc1cccnc1 84682,CC1CN(C(c2ccoc2)=O)CC2(CCN(C(c3cccc(N)c3O)=O)CC2)O1 84683,C1(NC(CSCCOC)=O)CC(O)CN(C(c2ccc(O)nc2Cl)=O)C1 84684,C(=O)(C(O)CC[S+](C)C)NC1CC(CNC(CC(C)SC)=O)C1 84685,c1(CC)nc(NCC(=O)NCC2CCN(N(C)C)C2)[nH]c(=N)n1 84686,Cc1cc(CNC(=O)COC2(C)CN(C(=O)CC3CCCCC3)C2)cnc1O 84687,CN1C2CCC1CC(C(N1CC3(CCC3NC(c3cccn(C)c3=O)=O)C1)=O)C2 84688,c1(N2CCC(NC(C3(C)CC3(F)F)=O)C(CO)CC2)ccc([N+](=O)[O-])cc1F 84689,S(=O)(=O)(c1cn(C)nc1C)Nc1scc(-c2c(C)ccc(Cl)c2)c1 84690,C1(=O)C(C)(C)C2CCCN2N1.C1(CCCC2(C)CC2)CC(=O)C1 84691,CC(CN(C)C)CCC(=O)NCC1C=CC(NC(=O)CN2CCSCC2)C1 84692,c1(C(N2CCN(CC)CC2C)C(=O)NC2CCCC2)nc(Cl)cc(C)c1Br 84693,c1(CN2CCC(c3cccc(C(=O)Nc4cnoc4)c3)CC2)cc(Cl)cc(Br)c1F 84694,C(=O)(CC1OCCc2ccccc21)NC(CNC(C1(OC(C)C)CCC1)=O)(C)C 84695,C(CCCCCCC(=O)NC1CCN(C(C2COC3(CCC3)CO2)=O)C1C)SC 84696,c1(SC)cc(C(=O)NC2CC2NC(=O)Cc2cncn2C)ccn1 84697,CCC(C)CCCCC(=O)NS(=O)(=O)c1ccc(C#N)o1 84698,c1(OC(C(=O)NCC(C)NC(=O)CC(O)c2ccccc2)C)ccc(CO)cc1 84699,c1(C(=O)NCCC(C)NC(c2cnn(C)c2Br)=O)ccc(C(=O)CF)cc1 84700,C1(C(=O)NCC2(CNc3ncc(Cl)c(O)n3)CCCC2)CCc2nnc(O)n2C1 84701,CC1(CCNC(C2(n3cncn3)CC2)=O)CCN(C(C2CCCC(=O)O2)=O)C1 84702,c1(C(N(C2CCCN(C(C3C(OCC)C3)=O)C2)CC)=O)cnc(CO)nc1C 84703,C1(C(N(CC#C)CCO)=O)N(C(=O)C(C)CSC)CCC1(C)C 84704,Cc1ccc(F)cc1C(N1CCC(CNCC(c2ccccc2)C)C1)=O 84705,C(=O)(C1=NOC(C)(C)C1)NC1CCCC(NC(c2c(C)ncc(C)c2)=O)CC1 84706,C1(NC(C(C)(C)NC(Cc2cn(C)nc2)=O)=O)CC12CC(O)C2 84707,C(=O)(CCCC(=O)N(c1ncnc(C)c1Br)C1CCNCC1F)OC 84708,C#CCC(C)(C)C(=O)NCCCCC1CCCN(C(c2cn(CCF)nn2)=O)C1 84709,Cc1cc(C(=O)NCC(C(=O)NC23CC2COC3(C)C)C(C)C)cnc1C 84710,NS(=O)(=O)c1ccc(NCC(N2CC(C3=NOC(C)(c4nn[nH]n4)C3)C2)=O)cc1 84711,N1(C(CCN(CCC)C)=O)CC(c2ccccc2)(NC(c2occc2Cl)=O)C1 84712,C1(NC(c2ccns2)=O)CCN(C(=O)CCOc2ccccc2Cl)CC12CCC2 84713,c1(NC(C2C3(CCN(Cc4cc(C)c(Cl)nc4)C3)C2)=O)c(Br)cc(F)c(F)c1F 84714,c1(CN(C)C(C2(CNC(C34CCC(C3)C4)=O)CC2)=O)ccn(C)c1 84715,c1(C(N2CC(C)(CC(=O)Nc3ccc(Cl)cc3)C2)=O)cc2cc(Br)ccc2s1 84716,C(=O)(CCCCC(=O)NC1CN(C(C2(O)CCOC2)=O)CC2(CC2)C1)NC 84717,C1(NC(C=C(C)CNC(=O)CCCC2CCOCC2)=O)CCOC1(C)C 84718,C(C(C)(C(=O)NC1CCC1NC(C1(CCCc2ccccc2)CC1)=O)OC)OC 84719,n1(CCCC)nc(C)c(C(=O)NC23CC2CN(C(=O)CN2CCCC2C)C3)c1Cl 84720,N1(CC2(C)CCN(C(Cn3c(C)cc(C(F)F)n3)=O)C2)CCC(O)C(C)C1 84721,Cc1cc(C(=O)NC2(C)CC(NC(C3CC(=O)NC(C)C3)=O)C2)cc(C)n1 84722,N1(C(c2scc(OC)c2)=O)CC2CC(NC(c3cn(C(C)C)cc3C)=O)C1C2 84723,N1(C(C2CC(OC)C2)=O)CCC2(CC2)CC1C(=O)NC(CCO)C1CCC1 84724,CC1OCCC1(F)C(=O)NCCC1CCCN(Cc2nccn2C)C1 84725,C1(CNC(c2ccc(C(C)(C)C)[nH]2)=O)CN(C(=O)CSC2CC2)CCC12CCC2 84726,c1(NC(C2NCCN(C(c3c(C)ncnc3)=O)C2)=O)ncnc2[nH]c(Br)nc12 84727,N1(C(c2c(CC)occ2)=O)CC(NC(C2CC(C#N)C2)=O)CCC1C 84728,CC1CCOC1CCNC(=O)C(C1(C)CC1)NC(=O)Cc1ccon1 84729,C1(NC(c2ccc(SC)s2)=O)CCN(C(c2ccc(N)c(N)n2)=O)C(C2CC2)C1 84730,c1(C(N2CC(C)(NC(C)=O)C2)=O)ccc(NCc2ccc(Cl)s2)cc1 84731,C1(C(=O)NCCC2(C)CCCO2)CCN(C(=O)CC2CCCC3CC23)CCO1 84732,C1(NC(CC(C)C)=O)CC2CC(NC(C3CNC(=O)N3)=O)CC12 84733,S(=O)(=O)(c1cccc(=NCC(C)C(C)C)[nH]1)N1CCC(C(C)C)CC1.CCCO 84734,N1(CC)CCC(CNC(c2conc2NC(=O)CC2CC3CC3C2)=O)C1 84735,c1(C2(C(=O)NCC(C)(O)CNC(c3csc(Cl)n3)=O)CC2)cccnc1Cl 84736,C1(CNC(=O)C(N2CCCC2c2ccc(Cl)cc2)=O)CCCS(=O)(=O)C1 84737,C1(=CCNC(C=CCCC(C)C)=O)CCN(C(c2c(C(C)C)cnn2C)=O)CC1 84738,C(=O)(C(F)CC(CC)CC)NCC(=C)CCNC(C1(C(=O)NC)CCOCC1)=O 84739,CC1(CS(=O)(=O)Nc2ccc(Cl)cc2)CCCN(CC(N2CCCC(CO)C2)=O)C1 84740,N1(C(C(CC(C)(C)NC(c2cc(OC)ns2)=O)F)=O)Cc2ccc(C#N)cc2C1 84741,CC1C(NC(=O)CNC(C2CCCCC2)=O)CC2CCC1N2C(=O)CCC1CC1 84742,c1(C(C(=O)NCC#CCNC(C2OCCN(C)C2)=O)=O)ccc(F)cc1F 84743,C1(C(N2CCC(Cc3onc(C)n3)CC2)=O)CCOC2(CCC2)C1 84744,Cc1cc(C)c(C(N2CC(C)(C)C2Cn2cc(CCC3CCCC3)nn2)=O)[nH]1 84745,C(=O)NNc1ccc(Br)c(F)n1.C1(NC(c2ccco2)=O)CCC(N2CCCCC2)C1 84746,C1(C(=O)NCCOCCOCC)CCOCC1NC(=O)C=NOC 84747,CC1CN2CCN1C(C(=O)NC1CCN(C(=O)CC3CC(F)C3)CC1F)C2 84748,C1(CC)CN(C(c2coc(CNC(C3(N(C)C)CCC3)=O)n2)=O)C(C)CO1 84749,C(C(C)(O)CC(=O)N1CCC1CNC(=O)C(C)(C)Nc1ccc(Cl)cc1)OC 84750,N1(CC(=O)NC(C(CC)C)CO)CC(C(=O)OC)C2(CN(C(C)(C)C)C2)C1 84751,N1(C(C2CC3CN(C(CCC(C)C)=O)CC2C3)=O)CCC2CN(C)CC2C1 84752,C1(NC(CCC)=O)CC(C)(C(=O)NCC(CO)C2CC2)C1 84753,n1(CCCC(=O)NC2CN(C(C34CCCC(CO3)C4)=O)C2)cnc2ccccc12 84754,C1(C(=O)NC2C(CC)N(C(=O)C(C)n3cccn3)CCC2)CC(C)(C)C(C)(C)C1 84755,C1(NC(=O)C(C2CCCCC2)O)CCCC1OCc1cccnc1 84756,FC1CC2CC1CC2NCc1cccc(C2CC2)c1 84757,N1(C(=O)CC2CCCC2(F)F)CC2CCCC(C1)N2C(c1cncc(Cl)c1)=O 84758,c1(C(=O)NC(C)CCNC(c2cc(Br)co2)=O)n[nH]cc1[N+](=O)[O-] 84759,c1(C(=O)NCC2CC(F)(CNC(CCN(C)CC)=O)C2)sc(C#N)cc1Cl 84760,Cn1cc(C(=O)NC2C3CC2N(C(=O)Cc2ccc(C#N)nc2)C3)ccc1=O 84761,C#CCCCCCC(=O)N1CC2CCC1CN2C(=O)CCCC 84762,N1(CC)CC(C(=O)NCCOCCNC(C2CC(=O)N(O)C2)=O)c2ccccc21 84763,c1(C2OCCN(C(c3nscc3Br)C(=O)NCC3CC3)C2)ccc(F)c(F)c1 84764,N1(C(c2n(CC)cc(Cl)c2)=O)CCCC(N(CC(N2CCC(C)CC2)=O)C)CC1 84765,c1(C(=O)NCCNC(CC2C(C)C2)=O)cccc2c1NC(=O)CC2 84766,C12=CC(=NC(=O)N3CCCCC13)NN2.c1(C(=O)OC)ccc([N+](=O)[O-])cn1 84767,N1(C(c2c(C)cno2)=O)CCC2(CCCN2C(c2ccc(C(C)C)c(Cl)c2)=O)C1 84768,C1(F)(CNC(c2ccoc2)=O)COCCN(C(=O)Cc2ccc(Br)cn2)C1 84769,C1(SCC)CC(C(=O)NCC(C)(C)CCNC(c2nc(O)sc2C)=O)CCO1 84770,c1(C(N2CCN(C(C(C)=C3CC3)=O)CC2C2CC2)=O)cc2cc(Br)ccc2[nH]1 84771,N1(C2CCN(C(CSCC(N)=O)=O)CC2)CCN(C(=O)CO)CC1=O 84772,CC(=O)CCCC(=O)N1CCC(C)C1CNC(=O)C(O)C1CCC1 84773,C1(NC(c2cc(OC)no2)=O)CS(=O)(=O)CC1NC(c1c(Cl)cnn1C)=O 84774,c1(CNCC2N(C(c3c(OC)cncc3)=O)CCOC2)cc(F)ccc1Br 84775,N1(C(C#C)C)CCN(C(CC2CC2(Cl)Cl)C(=O)NCc2ccccn2)CC1 84776,CS(=O)(=O)C1CC(C(=O)NCC2CCN(C(=O)CC3C=CCC3)C2)C1 84777,C1(CNC(C=C(COC)C)=O)CCN(C(c2cc(OC)cc(C)c2)=O)CC1C 84778,C(=O)(C1CC(=O)c2c(F)cccc21)NCC(CNC(c1c(C)cccc1Cl)=O)C 84779,c12c(cccc1NC)NC(=O)CCNC2c1n(CC=C)nnn1.C1CC1.N(C)(C)CC 84780,C1(NC(c2c[nH]cc(Cl)c2=O)=O)CC(N=c2ccn3ccnc3[nH]2)C12CCC2 84781,N1(C(c2ccc(C#C)c(Cl)c2)=O)CC2(C)CN(C(=O)CC(C)SC)CC2(C)C1 84782,N1(CC)CC2CN(C(=O)C(C3CCCN(C(=O)CCCOC)C3)(C)C)CC2C1 84783,c1(C(N2CC(OC)C(NC(C3(C)CC=CCO3)=O)C2)=O)cc(Cl)cc2c1CCC2 84784,C(=O)(C=CS(C)=O)NC1(CNC(C(C)OC(=O)NCc2ccccc2)=O)CC1 84785,c1(NCCCN2CC(C)OCC2)ccc(O)c(-c2ccc(Cl)cc2)c1 84786,C1(NC(c2c(CC)n(C)nn2)=O)CC(CNC(=O)CCc2cnn[nH]2)C12CCC2 84787,C(=O)(C(CNC(=O)C1=CCCC1C)C(C)C)NC(COC)(C)C(N)=O 84788,CN1CCn2ncc(C(=O)NC3CC(NC(=O)Cc4cccs4)C34CCC4)c2C1 84789,N1(C(c2ccc(N)cc2F)=O)CCC2(NC(=O)C(F)CC3CC3)CCCCCC12 84790,C1(C(=O)NC2C=CCN(C(Cc3scc(C)c3)=O)C2)CCc2cnnn2C1 84791,Cc1ccc(C(N2CCC(NC(=O)CC3CCC(C)(C)C3)CC2)=O)c(O)c1 84792,CC1CC=C(C(=O)NC2(C(=O)NCC3(CO)CCC3)CSC2)CC1 84793,CN1CCCC(CCC(N2CCC(C)(NC(=O)Cc3nc[nH]n3)C2)=O)C1 84794,c1(C(=O)NC2CC(NC(c3cc(C)c(Br)s3)=O)C2)cccc(Br)c1O 84795,N1(C(C(Cc2c(C)nc[nH]2)O)=O)CCC(NC(=O)CCCCCN(C)C)C12CC2 84796,O=C(C1=CSCS1)NCC1CCCCN1C(=O)Cc1ccccc1Cl 84797,N1(C(c2c(C(C)C)cco2)=O)CC(NC(c2ccc(Cl)s2)=O)C2(CCOCC2)C1 84798,N1(C(C(C(C)C)F)=O)CCCC(F)(CNC(=O)C=CC2CC2)CC1 84799,c1(CC)ncccc1NC(=O)CC1CCCN1C(c1cncc(Br)c1)=O 84800,c1(C(=O)NCC(CN(C(CC(n2ccc(C)n2)C)=O)C)O)cccnc1C1CC1 84801,CC1=C(C(=O)N(C2CC(NC(c3ccnc(OC(F)F)c3)=O)C2)CC)SCCO1 84802,C1(CNC(C(C(C)C)N2CCCS2(=O)=O)=O)CN(C)CCN1C(c1cnco1)=O 84803,c1(C(c2nnnn2C(C)C)Nc2c(OCC)cccc2)cc(Cl)ccc1[N+](=O)[O-] 84804,C(CC(=O)NC1CC12CCCC2)(CC(C)C)NC(c1cn(CC)nc1C)=O 84805,c1(OC)cccc(C2CCN(C(=O)NC3CCN(c4ccccc4)C3)CC2)c1 84806,c1(C(=O)NC(CC=C)CNC(c2coc(C(N)=O)c2)=O)c(F)ccc2n[nH]cc12 84807,C1(C(C)C)CN(C(C2CC(=O)C2C)=O)CCN1C(C1CS(=O)(=O)C1)=O 84808,C(=O)(C(C)(C)C(=O)N1CCC(C(C)NC(=O)C(C)=CC2CC2)CC1)OCC 84809,c1(C(N2C(CC)C(NC(=O)C(O)C=C(C)C)CC2)=O)coc2ccccc12 84810,c1(C(=O)NCC(CC=C)NC(=O)C(C)(F)CCCC)cnc2c(ccn2C)c1 84811,N1(CCC(N2CCC(NC(C3CCC(C#C)CC3)=O)C2)=O)Cc2ccccc2C1 84812,c1(CC)ccc(C(=O)N(C(C)CNC(c2cnn(C)c2Cl)=O)CC)c(F)c1 84813,N1(C(c2c(C)ccc(CC)c2)=O)CCC2(CCC2NC(=O)C2=CCCC2C)CC1 84814,C=CC1(C(=O)NCCCCCN(C(=O)Cc2csc(NC=O)n2)C)CCC1 84815,C1(N(C(=O)C=Cc2cc[nH]n2)C)CCCC(NC(=O)C=Cc2cnc[nH]2)C1 84816,C1(C)(C(=O)NC2CCC(C(=O)NC(CCC)c3ccco3)C2)CCC(=O)N1 84817,C1(C(=O)NC(C)C2CC2)CC2CC2N1C(C1(F)CC1)=O 84818,c1(CNC(C(C)N(C(C2C(CC)C2)=O)C)=O)ccnn1C 84819,c1(C(=O)NC2CC(NC(c3ncnc4sccc34)=O)C2)ccc2cc[nH]c2c1 84820,c1(C(C(=O)NCCC)N(CC)Cc2ccc(OC)cc2)ccc2c(c1)CC(C)O2 84821,c1(C(=O)NCCC(C)NC(C2CC(CCC)OCC2)=O)nc(O)nc(O)c1OC 84822,C1(C)(NC(C2C(C)OCC2)=O)CCCN(C(c2c[nH]cc2Br)=O)C1 84823,C(N=c1[nH]cncc1Br)C1OCC(CNC(C(C(CC)C)O)=O)C1 84824,Cc1ccc(C)c(C(=O)NCCN2CCN(C(C3(C)CCCCC3)=O)CC2)c1C 84825,N1(C(C2CCC(=O)NC2)=O)CCN(C(=O)Cc2cc(Cl)ccc2Cl)C(CCO)C1 84826,Cc1cc(C(=O)NC2CCC2NC(=O)C#CC(C)C)c(C)c(O)c1 84827,C1(NC(=O)CC2(O)CCOC2)CN(C(C2CCN(CCF)CC2)=O)CC12CCC2 84828,c1(C(=O)NCC(N(C(c2cc(C)ncn2)=O)C)C2CC2)ccc(Cl)cc1O 84829,c1(C(=O)NC(c2ccccc2)CCC)cncc(OCC)c1.C1(=O)C(CC)N1 84830,CC1CC(NC(C2CC2(C)C(F)F)=O)CCN1C(c1cc(F)cc(Cl)c1)=O 84831,C1(CNC(c2ccc(CSC)o2)=O)CCCCC1NC(=O)CCc1n[nH]c(=N)s1 84832,C1(NC(C(COC)(F)F)=O)COC2(C1)CN(C(=O)Cn1nc(C)oc1=O)C2 84833,c1(C(N2CCCC(CNC(CC(CCSC)O)=O)CC2)=O)cnc2sccc2c1 84834,C12(CNC(c3ccccc3F)=O)CC(C1)C(NC(C1CC13CCC3)=O)CO2 84835,C1(C(N2CCC(N(C(C3C(=C)C3)=O)CC)C2)=O)CC2(C1)CS(=O)(=O)C2 84836,CCC(C)C(C(=O)NC1CCN(C2CC2)C1)N(C)C(c1sncc1C)=O 84837,C1(NC(CCC=CC)=O)CN(C(C2(F)CCCC2)=O)CCC1CO 84838,N1(C(C(c2ccn(C)n2)(C)C)=O)CC(S(N)(=O)=O)C1 84839,N1(C(C2CC(NC(c3ncc(C)[n+]([O-])c3)=O)C2)=O)CC2CC3CC2C1C3 84840,C1(CNC(c2c(C(C)C)ncs2)=O)CN(CC(C)CS(C)(=O)=O)CCC1(F)F 84841,Cc1cn2c(n1)CC(C(=O)NCCCCNC(C1CCCS1(=O)=O)=O)CC2 84842,c1(OC)cc(OC2CC2)ccc1C(=O)NC1CC(CNC(=O)CC2CCCO2)C1 84843,C1(CCNC(CC2(C#N)CCC2)=O)CCCN(C(=O)COc2cccnc2)C1 84844,N(C1COc2ccccc21)C(=O)CCn1cc(Cn2cccc2)nn1 84845,c1(CC(N2CCC(=CCC)CC2)=O)ccc(-c2ccccc2)c(F)c1 84846,CCCC(C(=O)N(C)CC1CC(O)C1)NC(c1cn(C)cc1C)=O 84847,C1(OC)(CNC(c2nnnn2C2CCOC2)CCc2ccccc2)CCCCC1 84848,n1(CCC)cccc1C(=O)N(CC)Cc1ccn(CC)n1 84849,C=CCC(C)(CC)C(=O)N1CCC(N2CCN(C)CC2)C(C)C1 84850,C1(NCc2c(OC(C)C)cccc2)CC12CCNCC2.N1CCCCC1 84851,C1(S(C)(=O)=O)(C(=O)NC(CNC(C(CC)(C)OC)=O)C)CCOCC1 84852,c1(C(=O)NCCC(C)NC(=O)C(C)(F)F)cc(Br)cc2ccccc12 84853,N1(C(c2ccc(C)nc2)=O)CCN(C(C2(F)CCS(=O)(=O)C2)=O)CC1C1CCC1 84854,N1(C(c2cnn(-c3ccccc3)c2F)=O)CCCN(C(C2(F)CCOC2)=O)CC1 84855,C(=O)(C1=CCCC1C)NCCN(CCC)C(C1CC1c1cnc[nH]1)=O 84856,C1(N(C(CN(C(C=C(CC)CC)=O)C2CC2)=O)C)CCOCC1 84857,c1(C(=O)NCC2CCN(C(CSCC=C)=O)C2(C)C)ccc2c(C)noc2c1 84858,N1(C(C2CN(C(=O)NC)C2)=O)CC(C)(C)OC2(C1)CN(C(=O)Cc1cnoc1)C2 84859,C=CCCCCC(C(=O)NCCC)N(C1CCN(S(C)(=O)=O)CC1)C 84860,c1(CC(=O)NCC(C2CC2)NC(C(C)(O)C2CC2)=O)ccc2c(c1)OCCCO2 84861,N1(C(c2ncc(C(F)(F)F)[nH]2)C(=O)NC2CC2)CCc2[nH]c3ccc(F)cc3c2C1 84862,C1(OC)CC(CNC(=O)C(F)(F)CN2CCCC2)N(C(=O)C=C(C)C(F)F)C1 84863,NC(=O)C(O)CNC(=O)CC1CC(NC(=O)CC2CCCOC2)C1 84864,C=CC(C)(CC)NC(C1CC(N(C(=O)C(C)N2CC(C)C2)C)C1)=O 84865,c1(N(C)Cc2c(C)nco2)nc(=NCCCCCO)[nH]c2c1SCC2 84866,C(C(CC(F)(F)F)NC(C1(c2cc[nH]n2)CCC1)=O)NC(=O)Cc1cn[nH]c1 84867,C(C)(CC(C)NC(c1cc(F)n[nH]1)=O)NC(C=C(C)C(F)F)=O 84868,c1(C(=O)NCC(C(C)(C)C)NC(c2cnn(C)n2)=O)cc2n(n1)CC1(CC1)C2 84869,C(=O)(C#CC1CCOCC1)N1C(C(N2CC(C=C)C2)=O)CN(C)CC1 84870,C1(OC)CN(C(c2ccc(O)nn2)=O)C(C)(CNC(c2ccnc(S)c2)=O)C1 84871,C(=O)(C1=CCN(C(=O)CC23CCCC2C3)CC1)NCCN(C(CC)C)C 84872,c1(OC)cnc(F)c(C(=O)NC2CCC(NC(c3cccc(CO)n3)=O)CC2)c1 84873,N1(C(C=CCCC)=O)CCOC2(CCN(c3nc(O)c4ccccc4n3)C2)C1 84874,N1(C(C2C(C)OCC2)=O)CCC(C2CCN(C(c3cccnc3N)=O)CC2)CC1 84875,c1(C(=O)NC2C(C)N(C(c3ccns3)=O)CC2)cc2c(F)ccc(Cl)c2[nH]1 84876,C1(NC(c2cnc(C)nc2)=O)C(C)(C)C(NC(=O)CC2CC2C2CC2)C1(C)C 84877,c1(N(CC(=O)NCC2C(NC(CSCC)=O)CC2)C)c(Cl)cccc1[N+](=O)[O-] 84878,C1(CNC(c2scc(OC)c2)=O)COC(C)(C)CN1C(C1CCCO1)=O 84879,c1(C(=O)NC2CC(CNC(c3c(Cl)nc(OC)s3)=O)C2)cnc(O)cc1C 84880,N1(C(CC2N(C(c3ccc(C(N)=O)[nH]3)=O)CC2)=O)CCSC2CCC12 84881,CCCCC(C(=O)NCCCF)NC(=O)CCOC1CC1 84882,C(CC(C)(C)C(=O)N1CCN(C(=O)CCCc2ccc(OC)cc2)C(C)C1)OC 84883,c1(C(C)(C)C)cnc(CNc2nccn2CC(F)(F)F)o1 84884,C1(C(=O)NC2CCC(NC(c3cccc(Cl)c3Cl)=O)C2)CCC2CC1CO2 84885,N1(C(c2[nH]cc(C(C)=O)c2)=O)CCC(C2CCCN2C(C2CC3CC2C3)=O)CC1 84886,CC1(C)C(C(=O)NCC(C)(C2CC2)NC(c2cc(F)cc(F)c2)=O)CCS1(=O)=O 84887,C1(C(N(CC(C2CCC2)OC)C)=O)CNC(=O)CN1C(c1cc(C)ccc1C)=O 84888,Cc1cc(C(=O)NC2CC2CNC(=O)Cn2nc(C(F)(F)F)cc2C)cc(C)c1 84889,C1(C)(CC)CCC(CS(=O)(=O)NC(c2ccsc2Br)=O)O1 84890,C1(NC(Cc2c(C)non2)=O)CCCC2CN(C(c3cn(C)nn3)=O)CC12 84891,C1(C(=O)NC(C2CN(C(=O)CCCn3cccn3)C2)C)CCc2cnn(C)c2C1 84892,Cc1cc([N+](=O)[O-])cc(C(=O)NCC2CCN(C(=O)C#CC3CC3)C2)c1Cl 84893,C#Cc1ccc(F)c(C(N2CC(C)C(NC(=O)CC3CCSC3)C(C)C2)=O)c1 84894,c1(OC)cccc(CC(=O)N(C2CC(O)C2)CC2CCNC2)c1Cl 84895,C1(C(C(N2CC(OCCNC(CNC(CC(C)C)=O)=O)C2)=O)F)CCCC(=O)N1 84896,n1(CC)cc(C(=O)C(=O)NCC(C)(C)OCCNC(C2(C)CCCS2)=O)cn1 84897,C1(OCc2cn(C3(C(C)=O)CC3)nn2)CCN(c2ccc(Br)cc2)C1=O 84898,C1(C#N)(C(N2C(CNC(C3CC(CCC)OCC3)=O)CC2)=O)CCCCC1 84899,c1(C(=O)NC2(C(C)(C)O)CN(C(C3C(C)(CC)C3)=O)C2)nn(C)nc1C(=O)OC 84900,CCC(CC(=O)NCC1(C(=O)Nc2cccc(O)c2)CC=CC1)SC 84901,N1(C(C2(C)COC2)=O)CCOCC(F)(CNC(c2cn(C3CCC3O)nn2)=O)C1 84902,C1(CC)CC(N=c2[nH]c(=NC(CF)c3ccc(C)cc3)[nH]c3c2COCC3)C1 84903,C(CSC)(C(=O)N(C)CC1(O)CN(C(=O)C(C2CC(F)(F)C2)O)C1)OC 84904,N1(C(C(C)N(C(C)=O)C)=O)CCSCC1C(=O)NC(c1ccncn1)C 84905,C(=O)(CC1=NNC(=O)C1)N1CC(C(N)=O)(CNC(c2ccc(OCC)cn2)=O)C1 84906,N1(C(CCNC(C)=O)=O)C(C(=O)NCc2ccco2)C2CC(O)C1C2 84907,C(CCC)(CCCNC(=O)CCc1ncc[nH]1)NC(C(CC=C)NC(C)=O)=O 84908,c1(C(=O)NC(CC)CN(C(=O)CCC(C)C)C)cccc(F)c1C#N 84909,N1(c2snc(C)c2C#N)CCC2(NC(=O)CCCN3CCCC3)CCCCCC12 84910,c1(-c2cc(C(=O)OC(CC)C)n[nH]2)c(C)[nH]c2ccccc12.C12CSCN1C2=O 84911,N1(Cc2cc(OC)ncc2Br)CC2CCN(C(c3nc(C)cs3)=O)C2C1 84912,c1(C(CC)C(=O)N(CCC2(O)CN(C(C)=O)C2)CC)cc(C(F)(F)F)ccc1F 84913,n1(CC)cnc(C(=O)NCCCNC(=O)CNC(=O)NC2CC2)n1 84914,c1(C(=O)NCC(C)NC(c2oc(Br)nc2C(F)F)=O)cn2ccccc2n1 84915,N1(C(CCSCCCC)=O)CCC2(C1)CN(C(C1(C)CCN(C)CC1)=O)CCO2 84916,N1(C(C(C)c2cc[nH]n2)=O)CC2CCC(NC(=O)C3=CCN(C)C3)(C2)C1 84917,C1(C(=O)NC2CCN(c3ccncc3)CC2)COCCN(Cc2ccc(Br)o2)C1 84918,C1(NC(C(CC)c2ccccc2)=O)CCC(NC(=O)C(C)(C2CC2)OC)CC1 84919,c1(CCCC)nc(C(=O)NCC2C(CNC(=O)CC(=O)N(C)C)C2(F)F)cs1 84920,C1(C(=O)OC)CCN(C(=O)C(=O)NCC23CCCN(CC2)C3)C2(CC2)C1 84921,C1(CC(=O)N(C(C(N2CCC(COCC)C2)=O)C2CC2)C)CCN(C)CC1 84922,N1(C(CN(C(CCc2c(C)noc2)=O)C2CC2)=O)CCCC1(C)CC(C)C 84923,c1(C(N(CCNC(c2c[nH]nc2Br)=O)CC)=O)nccc(OC)c1N 84924,N1(C(c2ccc(C#C)cc2C)=O)CCC(C2CCN(C(=O)Cc3cnc[nH]3)C2)C1 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84942,CCC(C(=O)OCCNC1(C)CC1)n1ccnc1.C12(CC1)C(C)(C)N2 84943,Cc1sc(N)c(C(=O)NCC2CCCC2NC(c2cnn(C)c2C(F)F)=O)c1C 84944,N1(C(c2c(C3CCC3)cnn2C)=O)CC2(CCCN(C(C3(NC(N)=O)CC3)=O)C2)C1 84945,N1(C(C(C2CCOCC2)OCC)=O)CCN(C(c2ccoc2)=O)C2COCC12 84946,N1(C(CC)=O)CCCC(C2(NC(=O)CCCCCF)CC2)C1 84947,Cc1n[nH]cc1CNC(=O)C=CCC1(NC(=O)CCn2ccnc2)CCC1 84948,C12(CNC(CC=CCC)=O)CC1CN(C(C13CC(c4ccccc4)C1C3)=O)C2 84949,c1(OC)ccccc1C(C(C)(C)C)NC(c1ccc(N2CCCC2)cc1)=O 84950,N1(C(c2cc(C)n(CC)c2C)=O)CCC(N(C(=O)CCCOC)C)C2(CC2)C1 84951,c1(C(N2C(CNC(C(C)CN(C)C)=O)CC3(CC3)C2)=O)cc2cc(N)ccc2[nH]1 84952,c1(NC2C(NC(=O)CCNC(=O)CC(F)(F)Cl)CCCC2)ccc2occc2c1 84953,Nc1ccc(Cl)c(C(=O)NCC2CC(NC(=O)C3=CCCOC3)C23CCC3)c1 84954,N1(C(c2n(CCC)ncc2)C(=O)NC2CC2)CCCC(O)C1 84955,CC1(C)NC(=O)N(CCC(=O)NC2CCN(C(C3C=CCC3)=O)C2)C1=O 84956,S1(=O)(=O)c2cc(ccc2OC)N1.C1(C(CC)CC)CN(C(=O)OC)CCO1 84957,c1(-c2nc(C)sc2)cccc(C(N2CC3(NC(C4COC4)=O)CC2C3)=O)c1 84958,N1(C(C(CO)N(C)C)=O)C2CC=C(C(=O)NC3CCC4(CCCC4)C3)C1CC2 84959,C1(C(N2C(CC(=O)NC)CC2)=O)CN(C(c2cc(O)ccc2C)=O)C(C)(C)C1 84960,C(N=c1cc(C)nc(N2CC(C3CC3)OC(C)C2)[nH]1)C1(CCOCC)CCC1 84961,c1(CN(C(=O)C(F)(F)c2nccs2)CCNC(CNC=O)=O)ccc(F)cc1F 84962,N1(C(CCOC)=O)CCN(C(C23CC4CC2C3C4)=O)C2CC12.c12csc(n1)C2 84963,CCN=C(NCC1CCCC1OC)NCC(C1CCN(C(=O)NC)CC1)(C)C 84964,C1(NC(CC(C)CF)=O)CCC2(CCN(C(c3cc[nH]c4nccc3-4)=O)CC2)C1 84965,C1(N(C(CSCC#C)=O)C)CN(C(c2c[nH]nc2C)=O)CC1F 84966,c1(NC(CC)(CCCl)c2nnnn2C(C)C)cc(Br)ccc1OC 84967,C1(CC)C(=O)NCCN1C(C1CCCN1C(=O)CCCc1cnn[nH]1)=O 84968,CCCC(C)C(=O)NC1CCCC1CNC(c1sc(=N)[nH]c1C1CC1)=O 84969,c1(N2CCC(c3c(CNC(C4(SC)CC4)=O)c[nH]n3)C2)ncnc2onc(C)c12 84970,C1(NC(c2c(Br)cn(C)n2)=O)CN(C(c2ocnc2C2CC2)=O)CCC1F 84971,C1(CNC(C(C)(C)c2cnsc2)=O)COCCN1C(=O)C=Cc1cccs1 84972,S(=O)(=O)(c1cccc2c1OCCO2)Nc1ccc2c(c1)N(C)CC2 84973,C=CC1OCCCC1C(=O)NCC1CN(C(=O)CSCC(N)=O)CCC1C 84974,C(C(C(=O)NCC1(O)CC(N(C)C)C1)NC(=O)C(O)C1CCCC1)OC(C)C 84975,C(C(C)C(=O)NC(CSC)C(=O)NCCCNC(C)=O)OCC 84976,Cn1ncc(C(N2CC=C(CNC(C3CC34CCOCC4)=O)CC2)=O)c1C#N 84977,C1(C(C(=O)NC2CCCN(CC(F)(F)Cl)C2C)NC)CCC(F)(F)CC1 84978,N1(C(=O)OCCC=C)CC2CCC1(C(=O)NCCC(F)(F)F)CC2 84979,Cc1c(O)nnc(N2CCCC(N3CCCCC3=O)C2)c1C 84980,N1(C(CN(C(=O)NC)C2CC2)=O)CCN(C(c2nn(C)cc2C(F)(F)F)=O)C2CC12 84981,c1(CC(N2CC=CC(NC(c3cc(C(C)C)sn3)=O)C2)=O)ccc(F)cc1F 84982,C1(C(=O)NC(C)CCCCNC(=O)C(C)(C)c2cscc2Cl)CC2CC1CC2O 84983,N1(C(C=C(CC)CC)=O)CCCCC12CC(NC(=O)C(C)Cc1ccncc1)C2 84984,N1(C(COCCC)=O)CC2CN(C(=O)C(c3ccccc3F)(C)F)CC2(C)C1 84985,c1(N2CCC(CCOC)(NC(=O)C(C)SC)CC2)ccc([N+](=O)[O-])cc1C#N 84986,N1(C(CCc2onc(SC)n2)=O)CCC2(NC(c3ccnc(C)c3)=O)CCCC12 84987,C1(C(=O)NC(CCCN(C(=O)C2=COCC2)C)c2ccccc2)CC2(C1)CC21CC1 84988,C(=O)(C#CC1(C)CCCO1)NC1C(NC(Cc2n(C(C)C)cnn2)=O)CCCC1 84989,N1(C(C(CNC(=O)Cc2c(C)noc2C)OC)=O)CCCC(C2(C)CC2)C1 84990,c1(OCC=C)ccc(C(=O)NC23CC(CNC(=O)C(F)=C4CCCC4)(C2)C3)cc1 84991,C1(CNC(CSC(C)C)=O)CCCCCN1C(C1CC1c1cnc[nH]1)=O 84992,Cc1ccnn1CC(=O)NCC(O)C(=O)NC(c1cn[nH]c1)C 84993,N1(C(CC(C(C)C)O)=O)CCN(C(c2ccn(C(C)(C)C)n2)=O)C(C)C1C 84994,CCC(C#N)C(=O)N(C1CCN(C(C2CCN(C(C)C)CC2)=O)C1)CC 84995,c1(C(N2CC(CNC(c3c(C)nsc3)=O)C2)=O)ccc(C2CC2)nc1O 84996,C1(CC(N2CCCC(NC(c3n[nH]cc3F)=O)C2)=O)NC(=O)CNC1=O 84997,C1(C(=O)NCCn2ncc(CC)c2)CN(C)CCN1C(C1CCCC(=O)N1)=O 84998,C1(CNC(CC=CC=C)=O)CCC2CN(C(c3ncc(C(F)F)s3)=O)CCC2C1 84999,C1(NC(C2C(CC)CCC2)=O)CCC(NC(c2cc(OC)c(Cl)s2)=O)CC1 85000,S(=O)(=O)(c1cccc(F)c1)NCCNC(c1cn(CCOC)nc1)=O 85001,N1(C(=O)CCCCCn2cc(C3CCCOC3)nn2)CCCC2(CCNC2)C1 85002,N1(C(c2cccc(OC)c2OC)=O)CCCCC12CN(C(c1ccoc1C)=O)C2 85003,C1(CNC(C(CSC)O)=O)CN(C(c2ccc(F)c(F)c2)=O)CC(C)(C)C1 85004,Cn1ccc(C(=O)NC2(C(=O)NC3CC(CO)C34CCC4)CCC2)cc1=O 85005,N1(Cc2cn(CCC)nc2)CCC2(CN(C(=O)C3=COCCC3)C2)C1 85006,C1(O)(CNC(c2occc2C2CC2)=O)CN(C(c2cc(C3CC3)cs2)=O)C1 85007,CCC(CC(=O)NC1(CC(=O)NCC2CC[Si](C)(C)C2)CC1)C(C)C 85008,Cc1cccc(CC(=O)NC2CCC(CNC(C3(C)CSC3)=O)C2)c1 85009,Cc1ccc(C)n1CC(=O)NC1C=CC(C(=O)NCC2CCC(C)C2)C1 85010,c1(OC)cc(O)c(CN2CCCC2CN2CCCC2c2c(F)cccc2Cl)cc1O 85011,C1(C(N2CC(N(C(C(CC)CC)=O)C)C(C)CC2)=O)CCCC2(CCC2)C1 85012,c1(C(=O)NCCN(C(CC(=C)C)=O)C2CCCC2)csc(C)c1C1CC1 85013,CC(C)(C#N)CCCCNC(=O)Cn1cc(C2CCCCCC2)nn1 85014,C(=O)(C1COc2ccccc21)NC1CCN(C(c2n[nH]c(C)c2C)=O)CC1C 85015,C(=O)(CC1OC(=O)c2ccccc21)NCCCCNC(CCCC(CCC)C)=O 85016,C1(NC(C2(F)CCN(C(C3N(C)C(=O)OC3)=O)CC2)=O)CC2CC1CC21CC1 85017,c1(C(=O)NC(CNC(C(CC)=CC)=O)CC)nccc(C)c1N 85018,N1(C(c2nn(C)c(OC(F)F)c2)=O)CC(NC(=O)CCCn2ccnc2)CC(O)C1 85019,C(C(=O)NCC1COC(CNc2ccc(C(F)F)cn2)C1)(C(C)C)N(CC)CC 85020,c1(C(N2C(C)CC(NC(=O)C(C)(Cl)Cl)CC2)=O)ccc2n[nH]cc2n1 85021,O=C(CC(F)(F)F)N1CCC(N2CCN(C(c3c[nH]ccc3=O)=O)CC2)C1 85022,C(=O)(C1=NOC2(CCOC2)C1)NCC1(OC)CN(C(=O)C(F)n2cccn2)C1 85023,N1(C(c2ccc(SC)s2)=O)CCC(O)C(NC(C2(C)CCCCO2)=O)C1 85024,C1(NC(CCOCCCOC)=O)CN(C(=O)C=CSC)C(C)(COC)C1 85025,N1(C(C2C(C)OCC2)=O)CCC(C(C)(C)C)(CNC(=O)COC(F)(F)F)C1 85026,N1(C(c2ncccc2Cl)=O)CCC2(CCCC2Nc2nccc(CO)n2)CC1 85027,c1(C(=O)NC(CNC(C2(C(=O)OCC)CC2)=O)C)ccc(N)cc1C 85028,C1(CNC(C(C)(C)CO)=O)COCC2(CCN(C(=O)CC3=CCCCC3)C2)O1 85029,CC1CN(C(C2CCC(n3cc(-c4c[nH]nc4F)nn3)C2)=O)CC1C(N)=O 85030,C1(C)(CC)C=C(C(=O)NC2CC(NC(=O)C(C#N)Oc3ccccc3)C2)C1 85031,N1(C(C)=O)CC(C)CN(C(=O)NC2(c3ncccc3F)CCC2)c2ccccc21 85032,N1(C(Cn2cc(C(C)O)nn2)=O)CC2(C1)SCCC2NC(=O)C1=CCCCO1 85033,N1(C(c2c(C)ncnc2O)=O)CC(O)(C2(CNC(=O)C3=CCCC3)CC2)C1 85034,C1(CCN)CC2CCC(C1)N2N1CC(c2onc(C)n2)C1.c1(C=O)ccnc(Cl)c1F 85035,C12(NC(COCCCCC)=O)CC(C(=O)NCC3(F)CC3)(C1)C2 85036,C1(O)(CN(C(c2ncn(CC)c2)=O)C)CCN(C(c2ccoc2Cl)=O)C1 85037,C=C(C)CC(C(=O)NC1CCN(C(=O)CN(C)C2CC2)C(C)C1)OC 85038,C12(CNC(CNc3[nH]c(=N)sc3)=O)CNCCN1CCOC2 85039,C(=O)(CS(=O)(=O)CCO)NCC(CCNC(c1cc(CC)ncc1)=O)O 85040,N1(C(C)=O)CCCCC1C(=O)NCC1(O)CCN(C(c2cn(C3CC3)cn2)=O)C1 85041,C1(OC)(OC)CC2(CN(CC3CC(C4CC4)=NO3)C2C(C)C)C1 85042,N1(C(C(CC=CCC)C)=O)CC(C)N(C(=O)CSC(F)(F)F)CC1C 85043,Cn1ccn2ncc(C(=O)NC34CCCC3N(C(c3ccncn3)=O)CC4)c12 85044,N1(C(C2CCC(=O)N2)=O)CCC(CNC(c2cnc3n2CCC3)=O)C(F)(F)CC1 85045,C=C(C)CCCC(=O)NCC(CC(=O)N1CCCC1(CO)CO)OC 85046,N1(C(c2c(CC)scn2)=O)CCC2(CCCN(C(c3nncs3)=O)C2)C1 85047,c1(NC(=O)C=CC(F)(F)F)cncc(CO)c1.C12CCC(C1)NC2=O 85048,c1(C(N(C(CNC(C=CSC)=O)C2CC2)C)=O)cccc(NC(C)C)c1 85049,C1(CNC(CCSCCNC(=O)OC(C)(C)C)=O)CCC(=O)NC1 85050,CC1CCCC(N(C(=O)Cc2csc(NC3CN(c4nncs4)C3)n2)C)C1 85051,C(c1ccncc1)=C(C)C(=O)NCC1CCCCC1NC(C1CCC2CC12)=O 85052,N1(C(CC2N(C(C=CC(=O)OCCCC)=O)CCOC2)=O)CCCC(O)(CC)C1 85053,n1(CC(=O)NC2C=CCN(C(=O)C(=O)NC3CC3)C2)nc2c(n1)CCCC2 85054,C1(NC(CC2C(C(=O)OCC)C2)=O)CCCC1NC(c1c[nH]nc1OC)=O 85055,c1(OC)ccc(CC(N2CC(O)(C(C)NC(C3(C4CCC4)CC3)=O)C2)=O)c(F)c1 85056,C1(C(=O)NCC2(CNC(C(C(C)C)C3CCC3)=O)CCC2)Cc2nccn2C1 85057,c1(C(=O)NCCC(C)N(C(CC(CC)C)=O)C)cc[nH]c(=N)c1Cl 85058,c1(OC)nc(C)ccc1C(N1CC(NC(c2sc(CC3CC3)nc2C)=O)C1)=O 85059,N1(C(c2c(CC)nc(C)[nH]2)=O)CCC(NC(=O)C(O)C(C)(C)C)C12CCCC2 85060,c1(OC)ccc(F)cc1CCC(N1CC(NC(=O)Cc2cncn2C)C(C)C1)=O 85061,C1(C2CC2)(C(=O)NCC(C)(C)OCCNC(C2C3CCCOC23)=O)CC=CC1 85062,C12(CNC(=NC)NCc3nocc3C(C)(C)C)CCC(OCC)(CC1)CC2 85063,C1(C(C)C)(C(=O)NCCOCCCO)CCN(C(c2cncc(OC)n2)=O)C1 85064,N1(C(C2CCN(C)S2(=O)=O)=O)CC2(CCN(C(=O)CC3(C)CC3)CC2)C1 85065,C(=O)(C(C)CC(F)(F)F)NC1CCCCN(C(C2CC(OC)C(OC)C2)=O)C1 85066,CCCC(CNC(C1CC1OC(C)=O)=O)C(=O)NCC(C)(CC)CO 85067,N1(C(C(=C(C)C2CC2)F)=O)CC(CCNC(C2(C)CCN(C)CC2)=O)OC(C)C1 85068,N1(C(C2C3CN(C(CCOCCOC)=O)CC32)=O)CCC(C(N)=O)C(O)C1 85069,C1(C(=O)NCCOC2(C)CCC2)(CNC(CCCSCC=C)=O)CC2(CC2)C1 85070,C(=O)(C(Cl)=CCl)NC(C1CCOC1)CNC(CC1CN(C)C1)=O 85071,C1(NC(c2nc(CC)oc2)=O)CC(CNC(c2ncc(F)cn2)=O)C1(C)C 85072,C=C(C)CC(C(=O)NC1CN(C(=O)CSC2CC2)CC1CO)NC(C)=O 85073,Cc1ncc(C#N)c(N(C23CCC(N)(CC2)C3)C(c2ccc(O)c(O)c2Cl)=O)n1 85074,C1(NC(c2ccc(C(C)O)cc2)=O)CN(C(c2ccc(C#N)nc2)=O)CC1C#N 85075,C1(NC(C(c2cc(C)sc2)(F)F)=O)CCN(C(=O)C(C)C#N)C(C)C1 85076,Cc1nc(C(N2CCC(C(C)NC(C3(C)SCCCS3)=O)C2)=O)cn1C(F)F 85077,c1(OC)c(C(=O)NC2CC(CNC(=O)CN3CC=CC3)CC2O)ccnc1F 85078,C(=O)(C1=Cc2ccccc2C1)NC(C(=O)NCC(C)SC)c1cccs1 85079,C(=O)(C1=CCN(C(C2C3CCCOC23)=O)CC1)NCCc1ccn(CC)n1 85080,CCC(C(=O)NCC1(NC(=O)C(C)(C)C)CN(C(=O)CCCCOC)C1)N(C)C 85081,Oc1cc(C(C2CC2CO)NC(CC2CCOC2)CO)cc(F)c1 85082,N1(C(c2scnc2Cl)=O)CCCN(C(=O)C(O)c2ccco2)CC1 85083,N1(C(C(C2CC2)OC)=O)CC2CCC1C(CNC(=O)CC1CCCC(C)C1)C2 85084,CC(C(=O)N(CCC(=O)NCCC1CC(=O)N(C)C1)CCCO)C(F)F 85085,N1(C(CC(C(C)OC)NC(C23CCC(CC2=O)C3)=O)=O)CCC2(CC1)CSC2 85086,CC1CCn2cc(C(=O)N(C3CC4CCC(C3)N4c3nccnc3F)C)nc2C1 85087,CC1CN(C(=O)C(CO)NC(=O)C(=O)NC2CC2)C(C)C1C 85088,C(C1CCN(C(C2CCCCS2(=O)=O)=O)CC1)=CC(N1CC(C2(C)CC2)OCC1)=O 85089,Cc1cc(C(N2CCN(C(=O)CC(=O)N(C)C)C(CO)C2)=O)ncc1Cl 85090,N1(C(C(CC)Oc2ccccc2C)=O)CCC2(CCC2NC(=O)CC#N)CC1 85091,Cc1cc(C(F)(F)F)ccc1COC(C1CN(C)C(=O)N1)=O 85092,CCC(F)(F)CC(=O)N1CCC(C)(C)C1CC(=O)NCCN1CCOCC1 85093,C1(NC(C=C(CCC)C)=O)CC2(CCN(C(c3cncc(OC)n3)=O)C2)C1 85094,C1(CCC)(NC(=O)CCc2cnc(C)s2)CCN(C(=O)CC2CCOC2)CC1 85095,c1(C(=O)OC)cnc(Cl)cc1NCC1CC(C)CN1CCO 85096,c1(CC)noc(C(N2CCOC(CCNC(C3(CC(=O)OC)CC3)=O)C2)=O)c1C 85097,c1(CCC(=O)NC(C(C)NC(CNC(C)=O)=O)C)ccc(OC(C)C)cc1 85098,N1(CCc2cn(OC)nn2)CCN(C(C2CSCN2C(C)=O)=O)CC1.C1CCOC1 85099,c1(C(N2CCC(CCNC(C(C3CC3)OC)=O)C2)=O)ccc(C(C)C)cc1F 85100,C1(C(N2CC(c3nc(C)on3)C2)=O)CC(C)CN1C(=O)Cc1cnc(C)s1 85101,CC1OCCOC1CC1CCN(C(=O)Nc2cnn(N3CCOCC3=O)c2)CC1 85102,Cc1cc(C(=O)NC2CCN(C(=O)Cc3nc(Cl)cs3)C2)cc(F)c1 85103,C(=O)(C(CO)N(C)C)NC(CC1CN(C(C(C)OC2CCOC2)=O)C1)C 85104,N1(C(CN2CCCC(CC)C2)=O)CC2C3CCC(C2C1)N(C(C1CC1C)=O)C3 85105,C(=O)(C(C)(F)C(=O)NCC1(F)CC(NC(c2ncc(Cl)cc2Cl)=O)C1)OCC 85106,N1(C(C(C2CCC2)OC)=O)CC2CC(NC(C3(F)CCCCC3)=O)C1C2 85107,N1(C(CCCN(C(C)=O)C)=O)CC(CC(=O)OC(C)(C)C)CC12CCC2 85108,c1(OC)ccc(NC(=O)C(C(C)C)OC(c2cc(Cl)cs2)=O)cc1 85109,C12(NC(c3cccc[n+]3[O-])=O)CCN(C(=O)C=CCF)CCC1C2 85110,C1(C)(C(=O)NCC(COC)O)CCN(C(c2cccnc2O)=O)C1 85111,C1(C)(C(=O)NCCN(CC(C)C)CC)CN(C(c2c[nH]c(=NC)o2)=O)C(C)(C)C1 85112,c1(CC)nccnc1C(=O)NC1(C(=O)NC2CCOCC2C)CCOCC1 85113,Cc1cncc(C(=O)NC(C)C(C)NC(c2scc(C)c2Br)=O)c1 85114,CC1CCC(C)(CNC2(c3nnnn3Cc3nnn(C)n3)COCC2C)CC1 85115,Cc1ccc2oc(C(N3CCN(C(C4CC=CCO4)=O)C4CCCC34)=O)cc2c1 85116,CC1CCN(C(=O)CCCc2ccc(Br)cc2)C(CNC(c2cn[nH]c2)=O)C1 85117,S(=O)(=O)(CCC(=O)NCCN(C)C(c1ccc(Cl)s1)=O)NCCNC(C)=O 85118,C(CCC(C)C(=O)N(CC(C)NC(=O)Cn1cnccc1=O)C)OC 85119,CC(CNC(=O)CCn1cncn1)CNC(C1CC(N2CCCC2)C1)=O 85120,Nc1cc(F)c(C(=O)NC(CNC(c2cnc(O)o2)=O)C2CCC2)cc1Cl 85121,c1(C(N2CC(NC(C=C(COC)C)=O)C(C3CC3)C2)=O)cc2c(cc1O)OCO2 85122,N1(C(C(c2ccc(Cl)c(Cl)c2)(C)C)=O)C2CCC1(CNC(C1CC=CC1)=O)CC2 85123,CC(CN=c1ccc2ncc[nH]c-2n1)NC(=O)C1CC1 85124,C12(NC(=O)C=Cc3cnc[nH]3)COCCC1CN(C(=O)CC13CC(C1)C3)C2 85125,N1(C(CCC=C)=O)CCC(C)N(C(=O)CC2CCOC(C)(C)C2)CC1 85126,C1(NC(C(C)N(C)C)=O)CCN(C(=O)CC2CC2(Cl)Cl)CCC1CO 85127,c1(OC)ncc(C)c(C(=O)NC(C)CNC(c2nc(C3CC3)cs2)=O)c1Cl 85128,c1(NC(=O)NC2CCCN(C(C(CN)O)=O)C2)cc(Cl)ccc1Cl 85129,C#CCC(C)C(=O)N1CCCC1CNC(c1ccc(-c2ccsc2)nc1)=O 85130,c1(NC(=O)NC(CCCCC)c2ccccc2)cc(F)ccc1NC(C)=O 85131,CCC(C)C(C)C(=O)NCc1ccccc1CNC(=O)Cn1cnnc1O 85132,N1(C(=O)CC2CSC2)CCN(C(c2cnccn2)=O)C(CC(F)F)C1 85133,c1(CNC(CC2N(C(C3C(CC)C3)=O)CC2)=O)nc(C)ns1 85134,C1(NC(CCc2cncc(C)c2)=O)CN(C(=O)C(C)c2cccs2)CC(F)(F)C1 85135,c1(OC2(C(=O)OC)CC2)cc(NC(=O)C(c2ccc(F)cc2)OC)cc(F)c1 85136,CC1CC(NC(C23CC(C(F)(F)F)(CO2)C3)=O)CCN1C(c1cncc(Cl)c1)=O 85137,C(=O)(C(C)(F)C(=O)OC)N(CC(CNC(c1c(CC)ccs1)=O)C)C 85138,C1(C(N2C3C(NC(CNC(CC)=O)=O)CC(C3)C2)=O)CC2(C1)NC(=O)NC2=O 85139,c1(C(=O)OC)sc(C(=O)NC2CN(C(C3CCC4CC34)=O)C2)cc1C 85140,C(=O)(C1Cc2ccccc21)NCC1CCN(C(c2c(C)noc2C)=O)C(=O)CO1 85141,c1(C(N(CCNC(C2CC2(Cl)Cl)=O)C2CC2)=O)cc(Cl)c(C2CC2)cc1F 85142,C1(C(N(C(CC)CC)CC(C)C)=O)COCCN(C(c2ccc(O)nc2C)=O)C1 85143,CC(C#N)CCC(=O)NC1CCCC1NC(C1(c2cccc(Cl)c2)CC1)=O 85144,N1(C(C2(F)CN(C(=O)C=CCN3CCCC3)C2)=O)CCOC2CCCC12 85145,C1(CC(=O)N(C(C)CC(=O)NCCCCOC(C)C)C)CCCNC1=O 85146,n1(C(COC)(C)C)cnc2c(N(CCF)Cc3cccc(Cl)c3Cl)ncnc12 85147,CC1(C)NC(=O)CCC1NC(=O)CC(C(F)(F)F)NC(c1ccncc1N)=O 85148,N1(C(c2cc(F)ccc2F)=O)CCC2CCCC(C1)N2c1ncc(F)cn1 85149,C1(C)(C(N2CCC(N(C(CC=C)=O)CC)CC2)=O)Cc2ccc(F)cc2C1 85150,N1(S(CC(C)C)(=O)=O)CC2(CC(CC(=O)NC(c3ccccc3Cl)C)C2)C1 85151,C1(C#N)(C(=O)NCCC(C)NC(c2n[nH]cc2C2CC2)=O)CC2(CCC2)C1 85152,c1(C(=O)NC2(C)CN(C(Cn3c(=O)ccc(C)n3)=O)C2)nc2ccccn2c1F 85153,CC(C)C(C(=O)NC(C)C(=O)NO)C(C)NC(c1c[nH][nH]c1=N)=O 85154,C(C(C)(CCC)OC)(c1nnnn1Cc1ccccc1)NCCCSCCCC 85155,c1(CNC(C2(CSC)CC2)=O)cc(C(=O)NCCC2CCCC23CC3)n(C)n1 85156,CCCCCC(C)CC(=O)NCC(C(C)(C)C)NC(c1ncc2[nH]ncc2n1)=O 85157,c1(OC)c(Cl)ccc(C(N2CCC(C3CC3)(NC(=O)CS(C)(=O)=O)C2)=O)c1N 85158,CC1(CN=c2ccnc[nH]2)CCCN(c2cc(C3CC3)ccn2)C1 85159,C(=O)(C(F)(F)C(O)C(C)C)N1CC2C(Nc3cc(OCC)nc(C)n3)C2C1 85160,C1(CNC(C(C)=CC)=O)CC2(CO1)CN(C(c1ccc(OC)c(Cl)c1OC)=O)C2 85161,c1(C(=O)Nc2ccc(NC(C(CC)OC)=O)cc2C)cc(C)cc(Br)c1F 85162,c1(C(N(CC(CC)NC(CC(CC)C2CCC2)=O)C)=O)ccc2ncncc2c1 85163,c1(COC)nc2n(n1)CCCC2NC(=O)NC(C1(n2ccnn2)CC1)C 85164,C1(C(N2CCC(C)(CNC(c3n(C)ncc3)=O)C2)=O)CCC(S(N)(=O)=O)CC1 85165,CCC(C)(C)C(C)CC(=O)NC1CCN(C(=O)CCc2nccn2C)C12CCC2 85166,C1(O)(CC)CCC(NC(=O)C(C)C(C)NC(=O)Cc2nonc2C)CC1 85167,C1(NC(c2c(COC)nn[nH]2)=O)CC2CN(C(C3CCSCC3)=O)CC2C1 85168,C(CC(C)(C)CC(=O)NC(C)(C)C=CC(=O)NC(C1CCCC1O)C)OC 85169,N1(C(C(CC)=CCCC)=O)CC2CC(C)N(C(=O)CC=Cc3ccccc3)C2C1 85170,c1(OC)cccc(C(N2CCN(C(=O)C(O)C(C)(C)C)CC2CC(F)F)=O)c1C 85171,C1(C(=O)NC(C2CCCC2)CNC(c2nc(Cl)cs2)=O)CCNC1=O 85172,C1(NC(c2c(C(C)C)n[nH]c2)=O)CC2CC1N(C(=O)CC(C)F)C2 85173,C(C(C)(C)C(=O)NCC(C)CN(C)C(C1CCCC(=O)C1)=O)NC(C)=O 85174,C(C(N=c1nc(CCOC)[nH]s1)C(C)C)N(C(C(C)(C)NC(=O)NCC=C)=O)C 85175,c1(C(=O)OC)ccc(CC(=O)NCC(F)CNC(c2nn(C)cc2Cl)=O)c(Cl)c1 85176,C1(NC(C(c2c(C)cccc2)C)=O)CC2CC1CN(C(c1ccsc1)=O)C2 85177,c1(C(N2CCC(CCNC(c3cc(CC)sn3)=O)CC2)=O)cn2ccsc2n1 85178,C1(NC(c2ccc(C)n2C)=O)CCCCN(C(C2(C(F)F)CC(=O)C2)=O)C1 85179,C1(NC(C)=O)CN(C(=O)Cn2cc(CNc3cccn3C)nn2)CC1C 85180,C1(=CC(=O)NCC(CNC(c2n(CC)ccn2)=O)(C)O)C2CC3CC(C2)CC1C3 85181,c1(C(=O)NCCCNC(C2CC2(F)Cl)=O)ccc(Br)nc1O 85182,C1(NCc2scc(C)c2)CCN(C(=O)C2CC(=C3CCC3)C2)O1 85183,N1(C(C2CC(C)=C(C)CC2)=O)CCC=C(C(=O)N2CCOCC(C)(O)C2)C1 85184,N1(C(C(=C)COC(C)C)=O)CCC2(CC=CCO2)CC1 85185,CC(C)CC(C(=O)N1CC(S(C)(=O)=O)C1)ONC(C1(C#N)CCCCC1)=O 85186,N1(c2snc(COC)n2)CCCCC(CNC(=O)CCN2CCOCC2)C1 85187,N1(C(C(=O)NC(C)C)=O)CCC2COC(CC(=O)N(C)C)C2C1 85188,C1(CNC(C=CCCC=C(C)C)=O)CN(C(C2CC3C=CC2C3)=O)CC12CCC2 85189,C1(CC(=O)NCC(C)N(C(=O)C(c2ccccc2Cl)O)C)OCCCC1(C)C 85190,c1(NC(C(CSC)O)=O)ccc(C)c(Cl)c1.C1CCC(=O)NC12CC2 85191,N1(C(C2(C)C(C)(C)C2)=O)CCC(C(N2CCC(CO)(CO)C2)=O)C(O)C1 85192,N1(C(CNC(CC)=O)=O)CCN(C(=O)CCc2cccc(OC)c2F)C2CC12 85193,O=C(C1=CCCS1)NCC(C1CCN(C(C2(F)CCOC2)=O)CC1)F 85194,c1(NC(C)CCOC)ccc(S(=O)(=O)NCC(c2ccco2)O)cc1Br 85195,CC(CC(=O)N1CCC(CN(C(=O)C=Cc2ncc[nH]2)C)C1)P(C)(C)=O 85196,c1(OC)c(C(=O)NC(C)CN(C(=O)C#CC2CCCCO2)C)oc2ccccc12 85197,N1(C(C2CC(SC)C2)=O)CCn2c(CNC(=O)C(C)=C3CC3)nnc2C1 85198,c1(C(N2CCC(C(C)NC(C=CCOC)=O)C2)=O)ccc([N+](=O)[O-])cc1 85199,c1(N2CC=CC(NC(C(C)CC(C)(C)C)=O)C2)ncc([N+](=O)[O-])cc1F 85200,C1(C(=O)NC(CCNC(Cn2ccc(C)n2)=O)(C)C)CC2(CCOCC2)CO1 85201,c1(C(N(C2(C)CCS(=O)(=O)C2)C(C)C)=O)c(NC(=O)OC(C)(C)C)cncc1F 85202,C1(CC(=O)NCC(N(C)C)C2CC2)CCN(C(C2(Cl)CC2(F)F)=O)C1 85203,C(=O)(C1CCCc2nc[nH]c21)NCCCN(C(C1CC(C)C1)=O)CCO 85204,c1(SCCCC(=O)NCC(C)(CC)NC(C(C=C)O)=O)nc2ccccc2[nH]1 85205,c1(CC)noc(C)c1C(=O)NCC(CC(=O)N1CCC(O)(CN(C)C)C1)OC 85206,C1(NC(CC(OCC)OCC)=O)CC12CCN(C(c1sc(C)cc1C)=O)C2 85207,c1(C(=O)NC2(COC)CN(C(C3(C)CC4CCC3C4)=O)C2)cn2nc(C)sc2n1 85208,CCC(C)C(C(=O)N1CC(C)(C)CC1CC(=O)NC1CC(CCF)C1)N(C)C 85209,C1(NC(C(CC)CC(F)F)=O)CN(C(c2ccccc2)=O)C2CCCCC12 85210,C1(N(C)C)CCC(C(=O)COC(c2c[nH]nc2-c2ccoc2)=O)CC1 85211,C1(CC=C)(NC(=O)CSC(C)(C)C)CCCN(C(c2cc(Br)c[nH]2)=O)C1 85212,c1(C(=O)Nc2ccsc2C(N2CCCC(F)C2)=O)cc(O)cc(Cl)c1 85213,C1(NC(c2cnc[nH]2)=O)CN(C(=O)Cc2cnccc2Cl)CC12CCC2 85214,C1(NC(C(C)(C)C(F)(F)F)=O)CN(C(C2CCC(C)(C)O2)=O)CC12CCOCC2 85215,Cc1cncc(CC(=O)NCC=CC(=O)NCCCn2cncn2)c1 85216,C(=O)(C(F)CC(C)C)N(CCN(C(C1CCN(C(CCC)=O)CC1)=O)C(C)C)C 85217,N1(C(c2cc(CC)no2)=O)CCCCCC1CNC(=O)COC1CCN(C)CC1 85218,C(C)(C)(CC(=O)N1CCCCC1C(C)NC(=O)C=Cc1scnc1C)OC 85219,C1(C2CCCN(C(=O)CC3CCC4CC4C3)C2)(NC(C2(C)CC(C)C2)=O)CC1 85220,c1(C(N2CC3CN(C(Cc4nnc(C)o4)=O)CC32)=O)cc2cc[nH]c2cc1Cl 85221,CC(C)(O)C(C)(C)NC(C1CCC(CNC(c2ccn(CCF)n2)=O)O1)=O 85222,C(CCC(=O)NCCCC1CCCN1C(=O)C(CC)OCC)N(CCCC)CC 85223,c1(NCC=CCNC(C(c2cccc(Cl)c2)CC)=O)cc(C)ccc1[N+](=O)[O-] 85224,c1(NCC2N(C(C3CCC(C)(C)O3)=O)CCCC2)ncc([N+](=O)[O-])c(=N)[nH]1 85225,c1(CCC(=O)NCC2C(NC(Cn3c(C)ccn3)=O)CC2)ccc(O)nn1 85226,C1(COC)(NC(=O)Cc2nnc(S)n2C)CCN(C(c2c(O)noc2C)=O)CC1 85227,Cn1nnnc1SCCC(=O)NCC1CC(F)(CNC(=O)Cc2cnoc2)C1 85228,C1(NC(C2(OC)CCN(C(c3nocc3C)=O)C2)=O)CN2CCC1CC2 85229,c1(N2CCC(CC=C)C2)nc(=NCCC(C)(C)OC)[nH]c2c1SCC2 85230,C1(C(=O)NCC(COC)(C)CO)CCCN(C(C2CC3CCCC3C2)=O)CC1 85231,C=CCC(C)(CC)C(=O)N1CCN(C(c2ccc(OC)c(N)n2)=O)C(CCO)C1 85232,Cc1ccc([N+](=O)[O-])cc1-c1csc(C(=O)Nc2ccc(I)nc2)c1 85233,N1(C(c2cc(CCC)on2)=O)CCC(NC(=O)CC2CC2(C)C)C(O)C1 85234,Cc1ncc2cc(C(N3CCC4(CCN(C(C5(O)CCC5)=O)C4)C3)=O)ccn12 85235,CN1CC(C(=O)NCC(N)=O)C1.C12(CC1)CC(=O)NC2 85236,c1(C(=O)NC23C(CN(C(CC4ON=C(C)C4)=O)C2)CC3)csc2c1CCC(C)C2 85237,N1(C(C(=O)NC2CC(NC(c3cc(C)no3)=O)C2)C)CCCCCC1 85238,C12(C(=O)NCc3c(C)nn(C)c3)CCCC1CN(C(C1CCCCS1)=O)C2 85239,O=Cc1ccnc(N2CCN(C(=O)NCCCOC(F)F)CC2)c1 85240,N1(C(CCC(N)=O)=O)CCC2(NC(c3cc4n(n3)CCCO4)=O)CCCCCC12 85241,c1(SCC)cncc(C(=O)NC(C)CNC(=O)CNC(c2ccsc2)=O)n1 85242,c1(C(=O)NCC(CC)NC(=O)C=CC2CCC2)cc2cc(C)cc(C)c2[nH]1 85243,CCCCCCC(F)C(=O)N(C1CCN(C(c2cccc(Cl)c2N)=O)C1)C 85244,C1(C(N(C2CCN(C(=O)Cn3cc(Cl)c(C)n3)CC2)CC)=O)CC(C2CC2)C1 85245,O=C(C1=CCCCC1)N1CCC1C(N1CCC(NC(C2CCC2)=O)C1)=O 85246,CN1CCN(C(C2(CO)CCCC2)=O)CC1C(=O)NCC12CCCC(CO1)C2 85247,C=CC(CC)CC(=O)NCC=CCC(=O)NCC(C)N(C)C(C)C 85248,C1(C(C)C)CN(C(c2cncc(F)c2)=O)CCC1NC(=O)C=CC1CC1 85249,c1(NC(C(CC)NC(=O)CC2C=CCCC2)=O)cccc(CN(C)C)c1 85250,C1(C(=O)NC2CCCN(C(c3oc(C)c(CO)c3)=O)CC2)CC2CC1CC2(F)F 85251,CCCC(CCCNC(C1OCCC1(C)C)=O)NC(=O)CNC(=O)C1CC1 85252,CC1CN(C(C2(O)CC(F)(F)C2)=O)CC1NC(C1(F)CC1)=O 85253,CCC(CCC(=O)NCC1CC2(CCC2)CO1)NC(=O)C=CC1CCC1 85254,C12(C(C)=O)CCCC1CCN2C(=O)Cc1c(C)nn(CC(C)C)c1C 85255,CON=C(C(=O)NCCC(C)N(C)C(c1coc(S(N)(=O)=O)c1)=O)c1ccco1 85256,C1(NC(CSC)=O)CC2CCC1N2C(=O)Cc1cccc(Cl)c1 85257,C1(C(=O)NC(C)CCNC(=O)C=C2CC2)CC2(CCCCO2)C1 85258,C(=O)(CC(C(F)F)NC(C1C2CCC(C2)C1C)=O)NCCc1ccc(C)s1 85259,c1(C(N(CC(CC)NC(=O)Cn2ncccc2=O)C)=O)cc(C)c(C(N)=O)cn1 85260,c1(CC)nc(CCNC(=O)Nc2csc(Cc3ccccc3)c2)no1 85261,N1(C(c2c(OC)nsc2)=O)CC2CCC1(CNC(C1CC1C(C)C)=O)CC2 85262,N1(C(C2(CCC)N(C(C=C(CCC)CCC)=O)CCC2)=O)CC(O)C(O)C1CO 85263,O=C(C1CCCc2scnc21)N1CCCCC2(CCOCC2)C1 85264,c1(C(=O)NC(C(C)C)CCN(C)C(c2cnn[nH]2)=O)ccccc1N=S(C)(C)=O 85265,C1(C(=O)NC(Cc2ccco2)C(=O)N2CCC(CCO)C2)CC2(CCC2)C1 85266,c1(C(N2CC(NC(=O)CCC(=O)N3CCOCC3)C2)=O)ccc2c(c1)CC2 85267,c1(CN2CCC(C(C)NS(=O)(=O)Cc3ccccc3)C2)c(O)cccc1F 85268,c1(COC)nocc1COC(C1(S(=O)(=O)Cc2ccon2)CC1)=O 85269,N1(C(C(=O)N(C(C)COC)CCOC)=O)CCCCCCCCCC1 85270,c1(C(C(=O)NCC(CNC(C2(CC(C)C)CCC2)=O)C)(C)C)cc(Cl)cc(Cl)c1 85271,c1(CC)ccccc1C(=O)NC1CC(C)N(C(=O)CC2CN(C)C2)C1 85272,O=C1CCC(C(=O)NC(CNC(c2cccn3ccnc23)=O)CO)=NN1 85273,c1(C(=O)NCCC2(OC)CN(C(=O)CSSC(F)(F)F)C2)ccccc1C(F)F 85274,C(CCC)(C(=O)N1CCC(C(=O)NCCOCCOC)C1)=CC 85275,C1(CNC(C2CC(OCOCC)C2)=O)CCCCC1N1CCC1.N1(C=O)CCC1 85276,CC(C(=O)NC(c1ccccc1)C12CC(C1)C2)C(C)NC(=O)OC(C)(C)C 85277,C(=O)(CCCCC(=O)OC)N1CCC(N(C(CC(CCC)O)=O)CC)CC1 85278,c1(C(=O)NCC2CCN2C(=O)CNC(=O)C2CC2)nnc2ccccc2c1O 85279,C(C)(C(=O)NCC(c1ccccc1)NC(c1nc(Cl)c(Cl)s1)=O)(C(C)C)OC 85280,C1(NC(N(C(CC)C(C)O)C)=O)CCOC(CSC)C1 85281,c1(C(N2CC(CNC(c3cn(C)nc3O)=O)C2)=O)c[nH]c2cccnc12 85282,c1(C(=O)NC2C(NC(CCc3ccc(C)cc3)=O)CC2)ccc(S(N)(=O)=O)cc1 85283,c1(CCC(=O)NCCOCCC2=NCC(O)CO2)cnc2cccc(Br)n12 85284,CC(=O)CCN=C(NCC1CC2(C1)CC(C)(C)C2)NCC1CCC2CC1C2(C)C 85285,c1(N(C2CCN(C(C3(C)C=CCC3)=O)CC2)C)ncc2ncnc-2[nH]1 85286,c1(C(=O)NCCC2CSCCN2C(C2CC23CC3)=O)nc(O)[nH]c(=O)n1 85287,C(=O)(CCC(=O)NCC1CC(O)CN1C(=O)CCc1cnc(C)s1)NCCC 85288,c1(OCCCC)ccc(C(=O)NCC2CCN(C(C3CCCOC3)=O)C2)c(Cl)c1 85289,CC(CC(C)(F)F)C(=O)NCC1CN(C(=O)CC(F)(F)C(F)F)CCO1 85290,c1(OC)ccc(CC(=O)NCCC(C)NC(=O)C(C)(CO)OC)c(OC)c1 85291,CN1CCCC2CN(C(c3ccnc(Cl)c3Cl)C(=O)NC3CC3)CCC12 85292,C1(CNC(C2C(C)(C)C2)=O)CCCCN1C(=O)Cc1cnsc1 85293,N1(C(c2c(OC(F)F)cc(C)s2)=O)CC2CCC(C1)N2C(=O)CCS(C)=O 85294,CC1=C(C(=O)N2CC(O)(CCNC(C3CC4CCC(C3)C4)=O)C2)SCCO1 85295,C(=O)(C1=CCC2CCC1N2C(c1cccs1)=O)Nc1c(C)n(C2CC2)nc1 85296,C1(C(=O)NCC(CCOC)NC(COCCCC)=O)CC2CCC(C1)O2 85297,c1(C(N2CCC(F)(C(=O)NC(CCCC=C)C3CC3)C2)=O)ccc(F)c(C)c1 85298,Cc1cc([N+](=O)[O-])cnc1C(=O)NCC1CC(NC(c2c[nH]c(Br)c2)=O)C1 85299,N1(C(C2(C)CC(NC(CCc3n(C)cnc3)=O)C2)=O)CCC2(CCCOC2)C1 85300,C1(C2CCN(C(C3CC3C)=O)CC2)(NC(c2cc(C)cc(Br)c2N)=O)CC1 85301,N1(C(CN(C(c2n(C=C)nnc2)=O)CCC)=O)CCN(C)C(C)C1C 85302,CC1CC(NC(c2cn(C(F)(F)CO)nn2)=O)CN1C(c1snc(O)c1Cl)=O 85303,c1(NC)ccnc(C(=O)N(CCC(=O)NCc2cc(C)on2)C)c1 85304,C1(NC(C2CC23CCC3)=O)CN(C(c2snc(Cl)c2Cl)=O)CC1C(F)(F)F 85305,Cc1ccc2c(c1)CC(C13CC(C(=O)OCC4CC4)C1C3)S2 85306,c1(CC(=O)N(C(C)CN(C)C(=O)C2CC2)C)ccc(NC(=O)NC2CC2)cc1 85307,C(=O)(C(CC1CCC1)NC(=O)CSCCOC)NCC(C)OCC#C 85308,CCC(F)(F)C(=O)N1CCC(C(C(C)C)NC(=O)CN2CC(C)(OC)C2)CC1 85309,c1(C(=O)NC2CC(C)(CNC(CCCOCC)=O)C2)ccc2[nH]cc(C#N)c2c1 85310,CCC(C)C(C)(O)CNC(=O)C(C1(O)CCC1)NC(=O)CCCn1cccc1 85311,c1(N2CCN(C(C)C#N)CC2)nccc(=NCCc2cccc(Cl)c2)[nH]1 85312,c1(-c2cc(OCC)cc(F)c2)cc(C(=O)NC2(C(C)C)COC2)c2cn[nH]c2c1 85313,c1(C(N2C(C(=O)NCCc3ccncc3)CSCC2)=O)ccc(O)cc1O 85314,C1(CC(N2CC(C)(NC(C3C(C)OCCO3)=O)C2)=O)COC2(CCC2)CO1 85315,CC1=C(C(=O)NCc2cc(C(=O)N(C34CC(C3)C4)C)on2)CCO1 85316,C1(C(N2C(CNC(C(CCC)C#N)=O)C3CCC2C3)=O)CCc2nnnn2C1 85317,c1(OC)ccnc(F)c1C(=O)NCC1CCN(Cc2csc(Br)n2)C1 85318,C(CC(C)(C)C(=O)N1CCC(C)C(CNC(c2ncccc2F)=O)C1)OC 85319,c1(OC)cccc(C(C)CC(=O)NC(C)CCNC(=O)CCc2ccon2)c1 85320,S(=O)(=O)(c1cccc(=NCc2cc(C(N)=O)no2)[nH]1)NCc1c(COC)cccc1 85321,C#CCCC(C(=O)NCC(=O)NCC(=O)NC)NC(=O)C(C)N(C)C 85322,c1(C(=O)NC(C)(C)C)cn(C2CC2)cn1.CC1C(=O)N1.C1(=O)CO1 85323,C1(CC(=O)NC2CCN(C(c3ccc(CCC=C)cc3)=O)C2)CC(F)(F)C1(F)F 85324,C1(CCC)CN(C(C2(Cl)CC2(C)C)=O)CCN1C(=O)C=CBr 85325,N1(C(C(C)Oc2ccccc2)=O)CC2CCC(C(=O)NCC3(C)CSC3)(C2)C1 85326,N1(C(c2c(CNC(C(C)(C)n3cnnn3)=O)cco2)=O)CC2C=CC2C1 85327,CC(C)(C)CC(=O)NC1CC1NC(c1cc(CO)ccn1)=O 85328,c1(C(C2CCC2)NC(=O)NC(C)CC2CCC2)ccc(F)cc1F 85329,N1(C(COC)=O)CCCC(NC(=O)CC2CC2)CC1 85330,c1(NC(C2=C(C)OCC2)=O)ccc(C2=CCN(C(C3CCC(C)O3)=O)CC2)cc1 85331,C(=O)(C1=C(Cl)CCCCC1)N(CC(C)N(C(=O)C(F)Cc1ccccc1)C)C 85332,N1(CC(=O)NCCCCN(C(=O)C=CC2CC2)C)CCC(F)(F)C1 85333,CC1CCCN(C(c2cccnc2)=O)C1CNC(C12CC3CC1C2C3)=O 85334,CC1OCCOC1C(=O)NCC1CCCN1C(c1ccc(C(N)=O)s1)=O 85335,CCC(O)CN(C(=O)C(F)OC(F)(F)F)CC1CC1 85336,c1(CC)[nH]c(=N)sc1C(N1CC(NC(=O)Cc2ccnc(F)c2)C(C)C1)=O 85337,Cc1cc(C(=O)NC(C2CCCCN2C(=O)CCSc2nnnn2C)C)ccn1 85338,C(CC(C)C(=O)N1CCCC(C(=O)NCCN2CCOC2=O)C1)=CC 85339,Cc1nc(C(N2CC(C(C)NC(=O)C(O)Cc3ccccn3)C2)=O)c(=O)[nH]c1C 85340,Cc1ccc(C(=O)NCCCCC(C)NC(=O)C2=NOC(C)C2)c(Cl)c1 85341,C1(C)(CNC(c2ccn(C)n2)=O)CN(C(=O)CCOC2CC2)CCO1 85342,c1(CN2C(C(=O)Nc3nc(O)cs3)CC(O)C2)ccc(O)cc1Br 85343,N1(C(C(=O)NCC2CCSCC2)=O)CC=C(c2ccc(Br)cc2)CC1 85344,C#CC1(NC(C2(NC(=O)CN(C)C(C)=O)CCCC2)=O)CCCCCC1 85345,c1(C(N(CCCCNC(C2CCCC2O)=O)C)=O)c(Cl)nc2ccccn12 85346,c1(CC(C)NC(C(C)SC(F)(F)F)=O)ccc(CNC(C2(C)CCOC2)=O)cc1 85347,c1(CC)cc(NC=O)cc(CC)c1-c1nccn1-c1ccc(-c2ccc(C(F)(F)F)c(CC)c2)cc1 85348,c1(CC)ccccc1NC(=O)CNCC(C(C)CC)N1CCC1 85349,N1(C(C(CC)(C)OC)=O)CCCCC2(CCN(C(C3(CCF)CC3)=O)C2)C1 85350,Cn1ncnc1C(=O)NCCCOCCNC(=O)CC1(C)CC1F 85351,c1(CN(C(=O)COCC2CC2(C)CC)CC)cn(C(C)(C)C(=O)O)nn1 85352,C(=O)(CCCCCF)NCC1C(NC(c2c(CC)ncs2)=O)C1 85353,C1(CNC(C=C(C)C2CC2)=O)CC12CCN(C(=O)C=CCN1CCOCC1)CC2 85354,C(=O)(C1(C)OCCc2ccccc21)NC1CC(N(C)C(c2cncs2)=O)C1 85355,Cn1nnc2c1CCN(C(=O)C(C1(C)CC1)NC(C1CCCOC1)=O)C2 85356,C(C)(C(=O)OC)(C(C)C)NCc1ccc(Cl)cc1.n1(CCC)c2nnc1SC2 85357,n1(CC)ccc(CC(=O)NC2CCN(C(=O)C(C)(C)c3cscc3Cl)C2)n1 85358,CC1CC(N(C(=O)C(C2CC2)N(C)C(c2ccoc2Cl)=O)C)CC(C)C1 85359,N1(C(C(C)S(N)(=O)=O)=O)CCN(C(C2Cc3ccccc3C2)=O)C2CCCC12 85360,Cc1c(C(=O)N(CCCCN(C(=O)CC2(C)CCCCC2)C)C)cnn1CCO 85361,C1(N(C(C=CC=CCC)=O)C)CCN(C(=O)C(C)(C)C2CCCCO2)C1 85362,C(=O)(CCCC(CC)CC)N1CC(CC(=O)NCCC(CCC)C2CC2)C(C)C1 85363,C1(CC(=O)O)CSCCN1C(c1ccc(C2CCCC2)nc1)=O 85364,N1(C(C=CC=CC)=O)CCC(C)C(CNC(c2cc(C3CCOCC3)[nH]n2)=O)C1 85365,c1(CCCCNC(=O)NCc2cc(C)ncn2)ccc(F)c(F)c1 85366,N1(C(C(C#C)(C)C)=O)CCCN(C(C2CCC(=O)N(C(C)C)C2)=O)CC1 85367,c1(C(N2CC(CN(C)C(c3ncc[nH]3)=O)C2)=O)cn(C)c2ccccc12 85368,C(=O)(CN=S(C)(C)=O)N(CCCNC(C(C(C)O)C)=O)C 85369,c1(C(N(CC(C)NC(c2nn[nH]c2Cl)=O)CC)=O)cnc(O)c(Cl)c1 85370,N1(C(C(=O)NCCOC)CCC2CC=CCC2)CC2CC1CN2C1CC1 85371,C12(C(=O)NC3CCN(C(C4CCSCC4)=O)C3)CC(CO)(C1)OC21COC1 85372,N1(C(CCCC#CC)=O)CC2(CNC(C3CCCCS3)=O)CC1CCO2 85373,C1(CNC(C=CC=CC)=O)CN(C(c2nn(C(C)C)nc2Br)=O)C2CC12 85374,Cc1nc(C(=O)NCC2CC2NC(c2ccn(-c3ccncc3)n2)=O)co1 85375,CC1(C)CCCCC1=CC(N1CC2CC1C2CNC(c1ccc(Cl)o1)=O)=O 85376,CC(CC(=O)NC1CCC(CNC(C2CCOCC2)=O)C1)C(C)(C)C 85377,c1(CC(=O)NC(C2CCN(C(CCCC(C)C)=O)C2)C)ccc2cnccc2c1 85378,c1(CC(=O)NCc2ccc(CO)o2)ccc(C(=O)O)o1 85379,c1(C(=O)NCCCNC(C2CC(CC)C2)=O)cc([N+](=O)[O-])cnc1N 85380,Cn1cnc2c(C(=O)Nc3nc(-c4ccc(F)cc4)cs3)ccnc12 85381,CC1CC(NC(C2CCCCC2)=O)CCN1C(C1CC(=C2CCC2)C1)=O 85382,CC1(C)CC(NC(C2CC(C)N2C(C2(Cl)CC2)=O)=O)C1 85383,C(c1scnc1C)=CC(N1C(C(CNC(Cc2c(C)nc[nH]2)=O)(C)C)CCC1)=O 85384,C1(CC)C(NC(c2ncncc2N)=O)CCCN1C(=O)CN(C)C(=O)C1CC1 85385,N1(C(C(COC)NC(C)=O)=O)C2CCC1C(NC(c1cc(C3CC3)no1)=O)C2 85386,C(C(CC1CC1)C(=O)NCc1cccnc1F)NC(c1nc(CC)oc1)=O 85387,Cc1nc(C(=O)NCC2C=CCN2C(C2COCC3(CCC3)O2)=O)c(=O)[nH]c1C 85388,N1(C(=O)NC(C)CCc2ccccc2F)CC2(C(=O)N(C)C)CCCC1C2 85389,N1(C(c2c(OCC)cccn2)=O)CC(C(=O)Nc2cncs2)CC2OCCC12 85390,C=CCC(C)C(=O)NCC(C(C)C)NC(c1cc(C(C)=O)c(C)o1)=O 85391,S(=O)(=O)(c1ccc(C(=O)NCC(CO)NC(c2ccc3cnnn3c2)=O)o1)NC 85392,Cc1scc(C)c1C.c1(C(=O)OCC(O)CN(C)C)ccccc1 85393,c1(OC)cc(OC)cc(CC(=O)NC2CC(C)CN(C(=O)CC3CN(C)C3)C2)c1 85394,C(C(=O)NNc1ncnc2c1ncn2C)NC1(CO)C(C)CCCC1 85395,CC1(C2CCN(C(=O)CC3C4CCCC4N3C(=O)C=CC3CCCC3)C2)CC1 85396,c1(CC)c(OC)cc(C(=O)NCC2CCN(C(=O)C=CC(F)(F)F)C2)cc1OC 85397,CC(C)CC(=O)NCC(C1CCCC1)NC(=O)Cn1cc(Br)cn1 85398,c1(C(N2CCCCC(NC(C(C)CC3CC3)=O)C2)=O)cc(C#N)c(O)nc1N 85399,c1(OC)ccc(N(C(=O)CONC(=O)Cc2cn[nH]c2)C)cc1 85400,c1(C(=O)OCC)cccnc1N1CCC(C(C)NC(=O)CC2CCC(=O)N2C)C1 85401,C1(CNC(c2c(OC)n[nH]c2)=O)CN(C(c2ccccc2C)=O)C2(CCC2)C1 85402,C1(NC(C(c2scc(C)n2)C)=O)CN(C(=O)CC2CC2(Cl)Cl)C2CCCCC12 85403,C1(C(=O)OC)CN(C(c2sc(C)cc2Cl)=O)CC1(C)C 85404,c1(OCCCC(C)C)ccc(NC(N2CC(N)C2)=O)cc1 85405,CC1CC(C(=O)NCC(C2CCCN2C(=O)Cn2nccn2)(C)C)CCS1(=O)=O 85406,c1(C(N2CCC(C(=O)OCC)(CC)CC2)=O)[nH]c2nccc-2cc1Cl 85407,N(C1CCCc2c[nH]nc21)C(C1=CCC(NC(C#CC(C)C)=O)C1)=O 85408,N1(C(c2c(C)[nH][nH]c2=N)=O)CC2(C1)CN(C(c1ccc(C(C)(C)C)cc1)=O)C2 85409,N1(c2nnc(CC)o2)CCC(NC(C2CCCOC2)=O)C1(C)C 85410,c1(NC(C(C)N(C(=O)C(c2ccccc2)C)CC)=O)cccc(OC)c1C 85411,c1(C(C(=O)NCCN(CCOC)C(c2cscc2Cl)=O)C)ccccc1Cl 85412,c1(SC)cc(N2CCCC(C(=O)Nc3ccc(-c4cc[nH]n4)cc3)C2)ncn1 85413,c1(C(=O)NCC(CO)NC(c2c(C)nc(CC)s2)=O)nc(C)n(C)c1C 85414,C1(C(=O)NCC2CC(NC(=O)Cc3cnn(C(F)F)c3)C2)CCc2nncn2C1 85415,C(CCCC(=O)N1CCCC(N(C)CCC)C1)N.C(=O)(C(C(C)C)SC)CCC=C 85416,c1(CNC(C2CCC(NCc3cc(F)nc(F)c3)CC2)=O)ccc2c(c1)OCO2 85417,Cc1cccnc1C(=O)NC1C2CC(NC(c3cnnc(O)c3)=O)CC12 85418,C=Cn1nncc1C(=O)NC1(CN2CCN(C(=O)C(C)SC)CC2)CC1 85419,c1(C(C)(C)OC)nc(=NCC2(c3ccc(C)cc3)CC2)s[nH]1 85420,c1(C(N2CCCC(C3(C)N=N3)C2)=O)cc2cc(C#N)ncc2[nH]1 85421,Cc1cnc(C(=O)NC2CN(C(=O)CCc3cnc(C4CC4)o3)C2)c(Br)c1 85422,c1(C(=O)NCC2C(CNC(C3CCC(C)(O)CC3)=O)C2)cc2n(n1)CC(F)C2 85423,C(=O)(CS(=O)C(F)(F)F)NCCN(C(c1c(C)ccs1)=O)CCOCCO 85424,c1(-c2c(-c3cn(CCC=C)nn3)cccc2)ccc(F)cc1F 85425,N1(C(C2(C)CCN(C)C2)=O)CC(C2CCCN(C(=O)C(C)(C)CS(N)(=O)=O)C2)C1 85426,Cc1cc(C(=O)N(CCC(C)NC(=O)CSc2n[nH]c(C)n2)C)c2n[nH]cc2c1 85427,Cc1n[nH]c(C)c1C(C)C(N1CCC(NCCN(c2ccnc(Cl)n2)C)CC1)=O 85428,C1(C(=O)NC(c2cncnc2)C)C2CC(O)C(C2)N1C(c1cc2n(n1)CCO2)=O 85429,C(=O)(C(CC(C)(C)C)OC)NCC1OCC(C(=O)NCCOCCC#C)C1 85430,c1(OC)cc(OC)cc(C(N2CC(C(C)NC(C3CCCC3(C)C)=O)C2)=O)c1 85431,N1(C(CC(CC)(C)C)=O)CCCC2(CCN(C(=O)Cn3cc(CO)nn3)CC2)C1 85432,C1(C(N2CCC2CC2CC2)=O)C(C2CC2)CCN1C(C1CCCCCC1)=O 85433,Cc1ncc(CNC2CCCC2NC(=O)CC2CN(C3CCCCC3)C2)[nH]1.C=O 85434,c1(C(N2C(CNC(c3ccoc3Cl)=O)C=CC2)=O)cc(O)c2ccoc2c1 85435,C1(CNC(COCCCC)=O)(COC)CCN(C(=O)C(C2CC2)SC)C1.C(=O)COC 85436,c1(C(N2CC(CC(=O)N(C)Cc3ccc(C(=O)O)o3)C2)=O)cnc(O)c(Cl)c1 85437,CC(C)(C)CCC(F)C(=O)N1CC(CNC(=O)C=C2CCOCC2)C2(CCC2)C1 85438,C(=O)(C(C)(CN(C)C)CC(C)C)OC(C(c1ccccc1)C)OCC 85439,C(C(O)C(F)(F)F)C(N1CCC1CC(=O)NC1C(C)(C)C1)=O 85440,c1(NC(c2cc(CNC(c3scc(C)c3Cl)=O)ncc2)=O)ccc(I)cc1Cl 85441,c1(C(CC)=O)ccc(NC(=O)C(N2CC(c3ccc(F)cc3)C(N)C2)=O)cc1 85442,c1(SC)ncc(N)c(C(=O)N(C2CCN(C(=O)CSC)C2)CCO)n1 85443,c1(N2CCC(CS(N)(=O)=O)CC2)nc(NCCN2CCCC2=O)c2ncsc2n1 85444,C(=O)(C(C(C)(C)C)NC(c1cc(OC)ccc1N)=O)NCC(CC)OC(C)C 85445,CC1(C)CN(C(C2CCCN2Cn2cccnc2=O)=O)CC1C(=O)NC1CC1 85446,c1(C(=O)OCC(N)=O)ccn2[nH]c(=NC(=O)C3CC3Cl)nc2c1 85447,Cc1c(Br)ccc(NC(C2CC2NCc2ccc(C(F)(F)F)cc2Cl)=O)c1F 85448,C=CC(CC(=O)NC12CC(C1)N(C(c1cncc(NC)c1)=O)C2)c1ccccc1 85449,c1(OC)c(F)cc(C(=O)NCC2CC2NC(=O)C(C2CC2)C2CC2)cc1Br 85450,C1(CNC(C=Cc2ccc(C)nc2)=O)CN(C(c2ns[nH]c2=O)=O)CC(C)(C)C1 85451,c1(C(C)NC(c2n(CC)ncn2)=O)ccc(CNC(C2CC2C2CC2)=O)cc1 85452,CC(CC(=O)NCC12CCCC(CN1C(C1COCCOC1)=O)C2)CC(F)(F)F 85453,CC(C)C(C(=O)NC1CN(C(=O)CCCCO)CC1n1ccnn1)N(C)C 85454,C(CCCCCN=c1[nH]c2ccc(F)cc2o1)NC(C(CC)SC)=O 85455,C=CCC(CNC(c1c[nH]c(C(N)=O)c1)=O)NC(c1occc1C1CC1)=O 85456,c1(C(=O)NCCN2CCC3(CC2)CC3)nc2ccc(O)cc2s1 85457,CCC(CC(=O)N1CC(CO)C2(C1)CN(C(C1CCCC(C)C1)=O)C2)C(C)(C)C 85458,N1(C(C(CCC)OCC)=O)CCC(C)(C)CC1C(=O)NCc1cc(C)nc(C)c1 85459,Cc1c(S(=O)(=O)Nc2cc(Cl)nn2C)sc2cc(F)ccc12 85460,c1(C(N(C2CN(C(CC(C)C3CC3)=O)CC2O)C)=O)cc2c(cnn2C)nc1O 85461,N1(C(C(=O)N(C)C)=O)CCN(C(C2CCC3CC23)=O)C2(CC2)C1 85462,CC1=C(C)CC(C)(C(=O)NCCC(C)NC(c2sc(C(C)C)nc2C)=O)CC1 85463,c1(CNc2scc(-c3ccc(OC)cc3)n2)c(OC)ccnc1O 85464,Cc1cn2cc(C(=O)NCC(CC(C)C)NC(=O)C(C)n3cnnn3)sc2n1 85465,Cc1cc(C)c2nc(N(C3CCN(C(=O)C(C)(O)C4CC4)C3)C)sc2c1 85466,c1(C(=O)NCC2N(C(C(CCC)OCC)=O)CC2)c(N)sc(C)c1C 85467,Cc1cc(Cl)nc(N)c1C(N1CCCC(O)(CNC(=O)CC2CCCC2O)C1)=O 85468,c1(C(C)=O)ccccc1OCC(=O)NCC(C)(C)CNC(=O)C=CCO 85469,c1(CC(=O)NCC2(C)CCCN2C(c2csc(C3CC3)n2)=O)ncn2c1CCC2 85470,c1(NCc2cc(C)ncn2)nc(N(C)Cc2nc(C#N)cs2)nc2sccc12 85471,C1(C)(NC(CCc2ncn(C)c2)=O)CCN(C(C2(CCF)CCC2)=O)C1 85472,N1(C(C2N(C)C(=O)CC2)=O)C2CC=C(C(=O)NCc3n[nH]c4c3CCC4)C1CC2 85473,c1(C(N(C(CN(C(c2nc(C(C)=O)sc2)=O)C)C)C)=O)ccc2sncc2c1 85474,Cn1ncc(Br)c1CC(N1CCC(c2cn(-c3cccc(Cl)c3)nn2)C1)=O 85475,N1(C(CC(C)C)=O)CCCC(N(C(=O)Cn2ccccc2=O)CCO)C1 85476,N1(CC)CCC(Cc2c(-n3cc(C4CCCCC4O)nn3)noc2CN)C(C)C1 85477,C#Cc1ccc(NC(=O)C(N2CC(c3ccccc3C)OC(C)C2)=O)cc1Cl 85478,C1(CNC(c2c(C)nc(O)[nH]2)=O)CCC12CCN(C(=O)Cc1csc(Cl)c1)CC2 85479,C1(C(=O)NCCSCCCc2nccc(C)c2)CCC2(CC1)CNC2 85480,Cc1cc(C(=O)NC2CCC(NC(c3ccc(O)nc3C)=O)CC2)cnc1C 85481,C=C(C)CN=C(NC(C)C)N(C)CC12CC3CC1C2C3O 85482,C1(C(=O)NC(CC)CNC(=O)C(C)C)CC(c2cnn(C)c2)=NO1 85483,C#CC1(O)CCN(C(C2(CF)CCN(C(=O)CCc3cn[nH]c3)C2)=O)C1 85484,Cc1ccccc1C(=O)NC1COCC1CNC(C1(c2ccccc2)CCOC1)=O 85485,Cc1ccc(C(=O)NC23CCC2CN(C(c2cc(C4CC4)on2)=O)C3)nc1C 85486,N1(C(C2CC(OC)C2)=O)CCCC(C)C1CNC(c1cnn(C)c1Cl)=O 85487,Cn1ccc2[nH]c(C(N3CC(CNC(=O)NCCCCl)C3)=O)cc12 85488,N1(C(c2c(OC)n[nH]c2)=O)CCC2(CC1)CC2CNC(C1CC(F)C(=O)N1)=O 85489,N1(CC(=O)NCC(CC)NC(=O)Cn2ccnc2C#N)CCCc2ccccc21 85490,NCC(C(F)(F)C(F)(F)F)NC1CCCCC1c1ccnn1C 85491,S(=O)(=O)(c1c[nH]ccc1=NCCn1cnc(C)c1C)NC(C=C)(C)CC 85492,c1(C(=O)NC23CC(NC(=O)CCC4CCOCC4)(C2)C3)cc(O)ncc1Br 85493,C1(CCNC(C(=O)Nc2cccc(N3CCN(C)C3=O)c2)=O)CCC(F)(F)CC1 85494,C(CC(C)(C)NC(C1(C#N)CC1C)=O)OC.C1(=O)C(OC)C2CN1C2 85495,c1(C(=O)NCC2(F)CC(CNC(C3(F)C(C)C3)=O)C2)ccc2nc(=N)[nH]n2c1 85496,C=CC(CC)C(=O)NCC=CC(=O)N(CC(C)(CO)CO)CC 85497,C1(NC(CC2(C(=C)F)CCC2)=O)C(C)CCN(C(=O)CC(F)(F)C(F)F)C1C 85498,Cc1cn2cc(C(=O)NCC3CCN(C(c4ccc(N(C)C)nn4)=O)C3)sc2n1 85499,N1(C(C(C2CCOC2)OC)=O)CCN(CCNC(c2cnc(C)s2)=O)CC1 85500,c1(OCC)ncc(C(=O)NCC2CCCN(C(C3(C)CCCO3)=O)CC2)cc1Cl 85501,C=CCCCCCCCCC(=O)NC1CCSC12CN(C(=O)Cc1ccoc1)C2 85502,c1(C(=O)NC2CC(CCNC(COC)=O)C2)cc(C2CC2)nc2onc(C)c12 85503,CC(O)C(F)(F)C(=O)NC1(c2ccc(Br)cc2)CN(C(=O)C(N)=O)C1 85504,C1(NC(C(CC)F)=O)CN(C(=O)CN(C)CCO)CC2(CCC2)C1 85505,N1(C(CCCC#C)=O)CC2(C1)CN(C(c1sccc1Br)=O)CC2C(=O)O 85506,N1(C(C2(NC(C(CC=C)C)=O)CC(O)C2)=O)CC2CN(C)CC2C1 85507,Cc1nc(C2CC2)nc(C)c1C(=O)NCC(F)CNC(C1CC1(Cl)Cl)=O 85508,C1(NC(C2C(NC(C3CCCC(=O)C3)=O)CCCCC2)=O)CCn2ncnc2C1 85509,C(=O)(C(C(F)(F)F)C(F)(F)F)N1CCC2(C(CNC(CC(CC)CC)=O)C2)CC1 85510,C1(CCNC(C2(CC=C)CC=CC2)=O)CCCN(C(=O)CC2C(C)C2(F)F)CC1 85511,C12(NC(C(C)CF)=O)CCCC1N(C(c1ccnc(S)c1)=O)CC2 85512,c1(C(N(C(CNC(C2CN(C(C)=O)C2)=O)C2CC2)C)=O)cc([N+](=O)[O-])cnc1O 85513,C(C(CNC(=O)C(=O)NCC(F)F)S(C)(=O)=O)NC(C1(CO)CC(C)(C)C1)=O 85514,N1(C(C2(CC#C)CCOC2)=O)CCCC(CN(C)C(c2ccoc2C2CC2)=O)C1 85515,C(CC(C)C(=O)N(C1CCCN(C(c2ccccc2NCCO)=O)C1)C)OC 85516,N1(C(CN(CC)CC)=O)CC(C(=O)OC)(C(=O)NCCN2CCCCC2)C1 85517,C1(OC)CC2CC(NC(=O)CC3CCCN3C(=O)CC(=O)NC3CC3)CC12 85518,CCCC(C)(CCC)C(=O)N1CC2CC(NC(c3[nH]nnc3C)=O)CC(C2)C1 85519,c1(CC(=O)NC2C(NC(COC(CC)(C)C)=O)C2)ccc(OC(F)F)c(F)c1 85520,N1(C(c2c(C)ccs2)=O)CC2(CC2)CC1CNC(C1CC2CC1CO2)=O 85521,c1(C(=O)NCC2C(NC(C3(C#C)CCCC3)=O)C2)cc(NC(C)=O)cnc1C 85522,N1(C(CC(=O)OCC)=O)CC(F)CC1CN(C)C(c1ccccc1)=O 85523,c1(CN(C)C)ccc(C(=O)NC(c2ccccc2)CNC(C2(Br)CC2)=O)cn1 85524,c1(OC)cc(C)ccc1NC(C12CC(CO1)N(C(c1ccnc(O)c1)=O)C2)=O 85525,N1(C(CNC)=O)CCC2(C(=O)NCCN3CCNC3=O)CC2C1 85526,C(=O)(CC(C)(C)C)N(C(C)C(=O)NCC(C)(C)C(C)O)C 85527,C(Cc1ccccc1)(C(=O)NC(C)(C)CN(C)C(C1(CCO)CC1)=O)NC(C)=O 85528,N1(C(c2c(C(C)(C)C)ncs2)=O)CC2CC(NC(=O)CCCCCF)CC1C2 85529,C#CCC(C(=O)N(CCCC(F)(F)F)C)NC(C1CCC(OC)CC1)=O 85530,C(C(C(=O)N(C1CCC1(C)C)C)C(C)C)NC(C=CC(C)C)=O 85531,c1(C(=O)NCC2(NC(=O)C(C)NC=O)CC(OC)C2)cccc(C(C)C)n1 85532,N1(C(C(CCC)O)=O)CCCC(C)(NC(c2occc2Cl)=O)C1 85533,C1(C(=O)NCCC2N(C(=O)C=CBr)CCC2)(CF)CCC(F)(F)CC1 85534,O=C1COc2cc(CC(=O)NCCCOCCCO)ccc2N1 85535,c1(C(=O)NCC(CNC(c2cc(F)n(C)n2)=O)OC)cc(F)c2ncccc2c1 85536,Cc1ccc(=O)n(CC(N2CCC23CN(C(C2CC24CCOC4)=O)C3)=O)n1 85537,c1(C2C(C(=O)NCCN(C(=O)Cn3cc(CO)nn3)CC)C2)ccccc1Cl 85538,N1(C(CNS(CC)(=O)=O)=O)CC2CS(=O)(=O)CC2(NC(C2(CSC)CCC2)=O)C1 85539,c1(-n2ccc(CNC(Cc3c(C)cccc3)CO)n2)ccc(F)cc1F 85540,c1(CC)cc(C(=O)NC2CN(C(c3coc(C)n3)=O)C2)oc1CC 85541,Cc1cccc(CNCC2(C)CCN(C(c3nc(-c4nc[nH]n4)sc3C)=O)C2)c1 85542,c1(OC)ccc(C(=O)NCC2CCN(C(=O)C=CCF)C2(C)C)c(F)c1Cl 85543,C1(C(=O)NCC2C(C)(C)C2)CC2(CCN(C(=O)COCCCF)C2)C1 85544,N1(C(C)Cc2ccccn2)C(=O)NC(Cc2cccc(Br)n2)C1=O 85545,c1(OCC)cc(Cl)c(C)cc1CNC(=O)C(N1CCC1C(=O)OCC(C)C)=O 85546,N1(C(c2cc(C)ns2)=O)CCC(C(=O)N(C)CCO)CC1C 85547,c1(C(N2CC3(CN(C(C=CC(=O)OCC)=O)C3)C2)=O)cc(C)c(Br)cc1C 85548,N1(C(c2cc(OC)n[nH]2)=O)C2CCC1(CNC(=O)C(C)CC1CCCO1)CC2 85549,c1(C(=O)NCC(N(C)C)C2CC2)cc(O)nc2c(Br)cccc12 85550,C1(NC(C(CCSC)O)=O)CC2CCC1(C(=O)NCc1nncn1C(C)C)C2 85551,C1(C)(CC)C=C(C(=O)NC(C2CCCN2C(C2CC=CCC2)=O)(C)C)C1 85552,c1(C(=O)NCC(CNC(C2CCC(C)O2)=O)(C)C)ncccc1N 85553,Cc1cc(C)c(C(=O)NCC2CCN(C(=O)C(C)N(C)Cc3ccccc3)C2)[nH]1 85554,c1(C(=O)NCCOCCCN(C)C(c2cnccn2)=O)cc(C(F)(F)F)n[nH]1 85555,Cc1cc(=NC2CC(C)n3ncnc32)[nH]c(=NCCC(=O)Nc2ncc[nH]2)[nH]1 85556,Cc1ccc(C)c(C(=O)C(C)NC(c2ncccc2Oc2ccccc2)=O)c1 85557,C(=O)(CCCN(C(=O)CC1CC1)C)N(CC=C)CC=C 85558,N1(C(c2cncc(C#C)c2)=O)CC2CC(O)C1C2NC(=O)CC1C(C)(C)C1(C)C 85559,Cc1ccc(OCC(O)CNCCCC2CC2C)c(C)c1Br 85560,c1(NC(C2CC(=C)CN2C(C2(C)CC2)=O)=O)cccc(Br)c1OC 85561,C1(NC(c2cnc3ccsc3c2)=O)CC2CCC1N(C(=O)C=CC1CCOC1)C2 85562,c1(C(=O)NCC2CCCN(C(C(CC=C)(C)C)=O)CC2)c(Cl)nc2ccccn12 85563,c1(C(NNC(=O)C2C(C)N(C)CC2)=O)cc(F)c(Cl)c([N+](=O)[O-])c1 85564,CC1(CNC(=O)CNC(=O)CNC(c2c[nH]nc2C2CC2)=O)CCCCC1O 85565,n1(CC)cc(Br)c(C(N2CC3CC2C3NC(=O)C(C)(C)OC)=O)n1 85566,N1(C(=O)OC)CC(OC(c2csc(-c3ccc(Cl)cc3)n2)=O)C(OC(C)C)C1 85567,N1(C(c2c(C)oc(C(C)(C)C)c2)=O)CCC2C(C1)CN2C(=O)C(=O)C(C)(C)C 85568,C1(C(=O)NC2C=CCN(C(C3(C(F)F)CCC3)=O)C2)CC2CCCC(C1)C2 85569,n1(CC(=O)NC2CCCN(C(c3csc(C)c3N)=O)C2)cccc([N+](=O)[O-])c1=O 85570,C1(C(=O)NC(C(=O)OCC)C2CC2)CCC(C)(C)N(C(c2cccc(CC)n2)=O)C1 85571,C(=O)(C(C)(CC)CO)NCC1(Cc2cn(CCCC(=O)OCC)nn2)CC1 85572,N1(C(C(=O)NC2CC2)=O)CCCCC1C(=O)NCC1(c2cccc(F)c2)CCC1 85573,c1(C(CC)C)nccc(N2CCCC2CCCNC(=O)C(c2ccccc2)F)n1 85574,CON(CCC(=O)N1CCC(F)(F)CC1)C(=O)C(C)N1CCOCC1 85575,C1(C(=O)OC(C)(C)C)CC(NC(=O)OCC(C=C)Sc2ccccc2)C2CC12 85576,N1(C(C2(OC)CCCCC2)=O)CCCN(C(C2CCCC(C)(C)C2)=O)CC1 85577,c1(C(N2CCN(C(CCCC=C)=O)CC2CC(F)F)=O)n[nH]c2ccc(C)cc12 85578,N1(C(=O)C=CC2CCCC2)CCN(C(c2ccc(CF)cc2)=O)C(CCO)C1 85579,N1(C(CC(CNC(C(CC)(C)OC)=O)O)=O)CCC2(CCC2)C1 85580,Cc1cc(=NC2COCC2F)[nH]c(=NCc2ccc(N(S(C)(=O)=O)CCO)cc2)[nH]1 85581,c1(C(=O)NCC2N(C(c3ccc(OC)cn3)=O)CC=C2)ccc(C(C)=O)c(F)c1 85582,C1(CCNC(c2cc(COC)sc2)=O)CCCCN1C(C1COC(=O)N1)=O 85583,CCC(C)C(O)C(=O)NCC1CC(O)(CNC(c2ccn(C(C)(C)C)n2)=O)C1 85584,c1(-n2cc(CNC(Cn3c(C)cc(C)n3)C)nn2)ccc(C)c(NC(N)=O)c1 85585,C12CCN(C(=O)CNC1=O)O2.C1(C(C)C)CCN1C(N)=O 85586,C(c1cnc(C(C)(C)C)s1)=CC(=O)NCC(CC)NC(C1(CC(C)C)CCC1)=O 85587,CCC(Cc1ccccc1)CC(=O)NCC12CC1CN(Cc1cc(CF)on1)C2 85588,c1(-c2c(COC)n[nH]c2)nc(C2CCCO2)nn1CC1CCSC1 85589,c1(CC(=O)NCC(C2CCCCC2)NC(CSCCCC)=O)cccc(Cl)c1 85590,C1(NC(C2OCCO2)=O)CC2(CCOC2)C1 85591,c1(OC)ccc2nc(N3CC4CC4C3)[nH]c(=NCCc3ncnn3C)c2c1 85592,C1(C(=O)NC(c2ccc(F)cc2)CNC(C(CO)N(C)C)=O)CSCC(=O)N1 85593,c1(C(C)=O)ccc(Cl)cc1NC(C1CC2(C1)CN(C(c1ccon1)=O)C2)=O 85594,CC1=NOC(C)(C(N2CC(C)(NC(c3cc(C)c(C(F)F)s3)=O)C2)=O)C1 85595,c1(-c2n(CCCO)nc(-c3cc[nH]n3)n2)cnc2ncnn2c1O 85596,C1(CC)CN(C(c2cnc(C3CC3)[nH]2)=O)CCN1C(c1cccc(C(F)F)c1)=O 85597,C1(C(=O)NC(CN(C)C(C2CC23CC3)=O)(CO)CO)CCCCCCC1 85598,C(CCN(C)C(C1(C)CC=CC1)=O)(C(C)(C)C)NC(C(c1ccccc1Cl)C)=O 85599,C1(NC(c2ccc(OCC)cc2F)=O)CCCCN(C(=O)CC2CCCO2)CC1 85600,C1(C(=O)NCCCN(C(=O)CCc2cccn2C)CC)CCNC1=O 85601,C1(C(N2C(CNC(Cc3cn(CC)nn3)=O)C(C)CC2)=O)CCn2cncc2C1 85602,c1(CNC(C2(C3CCC3)CCC2)=O)ncc(CO)cc1Cl 85603,N1(C(C(C(C)C)SC)=O)CCC2(CC1)CCN(C(C1CCC3CCCCN13)=O)C2 85604,Cc1nc(N2CC(CN(C)C(c3cnccc3C(F)(F)F)=O)C2)c2sccc2n1 85605,C1(NC(C2(CCNC(=O)CC34CCCC3C4)CCCC2)=O)CC2CC1C(O)C2O 85606,c1(N(C)C)nc2ccc(C(N3CC(F)(CNC(=O)C(F)n4cccn4)C3)=O)cc2[nH]1 85607,N1(C(C(C)CO)=O)CCCC(C(=O)NCCn2cccnc2=O)CC1 85608,C(=O)(C(C)(O)C(C)C)N(C)CC1N(C(c2cc(CCOC)on2)=O)CCCC1 85609,C1(=CC(=O)NC(C2CCCC2)CNC(C(CCSC)O)=O)CCCCC1(C)C 85610,c1(CNC(CN(S(CC)(=O)=O)C2CC2)=O)ccc2c(c1)oc(=O)n2C 85611,Cc1cc(OCCN(C)C(=O)NCC2CC2F)cc(C)c1 85612,c1(CC(=O)NC(C2CC=CCC2)C(=O)N(CCCOC)CCO)ccnc(O)c1 85613,c1(CC(=O)N(C2CCN(C(CN3CC(CC)C3)=O)C2)C)c(C)noc1Cl 85614,C1(NC(C2N(C(C)C)CCC2)=O)COC2(C1)CN(C(c1cncs1)=O)C2 85615,C(=O)(C1CCOc2ccc(Br)cc21)N1C(c2cn(C)nc2)C(=O)NCC1 85616,C1(C)(CC)CC(NC(c2ccc(CO)cn2)=O)CN1C(=O)C(C)C 85617,c1(C(=O)NCCN(C(C(c2scc(C)n2)C)=O)CC(C)O)csc(C#N)c1 85618,C1(C(=O)OCC)CN(C(C2CCC(NS(=O)(=O)C(C)C)CO2)=O)CCO1 85619,C1(C(N(CC)CC)=O)CCC2CCC1N2C(=O)Cn1ncccc1=O 85620,CC(C)C(C)(O)C(=O)N1CCC(C(C)(C)C)(CNC(c2nc(Cl)ccc2N)=O)C1 85621,C1(C(C)C)(C(=O)NCC2CC(C)(C)C2)CCN(C(c2cc(Cl)n(C)n2)=O)C1 85622,C1(N(c2n[nH]c3c2CCC3)C(c2ccccn2)=O)CCC2(CCNC2)CC1 85623,C1(C)(C(N2CC(CNC(c3c(CC)c(C)sc3)=O)C2)=O)CC(=O)N(C)C1 85624,N(C1CCc2c(Cl)ccc(Br)c21)S(c1c(C)cccc1Cl)(=O)=O 85625,C(=O)(C(C)(O)C(F)(F)F)N1C(C#C)CCC1 85626,C12(C(=O)NC3C=CCN(C(c4ccn(C)c(=O)c4)=O)C3)CC(C)(C1)OC21CCC1 85627,C1(CC)C(NC(c2cn(CC)nn2)=O)CCCN1C(=O)C=CC=C(Cl)Cl 85628,c1(C(=O)NCCCCCNC(=O)C=Cc2ccccc2)c[nH]c2c(F)cccc12 85629,C1(C(=O)NCC(CC)(CC)NC(c2cnccc2OC)=O)CC2(CCCC2)CO1 85630,c1(C(c2n(C(CC)C)nnn2)NCc2cnc(Cl)s2)ccc(C2CC2)cc1 85631,Cc1ncc(CNC(C2CCN(C(C3(O)CCOC3)=O)C2)=O)o1 85632,CCC(CCC(=O)NC1CCC(CC(N2CCN(C)CC2C(C)C)=O)CC1)OC 85633,C1(CN(CC(C)(C)C)C)CCN(C(C2CC=CCC2)=O)CC1 85634,CC1CC(NC(=NCCNC(=O)OCC)NCCC(F)(F)F)CCN1C.C(C)(C)(C)O 85635,c1(C(=O)NCCC(C)N(C)C(C2CCCN2C2CCCC2)=O)ccncc1N 85636,c1(NC(C(C)(C)NC(c2cn(CC)nc2)=O)=O)cn(C)nc1C 85637,Cc1nocc1CNC(C1(NC(=O)CCc2ccccc2)CC1C)=O 85638,c1(C(=O)NC(CCOC)CNC(C2CC3(CCCO3)C2)=O)[nH]nc2cnccc12 85639,C(C)(CCCC(C)C)N1CCC(c2ccc(Br)cc2)(C(=O)OC)C1 85640,CN=c1ccc(C(=O)NC2(C(=O)NCc3cccnc3F)CCCC2C)c[nH]1 85641,C1(OC)CN(C(c2cccnn2)=O)CC1NC(=O)COC1CCCOC1 85642,c1(CCNC(C(c2ccco2)NC(COC(CC)C)=O)=O)c[nH]nc1O 85643,c1(-n2c(C3CCC(OC)C3)nc(-c3ccoc3C)n2)cc(F)cc(F)c1 85644,C1(C(N2CC3C(CNC(=O)C4=CCCCO4)(C3)C2)=O)CCC2(CCC2)CC1 85645,C=CC(C)(CC)C(=O)NC1C2CC1N(C(c1ccsc1OC)=O)C2 85646,C(=O)(C1(C)CCn2ccnc21)N(C)CC1(O)CCN(C(=O)COc2cccnc2)C1 85647,Cc1cc(=NC2C(C)C2C)[nH]c(=NCC(=O)N2CCN(C)CC2)[nH]1 85648,c1(C(N2C(C)CC(CNC(=O)C(C)(C)CC3CCOC3)C2)=O)cnc(O)c(F)c1 85649,C1(C)(CNC(c2cnc(CC)[nH]2)=O)CCN(C(=O)C(C)C(C)O)C1 85650,c1(C(=O)NCCOC2CN(C(C(CN(C)CC)F)=O)C2)cccc(COC)c1 85651,C(=O)(CC(=O)N1CC(NC(C2CC(OC)C2)=O)C1)OCC 85652,c1(C(=O)OC)cc(C(N2CCC(CNC(=O)COc3ccsn3)C2)=O)cc(F)c1 85653,C1(NC(CCC#CC)=O)CN(C(c2cccc3ccoc23)=O)C2(CCCC2)C1 85654,CCCC(C)CC(=O)N1CCCC1CN(C)C(C1(C(O)C(F)(F)F)CCC1)=O 85655,c1(C(=O)NC(C)(C)CNC(=O)C=CC(=O)NC2CC2)ccc(C(O)CF)cc1 85656,n1(CC(=O)NC2CC(CCNC(=O)Cc3cnoc3)C2)sc(=O)c2ccccc12 85657,Cc1cc(C(=O)NC(CO)C(C)NC(=O)C(c2ccc(Cl)cc2)O)cc(C)n1 85658,C(C#Cc1cccnc1)NC(c1cccc(-c2cccs2)c1)c1n(CC)nnn1 85659,Cc1ncc(CCC(N2CCN(C(=O)CCNS(C)(=O)=O)C3CC23)=O)c(O)n1 85660,C=C(C)CC(C(=O)N1CCC(CNC(=O)CN(C(=O)C(C)C)C)(OC)C1)OC 85661,CC1OCCC1CCNC(=O)CNC(=O)CC1CCOCC1 85662,O=C(CC1COCCO1)NOC1CCN(C(=O)CSC2CC2)C1 85663,c1(C(=O)OCCCNC(C#CC(C)C)=O)cccc(S(=O)(=O)NC(C)C)c1.OCCC 85664,c1(C(=O)N(C2CC2)CC2CCCCO2)cc2c(=O)cc[nH]c2s1 85665,CC1(C)CC(CO)CN1C(=O)CN(C1CC(C#N)C1)C(=O)CC1CNC(=O)O1 85666,CC(C)(C#N)CC(=O)NC(C)(C)CCNC(c1cc(F)cc(Br)c1)=O 85667,C1(C(N2CCC(CC(=O)NC)C2)=O)C(O)CCN1C(=O)C=CC1CC1 85668,C(Cc1cc[nH]n1)(C(=O)NCC1(C)CNC(=O)O1)NC(CCC=C(C)C)=O 85669,c1(C(=O)NC2C(F)CCN(C(C(C)c3cccs3)=O)C2)cc2ccc(F)cc2[nH]1 85670,C1(CO)CCN(CCn2cc(-c3ccncc3F)nn2)CC1(F)F.N1CCOC1=O 85671,C(=O)(CCCC(=O)NC(C)CN(C)C(c1nccnc1Cl)=O)NC(C)C 85672,N1(C(CC=CC=C)=O)CC2C3CCC(C2C1)N(C(=O)CCc1ccnn1C)C3 85673,c1(OC)nn(C)cc1C(=O)N(C1CC1)CC1CCCN1C(c1ccc(C)s1)=O 85674,c1(C(=O)NCC2CC(NC(=O)C=CC3CCOC3)C2)cc2c(cn1)CCCC2 85675,Cc1c(C(=O)NC(C)(CNC(C23COCC2C3)=O)C2CC2)cnn1C1CCC1 85676,C=CCC(CNC(C1C(C)C1(F)F)=O)NC(=O)Cc1csc(NS(C)(=O)=O)n1 85677,c1(OC)cc(N)c(C(=O)NCCC2(OC)CN(C(=O)C3=CCCCO3)C2)cc1F 85678,N1(C(CCN(CCCCC)C)=O)CCN(C(C2(C)CC=CCC2)=O)CC1C 85679,C12(N(c3cccs3)C(c3ncc(-c4ccc(C)cc4)[nH]3)=O)C3CC(CC13)C2(F)F 85680,C(CC(C(C)C)NC(C1(NC(=O)CC2CCCC2O)CC(O)C1)=O)OC 85681,N1(C(c2c(C)n(C)nc2)=O)CC2CN(C(c3cc4c(s3)CCOC4)=O)CC2(C)C1 85682,c1(C(=O)NCC(CC)NC(c2ccc3snnc3c2)=O)cccn2cc(C)nc12 85683,N1(CC2OCC(=O)C2c2ccccc2)CCn2c(C(=O)O)nnc2C1 85684,N1(Cc2c(C)n[nH]c2C)CC2CCC(NC(=O)CCCC(=O)N3CCCC3)CC2C1 85685,C(C(CN=c1cc(C(N)=O)nc[nH]1)C(F)(F)F)NC(C(CC)N(C)C)=O 85686,c1(C(=O)NC2CN(C(CCc3c(C)cccn3)=O)CC2C)nnn2c1CSCC2 85687,c1(OCCSCC(=O)NCC(C)NC(CC(=O)OCC)=O)ccccc1COC 85688,C(=O)(C(C)(C)CS(N)(=O)=O)NCC1CC(C)CC(C)C1 85689,CC1CN(C)CC(C(=O)NCC2(NC(c3cc(=O)cc(Cl)[nH]3)=O)CCC2)O1 85690,c1(C(=O)NCC2(CNC(C3CCC(F)C3)=O)CCCC2)cc(F)ccc1Cl 85691,Cn1ncc2c(O)nc(=NCCCOCCNC(=O)C(N3CCCC(O)C3)C)[nH]c12 85692,c1(SC)cscc1C(N1CC(C(=O)NCCNC(C23CC(CO2)C3)=O)C1)=O 85693,C(N=c1[nH]nc(C)o1)C1CCCC(NC(c2cc(OC)no2)=O)C1 85694,N1(C(c2c(CCC)occ2)=O)CCN(C(=O)C(O)Cc2cnn(C)c2)CCC1C 85695,CC(CC#N)C(=O)NC1CCCC1C(N1CC(N=[N+]=[N-])C1)=O 85696,C1(C(=O)NC2C(NC(c3cc(C)sc3)=O)CCC2)OCCOC1(C)C 85697,N1(C(c2cnc(CC)nc2C)=O)CC2CN(C(C3CC3C3CC3)=O)CCC12 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85750,C12(CNC(C(CCSC)O)=O)CC(C(N)=O)(C1)C1(CN(C(=O)C=CC(C)=O)C1)O2 85751,C1(NC(c2csc(C)c2N)=O)CCC(C)N(C(=O)C=CSc2ccccc2)C1 85752,CCCC(C)(O)CC(=O)N(CC(C)C(=O)Nc1c(C)cccc1C)C 85753,C12(CC(=O)NC3CN(C(=O)Cn4nnc(=O)[nH]4)CC3O)CCC(CC1)OC2 85754,N1(C(CCCn2cc(-c3occ(C(=O)O)n3)nn2)=O)CCC(O)C(F)(F)C1 85755,CCC(C)CCCCC(=O)N1CC(OCCNC(c2c(F)cc(O)cc2F)=O)C1 85756,C1(C)(CNC(C23CC(C(=O)OC)(C2)C3)=O)CN(C(c2ccc(O)nc2)=O)CCO1 85757,C1(C(N(CC)Cc2ncc[nH]2)=O)CC(NC(=O)C=CCCC(C)C)C1(C)C 85758,c1(CNC(=O)NC(c2nc(C)sc2C)C(C)(C)C)ccc(C)c(Br)c1 85759,N1(C(CCCSC)C(=O)Nc2ccccc2Cl)CCC(CO)C(O)CC1 85760,C(C)(c1ccc(OC)cc1)=CC(=O)NCC(C)(CC)NC(C1C(=C)CC1)=O 85761,C1(O)(CNC(CCN(CCCCC)C)=O)CCCN(C(=O)C(F)C(C)C)CC1 85762,C1(C)(CC)C=C(C(=O)NCCN(C(=O)C(N2CCP(C)(=O)CC2)C)C)C1 85763,CC1(C(=O)Nc2ccns2)CC12CCN(CC(N1Cc3ccccc3C1)=O)CC2 85764,c1(CC2CCOC2)ccccc1.C1(=O)CC2(CC2)C(=O)N(C)CCOCCN1C 85765,c1(OC)ccc(C)cc1C=CC(N1CCCCC1CNC(c1n[nH]cc1C)=O)=O 85766,N1(C(C2CC3CC3N2C(=O)CCN2CCCCC2)=O)CC2(CCOC2=O)C1 85767,c1(C(N2C3CN(C(C(C=C)(C)CC)=O)CC2C3)=O)coc2ccc(F)cc12 85768,C1(NC(C23CC(CC)(C2)C3)=O)CN(C(=O)CCC(=O)c2cccc(F)c2)CC1O 85769,N1(CC(=O)NCC(n2cc(-c3cc(C4CC4)no3)nn2)C)CCC(=O)CC1 85770,C1(C(=O)NCCN(C(C(Cc2ccc(OC)cc2)O)=O)C)CCN(C)S1(=O)=O 85771,C1(C(=O)N(CC(O)CNC(=O)COC2(C)CCOCC2)C)(OC)CCC12CCC2 85772,N1(C(c2cc(CCC)oc2C)=O)CCC(C)C(N(C(=O)C(C)OCC(C)C)C)C1 85773,c1(NC(C2N(C(CCOCC#C)=O)CCCC2)=O)ccc2oc(CO)cc2c1 85774,c1(C(CC)C)nccc(=NCCNC(C2CC2CC)=O)[nH]1 85775,C12(CNC(C(CN(C)C)NC(C3CC(O)(C(C)C)C3)=O)=O)CC(CN1C)C2 85776,O(N(C)C(=O)CCc1cnc(C)[nH]1)CC(=O)OC 85777,Cc1ccsc1CC(=O)NC1(CNC(=O)C(C)CN(C)C)CCOC1 85778,C1(C(N2CC(=C(CNC(C(C)(C)C3CCCCC3)=O)F)C2)=O)CCCCCC1 85779,C1(c2scc(C)n2)CN(C(=O)Cn2cc(CN(C)C)nn2)CCO1 85780,N1(C(CC(=C)Br)=O)CC(NC(=O)CCOc2ccc(Cl)cc2)CC1CO 85781,CC1(O)CCN(C(=O)CCCNC(=O)CC2(N(C)C)CCC2)CC1O 85782,N1(C(C(c2nc(F)ccc2Cl)C)=O)CCSCc2ccccc21 85783,C(C)(C)(CCCNC(C1NC(=O)CC1C)=O)NC(COCc1nnc(C)s1)=O 85784,C1(C)(CC)CCN(c2nccc(C(C)(F)F)n2)C1 85785,CCCCC(F)(F)C(=O)NC(CC1CCCC1)C(=O)NOCC(=O)OCC 85786,C1(S(C)(=O)=O)(C(=O)NC2CCC(C)N(C(C3CCC(=O)N3)=O)C2)CCOCC1 85787,c1(OC)c(C)cc(C(=O)NC2CCC(CNC(c3cccc(C)n3)=O)C2)cc1C 85788,C(=O)(NNC(=O)c1cccs1)C1CC(CC(C)(C)C)C1.C1CCCC1 85789,C1(NC(c2c(CNC(Cc3cc(C)[nH]n3)=O)noc2)=O)CCCC1(C)O 85790,c1(OC)ccc(C=CC(=O)NC2CCCC2NC(c2cccn2C)=O)c(C)c1 85791,C1(=O)C(CCC2CC2)N1.C(=O)(C(C#N)C1CC1)NC.N1(CC)CC1 85792,C1(C(N2C(C=C)CC2)=O)CC2C=CC1N(C(=O)CCCOCC)C2 85793,O1P(C)(=O)COC2=CC=CC=CC(CC2C)N(C)C(=O)C1 85794,c1(C(N2C3(CNC(C4(O)CCC(CC)C4)=O)CC(C2)C3)=O)c(C)[nH]c(C)c1C 85795,O=C(C(O)CC(F)F)N1CCN(C(=O)CCC2CCCCO2)CC1 85796,C1(OC)(CNC(=O)CCSc2ccccn2)CN(C(C2CC2(C)C(F)F)=O)C1 85797,N1(C(CCOCC(C)(C)C)=O)CCOCC(C(=O)NCCCCF)C1 85798,C1(NC(C2CN(C(C)C)C2)=O)CN(C(C2CC3(CSC3)C2)=O)CC1N=[N+]=[N-] 85799,Cc1nc(C)c(C(N2CCOC(CNC(C3CC3(C)C)=O)C2)=O)o1 85800,N1(C(c2cccc(COC)c2)=O)CC(NC(c2cccc(OC)n2)=O)CC(C)C1 85801,CCC(C)C(C(=O)NC1CCCC1C#N)NC(=O)C(N1CCCCC1)C 85802,C(=O)(C(C)(CC)OC)NCC(CC=C)NC(c1ccoc1Br)=O 85803,c1(CC)cccc(CC)c1CC(=O)Nc1nc(C)c(CSc2ccccc2)s1 85804,Cc1cnc(C(=O)NC2C=CCN(C(=O)C(c3ccc(F)cc3F)=O)C2)cc1C 85805,CC(C)CC(C(=O)NC1CCN(C)C1)ONC(=O)c1cc[nH]c1 85806,c1(C(=O)NC23CN(C(CC(=O)NCC#C)=O)C(C2)C3)cc[nH]c(=NC)c1 85807,C1(OC)CC(CNC(C2CCCC3CC23)=O)N(C(c2ccoc2Cl)=O)C1 85808,C(=O)(CCCC(C)C)N1CCN(C2CN(C(CS(CC)=O)=O)C2)CC1 85809,C1(CC(=O)NCc2ccccc2CNC(c2ccncc2O)=O)CCC1C1CC1 85810,Cc1c(C(N)=O)cccc1C(=O)NCC1(O)CCN(C(C2CCC(=O)O2)=O)C1 85811,CC(CN(C)C)CCC(=O)N1CC2C(C(=O)NC(C)Cn3cnnc3)C2C1 85812,N1(C(COC(C)C)=O)CCC2CCCC12CNC(=O)C(F)(F)CO 85813,C(=O)(C1CSc2ccccc21)N(CCCN(C)C(c1n[nH]cc1Br)=O)C 85814,C(CC(C(=O)NCCCCC1CC1C)N(C)C)NC(CC1C(CC)C1)=O 85815,N1(C(c2csc(Cl)c2)=O)CCCC(C2CC2NC(C2(CO)CCCO2)=O)C1 85816,c1(C(N2CCC(CN(C(C3CC(OC)C3)=O)C)C2)=O)nc2c(cc1Cl)OCCO2 85817,N1(C(C)=O)CCCC1CNC(C1CC(NC(=O)CCC=CC(C)C)C1)=O 85818,N1(C(C2(N(C)C)CCC2)=O)CC2(C1)CN(C(=O)CCc1cccc(F)c1Cl)C2 85819,c1(CN2CCCC(C(=O)NC(c3nnc(C)o3)C)C2)ccc(F)c(Br)c1F 85820,N1(C(C=CCN(CC(F)(F)F)C)=O)CCC2CN(C(C3CCCO3)=O)CC2C1 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86031,N1(C(CCCCC=CC)=O)CCC(C2CCN(C(=O)COCC(F)F)C2)C1 86032,c1(SCC=C)n[nH]c(=NC(=O)N2CCOC(C(c3ccccc3)O)C2)s1 86033,c1(N(C)CCO)cc(C(N2CCC2CNC(=O)Cc2nnc(S)n2C)=O)ccn1 86034,C(=O)(C1=CCOCC1)N1CCC(CCNC(c2cccc(F)c2F)=O)C1 86035,C1(NC(C(c2cccs2)OCC)=O)CC2CN(C(c3sccc3OC)=O)CC12 86036,N1(C(C2CCCN(C(C(C)S(C)(=O)=O)=O)CC2)=O)CC2CC(C)(C)C2C1 86037,c1(CN(C(Cc2ccc(C)o2)=O)CCNC(C2COCCO2)=O)ccc(Cl)nc1 86038,c1(C(=O)NCC(C(C)C)(C)NC(=O)C=CC2CCC2)c(F)cccc1Br 86039,CC#CCC(C(=O)NCC(O)CC1CCC1)NC(=O)CCc1ncnn1C 86040,C(C1CSc2ccccc21)N(C(=O)N=c1nc(C(F)(F)F)[nH]s1)CC 86041,C(CCCCCC(=O)N(C(C(F)(F)F)C1CC1)C)n1cc(COCC(C)O)nn1 86042,CCC(CC(=O)NC(C)C(C)C(=O)NCCc1cc(C)on1)C(F)F 86043,C1(C2CCCN2C(=O)OC(C)(C)C)C=CCN(N(CCC(=O)OC)CC#C)C1.C(C)=O 86044,CCCC(C(=O)NC1CCCCC1NC(=O)C(C)(C)OCC(F)(F)F)S(N)(=O)=O 86045,Cc1ccc(C(N)=O)c(NC(=O)C(=O)NCCCSc2ccc(C)o2)c1 86046,C1(NC(c2cncc(-c3ccccc3F)c2)=O)CCCC(C(F)F)CC1 86047,c1(C(=O)NC2CN(C(Cn3nc(C)oc3=O)=O)C(C)C2)cnc2ccncc2c1 86048,C1(NC(C(C)N(CCC)C(c2nnccc2C)=O)=O)CN2CCC1(F)CC2 86049,N1(C(C(CC2CC2)OC)=O)CCN(C(=O)COC(C)C(C)C)C2(CC2)C1 86050,C1(CNC(C(C)(C)NC(=O)NCC)=O)COCCN1C(c1cnc(OCC)s1)=O 86051,CC1CN(Cc2ncc(Br)cn2)c2ccc(C(F)(F)F)cc2O1 86052,C(=O)(C#CC1CCCCC1)N1CC(C(=O)NCC2(CCOC)CC2)OC(C)C1 86053,CC1CC(CNC(C2(C)C=CCCC2)=O)CCN1C(c1cc2scnc2[nH]1)=O 86054,C(=O)(CCC(C)C)N1C2CCCN1C2.C1(C=O)C2CCC1(c1ccnn1C)C2.CO 86055,C(=O)(CC(O)CC(C)(C)C)N1CCCC(C(=O)NC2(C3CCCC3)CC2)(CC)C1 86056,c1(CC(C(=O)N(CC(CNC(COC(C)=O)=O)O)C)C)c(C)noc1C 86057,CCN=c1[nH]c(C(=O)NCC2CCC(C)CN2C(c2nccc(Cl)c2F)=O)cs1 86058,Cc1cc2ccc(C(=O)NCC(C3CC3)NC(=O)CN3CCCC3C)cn2c1 86059,CC(C)(C)CCCCCC(=O)N1CCN(C(=O)C#CC2CCC2)CC1C(F)F 86060,O=C(C(O)COC(F)F)NCC(=O)NC1CN(C(c2cocn2)=O)C1 86061,C(c1cncnc1O)=CC(N1C(CN(C(C2(C)C(C)OCC2)=O)C)CCC1)=O 86062,O=C(C(C(F)(F)F)C(F)(F)F)NCC1(F)CC(CNC(C2CC2Cl)=O)C1 86063,Cc1cc(Cl)cc2cc(C(N3CCC(C)C3CNC(C3(CO)CC3)=O)=O)[nH]c12 86064,C1(CCOC)(NC(CCCOCC)=O)CCN(C(C2CCC(O)CC2)=O)C1 86065,c1(OCC=C)cccnc1C(=O)NCCC1CCC(NC(c2cc(C)co2)=O)C1 86066,C(CN=c1[nH]c2ccc(S(=O)(=O)NC(C)CC#N)cc2s1)c1nccc(OC)n1 86067,c1(C(N(C(C)CNC(=O)Cc2cccc(OC)c2)CC)=O)cc2sccc2[nH]1 86068,Cc1nc(-c2cccs2)sc1NCCOC1CNC(=O)C1 86069,C=C(C)CC(C(=O)OC)NC(C1CC=CC(n2cc(C(CC)OC)nn2)C1)=O 86070,C1(CC)CN(C(=O)C=C(C)C)CCC1NC(C1CC(F)(F)C1(C)C)=O 86071,CC1CC(=O)NCC1C(N1CCCN(C(=O)CCC23CCC(CC2)C3)CC1)=O 86072,N1(C(C(=O)NCSc2cccc(F)c2)C2C(C)C2)CCC(C(N)=O)CC1 86073,C1(NC(=O)Cc2ccc(Cl)nc2)CN(C(C2(F)CCC2)=O)CC2(CC2)C1 86074,CC1CN(C(=O)CC2(N(C(=O)C(n3cc(Cl)cn3)C)C)CC2)CC1N(C)C 86075,C1(C(=O)NCCC2C=CCC2)C2CC1N(C(C1(C(F)(F)F)CC1)=O)C2 86076,C1(NC(=O)C2CC2)CC(CO)C12CCC2.C1(C=O)CCOC1=O 86077,C1(NC(CC(CC=C)NC(c2cncc(C)c2)=O)=O)COC2(CCCC2)C1 86078,N1(c2cccc(S(=O)(=O)NCCC(=O)NC(C)C)n2)CCCC2(CCN(C)C2)C1 86079,C1(N(C)C(c2n[nH]cc2Cl)=O)CCCN(C(C2CC23CC3)=O)CC1 86080,C1(CNC(COCC=C)=O)CN(C(C2(NC(C)=O)CCC2)=O)C(C(F)(F)F)CO1 86081,C1(NC(c2ccc(COC)[nH]2)=O)CC2CC(C1)N(C(=O)CC1NC(=O)NC1=O)C2 86082,c1(NS(C)(=O)=O)ccccc1NC(=O)C(N1CCCCC1CO)=O 86083,c1(C(N(C(CN(C(CCOCCCOC)=O)C)C)C)=O)ccccc1 86084,N1(C(CC2(CSC)CC2)=O)CCCN(C(=O)Cc2ccnn2C)CC1C 86085,N1(C(CCCC2(NC(=O)C=C(C3CC3)C3CC3)CCC2)=O)CCOCC(C2CC2)C1 86086,c1(C(C)(C)C)noc(CCC(=O)NC2CC2CNC(c2cc(C3CC3)no2)=O)n1 86087,C12(C(=O)NCCOCCOC)CC(CN(C(C3CCSC(C)C3)=O)C1)C2 86088,N1(C(c2c(C)cc(=O)n(C)n2)=O)CCC2CN(C(c3cnc[nH]3)=O)CC2C1 86089,C(=O)(CCCN(C)C)NC(C1CCCN1C(c1ncsc1Br)=O)C 86090,c1(C(=O)NCCNC(c2c(C)nccc2Cl)=O)ccc([N+](=O)[O-])c(S(N)(=O)=O)c1 86091,N(C(=NC(C)CN(C)C)N(C)Cc1ccccc1)C(COC)C 86092,Cc1ccc(Cl)c(C(=O)NC(CNC(C2(C(F)F)CC2)=O)CC(C)C)c1N 86093,c1(OC)cccc(C(N2CCCC(N(C)C(C3COCC3(C)C)=O)C2)=O)n1 86094,C(C)(N=c1[nH]c2c(c(=NCCNC(=O)C3CC3)[nH]1)COC2)c1cc(C)c(F)cc1 86095,C1(NC(C2(C(=O)OCC)CCO2)=O)CC2CCC(C1)N2C(=O)C(C)CC(F)(F)F 86096,N1(C(C2C(=C)C2)=O)CCCC(C(=O)Nc2cnn(C(F)F)c2)CC1 86097,C1(C(=O)NCCOCCNC(c2ccncc2)=O)(C(=O)O)OC2CCC1CC2 86098,CC1CN(C(C2(CF)CCC2)=O)CCC1CNC(c1nccc(C(F)(F)F)n1)=O 86099,C1(C(=O)NCC(C)N(C(c2[nH]cc(C)c2)=O)C)CCCCN1C(C1CCCC1)=O 86100,c1(C(N(C(C)CC(=O)NOCC(=O)N(C)C)C)=O)cc2cc[nH]c2cn1 86101,C1(NC(C(CC)(C)F)=O)COC2(C1)CN(C(=O)C(C)(C)C(=O)OC(C)(C)C)C2 86102,C1(C(N2CC(OCC)(CNC(c3cnc(CC)nc3)=O)C2)=O)CCOCC1(C)C 86103,N1(C(c2ncc(OC)cn2)=O)CCC2(C1)CN(C(c1cc(Cl)c(Cl)s1)=O)C2 86104,c1(OC)ccc(F)c(NC(=O)C(C)(CSC)NC(=O)CC(C)C)n1 86105,C1(CC(=O)NCC2CC(NC(=O)Cn3cnnc3)C2)CC2(CCC2)CCO1 86106,Cc1cc(C(N2CC(O)(CN(C(=O)CC(c3ccccc3)N(C)C)C)C2)=O)co1 86107,N1(C(C2(C)CC2)=O)CC2(CCN(C(C3(c4cccnc4)CCCCC3)=O)CC2)C1 86108,c1(OC)ccc(C(N2CCCC2CC(N2CCc3sccc3C2)=O)SC)c(F)c1F 86109,C1(CCNC(C=CSC)=O)CCCN(C(=O)CC2COC(C)(C)CO2)CC1 86110,C1(NC(c2cc(OC)ncc2)=O)(CNC(c2ccc(Cl)cc2)=O)CCCCC1C 86111,CC1(C)C(CC(=O)NC2(C)CCN(C(c3ccccn3)=O)C2)C1(C)C 86112,N1(C(CC(CC)SC)=O)C2CC=C(C(=O)NCC3C(C)C3(F)F)C1CC2 86113,N1(C(C(C(C)C)CO)=O)CC2(CCC2)CC1CNC(=O)COC1(C)CCOCC1 86114,c1(NC)cnccc1C(=O)NCC=CCC(=O)N1CCC1C(N)=O 86115,C12(CNC(C3(CCCC)CC3)=O)CCC1CN(C(=O)C=Cc1ccc(C)s1)C2 86116,N(C(=NCC1CC1)N1CCC(CN2CCOCC2)C1)CC1(S(C)=O)CC1 86117,C1(F)(CNC(c2c(C)nc(C(C)C)o2)=O)CC(N=c2[nH]cnc3cc(Br)sc23)C1 86118,c1(NC(=O)NC2CCC(NC(c3nc(C(=O)OC)sc3)=O)C2)cccc(C#N)c1 86119,CC(CC(=O)NCC1(F)CN(C(C2(F)CCOC2)=O)C1)c1ccncc1 86120,CCCCCCCCCC(=O)N1CC(C)(NC(=O)C(c2ccccn2)O)C1 86121,N1(C(=O)NC)CCN(C(C2(Nc3ccc(-c4nn[nH]n4)cc3)CC(F)(F)C2)=O)CC1 86122,C12CCCCC1C(=O)N2.C(CCN=[N+]=[N-])OCC(N1CC(C(CO)OC)C1)=O 86123,C1(CNC(c2cccc(O)n2)=O)CCN(C(c2cnnc(O)c2)=O)CC1O 86124,Cc1ccc(CCCN2CC(COCCNC(=O)C(C)(C)C3CCCO3)C2)cn1 86125,C(=O)(C(C)C(CC)CC)N(C1CCN(C(c2c(CCC)n[nH]c2)=O)C1)CCC 86126,N1(C(c2c(C)nc(C)s2)=O)CC(NC(=O)COCC(F)F)C(C2CC2)C1 86127,c1(N(CCNC(=O)C(C)CC2CCC2)CC)ccc(F)cc1C#N 86128,C1(NC(c2nc(C(C)C)sc2)=O)CCCC1(C)NC(=O)C(C)C1CC1 86129,c1(C(=O)NCCC(=O)NC2C(CNC(C(CC)NC(C)=O)=O)C2)ccc(C)cc1 86130,Cc1[nH]c(=N)nc(O)c1CCC(=O)NCC1CN(C(=O)CCC2CCCCO2)C1 86131,c1(NC(=O)NCC2(c3ccc(OCC)cc3)CCCCC2)c(Cl)nc(C)nc1Cl 86132,C1(N2C(C(=O)NCc3ccn(C)n3)CCC2)CCN(C(c2ncccn2)=O)CC1 86133,n1(C(C)C)cnc(C(=O)NC(C)(C)CNC(=O)Cc2cncs2)c1 86134,N1(C(c2n(C(CC)C)ncc2)=O)CCCC(NC(C2CC2OC(C)=O)=O)C1 86135,N1(C(C2C(C)C2C)=O)CCN(C(=O)C(Cl)=CCl)CCC1C 86136,C1(NC(c2cc(C)n(C)n2)=O)CN(C(=O)C(Cl)=CCl)C2(CCCCC2)C1 86137,N1(C(C2C(C(N)=O)C2)=O)CCN(C2CCCN(C(c3ccco3)=O)C2)C(=O)C1 86138,CC1(c2cn(-c3ccccc3Br)nn2)CCN(C(C2CC2(C)C(F)F)=O)C1 86139,C(CCCC#N)(c1nnnn1C1CC1)NC(c1ccc(N2CCCCC2)cc1)C 86140,c1(C(N(CC(CC)NC(=O)C=CCn2cncn2)C)=O)ccccc1C(C)(C)C 86141,N1(C(Cc2c(COC)cccc2)=O)CCN(C(=O)C2=NOCC2)C2CC12 86142,C12(C(=O)NCC(C)(O)CCO)CCC1CN(C(=O)CCOCC(F)F)C2 86143,CCCC(CNC(C1C=CCCN1C(c1ccccc1C)=O)=O)CCO 86144,c1(C(N2C(CN(C(CC(C)SC)=O)C3CC3)CCC2)=O)sc2nccnc2c1N 86145,C=CCC(CNC(C1CCC(C)(C)CC1)=O)C(=O)Nc1cccc(OCC)c1 86146,N1(C(C(CC)N(C)C)=O)CC(NC(c2ccnc(OC)c2)=O)C2CCCCC12 86147,N1(C(c2c(C)cco2)=O)CCC(N=[N+]=[N-])(C(=O)N(C)CC2CC2(C)C)C1 86148,c1(C(N2CCC(N(C(=O)C(O)CC)CCC)C2)=O)cn(C)c(=O)nc1O 86149,C12(CNC(c3cccc(C)c3)=O)CCCC1CCN2C(c1cccc(O)n1)=O 86150,CCN=C(NCCCC(C)(F)F)NCCC1CCCC1(C)C 86151,Cc1ccc(C(=O)NC(C(=O)N(C)Cc2cnco2)C(C)C)c(C)n1 86152,C1(CNC(C2(O)C(C)(C)C2)=O)CCC2(CO1)CC(NC(c1cc(O)ncn1)=O)C2 86153,N1(C(c2cnc(C(C)C)nc2)C(=O)Nc2c(C)cccc2)CC2CC3CC2C1C3 86154,c1(C(N2C(C)CC2C(=O)N(CCF)C2CC2)=O)cc[nH]c(=N)n1 86155,c1(OC)ccc(C(N)=O)cc1C(=O)NCC(C)(C)NC(=O)C=CCO 86156,Cc1cc(C(=O)NC(C2CCCCC2)CNC(C2CC(=O)N2)=O)ccc1[N+](=O)[O-] 86157,c1(OC)ccc(C=CC(=O)NC2(C)CCN(C(=O)C(C)C(C)(C)C)C2)cc1F 86158,c1(C(N2CCCCC(NC(C3C(C)C3)=O)C2)=O)cccnc1S(=O)(=O)C(F)(F)F 86159,c1(CC)ncccc1C(=O)N(C1CCC(NC(c2cccnc2)=O)C1)C 86160,c1(SC)ncc(C(=O)NC2CC(NC(C3(n4ccnn4)CC3)=O)C2)c(O)n1 86161,c1(C(=O)NC(C(=O)NC2CC(C(C)C)OC2)CC2CC2)ccn2ccccc12 86162,c1(C(N(C(CNC(c2c(C)ccc(Br)c2)=O)C)C)=O)coc2c(C)cccc12 86163,C=C(C)CC(C(=O)N(C1CCCN(C)C1)C)NC(c1cc(OC)ccn1)=O 86164,CC1CC(NC(c2cccc(=O)o2)=O)CN1C(=O)Cc1ccccc1Br 86165,N1(C(COCC(=C)C)=O)CC(NC(=O)COCc2ccccc2)CC(O)C1 86166,Cc1ccc2snc(C(N3CCC(O)(CNC(=O)C(C)CC(F)F)C3)=O)c2c1 86167,c1(C(N2CC3C(CNC(CC(C)(C)C4CC4)=O)(C3)C2)=O)cc(O)ccc1Cl 86168,S(=O)(=O)(c1cnc(NCC23CCCC2OCC3)c(Cl)c1)NCCCN(CC)CC 86169,c1(C(=O)NC2CCN(C(CCC(=O)NCC)=O)CC2F)cccn2c(C)nnc12 86170,c1(C(=O)OC)c[nH]ccc1=NC(=O)CC1CC(OC)C1.C12CN(CCO1)C(=O)C2 86171,CC(F)(F)CCNC(=O)CC1CCN(C(=O)CSCC(N2CCCC2)=O)C1 86172,CC1(NC(c2coc(Br)n2)=O)CCN(C(=O)CCCn2ccccc2=O)C1 86173,N1(C(CCC(=O)OCC)=O)CCC(CO)C(NC(=O)CCCn2ccnn2)C1 86174,N1(C(C(CC)O)=O)CC2CC3CC2C1C3NC(=O)CCc1cscn1 86175,N1(C(CC=CCC)=O)CC(NC(=O)Cc2ccc(Cl)s2)C(C#N)C1 86176,N(C(=NCCc1nc2c(s1)CCC2)NCC1CCC1)CC(C(C)C)N1CCCC1 86177,c1(CC(=O)N(CCC(C)NC(c2c(OCC)cccn2)=O)C)cc(C)cc(C)c1 86178,N1(C(C(C=C)(C)O)=O)CC2CC(NC(c3ccc(CC)c(Br)c3)=O)C1C2 86179,C1(C(=O)O)CCCC(CNC(c2occc2-c2ccccc2)=O)C1 86180,c1(C(=O)NC2C(CNC(c3cccc(C(=O)NC)c3)=O)C2)ccc(Cl)c(N)c1Cl 86181,N(C(=NCCF)NC(c1cc(Cl)ccc1O)=O)CC1CCN(C)CC1 86182,c1(N(CCCNC(=O)CC(C)C2CCCO2)CC)ncncc1OC 86183,CC(C)(CCCNC(=O)CC(F)(F)F)C(=O)NCC1CCC(=O)N1 86184,c1(OC)cc(C(=O)NC(C)(C)CCCNC(C23CCN(CC2)CC3)=O)cc(F)c1 86185,c1(N2CCC(CSC)C2)nccc(=NC(C)COC2CCCC2)[nH]1 86186,N1(C(CC2(C)CC2)=O)CCC(O)(C(F)(F)C(N)=O)C1.n12cc(nn1)C2 86187,CN(Cc1cc(-c2cccc(Br)c2)no1)N1CC(C2(C)N=N2)C1 86188,N1(C(C2C(COC)CC2)=O)CC2CC2(NC(C2CC(C(C)C)C2)=O)C1 86189,c1(C(N2C(C)C(=O)NCC2)C(=O)NCc2ccco2)cc2ccccn2n1 86190,N(C(=NCCCC(C)(F)F)NC(C)C1CC1)C(c1cccnc1)C 86191,C1(CC(=O)NC(C=C)(C)C)CN(C(C2CC3C=CC2CC3)=O)CCC1C 86192,c1(OCC)cc(Cc2nc(CC)n(-c3c(F)cccc3Cl)n2)ccc1C 86193,C(CCCC#N)(c1nnnn1C1CCOCC1)NCC(C)OCC 86194,N1(C(C(CO)OC)=O)CC(CNC(C23CCCC2OCC3)=O)CC12CCC2 86195,c1(CC(C(=O)O)n2cc(CC(CC(=O)C3C(C)C3)N)nn2)cccc2ccsc12 86196,C(=O)(C1=COc2ccccc2O1)N(C1C2CN(C(c3cnc(C4CC4)[nH]3)=O)CC12)C 86197,N1(C(CN2C(C)CCC2)=O)CCC(N(C(=O)COc2ccc(F)cc2)CCO)CC1 86198,c1(C(N2CC(C(C)NC(C3(CC=C)CC3)=O)OCC2)=O)cc2c(cn1)OCCO2 86199,C=C(Br)CCC(=O)NC1CCC(CNC(c2ccc(C(F)F)nc2)=O)C1 86200,Cc1c(O)c(=O)ccn1CC(N1CC2CC(NC(=O)C(F)C3CC3)C1C2)=O 86201,c1(C(=O)NC2(C)CC(NC(C3(Cl)C(C(C)=O)C3)=O)C2)c(C(C)C)cnn1C 86202,Cn1cnc2cnc(N3CC4CC3CCC4NC(=O)COCCN(C)C)nc12 86203,C(CC(C(C)(C)C)NC(=O)C(C)OC1CCOC1)N(C(c1c(C)noc1N)=O)C 86204,CC(C)(CC(=O)N1CC(NC(C2CCCCN2N=O)=O)CC(F)C1)CC(F)F 86205,C1(NC(C(C)O)=O)CC2(C1)CC(NC(c1c[nH]cc(F)c1=O)=O)C2 86206,c1(C(N(CCCNC(C2CCC=CCC2)=O)CCO)=O)ccnnc1S 86207,C1(NC(C(CCC)F)=O)Cc2ccccc2C1NC(=O)CC1C=CCC1 86208,CC(Cc1ccccn1)N=c1[nH]c(=NCCN2CCC(O)C2)c2sccc2[nH]1 86209,N1(CC(=O)N(C2C(NC(CCN(C(C)=O)C)=O)CCCC2)C)CCN(C)C(=O)C1 86210,c1(N2CC3C(NC(C(C(C)C)SC)=O)C3C2)ncnc2ccccc12 86211,c1(C(=O)NC2C(NC(Cn3ncn(C)c3=O)=O)CCC2)c(N)cccc1[N+](=O)[O-] 86212,C(C(C(=O)N1CCCC1CCNC(c1ccc2c[nH]nc2c1)=O)C(F)(F)F)OC 86213,c1(C(N(C2C(C)CCN(C(=O)CC3(C)CC3)C2)C)=O)ccc(Cl)c2ccccc12 86214,C1(NC(C(c2c(C)nn(C)c2)C2CCCCC2)=O)CCC2CN(C(C)C)CC2C1 86215,C#CC1CN(C(=O)CCc2nncn2C)CCN1C(=O)COCCN(C)C 86216,N1(C(C2(C(=O)OCC)CC2)=O)CC(C(=O)NC2CCCC(C)C2C)C(C)(C)C1 86217,C1(C(=O)NC2(C)CN(C(C3(CC=C)CCOC3)=O)C2)CC2CCC(C1)C2 86218,N1(C(c2cnc(C)o2)=O)CC=CCC1C(=O)N(C)C1CC1 86219,c1(CC(=O)N(C)CC2CCCN2C(=O)CN2CCOC2=O)c(F)cccc1Cl 86220,c1(OC)ccc(C(=O)NCCC2CCN(C(C3(C(C)C)CC3)=O)CC2)nc1 86221,C(=O)(C1=CCCOCC1)N1CCC(CC#C)(C(=O)NCc2ncc(CO)o2)C1 86222,C1(CC(=O)NCC2N(CC)CCC2)N(C(c2cccnn2)=O)CCC1(C)C 86223,C(=O)(C1=NNC(=O)CC1)NCC(C1CCCCC1)NC(C1C(CN(C)C)C1)=O 86224,N1(C(c2cc(CN(C)C)on2)=O)CCC2CN(C(=O)Cn3ccnn3)CC2C1 86225,N1(C(c2c(CC)n(CC)nn2)=O)CC(O)(C2(CNC(C3CC(C)CO3)=O)CC2)C1 86226,c1(CC(N2C(CN(C(COCCOC)=O)CC)COCC2)=O)cc(C)ccc1O 86227,CC(C)C(CNC(=O)COc1ccsc1Cl)NC(c1cnn(C)c1)=O 86228,C1(C(=O)NCC2(NC(CCN(CCC)C)=O)CCC2)CCc2nn(C)cc2C1 86229,c1(C(=O)NCC(CC)NC(=O)C(C#N)CC)cn(C)nc1-c1cccs1 86230,C1(C)(C(N2CCC(N(C)C)CC2)=O)CCCN(Cc2sccc2Br)C1 86231,C1(NC(CN(c2ccccc2)CC)=O)CCC2CNCCC2C1 86232,Cc1cccc(C)c1C(C(=O)O)NCc1cc(Br)sn1 86233,N1(C(CN(C)CC)=O)CCC2CCCC(C1)N2C(c1cc2c(nn1)CCCO2)=O 86234,c1(C(=O)NC(CC=C)CNC(c2cc3scnc3[nH]2)=O)cc(F)c(F)cc1F 86235,N1(C(C(COC)OC)=O)CC(CCNC(=O)CC=C(C)C)C(C)C1 86236,C1(CN(C(CN(CCC)C(c2ccc(C#N)o2)=O)=O)C)C(C)(C)C1(C)C 86237,N1(C(=O)CC2CCCC23CC3)CC=C(C(=O)N(CC(F)F)C2CCC2)CC1 86238,c1(C(=O)OC)cc2n(n1)CCCC2NC(c1ncoc1-c1cnn(C)c1)=O 86239,c1(CC(=O)NCC(C)N(C(C2CCSCC2)=O)CC)ccc(F)cc1[N+](=O)[O-] 86240,C12(CNC(C(CCC)C#N)=O)CN(C(c3c[nH]nc3C3CC3)=O)CC1CCO2 86241,Cc1nc2cncc(C(N3CC4(CCN(C(c5c[nH]cc5Br)=O)C4)C3)=O)c2[nH]1 86242,CC(C)CCCCN(C(c1ccnn1C)C(=O)N)C.C(C)(C)(C)ON.C1COC1=O 86243,C1(NC(CC2(OC)CCC2)=O)COCCC1NC(C1CCC(C(C)C)CC1)=O 86244,c1(C(=O)NC(CC(C)NC(C2C(C)C2)=O)C)n[nH]c2c1CC(C)CC2 86245,C(CNC(=O)CCC1CC1C)(C(C)(C)C)NC(c1cc(CCCCC)[nH]n1)=O 86246,c1(-c2n(C)nc(CO)n2)cc2c(s1)C(C)(C)CCC2 86247,C=CC(C)CC(=O)NCCC1CC(NC(=O)CCc2ccccc2O)C1 86248,c12cc(ccc1F)C(=O)N2.C(CCCCNC(=N)N)OC 86249,Cc1cc(C(=O)NC2CCN(C(=O)C(=O)Nc3ncc[nH]3)CC2C)ncc1C#N 86250,N1(CCOC)CC(NC(C2CC(CCNC(=O)C(C)N3CC(C)C3)C2)=O)CC1=O 86251,N1(C(c2nnc(-c3ncccc3Cl)s2)=O)CCC2(CCNC2=O)C1 86252,c1(C(=O)NC(CC)CNC(=O)CC(C)(C)C#N)cc2c(C)cc(OC)cc2o1 86253,c1(C(=O)NC(CC)(C)CNC(=O)C#CC(=O)N(C)C)n[nH]c2ccc(O)cc12 86254,N1(C(C(CN(C)C)(C)C)=O)CCOCC(CNC(=O)CCCCCO)C1 86255,C1(O)(CC(=O)NCCCCNC(CSc2nc(C)[nH]n2)=O)CCCOC1 86256,Cc1ccc2cc(C(=O)N(C)CCN(C(=O)C=CC(F)F)C)nn2c1 86257,CC1CC(C(N2CCOC(C(N)=O)C2)=O)N(C(=O)CCC2(C#N)CCC2)C1 86258,C=CC1(CC(=O)Nc2c[nH]ccc2=O)CN(C(=O)COCCC)C1 86259,c1(N2CCCCC(NC(CC(=C)C)=O)C2)nccc(S(C)(=O)=O)n1 86260,c1(C(=O)OC)cccc2c(C(=O)NCC3CCCCC3C)cccc12 86261,N1(C(C(CSC)OC)=O)CCCC(NC(C2C(c3ccccc3)C2C)=O)C1 86262,C1(CNC(CC=C)=O)CCN(C(=O)CCc2nc3ccccc3o2)C12CCC2 86263,C(=O)(CC(C)(C)C=C)N(C(CC(=O)NC(C#C)CC1CCCC1)CC)C 86264,N1(C(C(C(=O)OCC)(C)C)=O)CCc2sc(CNC(=O)CS(N)(=O)=O)nc2C1 86265,N1(CC)CC2(CCCN(Cc3ccc(Cl)c(O)c3)C2)C1.c12ccc(cc1)CN2C 86266,C1(CCC(=O)N(CC)Cc2cnn(C)c2)CCCCN1C(C1C=CCCC1)=O 86267,c1(C(=O)OCC)nn(C)[nH]c1=NC(=O)c1noc(C)c1I 86268,N1(CC)C(=O)CCC1CC(N1CC(CNC(c2c(C)nsc2N)=O)C1)=O 86269,CC1(C)NC(=O)CCC1NC(C1CSCN1C(=O)CCOCCN(C)C)=O 86270,C1(NC(=O)C=CC2CCC2)CCC12CN(C(C1CCN(C3CC3)C1=O)=O)C2 86271,C=CC(O)C(=O)NC(C)(CNC(c1cc(OC)ns1)=O)CO 86272,O=C(CCC(CF)CF)NCC(C1CC1)NC(=O)CCc1ccc(F)cc1 86273,N1(C(C=C(C)c2ccco2)=O)C(CC(=O)NC2CCCC2O)C2CCCC12 86274,c1(C(N2C(C)C(NC(=O)Cn3cccnc3=O)CC2)=O)cccc(S(N)(=O)=O)c1 86275,C1(C(N(CCN(C(c2cc(C(C)(C)C)on2)=O)CC)CC)=O)CCc2nnnn2C1 86276,CC1CN(C(=O)CCn2ccnc2)CC1CNC(=O)CN1CC(=O)NC1=O 86277,c1(C(N2C(C)C(C)N(C(C3CC(=O)CCO3)=O)CC2)=O)cn2cc(Cl)cnc2n1 86278,c1(C(=O)NCC2CC(OC)CN2C(=O)CNC(C2CC2C)=O)cc(C)n(C)c1C 86279,c1(CC)nc2c(C(=O)OCC#Cc3cccc(Cl)c3)cccn2n1 86280,C(=O)(CCCC(=O)OC)NC(CNC(CC1(OCC)CC1)=O)(C)CO 86281,C1(C(=O)NC(C2(O)CN(C(C3(OCC)CCCC3)=O)C2)C)CCOC(C)(C)C1 86282,CCC(F)(F)CC(=O)NC1CCCC(NC(c2ncccc2NC(C)=O)=O)CC1 86283,c1(C(N2C3CCC(NC(C=CC=CCC)=O)C(C3)C2)=O)cnn2ccc(O)nc12 86284,c1(NC(C2CC3CC3N2C(=O)CC2CCCCO2)=O)ncc(Br)nc1Br 86285,Cc1cc(=NCCOc2nc(O)n[nH]2)[nH]c(NC2CCC3(C(C)C)CC23)n1 86286,c1(CC)cc(N2CCC(CCNC(=O)C(F)(F)c3ccnn3C)C2)ncn1 86287,c1(NCC2C(NC(c3cn(CCCC)nc3C)=O)CCC2)ccc(C#N)nc1 86288,C1(CC(=O)NC(C2CCCN2C(c2c[nH]nc2C(F)F)=O)(C)C)CCC2CC2C1 86289,C1(NC(c2cc[nH]n2)=O)CCCC(NC(C23CSC(C2)C3)=O)C1 86290,N1(C(c2c(C(C)(C)C)nc(N3CCOCC3)nc2)=O)CCc2ccccc21 86291,c1(NC(=O)NC2CC(c3ccc(Cl)cc3)C2)ccc2nc(O)sc2c1 86292,CC1NC(=O)CCC1NC(c1cc(CNC(c2ccn(C(F)F)n2)=O)no1)=O 86293,c1(NCCCCC(C)NC(=O)Nc2ccccc2)snc(-c2ccccc2)c1C#N 86294,N1(C(C(C)c2cc[nH]n2)=O)CCCCC(C(=O)NCCc2cc[nH]n2)C1 86295,C#Cc1ccc(C(=O)NCC(C)(C)CNC(c2c[nH]cc2C2CC2)=O)nc1 86296,N1(C(C(C)NC(C)=O)=O)CCCC(CCNC(c2conc2C(C)(C)C)=O)CC1 86297,Cn1cc2ncc(C(=O)NCC3(O)CN(C(=O)C(C)(F)C(C)(C)F)C3)cc2n1 86298,C1(c2n(C)cnc2)CN(C(C2(C)CNC(=O)C2)=O)CC1NC(=O)C=CC(F)(F)F 86299,c1(C(N2CCC(OC)C2)C(=O)NCCSC2CCOCC2)ncc(C)cc1C 86300,Cc1noc(C(=O)NC(Cc2ccccc2)C(=O)O)n1 86301,CC(F)(F)C(C)(C)CNC(=O)NCc1c(C2CC2)cccc1F 86302,C(C(C)(CC)C(=O)N(C1CC1)CC1CCN(C)CC1)NC(c1ccc(C(C)=O)o1)=O 86303,C12(NC(C3CC(F)C3)=O)CC3CCC(C1C2)N3C(=O)Cn1ncc2ncccc12 86304,C(CC(O)C(=O)NCC(=O)NCc1cn(CCc2cccnc2)nn1)SC 86305,C(=O)(C1CCCc2scnc21)NCC(C)(C)Nc1nc(Cl)nc2c1CCC2 86306,N1(c2nnc(CCC)s2)CCN(C(c2ccc(CCC)[nH]2)=O)CC(C)(F)C1 86307,CCCC(C(O)C(=O)N1CC(N2C(=O)CCC2=O)C1)NC(C12CCCC1CCC2)=O 86308,N1(C(c2cc(CC)[nH]n2)=O)CCOC(CN(C)C(C2CCCN(C(N)=O)C2)=O)C1 86309,C1(C(C)NC(=O)CC2CCC2)CN(C(=O)Cn2cccnc2=O)CCO1 86310,Cc1cc(CNC(C2CC(C)CN(C(c3c[nH][nH]c3=N)=O)C2)=O)cc(F)c1 86311,N1(CC)C(C)CN(Cc2c(OC)nsc2OC(C)C)CC1(C)C 86312,CCCC(C)(CC)C(=O)N1CC(C(=O)NC(CCO)CC(C)C)C(C2CC2)C1 86313,N1(C(c2nnc(C(F)(F)F)s2)=O)CCn2c(cc3ccc(Cl)cc23)C1 86314,c1(C(N2C(CNC(=O)CCC(C)C)CC(OC)C2)=O)nccc2c(F)cccc12 86315,C1(C2CCCCC2)(C(=O)NCC(CNC(c2ncn(C)n2)=O)OC)CCCCC1 86316,c1(CN2CCC(C)C(C)(C)C2)ccc2cc(F)cc(Br)c2n1 86317,c1(-c2c(OC)cccc2CN=c2[nH]nc(C)n2C)ccc2[nH]nc(CO)c2c1 86318,N1(C(c2ccc(F)c(Br)c2F)=O)CCOC2CCNCC12 86319,Cc1nn(C)c2sc(C(=O)NC3CC(F)CN(C(=O)CC(C)F)C3)cc12 86320,Cc1c(C(=O)NC(CNC(c2ccsn2)=O)CO)cnc2ncnn12 86321,C1(NC(C=CC(=O)N(C)C)=O)C=CC(C(=O)NCC(F)Br)C1 86322,c1(SC)cnn(C)c1C(=O)N(CCCNC(=O)C(c1ccc(C)s1)C)C 86323,c1(C(N2CC3CC2CN3Cc2cscc2Br)=O)cc2n(n1)CCC2 86324,C12(CNC(C3(SCC)CC3)=O)CCC1CN(C(=O)Cc1ncsc1Cl)C2 86325,CC(C)(CO)C(=O)NCc1ncoc1C1CN(C(=O)COC(F)(F)F)C1 86326,C=C(Cl)CC(C(=O)NC1CCC(=O)NC1)NC(=O)C(F)CCC 86327,Cc1c(C(=O)NC(C)C(CO)NC(=O)CSc2cn[nH]c2)cnn1C(C)(C)C 86328,C1(NC(c2c(C)n(C3CCC3)nc2)=O)CC2(CCN(c3ccnc(C#N)n3)C2)C1 86329,Cc1nc(NCCc2nnc3n2CCS3)cc(=NC(C)c2cc[nH]n2)[nH]1 86330,Cc1cccc(C(O)C(N2CC(C)(NC(c3cncc(N(C)C)c3)=O)C2)=O)c1 86331,N1(C(C(C(C)(C)C)O)=O)CCN(C(=O)CC2=NNC(=O)C2)C2COCC12 86332,c1(C(=O)NCC(Cn2cc(C(C)(C)O)nn2)(F)F)c2c(co1)CCC2 86333,N1(C(C2N(CC)CCC2)=O)C2CCC1CC(C(=O)NCC(F)C1CCC1)C2 86334,c1(C(=O)NC(C2CN(C(c3cn(CCC4CC4)nn3)=O)C2)C)c[nH]nc1[N+](=O)[O-] 86335,C12(C(=O)NCCCC#C)CC1CN(C(=O)C(N1CCN(CCO)CC1)CC)C2 86336,Cc1nncn1NC(=O)C1CC(NC(c2csc(CO)n2)=O)CCO1 86337,CC1CCN(C(=O)Cc2cccs2)CCC1N1CCCC1c1c(F)cccc1Cl 86338,c1(C(=O)OCC)cc(C(=O)OCc2cc(C)c(C)o2)c(C)cc1OC 86339,C1(C(N(CC(C)NC(c2ccncn2)=O)C)=O)C(C)CCN1C(=O)OC(C)(C)C 86340,C(=O)(CCN=[N+]=[N-])N(C1(C(=O)NC(CC=C)C)CC1)C 86341,N1(C(c2cc(CC)n(C)n2)C(=O)NCCC#N)C2C=CCC1CCC2 86342,c1(C(N(C2CN(C(C3CC34CC(O)C4)=O)C2)C)=O)ccnc(F)c1 86343,c1(C(N2CC(O)(CCNC(C3(CC#C)CCOC3)=O)C2)=O)cc(C#C)ccn1 86344,c1(NC(c2nnc(O)o2)C)[nH]c(=NCc2ccc(=N)[nH]c2)nc2scnc12 86345,CCCC(C(O)C(=O)NC1CCN(C(C)(C)C)C1)NC(=O)CC(C)(C)COC.OCC 86346,CN1CCC(C(=O)NC2CCN(C(c3cccc(NS(C)(=O)=O)c3)=O)C2)C1=O 86347,c1(C(N(C)CCOCCNC(=O)Cn2cnnc2O)=O)cn2ccsc2n1 86348,O=C1CS(=O)(=O)CC(C(=O)NC2CC(CCNC(C3CC(F)(F)C3)=O)C2)N1 86349,c1(CC2(C(N(CC(C)NC(c3cnn(C)c3)=O)C)=O)CCCC2)ccc(Cl)nc1 86350,N1(C(C(CCC)OCC)=O)CC2(C(=O)NCC(CO)C3CCC3)CC1CO2 86351,Cc1cnc(C)c(NC(C2C=CCN2C(=O)Cc2ccccc2Cl)=O)n1 86352,C1(CC)OCCCC1C(=O)NCCC1CC(NC(C2NC(=O)OC2C)=O)C1 86353,N1(C(C(C)C)=O)CC(CNC(C2NC(=O)CC2C(F)(F)F)=O)C(C)C1 86354,C(=O)(C1=CCCN(Cc2cccc(F)c2I)C1)Nc1ccc(OC)nc1OC 86355,c1(N(C(c2c(CNC(CC3(C#N)CC3)=O)noc2)=O)CCO)cccc(F)c1 86356,C1(NC(c2c(C)con2)=O)C(C)CCN(C(c2cnc3sccc3c2)=O)C1C 86357,c1(C(C(=O)NCCCC)N(C2CCN(CC(F)F)C2)C)cc(F)cc(C#N)c1 86358,C(C(C(=O)N1CCCC1CNC(c1cc(C)ns1)=O)C(C)(C)C)OCC=C 86359,C(=O)(C1=C(Cl)CCCC1)NCC(C(C(=O)NCC(=C)Cl)F)C 86360,N1(C(C)C)CCCCC1C(=O)NC1(C)CN(C(C2(S(C)(=O)=O)CC2)=O)C1 86361,CC(CN(C)C)CCC(=O)NCc1ccc(C(=O)NCC2C3CCCC23)s1 86362,N1(C(CCC)=O)CCCC(C(N2CC(O)(CNC(=O)CCC(N)=O)C2)=O)C1 86363,C(=O)(C1CCCc2scnc21)NCC(CC)NC(C1CCc2nncn2C1)=O 86364,c1(CNC(C)C(=O)Nc2ncccn2)ccc(C#N)c(F)c1 86365,C1(NC(CSCCCC)=O)CCCN(C(=O)CCc2ccoc2)C1C 86366,N1(C(C(C(C)(C)C)=O)=O)CCC(C(N2CC3C=CCC(C3)C2)=O)C(C)(C)C1 86367,Cc1noc(C)c1-c1cn(C2CCC(C(=O)N(C)CCN(C)C)C2)nn1 86368,N1(CCNC(C2(CCNC(C3(CC)CCC3)=O)CC2)=O)CCNC(=O)C1 86369,c1(CC(=O)OC)cccc(C(=O)NC2CC2NC(=O)C(O)Cc2cnc[nH]2)c1 86370,CC1(COC(C2CC2c2ccc(Cl)c(Br)c2)=O)NC(=O)NC1=O 86371,Cc1c(C(=O)NCCCCCN(C)C(c2cncc(C(C)C)c2)=O)ncn1C 86372,c1(C(=O)NCCNC(C2CCCOC2)=O)ccc2c(Br)cccc2c1 86373,C1(NC(C(C)OCCN(C)C)=O)CCCC1CNC(C1(F)CC1)=O 86374,c1(CN(C)NC(=O)CC23COC(C)(C2)C3)nc(-c2ccccc2)sc1N.C1(C)(N)CC1 86375,CCC(CNC(C1CN(C(N)=O)C1)=O)(CC)NC(C1CCNC1=O)=O 86376,C1(CNC(C2(COCC)CC2)=O)CC(C)(C)CN1C(c1ccc(SC)cc1)=O 86377,c1(C(=O)NC2C(C)CCN(C(=O)CC3(CO)CC3)C2)cc2ncccc2[nH]1 86378,c1(N2CC(CC)N(c3cc(OC)nc(C)n3)CC2)nc(NC)cn2ccnc12 86379,c1(C(=O)NCC2(C)CCCN2c2cc(Cl)ncn2)cnc2cnccc2c1 86380,c1(C(=O)NC(C)CNC(c2ccncc2N)=O)cc2nccc(C(F)(F)F)n2n1 86381,C1(NC(C(C)OCC#C)=O)CCS(=O)(=O)C12CN(C(=O)CN(S(C)(=O)=O)C)C2 86382,N1(CC(=O)NC2CC(CNC(C(C(C)C)F)=O)C2)CCc2ccccc2C1=O 86383,C(=O)(CCS(=O)(=O)CC(C)C)N1CC(NC(C2=C(C)S(=O)(=O)CC2)=O)C(C)C1 86384,Cc1cc(C(N2CCOCC(NC(c3ncc(Cl)s3)=O)C2)=O)c(N)c(Cl)c1 86385,C(=O)(C(F)(F)CCNC(C1CCS(=O)(=O)N1C)=O)OCC 86386,C1(CNC(CCSc2n(C)ccn2)=O)CCN(C(C2(C)CC3CC3C2)=O)CC1 86387,C(=O)(C1=CC(O)CCC1)NCC1CC(OC)CN1C(c1ccc(F)cc1)=O 86388,n1(CC)nc(C)c(C(=O)NCC2CN(C(c3cc(F)n[nH]3)=O)CCC2C)c1Cl 86389,c1(C(N(C(c2ccc(Br)cn2)C)C)=O)cc2c(C(F)(F)F)cc(N)cc2s1 86390,c1(C(C(=O)NCC(=C)C)N(CCC(=O)OC(C)(C)C)C)cn2c(Br)cnc2s1 86391,N1(CC)CCC(C23CC(C2)C3)C1.c1(-n2c3nc(n2)C(C)S3)ccc(C)c(F)c1 86392,CC1Cc2cccc(C(=O)NC3CC(N)C3)c2O1.c1(C(=O)N)ccc2ncccc2c1 86393,C1(CC(=O)NCC2C(C(=O)NCC(CC)C#N)CC2)CCC(C)(C)C1 86394,c1(C(N2CCC(NC(C(CCC)C)=O)C2)=O)cc(OC(F)F)ccc1C 86395,N1(C(c2cc(NC(C)=O)ncc2)=O)CCN(C(C2(C)CCCCC2)=O)CC1C#N 86396,c1(CC(=O)NC2CC(CCNC(C3(C)CCCS3)=O)C2)ccc(C#N)c(F)c1 86397,C1(CC(=O)NCC(C(C)C)(C)NC(=O)CN2CC(C)(C)C2)CCCC(C)(C)O1 86398,C1(C(N2CC(O)(C(C)NC(c3c(OC)c[nH]n3)=O)C2)=O)C2CCCCC12 86399,c1(C(=O)NCCC2CCN(C(C(C)=CC3CC3)=O)CC2)c(F)ccnc1Cl 86400,CC1(C)CC(CNC(c2cnc(C(N)=O)s2)=O)CN1C(c1cccc(F)c1)=O 86401,C(=O)(C(O)CC(C)(C)C)N1CC2C(CNC(C(C)N=[N+]=[N-])=O)(CC2)C1 86402,c1(C(=O)NC(C)C(C)NC(=O)CCCCNC(N)=O)ccc2cccc(F)c2n1 86403,c1(CC)ccc(C(=O)NCC2(NC(=O)Cc3c(C)nn(C)c3C)CCC2)cc1N 86404,N1(C(CSCCC(C)C)=O)CCC2CC1CN2C(=O)C(c1cncc(F)c1)C 86405,N1(C(C2(NC(=O)Cc3ccccc3O)C(C)(C)C2)=O)CC2(C)COCC2(C)C1 86406,C1(OC)CC(NC(c2cnn(-c3nccs3)c2)=O)CN(C(C2CCCSC2)=O)C1 86407,c1(C(=O)NCCN(C(=O)C(C)(C)Br)CCC)ccsc1OC 86408,C1(C(C)C)CN(C(c2cc(N(C)C)ccc2F)=O)CCC1NC(C1CC=CC1)=O 86409,C(=O)(C(C)(O)C(C)(C)C)NCC(CNC(C1CC2(CC(=C)C2)C1)=O)O 86410,Cc1cc(C(=O)N(CCCNC(C2(C)CC(=O)N(C)C2)=O)C)cc(C(F)F)c1 86411,CC1(C)CCN(C(C2C3CCCOC23)=O)CC1NC(c1ccc(C2CC2)nc1)=O 86412,c1(C(N2CCC(C(CNC(CC(C)OC)=O)F)CC2)=O)cc(N)c(F)cn1 86413,Cc1cc(C(N2CCOC3(CCN(C(=O)C4=CC4)C3)C2)=O)c2cc(F)ccc2n1 86414,N1(C(CCCCCC#C)=O)CCc2[nH]nc(CNC(=O)C(C(C)C)N(C)C)c2C1 86415,N1(C(CCc2cnc(C)o2)=O)CC2CC1C2NC(=O)CCSc1nccn1C 86416,c1(C(=O)NCC2C(NC(CCCn3c(C)ncc3)=O)C2)ccc(C(O)CF)cc1 86417,N1(C(CCCNC(CC2(NC(C)=O)CC2)=O)=O)CC(C)C(C)C1C 86418,N1(C(c2ccc3occc3c2)C(=O)NCCC2CC2)CCC2(CCCCO2)CC1 86419,C1(NC(C(C(C)C)O)=O)CC2CCC(C1C)N2C(=O)Cc1c[nH]c2cccnc12 86420,C1(NC(C(N)=O)=O)CCCC2CN(C(=O)CC3CCCCCC3(F)F)CC12 86421,c1(C(C)C(=O)NCCN(C(C2CC(C)(C)O2)=O)C2CC2)ccc(F)cc1F 86422,C1(C(=O)NCC2CC(C(=O)NC3CCS(=O)(=O)C3)CO2)(CC)CNC(=O)C1 86423,N1(CCC(=O)OC)CCC(C(C)NC(C2(C(F)(F)F)CCC2)=O)CC1 86424,C1(NC(=O)Cn2ncnn2)(CF)CCN(C(c2cccc(Br)c2)=O)C1 86425,Cc1cc(C)n(CCNC(C2OCCC2NC(=O)CCc2ccncn2)=O)n1 86426,C1(CC(=O)NC2C(CNC(COC(CC)(C)C)=O)C2)CCOC1C 86427,Cn1cnc2cc(C(N3CCC(C)(C)C(c4cn(CC(N)=O)nn4)C3)=O)cnc12 86428,N1(C(CC(CC)OC)=O)CCC(CNC(c2ccc(Cl)c(Cl)c2)=O)C(C)C1 86429,N1(C(c2c(C)nc(S)s2)=O)CCCN(CC(C2CN(S(C)(=O)=O)C2)=O)CC1 86430,c1(C(N2CCC(N(C(C(C)C(C)(C)C)=O)CC3CC3)C2)=O)cccc2occc12 86431,C1(CC(C)C)CCN(C(C2(CNC(=O)CCn3cnnn3)CCCC2)=O)C1 86432,CN1CCC(NC(=O)CCN(C(=O)Cn2c(O)nnc2O)CCO)C(C)(C)C1 86433,c1(C(=O)NCCC(=C)CNC(=O)CCc2nc[nH]n2)ccc(Cl)cc1 86434,c1(C(=O)OCCCC#C)nn(CC)c2c1COCC2 86435,N1(C(c2c(CCC)nco2)=O)CC2CCC(C1)C2NC(=O)COC(C)C 86436,C1(C(=O)Nc2cn(C(C)C)nc2)CCCC12CCN(Cc1cnc(Cl)cc1F)C2 86437,N(C1CCN(C(=O)Nc2cc(C)c(C(F)F)cn2)c2ccc(Br)cc21)C(C)(C)C 86438,C1(CC(N2CCC(CN(C(=O)CSCc3ccccc3)C)C2)=O)NC(=O)NC1=O 86439,C(=O)(C(C(=O)N1CCC(F)(CNC(=O)C#CC(C)C)C1)OC)OC 86440,CCC1=NOC(C(=O)NCC(O)CNC(=O)C(C)(C)NS(C)(=O)=O)C1 86441,CC(C)(C(=O)N1CCC(NC(C2CCOC2C(F)(F)F)=O)C1)c1cccs1 86442,Cc1cc(=NCC(O)c2cnc(C(F)(F)F)nc2)nc(N2CCCCC2)[nH]1 86443,C1(C(N(C)Cc2cccc(C)n2)=O)CCCCCCN1C(C1CC1C(N)=O)=O 86444,N(C(=NCc1cc(C2CC2)on1)NC1CC(=O)N(c2ccccc2)C1)C(C=C)C 86445,Cn1cc(C(F)=CC(=O)NCC2(CNC(c3cc(N)ccc3F)=O)CC2)cn1 86446,c1(CC)cccc(C(=O)N(CCCCCCNC(C23CC(O)C2C3)=O)C)c1 86447,c1(C(=O)NC2(C)CCCN(C(C3ON=C(CC)C3)=O)C2)cc2cccc(C)n2n1 86448,c1(C(N2CC(C(=O)OC)OCC23CC3)=O)[nH]nc2c1COC2(C)C 86449,C1(NC(C2CCC(CC)CC2)=O)CC(O)CN(C(=O)CSCc2ccccc2)C1 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86468,CCCC(CCC)=CC(N1CC(C(=O)N(C)Cc2cn(C)nn2)C(F)C1)=O 86469,c1(C(N2CC3C(CCNC(CCOCC#C)=O)(CC3)C2)=O)nc[nH]c2ncnc1-2 86470,C1(NC(C2CCS(=O)CC2)=O)C2CCC1N(C(=O)CC1=CCCC1)C2 86471,C#CC1(C)CCCN(C(=O)C(O)CCCNC(=O)C(C)(O)C=C)C1 86472,c1(C(=O)NCC(C)(C(C)C)NC(c2ccn(CCC)n2)=O)ccnc(F)c1N 86473,c1(C(=O)OC)ccc(C(CNC(=O)C2CC2)=O)[nH]1.C1(=O)CO1 86474,c1(CC(=O)NC23CC(C(=O)NC4CCC5(CCC5)C4)(C2)C3)c[nH]c2ncccc12 86475,n1(CC(=O)NC(CCNC(C=CC)=O)(CC)CC)cc([N+](=O)[O-])c2ccccc12 86476,C#CC(C(C)(C)OC)NC(=NCc1ccccc1)NC1CC1(CC(F)(F)F)CC 86477,C1(C)(CNC(=O)NC(C2CC3CCC2C3)C)CCN(C)CC1 86478,C1(NC(C(C)=C(CC)C)=O)CN(C(=O)COCC2CCC2)CCC1CO 86479,Cc1nc(=N)[nH]c(C)c1C(N1CCC(NC(c2cc(Cl)on2)=O)C(C)C1)=O 86480,c1(C(N2CCC(C(C)NC(c3c(C)c(O)ccc3)=O)C2)=O)cnc2[nH]cncc1-2 86481,N1(C(CSC)=O)CCCC(N2CCN(C(=O)CC3CCCC34CC4)CC2)C1 86482,C(=O)(CCCC(N)=O)N(CC(C)N(C(=O)Cc1ccn(C)n1)C)C 86483,N1(CC(=O)N(C(C)C)CCNC(=O)Cc2cncnc2)CCC(C(F)(F)F)CC1 86484,C(=O)(C1COc2ccc(Cl)cc21)NC(CC=C)CNC(c1ccsc1OC)=O 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86520,C1(C(=O)NCC2CCCN(CC(F)F)C2)CC2(CCCCCCC2)N1 86521,C1(C)(CCC(=O)NC2CC(C)C2)CCCN1C(C1CCC1C(C)(C)C)=O 86522,C1(C(=O)NC2CC(NC(c3ccc(NCCO)cc3)=O)C2)CCC(F)(F)CC1 86523,c1(-c2cnc(NC(c3nn(C(CC)CC)c(C)c3)=O)s2)cccc(C#N)c1 86524,C1(CNC(C=CC)=O)CC(F)(F)CN1C(=O)C(O)Cc1[nH]cnc1C 86525,c1(C(=O)NC2CC(OCC(N3CCC(SC)C3)=O)C2)cc[nH]c(=N)n1 86526,Cc1nn(CC(=O)NCC(O)CCNC(C2CN(C3CCCCC3)C2)=O)c(=O)n1C 86527,C1(CC(=O)NC2C(F)CCN(C(COC(C)C)=O)C2)CS(=O)(=O)CCN1C 86528,c1(C(=O)OCC)c(C)ccnc1CNCc1cc(C(F)F)n[nH]1 86529,N1(C(C(C)c2cccs2)=O)CC(C2CCCN(C(C3(C4CCC4)CCC3)=O)C2)C1 86530,c1(CN(C(c2c(C)cc[nH]c2=N)=O)C)c(Cl)cc(Cl)cc1Cl 86531,CON(C(=O)c1c[nH]nc1CNC(=O)C(C1CCCCC1)C)C1CCCC1 86532,C(=O)(CS(=O)(=O)C1CC1)NC1C(CC)CN(C(C2(F)CCN(C)CC2)=O)CC1 86533,CC(C)(CNC(C1C(CNC(C2C=CCS2)=O)C1(C)C)=O)CN=[N+]=[N-] 86534,C(=O)(CCC(C)(C)[N+](=O)[O-])NC(CC)(CNC(c1cnco1)=O)CC 86535,C(=O)(CC(=O)NC1CC1)NC(C1CCCN1C(c1csc(-c2ncc[nH]2)n1)=O)C 86536,CC(C)C(O)C(F)(F)C(=O)N1CC2CCN(C(=O)CCCC(C)(C)C)CC2C1 86537,C1(C(=O)NC2(CC=C)CN(C(C(CC#C)C3CC3)=O)C2)CC2(C1)CC2(F)F 86538,C1(C(=O)NCCCN(C(=O)Cc2cccs2)C)CCCC(N(C)C)C1 86539,CCC(CC(=O)NCC1(NC(=O)CC2(CO)CC2)CCCCC1)SC 86540,c1(CNC(C2(OC)CCC2)=O)cc(C(N2CCCC2CCC2(C)N=N2)=O)on1 86541,C(=O)(C(CC)CC(F)(F)F)NCC1CN(C(CCCC)=O)CC(C)(C)C1 86542,c1(C(=O)NCCC2N(C(C(C=C)OC)=O)CCOC2)cc(C)c2occc2c1 86543,CCC(C(=O)NC(C)Cn1cc(C2CCCO2)nn1)N(C)C 86544,c1(C(=O)NCC2CCS2(=O)=O)ccc2c(c1)NC(=O)CCN2 86545,Cc1ccnc(C(C)(C)C(=O)NC2CCC2NC(C2COCC2(C)C)=O)c1 86546,c1(CNC(=O)C(F)(F)F)cc(F)c(Nc2cc(-c3ccncc3)ccn2)c(F)c1 86547,C1(NC(CCC(=O)NCC)=O)CN(C(c2ccc(N)c(F)c2)=O)CCC1(C)C 86548,c1(SC)cncc(NC(C2(C)C=CCN2C(C2CC2C(N)=O)=O)=O)c1 86549,C1(NC(c2cnc(C)o2)=O)CCS(=O)(=O)C12CN(C(=O)CCS(C)=O)C2 86550,C1(NC(C2C(OC)C2)=O)CCCCC1C(=O)NCc1ccccc1OC(F)(F)F 86551,c1(C(N2CC(NC(CC(C)(C)O)=O)C3(C2)CC3)=O)cc2ccc(F)cc2[nH]1 86552,C=CCC(C)(C)CC(=O)N1CCC(C)CC1CNC(=O)CC1(N(C)C)CCC1 86553,c1(C(N2CCCC2CNC(C2CC(F)(CF)C2)=O)=O)ccc2c[nH]nc2n1 86554,c1(C(N2C(CNC(CS(CC)(=O)=O)=O)CC2)=O)cc(Cl)c(C)cc1[N+](=O)[O-] 86555,c1(C(N(C(CC)CNC(=O)C(c2ccnn2C)C)C)=O)cc(O)ncc1F 86556,CC(C)CC(C)C(=O)N1CC=CC1C(=O)NCC(O)(CO)CO 86557,Cc1cnc(C(=O)NC(C)(C)CN(C)C(c2ccc(C(C)(F)F)nc2)=O)cc1C 86558,N1(C(C2C(NC(c3c(C)cco3)=O)C2(C)C)=O)CCCC(C)(F)C1 86559,c1(CCN)cccnc1C(c1nnnn1CC(C)C(C)(C)C)OC 86560,C1(CNC(C(C(CC)(C)C)O)=O)CN(C(=O)CC(O)C(C)C)CCC12CCOC2 86561,C1(c2nnnn2C2CC2)(NCc2ccncn2)CC2COCC2C1 86562,C1(CNC(c2[nH]cc(C)c2)=O)(NC(=O)CCSCC(N)=O)CCCCC1C 86563,C(=O)(C1CCCc2ncnn21)NCCCN(C)C(c1cc(Br)ccc1F)=O 86564,c1(OC)ncc(C(=O)NC2CC(F)(CNC(=O)CCCN(C)C(C)=O)C2)c(C)n1 86565,N(C(=NCC1CC1)NCC1(C)CCCC1)C(COC)C 86566,n1(CC)ncnc1C(=O)N(CC(C)NC(C1(COC(C)C)CC1)=O)CC 86567,c1(OCCC(N2CC(NC(C(C=CC)O)=O)C(F)C2)=O)ccc(C)cc1C 86568,c1(C(N2CC(CNC(Cc3cccc(SC)c3)=O)OCC2)=O)c(Cl)cc(Br)cc1Cl 86569,c1(C(=O)NC2C=CCN(c3nnc(C4CC4)s3)C2)ccc2c(c1)CCCC2 86570,N1(C(C(c2c(C)cccn2)(F)F)=O)CCOC(C)(CNC(c2ccc(Cl)o2)=O)C1 86571,c1(CC)ncsc1C(=O)NC1(CNC(=O)C(F)CC2CC2)CC1 86572,c1(NC(c2scc(CC)n2)C)nccc(=NC(C)c2ccccc2OC)[nH]1 86573,C1(NC(CC(C)(C)O)=O)CC2CC(C1)N(C(c1cnncc1C(F)(F)F)=O)C2 86574,CCCC(C(=O)N1CCCCC(NC(c2ccnn2C2CCC2)=O)C1)S(N)(=O)=O 86575,c1(C(=O)NCC(O)Cc2ccccc2Br)coc2c(Cl)cc(Br)cc12 86576,CC(CNC(=O)CN(C(c1cc(C#N)c[nH]1)=O)C1CC1)CC(C)O 86577,C1(NC(=O)Cc2cccnc2O)CN(C(c2ccoc2)=O)CC2CCCC12 86578,c1(NC(C(C)NC(=O)NC)=O)nc(OC(C2(O)CCN(C(=O)NC)C2)=O)ccc1F 86579,c1(CN2C(C(N3CCCC(C(N)=O)C3)=O)CC(=C)C2)c(O)ccc2ccccc12 86580,C1(CNC(C2(CC#C)CCOC2)=O)(NC(=O)C(O)P(C)(C)=O)CC2CCC1CC2 86581,C1(C(N(C(c2ccc(F)cc2)C)C)=O)COCCN(CC2COC(=O)N2)C1 86582,c1(N(C)C)ccccc1C(=O)NC1(CC(=O)NCc2ncsc2Br)CCC1 86583,c1(C(=O)NCCN(CCC)C(C2CC2(C)Br)=O)cn[nH]c1 86584,c1(CCC(=O)NCCN(C(C2(C)CCC(=O)C2)=O)CC)ccc2ccccc2c1 86585,C1(CNC(C=C(C)C(C)(C)C)=O)CC2CN(C(C3CC3C(=O)NCCO)=O)CC12 86586,c1(N2CCCC(CO)CC2)ncnc2ccc(O)cc12 86587,CN1CCc2[nH]nc(C(N3CCC4(CCCN4C(C4COC(=O)C4)=O)C3)=O)c2C1 86588,c1(C(N2CCC(NC(C(C(C)C)SC)=O)C23CC3)=O)ccc2c(C)noc2c1 86589,CCC(C)C(C(F)(F)F)NC(=O)Cc1ccccc1NC(=O)C(C)(C)C 86590,N(C1COc2ccc(Cl)cc21)C(C(Cc1ccccc1Br)NC(C(C)O)=O)=O 86591,c1(CC)cnc(NC(=O)Cn2cncn2)c(C)c1 86592,c1(-c2n(C(C)C3CC3)nc(C3CCOC3)n2)cnc(O)c(Br)c1 86593,S(=O)(=O)(c1cc(F)c(Br)c(F)c1)NC1C(OC)CN(C(c2cc(Cl)cs2)=O)CC1 86594,c1(OC)ccc(C)cc1C(=O)N(C1(CC(=O)N(CC(O)C2CC2)C)CC1)C 86595,C12(C(N(C3CCCCC3)CCCN)=O)CC3CC(C1)CC(Cl)(C3)C2 86596,c1(C(N2CC3CCC2CC3)C(=O)NC(CC)C)ccc2cccc(Br)c2n1 86597,N1(C(c2c(NC)cncc2)=O)CCC(C(=O)NCCCS(C)=O)C12CC2 86598,C1(=CCNC(=O)CC(F)F)CCN(C(C2(F)CCOC2)=O)CC1 86599,C(CCC(=O)N(C1CCCCC1)CCNC(=O)C=CC1(C)COC1)N(C(C)=O)C 86600,N1(n2cc(C=O)ncscc2)CC(F)(F)CC1CNC(C1(C(=O)O)CCCC1)=O 86601,C(=O)(CCC(=O)NCc1cn(CC(N2CCC(C)CC2)=O)nn1)NC.C1C(=O)N1 86602,c1(C(N2CCN(C(COC(CC)C)=O)CC2C)=O)nc(C)c(C)nc1C 86603,C=C(Cl)CCC(=O)N(CCCNC(=O)CSCC1CCCC1)CC.c1(N)cccnc1 86604,c1(C(CC)NC(=O)C(N2C(C)CC2(C)C)CC)ccc(OCCOC)c(OC)c1 86605,c1(C(N(CCCCCNC(=O)C#CC2CCCO2)C)=O)ccc2nnc(S)n2c1 86606,c1(C(=O)NC(CNC(c2cocn2)=O)C2CCC2)cc(Cl)nnc1O 86607,c1(C(C)NC(=O)NCC2CC2c2cn[nH]c2)cccc(O)n1 86608,c1(NC(N2Cc3n(cc(C)n3)CC2)=O)nc(C2=CCC(C)(C)CC2)cs1 86609,c1(NC(C2(CC)CC2)=O)cn(C)c(C(=O)NCc2cocn2)n1 86610,CC1=C(C(=O)NCCOC2CCN(C(c3oc(C)nc3C)=O)C2)CC1 86611,N1(C(c2ccc(CC)s2)=O)CC(C(=O)NC2CCOC(C)C2)CC1(C)C 86612,c1(N2CCCC(C(N)=O)C2)nc2ccc(Cl)cc2c(=NCCSC2CCCC2)[nH]1 86613,C1(CNC(C(CSC)(C)C)=O)CN(C(=O)CNC(C)=O)CC1O 86614,c1(OC)cc(C(N2CCN(c3ccc(C(F)(F)F)nc3)CC2)=O)ccc1N 86615,c1(C(N(C)CC2CN(C(C3CCOC3)=O)C2)=O)csnc1Cl 86616,n1(CC)nnc2cc(C(N3CCCCCC(NC(C4CC(F)C4)=O)C3)=O)ccc12 86617,CCCCC(O)CC(=O)NC1(CC(N2CCCN(CCC)CC2)=O)CC1 86618,CC(CCCc1cn(C(C)(C)C(=O)O)nn1)C(=O)NC1(Cc2ccncc2)CC1 86619,C(CC(C)C)(C(=O)N1CC(N2CC(N(CCO)CCO)CC2=O)C1)NC(=O)OC 86620,N1(C(C(CCC2CC2)NC(C(C)SC(C)C)=O)=O)CC2(CCNC(=O)O2)C1 86621,N1(C(CCCC#C)=O)CCCC(C2CCN(C(c3cscc3Cl)=O)C2)C1 86622,C1(C)(CC(=O)N(CCC(=O)NC(c2ccn(C)n2)C)C)OCCO1 86623,N1(C(c2c(CC)occ2)=O)CCC(C(=O)NCC(=O)N(C)C)C12CCC2 86624,N1(C(C23CC(C2)C3)=O)CCC12CCN(Cc1cccc(F)c1O)CC2 86625,N1(C(c2c(CCC)n(C)nc2)=O)CCCN(C(=O)CC=C(Cl)Cl)CC1C(C)C 86626,c1(N(C)C)ccc(Cn2nc(-c3cccc(F)c3)nc2-c2cccnn2)cc1 86627,C1(C(=O)NC2(C3N(C(C=C(CCC)C)=O)CCC3)CC2)C(C=C(C)C)C1(C)C 86628,S(=O)(=O)(c1cc(Cl)c(Br)cc1F)N(C1(Nc2c(C)cncn2)COC1)C(C)C 86629,c1(CN(CC(=O)N(C)Cc2ccccc2)C(C)(C)C)ncccc1Br 86630,c1(C(N2CCN(C(C(CC)C)=O)CC2CC(=O)NC)=O)ccnc2c1CC(=O)N2 86631,C(=O)(C(CC1CC1)NC(C1CCNC1=O)=O)NCC(c1cccs1)C 86632,c1(CC(C(=O)O)NCc2cnc3cccnc3c2)cccc2ccccc12 86633,N1(C(c2ccc(C)o2)=O)CCC(C(C)(C)C)(CNC(C2CCC3CC3C2)=O)C1 86634,c1(NC(=O)NC)cccc(C(N2CC3CC3(CNC(=O)CN(C)CCO)C2)=O)c1 86635,c1(CC(=O)NCc2ccc(CNC(=O)CC3(O)CCC3)cc2)cc(Cl)cc(Cl)c1 86636,c1(-c2cn(CCN3C(N4C(=O)OCC4)COCC3)nn2)ccc(F)c(Br)c1 86637,N1(C(Cc2c(C)cco2)=O)CC2CC(C1)C2NC(=O)CNS(=O)(=O)N(C)C 86638,CC1(NC(=O)C(C2CCCCC2)O)CCCCC1C(=O)NC1C=CCCC1CO 86639,C1(NC(C(C)C2CCCC2)=O)COCC1NC(c1cn(CC(=O)N(C)C)nn1)=O 86640,Cc1c(C(N2CC(C)N(C(C3CC3F)=O)CC2C)=O)cc(F)cc1[N+](=O)[O-] 86641,CCCCCCC(C)CC(=O)NC1CCC(NC(c2cc[n+]([O-])cc2)=O)C1 86642,N12CCN(CC1)C(=O)C(C)N1CC2C1.c1(OC)ccc(C(F)(F)C(=O)OC)cc1 86643,n1(CCC)ccc(=NC(=O)C2CCC(C(C)C)N2C(C2CC2C#N)=O)[nH]1 86644,C1(c2c(C)c[nH]n2)COCCN1N1CC(CCS(N)(=O)=O)C1.c1cccs1 86645,c1(OC)cc(O)ncc1C(=O)NC(CNC(c1nc(C)oc1C)=O)CC(C)C 86646,C(=O)(CC(O)C(C)CC)NCC(CC(=O)N(CC(C(=O)NC)C)C)O 86647,C(C(CNC(c1ccns1)=O)S(C)(=O)=O)NC(C1N(C(C(CC)C)=O)CSC1)=O 86648,C1(C(=O)NCCc2c(C)cc(C)cc2C)CCCN1NC(=O)Cc1ccsc1C 86649,C1(C(=O)OC)CCN(C(=O)Nc2c(F)c(F)cc(F)c2F)CCC1(F)F 86650,N1(C(C2C=CCCC2)=O)CCC2(CC1)CCN(C(C1CCC(F)(F)CO1)=O)C2 86651,c1(C(=O)NC(CNC(C2CN(C)C(=O)CC2)=O)C2CC2)csc(=NC2CC2)[nH]1 86652,CS(=O)(=O)c1ccc(F)cc1C(=O)NC1CC(F)CN(C(C2CCC(=O)N2)=O)C1 86653,C1(CN(C)C(c2cnn(C3CCC3)c2)=O)CN(C(C2CC(F)C(=O)N2)=O)CCO1 86654,c1(N(C)C)ccc(C(=O)NCCCCCCNC(=O)Cc2cnn(C)c2)nc1 86655,CC1OC2(CNC(=O)C(=O)NCC(F)(F)F)CC1(NC(C1CCN(C)C1)=O)C2 86656,C1(NC(C(CCSC)O)=O)CCN(C(=O)Cc2ccc(Cl)s2)C12CC2 86657,C=CCC(C)(C(=O)NC1(CNC(=O)C(C)CC)CCC1)N(C)C 86658,C(=O)(C1Cc2ccc(C)cc21)N1CCCN(C(C(CC)CCOC)=O)CC1 86659,c1(C(=O)NC2C(NC(c3c(C)noc3C3CC3)=O)CC2)onc2ccccc12 86660,C1(C(N(C)CCc2ncccn2)=O)CN(C(C2(C)CNC(=O)N2)=O)CCO1 86661,c1(C(C(=O)NCC)N(C2CCN(CC(F)(F)F)CC2)C)noc2c1CCCC2 86662,CC1(C)CCC(C(=O)NC2(C)CN(C(=O)CC3(C(F)(F)F)CNC(=O)C3)C2)O1 86663,S(=O)(=O)(C(Cl)(Cl)Cl)NCC(N1C(C(=O)Nc2scc(C)n2)CCC1)=O 86664,N1(C(c2cc(CNC(C(CC3CC3)OC)=O)[nH]n2)=O)CCC(C)(F)C1 86665,N1(C(COc2cc(C)on2)=O)CCN(C(c2nc3c(s2)COCC3)=O)C(C)C1C 86666,C1(CNC(C(CSC)(C)C)=O)CC(C)CN(C(=O)CC2CC(F)C2)C1 86667,C(CC(=O)NOCC1CCOC1)(C(F)(F)F)NC(CCNC(N)=O)=O 86668,C(=O)(C1=CCCC1(C)C)NC(C(C)C)CNC(c1cc(OCC(F)F)ccn1)=O 86669,C1(C(N2CCC(C(C)(C)C(=O)O)CC2)=O)(OC)CCCOC1 86670,C1(O)(C(=O)NCC(CCOC)NC(CSCCOC)=O)CCCCC1 86671,Cc1nnc(NC2CCN(C(c3nc(C)n(-c4nc[nH]n4)n3)=O)C2)c(C#N)c1C 86672,O(NC(=O)C(C)(C)CCCNC(=O)CCC(C)CC)C(C=C)C 86673,c1(C(=O)OC)ccc(I)cc1NC(C1CCN1Cc1ncco1)=O 86674,C1(C)(OCC(=O)NC(C2(NC(C)=O)CC2)=O)CN(C(C)=O)C1.C(C)(C)(C)O 86675,C1(F)(C(=O)NC2CC(NC(c3cc(C(=O)OC)[nH]c3)=O)C2)CCS(=O)(=O)C1 86676,c1(OC)ccnc(C(=O)NCC(C)N(C(=O)CC(C)n2ccnc2C)C)c1F 86677,C1(CC(=O)NC(C(=O)NCC(N2CCCCC2)C)CO)CCC(C)(C)C1 86678,Cc1ccc(NC(N2CCOCC(C(=O)OC(C)C)C2)=O)c(C)c1 86679,N1(C(C=CC)=O)CCOC(CN(C)NC(C2CC2C(N)=O)=O)C1 86680,C1(NC(C2C(C)(C)C2)=O)CC12CCN(c1cc(=O)n(-c3ccccn3)[nH]1)CC2 86681,C1(NC(C2(CC=C)CCCC2)=O)CN(C(C2CC2=C)=O)CC(C)(C)C1 86682,N1(C(C2(COCC)CC2)=O)CCC(NC(=O)C(C(C)C)NC(N)=O)C1(C)C 86683,c1(OC)ccc2nc(N3CCc4sc(Br)cc4C3)[nH]c(=NCC3CCSC3)c2c1 86684,c1(C(C(=O)NC2C(NC(CC(C)SC)=O)C2)NC(C)=O)c(F)cccc1F 86685,C1(NC(C=CCC)=O)CN(C(c2ccc(-n3ccnc3)cc2)=O)CCC1C 86686,C1(C(N2CC=CC(NC(c3cc(Cl)c(Cl)s3)=O)C2)=O)(OC)CCCCC1 86687,c1(CC(=O)N(CCCn2cc(-c3cnccn3)nn2)C)c(Cl)cccc1Br 86688,c1(C(N(CC(C)NC(=O)Cn2cc(C#N)cn2)C)=O)ncccc1OC(F)F 86689,c1(SC)ccc(C)c(C(N2CCCC3(NC(c4ccns4)=O)CC23)=O)c1 86690,CS(=O)(=O)c1ccc(CN2CC3CC3(C(=O)Nc3ncc(I)nc3Cl)C2)cc1 86691,c1(C(N2CC(CC=C)(NC(c3cnn(C)n3)=O)C2)=O)ccc2ncn(C)c2n1 86692,C(C)(CCC(=O)NOCc1cccc(C)n1)NC(c1cc(C)no1)=O 86693,C1(NC(C2(CC=C)CC2)=O)CC2CC1CC2C(=O)NC(CO)C1CC1 86694,C1(CC(=O)NC(C2(O)CN(C(=O)Cc3ccccc3O)C2)C)CCS(=O)(=O)C1 86695,C1(NC(C2CCCCS2)=O)CCC2(CC1)CN(C(c1ccc(C3CC3)cn1)=O)C2 86696,C1(NC(c2cc(C=C)cc(F)c2)=O)CC(C2CCN(C(=O)CC3=CCCC3)C2)C1 86697,C=CCC(CNC(C1CCCCS1)=O)C(=O)Nc1ccc[n+]([O-])c1 86698,C1(COC)CC(Cn2cc(C(C)OC)nn2)N(C(=O)CCC2CC(F)(F)C2)C1 86699,N1(C(c2ccc(OC)s2)=O)CCC2(CC2C(=O)NCc2cc(C)ccc2F)C1 86700,c1(C(=O)NC(C)Cc2nc[nH]n2)c(CNC(=O)CC(C)(C)N(C)C)cnn1C 86701,CS(=O)(=O)CCC(=O)N1CCN(C(=O)Cc2nc[nH]n2)C(CC(=O)NC=O)C1 86702,N1(C(c2ccc(C)cc2O)=O)CC2CCC(C1CO)N2C(=O)Cc1ccco1 86703,C12(C(=O)NC(C)CCNC(=O)C(C)C3CCOC3)CC=CC(C1)OC2 86704,C1(C(=O)NC(C)C(N)=O)CC(F)(F)CN1Cc1cccc(-n2cncn2)c1 86705,c1(C(=O)NCC2C(NC(=O)Cc3ccn(C(F)F)n3)C2)cccc(Cl)c1 86706,N1(C(C2C(C)C2C)=O)CCC(CCCNC(C2(C)CCCOC2)=O)CC1 86707,c1(C(N(CCNC(c2ccccc2)=O)CC)=O)ccc2nnn(C)c2c1 86708,C1(CNC(c2c(C)[nH]nc2Cl)=O)COCCN(C(c2cc(Br)c[nH]2)=O)C1 86709,c1(C(NNC(=O)C2CC(C)OC2)=O)cc(-c2cn(-c3nccs3)nn2)ccc1Cl 86710,c1(C(=O)NC(c2cn(C(C)C)nc2)C)cccc2c1CCO2 86711,C1(C(=O)NCCOCCCNC(C2C=CC=CC=C2)=O)CCC2(CCOC2)O1 86712,C(=O)(C(CCC(C)C)NC(C1CCC(=O)C1)=O)NC1(COC)CC1 86713,N1(C(C2C(C(N)=O)COC2)=O)CCC(C2CN(C(C3CCCCO3)=O)C2)CC1 86714,C1(C(=O)NC2C(C(=O)OCC)C2)CCN(C(c2ccc(CN(C)C)[nH]2)=O)CC1 86715,C1(NC(C2(CC=C)CCCC2)=O)CCN(C(c2ccnn2C(F)F)=O)CC1CO 86716,Cc1cnccc1C(=O)NCC1C2CN(C(c3cc[nH]c3)=O)CC12 86717,C1(C(N(CCCC)C)=O)CCC(O)CN1C(C1CC2C=CC1O2)=O 86718,C(CCC(O)CO)N(C(CC1(C)N(C(C=CC=CCC)=O)CC1)=O)C1CC1 86719,N#Cc1cccc(F)c1NC(C1CC(F)CN1C(C1CCCS1)=O)=O 86720,C1(NC(c2cc(CNC(c3cc(C)nnc3)=O)on2)=O)CCCC1C1CC1 86721,N1(C(=O)OC(C)(C)C)CC(C(N2CCC3(CCC3O)C2)=O)C(C2CCCC2)C1 86722,C(=O)(C(CC(C)(C)C)OC)NC(C(=O)NCC(COC)(C)O)(C)CO 86723,C1(C(=O)NCCCN(C(=O)CC2CCCC(=O)N2)C)Cc2c[nH]cc2S1(=O)=O 86724,N1(C(CN2C(C)CC2)=O)CCC(CNCCNC(C2(NC(N)=O)CCC2)=O)C1 86725,C1(C(=O)NCCCN(CCCNC(C2(C(C)C)CC2)=O)C)CCCC1(C)C 86726,C1(CNC(C=CS(C)=O)=O)CC(C)(C)CN1C(=O)Cc1nc(=N)[nH][nH]1 86727,C1(NC(c2c(N)c(Cl)ncc2)=O)CC12CCC(NC(C1CC1F)=O)CC2 86728,CCS(=O)CC(=O)N1CCC(C(=O)NC(C)C(C)(C)C#N)(CF)C1 86729,N1(C(c2c(N)c(F)ccc2)=O)CCCC2(CNC(c3coc(Br)c3)=O)CCCC12 86730,Cc1ccc(NC(=O)C(C)(C2CC2)N(C(=O)C(O)C(F)(F)F)C)cc1Cl 86731,c1(C(=O)NCC(CNC(C2C(CCC)C2)=O)(C)O)ccc(N)cn1 86732,C(=O)(CC(C)(C)NC(=O)CN(C)C)OC(C)(C)C.c1(C(C)NC(N)=O)ccc(N)cc1 86733,c1(CNC2C(C(=O)NC(C=C)CO)C2)csc(Br)n1 86734,CN1N=C(CC(=O)N2CC(=O)NCC2C(N2CC3C(C(N)=O)C3C2)=O)CC1=O 86735,Cc1cc(F)c(C(=O)NCC2CC3CCC2N3c2cc(C)nc(CO)n2)c(F)c1 86736,C#CC1(CC)COCCN1CC(=O)NC(C(=O)NCCOCC)c1cscn1.C1CC1 86737,c1(N2CCC(NC(C(CCCC)(C)F)=O)C(C)(C)C2)nc(Cl)nc2c1ncn2CC 86738,C1(NC(C2CC(C#N)C2)=O)CCC(NC(=O)CN2CCS(=O)CC2)CC1 86739,C(=O)(C(F)C(C)(F)F)N1CCC(CC(=O)N(C2CCS(=O)(=O)C2)C)CC1 86740,N1(C(CC2(OC)CN(C(=O)CC3CCCSC3)C2)=O)CCC12CN(C)C2 86741,N1(C(C(C=C)OC)=O)CCC(C(=O)NC2CC3(CC3)C2)C12CCC2 86742,Cc1cc(C(=O)NCC(C)(O)CNC(=O)CCSCC(C)C)nn1C(C)C 86743,C(=O)(CCC(C)(C)C)N(CCCCN(C(=O)CC(O)c1cnc(Cl)s1)C)C 86744,C1(C(C)C)CCOCCN1C(=O)CC1CC(O)CN1C(c1cccs1)=O 86745,N1(C(c2c(NC)nccc2)=O)CCC2CC2(C(=O)N(C)C(C)C)CC1 86746,c1(OCC(=O)NC2(CC=C)CCN(C(=O)C=C(C)Cl)C2)cc(F)ccc1F 86747,c1(-c2cccc(CO)c2)c[nH]c2ccc(Oc3ccccn3)cc12 86748,c1(N(C)C)cnccc1C(=O)NC1CCN(C(C2C3CC(=O)CC23)=O)C1 86749,C(CC(C(=O)NC(CC1CCCC1)CO)NC(C12CC(F)(C1)C2)=O)=CC 86750,CC(C(=O)N1CCSCC1CCNC(c1csc([N+](=O)[O-])c1)=O)P(C)(C)=O 86751,C(C(C)(C)C(=O)NCC(C(=O)NCC1C(CO)C1(C)C)N(C)C)OC(C)C 86752,C(C(C)(C)CC(=O)NC1(CO)CCCCCC1)NC(c1n[nH]c(CC)c1C)=O 86753,c1(C(=O)NC2C(CNC(C(C)OCCCCCC)=O)CC2)ccn2cccc2c1 86754,C1(CNC(c2cnn(C)c2C(N)=O)=O)CCC2(CN(C(=O)OC(C)(C)C)C2)O1 86755,N1(C(C(C=CC)O)=O)CC2CCN(C(c3nn(C)c(Cl)c3Cl)=O)C2C1 86756,c1(C(N(C2CCC(NC(C3CC4(C3)CC4F)=O)CC2)C)=O)cc(N)c(Cl)c(O)c1 86757,c1(C(N2C(CN(C(c3cccc(C#C)c3)=O)C)CCC2)=O)ccc2c(c1)OCC2 86758,Cc1cc2[nH]c(C(=O)NC34CCN(C(c5cnn(CCO)c5)=O)CC3C4)cc2s1 86759,N1(C(CCC=C(C)C)c2nnnn2C)CCCC(O)(CSC2CCCN(C)C2=O)C1 86760,N1(C(c2nc(CNC(=O)Cc3ccon3)oc2)=O)CCC2(CCCO2)C1 86761,c1(CCC(=O)Nc2cc(OC)c(F)cc2)ccc2[nH]ccc2c1 86762,c1(C(=O)NC2CN(C(C(C=C)(F)F)=O)CC2C(F)F)ccc(Cl)c(C)c1N 86763,N1(C(C)=O)CCc2c(NC(C3(C)CCCOC3)=O)cccc21 86764,CC1CCC(C(=O)NC2(CO)CC(F)(F)C2)N(C(c2cn(C)cn2)=O)C1 86765,C1(CNC(COCCC=C)=O)CCCC12CCN(C(C1CCCC3CC13)=O)CC2 86766,Cc1cc(C(N2CCOC(CNC(=O)Cc3conc3C)C2)=O)ccc1Cl 86767,Cc1cc(C(=O)NC2CC3CC2N(C(C2(C)CCC(O)CC2)=O)C3)c(F)cc1F 86768,N1(C(C(C2CCCC(=O)N2)C)=O)CC2CCC1CN2C(C1CCOC(=O)CC1)=O 86769,C(CCCCCN=c1[nH]nco1)N(C(c1c(CCN(C)C)cccc1)=O)C 86770,CC1CCn2c(C(=O)NC3CCN(c4cc(C5CC5)nc(Cl)n4)CC3)cnc2C1 86771,c1(OC)cc(C=CC(N2CCN(C(=O)C=CBr)C(CCO)C2)=O)ccc1O 86772,CCCC(C(=O)N1CCC12CN(C(=O)C(C)Cc1ccnn1C)C2)S(N)(=O)=O 86773,c1(C(N2C(C)CCC(CNC(CSCC(=O)OC)=O)C2)=O)cnn2ccccc12 86774,N1(C(CCN(C(C)=O)C)=O)CCN(C(c2cc(Br)ccc2Cl)=O)CC1C#N 86775,c1(C(N2C(CN(C(c3c(SC)nccn3)=O)C)COCC2)=O)ccc(F)cc1C 86776,C(=O)(C1(CC)CCCc2ccccc21)N(CCNC(C(CCC)C)=O)CCC 86777,C1(C(=O)NCCC(C)SC)N(C(c2cc(C)cc(O)n2)=O)CCCC1(C)C 86778,C(=O)(C(CNC(c1ccc(COC)o1)=O)CC(C)C)NCCCCC(=O)NC 86779,c1(C(N2CC(OCCC(=O)NC3CC(C)(C)OC3)C2)=O)cc(F)ccc1Cl 86780,CN1CC2CN(C(C3OCCC3N)=O)CC2(C)C1.C12(C=O)CCC(C1)C2 86781,CCCC(C)(C)CC(=O)NCC1CN(C(C2(C)CCC23CCC3)=O)CC(C)(C)O1 86782,C(CNC(=O)C(C)NC(=O)C(C)(C)C)(CC)(CC)NC(C(C)OC)=O 86783,C1(C(N(CC(C)N(C(C=COCC)=O)C)C)=O)CC(=O)N(C(C)(C)C)C1 86784,c1(OCCC)ccc(C(=O)NCC2N(C(C3CC=CCC3)=O)CC2)cc1C 86785,C1(N(C)Cc2cn(C(C)C)nc2)CCN(N2CCCN(S(C)(=O)=O)CC2)C1 86786,c1(C(=O)NCC(CN(C(c2cc(CC)sn2)=O)C)C)ccc(C)nc1 86787,c1(N2CC3CCCC(NC(c4c(C)coc4)=O)C3C2)ncc([N+](=O)[O-])cc1C#N 86788,C1(n2cnnn2)(COC(c2ccc(OC3CCOC3)cc2)=O)CCCCC1 86789,C(=O)(C(C)(C)C(=O)NC)N(CC(CN(C(C(CC)n1ccnc1)=O)C)O)C 86790,C(C(C)C(=O)NC1CC(C(C)NC(C2CC2C(=O)OC)=O)C1)OC 86791,N1(C(=O)CSC(F)(F)F)CC2(C1)CN(C(c1n[nH]c3c1COC3)=O)C2 86792,C1(CC(=O)NC(CNC(C(COC)(C)OC)=O)(C)C)CCCS(=O)(=O)C1 86793,N1(CCOCC=C)C(=O)CN(Cc2cnn(C)n2)C1=O 86794,C1(CNC(C2(C)CC=CC2)=O)C2CC1N(C(c1ccc(-n3ccnn3)cc1)=O)C2 86795,c1(C(N(C)CC2OCCN(C(C(CC)=CC)=O)C2)=O)ccc2c(c1)ncn2C 86796,C1(O)(CNC(C(C(C)(C)C)SC)=O)CC2CCC(C1)N2C(=O)Cc1cncn1C 86797,N1(C(Cc2c(F)ccc(C)c2)=O)CC2(CCN(C(=O)CCCCN(C)C)CC2)C1 86798,C(=O)(CC(C(C)OC)NC(C1(CO)COC1)=O)NCCCOC 86799,Cc1ccc(C(C)C(N2CCN(Cc3nccs3)CC2)=O)cc1 86800,CC1CN(Cc2cc(C#N)ccc2Oc2ccc(Cl)cc2)c2cccnc21 86801,C=CCC(CC(=O)N(C)CC1CCCC1)NC(C1CC2(C1)CC2(F)F)=O 86802,c1(C(=O)NC(C2CCOC2)CNC(CCOCC)=O)c(O)cc(Br)cc1F 86803,Cc1cc(F)c(C(=O)NC2CCCC2NC(=O)Cc2ccsn2)cc1F 86804,N1(C(Cc2cnc(C)[nH]2)=O)CCC(N(CCO)C(c2nccn2C)=O)CC1 86805,C1(C(=O)NCc2ccccn2)CSCCN1C(=O)CC1CC2C=CC1C2 86806,CC1(C)CCCC(C(=O)NC2CC3(C2)CC3NC(c2csc(C3CC3)n2)=O)CC1 86807,Cc1cc(Cl)c(C(=O)NC2C3CC2N(C(c2ocnc2C(F)(F)F)=O)C3)s1 86808,Cc1cccc(C(F)C(=O)NCCCCCNC(C2CS(=O)C2)=O)c1 86809,N1(C(C(C)(C)C2CCC2)=O)CC(CNC(=O)CCc2cc[nH]n2)C2(CCC2)C1 86810,c1(CC)noc(C(=O)NCC(C(C)C)NC(=O)C(C2CCOCC2)C)n1 86811,N1(C(C2(C=C)CCC2)=O)CCCC(OCCCOC(c2cncc(C)n2)=O)C1 86812,CC1(C)CC(C)(C(=O)NC2CCSCC2)CN1C(=O)CC1CC(F)(F)C1 86813,c1(C(=O)NC(c2ccc(O)cc2)C)n[nH]c2c1CN(C(=O)Cc1ccco1)C2 86814,N1(C(Cc2n(C)ncc2Cl)=O)CCCC2CN(C(c3csc(O)n3)=O)CC12 86815,CS(=O)CCCCNC(c1cc(CNC(=O)CC2CCCC(=O)C2)[nH]n1)=O 86816,N1(C(C(C)C2(O)CCC2)=O)CC2(CCC2)CC1C(=O)NC1C2CCC1CC2 86817,N1(C(CCC2N(C(C(CSC)OC)=O)CCCC2)=O)CC(=O)NC(C)C1 86818,C1(CNC(C(c2ccc(Cl)cc2)CC)=O)C2CN(C(=O)CSC(C)C)CC12 86819,c1(C(C)=O)ccc(S(=O)(=O)NC2CC(NC(c3cccnc3S)=O)C2)cc1 86820,CC1CCN(C(c2ccccc2Cl)=O)CCN1C(=O)C1=CS(=O)CCC1 86821,C1(NC(C2ON=C(CC)C2)=O)CC2CC1CC2C(=O)NOCC(F)(F)F 86822,C1(C(=O)NCCC2(O)CCN(C(C3CCC=CO3)=O)CC2)CCC2C(C1)C2(F)F 86823,Cc1cc(C)n2nc(C)c(C(N3CCC(C)(NC(=O)C(C)S(N)(=O)=O)C3)=O)c2n1 86824,c1(C(C)NC(c2c(O)ncc(C(C)C)c2)=O)ccc2ccccc2c1 86825,C(C(C)(COC)CC)NC(C(c1cccs1)NC(c1c(COC)cc[nH]1)=O)=O 86826,c1(OC)nc2ccccc2cc1C(=O)N=c1cncc[nH]1.c12csc(n1)C(=O)N2 86827,N1(C(C2OCCC(C)C2)=O)CCC2(CCC2CNC(=O)CN2CCCCC2)CC1 86828,Cc1cc(F)ccc1C1(C(=O)NC(CO)C(C)NC(C2(O)CCC2)=O)CC1 86829,N1(C(CCC(C)(C)C)=O)CC(NC(=O)CN=c2cc[nH]cc2)CC2(CCC2)C1 86830,N1(C(CN2CCN(C(C3CCCN(CC)C3)=O)CC2)=O)CC2C(C1)C2(C)C 86831,C(=O)(C1=Cc2ccccc2C1)NCC(CC(=O)N(CC(F)F)C)C1CC1 86832,C1(CCNC(=O)Cc2csnn2)COCCN1C(=O)CC1(CC2CC2)CCC1 86833,c1(C(=O)NCC2C(NC(c3cccc(OCCOC)c3)=O)C2)cc(N)cnc1Cl 86834,CCCC(C(=O)N1CC2CC(NC(C3CC4(C3)CC4(F)F)=O)C2C1)C(C)C 86835,C(CC1CCC1)(C(=O)N(C)CC1CC(O)C1)NC(C(C)OCCCC)=O 86836,c1(C(=O)NCC2CC(NC(C3CCC(C)NC3=O)=O)C2)ccc2n[nH]cc2c1 86837,N1(C(C=CC(C)(C)SC)=O)CCCCC1CC(=O)NCCc1cc[nH]n1 86838,CC#CC1CCN(C(=O)C(F)CC2CN(C(c3coc(OC)n3)=O)C2)CC1 86839,C1(C(N2C3(CN(C(c4cn(C5CCC5)nn4)=O)C3)CC2)=O)CC2CCCCN2C1 86840,N1(C(CN(C2CCCC2)C)=O)CC2C(CNC(C3CCC(C)(C)C3)=O)C2C1 86841,C1(NC(C2CC(Cl)(Cl)C2)=O)CCC2(CCCN(C(c3ccncc3)=O)C2)C1 86842,c1(NC(C(CCSC)NC(c2sccc2C#N)=O)=O)cc(C)cnc1C 86843,N(C1CCCc2ccoc21)C(=O)NC1C(C(N)=O)CCC1 86844,C1(C(=O)OC)CCC=CC1NC(=O)CCN(C)C(c1ccc(C)cc1)=O 86845,c1(C(N2CCCC(NC(C3C4COCC34)=O)C2)=O)ccc(C(F)(F)F)cc1Br 86846,N1(C(CC(C)C)C(=O)Nc2ccccc2)CCS(=O)(=O)CC(C)C1 86847,N1(C(C(CCC2(OC)CCC2)N)=O)CCN(C2CCCC2)C(C)C1 86848,CC(O)CCCC(=O)N(C(C)CCNC(C1(S(C)(=O)=O)CCC1)=O)C 86849,C1(C(N(CC(C(=O)Nc2c(CCC)cccc2)C)C)=O)CC(=O)OC1(C)C 86850,c1(C(=O)NCC(CNC(CN(C(=O)OCC)C)=O)(C)F)ncncc1C 86851,C(=O)(C(CO)C(C)(C)C)N1CCC(O)(CNC(C(n2ccc(Br)n2)C)=O)C1 86852,C(=O)(C1=NOC(C)(C)C1)NC1CN(Cc2nc(C)sc2C)C(C)CC1 86853,CC(CC(F)F)C(=O)N1CCCCC(N(C(=O)COCC2CC2)C)C1 86854,CC(C)S(=O)(=O)CC(=O)NC(C)C(CO)NC(c1ccccc1Br)=O 86855,c1(C(N2CCNC(CC(F)(F)F)C2)=O)[nH]nc([N+](=O)[O-])c1Cl 86856,c1(CC)ccccc1CC(=O)NC(CN(C(=O)C(CC)NC(C)=O)CC)CC 86857,C1(N(C)CC)CCN(C(C2CCOCC2NC(C2CCN(C)C2)=O)=O)CC1 86858,Cc1ccncc1C=CC(N1CC2CC(NC(=O)CC3CCC4CC34)C2C1)=O 86859,CS(=O)(=O)C1CN(C(c2c[nH]nc2CNC(=O)C(F)(F)C2CC2)=O)C1 86860,C1(C(=O)NCC2CN(C(c3c(SC)ccs3)=O)CC2O)CC2(CCC2)CCO1 86861,c1(C(=O)NCCCC(c2ccccc2)NC(CN(CC)CC)=O)sc(C)cc1Cl 86862,C1(C(=O)NC(CCSC)C(N)=O)CC12CCN(C(=O)Cc1ccccc1Cl)CC2 86863,C1(C(=O)NCCCOCCN(C(CC=C=C)=O)C)Cc2ccccc2O1 86864,CC(C)C(C(=O)N1CCC(c2cccc(F)c2)(NC(c2cocn2)=O)C1)NC=O 86865,C(=O)(N=c1[nH][nH]c2c1CN(S(=O)(=O)CCCCCl)C2)c1cc(C)c(Cl)nc1 86866,C12(CC)CN(C(=O)CCCSC)C(CNC(c3sc(C)c(C)c3C)=O)(C1)C2 86867,C1(C)(C(N(C(CC)CSC)C)=O)CC(NC(=O)C(C)NC(=O)OC)C1 86868,c1(C(=O)NCC(CN(C(c2c(SC)ccs2)=O)C)O)ccc([N+](=O)[O-])c(C#N)c1 86869,c1(C(=O)NC2CC(C)(CNC(C3(C)ON=C(C)C3)=O)C2)cc(C)c(C)cn1 86870,N(C(=NCCN1CCSCC1)NC1CCS(=O)(=O)C1)C1C(C)C1C.N1CCOCC1 86871,c1(COC)cc(C(=O)NC(CC(=O)NC2CC(C(F)(F)F)C2)C2CC2)no1 86872,N1(C(C2(OC)CCSC2)=O)CC2CCC(C1)C(NC(=O)C1=CCS(=O)(=O)C1)C2 86873,C1(c2cn(CC(=O)NCCOCC)nn2)CCCCC1OC.N1CCCOCC1 86874,N1(C(c2c(C)[nH]c(C#N)c2)=O)CCN(C(=O)C(C)(C)C2CCC2)CCC1C 86875,N1(C(C23N(C(c4cc(C)n(C)c4C)=O)CC(C)(C2)C3)=O)CCC(C)C(C)(C)C1 86876,N1(C(C(C=C)(C)C)=O)CCC(C)N(C(c2ccc(C(F)(F)F)s2)=O)CC1 86877,c1(C(N2CC(CCNC(c3cc(OC)ncc3F)=O)C2)=O)cc2c([nH]1)CCCC2 86878,N1(C(CCCOC)=O)CC=CC1(C)C(=O)NC(c1nnc(C)o1)C 86879,C(=O)(C1=CCCC1)NCCC(C)N(C(=O)CCC1CCCO1)C 86880,c1(OC)ccc2c(C(=O)NCC3CCC4(CN(C(=O)C(C)OC)C4)O3)csc2c1 86881,CC1CCC(NC(=O)CCN2CCN(C)CC2)CN1C(C1SCCS1)=O 86882,c1(NC(c2ccc[nH]2)=O)ccccc1OCCO.C12CC(F)C(C1)C(=O)N2 86883,C(CC(O)C(=O)NC1COCCC1C(=O)NC(CO)CCO)N(C)C 86884,c1(CNC(c2c(C)n[nH]c2)=O)cc(F)cc(F)c1.c12c[nH]nc1C1CCN(C1)C2 86885,N1(C(Cn2nc(C)n(C)c2=O)=O)CCC2CN(C(=O)C(C)n3cncn3)CC2C1 86886,C(C)(C(C(=O)NCCC(C)N(C(=O)CSc1cn[nH]c1)C)N(C)C)OC 86887,c1(C(=O)NCC2CCCC2n2cccn2)ccc2c(c1)CCC2 86888,c1(C(=O)NCC(C)(C)OCCNC(C2CCN(C)C2)=O)cccc(C#N)c1 86889,N1(C(C(=C)F)=O)CC2CCN(Cc3ccc(O)c(O)c3)CC2C1 86890,CC1=NNC(=O)C1CCC(=O)NCC(C1CCC1)NC(C1(n2cccn2)CC1)=O 86891,N1(C(C(CN(C)C)N(C(C2ON=C(C)C2)=O)C)=O)CC(S(C)=O)C1 86892,C1(C(=O)NC(C2CN(C(=O)C(=C3CCCCC3)F)CCO2)C)(CC)CCOCC1 86893,C1(NC(C2(CC)CCNC2=O)=O)CCN(C(C2(NC(N)=O)CC2)=O)CC1O 86894,N1(C(C2(OC)CC(C)C2)=O)CCC(F)(C(=O)NCC2COC(C)(C)C2)CC1 86895,N1(C(CC(C)=C(C)C)=O)CCN(C(c2cnn(C)c2)=O)CC(O)C1 86896,C1(C(=O)NCCC2(C(N(CC(F)F)CCOC)=O)CC2)OC2CCC1C2 86897,C(=O)(CCCCCCCO)N(C1CC(n2cc(-c3cn(CC)nc3)nn2)C1)CC 86898,C1(NC(=O)Cc2csc(S)n2)CN(C(=O)C=Cc2ccncc2)C2(CCOC2)C1 86899,C(=O)(C1=COCCO1)N(CCN(C(=O)C(N1C(C)CCC1C)C)C(C)C)C 86900,c1(-c2cn(COC)nc2)ccc2nc(O)cc(C(N3CCCC(Br)C3)=O)c2c1 86901,C1(CC(=O)N(C2C(OC)COC2)C)(NC(=O)CC2COC3CC2C3)CCCCC1 86902,N1(C(C(CCC)OC)=O)CC(CNC(=O)CCn2cncn2)C2(CCOCC2)C1 86903,N1(C(C(CC#C)O)=O)CC2(CC(NC(=O)Cc3cn(C)nc3C)c3nccn32)C1 86904,C(=O)(CC(C1CC1)NC(=O)CN1CCCCC1)NCCN(CC)CC.C1C(C)O1 86905,CON(C)C(=O)C1(NC(=O)C(O)C2CCCC2)CCC1 86906,c1(OC)cncc(C(=O)NCC(C(C)C)NC(C2CC2c2ccc(F)cc2)=O)n1 86907,C(=O)(C1Cc2c(Cl)cccc21)N1CCC(C)(CNC(=O)CC2CCSCC2)CC1 86908,C1(Cc2cn(CCOCC)nn2)COCCN1C(c1cc(-c2ccco2)[nH]n1)=O 86909,C1(CNC(C2CC2c2ccncc2)=O)CCCN(C(C2(c3nc[nH]n3)CC2)=O)C1 86910,N1(C(C)=O)CCCC(O)(C(=O)Cn2cc(C(c3ccc(F)cc3)O)nn2)C1 86911,Cc1cc(=NCc2ccc(CO)o2)[nH]cc1S(=O)(=O)NC(c1ccco1)CO 86912,c1(CC(N)C(N2CCNC(=O)C2c2ccccc2Br)=O)cn2c(n1)CCCC2 86913,c1(NC(CC2(C)CN(Cc3cc(F)c(F)cc3I)C2)=O)ncc(Cl)cc1[N+](=O)[O-] 86914,c1(CC)sc(NC(C2(CNC(=O)CCF)CC2)=O)cc1Br 86915,c1(N2CCN(CCC)CC2)nc(=NC2CCC(N(C)C)C2)[nH]c2c1ncn2CC 86916,Cc1nc(C(N2CCC(F)(CNC(=O)CC3NC(=O)NC3=O)C2)=O)sc1C 86917,c1(C(=O)NCCN(C(C(C)c2cc[nH]n2)=O)C2CCCC2)c(F)cccc1F 86918,C1(C)(C(N2CC(SC)C(N(C)C)C2)=O)COC(C)CO1 86919,c1(C(C)C)nccc(N2CC(NC(c3cccc(Cn4ccnn4)c3)=O)CC2C)n1 86920,C#CC1(N(C)C)CN(C(C2C=CCCN2C(=O)CC2CCCC2O)=O)C1 86921,Cc1cc(CC(=O)NCC23CC(NC(=O)CCc4ccccc4Cl)(C2)C3)c(C)s1 86922,CC1CC(C(N2CCC(CCNC(=O)CC3CCCCO3)CC2)=O)CCO1 86923,Cn1nccc1C1CC1C(=O)NC(C)(CNC(=O)COc1cccnc1)CO 86924,c1(C(=O)NC(CC=CC)C(=O)NCC2(C)CCCOC2)cc2n(n1)CCC2 86925,Cn1cc(CN2CCCC(NC(C3CNC(=O)C3)=O)CC2)c2ccc(F)cc12 86926,Cc1cc(CNC2C3CN(C(=O)C(c4ccccc4)N(C)C)CC23)c(C)s1 86927,N1(C(CC(=C)C)=O)CC(NC(C23CC(C)C2C3)=O)C(c2nccn2C)C1 86928,c1(CN2CCC(C)(C(=O)Nc3c[nH]nc3Cl)C2)ccc([N+](=O)[O-])c(F)c1 86929,c1(C(C)C)ccc(C(=O)NCC2CCN2C(=O)CC2CCCCC23CC3)cc1F 86930,C(=O)(C(O)C(C(C)C)OC)N1C(C(=O)NCC(=O)NC)CC1 86931,Cc1ccc(F)cc1C(=O)NC1CN(C(c2cscc2Br)=O)CC1O 86932,c1(N(C)Cc2ccc(C)s2)nc(=NC2CC(C3CCCC3)C2)[nH]c2c1COC2 86933,C1(NC(c2ccc(SC)cc2)=O)CCCC12CN(C(=O)CC13COC(C)(C1)C3)C2 86934,C1(NC(CNC(=O)OCC)=O)CC2CC(NC(C3(O)CCCCC3)=O)CC12 86935,C(=O)(C1=COCCO1)N(C)CC1CCCN1C(C1(C)CCCO1)=O 86936,c1(OC)cc(CN2C(C(=O)Nc3ncc(F)cc3Cl)CC3CC23)cc(O)c1O 86937,C1(CNC(C(CC)(C)O)=O)CC(F)CN(C(=O)Cc2cncc(Br)c2)C1 86938,C(=O)(CC(C)C(C)C(C)C)NCCN(CCC)C(c1[nH]c(C)cc1C)=O 86939,C1(OCC)CN(C(c2ccn(CC)c2C)=O)CC1CNC(=O)CC(C)(C)O 86940,c12cnc(nc1)CN2.c1(NC(C2C(C(=O)O)C2)=O)cc(-c2ccccc2)on1 86941,C12(CNC(C3N(CC)C(=O)CC3)=O)CN(C(C3CCCO3)=O)CC(F)(C1)C2 86942,CC(C)C(O)C(=O)NCCC(C)N(C(=O)CC1(c2ccccc2)CS(=O)(=O)C1)C 86943,C(=O)(C(F)CC(C)(C)C)N(CC(=O)NCC1(C)CC1(C)C)CCOC 86944,CC1(CNC(=O)NC2CCO2)CCCN(C(C2CN(S(C)(=O)=O)C2)=O)C1 86945,c1(C(N2CC(NC(Cc3c(COC)cccc3)=O)C2)=O)cc(Br)cnc1N 86946,C1(NC(CC2(C=C)CC2)=O)CN(C(c2cc(CC)ccn2)=O)CC1C 86947,N1(C2CN(C(CN(C)C)=O)C2)CC(NC(c2cc(O)cs2)=O)CC1=O 86948,C1(C(=O)NC(C2CCCN2C(=O)CCc2ccc(O)cc2)C)OCCN(C)C1=O 86949,c1(C(N2C(CNC(C(CCC)CC(C)C)=O)CC2)=O)cccc2nc(O)ccc12 86950,CCC(CC(=O)NCC1(CNC(=O)C(C)(C)c2cccs2)CC1(F)F)SC 86951,CN1C(=O)C(NC(=O)C(=O)NC2(C3CCCO3)CCC2)CCc2ccccc21 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86969,C=CCC(C(=O)NC1CC1NC(c1sccc1C)=O)NC(=O)OC(C)(C)C 86970,C1(NC(C2CC(CNC(C(n3ccc(C)n3)C)=O)OC2)=O)CCC=CCCC1 86971,CC(CC(F)F)C(=O)N1CC(NC(c2cnc(Cl)s2)=O)C(C(F)F)C1 86972,C1(C(=O)NCCN)CCC2(CCCCC2)CC1.CCCC(CC)C(=O)N(CC)CC 86973,c1(C(N2CCC(COC)(NC(=O)CC34CC(C3)C4)CC2)=O)cc2c([nH]1)CCCC2 86974,c1(NC(c2n(C)ncc2CNC(C2CCCCC(=O)C2)=O)=O)ccc2c(c1)CCC2 86975,S(=O)(=O)(CCC(=O)N(C)CCNC(c1cc(Cl)nnc1O)=O)NC 86976,Cc1cc(C)c(C=CC(=O)NC2CN(C(c3cc(C)[nH]c3C)=O)C2)c(C)c1 86977,O=C(CC1=CCN(C(C2CCCC2O)=O)CC1)Nc1cccn2nccc12 86978,C1(NC(c2nnc(C)s2)=O)CN(C(c2ccc(N(C)C)cc2F)=O)CC1C1CC1 86979,C12(C(=O)NC34C(CN(C(c5cc(CC)ncc5)=O)C3)C4)CCC(CC1)OC2 86980,C1(CCN(C)C(C2(C)SCCCS2)=O)CCN(C(=O)CC2CCCCO2)CC1 86981,C1(C(=O)NC(CC(C)NC(c2cc(C)n(C)c2)=O)C)CN2CCN1CC2C 86982,CON(CCC(=O)Nc1cnc2ccnn2c1)C(=O)CC1CC2C=CC1C2 86983,c1(C(C(N2C(C(C)NC(=O)Cc3cn(C)nn3)CC2)=O)C)noc2ccccc12 86984,N1(C(C(C=C=C)C)=O)CC(C2CCN(C(=O)Cn3ccc(=O)n(C)c3=O)CC2)C1 86985,C#Cc1ccc(NC(C2COCCC2NC(=O)CNC(C)=O)=O)c(C)c1 86986,C1(C2CCN(C(C3CCC(C)O3)=O)C2)CN(C(=O)CCc2ccn(C)n2)CCO1 86987,C12(NC(CC(C(=O)OC)C)=O)CCC(CN(C(c3ccnnc3C)=O)C1)C2 86988,C(=O)(CCCC(=O)NC(CNC(=O)CSCc1cccs1)C(C)C)NCCC 86989,CS(=O)(=O)c1ccccc1NC(C1CSCCN1Cc1cncc(Cl)c1)=O 86990,N1(C(C(=O)N(CCC)CCNC(=O)C(c2ccccc2)OC)C)C(=O)CCC1=O 86991,C1(C)(C(=O)NC(CC(=O)NCC(CC)CC)C2CC2)CNC(=O)C1 86992,c1(CNC(C2C(OC)(OC)CC2)=O)ccc(C2SC(=O)CN2CCSC)cc1 86993,C1(CNC(=O)NC(c2ccc(F)cc2)C2CC2)CCC2COCC2O1 86994,C(=O)(CCC(C)(C)[N+](=O)[O-])NC(CCCC=C)C(=O)N1CCOC(C)C1C 86995,c1(C(N(C)CC2OCCN(C(C(CC)(C)F)=O)C2)=O)ccc(S(N)(=O)=O)s1 86996,c1(C(=O)NCC2N(C(C(C)=C3CCC3)=O)CC(C)CC2)ccc2sccc2c1 86997,c1(C(=O)NC(C2CCCN2C(=O)Cc2cncs2)C)nc[nH]c2ncnc1-2 86998,C(=O)(C1CCc2nccn21)NC1(C)CCCN(C(c2cccc3ncsc23)=O)C1 86999,CON(C(=O)C1=CCC(NC(c2ccc3occc3c2)=O)C1)C1CCC1 87000,c1(CN2CC(NC(C(CCC)C)=O)C(F)C2)cc(Br)cc(Cl)c1O 87001,c1(C(c2n(CCCC)nnn2)NCc2nc(C)co2)nc(F)ccc1Br 87002,c1(C(=O)NCC2(CN(C)C(C3(C(F)(F)F)CCC3)=O)CC2)ccc2n[nH]cc2c1 87003,N1(C(C)(C)C)CCC(N=c2[nH]c3c(c(=NCC(Cl)Cl)[nH]2)CCC3)CC1 87004,N1(C(Cc2cc(C)on2)=O)CC(NC(C2(C)CC2(F)F)=O)C(C)C1 87005,n1(CC)ccc(C(=O)NCC(O)CNC(c2scc(C)c2Cl)=O)cc1=O 87006,CN1CCOCC1CC(=O)NCc1ccc(C(N2CCC(O)(CO)C2)=O)o1 87007,Cc1nsc(N2CCN(CCNC(=O)CC3CC=CCC3)CC2)c1C#N 87008,N1(C(C=C(C)Cl)=O)CCCC2(C1)CN(C(c1cnc3c(Cl)cccn13)=O)CCO2 87009,C=CC1(C(=O)NCC2C3CCCCCC23)CCN(C(=O)CC2CCC(C)(C)O2)C1 87010,c1(C(=O)NCC(=C)CCNC(c2cc(-c3cccnc3)on2)=O)oc(C)cc1C 87011,C1(C(N2CCCC(C)C2CNC(=O)Cc2cnsc2)=O)CCC2(CC1)CC(O)C2 87012,C1(CN(C(=O)CC2CC(C)(C)CO2)C)COCCN1C(=O)CC1CSCCS1 87013,Cc1nn(C)c(C)c1C(=O)NCCCN(CCCNC(c1ccsc1)=O)C 87014,c1(CC(=O)NCC(CN(C(C2CCC3CCC23)=O)CC)(C)C)cc(F)ccc1F 87015,N1(CC)CCOC(C(=O)NC(C)CNC(=O)C(c2ccc(F)cc2)C2CC2)C1 87016,C=C1COCCN(C(C2(C=C)CCN(C(c3cn(CC)cn3)=O)C2)=O)C1 87017,C1(NC(CCCC#CC)=O)C2CCN(C(c3c[nH]ccc3=O)=O)CCC12 87018,n1(CC)c(C(N2CC(=O)CC2C(=O)N(C)CCF)=O)cnc1O 87019,C1(C2CCN(C(C(CC)C)=O)C2)CCCCN1C(=O)CSCCN(CC)CC.CCO 87020,c1(C(=O)NCCn2cc(CNC(CC(C)OC)=O)nn2)cccnc1S 87021,C1(F)(CNC(C2CC=CCC2)=O)CN(C(=O)C(F)(F)c2csc(Cl)c2)C1 87022,c1(NC(C2CCN(C(=O)CCF)C2)(C)C)cnc(C(=O)OCC)s1 87023,N1(C(C(CNC(C2CCCC(F)C2)=O)N(C)C)=O)CCn2cncc2C1 87024,c1(C(=O)OCC)ccc(OC(C2COCCC2(F)F)=O)c(OC(F)F)c1 87025,c1(CC)ccc(C(N2CC(NC(C3CSCCS3)=O)C(F)C2)=O)cc1 87026,c1(C(CNC(C(C(CC)(C)C)O)=O)NC(=O)C2CC2)ccc2ccccc2c1 87027,N1(C(C2C(C)CC2)=O)CCN(C)C(CC(=O)NC2COCC2F)C1 87028,C1(C(N2CC(CC(C)NC(=O)CNC(N)=O)C2)=O)CCC12CCOCC2.C(C)(C)(C)O 87029,C=CC1CN(C(=O)C(C(C)C)NS(C)(=O)=O)CC1NC(C1CC(=C(F)F)C1)=O 87030,n1(CCC(=O)OCC)nnnc1C(c1cnccn1)NCC(C)C(C)C 87031,C(=O)(C#CC1CCCOC1)NCC(C)N(C(c1c(C)cc(N)cc1)=O)C 87032,C1(C(N(CC(F)F)C(C)C)=O)CCC(C)(C)N(C(=O)CC2CCCO2)C1 87033,c1(CC)nn(C)c(Cl)c1C(=O)NCC(C(C)C)NC(C1CN2CCC1CC2)=O 87034,N1(C(c2cc(C)c(C)o2)=O)CC(O)CC1(C)C(=O)NCCCCF 87035,c1(CCC(=O)NC(C)CC(C)NC(c2cncc(F)n2)=O)ccc(C#N)cc1 87036,O=C(C1CCCc2c[nH]nc21)NCC1CN(C(=O)Cc2ccc(Cl)cc2)CCO1 87037,N1(C(=O)NC(COc2ccc(C(=O)OC)cc2)C)CC(O)CC12CCC2 87038,c1(CC)cc(C(=O)NC2COCCN(C(C3CCCC(C)(C)C3)=O)C2)c(C)nn1 87039,C1(C(N2CC(C#C)(F)C2)=O)CC2C=CC1N(C(=O)CC1C(C)(C)C1(C)C)C2 87040,O=C(CCS(=O)(=O)c1ccc(F)cc1)NC1CCOC(C2CCOCC2)C1 87041,c1(CNC(c2cnn(C)c2)CC)cccc(CC(F)(F)F)c1 87042,C(=O)(C(CCCCCCO)N1CCC1(C)CCO)NCCSC 87043,c1(C(=O)NC(CN(C(c2c(CC)nc[nH]2)=O)CC)C)oc(SC)cc1C 87044,C12CCCC(CC1)N2.N1(C(C(N)=O)=O)CCC(OC2CCC2)CC1 87045,N1(C(c2cnc(CC)nc2)=O)CCCC(C)(C)C1C(=O)NCC(F)CO 87046,c1(N2C(CC)CN(C(C3CCC(=O)N3)=O)CC2)ncnc2c1ccn2C(C)C 87047,c1(OC)cc(C)c(Cl)c(C)c1.C12CCN(CC1)C(=O)NC2CC(=O)OC(C)(C)C 87048,C1(CNC(C(CC)NC(c2n[nH]cc2Cl)=O)=O)C2CCCCCC12 87049,N1(C(C(CC)(C)OC)=O)CCC2(C1)CN(C(c1ccc3nn[nH]c3n1)=O)CCO2 87050,N1(C(COCC=C)=O)CCC(CCNC(c2cc(C)nnc2O)=O)C(F)(F)CC1 87051,c1(C(=O)NC2C(NC(C=C(C)Cl)=O)CCC2)[nH]c2ccc(Cl)cc2c1Cl 87052,C1(F)(C(=O)NCCCOCCN(C)C(C23CC(F)(C2)C3)=O)CC1(Cl)Cl 87053,CC1(C)CCOC1C(=O)NCC1CC(O)CN1C(=O)C=CCF 87054,c1(C(=O)NCC(CCOC)NC(=O)C(C)OC)cncc2nc(C)[nH]c12 87055,C(C)(C)(C(c1ccc(-c2ccccc2)s1)NCC1(c2nn[nH]n2)CCCO1)OC 87056,C(C(=O)OC(C)(C)C)(C(=O)N1CC(NC(c2cccc(C(=O)NC)n2)=O)C1)OC 87057,c1(C(=O)NC2C(OC)CN(C(c3csc(CC(C)C)n3)=O)C2)cnc(C)c(C)c1 87058,CP(C)(=O)c1cnn(CCn2cc(CN3CCCC(CO)C3)nn2)c1 87059,N1(C(CNC(CC)=O)=O)CC(CNC(c2cnccc2Cl)=O)C2(CCC2)C1 87060,C1(C(N(CC(=C)C)CCc2ccncc2)=O)CCCC(NC(=O)OCC)C1 87061,c1(NC(C2N(Cc3cnc(OC)c(Br)c3)C3C(C2)C3)=O)ccc(F)cc1[N+](=O)[O-] 87062,N1(C(c2c(C)nccc2)=O)CCC2C1CCN2C(c1cc2cccnn2n1)=O 87063,c1(OC)cc(F)c(C)cc1NCc1ccnc(Br)c1Br 87064,C(CCCC(=O)N1CCC(O)(CNC(C2CCC(OC)CC2)=O)C1)OCCC=C 87065,N1(C(C2(C#N)C(C)C2)=O)CC2CCC1CN2C(c1nc(C2CC2)cs1)=O 87066,C1(CN(C2CN(C(=O)C=CC3CC3)C2)C)Cc2ccccc2O1 87067,C(C(CC(F)(F)F)NC(c1snc(O)c1Cl)=O)NC(C(C(C)C)OC)=O 87068,C1(O)(C(C)NC(CCOCCC)=O)CCN(C(=O)CNC(=O)C(F)(F)F)C1 87069,C1(C)(NC(CCc2ncc(C)[nH]2)=O)CCN(C(c2cc(C(F)F)n(C)n2)=O)CC1 87070,C1(NC(CC2(C#N)CC2)=O)CC(O)CN(C(=O)Cc2csc(C3CC3)n2)C1 87071,N1(C(CCCCOC)=O)CCC2CN(C(=O)C(CCC(C)C)NC(C)=O)C(C)C12 87072,C(=O)(C(C)S(C)(=O)=O)NCC=CC(=O)NC(C(C)O)(C)C 87073,C1(NC(CC2(C)CCN(C(c3cc(C(N)=O)[nH]n3)=O)C2)=O)(CO)CC2CCCC12 87074,C1(CNC(c2c(C(C)C)ocn2)=O)CCCC2CN(C(C3(C#N)CCC3)=O)CC12 87075,CC(C)CC(O)C(=O)NCC1(F)CCCN(C(=O)C(N2CCCCCC2=O)C)C1 87076,Cc1ccc(O)cc1C(=O)N(CCC(=O)NC1CCCCC1(C)O)CC1CC1 87077,CCC(C(=O)NC1CC(NC(C2(CC(C)C)CCC2)=O)C1)C(C)(F)F 87078,N1(C(CNc2cncc(C(N)=O)c2)=O)CCC(NC(c2ccoc2Cl)=O)C12CC2 87079,N1(C(c2c(C)nc(C)s2)=O)CCN(C(C2CCCC3CC23)=O)C(C)C1 87080,N1(C(C(CC#C)(C)C)=O)CC2(C)CN(C(C)C(=O)NC3CC3)CC2(C)C1 87081,c1(C(=O)NC(C2CCCCN2C(=O)Cc2ccccc2)C)cc2c[nH]cnc-2n1 87082,c1(-c2nc(NCC3C(OCC)COCC3)on2)cc(F)cc(Br)c1 87083,C12(CNC(c3n(CC)ccc3)=O)CCCC1CN(C(=O)Cc1ccn(C)n1)C2 87084,N1(C(CC=CC)=O)CCC2CCC12CNC(c1c(O)cccc1Cl)=O 87085,C(CCCC(=O)NCC(C)(Cn1cccn1)NC(=O)CCc1cnn[nH]1)SC 87086,C(=O)(C(C(=O)NC1(C(=O)NC2C=CCCCC2)CCCCC1)OC)OCC 87087,c1(C(=O)NC(c2ccccc2)CNC(CC(=C)Br)=O)cn(C)nc1OCC 87088,C=CC(C)(CC)C(=O)NCc1csc(CNC(c2[nH]c(C3CC3)nc2C)=O)n1 87089,N1(CC)CC(C(=O)NCC2(O)CC(NC(C34CC(CCO3)C4)=O)C2)CCC1=O 87090,C1(NC(c2n(CC)ccn2)=O)CCC2(CC1)CN(C(C1CC3(CCC3O)C1)=O)C2 87091,C1(C(=O)NC2CCCN(C(CCn3ccc(C)n3)=O)C2)CN2CCC1(C)CC2 87092,Cc1oc(C#N)cc1C(=O)NC12CC1CN(C(c1ccnn1C(C)(C)C)=O)C2 87093,C(=O)(C(O)CCNC(C1(SC)CC(=O)C1)=O)N(CC)CC1CCC1 87094,c1(C(N(CCOCCC(=O)NCC2(CC)CCC2)C)=O)cc(C)ncc1C 87095,N1(C(c2n(CC#C)ccc2)=O)CCC2CC1CN2C(c1n[nH]cc1CC)=O 87096,C(CCC(=O)N1CCCC1C(C)NC(c1c[nH]nc1-c1cnccn1)=O)=C(C)C 87097,N1(C(CCCOCC)=O)CCN(C(c2ccc(C)cn2)=O)C2CC12 87098,N1(C(c2cc(OC)ns2)=O)CCSCC1C(=O)N(C)Cc1ncccn1 87099,C1(C(N(C)CC2CN(C(=O)C(O)c3ccsc3)C2)=O)CCCN1C1CCCCC1 87100,[N-]=[N+]=NC1CCC2(C(N3CCN(C(c4cncc(C(F)(F)F)c4)=O)CC3)=O)CC12 87101,c1(CC(=O)OC2C=CCC2)cc2cc(Cl)ccc2[nH]1 87102,N1(C(Cc2c(C)ocn2)=O)CCC2(CC2)CC1C(=O)NCC(C)(O)CO 87103,N1(C(C(CC)C)=O)CCC(NC(c2cn(CC3CC3)nn2)=O)C(CO)C1 87104,c1(OC)ccc(C2(C(N3CCC(Nc4ccnc(C)n4)CC3)=O)CC2)nc1 87105,CC(C(=O)NCC1CC(NC(=O)Cc2cccs2)CCO1)C(F)(F)F 87106,C(=O)(C(C)S(C)(=O)=O)N(C(C)C(N1CCCC(CN=[N+]=[N-])C1)=O)C1CC1 87107,C#CCC(CC(=O)OC)NC(=O)CC(CCC)NC(=O)C1=C(Cl)CC1 87108,C1(CNC(=O)C(C(F)(F)F)C(F)(F)F)CN(C(=O)C2CC2)CCC12CCOC2 87109,c1(C(N2CCN(C(C3CC(C#C)(O)C3)=O)CC2)=O)cc(Cl)c(Cl)n1C 87110,c1(OC)c(C(N2CC3CCN(c4ncncc4Br)C3C2)=O)cccc1[N+](=O)[O-] 87111,c1(C(=O)NCC(CN(C(=O)CC23COC(C)(C2)C3)C)O)c(N)cccc1Cl 87112,C1(CC)C(C(=O)NC(C)(C)CNC(=O)C=Cc2ccco2)CCN1C 87113,CC1=NNC(=O)C1CNC(c1ccccc1)Cc1ccc(F)cc1 87114,N1(C(C2=NNC(=O)C2)=O)CC2(CCC2)CC1CNC(C1CCOCC1)=O 87115,C(C(=O)NNC(=O)C(N)C(C)C1CC1)n1cc(CCCCOC)nn1 87116,Cc1noc(C(=O)N(C)CCC2CCCCN2C(=O)COC2CCOC2)c1C 87117,C1(C(N2CC(O)(CCNC(C3(OC)CCSC3)=O)C2)=O)CCN(C)S1(=O)=O 87118,c1(C(=O)NC2CC(C(=O)C)C2)cnc(OCC(F)F)cn1.C12CC1C(=O)N2.C1(N)CC1 87119,C#CCCN=C(NC(C#C)CNCC)N1CCC(NC(N)=O)C1 87120,Cc1n[nH]c2cc(C(=O)NC(CNC(=O)CCC3CCCO3)C(C)C)ncc12 87121,C(=O)(C(=O)N(C)C)N(C(CNC(C1(CC(C)C)CC1)=O)C)C 87122,c1(NC(C(c2cn[nH]c2)N(CC)Cc2ccon2)=O)ccc(OC)cc1 87123,N1(C(c2ncoc2C(F)(F)F)=O)C2CCCC1CC(NC(C1(O)CCCC1)=O)C2 87124,C(C)(C)(CCC(=O)NC1CC(C)CCC1O)NC(c1ncn(CC)c1)=O 87125,C1(C(C)C)CN(C(=O)C2=NNC(=O)C2)CCCN1C(c1ccc(Cl)cc1Cl)=O 87126,Cc1ccc2c(C(=O)NC(C)(C)CCNC(C3CC(F)C(=O)N3)=O)c[nH]c2c1 87127,c1(C(=O)NC2C(NC(C(CC)OCC)=O)C2)ccc(-n2cccc2)nc1 87128,C#CC(CNC(=O)C(C(C)(C)C)n1cc(C2(O)COC2)nn1)CC(C)(C)C 87129,S(=O)(=O)(c1ccc(C)cc1)NCCN(C(CC)C)C.N12CCC(F)(F)C(C1)C2=O 87130,c1(C(=O)NCCN(C(C2CCCN(C(C)=O)C2)=O)C2CC2)ccc(O)c([N+](=O)[O-])c1 87131,N1(C(=O)NCC2CCCN(C(C3CC(F)(F)C3)=O)C2)CCN(C2CCC2)CC1 87132,CC(C(=O)N1CC(n2cc(C3(O)CC3)nn2)CO1)N(C)C 87133,c1(C(N(C(C)CNC(C2CCCCS2)=O)CC)=O)cccn2cc(C)nc12 87134,c1(CNC(C2=C(C)CCCC2)=O)n[nH]c2c1CN(C(c1csc(C)n1)=O)CC2 87135,N1(C(CC(C)(C)CC(F)F)=O)CCC2(CCC(CN=c3ccnc[nH]3)O2)CC1 87136,N1(C(C(CC(N)=O)NC(C2C(C)(C)COCC2)=O)=O)Cc2cccnc2C1 87137,CCC(COC)C(=O)NCCC(C)(C)NC(C1CC=C(C)CC1)=O 87138,C1(O)(C(C)NC(=O)C=CC(=O)N(C)C)CCN(C(C2CC(=O)CO2)=O)CC1 87139,O(C1CCc2c(Br)cccc21)C(c1ccc(C2CCC2)cc1)=O 87140,C12CC3(CCN1CCNC2=O)CC3.c1(SCC(=O)OCC)n[nH]c(=N)[nH]1 87141,C(c1c(F)ccc(Cl)c1F)=CC(N1CCC(NC(C(C)=C(C)C)=O)C1C1CC1)=O 87142,c1(C(N2C3CC(C(=O)NCCC(O)CO)C2CC3)=O)ccc2nccc(Cl)c2c1 87143,N1(C(c2ncc(C)nc2)=O)CCOC(C)C1C(=O)NCCC(CO)C(C)C 87144,CCC(CCC(=O)NCC1(C(=O)NCCc2cc(C)ns2)CCC1)OC 87145,C(=O)(C#CC1CCCCO1)N1CCCC(CNC(c2c(C)cn(C)c2)=O)CC1 87146,Cc1nccc(CN(C)CC2CCCCN2C(c2nc(Cl)oc2C)=O)n1 87147,C1(NC(C(CC#C)C2CC2)=O)CC12CCN(C(c1ccc(Cl)c(C)c1N)=O)CC2 87148,c1(C(=O)NCCN(C(=O)CCc2cnoc2)CC(C)O)cccc2ccccc12 87149,Cc1cc(N2CCOC(CN(C)C(C3CC3Cc3ccccc3)=O)C2)nc(Cl)n1 87150,Cc1cnccc1C=CC(=O)NC1CCC1NC(c1cn(C)ccc1=O)=O 87151,C12(C(=O)Nc3ccc(CC)nc3)CCC(NC(=O)C(F)=C(C)C)(CC1)C2 87152,N1(C(CN2CCC(C)(C)C2)=O)CCCC2CCN(C(c3ccc(Cl)cc3)=O)CC12 87153,C(=O)(C(CNC(C1CC1(C)C)=O)CC(C)C)Nc1c(C(C)C)scc1 87154,CC(CC(C)(F)F)C(=O)OCC1OCCCO1 87155,N1(C(CCc2cc(C)no2)=O)CC2CCC(C1)N2C(c1cc(C)c(Cl)cc1F)=O 87156,N1(C(c2c(C)cn(C(C)C)c2)=O)CCC2(CC2C(=O)Nc2ccc(O)c(Cl)c2)C1 87157,C12(C(=O)NCC(CC)C#N)CCC(CC1NC(C1CC3(C1)CC(O)C3)=O)C2 87158,c1(C(N2C(CNC(=O)C3=COCCC3)CC(C)(C)C2)=O)ccc2c(c1F)CCC2 87159,C(=O)(CCCCN(C)C(c1ncccc1Cl)=O)NCC(CC1CC1)OC 87160,C(CCC(C)C)(C(=O)NCCNS(N)(=O)=O)NC(C(CC1CC1)OC)=O 87161,c1(C(=O)NC(CN(C(C2CC(=C)C2)=O)C)(C)C)cc(CC)nnc1C 87162,c1(CN(C)C)c[nH]nc1C(=O)NCC1C=CC(NC(C2CC(=C3CCC3)C2)=O)C1 87163,C#Cc1ccc(C(=O)NCC(C)(C)C(=O)NC2CCN(C(=O)CC)C2)cc1 87164,CS(C)(=O)=Nc1ccc(C(N2CCN(C(=O)CC3CCOC3)C(CF)C2)=O)cc1 87165,Cc1nc(C(=O)NC(CC(=O)N2CCC(n3cncn3)C2)C2CC2)c(C)o1 87166,c1(N2CC(C(=O)Nc3ccc(-c4cn[nH]c4)cc3)C(O)CC2)ncnc2occc12 87167,c1(CC)ncncc1C(=O)NC(C1CCN(C(=O)CCc2cccnc2)C1)C 87168,C(C(C)C(F)C(=O)Nc1cn(C)nc1C#N)NC(c1ccnc(OC)n1)=O 87169,c1(CC)nc(C(C)C)ccc1C(N1CC(CNC(c2cscc2C)=O)C(O)C1)=O 87170,C12(C(N3C(C)(C(=O)OC)CC3)=O)C(NC(=O)CN=[N+]=[N-])C3CC1C2C3 87171,C1(NC(C2(C)CC=CCC2)=O)CN(C(c2cc(Cl)cnn2)=O)CCC1F 87172,C1(NC(C(C)N(C)C)=O)CCN(CC2CCC(C)C2)CC1(C)C 87173,c1(C(=O)OC)ccccc1NC(CN(C(=O)NCc1cncc(OC)c1)C)=O 87174,Cn1nccc(C(=O)NC2CN(C(=O)Cn3nccn3)CC2O)c1=O 87175,N1(C(CC=C)=O)CC(NC(c2ccnc(CC(C)C)n2)=O)CC(F)C1 87176,N1(C(c2nc(C)n(C)c2)=O)C2CCCC1CN(C(C1CC=CCO1)=O)C2 87177,c1(OC)c(Cc2nnnn2Cc2ccc(-c3ccc(C#N)s3)cc2)cccc1Cl 87178,C1(C)(C(=O)NCC(=C)CCNC(C2(c3ccsc3)CC2)=O)CC(O)CN1C 87179,C1(C(N(C(C)CNC(C2CCCS2)=O)CC)=O)(OC)CCC1 87180,C12(C(N3CCCCC(NC(CC4N(C)CCC4)=O)C3)=O)CCC(CO)(CC1)CC2 87181,N1(C(C2N(N(C)C)CCCC2)=O)CCC(C)(C)C(C(=O)N(C)C)C1 87182,C(C(C(=O)N(C)CC1(O)CCOC1)C(C)(C)C)NC(C(C(=O)OCC)(C)C)=O 87183,c1(CC2(C(=O)NC(C)CC(C)NC(=O)CC3(O)CCC3)CC2)ccc(O)cc1 87184,c1(CC)cccc(C(=O)NC2CC(NC(=O)Cc3c(Cl)cnn3C)C2)c1F 87185,[N-]=[N+]=NC1CN(C(=O)NC(c2cnco2)C2CCCC2)C1 87186,N1(C(c2cccc(OC)n2)=O)CCN(C(=O)C(C)OC(C)(C)C)C(C)C1 87187,CC1(C)CCCC(CC(N2CCN(C(c3ccnc(S)c3)=O)CC2C2CC2)=O)O1 87188,c1(C(N(C2CN(C(=O)C3=CCCCO3)CC23CC3)C)=O)c2c(nn1C)CCC2 87189,C1(F)(C(=O)NCCc2cn(C)nc2)CCN(C(C2(CO)CCOC2)=O)C1 87190,c1(CC)nc(O)c(C(N2CCC3(NC(=O)CC4CCSCC4)CC3C2)=O)cc1C 87191,N1(C(c2ccc(C#C)o2)=O)CCCCC2C1CCCN2C(=O)C(F)C(C)C 87192,C1(NC(C(CSC)(C)C)=O)CC2(CCCN(C(=O)C=Cc3cccnc3)C2)C1 87193,Cc1scc(C(=O)NCCC2CN(C(C3CCCC(=O)N3)=O)CCO2)c1N 87194,C(=O)(C(CNC(=O)CN1CCCCC1=O)(CC)CC)NC(C#C)C(C)(C)C 87195,C1(N(C(=O)CCOCC(F)F)C)CCCCN(C(=O)Cc2cnc[nH]2)C1 87196,Cc1nc(N)cnc1C(=O)N(CCCOCCNC(=O)CC(C)n1ccnc1)C 87197,C1(NC(c2cnn(C)c2F)=O)CN(C(C2CC3CCC2O3)=O)CC2(CCC2)C1 87198,c1(C(C)C)cc(N2CCC(NC(=O)C3=CCCCC3)C(C)C2)n2ncnc2n1 87199,CC(C)CCCC(C)C(=O)N1CC(C(=O)NC2(C(=O)N(C)C)CC2)C(C)(C)C1 87200,C=C=C(C)CC(=O)N1CCC(N(C(=O)CCSc2ccccc2F)C)C1 87201,C1(CCC)CN(C(C2(CF)CC2)=O)CC1C(=O)NC(c1cccnc1)CC 87202,CC1CCN(C(=O)C(=O)NCc2cc(C(F)(F)F)ccn2)CCS1=O 87203,c1(C(C(=O)N(CC(C)NC(c2c(C)ccnc2)=O)C)(F)F)cccc(F)c1F 87204,c1(C(N2CC(C)(C(=O)Nc3c(C)cc(O)cc3)C2)=O)c(F)c(F)c(O)c(F)c1F 87205,C1(NC(CN2C(C)CCC2)=O)CCC2(CC1)CC2NC(C1C2CC3C(C2=O)C13)=O 87206,c1(OC)ccc(C(=O)NCC#CC(=O)NCC(=O)NC2CCCC2)s1 87207,N1(C(C(C#C)(C)C)=O)CCOCC(C)(CNC(C2CCC3CC2CO3)=O)C1 87208,c1(C(=O)NCC2(F)CCC(CNC(C3(CO)CCCO3)=O)C2)ccc(F)cc1Cl 87209,c1(NC(C(=O)N(C)CC)=O)c(SCC(C2CCC2)C2CCC2)cc(Br)cc1C 87210,N1(C(C)C)CC(C(=O)NCCOCCCN(C)C(C2(C)CCOC2)=O)CC1=O 87211,N1(CC)CCCCC1C(N1CCCCC1C(=O)NC1CCC(OC)C1)=O 87212,C(CN=c1[nH]c(=NCCC2CCCCO2)[nH]c2cc[nH]c12)c1ccc(SC)cc1 87213,c1(NC(C2(CNCc3cccc(Br)n3)CC2)=O)cc(F)c(Cl)c(Cl)c1 87214,N1(C(CONC(=O)C2(CCC)CC2)=O)CCCC[Si](C)(C)C1 87215,CCCCN=c1[nH]c(=NCc2n[nH]c3c2COCC3)[nH]c2c1SCC2 87216,c1(C(N2C(CO)CC(NC(C3CCC(C)O3)=O)C2)=O)c[nH]cc(Br)c1=O 87217,N1(C(CC(C(F)F)NC(c2cc(C)c(F)cc2)=O)=O)CCC2CCCC2CC1 87218,Nc1sc2c(c1C(N1CCC3(CC(NC(=O)CCC4CC4(F)F)C3)C1)=O)CCC2 87219,[N-]=[N+]=NCCCCCC(=O)N1CCOC(CC(=O)NOCC2CC3C=CC2C3)C1 87220,c1(C(=O)NCC2C3N(C(C4C(CCC)C4)=O)C(CC3)C2)ccc2oc(O)nc2c1 87221,c1(CC=C)ccccc1C(N1CCC(CNC(=O)C(C)n2cccn2)(OC)C1)=O 87222,C1(NC(=O)C=CC=C(Cl)Cl)CCCCC12CCN(C(=O)C=Cc1cccs1)C2 87223,c1(OCCC)ccc(C(N2CCCC2CNC(=O)CC2CCOC2C)=O)cc1 87224,C(=O)(CCC=CBr)Nc1ccc(C(N(C(C)C)C(=O)C2CC2)=O)s1 87225,Cc1nc(C(=O)NCCCN2CCN(C(=O)COC3CCCC3)CC2)c(C)s1 87226,N1(C(c2cc(C)c(Cl)s2)=O)CC2CC1CN2C(C1CC(C2CC2)=NO1)=O 87227,N1(C(C2OCC(C)(C)C2)=O)CC(C2CC2)(C(=O)NC2C3CCCC2CC3)C1 87228,c1(CN2C(C)(C(=O)Nc3ccc(N(C)C)cc3)COCC2)c(F)ccc(Br)c1F 87229,c1(C(=O)NCCCCN(C)C(C2CCC2)=O)csc(C2CC2)c1 87230,N1(C(Cc2cc(C)[nH]n2)=O)CCCC(NC(c2nnc(O)cc2C)=O)CC1 87231,C(C1=CCN(C(=O)C(c2ccncc2)C)CC1)NC(C1C(COC)C1)=O 87232,c1(C(=O)NCCCNC(c2c(NC(=O)OC)cccc2)=O)cn(C)c(=O)nc1O 87233,C1(C2CCOCC2)(CNC(C2(C)CCCCC2)=O)CCN(C(C2CC=CC2)=O)C1 87234,N1(C(C2N(C(CCC)=O)CCCC2)=O)CC2(CCCCN(C(=O)C(C)CO)C2)C1 87235,C1(NC(c2cc(C3CC3)no2)=O)CC2CCC1(N=c1[nH]nc(C(F)F)o1)C2 87236,C(=O)(CC(O)CC(C)(C)C)NCC(=O)NCC(=O)NCCCOCC=C 87237,C1(C(=O)NCC(C)CO)CC(O)CN1C(c1cc(Cl)no1)=O 87238,N1(C(C2CCC(=O)C2)=O)CCC2(CCCN2C(c2cscc2F)=O)C1 87239,C(=O)(CCCCCN(C)C)N1CC(CCC)C(C(N2CC(F)C2)=O)C1 87240,c1(NC(CCC)CCCNC(C2CCC2(C)C)=O)c([N+](=O)[O-])c(CC)nn1C 87241,CC1(C(N2CCCC2CNC(=O)CC2CCCC2O)=O)CC1(F)F 87242,N1(C(CN(C)S(N)(=O)=O)=O)CCC2(CC1)CC2NC(=O)CCSc1nccn1C 87243,N1(CC(CC(=O)OC)NC(C)=O)CCCN(Cc2noc(C3CC3)n2)CC1 87244,C1(CNC(CN(C)C(c2ccccc2)=O)=O)CCCCC1NC(=O)CC(F)F 87245,c1(OC)ccc(C2(C(=O)NC(C)CC(C)NC(C3CCC(=O)N3C)=O)CC2)cn1 87246,CC(C)(CCC(=O)NC1(CNC(=O)C(O)(C2CC2)C2CC2)CC1)[N+](=O)[O-] 87247,CC(CC(=O)N(C1CCN(C(C2(C#N)CCC2)=O)CC1C)C)C(F)F 87248,c1(C(C(=O)N2CC(F)C2)NC(CCOC(C)C)=O)cnn(C)c1 87249,C12(NC(CN(c3ccc(Cl)cc3)C)=O)CCC1CN(C(c1c[nH]c(=O)cn1)=O)C2 87250,c1(C(N(C2CC(NC(CN(CCC#C)C)=O)C2)C)=O)cc2occc2n1C 87251,N1(C(c2cn(C)nn2)C(=O)NCC(=C)C)CCCC(OCCOC)C1 87252,c1(CC(=O)N(C2CC2)CC2CCN(C(C(COC)N(C)C)=O)C2)c(C)noc1Cl 87253,C1(C(=O)NOCc2ccccc2F)C2CCCC2CN1C(=O)CCC1CCCO1 87254,CC1c2ccc(F)cc2CCN1C(c1cnsc1)C(=O)Nc1cccc([N+](=O)[O-])c1 87255,c1(C(=O)OCC)c(Nc2cc(NCCNC3CCOCC3)ncn2)ncnc1Cl 87256,CC(CC(C)NC(C1CCCN1c1cnccn1)=O)NC(=O)C(C)(C)C 87257,c1(CC)nn(C)cc1NC(C(=C1CCCN1C(=O)OC(C)C)C)=O 87258,c1(C(=O)NCCC(=O)NC(CC)C)c[nH]nc1CCNC(=O)CC1CC1 87259,C1(C(=O)NC(c2ccccc2)CC)CC2(CCC2)CN1C(=O)C(CO)C(F)(F)F 87260,C1(NC(COC(C)(C)CNC(C2(C)CCC(=O)C2)=O)=O)CCC(=O)NC1=O 87261,C1(C2CCCN(C(=O)C(C)(C)CC#N)C2)(NC(C(c2ccncc2)C)=O)CC1 87262,CC1CN(C(=O)Nc2nc(-c3ccc4c(c3)OCCN4)cs2)c2cnccc2O1 87263,C(=O)(C(CNC(C1CNC(=O)N1)=O)CC1CC1)N(CC(C1CCC1)OC)C 87264,c1(C(=O)NC(CC)CN(C)C(C2(CCF)CC2)=O)cc(C)c(Cl)c(C)c1 87265,CC(CNC(c1ccc(O)cn1)=O)C(F)C(=O)NCCc1cccnc1F 87266,N1(Cc2c(OC)nccc2)CC2CC1CN2C(c1ccc(O)c(F)c1)=O 87267,c1(COC)nc(OC)cc(N(C2CCCN(C(=O)CN3CCC3)C2)C)n1 87268,c1(C(C)NC(C(CC)NC(c2ccccc2)=O)=O)cc2ccccc2s1 87269,C1(NC(C23OCC(C)(C2)C3)=O)CC2CC1N(C(=O)CCCCc1cnn[nH]1)C2 87270,C1(CC(=O)NCCC2(O)CN(C(COCC=C)=O)C2)CCOC(C)(C)C1 87271,C1(C(=O)NC(C=C)C2CCC2)CN(C(=O)C(CC)=CCOC)CCC1(C)C 87272,c1(C(N2C(C(C)NC(c3cc(Cl)cnn3)=O)CCC2)=O)cncc2nc[nH]c12 87273,C1(c2nnnn2C(C)(C)CC)(NCC(CC)(C)CC)CCS(=O)CC1 87274,CON(CCCO)C(=O)C1(CO)CCCN(C(c2cnnc(C)c2)=O)C1 87275,C1(CN(C(C=CCOC)=O)C)CCCN1C(C1(c2cccnc2)CCCC1)=O 87276,CC1CN(C(C2CCC(C)(C)CC2)=O)CC1(C)C(N1CC(C)(F)C1)=O 87277,c1(NC(C(CC)NC(=O)CC(F)(F)F)=O)ccc(OC)cc1Br 87278,C=C(C)C1CCC(C)CC1NCCCOc1ccc(Br)cc1 87279,C1(CC)CCN(C(=O)CCC2(C)CC2)C1C(=O)N(CC(C)(C)COC)C 87280,c1(C(N2C(CN(C(C(C)CC3CC3)=O)C)CCC2)=O)ncccc1OC(F)F 87281,c1(C(=O)NC23CN(C(C(CC=C)C)=O)C(CC2)CC3)cc(C#N)c(O)nc1N 87282,C1(COC)N(C(=O)CCCN(C)C(c2csc(C)c2C)=O)CC1(C)C 87283,N1(C(C(CC)CC)=O)CC2CC1CC2NC(c1cnc(C)nc1C(F)(F)F)=O 87284,C1(CN(C)C(c2scc(Cl)c2Cl)=O)CN(C(=O)Cc2cncs2)CCO1 87285,N1(C(C2CC(CC)(CC)C2)=O)CC(C(=O)NC2CCCC2CCO)CCC1C 87286,C1(C)(OC)CCCN(C(=O)CC=CCNC(=O)C2=C(C)OCC2)CC1 87287,Cc1c(C(=O)NCC2COCCN2C(=O)Cn2cc(Br)cn2)cncc1Br 87288,C1(CC)CN(C(c2cocc2C)=O)CCC1NC(C1(C)CC(F)C1)=O 87289,c1(C(N2CCCC2)CNC(C(=O)NC(C)CCC2CCCO2)=O)cccc(Cl)c1 87290,C(=O)(CCCCNC(=O)C(C)(F)c1ccon1)N(C)Cc1cc[nH]n1 87291,c1(OC)ccc(CCC(=O)N(C2CN(C(=O)CC3CC(C)C3)C2)C)cn1 87292,CC(CC(=O)N(C)CC1(O)CCN(C(=O)C(F)(F)CO)C1)C(F)(F)C(F)(F)F 87293,c1(C(N)=O)ccc(C=CC(=O)NC2CC(NC(c3cscc3Cl)=O)C2)o1 87294,N1(CC2(NC(C=COCC)=O)CC2)CCN(C(=O)C(F)(F)c2ccccn2)CC1 87295,Cc1cc(C(=O)NCC(=C2CN(C(=O)Cc3ccn(C(C)C)n3)C2)F)n(C)n1 87296,C(CO)(CCCCNC(C1(C)COC(=O)OC1)=O)NC(C=COCC)=O 87297,C1(CNC(CC=CC=C)=O)(CNC(=O)CCNC(=O)CC(C)C)CC12CCC2 87298,CC(C)CCCCC(=O)NC1CC1CNC(c1ccnc(OCC(F)F)c1)=O 87299,CC1(C)CC(C)(C(=O)NCCC2(CNC(C3CNC(=O)C3)=O)CC2)C1 87300,Cc1cc(C(N2CCCC2CNC(c2ccc(=N)[nH]c2)=O)=O)ccc1Br 87301,c1(C(N2CC(OCCNC(C3C=CCS3)=O)C2)=O)nnc2ccccc2n1 87302,C12(C(N(CC(CC)NC(=O)Cc3cc(C4CC4)on3)CC)=O)CCCC1CC2 87303,c1(C(N2CCC(OC)(CN)C2)=O)c2c(nn1C)CCS(=O)(=O)C2 87304,CCCC(C)C(CC)(c1nnnn1CC1CC1)NCCOCc1ccc(Cl)cc1 87305,N1(C(C(C)=C(CC)C)=O)CCC2CN(C(c3cn(CC4CCOC4)nn3)=O)CC12 87306,c1(CC(=O)NCC2C(CNC(CSCC=C)=O)C2)ccc(C)nc1 87307,c1(C(N2C(C)CCC(CC)C2)C(=O)NCCCF)ccc(S(C)(=O)=O)c(OC)c1 87308,CS(=O)(=O)CC(=O)NC1CCCCC1NC(=O)CNC(=O)C(F)(F)F 87309,C12(CNC(c3n(C)cnc3)=O)COCCN1CCN(C(c1cnsc1)=O)C2 87310,CCC(CC(C)C)C(=O)N(CC(C)(C)CNC(=O)CC1CCC(C)(C)CC1)C 87311,c1(CC)ccoc1C(=O)NCC1(CNC(C2CN(C3CCC3)C2)=O)CCC1 87312,N1(C(c2cc(C3(C)CC3)on2)=O)CCCC(C2CC2NC(=O)CCP(C)(C)=O)C1 87313,C1(NC(C2CCC(=O)NCC2)=O)CCc2nn[nH]c2C1 87314,C(=O)(C(C)(C)CCCOC)N(CC(CC)NC(=O)Cc1ccnc(O)c1)C 87315,N1(C(C2C(C(C)C)CCC2)=O)CCCC(C)(C)C1C(=O)NC1CCC2(CCC2)C1 87316,c1(C(=O)NC(C2CCN(Cc3cccnc3Br)CC2)C)cc(Cl)cnc1Br 87317,C1(NC(C(CC)NC=O)=O)C=CCN(C(=O)COc2cccc(OC)c2)C1 87318,N1(C(CC=CC=C)=O)CC(C2CC2)(C(=O)NCC2CC(C)C2)C1 87319,Cc1ccc2c(c1)C(C(=O)NC(C)(C)CNC(C1CC1c1ccccc1)=O)C2 87320,c1(OC)ncccc1CN1CCC(N(C)C(C2CCN(C)CC2)=O)C1 87321,C(=O)(NNc1ncc(Br)c2ccccc12)C(C)(C)CNC(=O)OC(C)(C)C 87322,C1(CCC(N2CC(CC(C)NC(=O)CN(c3ccccc3)C)C2)=O)CCCN1C 87323,C12(C(=O)NCC(C)(C3CC3)NC(=O)CC34COCC(C3)C4)CCC(CC1O)C2 87324,N#CCCCC(=O)NC1CCN(C(=O)COc2ccc(Cl)cc2)C1 87325,c1(CC(N2CC(CNC(C3(C)CC(C#N)C3)=O)OCC2)=O)ncn2c1CCCC2 87326,c1(C(N2CCC(C(C)C(N3CC(CO)(CF)C3)=O)C2)=O)nnn(C)c1N 87327,C=CC1(C(=O)NCCOCCN=[N+]=[N-])CCN(C(=O)NCCCCl)C1 87328,c1(CC(=O)NCCCCCNC(c2sccc2F)=O)ccc2n[nH]cc2c1 87329,C1(NC(c2ccc(C(N)=O)cc2)=O)CC2CCC1N(C(c1cc(Cl)c[nH]1)=O)C2 87330,C(CCCCCO)NC(CC(C)N(C(CN1CCC(C)C1)=O)C)=O 87331,C(=O)(C(C)C(C)c1ccc(F)cc1)N(CCNC(=O)CCc1ccc(Cl)s1)CC 87332,CN1CCOC(CC(=O)NC(CCN(C)C(c2ccco2)=O)c2cccs2)C1 87333,Cc1cc(S(=O)(=O)NC(C2COC3CNCC23)=O)c(Cl)cc1Cl 87334,N1(C(CN(C(=O)OC)C)=O)Cc2ccnn2CC(NC(=O)CNC(=O)C2CC2)C1 87335,C12(n3cc(CCCCC)nn3)CCC(NC(c3cc(Cl)n[nH]3)=O)(CC1)C2 87336,Cc1cc(Cl)cc(C(=O)NCC2CC2CNC(=O)CCCC(F)(F)F)c1C 87337,CN1CCOC(C(=O)NCC(O)CCNC(c2cnoc2-c2ccco2)=O)C1=O 87338,c1(CC)ccsc1C(=O)NC(C(=O)NCCc1cncn1C)C1CC1 87339,Cc1ncc(N)cc1C(N1CC(C(C)NC(c2nc(Cl)c(Cl)s2)=O)C1)=O 87340,c1(C(N(CCCCNC(C(CC)C(C)(F)F)=O)C)=O)noc2c1CC(C)CC2 87341,c1(C(N2C(CC)CN(C(=O)CC(C)F)CC2)=O)cnc2scc(C)n2c1=O 87342,c1(C(C(=O)NCC(C(C)C)NC(=O)C(=O)NCC(F)(F)F)C)cncc(F)c1 87343,c1(CC(N2CCC(C(C)NC(c3nc(C)sc3)=O)C2)=O)ccc2c(c1)ncn2C 87344,c1(OC)cc(CCN2CCCC2)cc(OC(=O)COCc2nc[nH]n2)c1OC 87345,C(=O)(C(C)(C)C(N)=O)N1CC(NC(C2C(C)OCCC2)=O)C1 87346,CN1CCN(C(=O)C(O)CCn2cncn2)CC1CNC(C1(C(F)F)CCC1)=O 87347,c1(SCC(=O)NC2CCN(C(CC(CCC)C)=O)C23CC3)nnc2ccccn12 87348,c1(C(=O)NCCN(C(=O)C(C2CCC(=O)N2)C)C(C)C)ncc(F)cn1 87349,Cc1cc(=O)n(CCNC(C2CCC(C)(C)CC2)CO)cn1 87350,C1(C(N(C2CCC(CNC(C(C)(C)OC)=O)CC2)C)=O)CCC12CCCO2 87351,N1(C(c2c(COC)n(-c3ccc(C)cc3)nc2)=O)CCCN(C)C(=O)C1 87352,Cc1cccc(C(F)C(=O)N(CCCCNC(c2nn(C)cc2Cl)=O)C)c1 87353,N1(C(C(C)(C)OC)=O)Cc2occ(C(=O)NC3CN(C)CC3(C)C)c2C1 87354,C#CCCCC(C)C(=O)N(CCN(C)C(C1(C)COC(C)(C)CO1)=O)C(C)C 87355,C(CC(C(C)C)NC(=O)CC1CCC(=O)C1C)N(C(c1ccc(SC)o1)=O)C 87356,n1(C(C)(C)C)ncnc1CNC(=O)NCC1CCCCS1 87357,CC1CN(C(C2COC2)=O)CC(C)N(C(=O)Cc2ccn(C)c2)C1 87358,c1(C(c2n(CC=C)nnn2)NCC2(OCC)CC=CC2)ccnn1C=C 87359,Cn1cc(C(=O)NC23CCCC(NC(=O)C(F)C(F)(F)F)(C2)C3)ccc1=O 87360,CN1CCCCC(C(=O)N(C)CCN(C)C(c2cn(CC(F)(F)F)cn2)=O)C1=O 87361,C(=O)(CCCCn1ccnn1)N1C(CNC(C(C)NC(c2cccs2)=O)=O)CC1 87362,c1(C(N2CC(O)(CCNC(C3C(CC)N(C)CC3)=O)C2)=O)cc(O)ccc1C 87363,N1(C(c2c(Cl)ccc(C#C)c2)=O)CCCC2(NC(=O)Cn3ccc(C)n3)CC2C1 87364,Cc1cc(C)n(C(C)CC(=O)N(C)CC2CCN(C(c3ccc(F)o3)=O)C2)n1 87365,C1(NC(C(C)CO)=O)C2CC3C1C3C2C(=O)Nc1cc(O)cc(F)c1 87366,Nc1c(C(N2CC(NC(=O)Cn3ncnn3)CC(F)C2)=O)ccc(Cl)c1Cl 87367,S(=O)(=O)(c1c[nH]ccc1=NCc1ccc2occc2c1)N(C)Cc1cc(C)on1 87368,C12CCC(CC1)CC(=O)N(C)CC1CCCN1C2=O.CCCCCCO.C(C)(=O)O 87369,C(=O)(C(C)(C)C(C)(F)F)N1CC2C(C(N(C3CCOCC3)C)=O)C2C1 87370,N1(C(C2(SC)CC2)=O)CCC(C)C(NC(=O)C(C)(c2ccccc2)OC)C1 87371,C(=O)(C(CC)C(C)(C)CC)N1CCCC(N(C(CCCC(=C)C)=O)CC2CC2)C1 87372,C(CC(C)C)(C(C(=O)Nc1ccc2c(c1)OCO2)N1CCOCC(CO)C1)OC 87373,c1(OC)cc(C)c(C(C)Nc2cc(NCC(C)S(=O)(=O)NC)nc(C)n2)cc1C 87374,S(=O)(=O)(c1ccc(Br)s1)N1C(C(=O)Nc2cc(C(C)(C)C)no2)CCCC1 87375,C(=O)(C(CC(C)C)NC(N)=O)NCC(=O)NCC1(CC)CC1 87376,CCCCCC(O)C(C)C(=O)NCCOCCCN(C)C(C1CCOC(C)C1)=O 87377,CN1CC2C(CCCN2C(=O)NC2CCCN(Cc3ccccc3)C2)C1=O 87378,CC1(C)CCC(C(=O)NC(CCO)C2CC2)CN1C(C1(O)CCCC1)=O 87379,CCC(C)(COC)C(=O)N1CSCC1C(=O)NCc1nn(CC)nc1C 87380,C(=O)(C=C1SCC(=O)N1C)NCC(C)NC(C1CCCCC1)=O 87381,C1(CNC(c2c(CC)nccn2)=O)CN(C(C2CCOC(=O)CC2)=O)CCCO1 87382,N1(CC)CCCCC1CN=C(NCc1ccc(NC)cn1)NCc1cc(C)on1 87383,C1(F)(CNC(C(C)OC)=O)CN(C(=O)CCNC(c2ccsc2)=O)C1 87384,N1(C(=O)Nc2cc(C)on2)CCN(C(=O)C(C)N(C)Cc2ccccc2)CC1 87385,c1(CNC(CC)C(C)Cc2ccccc2)ccc(C#N)n1C 87386,C1(NC(C(CCC)C)=O)CN(C(c2ccn(-c3cccnc3)n2)=O)CCC1(C)C 87387,c1(C(=O)NCC(CC)(C)NC(C2C(C(=O)OC)C2(C)C)=O)ccc(CF)cc1 87388,C1(C(N(CC#C)CCF)=O)CN(C(=O)C=C(C)C2CC2)CC1(C)C 87389,c1(C(=O)NC2(CC=C)CCN(C(=O)C=CCOC)CC2)nc2ccc(Cl)nn2n1 87390,C=C=CC(C)C(=O)NCC1CCCN(C(C2(C)COC(=O)N2)=O)C1 87391,c1(C(=O)NCC(CNC(CC(=O)OCC)=O)(C)C)noc2c1CN(C(C)=O)CC2 87392,O=C(C1=CCCCCC1)NCc1cc[nH]c1C(=O)NCC1OC(=O)CC1O 87393,CC(C)S(=O)(=O)CC(=O)NC1CCN(C(C2CCCCCS2(=O)=O)=O)CC1O 87394,c1(C(N2CCC(C(=O)Nc3ccc(C4CC4)cc3)(CF)C2)=O)cccc(Cl)c1 87395,Cc1cc(C(=O)N(C2CCCCC2)CCNC(=O)CCCF)cc2c[nH]nc12 87396,c1(C2(NC(CCC(=O)Nc3cccc(C)n3)=O)CCC2)c(F)cccc1F 87397,CC(C)CCCC(=O)N1CCC(NC(=O)C=CC2CCCCC2)C(O)C1 87398,CC(C)C(C)(CNC(C1CCC(=O)C1)=O)NC(c1ccc(C2CC2)nn1)=O 87399,C1(C)(C(N(CC(C)NC(C2(CC#C)CCC2)=O)CC)=O)CCCOC1 87400,c1(C2N(C(c3ncccc3Br)C(=O)NC3COC3)CCC2)ccc2nonc2c1 87401,Cc1nnc2c(C(N3CCCN(C(C4CCCSC4)=O)C(C)C3)=O)nccn12 87402,O=C(CC1NC(=O)c2ccccc21)NCCC1CCN(C(C2SCCS2)=O)C1 87403,C(CCC(C)CC(=O)N(C)CC1(NC(=O)COC(C)(C)C)CC1)=C(C)C 87404,c12cc(Br)ccc1C(=O)OC2.C(C(C)C(=O)OC)OC 87405,N1(C(CNC(CC(c2c(C)n[nH]c2C)C)=O)=O)CCOC(C)(C(F)F)C1 87406,N1(C(C(CC#C)C)=O)CC(NC(c2ccn(C)c(=O)c2)=O)CCC1C 87407,CC(CN=c1[nH]cnc2c(F)c(F)ccc12)N(C)C(c1ccc(Cl)c(F)c1F)=O 87408,N1(C(C(C2CCOC2)NC(Cn2ncc(C)c2)=O)=O)CCCC2(CC1)CC2 87409,C(=O)C1=CC2C=CC(C1)C2.N1(N2CCC(CC)C2C=O)CCCC(C)(COC)C1 87410,C(C)(CCS(C)(=O)=O)NC(=O)NCc1ccc(CC)nc1 87411,c1(C(=O)NC(CNC(C2CCCSC2)=O)C2CC2)cccc(OCC(F)F)n1 87412,C(=O)(C1Cc2ccc(F)cc21)NC1(C)CC(NC(CC(C)c2cnn(C)c2)=O)C1 87413,Cc1cccc2nc(NC(=O)CC3CCCN3C)[nH]c12 87414,N1(C(C2N(C)CCOC2)=O)C2CCC1CN(C(c1ccc(C(F)F)c(F)c1)=O)C2 87415,N1(C(C)=O)CCC(CC(=O)NCCCN(C(c2cncn2C)=O)C(C)C)C1 87416,C=CCCC(=O)N(C(CNC(c1cscc1Cl)=O)Cc1ccccc1)C 87417,C1(C(=O)O)COC2CN(C(c3ccccc3-n3cc(C4CCCC4)nn3)=O)CC12 87418,N1(C(C(C(C)O)C)=O)CCCCC(NC(=O)CCc2ccsc2)C1 87419,C1(C(=O)NCCC(=O)NC)CCOCC1NC(c1ccc(O)cn1)=O 87420,C#CC1(C(=O)N(CCNC(=O)CC(=O)NCC)CC)CCCC1 87421,c1(OCC(=O)NCCN(C(C2(CF)CCCC2O)=O)CC2CC2)cccc(O)c1 87422,Cc1nc2ncnn2c(NC2CC3CC(C2)N(C(C2CN(C)CCO2)=O)C3)c1C 87423,c1(NCC2(CNC(=O)CCc3cc(Cl)cs3)CC2)ncnc2cc(C3CC3)nn12 87424,C12(C(=O)NCCC(C)NC(C3CC4(CCO3)CC4)=O)CC3CC1C2C3(F)F 87425,c1(CSC)nc(C(N2CCCC2CNC(=O)C=CCF)=O)c2ccccn12 87426,CCC(C)C(C(=O)NC1CC(NC(C2CCOC(C)(C)C2)=O)C1)c1ccccc1 87427,c1(C(N(C2CCC(NC(c3ccnn3C(F)F)=O)C2)C)=O)cnn(C(F)F)c1Cl 87428,C1(C)(OCC)CC(NC(=O)Nc2ccccc2OCC2CCCO2)C1(C)C 87429,c1(OC)cccc(CCC(N2CC3C(NC(C4(Cl)CC4(C)C)=O)C3C2)=O)c1 87430,C1(C(N2CCC2CNC(C2ON=C(C)C2C)=O)=O)(CC)CC(F)(F)C1 87431,c1(COC)nc(NCCC(C(C)C)OC)cc(=NCC(=O)OC)[nH]1 87432,C(=O)(C1=C(c2ccccc2)SCCO1)NCCN(C(CC=C)=O)CC(C)O 87433,C1(OC)(OC)CCN(Cc2ccc(Cc3ccccc3)cc2)CC1O 87434,c1(CN2CC(CC(=O)NCC(=O)N(C)C)C2)cccc(C#N)c1 87435,c1(CC)ncc(C(=O)NC2CN(C(C3CCC(C)(C)CO3)=O)CCC2C)c(O)n1 87436,C1(OC)CCCCN(CC(=O)NCC(C)N(C)C(C2C(C)(C)OC2(C)C)=O)C1=O 87437,N1(C(CCCC#CC)=O)CCC2(CC1)CC(NC(=O)CSC)CCO2 87438,Cc1cc(=NC(=O)C2(c3cccc([N+](=O)[O-])c3)CC2)cc[nH]1 87439,C1(CNC(C2(C)CCC2)=O)C2CN(C(=O)CCc3cccs3)CC12 87440,C1(C(N(C2CCNC2)CC(=O)O)=O)CC(=O)N(c2cccc(Br)c2)C1 87441,N1(C(C(C(C)C)n2cnnc2)=O)CCCN(C(=O)CCCCC2CC2)CC1C 87442,CC1=C(C(=O)N2CC=CC(NC(c3ccc(C(N)=O)c(Cl)c3)=O)C2)CCO1 87443,C(c1cc(Cl)c2c(c1)OCO2)=CC(N1CCC(C)C(NC(=O)COC(F)F)C1)=O 87444,C(c1ccc(C#N)cc1)=CC(=O)NC1(CN(C(C2CC(C)OCC2)=O)C)CC1 87445,Cc1cc(O)nc(C)c1C(N1CC(F)(CNC(C2(C)CC3CC3C2)=O)C1)=O 87446,C(=O)(C(C)(C)CC(C)C)N1CC(C(N2CCC(C=C)(O)C2)=O)OC(C)C1 87447,C1(OC)CC(C(F)(F)F)CN(C(=O)OC(C)(C)C)C1.C(C(C)C1CC1)N 87448,C(N=c1cccc(S(=O)(=O)NC2CC(F)(F)C2)[nH]1)c1ccc(C(C)OC)o1 87449,N1(CCn2c(C)ncc2)CCC2(CC1)CC2(C)C(=O)NCCNC1CCCC1 87450,Cc1cc(Cl)c(C(N2CCC(O)(C(C)NC(c3cccc(F)n3)=O)C2)=O)cc1C 87451,c1(OC)cc(C(N2CC(CCCCNC(=O)CCF)C2)=O)ccc1O 87452,c1(C(N2CCC(F)(C(=O)NCCC34CC(CO3)C4)C2)=O)ccc(Br)cc1 87453,C1(c2cn(C3C(F)(F)C3c3ccccc3)nn2)CC2(C1)CC21CCC1 87454,CC1(C)CC(CO)CN(C(CCC2CC2)C(=O)NCc2ccccc2Br)C1 87455,N1(CC#C)CCN(C(C2CSCN2C(=O)CCc2cnoc2)=O)CC1=O 87456,c1(C(N(CCOCCCN(C(CN2CC(C)(OC)C2)=O)C)C)=O)cc(Cl)ccn1 87457,C(=O)(C#CC(C)(C)CNC(=O)C(O)c1ccsc1)NC(c1ccc(C)cc1)C 87458,N1(C(C(C)OCC#C)=O)CCN(C(c2cnn(CC)c2C)=O)C2CS(=O)(=O)CC12 87459,C1(NCC2(C)CC2)CN(C(=O)CC2(c3cccnc3)CC2)C2(CCCOC2)C1 87460,C(=O)(CCCCC(N)=O)NC1(C)CCN(C(=O)C=Cc2ccccc2)C1 87461,C1(NC(C(CSC)OC)=O)CCC2(CC1)CN(C(=O)C1=COCC1)C2 87462,N(C)(C1CCc2cc(F)ccc21)CC(=O)N(c1ccccc1)CCOCCOC 87463,C(COC)(CC(C)(C)C(=O)OC)NC(C1CCC(CCCC)C1)=O 87464,c1(C(N2CCCC(C)(NC(C(C)=C3CCCC3)=O)C2)=O)ccn2cc(C)nc2c1 87465,C1(F)(C(=O)NC(CNC(C(CC)CC2CCCCC2)=O)CO)CCC(F)(F)CC1 87466,c1(N2CCCN(CCC)CC2)nc(=NCc2cnn[nH]2)[nH]c2cc(C)ccc12 87467,CCCCC(O)CC(=O)NCC(C1CCCC1)NC(c1ncccc1Cl)=O 87468,C1(n2cc(CN(CC(C)(C)OC)C)nn2)CCCCCC1O 87469,N1(C(CC(c2ccccc2)SC)=O)CC2CC1CCC2NC(C1CCCCC1)=O 87470,C(=O)(C1=CCC2CCC1N2C(=O)CC1(N(C)C)CC1)Nc1ccc(OC)c(C)c1 87471,C(c1cn(C)cn1)=C(C(=O)NC1(CC)CN(C(C2C(OCC)CCC2)=O)C1)F 87472,Cc1nc[nH]c1CC(=O)NCC1(CCNC(c2cc(C(F)F)cs2)=O)CC1 87473,c1(C(N2C(C)CN(C(=O)Cc3ccccn3)CC2)=O)cccc2ncsc12 87474,Cn1cc(NC(=O)CC2CCCN2C(C2CC(=O)CC(=O)C2)=O)c(O)nc1=O 87475,c1(N(C2CCCNC2)C(COC)=O)ncc(F)c(OC(C)C)n1 87476,C#Cc1ccc(CC(N2CCC(NC(c3c(C)csc3Cl)=O)C(CC)C2)=O)cc1 87477,c1(C(=O)NC2(CO)CN(C(=O)Cn3ccccc3=O)C2)ccnc(C(F)F)c1F 87478,C1(C(N2CC(NC(C(C(C)C)NC(N)=O)=O)C(F)C2)=O)CCCCCCC1 87479,N1(C(c2cc(C)ncn2)=O)CCN(C)CC1CNC(c1ccoc1C1CC1)=O 87480,c1(CCC(=O)NCCCCNC(CC2C(CC)C2)=O)cccc(O)n1 87481,Cc1cnc(NC2(C)CC2)c(S(=O)(=O)NCCC(C)c2cn[nH]c2)c1 87482,N1(C(C2C(C)CCC2)=O)CCC2(CCOCC2C(=O)Nc2cc(Cl)ccn2)CC1 87483,C1(C(NC)=O)CCN(C(=O)C(C)(C)C)CC1.C(CCC(=O)NC1CC1)CCN(C)CS 87484,c1(CCC)cc(=NC(CNC(c2coc(CCOCC)n2)=O)C2CC2)[nH]c(Cl)n1 87485,c1(CC(N2CC(C)C(NC(c3nccnc3Cl)=O)C2)=O)ccc2c(c1)CCC2 87486,C=Cc1cncc(C(N2CC(O)(C(F)C(=O)NC(c3cnn(C)c3)CC)C2)=O)c1 87487,N1(C(CC(CC)C)=O)CCC(O)C(NC(=O)CCCSC)C1 87488,C(=O)(CC(C)(C)N(C)C(C1CCOC1(C)C)=O)N(C)CC1CCOC1 87489,CC(CN1CCCC1=O)N=c1cccc(S(=O)(=O)NCCN2CCNC2=O)[nH]1 87490,C(=O)(CC1=CCN(C(C2(C)CCC(C)C2)=O)CC1)NCC(C)C 87491,c1(OC)cc(C(=O)NC2CCC(NC(C3CC(CF)C3)=O)C2)ccc1C 87492,Cc1sc(C(N2CCCC2CCNC(=O)C2=NOCC2)=O)cc1Br 87493,N1(C(C(C(=O)OC)(C)F)=O)CCC(C)N(C(c2cnn(CC3CC3)c2)=O)CC1 87494,c1(OC)ccc2nc(S(C)=O)[nH]c(=NCc3cnn[nH]3)c2c1 87495,c1(CC(=O)NCCN2CCN(C(c3c(C)onc3)=O)CC2)ccc(Cl)cc1Cl 87496,C(=O)(C(C)(C)CS(N)(=O)=O)N1CC(NC(C(C2CC2)OC)=O)C(C(F)F)C1 87497,Cn1cncc1C=CC(N1CCC(CCNC(C2C3CCCOC23)=O)C1)=O 87498,Cc1ccc(NC(C2CC(C)N(C(c3cnn4c3CCC4)=O)C2)=O)cc1C 87499,C#Cc1cnn(C)c1C(=O)NCC1COCCN1C(C1C2CCC1CC2)=O 87500,C1(NC(c2cc(Cl)ccc2F)=O)CN(C(=O)CCCC(F)F)CC1C1CC1 87501,c1(C(=O)NC(C(C)NC(C(CC)CCOC)=O)CO)cnn2cccc(OC)c12 87502,CN1CCc2ccc(C(=O)NC3CC3CNC(=O)C3=NNC(=O)CC3)cc21 87503,CCC(C)C(C(=O)NCC1CN(C(C23CC(C)(C2)C3)=O)CC1(C)C)OC 87504,C(=O)(C(C)CC(F)(F)F)N1CCC(NC(c2c(C)cc(N(C)C)cc2)=O)(CF)C1 87505,C(=O)(CCS(C)(=O)=O)NC1(C(=O)NC(CC)CN2CCCC2)CCSC1 87506,c1(C(=O)NC2CC(NC(=O)C=Cc3cc[nH]n3)C2)ccc(C2CC2)nc1 87507,N1(C(c2c(C)n(C)cc2)=O)CCC(NC(=O)C(O)C(F)F)C2(CCC2)C1 87508,c1(OC)ccc2nc(N3CC=CCC(C)(C)C3)[nH]c(=NCCOCCF)c2c1 87509,N1(C(c2c(C)n(-c3ccccc3Cl)nn2)=O)CCC(CNC(=O)C2CC2)C12CC2 87510,c1(CC(=O)NC2CC2NC(c2csc(-c3ccccn3)n2)=O)ccc(O)cn1 87511,c1(C(=O)OCC)ccn(CC(=O)NCCC2CC(NC(=O)CC3CCOC3)C2)n1 87512,O=C(C1=CS(=O)CCC1)NCCN(CCOCCO)C(C1(OC)CCC1)=O 87513,O=[N+]([O-])c1cncc(-c2ccn3ccnc3c2)c1 87514,c1(SC)ccccc1C(=O)NCC(C)CNC(=O)CC=C(C)C.c1(C)cccc(Cl)c1 87515,Cc1cc(O)nc(CNC(C2(F)CN(C(c3cccc(CO)c3)=O)C2)=O)n1 87516,N1(CCC(=O)NCC2CC(O)CN2C(=O)COC2CCCCC2)CCOCC1=O 87517,C(N=c1ccnc(C)[nH]1)C1CCCC(NC(C(c2cc(C)c(F)cc2)(C)C)=O)C1 87518,c1(C(=O)NC2C3(CN(C(C4(CC)COC4)=O)C3)CC2)coc(S(=O)(=O)NC)c1 87519,N1(C(C(c2ccc(OC)nc2)(F)F)=O)CCC2(NC(=O)CC(C)(C)O)CCCC12 87520,N1(C(c2cc(C)c(C)s2)=O)CC2(CC(NC(=O)CS(=O)(=O)N(C)C)C2)C1 87521,N1(C(C(C)=C2CC2)=O)CC(NC(c2cc(Cl)ccc2F)=O)CC12CCCCCC2 87522,C1(CC(=O)NCC2CCC(CC)O2)CN(C(=O)COc2cccnc2)CCO1 87523,c1(OC(COC)C)ccc(Oc2ccc(F)cc2)cc1.C1CC(=O)N1 87524,OC1CC(CNC2CC2c2cccnc2)CC1OCc1ccccc1 87525,CCC(CNC(=O)C(C(=O)OC)OC)(CC)C(=O)Nc1ccc(O)cc1Cl 87526,C(=O)(C#CC1(C(F)(F)F)CC1)NC1C(CNC(CCCN(C)C)=O)CCC1 87527,N1(C(c2c(CC)ncs2)=O)CCCC2(C1)CN(C(c1cccc(C)c1Cl)=O)C2 87528,CC1CN(C(=O)CS(=O)(=O)N(C)C)C(C)CN1C(c1cnn(CCN(C)C)c1)=O 87529,CN1CCN(C(C2CC(C3CC3)=NO2)=O)C(C(=O)NC2(CCF)CCC2)C1 87530,CCCCN=C(NCCc1ccc(Cl)c(Br)c1)NCCc1cccs1 87531,C1(C)(CC=C)CN(C(=O)CN(CCC)C(c2ccc(Cl)o2)=O)C1 87532,c1(C(N(C2CCCCN(C(C3(C)CC=CC3)=O)C2)C)=O)cc(Br)cnc1O 87533,N1(C(c2c(COC)cco2)=O)CCCCC1CNC(=O)C(COC)OC 87534,c1(NC(CS(N2C3CN(C(C)=O)C(C3)C2)(=O)=O)=O)cc(CO)c2ccccc2c1 87535,C1(C)(CNC(C2(COC)CC(=C)C2)=O)CCN(C(C2CNC(=O)CC2C)=O)CC1 87536,N1(C(C2CCC(C)CC2)=O)CC2N(C(=O)C(C)S(N)(=O)=O)CCC2(C)C1 87537,C1(C(N2C(CC(=O)NCC(C3CCCCC3)C)CC2)=O)C2CCCOC12 87538,c12sc3ccccc3c1CS2.c1(CC#N)cc(C(F)(F)F)cc(C(F)(F)F)c1 87539,c1(C(=O)NC2C(NC(C(C)(C)C3CCCO3)=O)COC2)cc[nH]c2nccc1-2 87540,C(=O)(C#CC1CCCOC1)NCC1(C)CCN(C(c2c(N)ccc(CC)c2)=O)C1 87541,C12(C(N3CCC(NC(C=C(C)Cl)=O)C3)=O)CCOCC1C2 87542,C(C1CN(C(=O)C(O)CC2CCCC2)CC1C(=O)NCC(C)C(C)C)=CC 87543,Cc1cccc2[nH]cc(C(N3CC(NCc4ccsc4Br)C(C)C3)=O)c12 87544,c1(C(=O)NC(CCN(C(Cc2cc(OC)ncc2)=O)C)C)c(OC)ccnc1F 87545,N1(C(C(N2CCSCC2)C)=O)CC(NC(c2ccc(F)s2)=O)CCC1C 87546,C1(CC(=O)NC2CS(=O)(=O)C2)(OC)CN(C(C2(C)CC=CC2)=O)C1 87547,N1(C(CCNC(c2nccn2C)C(C)C)=O)CC2CC1C2C(=O)OC 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87566,N1(C(C(SC)SC)=O)CCCC1C(C)NC(=O)CC1CCC1 87567,Cc1cc(C(=O)NCC2COC(CNC(c3cc(C(N)=O)cs3)=O)C2)nn1C(F)F 87568,N1(C(c2cncc(N(C)C)c2)=O)CCOCC(NC(C2CC=CCC2)=O)C1 87569,N1(C(CC2(OC)CCCC2)=O)CCN(C(=O)CCN2CCC(O)CC2)C(CF)C1 87570,N1(C(C(C)=C2CCCC2)=O)CCN(C(c2cc(-c3ccccc3)no2)=O)C(C)C1 87571,Cc1nc(NCC(=O)N=c2cc[nH]cc2)cc(=NCC2CCCC(CO)O2)[nH]1 87572,N1(C(c2oc(C)c(Br)c2)=O)CC(C)CN(C(=O)C(F)=C2CCC2)C(C)C1 87573,N1(C(C2(C#C)CCC2)=O)CC2COCC(C1)C2NC(C12CCCN(CC1)C2)=O 87574,C(CCCCC(=O)NC1C=CCN(C(c2cc(Cl)c(Cl)n2C)=O)C1)OCC 87575,c1(C(N2CCCC(CC(=O)NCc3ncccc3O)C2)=O)cccc2nccn12 87576,C(C(C)(C)CC1CC1)NC(c1nnnn1C1CC(F)(F)C1)(c1nccn1C)CC 87577,c1(C(=O)NC(CC2CC2)C(=O)NCC(F)Br)coc2ccccc12 87578,c1(C(=O)NCCC2CCCCN2C(=O)CC2CCOC2=O)cncc2nc[nH]c12 87579,CCCCCCN(CCC(=O)NCC1CCN1C(c1cnc(NCC)s1)=O)CC 87580,N1(C(CN2C(C)COCC2)=O)CC2CC(C(=O)NCc3ncc(F)cc3F)(C2)C1 87581,Cc1cc(OCC(=O)NC(CNC(=O)CC(C)(C)C#N)CO)cc(C)c1 87582,N1(C(CCC=CCC=C)=O)CC=CC(C(=O)NCc2ccccc2C)C1 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87654,C1(CC(C)NC(CCN(C(C)=O)C)=O)CN(C(=O)C(C)(C)COC(C)C)CCCO1 87655,N1(C(CCC=C=C)=O)CC(C(=O)NCC2(C(O)C(C)C)CC2)CC1(C)C 87656,c1(OC)ccccc1C=CC(=O)NCC(C)(CO)NC(c1cc(F)ccc1C)=O 87657,C1(C(N(CC(C)NC(CSc2n(C(C)C)cnn2)=O)C)=O)CCC(C)=C(C)C1 87658,c1(CC(=O)NCC2CC(F)(CNC(CCCC#N)=O)C2)ccc2ccoc2c1 87659,c1(OC)nc(NC(c2n[nH]cc2NC(c2scc(C)c2Cl)=O)=O)cnc1C#N 87660,c1(C(c2c(CNC(C)CCC3CC3)cccc2)=O)ccc2c(c1)OCCO2 87661,N1(C(C2(C)CCCCO2)=O)CC2CC(NC(=O)C(O)C3CC3)CC2C1 87662,C1(CN(C)C2CC2)CCN(C(=O)CCOC2CN(C(=O)CC3CC=CC3)C2)C1 87663,N1(C(CCC(C)(C)OC)=O)CC2(CCCN(C(c3cccc(C)c3C)=O)C2)C1 87664,C1(C(N2CCC(NC(=O)CSCCc3ccccc3)C2)=O)CCn2nccc2C1 87665,c1(N2CCC(OC)(CO)CC2)nc(NCC2(CF)CCC2)c2cnn(C)c2n1 87666,C1(N(C(CC(C=C)c2ccccc2)=O)C)CCCN(C(=O)C=CC=CC)CC1 87667,c1(OCCC)ccc2c(c1)OCC(C(=O)NCc1nc(OC)cc(Cl)n1)=C2 87668,CC1CC(C(=O)NCc2nocc2C(=O)NCC2CC(C)(C)C2)CCO1 87669,N1(c2nccc(C(=O)OC)n2)CC2(CCCC2NC(=O)CCC(C)C)C1 87670,Cc1cc2ccc(C(=O)NC3CCCCC3NC(C3CC3Br)=O)cn2c1 87671,Cc1cnc(NC2CC(NC(=O)Cn3nc(O)ccc3=O)C2(C)C)nc1O 87672,c1(C(N2CCC(O)(C(C)CNC(=O)CCNC(N)=O)C2)=O)ccc2nn[nH]c2n1 87673,C1(C(=O)NC2CCN(S(C)(=O)=O)C2)CN(C(C2(C)CCCCC2)=O)CCN1 87674,C1(NC(C(C)SCCCC)=O)CC(O)(CN(C(=O)CCc2csnn2)CC)C1 87675,N1(C(C(=O)NCc2nnn(C)n2)CCC2CCCOC2)CCC(S(=O)(=O)C(F)F)C1 87676,c1(C(=O)NC2CC(CCNC(C(C3CCCCC3)OC)=O)C2)c(F)cccc1F 87677,c1(OC)cc(CN2CC(NC(c3ccoc3)=O)CC(F)(F)C2)cc(I)c1O 87678,C12(CN(C)C(c3coc(CNC(=O)Cc4cncs4)c3)=O)CCC(CC1)C2 87679,Cc1cccc(CCCNC(c2ccnn2C2CC2(F)F)c2nnnn2C)c1 87680,CCC(CC(=O)N1CCN(C(=O)CCc2ccc(C)cc2)CC1COC)C(F)F 87681,c1(OC)cccc2c(CC(=O)NCCCN3CC(C)CC(C)C3)c[nH]c12 87682,Cc1cccc(N)c1C(=O)NC1CCN(C(=O)CC(C)(C)F)CC1C 87683,c1(CCC)onc(C)c1C(N1CC2CC2(C(=O)NCc2cccc(Br)n2)C1)=O 87684,c1(C(N2CCCC(OC(C)(C)C)C2)C(=O)NC(CC)(C)C)ccc2c[nH]nc2c1 87685,c1(C(N(CC(C)NC(c2cnc(C(C)O)s2)=O)C)=O)cnn(C)c1C1CC1 87686,C1(C(N(C2CCC2O)C)=O)CC(O)C(O)CC1CNC(=O)CC1(N(C)C)CC1 87687,C1(N(C(CC)C(N)=O)C(C2CCn3ccnc3C2)=O)CCCC12CCNCC2 87688,Cc1cc(N)c(C(=O)NC(C2CN(C(c3cccc(F)n3)=O)CCO2)C)cc1F 87689,c1(C(=O)NC2CCCC(NC(=O)C3=CCC3)C2)ccc2c(c1O)CCCC2 87690,C1(NC(C(CC#C)C)=O)CC2(C1)CN(C(c1ccnc(OCCO)c1)=O)C2 87691,c1(C(N2CCCC(C(=O)NCC#CCC)C2)C)cc2ccccc2o1 87692,c1(NCC(N2C(CN(C)NC(C(CC)OC)=O)CCC2)=O)ccc(C)cc1 87693,c1(OC(CC)C)cc(N2CCC(C3CC(N)CCO3)CC2)nc(C)n1 87694,C1(NC(C(=O)Nc2ccc(C3CCCNC3)cc2)=O)CCNCC12CC2 87695,CC(CCC(=O)NCC#CCNC(=O)C(O)C1CC1)NC(=O)OC(C)(C)C 87696,C(C1c2ccccc2CN1C(C1C2CCCOC12)=O)NCCn1cc(CN)nn1 87697,c1(C(N2C(C)CN(C(C3CCC(=O)N3)=O)CC2)=O)ccnc(P(C)(C)=O)c1 87698,C1(CC(=O)NCCC(=O)N(CCn2c(C)ncc2)C)CCCCN1C 87699,c1(C(=O)NCC2C(C(=O)NCC(=O)N(C)CC)CCC2)ccccc1C1CC1 87700,C1(C(N2CCCC(NC(c3cnc(CC)[nH]3)=O)C2C)=O)CC2CCCCCCC12 87701,c1(CN)ccc(CCC(=O)O)cc1.C12(CCOC1)CC(=O)N2CCC(=O)OC 87702,c1(CCNC(=O)CCOc2ccc3n[nH]cc3c2)cccc2c1OCCO2 87703,C1(C(=O)NC(C2CC2C(=O)NOCC2(C)CC2)C)C=CCOC1 87704,N1(C(C2CCC(=O)N2)=O)CC2(CCCC2NC(c2ccc3ncsc3c2)=O)C1 87705,c1(OC)cccc(C(F)F)c1C(=O)N(CC(O)CN(C)C(C12CC(C)(C1)C2)=O)C 87706,C1(CC(=O)NC2(CF)CCN(C(c3cc[nH]c3)=O)C2)CC2C=CC1CC2 87707,N1(C(CNC(CC)=O)=O)CCC(C(C)NC(c2sc(C)nc2CC(C)C)=O)CC1 87708,C(=O)(C1=NOC2COCC12)N(CCNC(C(C)SC)=O)CC1CC1 87709,C=CCCCCC(=O)NC1COCC1CNC(=O)CCc1c[nH]c(=N)[nH]1 87710,N1(C(c2occ(C)c2)=O)CC2OCCN(C(=O)CC3C=CCCC3)C2C1 87711,C(C1=CCCOC1)NC(C#CCNC(C1C(C)C1)=O)=O 87712,Cc1cc(C(=O)NCc2cc[nH]c2C(=O)NCC(F)C2CCC2)[nH]c1C 87713,c1(NC(C(=O)N(C2CC3CCC2C3)C)=O)cncc(SC(C)(C)C)c1 87714,N1(C(C(C(C)C)O)=O)CC2CN(C(=O)CNC(=O)CC3CCCCC3)CC2C1 87715,c1(C(C)(F)F)ccccc1C(N1CC(CNC(=O)CCC2CC3CCC2C3)C1)=O 87716,C1(NC(=O)Cc2cscn2)CC2(C1)CN(C(c1ncoc1C1CC1)=O)C2 87717,Nc1ccc(C(=O)NCC2CCCC2NC(C2COCCN2C)=O)nc1 87718,C1(C(NC(CC2(C(=O)OCC)CCC2)=O)(C)OC)CN(C)CCN1C(c1csc(Cl)c1)=O 87719,N1(C(COCCC#C)=O)CC(CNC(C2CCCCN2C)=O)C(O)C1 87720,c1(CCC(=O)NC2CCN(C(CCC(=C)C)=O)C2)cn2ccccc2n1 87721,c1(OC)cc(OC)[nH]c(=NC2CCC(C)N(C(c3ccc4cnsc4c3)=O)C2)n1 87722,c1(CNC(NC(CC)C)=NCC2CN(C)CCO2)ccc2c(c1)CCCC2 87723,c1(C(N2C(CNC(Cn3c(C)cnc3)=O)C(C)CC2)=O)cccc(O)c1F 87724,C=Cn1nccc1C(=O)NCC(C)CN(C)C(C1CCN(C2CC2)C1=O)=O 87725,CCCCCCCCC(=O)N1CC(CNC(=O)CSCC2CCCO2)C2(CC2)C1 87726,c1(OC)ncc(S(=O)(=O)NCCC2(CN)CC2)cc1C 87727,c1(NC(c2cc(Br)cnc2OC)c2n(C(CC)C)nnn2)cccc2c1OCC2 87728,C1(CC)CN(C(=O)CCOCC(F)(F)F)CCN1C(c1ccnc(C)c1N)=O 87729,N1(C(C(C)=CC)=O)CCC(CNC(c2ccc(Cl)c(COC)c2)=O)C12CC2 87730,Cc1csc2ncnc(N3CCCC(C(=O)NCC(C)O)C3)c12 87731,c1(CC(=O)NC(C)CCNC(c2csc(-c3cnc[nH]3)n2)=O)c[nH]c(=N)nc1O 87732,C12(CNC(C=Cc3ccc(C)o3)=O)CCCC1N(C(c1nc(Cl)sc1C)=O)CC2 87733,C(CC(F)F)(C(=O)NC(C)CSC)NC(COCCOC)=O 87734,C=CCC(C(=O)NCC(F)C1CCC1)NC(=O)CCCN(C)C 87735,Cc1nc(NCc2nnc(-c3ccoc3)s2)cc(=NCc2ccc(F)cc2Br)[nH]1 87736,C1(NC(C(CC(=O)OC)NC(=O)OCC2CCCO2)=O)CCCCC1C(F)(F)F 87737,c1(COC)nc(N2CC(CNC(C3CN4CCN3CC4)=O)CC2C)cc(C)n1 87738,c1(NC(C)=O)ccc(C(N2CCCC(NC(C3CCCS3)=O)C2)=O)c(Cl)c1 87739,c1(C(N(CC(C)NC(=O)CC2(CO)CCCC2)CC)=O)coc2c1COC2 87740,N1(C(C2CC(C)(C)C2)=O)CC2CC1(C(=O)NCC1CC3CCC1C3)C2 87741,c1(C(CO)NC(c2cnn(CCC)c2Cl)=O)cc(F)cc(Cl)c1 87742,c1(OCCCC(=O)Nc2cccc(CNC(CSC)=O)c2)ccc(C#N)cc1 87743,c1(CC)nn(C)c(CC)c1CC(N1CC(C)C(NC(C2CCC(=O)N2C)=O)C1)=O 87744,N1(CCC)C(=O)NC2(CCN(CC(C3CCOC3C)=O)CC2)C1=O.CCCl 87745,C(c1c(C)nn(C)c1Cl)=CC(=O)NC(CC)(C)CNC(C1CN2CCC1CC2)=O 87746,C1(C(N(CCC)CCNC(C2CC=CCC2)=O)=O)CCN(C(=O)OCC)CC1 87747,N1(C(C2N(C(CCC(C)NC(C)=O)=O)CCC2CO)=O)CCC2(CC1)CN(C)C2 87748,c1(C(=O)NC(C(C)C)C(C)NC(=O)Cc2cncs2)cccc2c1OCC2(C)C 87749,CC1CCN(C(C(=O)Nc2ccc(Cl)cc2F)c2ccco2)CCS1 87750,FC1(F)CCCC(Cc2nc(-c3ncccc3Br)no2)CC1 87751,C(=O)(C1CCCc2ccccc21)NC(CN=c1[nH]nc(C(=O)OC)s1)C 87752,CCC(C)C(O)CC(=O)N1CCC(CC(=O)NCC=C(Cl)Cl)CC1 87753,C(CO)(CCCNC(c1ccc(=N)[nH]c1)=O)NC(c1c(CC)cco1)=O 87754,c1(OC)ccccc1OCC(N1CCC(NC(C2C3CCCC23)=O)C1)=O 87755,C1(NC(CCc2cnc(C)o2)=O)CCCC(C(=O)N(CC(C)O)CC(C)O)CC1 87756,Cc1cnn(C)c1CC(=O)NCC1(CNC(C2CC2C)=O)CCCC1 87757,CCC(C)(C(=O)O)n1nnc(CCCCCO)n1.n12cc(nn1)CN1CC2C1 87758,c1(C(=O)NC2CCCC(NC(C3C(C(=O)NCC#C)C3)=O)C2)csc2nccn12 87759,C(CNC(=O)C(C)Oc1ccc(F)cc1)(CC(C)C)NC(c1c(CC)ocn1)=O 87760,c1(NC(C2(CC)CN(C(=O)Cc3ccoc3C)C2)=O)cnccc1CO 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87779,C1(C(=O)NCC(O)CO)(OC)CCN(Cc2ccc(F)cc2)CC1 87780,C1(CCC)CN(C(C2CCCSC2)=O)CCN1C(=O)CC1CCC1 87781,c1(C(N2C(CCNC(c3c(CC)nn(C)c3)=O)COCC2)=O)ccc(F)cc1Cl 87782,C1(NC(c2c(CC)cccc2)=O)CC2CC1N(C(c1cn(C)nc1Br)=O)C2 87783,C(=O)(C(CCC1CCC1)NC(=O)CC1CCC(=O)NC1)NCc1ccn(C)n1 87784,c1(C(=O)NC2CN(C(=O)COc3ccc(F)cn3)C2)cccc2ncc(Br)n12 87785,C1(C2(O)CN(C(=O)C3=C(Cl)CCOC3)C2)(CNC(CCC(CC)OC)=O)CC1 87786,N1(C(CS(CC)(=O)=O)=O)CCCN(C(C2CC(F)C2)=O)C(CO)C1 87787,C(=O)(C1OCCn2ccnc21)NC1C(CNC(c2c(C)cccc2Cl)=O)CC1 87788,c1(C(C(=O)NCCc2cccc(C#C)c2)C)ccc2c(c1)OCO2 87789,N1(C(=O)NCC=C(CCC)C)CCC(C)(C(=O)OC)CC1.C(C)(=O)O 87790,N1(C(CC(C(=O)OC)C)=O)CCC(C)(C)CC1C(=O)NCC(CO)OC 87791,c12ccc(Br)cc1O2.c1(C(=O)NCc2ccc(OC)cc2)cc(C)cc(C)c1 87792,C12COCCN(C1)C(=O)C2.C(C(=O)NCCSCCOC)=CCC 87793,c1(SC)cccc(C(N2CCC(CCNC(=O)C(C)CF)C2)=O)n1 87794,c1(-c2nc(CCNC(=O)NCC3(CO)CCOCC3)sc2)cccc(F)c1 87795,Cn1cc(N(C2CC2)Cc2nc[nH]n2)cc(Br)c1=O 87796,C(C)(C)(CC(F)C(=O)NC1(C)CC2CCC1C2)NC(C(CCCC)O)=O 87797,CC1(C)CCCCN(C(C2N(C(C3OCCC3(C)C)=O)CC23CCCC3)=O)C1 87798,C1(C(=O)NC2(C)CN(C(=O)CC3(O)CCOC3)C2)Cc2c(F)cccc2O1 87799,N1(C(c2c(C)c[nH]c2)=O)CCN(C(=O)CCc2cncnc2)CC(C)C1 87800,C1(CC(=O)NC2(C(=O)NCCC3CCCC3)CCC2)CCCOC1c1cn[nH]c1 87801,C=CC1(O)CCN(C(=O)CC(C(C)OC)NC(c2cncnc2CC)=O)C1 87802,C(=O)(C(C1=CCSC1)N(CCS(=O)(=O)C(C)C)C)NCCSC 87803,CCCCCCCCCCCC(=O)N1CCCC1CN(C)Cc1nnc(CC)o1 87804,C(C(C)(C)CC(=O)OC(=O)C(C)(C)C)NC1C(C(=O)NC)C1 87805,c1(OC)cccc(C(=O)N(C2CCCN(C(=O)Cc3cnc(C)o3)C2)CCF)n1 87806,C(C(CC(=O)NC1C=CCS1)NC(=O)C(C)NC(N)=O)OC 87807,c1(N(C)C)cncc(C(N2CCN(c3cc(N)ncn3)CC2)=O)n1 87808,c1(CCCC)ccc(CC(=O)N(C2CCC(SC)C2)C)cc1 87809,C1(C(=O)NCc2ccc(OC)cc2)CC12CCN(c1nc(Cl)ncc1Cl)CC2 87810,CC(C(=O)Nc1cnc(F)nc1)C(C)NC(c1ncc(F)cn1)=O 87811,CCCC(C)(C)C(=O)NCC(CNC(c1cnn(C)c(=O)c1)=O)OC 87812,CC1C(CO)SCCN1C(=O)C(=O)N(C1CCN(c2ccncc2)CC1)C 87813,N1(C(C(c2ccc(C)cc2)F)=O)CCC2C(CCCN2C(C2CCS2(=O)=O)=O)C1 87814,N1(C(CCSCCC)=O)CCC2CCN(C(c3nc(C)c(N)cc3C)=O)C2C1 87815,N1(C(C=C(COC)C)=O)CCN(C(=O)CC2CCC(C)C2)CC(O)C1 87816,CC(C)C(CNC(C1(C)CC1(C)C)=O)C(=O)NCc1c(F)cccc1F 87817,c1(C(C)=O)ccc(CC(N2CC=CC(NC(=O)CCN3CCC(F)C3)C2)=O)cc1 87818,c12cccc(c1)NC(=O)CO2.C(=O)(CC(C)n1cccn1)OCC 87819,C1(CNC(C2N(CC)C(=O)CC2)=O)CC(C)CN(C(=O)OC)C1 87820,C1(C(=O)OCC)CN(C(=O)CC2CCC(O)C2O)CC1(C)C 87821,C(N=c1[nH]c(=NCC(C(C)C)N(C)C)[nH]c2c1CCCCC2)c1snc(C)n1 87822,CC1(CCn2cc(CC(C(=O)OC)NC(=O)CCN=[N+]=[N-])nn2)CC1(F)Cl 87823,c1(C(=O)NC2CCN(C(C3CC4C(C3)C4(F)F)=O)CC2F)occ2c1CCOC2 87824,C(c1cccc(C#N)c1)=CC(=O)NC1C(OC)CN(C(C2CCCO2)=O)C1 87825,N1(C(C(C=C)O)=O)CC2COCC(C1)C2NC(c1cc(C)nc(C)n1)=O 87826,N1(C(C(C)OCC2CC2)=O)CCCC2CN(Cc3ccc(S(C)(=O)=O)o3)CCC12 87827,c1(C(=O)NC2C(NC(C3(C)CC(=C)C3)=O)CCCC2)nc2n(c1Cl)CCCC2 87828,c1(CC2(C(=O)NCC(C)CN(C(=O)CC(C)C3CC3)C)CC2)cccc(F)c1 87829,C1(OCC)CCCC1(c1nnnn1CCCF)NCC(C)(CC)CC 87830,c1(C(C(=O)NC(C)C(=O)NCCCOCC2CCC2)O)cccnc1 87831,CCC(C)(CC)C(c1nnnn1-c1ccccc1C)NCc1ccc(OC)nc1C 87832,N1(C(C(C)OC(C)(C)C)=O)CCC2(CCOCC2)C(NC(=O)C=CCO)C1 87833,C1(CC)CCN(C(=O)C=Cc2ccncn2)C1C(=O)NC1COC(C(F)F)C1 87834,N1(C(C=CCN(C)CC)=O)CCC(CNC(=O)C(C)(C)c2nccs2)C(C)C1 87835,C(CCCCCC(=O)NCC1CCN(C(c2ccc(C(=O)CF)cc2)=O)C1)SC 87836,N1(C(c2cn(C)nc2O)=O)CC(CO)C2(C1)CN(C(=O)C(C)(C)n1cnnn1)C2 87837,Cc1ccc(C=CC(=O)NC(C)CN(C(=O)CC23CCCC2C3)C)cc1 87838,CCS(=O)(=O)CC(=O)N1C2CCC(C2)C1CC(=O)NCc1nn[nH]n1 87839,C(CC(C)(C)C)(C(=O)N1CCC(C)(C(N2CCCCC2)=O)C1)OC 87840,C12(C(N(C)Cc3ccoc3)=O)CCC(CC1NC(=O)CSC(F)F)C2 87841,C(=O)(CCC(C)NC(C1CCC(N(C)C)CC1)=O)NCC(C)O 87842,C(CCCCC(=O)NCC1CCC(C#N)C1)n1cc(C2(CC)CCC2)nn1 87843,N1(C(C2CC(CC)OCC2)=O)CCC2(CC1)CCN(C(C1(Cl)CC1)=O)CC2 87844,N1(C(c2c(NC)nccc2)=O)C2CCC1C(C)C(NC(C1(Cl)CC1)=O)C2 87845,C1(C(=O)Nc2n(C)nc(C)c2Br)CC(N=c2ccnc(S(C)(=O)=O)[nH]2)C1 87846,c1(C(=O)NC2CCC(C)N(C(=O)Cn3ncnn3)C2)ccn2c1CSCC2 87847,C1(NC(C(=Cc2cccnc2)C)=O)CCN(C(=O)CC2(C)CCC2)CCC1CO 87848,c1(OC)ccccc1-c1n[nH]cc1CNCCC(C1CCCC1)C1CCCC1 87849,C(=O)(N=c1ccc(Cl)n[nH]1)C1C(C(=O)OC)C1 87850,c1(C(CNC(C(n2cc(C(C)O)nn2)C)=O)=O)ccccc1[N+](=O)[O-] 87851,C(c1ccccc1)=CCN(C(=O)CN(C1CN(C(=O)CC2(C)CC2)C1)CC=O)C 87852,c1(C(N(CCNC(=O)C(F)OC)CC)=O)n[nH]c(C(C)C)c1[N+](=O)[O-] 87853,C1(NC(c2cc(F)c(F)cc2O)=O)CC2CN(c3ccncn3)CC2C1 87854,N1(c2nnc(C(C)(C)C)s2)Cc2nccn2CC(NC(C2(C)CC2(F)Cl)=O)C1 87855,C=CCC(C)(CC)C(=O)NC1CCCC1CNC(c1cnnn1C)=O 87856,c1(OCC)nc(C)ccc1CNC(C1CCCN1C(=O)CCC(C)C#N)=O 87857,c1(C(N2CCC(N(C(c3cc(C)on3)=O)C)C2)=O)c(-n2nccn2)cccc1F 87858,C1(C(=O)Cl)(C(=O)NCc2ccccc2)CN(C(C2CCCC2)C2CCC2)C1 87859,Cc1nc(C(C)C)ccc1C(=O)NC1CCCC(NC(c2cc(F)n(C)n2)=O)C1 87860,C(=O)(C(C)(C)C(=O)NC1CCCC(C(=O)NC2CCCC2CCO)CC1)OCC 87861,c1(C(C(=O)OC)N(C(=O)COC2CCCOC2)C)ccccc1F 87862,C1(CCC)CN(C(=O)CCNC(=O)COC)CCN1C(C1CCCOCC1)=O 87863,C(=O)(CS(=O)(=O)C1CCCC1)NCC(C(C)(C)C)NC(C1CC2(C1)CC2(F)F)=O 87864,Cc1ccc2snc(C(=O)N(CC(C)NC(C3CC4CCCCN4C3)=O)C)c2c1 87865,C1(C(N2CC(C)(C)C2)=O)COC2(C1)CN(C(=O)CC1CCCOCC1)C2 87866,CC1OCCCC1C(=O)NC1(C(=O)NCC(C)(O)C2(C)CC2)CCCCC1 87867,Cc1ncnc(C)c1CC(=O)Nc1ccc(N2CCN(C)CC2)nc1 87868,CCC(COC)C(=O)N(C(C)(C(=O)NC(C)C(C)(C)CN(C)C)C1CC1)C 87869,C(CN=C(NCC1CC=CCC1)NC(C)CC(F)F)OCC 87870,Cc1cccc([N+](=O)[O-])c1C(N1CC(n2cc(S(N)(=O)=O)cn2)C1)=O 87871,N1(C(CC(C)N(C(C)=O)C)=O)CCCC(CC(N2CCC(CC3CC3)CC2)=O)C1 87872,O(NC(=O)C(F)C(C)CNC(c1c(C)ccnc1O)=O)CCCC#C 87873,CC1(NC(=O)CC2CCSCC2)CCCN(C(c2coc(CC3CC3)n2)=O)C1 87874,C1(O)(CNC(c2cc(OC)no2)=O)CCN(C(=O)C(C)(C)Sc2ccccc2)C1 87875,C1(C(=O)NC(CNC(C2(C(C)(C)O)CCC2)=O)CC)(COCC)CCC1 87876,N1(C(c2c(C)ncnc2)=O)CCC2(CCSCC2)CC1 87877,CC1CN(C(c2csc3nccn23)=O)CCCN1C(c1cc(F)n(C)n1)=O 87878,C1(CC(=O)NCC(C)NC(C(COC)C)=O)(CNC(C)=O)CCCCC1 87879,c1(C(=O)NC2CN(C(=O)C=Cc3ccccc3)CC2O)coc2ccc(F)cc12 87880,C1(C(N(CCNC(=O)Cc2csc(S)n2)Cc2ccccc2)=O)CCCC1(F)F 87881,N1(C(C(CCSC)OC)=O)CC2CC1CN2C(c1ncn(C(C)(C)C)n1)=O 87882,Cc1cc(Cl)ncc1C(N1CCOCC1c1noc(-c2ccccc2)n1)C1CC1 87883,C1(CC)CCC(O)(C(=O)NCCC2(CNC(=O)C=Cc3ccc[nH]3)CC2)C1 87884,C#Cc1cc(F)c(C(=O)NC(CO)C(C)NC(c2cnnn2C2CC2)=O)cc1F 87885,C12(c3cn(C)nc3)CCC(C1)C2C(=O)Nc1nnc(C2(CC3CC3)CCCO2)o1 87886,C(CCC(=O)N1CCCC1C(C)NC(=O)C(C)N1CC(C)C1)OCC 87887,CP(C)(=O)C(O)C(=O)NCCOC1CCN(C(=O)CCC2CCCC(=O)N2)CC1 87888,c1(C(=O)NC(C)CCNC(C2(CCF)CC2)=O)cc([N+](=O)[O-])ccc1OC(F)F 87889,c1(C(C(=O)NC2CN(C(C(C#C)(C)C)=O)CC2CC)(C)C)cc(F)cc(C#N)c1 87890,c1(OCC(=O)NCC(CNC(c2cnsc2)=O)OC)ccc(Cl)c(C)c1 87891,Cc1cc(C(=O)N(C)CC2CCN(C(=O)C=Cc3cn[nH]c3)C2)no1 87892,CC(C(F)F)N(C)N1CCC(C(N2CCOCC2)=O)CC1 87893,c1(C(=O)NCC(CC)NC(CSCC#C)=O)cn(C)nc1OC 87894,Cc1cncc(C)c1C(=O)NC(CCN(C)C(C1CCOCC1)=O)C(C)(C)C 87895,N1(C(c2c(CN=[N+]=[N-])ccs2)=O)CCN(C2CCN(C(C3CCO3)=O)C2)CC1.C1CC1 87896,c1(CNC(C2C(C)N(C(C3(CO)CC(C)(C)C3)=O)CC2)=O)ncc(F)cc1F 87897,Cc1nc(C(N2CC(O)C(O)C2CNC(=O)CCCc2nccs2)=O)cc(O)n1 87898,CC1=C(C(=O)N2CC=CC(NC(C3CCCSC3)=O)C2)CCCO1 87899,c1(N(CCCS(C)(=O)=O)C)nc(-c2ccccc2)nc(=NC2CCOC2C)[nH]1 87900,C1(C(N2CCCC(N(C)C)C2)=O)CCC2(CC2)N1C(C1(N(C)C)CCCCC1)=O 87901,N1(C(Cc2cccc(C#C)c2)=O)CCC2(CCCN(C(=O)CCCOC)C2)C1 87902,N1(C(c2ccc(C)cn2)=O)CC2(CCOCC2)CC1CNC(=O)C(C)C1CC1 87903,C1(C(=O)NCC2N(c3sc(C(=O)OC)c(Cl)n3)CCC2C)Cc2cccnc2C1 87904,C1(N(C(C(C=CC)O)=O)C)CCCC(NC(C2CC(=O)N(CC)C2)=O)C1 87905,c1(C(N(CCC(C)NC(=O)CN2CCOCC2)C)=O)cc2c(F)c(F)ccc2s1 87906,c1(C(C(N2CC(CCNC(CCCN(C)C)=O)C2)=O)O)ccc(Cl)c(F)c1 87907,C1(CNC(CNC(CNC(CC=CC)=O)=O)=O)CCCC(C#C)C1 87908,c1(OCC(=O)N(CCN(C(C2CCC2(C)C)=O)CC)CC)ccc(C#N)cc1 87909,C1(CC(C(=O)NC(CC)C)N(C(C)C)Cc2cc(C)n(C)n2)CCN(C)CC1 87910,c1(Nc2c(C(=O)NCC(C)(C)C)cc(OC)nc2)ncc2[nH]ncc2n1 87911,c1(C(N2CCC(C)(NC(C3CCC4CC4C3)=O)C2)=O)cc2n(n1)CCNC2=O 87912,C(=O)(C(F)CCC(C)C)N(CC(CC)OC)CC.C(CN=[N+]=[N-])S.C1(=O)CN1 87913,C1(c2nn[nH]n2)(C(=O)NC(C(C)C)c2nc[nH]n2)CC12CCCC2 87914,c1(C(=O)NCCOCCNC(c2c(C)nncc2)=O)cccc(CO)c1C 87915,c1(OC)cc(S(=O)(=O)N2CC(O)(CNC(c3cc4cccnc4[nH]3)=O)C2)ccc1Br 87916,n1(CC(=O)NCC(=C2CN(C(C3CCC(=O)O3)=O)C2)F)c(=O)cnc2ccccc12 87917,c1(C(=O)NC(C2CCCC2)CNC(c2n(CC#C)ccc2)=O)ncccc1CO 87918,C=CC1(C(=O)NCC(c2ccc(F)cc2)NC(C2CC2C)=O)CCOCC1 87919,C1(C)(CC(=O)OC)CCN(C(C2(n3cccn3)CCCC2)=O)CC1 87920,CC1CCCC(n2cc(CN(C)C)nn2)C1.OCP(C)(C)=O 87921,c1(CN(C(=O)C(C2CCCO2)NC(=O)CC2(C)CCC2)C)cncnc1 87922,N1(C(CC2C(C)OCC2)=O)CCC2(CC1)CN(C(c1ccc(F)c(C(F)F)n1)=O)C2 87923,N1(C(C2C(=C)C2)=O)CCCCC12CC(NC(=O)CCCSCc1ccccc1)C2 87924,C1(CNC(c2c(C)cc[nH]2)=O)CC2CCC(C1)N2C(c1csnc1C)=O 87925,CCC(CC)C(C)C(=O)NCCC1(OC)CN(C(=O)COCC(C)C)C1 87926,Cn1cnc2nc(N3CCN(CCCO)CC3)nc(NCc3cc(Cl)sc3Cl)c12 87927,CN1CCC(NC(=O)COC2CCCCC2)C1c1cccnc1 87928,N1(C(c2nccc(OC)c2)=O)CCCC(O)(CNC(C2CC3(CCC3)CO2)=O)C1 87929,C12(CNC(C(C3CC(F)(F)C3)NC(=O)OC(C)(C)C)=O)CCC(CC1)CC2 87930,n1(CC)cnc(S(=O)(=O)NC(c2ccc(-c3ccccc3Cl)o2)=O)c1 87931,CC1CC(NCCC(=O)NCC(c2ncccn2)=O)c2nccn21 87932,c1(C(=O)NC(C)CCNC(c2nnn(C(C)(C)C)n2)=O)cc(Cl)ccc1[N+](=O)[O-] 87933,C(=O)(C(CO)C(F)(F)F)NC1C2C(C(=O)NC(C(=O)NC)CC3CC3)C3C(C2)C13 87934,C1(c2c(C)nc(-c3c(OC)cccc3)s2)NC(=O)N(CC(C)C)C2=C1C(=O)OC2 87935,c12cc(Cl)ccc1OC2.C(=O)(C(C)N(CCNC(C)=O)C1CC1)OC 87936,c1(C(N2C3CCC2CC(CC(F)(F)F)C3)=O)ccc(OC(F)(F)F)cc1[N+](=O)[O-] 87937,c1(C(=O)NC(C(=O)NCC=C=C)C2CCCC2)ncoc1CC 87938,c1(NC(=O)NCCOC)cn(CC(=O)N(CCC(C)(C)O)C)nn1 87939,Cc1c(NCC2CCCC(F)(F)C2)ncnc1N1CC(C)SC(C)C1 87940,C1(C(C)C)CCOC1C(=O)NCC1(O)CN(C(=O)C(C)CN2CCCCC2)C1 87941,c1(-c2cn(CCN(C(c3cc(Cl)cnn3)=O)CC)nn2)cc(F)ncc1F 87942,C1(C)(CNC(C(C(C)C)OCC)=O)CCN(C(=O)CCc2ccoc2)CC1 87943,Cc1nc(CC(=O)NCC2C(C)CCN2c2nnc(-c3ccccc3)s2)[nH]c1C 87944,CCCCC(C)CCC(=O)NC1CCCC1(C)CN(C(=O)CNC(C)=O)C 87945,C1(C(N(C)CCNC(=O)Cc2cncnc2)=O)CCNC(=O)C1 87946,N1(C(C(=O)NCC=C)C)CCC(O)(C(=O)NCC(C2CCCCC2)C)CC1 87947,c1(CNC(C(CNC(c2cn(C)nc2C)=O)OC)=O)ccnc(F)c1F 87948,Cc1ccc(Br)c(NC(C2CC(NC(=O)Cn3cc(Cl)cn3)C2)=O)c1 87949,C1(C#N)(CC(C(=O)NC2CC2)N(CC(C)Sc2ccccc2)C)CCOCC1 87950,CON=CC(=O)NCCCCC1CN(C(c2csc(CC(F)(F)F)n2)=O)C1 87951,C1(C(=O)NCC(=O)NC)CSCCN1C(c1cnc(O)[nH]1)=O 87952,n1(CCC)ncc(-c2nc(C3CCCCCC3)nn2C(C)C(C)C)c1C 87953,Cc1[nH]c(C)c(C(=O)N(C)CCOCCN(C)C(C2(C)CCN(C)C2)=O)c1C 87954,C1(CNC(Cc2cc(C)ns2)=O)CCCCN(C(=O)C(N2CCSCC2)C)C1 87955,CC#CCCCC(=O)N1CCCC(CNC(=O)C(C)COC)CC1 87956,CC(C)(C)CCCC(=O)N1CCN(C(=O)Cc2csc3nccn23)C2CC12 87957,N1(C(COCc2cc(C)on2)=O)CC(C)CN(C(c2cnc(C3CC3)s2)=O)CC1C 87958,N1(C(c2cn(CC(C)C)nc2)=O)CCC(C(C)NC(=O)CCF)CC1 87959,C1(F)(C(=O)NC(C2CCOC2)CC)CCN(C(c2ccn(COC)n2)=O)CC1 87960,N1(C(c2cc(Cl)c(C)cc2Br)C(=O)NC)CCC(C2CCC(F)(F)CC2)C1 87961,N1(C(CCCCN(C(C)=O)C)=O)CC2(CCCN(C(=O)C(C)(C)S(C)(=O)=O)C2)C1 87962,C(=O)(C1=C2CCCN=C2NN1)NC1CCCN(C(C2C(C(N)=O)COC2)=O)C1 87963,C1(CC(=O)NCCOCCN(C)C(c2cc(C#N)on2)=O)SC2=NCCN2C1=O 87964,C(=O)(CCCC(F)(F)F)NC(CSCC)C(=O)NCCC1CCN(C)C1 87965,C1(NC(c2ccc(CNC(c3ccc(C#C)o3)=O)s2)=O)CCC(C)(C)CC1 87966,c1(C(C(=O)NCC(CNC(c2c(OC)n(C)nc2)=O)CO)=O)cc(F)ccc1C 87967,C1(NC(c2c(OC)c(F)ccc2)=O)CN(C(=O)C2=C(Cl)CCCC2)CC2(CC2)C1 87968,CN1CC(CN(C(c2ccc(I)cc2)C(=O)NC2(C)CC2)C)C(O)C1 87969,N1(C(c2nnn(CC)c2C)=O)CC(C)N(C(c2cccc(COC)c2)=O)CC1C 87970,C(=O)(C(C)(C)C(F)F)NCC12OCC(CNC(c3nn(CC)c(O)c3)=O)(C1)C2 87971,O=C(C1=CCCC1)NCC1CCCC(NC(C2(c3ccno3)CC2)=O)C1 87972,C1(CNC(c2n(C(C)C)nnc2)=O)CN(C(=O)CNc2ccccn2)CC12CC2 87973,N1(C(c2n(CC(C)C)ncc2)=O)CC2CN(C(=O)Cc3cnc[nH]3)CCC12 87974,c1(OC)c(C(N2C3CCC2CC(NC(c2ccnn2C)=O)C3)=O)ccc(Cl)c1C 87975,C1(C(=O)NC2C(CC(=O)NC(C#C)CCC)C(O)C2)NC(=O)OC1C 87976,C1(CC(=O)NCC#C)CCN(C(C(CC)CC)=O)CC1 87977,c1(C(=O)NC2CC(NC(CNC(C)=O)=O)CC2O)ccc([N+](=O)[O-])[nH]1 87978,Cc1nc2ccc(C(=O)NC3CCCN(C(C4(C)COC(=O)OC4)=O)C3)cc2o1 87979,C12(C(=O)NC3C(CN(C)C(c4ccc(C(N)=O)nc4)=O)CCC3)CCC(CC1)C2 87980,C(=O)(C(C)(C)CCS(C)(=O)=O)NC(Cc1ccc(OC)cc1)(C)C 87981,N1(C(CSCCC)=O)CC2CC(C1)C(CO)C2NC(=O)C(CC)N(C)C 87982,CC1(C)CCCCC(C(N2CCC(O)(CNC(c3nccc(N)c3Cl)=O)C2)=O)C1 87983,CC1CN(C(=O)C(=C2CCCCC2)F)CC1CC(=O)NC1CC2CCCC12 87984,C1(C(=O)NCc2c(CNC(c3c(OC)n(C)nc3)=O)nco2)CCC(C2CC2)C1 87985,C12(C(N(C(C=C)C)C)=O)CC1CN(C(=O)C=Cc1ccoc1)C2 87986,N1(C(c2ccc(C)cn2)=O)CC2CCCC(NC(c3csc4cncn34)=O)C2C1 87987,C1(CC)CCCC1(C)C(=O)NCC1CCN(C(=O)Cc2cccc(OCC)c2)C1 87988,C1(C[Si](C)(C)C)CCCN(C(=O)NCC(c2ccccc2)CO)C1 87989,c1(C(C)N(C2CCN(C)C2)C(=O)OCC)ccc(F)nc1 87990,Cc1ncc(C(N2CCC(C)C(CNC(c3ccc(O)cc3O)=O)C2)=O)c(C)n1 87991,c1(C(N(CCNC(c2cc(S(=O)(=O)NC)oc2)=O)C)=O)ccc2sc(C)nc2c1 87992,n1(CCC(N2CC3(C(NC(C(C)SC)=O)CC3)C2)=O)ncc(=O)c2ccccc12 87993,Cc1ncnc(C)c1OCC(N1CCN(C(=O)C=C2CC2)C(CC(F)F)C1)=O 87994,c1(CC)cnc(C(N2CCC(NC(=O)C(C)n3ccnc3)C2C)=O)cn1 87995,C=CCC(C(=O)NCc1nccn1C)NC(C1CCCC1CCC)=O 87996,c1(CC(=O)OC)cccc(C(=O)NCC2C3CN(C(C)C=C(C)C)CC23)c1 87997,c1(C(=O)NCC(CNC(c2c(C)onc2)=O)(C)C)nn2c(c1Br)CCC2 87998,CCCC(CC(=O)Nc1cscc1C)NC(C1CCCN(C)C1)=O 87999,c1(C(=O)NCC2(NC(CCCCSC)=O)CC2)cc(N2CCOCC2)nc(Cl)c1 88000,C1(NC(CSCC)=O)CCCC(N(C(=O)CC2CN(C)C2)C)C1 88001,N#Cc1cnn(CC(N2CC3C(CNC(C4CC5CCC4O5)=O)C3C2)=O)c1N 88002,c1(C(=O)NCCCCC(C)NC(CSCCCC)=O)cccc2c1OCCN2C 88003,Cc1ncnc(C(N2CCSCC2C(=O)N(CCCCC(C)C)C)=O)c1C 88004,Cc1cc(-c2ccsc2)ncc1C(=O)NC1CCC(NC(c2cscn2)=O)CC1 88005,N1(C(CC2CC(NC(CC3N(C)CC=CC3)=O)C(O)C2)=O)CC(=O)NCC12CC2 88006,N1(C(c2n(C)cnc2)=O)CC2C(NC(=O)C(c3cccc(Br)c3)O)C2C1 88007,c1(OC)ccc2c(c1)CCC2C(=O)NCC(C)N(C)C(C1(CF)CC1)=O 88008,C1(NC(C2(C)CC(=C)C2)=O)CCCN(C(c2ccc(C#N)c(Cl)c2)=O)CC1F 88009,Cc1cc(C(N2CCCC2(C)CNC(=O)C(F)(F)CC2CC2)=O)ncn1 88010,c1(CC(C)NCc2cccc(P(C)(C)=O)c2)ccc2c(c1)CC(C)O2 88011,C1(NC(c2ncc(C)nc2)=O)CC2CC1CC2C(=O)N(C1CC1C)C 88012,Cc1nc(C)n(CCC(=O)NC(CO)C(C)NC(C2CCN(C3CC3)C2=O)=O)n1 88013,C1(C(C)C)N(C(c2cnc3c[nH]nc3c2)=O)CC12CCN(C(=O)C1CC1)CC2 88014,c1(CC(=O)NCCC(C)CCNC(C2(F)CCCCC2)=O)cccc(Cl)c1Cl 88015,N1(C(CCC(C)C#N)=O)CCCC(C)(C)C1CNC(C1C2CCC1(C)C2(C)C)=O 88016,CC(C)CCC(C(=O)NC1CCS(=O)(=O)C1)NC(C1CCCC(=O)N1C)=O 88017,CC(CCCNC(=O)Cc1nccn1C)NC(c1cnc(Cl)s1)=O 88018,C1(CCC)CCN(C(C2CC(CNC(=O)C(C3CC3)OC)C2)=O)C1 88019,C1(C(=O)NCC(CNC(C(Cn2ccc(C)n2)C)=O)O)CC(C2CC2)=NO1 88020,C1(OC)CC(NC(C2(OC)CCSC2)=O)CN(C(=O)Cc2occc2C)C1 88021,c1(OC)c(NC(=O)CC(C)OC2CC2C(=O)OC)cccc1F 88022,CC(C)CC(C)(O)C(=O)N(C)CC1CCN(C(c2ccc(CN(C)C)[nH]2)=O)C1 88023,N1(C(CCCCOC)=O)CC(NC(C2(C(=O)N(C)C)CC2)=O)CC(F)(F)C1 88024,Cc1ccc(O)c(C(N2CCC(O)C(NC(C3CC4(C3)CC4F)=O)C2)=O)n1 88025,C1(NC(c2ccc(C#C)cc2)=O)CC2CN(c3nccc(SC)n3)CC2C1 88026,N1(C(CCC)=O)CCC2(C=C(C(=O)N(C)Cc3cncs3)C2)C1 88027,C1(CC(=O)NC2(CCO)CN(C(C3CN(S(C)(=O)=O)C3)=O)C2)CC2CCC1O2 88028,C1(C(=O)NCCn2ccnc2)CN(C(c2ccnc(-c3ccccc3)c2)=O)CCN1 88029,CP(C)(=O)c1ccc(C(N2CCC(NC(c3cn4c(n3)COCC4)=O)C2)=O)o1 88030,c1(CC(N2CC=CC(NC(CCCCSC)=O)C2)=O)cnc2n1CCCC2C 88031,CC1(C)CCCN1CCSC.n12cc(nn1)C(c1ccccn1)NC2=O 88032,c1(CC(=O)NC2CC(C)(CNC(=O)Cc3cnns3)C2)ccc(Br)cc1 88033,c1(C(=O)NCC2CCN2C(C23CC(F)(C2)C3)=O)cnc2ccsc2c1 88034,C=C(C)CC(C)C(=O)NC1CN(C(c2csc(CO)n2)=O)CC1O 88035,c1(C(=O)NC(CNC(C2C=CCC2)=O)C2CC2)ccc(Br)cn1 88036,C1(CC(=O)NC(C)Cn2ccnc2)C2CCC(C2)N1C(c1c[nH]c(=O)cn1)=O 88037,c1(C(=O)NCCCC(CC)N(C)C(C2CC3CC3C2)=O)cc(C2CCC2)on1 88038,N1(C(C(C)OCCCC)=O)CCCN(C(=O)C=CSc2ccco2)C(C)C1 88039,C(=O)(C1=CC(C)CC1)NCCC(C)NC(c1nc(C)sc1C)=O 88040,c1(CC)nc2ccc(NC(=O)N(C3CCC3)C3CC3)cc2s1 88041,C=C(Cl)CCC(=O)N(CC(C)NC(=O)C(C)(C)c1cscc1Cl)C 88042,Cc1cccc(C(C)(C)C(=O)NCCN(CC(C)O)C(=O)CCCCC(C)C)c1 88043,C1(C(=O)NC2CN(C(C(C)SCCCC)=O)C2)CN(C(=O)C=CC(C)C)CCO1 88044,Cc1ncccc1CCCNC(C1(NC(=O)COc2ccccc2)CCCC1)=O 88045,N1(C(=O)C(O)Cc2ccccn2)CCN(C(=O)Cc2ccsn2)C(CO)C1 88046,c1(CN2CC(C(=O)Nc3cc(OC)n[nH]3)SCC2)ccc(Cl)nc1C 88047,c1(CSC)ccc(C(N2CCC(N(C(=O)C(CO)N(C)C)CCO)CC2)=O)cc1 88048,c1(CNC(c2n(CCOC)nnn2)C2C3COCC23)cccc(F)c1OC 88049,Cc1ccc(C(C)C)c(C(N2CCSC(C)(C)C2)=O)c1 88050,N1(C(c2cc(C)c(N)cn2)=O)CCN(C(C2CN(C)CC(C)O2)=O)CC12CC2 88051,c1(C(N(C2CCCN(C(=O)Cc3ccccc3)CC2)C)=O)cnc2ccnn2c1 88052,C1(C)(CC(=O)N(C(C)CN(C(=O)CCOC2CC2)C)C)CCOCC1 88053,c1(C(N2CCC(NC(C3(CC#C)CCCC3)=O)C(C)C2)=O)cc(O)cc(C#N)c1 88054,C=CC(CC)CC(=O)NN(C(C)C(=O)N(C)CCN(C)C(=O)C1CC1)C 88055,N1(C(C(C(C)O)(C)C)=O)CC2CCC1CN2C(=O)CCc1ccccn1 88056,C1(CC(=O)NCC2(C(=O)OC)CC2)CCCCN1C(c1ccc(Cl)o1)=O 88057,c1(CN2CC(C(N3CCC(N4CCC4)CC3)=O)NCC2)cc(Br)cc(Br)c1O 88058,Cc1nc(O)nc(C)c1CCC(N1CC(C2(NC(c3csc(=N)[nH]3)=O)CC2)C1)=O 88059,c1(C(N2C3(c4cn(C(COC)COC)nn4)CCC2CC3)=O)ccccc1[N+](=O)[O-] 88060,N1(C(c2n(C)ccc2)=O)CCOCC(CNC(C2CCC2)=O)C1 88061,C(C)(C)(C(=O)NCC=CC(=O)NCC1CC1CC(C)C)SC 88062,c1(C(=O)NCC2C(C(=O)NCc3cn(CC)nc3)CCO2)cncc(OC)n1 88063,C(=O)(C1COc2ccccc21)N1CCC(NC(CC2(CSC)CC2)=O)C12CC2 88064,C1(CC(N)=O)(NC(=O)C2=COCC2)CCN(C(c2n[nH]c3c2CCC3)=O)CC1 88065,c1(C(N(C(C)CN(C(=O)C(C)(C)C#N)C)C)=O)ccc(P(C)(C)=O)cc1 88066,CCCCN=C(NCCc1ccc(F)cc1F)NCC1CC(=O)N(C(C)C)C1 88067,CC(C)C(C(=O)NCC1CCN1C(C1CCC1(F)F)=O)C(C)C 88068,Cc1csn1CC(=O)NCCN(C(=O)CC1CCCC1)C1CC1 88069,N1(C(CCC#C)=O)CC2(CCN(C(=O)CNCCOC)C2)C1.c1ccccc1 88070,C(CC(=O)NCCCC(=O)OC)(C(C)C)NC(C(CCC)OCC)=O 88071,S(=O)(=O)(c1cnn2ccc(=NC(C)CCOC)[nH]c12)NC(C(CC)CC)C 88072,C1(C(=O)NC2CC(C)(NC(c3cn(C)nc3)=O)C2)C2CCN(CC2)S1(=O)=O 88073,c1(C(N2C(CCCNC(c3cnc(S)[nH]3)=O)CCCC2)=O)ccc2nc[nH]c2n1 88074,N1(C(=O)Nc2ccnn2C2CNC2)CCC2(CCCCO2)C1 88075,C(c1ccc(F)cc1Cl)=CC(N1CC2CN(C(CCCC#C)=O)CC21)=O 88076,Cc1c(NC(C2CC(F)(F)CN2Cc2cn3ccccc3n2)=O)ccc(Br)c1Br 88077,n1(CCC)nc(C)cc1C(=O)NC1CCC1NC(c1cccc(C(N)=O)c1)=O 88078,c1(C(=O)NCC2N(C(c3cc(C)ncc3C)=O)CC2)ccc2nc(Cl)nn2c1 88079,N1(C(c2cncc(OC)c2)=O)CCC(C)C(NC(C2CCCN2C2CC2)=O)C1C 88080,C1(CC(=O)NCC2CCCS2)CC(F)CN1C(C1C(C2(C)CCC2)C1)=O 88081,c1(CCC)noc(CN2CCC(CCNC(=O)C(C)O)C2)n1 88082,Cc1ccc(F)c(O)c1C(=O)NCCC(C)(C)NC(C12CC(CC(F)F)(C1)C2)=O 88083,CCC1=NOC(C(=O)NCCC(C)(C)NC(c2ccn(C3CC3(F)F)n2)=O)C1 88084,CCCCC(C(=O)NC1CCN(c2nnn(C)n2)C1C)NC(N)=O 88085,N1(C(c2c(OC)nsc2)=O)CC2CCOC2(CNC(c2cc(F)cc(Cl)c2)=O)C1 88086,c1(NC(Cn2cc(C(=O)NC)nn2)=O)ccc(C)c(N(C)C)c1 88087,c1(C(N2C(CN(C(C(CC)SC)=O)CC)CCC2)=O)cc(N)ccc1Cl 88088,c1(OCCCC)ccc(C(=O)NCC2(C)CC2(Cl)Cl)cc1OCCC 88089,c1(CN(C(=O)CN(C(c2ccoc2Cl)=O)C2CC2)C)cn(C)nn1 88090,C1(CC(C)O)CCC(C)CN1C(=O)NC1CCCCC12CC2 88091,N1(C(c2scc(COC)n2)=O)CCS(=O)(=O)C(Cc2ccc(F)cc2)C1 88092,N1(C(CC=CCC)=O)CC2CCC(C1)C2CNCc1ccc(-n2cncn2)cc1 88093,C1(CC(=O)N(CC(N)=O)CCO)CC(N=c2ccnc(Cl)[nH]2)C12CCOCC2 88094,CC(C)CCC(O)C(=O)NC(CC1CC1)C(N1CC(=O)NCC1C(N)=O)=O 88095,c1(OC(CNC(=NC)NCCc2cnccn2)(C)C)ccccc1C#N 88096,N1(C(COCCC)=O)CCC(C)(C(=O)NCC2CN(C(C)C)CCO2)CC1 88097,C1(C(N(CCCCCNC(c2c(C)ocn2)=O)C)=O)CC12CCC(F)(F)CC2 88098,Cc1ccc(N)c(C(=O)NCC(CO)NC(=O)Cc2ccccc2)c1 88099,C1(N(C(=O)CCc2csc(C)n2)CC#C)CCN(C(C2CCC(C)S2)=O)CC1 88100,c1(CC(N2CC3CC(NC(CN(C)CC)=O)C3C2)=O)ccc2n[nH]cc2c1 88101,N1(C(CC(C)(C)C)=O)CC2CCCC(NC(c3coc4c(F)cccc34)=O)C2C1 88102,N1(C(COC(C)C)=O)CC(NC(=O)Cc2cc(C(C)C)no2)CC(O)C1 88103,c1(C(=O)NCC2C(NC(CCC=C)=O)CC2)c(C)ccc(F)c1O 88104,c1(C(c2nnnn2C2CCCCCC2)NCC(COCC)C)oc(CC)nc1C 88105,c1(C(N2C(CC(=O)NCCc3c(C)c[nH]c3C)COCC2)=O)nc(Cl)ccc1F 88106,C(=O)(C1CCc2c(Cl)cccc21)N(CCCNC(=O)COC1CC1)CC 88107,CC(C)CC(C)(C)C(=O)NC1CN(C(c2ccncc2Cl)=O)CC2(CC2)C1 88108,C(C)(C)(CCCC(=O)N1CCC2C(O)CC12)NC(CCc1n(C)cnc1)=O 88109,C(=O)(C(F)CC(C)(C)NC(c1cc2ccccn2n1)=O)NCC(c1cccs1)C 88110,C1(C(=O)NC(C)CCNC(=O)C(=Cc2cccs2)C#N)CCCC2C1C2(F)F 88111,C(C(Cc1ccc(Cl)s1)C(=O)N1CC(O)CC1c1ccc(F)cc1)OC 88112,CCC(C)C(O)C(=O)N1CCN(C(=O)Cn2cc(C)ccc2=O)CC1 88113,c1(C(=O)NC2CCC(N(C(c3ncc(CC)s3)=O)C)C2)ccc(C2CC2)cc1 88114,C(=O)(C(C)(CSC)NC(=O)C=CC1CCOC1)N1C(C)(CC)CC1 88115,N1(C(C2C(C)(C)C2)=O)CCC2CC1CN2C(=O)CCNC(C1CCCCC1)=O 88116,C(=O)(CC1OCCc2ccccc21)NC(CN(C(c1[nH]cc(CC)c1)=O)C)C 88117,C1(C(N2C(CN(C(c3[nH]cc(C(C)=O)c3)=O)C)CCCC2)=O)C(C)(C)OC1(C)C 88118,Cc1cc(C(N2CCCC2CC(=O)NC(C)CC2(O)CCC2)=O)c(N)s1 88119,C(C(=O)NCC1CCCN1C(=O)CC1OCCO1)(C(C)C)n1cc(C)nc1 88120,C#CCC(CC(=O)NC1CC(NCC2CCCCO2)C1)NC(C1CC1)=O 88121,C(=O)(C(C)(CSC)NC(=O)OC(C)(C)C)NC1CN(C(C=C(COC)C)=O)C1 88122,CC(c1cccnc1)=CC(=O)NC1CCN(C(c2conc2C)=O)CC1F 88123,Cc1cc(C(N2CCC(C(=O)NC(C34CC(CO3)C4)C)C2C)=O)c(C)nn1 88124,N1(CC(c2cccc(OC)c2)=O)CCC(O)C(C(=O)NCCc2nccs2)C1 88125,C(CCN=C(NCC(C(C)C)c1ccnn1C)N1CCC(C(C)(C)C)CC1)SC 88126,C(=O)(C(C(C)O)NC(=O)COC1(C)CN(C(C)=O)C1)NCCN(CC=C)C 88127,C(=O)(C(C)P(C)(C)=O)NC(CNC(C(C)(F)F)=O)C(C)(C)C 88128,N1(C(C(CCCC)=O)=O)C(CNC(=O)C(c2cnn(C)c2)C)CC2CCCCC12 88129,C(CO)(C(=O)N1CCCC1CC1CCC1)NC(CC(=O)N(C)C)=O 88130,CN(C)NC(=O)CCC(=O)NCCOC1CN(C(C23CCCC2CC3)=O)C1 88131,c1(C(=O)NC2CCN(C(C3COC3)=O)CC2O)ncn2ccccc12 88132,C1(C(N(C2CCN(C(=O)C(=O)N3CCCC3)C2)C)=O)CCc2cncn2C1 88133,C1(CCNC(c2sc(F)cc2Cl)=O)CCCN(C(c2ccc(CCO)cc2)=O)C1 88134,C(=O)(CC(C)(C)CC)NC(CC#C)C(=O)N(C1CCN(C(C)=O)C1)C 88135,c1(CC(N2CCC3CN(C(c4c(C)coc4)=O)CC32)=O)coc2cc(O)ccc12 88136,Cc1cncc2cc(C(=O)NC(C)CCCCNC(C3C4CCCOC34)=O)sc12 88137,Cc1ccnc(O)c1C(=O)N(CC(O)CN(C(=O)CC1(N2CCCC2)CC1)C)C 88138,N1(C(c2c(C)cco2)=O)CC2C3CCC(C2C1)N(C(=O)CSCC(N)=O)C3 88139,Cc1c(N)ccc(C(=O)NC(C)(C)CNC(C2CCC(C)(C)O2)=O)c1C 88140,N1(C(CNC(CC)=O)=O)CCCC2C1CCCCN2C(=O)C(O)C(C)C 88141,CC(O)(C(=O)NCC(O)CC(=O)NCC(O)CCC1CC1)C(F)(F)F 88142,C=CCCCCCCC(=O)NC1CCC(NC(=O)C=C(C)c2ccccc2F)C1 88143,N1(C(CONC(c2cncc(C=C)c2)=O)=O)CCn2c(cnc2C)C1 88144,c1(C(=O)NCCCC(=C)C)ccc(CNC(C2(C)CCOC2C)=O)nc1 88145,c1(C(=O)NC2CN(C(COC(CC)(C)C)=O)CC2(C)C)nccc2cccnc12 88146,C1(CNC(=O)CCc2nccs2)CN(C(C2CC2F)=O)CCC12CCOC2 88147,c1(C(N2CCC3CN(C(C4CC4F)=O)C3C2)=O)cc(Cl)cc(Cl)c1O 88148,N1(C(c2ccc(C(F)F)o2)=O)CCC2CCN(C(=O)CCc3cccs3)C2C1 88149,CC1CN(C(c2cc(O)nc(O)n2)=O)CCCN1C(=O)C(c1ccccc1)O 88150,c1(OC)cc(F)c(NC(=O)Nc2cc(NC(C)CC3CCCC3)ncn2)c(F)c1 88151,C1(C(=O)NC2C(NC(c3cn(CCF)nn3)=O)CCC2)CC12CCOC2 88152,CCCC(C(C(=O)NC)N1CCN(C2CC2)C(CS(C)(=O)=O)C1)OC 88153,CC1CN(C(=O)C(=O)NCc2cnn(C3CC3)c2)CCS(=O)(=O)C1 88154,C12(CC)CN(C(c3ccc(C4CC4)o3)=O)C(CNC(C3CN(C(C)=O)C3)=O)(C1)C2 88155,c1(OC)cc(F)c(C(=O)NCCC(O)CNC(c2cc(C)c[nH]2)=O)c(Cl)c1 88156,CC1(CNC(c2cc(C#N)cs2)=O)CN(C(c2csnn2)=O)CCO1 88157,c1(C(N2C(C(C)C)CN(C(=O)C(=O)C(C)(C)C)CC2)=O)cn2cccc(Cl)c2n1 88158,c1cccc(Cl)c1.O=C1CCN1.c1(C(=O)NCCOCCNC)ccco1 88159,C1(NC(c2ccc(C(C)=O)o2)=O)CCC(NC(C2C(C)C2(F)F)=O)CC1 88160,c1(C(=O)OC(c2c(OC)cccc2)C)c(C)ccc(F)c1Br 88161,N1(C(c2scc(C(=O)OC)n2)=O)CCC(NC(c2cccc(NC)c2)=O)C(O)C1 88162,c1(CNC(c2c(C(C)NC(c3cccnc3)=O)noc2)=O)ccc(C#N)cn1 88163,N1(C(C(=O)N(C2(CNC(CC#N)=O)CCOC2)CCl)C2CC2)CCS(=O)(=O)CC1 88164,N1(C2CCN(Cc3cc(OC)cc(O)c3)C3(C2)CC3)CCc2c(Cl)cccc2C1 88165,N1(CC(=O)Nc2c(OC)ccc(CO)c2)CC2COCC1CN(CCN(C)C)C2 88166,C1(N(C(=O)Cc2sccc2C)CC)CCN(C(=O)CCc2cnn[nH]2)CC1 88167,CN1CCCC(NC(=O)NNC(=O)C2CCC(=O)N2)CC1 88168,Cc1c(Cl)c(C(N2CC3(C2)CN(C(c2cc(Cl)ncc2O)=O)C3)=O)nn1C 88169,CCC(N=c1[nH]c(=NC(C)c2ccncn2)c2ncccc2[nH]1)c1ccncc1 88170,N1(C(C)=O)CCC(C(=O)NCCCNC(=O)Cc2cccs2)CC1 88171,c1(C(N2CC(C)(C)C(NC(c3cc(N)ccc3F)=O)C2)=O)csc(S(C)(=O)=O)c1 88172,C1(C2(O)CCOC2)(CNC(c2c(OC)cc(NC(C)=O)cc2)=O)CC1 88173,c1(OCC(N2CC(NC(c3c(C)csc3)=O)C(C)(C)C2)=O)ccc2c(c1)CCC2 88174,C1(NC(CCN(CCC)C)=O)CCC2CCN(C(=O)CC3CNC(=O)C3)C12 88175,C(=O)(CC(O)CC(C)(C)C)N1CCC(=C)CC1C(=O)NOCC1CCC(OC)CC1 88176,C1(NC(c2c(C)nc(CNC(C3CC(=C)C3)=O)o2)=O)CCOC(C)(C)C1 88177,C(C)(CCC(C)(C)C)(C(=O)O)NCc1ccc(CC)o1 88178,C(C(Cc1ccc(F)cc1)C(=O)O)NC(c1cccc(N2CCOCC2)n1)=O 88179,Cc1ccccc1NCC(=O)NC1CCCC(NC(C2CCN2C(C)(C)C)=O)C1 88180,Cc1nnccc1C(N1CCOC(C2CCCCC2)C1)C(=O)NCC1CCOC1 88181,Cc1nc(C)c(C(=O)NC(C)(CNC(=O)CCC2CCC(C(N)=O)O2)CO)[nH]1 88182,c1(C(=O)NCC2C(CNC(C=CCCC)=O)C2)c(Cl)cncc1Br 88183,c1(OC)ncc(NC(C2CCN(C(=O)CC3CC(OC)C3)C2C)=O)cn1 88184,N1(C(C(CN(C)C)(F)F)=O)CCCC(CCNC(c2ccc(Cl)s2)=O)CC1 88185,C1(CNC(c2c(C)occ2C(F)(F)F)=O)CCN(C(=O)C(C)(F)F)C1(C)C 88186,c1(C(=O)NC(C2N(C(C3ON=C(C)C3)=O)CCC2)C)cccc(-n2ccnc2)c1 88187,c1(C(N2CCC(NC(CSCC=C)=O)C2(C)C)=O)ccc(C)c(C)c1O 88188,CC(CNC(=O)CC1CCOC1(C)C)CC(=O)NCCC1(C)CCCC1 88189,C1(NC(C2N(C(C(C)NC(=O)OC)=O)C3(CC2)CC3)=O)CCN(C)CC1C#N 88190,O=C1CC2C(C(=O)NCc3cc(C(=O)NC4CCC(O)C4)ccn3)C2C1 88191,CN1CC(NC(C2CCC2NC(=O)CCN2CCOC2=O)=O)CC1(C)C 88192,N1(C(C2C(O)CCN(c3cc(C)cc(C)n3)C2)=O)CC2CC3CCCN3C2C1 88193,CC(C)C#CC(=O)NC(CCN(C)C)C(=O)NC(C)C(C)F 88194,[N-]=[N+]=NCCCCCCNC(=O)C(c1ccoc1)NC(=O)CC1(O)CCCCC1 88195,CCCC(C)(O)CC(=O)NC(C)CCNC(c1cc(Br)cnc1N(C)C)=O 88196,c1(OC)cc(C(N2CC(OC)CC2CNC(c2ccc[n+]([O-])c2)=O)=O)cc(Cl)n1 88197,c1(OCC=C)cccc(C(c2nnnn2CC(F)F)NCCC(C)CO)c1 88198,N1(C(=O)C#CC2CC2)C2CCC1CN(c1c(Cl)cncc1[N+](=O)[O-])CC2 88199,n1(CC)ncc(C(N2CC=CC(NC(c3cnc(N(C)C)cn3)=O)C2)=O)c1C 88200,c1(C(=O)NC2CC(O)(CNC(C(C3CC3)SCC)=O)C2)cnc2c(c1)COC2 88201,N12CCC(CC1)C2=O.c1(CC(c2cccs2)N(CC=C)CC=C)ccc(F)cc1 88202,C1(CNC(c2cn(C3CN(C(C(C)OCCC=C)=O)C3)nn2)=O)CCCOC1C 88203,C1(CNC(CCOCCNC(C2CC(CC(C)(C)C)C2)=O)=O)CC[Si](C)(C)C1 88204,C12(C(=O)NCCCCC(C)NC(C(C)c3ncco3)=O)CC3CC(CC(C3)C1)C2 88205,c1(C(=O)OC)ccc2oc(CNc3nccc(C)n3)cc2c1 88206,N1(C(CCC#CC)=O)CCC2(CC1)OCCC2NC(c1cc(OC)cs1)=O 88207,c1(C(N2CC3C(CCNC(c4c(C)cco4)=O)(CC3)C2)=O)cccc([N+](=O)[O-])c1 88208,C1(NC(C2CN(C)C2)=O)CN(C(C2(O)CCCC2)=O)CCC1F 88209,N1(C(CCC)=O)CC2CC(NC(C3OCC3(C)C)=O)CC2C1 88210,CC1(C)CCCC(CNCCn2ncc3ccccc23)CC1 88211,c1(OC)cc(C(=O)NCC(CNC(=O)C(O)C(C)C)C(F)(F)F)cc(N)c1O 88212,C(=O)(C(F)(F)C(F)F)N1CCC(N(C(=O)COC2CCC2)C)C1 88213,C12(C(=O)NCC3CC(NC(=O)Cc4cccc(O)c4)C3)CSCC1C2(F)F 88214,c1(OC)ccc(CCCC(=O)N2CCCC2C(C)(C)NC(=O)C(Cl)=CCl)cc1 88215,C1(CCCC)CCC(NC(C2CN(C(=O)CCOCC(F)F)CCO2)=O)CC1 88216,C1(NCCNC(=O)C(C)OCCOC)CCCCC1.C12(CC1)N(CCC)C2=O 88217,Cc1cnn2cc(C(N3CCCC3CCNC(C3(N(C)C)CC3)=O)=O)cnc12 88218,c1(CCC(=O)NCC2CCN(C(c3c(C)cco3)=O)C2)cccc2c1OCCO2 88219,c1(CC)cc([N+](=O)[O-])ccc1N1CCC(CCOC)(NC(=O)C(C)C(C)(C)C)C1 88220,C12(NC(C(C)(F)F)=O)CC1CN(C(c1csc(Cl)n1)=O)C2 88221,C1(CC(N2CC(OC)(CNC(=O)CC(=O)NC3CC3)C2)=O)CCN(C)CC1 88222,c1(CC)[nH]c(=N)sc1C(=O)N(CC(C)N(C)C(c1cncnc1C)=O)C 88223,N1(CC2CCC(Nc3n(C)ncc3)CC2)CCc2nc(C(=O)N(C)C)cn2CC1 88224,N1(C(C=Cc2n(CC)ccn2)=O)CCCC2(NC(c3n[nH]cc3OC)=O)CC2C1 88225,c1(C(N(CC(O)CNC(=O)C#CC2CC2)C)=O)cnc2c(F)c(F)ccc2c1 88226,c1(C(=O)NCCC(C(C)C)NC(C(COC)C)=O)cccc2ncc(Br)n12 88227,C1(CCC(=O)Nc2cc(CC)no2)CCCN(C(C2CCC(=O)O2)=O)C1 88228,CCC(C)(C)CC(=O)N1CCC(C)(C(=O)NC2CC3(CC3)C2)C1 88229,c1(NC(C)=O)cccc(C(=O)NC2CCCC(CNC(c3scnc3Cl)=O)C2)c1 88230,c1(C(=O)NC(C2(O)CCN(C(c3ccn(C)c3)=O)C2)C)cc2c(ccn2C)[nH]1 88231,N1(C(c2cc(-c3cn(CC=C)nc3)[nH]n2)=O)CCc2cc(C)ccc2C1C 88232,N1(C(C(CN(C(COCCC#C)=O)C)(C)C)=O)CC2OCCN(C)C2C1 88233,N1(C(CSc2c(C)cccc2)=O)CCC2(CCN(C(C3(C)CC4CC4C3)=O)C2)C1 88234,c1(C(=O)NC2CCC(NC(c3c(OC)cc(Cl)nc3)=O)C2)cc(C)c(F)cc1Br 88235,c1(C(C(=O)NCC2(C)N(C(c3onc(CC)n3)=O)CCC2)C)cc(C)cc(F)c1 88236,C1(C(=O)NC(C)(C)CNC(C2CC(C)(F)C2)=O)CCCC1(F)F 88237,c1(C(N2C(CCNC(=O)C3=CCCCC3)CCC2)=O)cc2cccn2cn1 88238,C#CC1(C(=O)NCC2(O)CCC(C)(C)C2)CCN(C(=O)COC2CC=CC2)C1 88239,CCC(CC(C)C)C(=O)N1CCC(CN(C(=O)C(C)(C)c2ccn(C)n2)C)CC1 88240,c1(C(=O)NC(CCNC(C2(CC)CCCC2)=O)C)nn(C)c2c1CC(C)(C)CC2 88241,C1(C(=O)NCC(CCNC(=O)CCc2cnco2)O)CCc2ccccc2C1 88242,C1(C(=O)NCCC2CC(NC(Cc3ccc(C)o3)=O)C2)CCCCN1S(N)(=O)=O 88243,C1(CN(C(C(=O)NCC)=O)C)CCCC(NC(c2csc(=N)[nH]2)=O)C1 88244,c1(C(=O)OCC)cnc(NC2CC3(C2)CC3NC(c2[nH]nc(OC)c2Cl)=O)cn1 88245,C1(C(F)(F)F)(C(=O)NC(CC)CNC(c2ccnnc2)=O)CC=CCO1 88246,N1(C(C)COc2ccccc2)CCC(O)(C(=O)NCC2COC2)CC1 88247,N1(c2nnc(C)s2)CCOC2(CCN(C(c3ccc4ncnn4c3)=O)CC2)C1 88248,N1(C(C=CC)=O)CCCCC1CCN(C(=O)C(C(=O)OC)OC)C 88249,c1(OC)nn(C)cc1N(C)C(C1CC(CNC(=O)CCCC2CC2)C1)=O 88250,N1(C(CN(CCC)C)=O)CCC(NC(c2ccc(OC)nc2C)=O)C12CCCC2 88251,N1(C(C=CCOC)=O)CCCCC1C(C)NC(C1(C)COC1)=O 88252,N1(C(c2cc(CCNC(c3cnc(C)o3)=O)on2)=O)CCOC2CC12 88253,c1(CC(CNC(C2CCCCC2)=O)NC(=O)CCC2CCCO2)ccccc1 88254,C1(CC)CC(C(=O)NCC(C)CC(=O)OC)CCN1C(c1c[nH]c(=N)c(C)c1)=O 88255,N1(C(CSCC#C)=O)CCC(O)(CCNC(=O)C(c2nc(C)cs2)C)C1 88256,C1(C(=O)NC2CCN(C(c3cocc3C)=O)C2)(COC)CCCCO1 88257,C1(CNC(C(CO)N(C)C)=O)C2CN(C(=O)C(F)(F)c3ccccc3)CC12 88258,N1(C(C(C2CCN(C(C3C(CCC)CCC3)=O)C2)F)=O)CC(OCC)C2(CC2)C1 88259,n1(CC)nc(C(=O)NCCC2CC(NC(=O)C(C)(COC)OC)C2)c(C)n1 88260,n1(CC)cnc(C(=O)NCC2(NC(c3ccn(CC(C)C)n3)=O)CCCC2)n1 88261,c1(C(=O)NCc2ncon2)cc2ccc(-c3cnn(C4CCCCO4)c3)cc2s1 88262,C1(NC(C2(CC)CCCN2C(=O)C(C2CCOCC2)=O)=O)CCC2(CCC2)C1 88263,C1(C2CN(C(=O)CN=S(C)(C)=O)C2)(NC(C(=C(C)C2CC2)F)=O)CC1 88264,c1(C(N2CC(C)C(F)(F)C2)C(=O)NC)cccc2c1CCO2 88265,N1(CC(N2C(CC(=O)NC(COCC)CO)CC2)=O)CC(=O)NC1=O 88266,c1(CC(N2CC(N(C(C3N(CC)CC3)=O)C)C(O)C2)=O)cc(C)ccc1OC 88267,C1(C(N2C(CC)CN(C(=O)CCCF)CC2)=O)CCC(C2CC2)CC1 88268,C1(C2(NC(C=NOC)=O)CC2)CCCCN1C(c1cccc(CF)c1)=O 88269,C#CC1(O)CC(C(=O)NC2(C(=O)NCCSCc3ccco3)CCSC2)C1 88270,CCC1C(=O)N(C2CC2)CC(=O)N1.C(=O)(C(C)(F)c1ccon1)NC 88271,c1(NC2(C)CCN(C(C(C=CC)O)=O)C2)ncc(C(=O)OCC)cc1[N+](=O)[O-] 88272,C1(OC)CCCC1C(=O)N(C(C)CN(C(=O)Cc1cccnc1)C)C 88273,CC(CNC(C1CN(C)CCN1C)=O)C(F)C(=O)NC1CCNC(=O)C1 88274,c1(CC(=O)NC2C(C)CN(C(=O)C(C)(C)C3CCC3)C2)ccc([N+](=O)[O-])cc1F 88275,c1(C(=O)NC2CCC(CNC(CS(N)(=O)=O)=O)C2)cnc2nccn2c1 88276,C1(NC(c2n(CC)nnn2)c2cnn(C)c2)COC(C)(C)C1 88277,C1(C(=O)NC(C2(CNC(c3cc(C)n(C)c3)=O)CC2)C)CCC(C)(C)OC1 88278,N1(C(COCCOC)=O)CC2CC2(C(=O)NC(CO)C(=O)O)C1 88279,N12CC3CC1CN3C(=O)C(O)C1CN(C3CN2C3)C1.C(=O)NC.C(C)=O 88280,N1(C(C2(C#C)CCCC2)=O)CCC2(CCCC2CNC(C2CCNC2=O)=O)CC1 88281,N1(C(=O)OCC)CSCC1C(C(=O)CCCc1ccccc1)=O.C12(CC1)NC2 88282,C1(NC(C(CNC(C(C2CCC2)OC)=O)OC)=O)CC(C)(C)C12CCC2 88283,N1(C(CSc2ccc(C)cc2)=O)CC2(CCN(C(=O)CC(C)C(C)C)C2)C1 88284,CC1OC2(C(=O)NC3CCN(C(c4cc(C(N)=O)co4)=O)C3)CC1C2 88285,C#CCCCCC(=O)NC1CCC(NC(C2(CCOC)CC2)=O)C1 88286,CCC(CC)CCC(=O)NCCCN(C(c1cc(OC)ccc1CC)=O)C1CC1 88287,Cc1cc(C(N2CC3CC3(CNC(=O)CC3CCCC3O)C2)=O)n(C2CCC2)n1 88288,N1(C(C2N(CC)CC2)=O)CCC(CNC(=O)C=CCN(CC)CC)C1(C)C 88289,N1(C(C=C(COC)C)=O)C2CCCC1CC(NC(C1CC(n3cnnc3)C1)=O)C2 88290,c1(-c2nnc(N3C(CCC)CCC3)n2CCCCCO)cc2ccccc2o1 88291,C1(F)(C(=O)NC(C(C)NC(C2(F)CC=CC2)=O)C)CCCCC1 88292,CC1(C)CCC(NC(c2cncnc2)=O)C(CNC(=O)C2=CCCOC2)C1 88293,c1(C(=O)NC2C(CNC(c3cnc4c(c3)CCC4)=O)C2)cccc2c1COCC2 88294,C1(CNC(C(CCC)C)=O)CC2CCC(C1)N2C(C1(C#N)CCCC(=O)C1)=O 88295,N1(CC(=O)NCC2C(C)CN(C(=O)C=CC3CCOC3)C2)CCCCCCC1=O 88296,Cc1cc(F)ccc1C(F)(F)C(=O)NC1C2CN(C(C3CCCOCC3)=O)CC12 88297,CCC(C)(CO)C(=O)NCc1cncc(C(=O)NCC(O)CC2CCC2)c1 88298,CN1CCC2CCC(C1)N2C(C1(C2CCCN2C(=O)C2=COCC2)CC1)=O 88299,C1(CNC(C2(C)ON=C(C)C2)=O)CN(C(=O)CC2(C)CC(F)(F)C2)CC12CCC2 88300,N1(C(C(=O)NC(CC)C)CCC2CC2C)CC(C(=O)OC)C(C2CCCCC2)C1 88301,c1(NC(C(F)=CC)=O)ccc(NC(c2cc(CC(C)C)c[nH]2)=O)cc1C 88302,N1(C(C(C)C(C)(F)F)=O)CCC(C2(O)CN(C(=O)CNS(N)(=O)=O)C2)CC1 88303,N1(C(COC(C)=O)=O)CC2CC1(CNC(c1ncc(C(F)F)s1)=O)C2 88304,c1(CC(=O)NCCN(C(C(C=CCCC)O)=O)C2CC2)ccc(C)cc1Cl 88305,c1(OC)ccc(F)cc1C(=O)N(C1CCCN(C(C2CCCOCC2)=O)CC1)C 88306,N1(C(C2C(C#C)C2)=O)CCOCC1CN(C(=O)C=CCOC)C 88307,CC(F)(F)C(C)(C)C(=O)NCCC1CC(F)(F)CN1C(C1COCCN1C)=O 88308,c1(C(N2CCC(N3CCOC3=O)C2)C(=O)NCCOC)cnc(OC)c(Cl)c1 88309,C(=O)(C(O)C(F)(F)F)N(CC(CC)NC(=O)C(O)Cc1ccccn1)CC 88310,c1(C(=O)NC2CCC(NC(C3N(C)CCCCC3)=O)CC2)cnc2c(c1)COC2 88311,N1(C(C(CCC)F)=O)CC(CNC(c2c(C)noc2C2CC2)=O)CC(C)C1 88312,C(CO)(C(O)c1cccnc1)NC(c1nc(Br)c[nH]1)=O 88313,c1(OCC(N2C3CC(NC(C4N(C)C(=O)OC4)=O)(C3)C2)=O)ccc(Cl)cc1F 88314,C(C(C(C)(C)C)NC(=O)C=CCOC1CCOCC1)NC(COCCC#C)=O 88315,CCC(C)C(=O)NC(C)CCCNC(c1cnoc1-c1cccs1)=O 88316,CCCCCC(C)C(=O)N1CCN(C(=O)COc2ccc(Br)cc2)CC1C#N 88317,C(=O)(C(F)C(F)(F)C(F)(F)F)NC1C(CNC(C(=O)N(C)C)=O)CC1 88318,N1(C2CN(C(C=CC(C)C)=O)C2)CC(NC(=O)C(=O)N(C)C)CC1=O 88319,C1(NC(c2cc(C3CC3)on2)=O)(CF)CCN(C(=O)CCF)C1 88320,c1(C(=O)NCC2CN(C(CC3C(C(=O)OCC)C3)=O)C2)n[nH]c2c1CCCCC2 88321,C1(CNC(C(=O)NCC2CC(C)(C)C2)=O)Cc2ccc(Br)cc2C1 88322,C12(CC(F)(F)C1)COC(C)C(=O)OC2.C1(C(=O)OCC)CCCN1C(CC=C)=O 88323,c1(NC)cnncc1C(=O)NC1CCC(CNC(c2cc(O)ncn2)=O)C1 88324,CC(CC(=O)N1CCCC1CCCNC(=O)C1=NNC(C(F)(F)F)C1)C(F)(F)F 88325,C1(C(=O)NC(CC(C)NC(c2cnc(C)s2)=O)C)Cc2ccccc2N1 88326,CCC(CC)CCCC(=O)NC(Cc1cc[nH]n1)C(N1CCCC(N=[N+]=[N-])C1)=O 88327,C1(NC(c2cc(C(N)=O)[nH]c2)=O)CC2CCC1(NC(C1CC=CC(O)C1)=O)C2 88328,C(=O)(C1c2c[nH]nc2CN1C(=O)C#CC1(C)COC1)N(CC(C)O)CC1CC1 88329,c1(CC)c[nH]c2ncnc(N3CCC(CF)(NC(C4C=CCC4)=O)C3)c12 88330,O=C1CCCC(C(N2CCCC(NC(c3cnn(C4CC4)c3)=O)C2)=O)CC1 88331,CON(C)C(=O)C(C)NC1CCCCC1n1cc(CC(C)(C)C(=O)O)nn1 88332,N1(C(C(C)C2CC2)=O)CC2(CCC(CNC(=O)Cc3ccc(Cl)c(F)c3)O2)C1 88333,c1(C(N2CC(SC)C(NC(C3(C)CCCO3)=O)C2)=O)ccc2n[nH]c(C)c2c1Cl 88334,N1(C(c2c(C)n[nH]c2)=O)CCOC2(C1)CN(Cc1cccc(C#N)c1)C2 88335,CC1CCc2[nH]c(C(N3CC(C)C(C)(C(=O)O)C3)=O)cc2C1 88336,N1(C(c2c(CC)nc[nH]2)=O)CCOCC2(COCCN2C(=O)C(O)C(C)CC)C1 88337,CC(C)C(C)CCNC12COC(C1)C2 88338,c1(C(N(CCC(=O)NC2CCSC2)CC#C)=O)ccnn1C 88339,c1(OCCN(C)C)ccc(NC(=O)NCC2CC(Cl)=NO2)cc1 88340,N1(C(CNC(CC)=O)=O)CC(NC(=O)CCN2CCC(C)CC2)CC1(C)CC 88341,CN1CCC(NC(=O)C(CN(C)C)NC(c2cncc(Cl)c2)=O)C(C#N)C1 88342,c1(NC2CCCN(C(C(C)Cc3ccccc3Cl)=O)C2)cnc(C#N)cn1 88343,C12(CC(=O)NC(CCO)C(F)F)CCC1CN(C(=O)CCC1OCCO1)C2 88344,N1(C(c2cc(CC)n(C)n2)=O)CCC(NC(C2C(C)C2C)=O)CC(C)(C)C1 88345,CC(C(C)(C)C)=CC(N1CCC(NC(=O)CCc2cc[nH]n2)C1)=O 88346,CCC(CO)C(=O)NCCC1(O)CN(C(=O)C(F)(F)C2CCOCC2)C1 88347,N1(Cc2c(OC)cc(Br)cn2)CCC(F)(F)C(NC(=O)C=CC2CC2)C1 88348,C(CCC(=O)NC1CCOC2(CCC2)C1)(C(C)C)NC(C(c1ccn(C)n1)C)=O 88349,c1(CC(=O)NCC2CCCC(NC(c3csnn3)=O)C2)nc([N+](=O)[O-])n[nH]1 88350,N1(C(C2(C)CC3CC3C2)=O)CCN(C(=O)CCCN=[N+]=[N-])C(C(F)F)C1 88351,c1(N(CC(C)C)C)ccc(C(N2CC(F)(CNC(C3CC3C#N)=O)C2)=O)cc1 88352,C1(NC(=O)C=CCN2CCOCC2)CCC2CN(C(c3cc(O)cs3)=O)CC12 88353,n1(CCCN(C)C(C2(C3CCCCO3)CC2)=O)cc(C2CCCO2)nn1 88354,O=C(CC1=CCCCC1)N1CCC(C(=O)NCc2ncco2)C12CC2 88355,C1(CNC(C(CC=C)NC(=O)C2=C(Cl)CC2)=O)CCCC12CCC2 88356,C1(CC)(NC)CCN(C(C2CCC(CO)CC2)=O)CC1 88357,CC(O)(CNC(c1conc1CNC(C1(CO)CCC1)=O)=O)C(F)(F)F 88358,c1(C(N2CCC(N(CCC)C(c3ccc(C)cc3)=O)C2)=O)cc(F)c(N)cc1F 88359,c1(CCNS(C)(=O)=O)ccccc1C(=O)NC1(C)C(C)C1 88360,C1(NC(=O)CCc2ncc[nH]2)CCC(c2cn(CCC(F)(F)CO)nn2)CC1 88361,C1(C(N(C)Cc2scc(C)c2)=O)C2CC1N(C(=O)Cc1ncoc1C)C2 88362,c1(CC(=O)NC2CC3CC(NC(C(C)OCC=C)=O)C3C2)c(C)cc(C)nc1O 88363,CN1CCN(CC23CC(c4ccccc4)(C2)C3)CC1.c12ccc(cc1)oc2=O 88364,c1(CC)ccc2c(c1)C(CC(=O)N1CCCC1CCNC(=O)C(C)(C)O)C(=O)N2 88365,N1(C(CCOCC#C)=O)CCC2CN(C(C3OCCN(C)C3=O)=O)CC12 88366,C1(CC)CCCN(C(C2CC(C#N)(OC)C2)=O)C1C(=O)NC1CCN(OC)CC1 88367,c1(N2C(=O)CC(C(=O)NCC(CN(C(=O)C(C)(C)O)C)O)C2)ccc(F)c(F)c1 88368,C1(CC(N2C(CNC(CCSCCCC)=O)C=CC2)=O)COCCN1CC 88369,C1(C(=O)NC)(CNC(C(C)OC2CCCC2)=O)CCCO1.C(COC)SC1CC1 88370,C(=O)(CS(=O)(=O)C1CC1)NC1C(C2CCN(C(C(F)=C(C)C)=O)CC2)OCCC1 88371,CN1C2CCC1CN(C(C1COCCN(C(C3CCCO3)=O)C1)=O)CC2 88372,c1(N(C(c2cnc(C)[nH]2)=O)CC2CC2)ccc(Cl)cc1 88373,C(=O)(C1CCCn2cnnc21)N1CCN(C(C(CC#C)C)=O)CC1COC 88374,CC1(C(=O)Nc2cncc(Br)c2Cl)CCCN(C(=O)CCc2cnccn2)C1 88375,c1(C(=O)NC2CCN(C(CSCCCC)=O)CC2)ccnc2c1ccn2C 88376,N1(C(Cc2c(C)cccc2)=O)CCC2CCC12CNC(c1c(C)nc(C)n1O)=O 88377,C(=O)(CS(=O)(=O)CCO)NCC1(CO)CCN(C(C(COC)O)=O)C1 88378,C(CCCC(C)NC(c1cnn(CC)n1)=O)NC(C(C)(C)OCC)=O 88379,c1(NC(C)CCc2ccccc2F)nccc(=NCC2(CCO)CC2)[nH]1 88380,c1(C(C)OC(CC(C)C)C)nc(-c2cnn(C)c2)nn1CC1CCC1 88381,N1(C(c2ncc(C)c(OC)c2C)C(=O)NCC2CC2)CCC2(C)C(F)(F)C2(C)C1 88382,C1(CCOCC)(NC(=O)C(F)CC(C)C)CCN(c2ccc(C#N)cn2)CC1 88383,N(C(=NC1CCS(=O)(=O)C1)NCC1CC(C)(C)C1)C1CC(OC)C1 88384,C#CCCCCCC(=O)NCC1C2CN(C(=O)CC(C)N(C)C)CC12 88385,S(=O)(=O)(CC(=O)NC1CCCC1Cc1ccccc1)NC(C)(C)C 88386,C1(CCNC(=O)CC2CCCSC2)CCCN(C(c2ccsc2)=O)CC1 88387,C(=O)(C1CCCc2ncnn21)N1CC(O)CC(NC(C2(C)CCCCC2)=O)C1 88388,Cc1nn(CC(=O)NC2C3CN(C(=O)C(C)CC4CC4)CC23)c(C)c1Cl 88389,Cc1cc(C(N2CC(O)(c3ccccc3)C2)=O)n2nccc2n1 88390,c1(CC(N2C(C(=O)OC)C=CCC2)=O)ccc(S(=O)(=O)NCCN(C)C)s1 88391,N1(CCC(=O)N(S(CC)(=O)=O)CC(F)(F)F)CCCC(NC(=O)CC(F)F)C1 88392,Cc1n[nH]c2cnc(C(=O)NCC(C(C)C(C)C)NC(c3nocc3Cl)=O)cc12 88393,N1(C(C(CSC)OC)=O)CC(NC(=O)CCc2cncc(O)c2)C(C2CC2)C1 88394,C1(C(=O)OC)CC(NCC(=O)N(c2ccc(Cl)cn2)C)CC(C)(C)O1 88395,N(C1CCCc2cc(CNC(=O)C=Cc3ncco3)ccc21)C(C(C)SC)=O 88396,C1(OC)(OC)CCC12CC(CNC(=O)Cc1cnn(C)c1Br)C2 88397,C(=O)(C(=O)CCC(C)(C)C)NCC1C(C)CN(C(c2cc([N+](=O)[O-])n[nH]2)=O)CC1 88398,N1(C(C=CCC)=O)CCN(C(C2CS(=O)(=O)C2)=O)CC1CC(=O)NCC 88399,N1(C(C(C(C)(C)C)O)=O)CCC2(CC1)CN(C(C1Cc3cccc(F)c3O1)=O)C2 88400,c1(C(N2C(C(N(CCCO)CC#C)=O)CC2C)=O)ccc(CC)cn1 88401,C1(C(=O)NC2(CCOC)CC2)COCCC1NC(=O)CC1CSC1 88402,Nc1ccc(C(N2CCC3(NC(c4ccoc4C4CC4)=O)CC3C2)=O)c(O)c1Cl 88403,C1(NC(CN2CCC(C)CC2)=O)CC(F)CN(C(c2cc(C(N)=O)no2)=O)C1 88404,CC(CC(F)(F)F)C(=O)Nc1ncc(C(C)(C)O)s1 88405,c1(OC)ccccc1C(C)(C)NC(=O)NCc1ncccc1C(F)F 88406,c1(C(N2C(CCCNC(C3C(C)C3(F)F)=O)CCC2)=O)cc(C(F)F)ncn1 88407,C1(OCC(=O)NC(C)CN(C(=O)CC2(CO)CCOCC2)C)CCC(F)(F)CC1 88408,c1(C(=O)NCCCN(C(C2(F)CC2)=O)C2CC2)ccc(CCc2ccccc2)s1 88409,N1(C(=O)Cn2ccc(C3CC3)n2)CCCN(C(c2n[nH]cc2[N+](=O)[O-])=O)CC1 88410,CC1=C(C(=O)N2CCC(NC(C34CCCC3C4)=O)CC2C)C(=O)OC1(C)C 88411,c1(CC(=O)NCCCN(C(c2csc(Br)c2)=O)CC)cc(OC)no1 88412,C1(OCC)CN(C(C2(CC)CC2(F)F)=O)CC1CNC(c1ncccc1NC)=O 88413,CCC(CC(F)F)C(=O)N1CCN(C(c2cscc2C(N)=O)=O)CC1 88414,N1(C(C(CCC)F)=O)C2CCC(C(N3CC4CC3CN4C)=O)C1CC2 88415,CC(Cc1cccs1)N=c1[nH]c2c(c(=NC(C)c3c(F)cccc3Cl)[nH]1)CCC2 88416,n1(C(C(=O)NCCN(CC(=O)OCC)CCNC(N)=O)C)cc(Br)cn1 88417,c1(CNC(CC2(OC)CN(C(C3OCCCC3(C)C)=O)C2)=O)ccnc(F)c1F 88418,c1(CC)[nH]nc(C(=O)NCCC(C)NC(=O)C(c2ccnn2C)C)c1[N+](=O)[O-] 88419,N#CC1(C(=O)NCc2cc(C(=O)NCCCc3cnn[nH]3)co2)CCOCC1 88420,Cc1cc(CNC(c2conc2C(C2CC2)NC(N)=O)=O)n(C)n1 88421,Cc1cn(C)nc1CON1CC(SCC(=O)O)C1 88422,Cc1c(F)cc(C(N2CCCC(N(C)C(C34COCC3C4)=O)CC2)=O)c(F)c1N 88423,Cc1nc(C(N2CCC(n3cc(CNC(c4ccnn4C)=O)nn3)C2)=O)c(C)o1 88424,c1(CC)ccc(C(=O)NCCOCCN(C)C(C2(C)CCC(F)(F)C2)=O)c(F)c1 88425,c1(N(CCC)C)ccc(C(=O)NCCN(C(C2SCCS2)=O)C2CC2)cc1 88426,C(CNC(=O)C(c1cccn1C)=O)(CC(=O)N(C1(CCO)CC1)C)OC 88427,Cc1nc(CO)sc1C(=O)NCC(C)NC(c1nc(=N)cc[nH]1)=O 88428,c1(C(N(CCOCCNC(C(C(C)O)C)=O)C)=O)ccc(F)c2ccoc12 88429,Cc1nc[nH]c1CC(=O)NC(C)(CNC(c1cccnn1)=O)C1CC1 88430,C1(NC(C2N(C(=O)OC)CC2)=O)C=CCC(C(=O)NC2CCCC2CCO)C1 88431,Cc1[nH][nH]c2ncnc(=NCC3(CNC(c4csc([N+](=O)[O-])c4)=O)CCC3)c1-2 88432,C1(O)(CNC(c2c(CNC(c3c(C)nc(CC)o3)=O)cco2)=O)CCC(C)(C)C1 88433,C=CCC(C)(C)CC(=O)NCCCCNC(c1c(C)ncnc1O)=O 88434,C1(NC(C(C=C)(C)O)=O)CN(C(c2cc3ccccc3o2)=O)C2(CCC2)C1 88435,Cc1cnc(Cl)c(S(=O)(=O)N2CCCC2CC(=O)Nc2ccnc(Cl)c2I)c1 88436,C=C(C)C1CN(C(C2C3CC3CN2C(c2cc(C(F)F)[nH]n2)=O)=O)CCO1 88437,c1(N2CCCC(C)(CO)C2)cc(Br)ccc1S(=O)(=O)NCc1ccnc(C#N)c1 88438,Cn1cnc2cc(C(N3CCCC(NC(=O)C4=CCCOC4)C3)=O)ccc12 88439,C1(C(C)C)CN(C(=O)CN2CCNC(=O)C2)CCN1C(=O)Cc1cccnc1 88440,C1(CC=C)(NC(c2csc(COC)n2)=O)CCN(C(c2cc(=O)cc[nH]2)=O)CC1 88441,c1(NC(=O)COC2CCCCC2)cccc(-c2nc(O)n[nH]2)c1 88442,N1(C(CC2(OCC)CC2)=O)CCN(C(c2cn(C3CC3)nc2C)=O)CC(C)(C)C1 88443,c1(OC)cc(C(N2CC(NC(c3cccc(F)c3C)=O)CC2C)=O)cc(N)c1N 88444,C12(C(=O)NC3CCC(NC(C4C=CCC4)=O)CC3)C3CC(CC13)C2(F)F 88445,CC1CN(C(=O)CNC(c2ccccc2)=O)CC1NC(C1(F)CC=CCC1)=O 88446,N1(C(c2c(C(C)C)occ2)=O)CC(S(C)(=O)=O)CC1(C)C 88447,N1(C(=O)OC)CC2CN(C(=O)CCn3cc(-c4ccc(SC)cc4)nn3)C2C1 88448,Cc1cc(F)ccc1C(=O)NCCC1CCCN1Cc1ccncc1 88449,C(CC(F)F)(C(=O)NC1CCCC1C#N)N(C)C.C1CCC(=O)NCCO1 88450,c1(C(N2CC3C(CNC(CCc4n[nH]c(=N)s4)=O)(C3)C2)=O)ccc2nccn2n1 88451,CC1COCCN(C(=O)CCN(C(=O)COC2(C)CCC2)C2CC2)C1 88452,N1(C(c2n(OC)cnc2C)=O)CCC2(CCOC2)C(CNC(=O)CSC(C)C)C1 88453,N1(C(C(CCOC)NC(=O)CCCCNC(C)=O)=O)CCNC(=O)C1C 88454,c1(C(=O)NC2CC(CNC(C(C)C3CCC3)=O)C2)n[nH]c2ccc(Cl)cc12 88455,c1(C(=O)NCCC2N(C(CC(C)NC(N)=O)=O)CCC2)nn(C)nc1Br 88456,C(C(=O)N(C)CC1CCOCC1)(C(C)CC)N(C(C1CCC(=C)CC1)=O)C 88457,CC1(C)CCOC1CS(=O)(=O)NC(c1cnc(CN2CC(N)C2)o1)=O 88458,Cc1cccc2c1CCOC2C(=O)N(CCCOCCC(=O)NCCNC(N)=O)C 88459,C(=O)(CC(C)(C)C(=O)OC)NCC1C(NC(CCC=C)=O)CC1 88460,C=Cn1nccc1C(=O)NCCCCC(C)NC(=O)CC1CCN(C(C)C)CC1 88461,C1(CNC(CCCC(C)=O)=O)CN(C(=O)C(C)(C)C2CCCCO2)CCC1(F)F 88462,c1(OC)coc(C(=O)NC2CC(CCNC(=O)Cn3cc(C#N)cn3)C2)cc1=O 88463,C(CC(C)(C)C)(C(=O)N1CCC(C)(C(=O)N(C)CC2(C)CCC2)C1)OC 88464,C#Cc1cccc(C(=O)N(CCN(C)C(c2cnn(C)c2Cl)=O)C(C)C)c1F 88465,c1(C(N(CC(CN(C(=O)CCC2CCCO2)C)O)C)=O)nccc2cccnc12 88466,CCCCCC(F)C(=O)N1CC(NC(=O)CCc2cnc[nH]2)C(C)(C)C1 88467,C1(NC(C2C(C#C)C2)=O)CCCN(C(C)Cc2cc(C)n(-c3ccccn3)n2)C1 88468,N1(C(CC)CC)CC(C(=O)N(C2CCC(CNC(=O)C(F)CC)CC2)C)CC1=O 88469,c1(C(=O)NCCC2(O)CN(C(CC3CC(=O)OC3)=O)C2)cc(C2CC2)ccn1 88470,C(=O)(CC(C)(C)CC(F)F)N1CC(C2(NC(C(C)NC(N)=O)=O)CC2)C1 88471,C1(NC(C(CC)NC(N)=O)=O)CCC2CC1CN2C(=O)C(C1CC1)OC(C)=O 88472,N1(C(C(CC)(F)F)=O)CCc2ccccc2C(NC(c2ccncc2Cl)=O)C1 88473,C1(C)(NC(CC2C=CC(NC(c3cc(C(C)C)on3)=O)C2)=O)CC(F)(F)C1 88474,c1(C(C)=O)[nH]c2ccccc2c1C(=O)NCC1CC1F.C12CCCC1NC2=O 88475,Cc1ncnc(C(=O)NCC(CC2CC2)C(=O)NC2(c3nn[nH]n3)CC2)c1C 88476,C12(NC(C(C)C3CCCC3)=O)CCC(CNC(=O)CN3C(=O)CCC3=O)(C1)OC2 88477,C(=O)(C(O)CC(C)(C)C)NCC1C(CC)CN(C(=O)C2=C(Cl)CC2)CC1 88478,C1(NC(=O)CC2CN(C(c3coc(Br)n3)=O)C2)CCc2ccc(O)cc2C1 88479,N1(C(C2CCC(n3cc(C4CC4)nn3)C2)=O)CCCc2cc(OC(F)F)ccc21 88480,CC(C(=O)N1CC(CCNC2(C(N3CCOCC3)=O)CC2)C1)S(N)(=O)=O 88481,C1(C)(c2cn(CCc3ncn(C)n3)nn2)COCCN1C(=O)Cc1nc(=N)[nH][nH]1 88482,C(=O)(C1CCCc2ncnn21)N1CC(N(C)C(c2csc(S)n2)=O)C1 88483,C(CC(C(C)(C)C)NC(=O)CC1CN(C(C)=O)C1)N(C(C(COC)(C)OC)=O)C 88484,c1(C(N(CCCN(C(=O)CCc2ccnc(Cl)c2)C)C)=O)cnn2ccn(C)c12 88485,C(=O)(C(C)(C)C(C)C)NCCC(N1CCC(N(C(CCCOC)=O)C)C1)=O 88486,c1(COC(CC2ON=C(CC)C2)=O)ccc2c(c1)CCCO2 88487,c1(OC)ccc2c(c1)CC(C(=O)NCC(C)(CO)NC(=O)C1=CCOC1)O2 88488,c1(N(CC(C)C)C)ccc(C(=O)NC2CC(C)(NC3CCCN3C(C)C)C2)cn1 88489,C(=O)(CCC(=O)N1CC(N(C(=O)CCCOc2cccnc2)C)C1)NCCC 88490,Cc1cc(C(N2CCCC2(C(=O)N(C(CO)C2CC2)C)C(C)C)=O)nc(O)c1 88491,c1(CCN(C(=O)CNC(=O)CN(C)CC2(CO)COC2)C)ccccc1 88492,N1(C(C(C)n2ccnc2)=O)CCC(O)C(NC(c2cc(=O)cc(Cl)[nH]2)=O)C1 88493,CCCCC(CC(=O)N1CCC(CO)C12CC2)NC(=O)CCC(C)(C)F 88494,S(=O)(=O)(c1ccc(NC2CCC(CO)C2)cc1Cl)NCCc1nc(C)sc1 88495,N1(C(C(CC)N(CC)CC)=O)CCCC(NC(C2CC2C2(F)CCC2)=O)C1 88496,N1(C(CCCOCCC)=O)CC(C(=O)NC(CF)C(F)(F)F)C(F)(F)C1 88497,C1(CNC(=O)CCCc2ccccc2)CCN(C(c2ccc(O)c(O)c2)=O)CC1O 88498,CC1=C(C(=O)N(C)CCC2CCN(C(C3(C(=O)N(C)C)CC3)=O)CC2)SCCO1 88499,C1(C(=O)NCc2ccc(Cl)s2)C=CCN(C(C2CCCCO2)=O)C1 88500,C1(NC(COCCOC)=O)CC12CCN(C(=O)Cc1cnc(C)s1)C2 88501,C1(C)(NC(CC2C(C)CCN(C(C3CNC(=O)O3)=O)C2)=O)CC(C)(C)OC1=O 88502,C1(NC(CC(C)(C)C2CC2)=O)CCCN(C(c2ccc(Br)c(O)n2)=O)CC1 88503,Cc1cnccc1C(N1CCC(NC(=O)COC(c2nccn2C)C)C1)=O 88504,c1(C(c2n(CC)nnn2)NCCN2CCOC2=O)cc2nccc(Cl)c2s1 88505,C1(NC(c2cncnc2)=O)C(CC2CC2)CCN1C(=O)CCC1CC1 88506,C(=O)(CCC(F)(F)C(=O)N1CCN(C(C2C=C2C)=O)CC1COC)OCC 88507,Cc1cccc2c1OCC2C(=O)N1CC(CCCCNC(=O)CCOC(C)C)C1 88508,c1(SCCOC)cccc(NC(N2CCCC(CC3CCOC3OC)C2)=O)c1F 88509,C1(C(=O)NCCCCCCN(C(CCC2CC(C)C2)=O)C)Cc2ccncc2N1 88510,C(C(CC(C)C)NC(=O)Cc1ccc(C)cc1)NC(C1(NC(C)=O)CC1)=O 88511,C1(C(N(CCN(C(CC2ON=C(CC)C2)=O)C)C)=O)Cc2cc(C)ccc2S1 88512,N1(Cc2cnc(CCC)s2)C(C(N2CCOC3(CC3)C2)=O)CC2CCCCC12 88513,c1(-n2cc(CC(C(=O)NC(C(CCCOC)C)=O)C)nn2)cccc(C#N)c1C 88514,C(C)(C(C(=O)Nc1cnn2ccccc12)C(C)C)NC(C1C(C(C)=O)C1(C)C)=O 88515,C(CC1CCCCC1)(C(=O)NCCCCCN(C(=O)C=Cc1cscn1)C)OC 88516,N1(C(C(CCOC)(C)C)=O)CCC2CC(NC(C3(O)CCSC3)=O)CCC2C1 88517,Cc1cn2c(n1)CC(C(=O)NCC(C(C)C)NC(c1cc(C3CC3)[nH]n1)=O)CC2 88518,C1(OCC(=O)NCC2(CC(=O)OC)CC2)CCN(C(C2(C)CCOC2)=O)C1 88519,c1(C(N2CCC(C)(NC(CN(CCOC)C)=O)C2)=O)[nH]c2ccc(Cl)cc2c1Cl 88520,CCC(C(=O)NCC(=O)NC(c1cn(C)nn1)C)NC(C)=O 88521,c1(C(N(CCOCCN(C(c2cn(CC=C)nn2)=O)C)C)=O)cc[n+]([O-])cc1 88522,c1(OC)ccc(Br)c(F)c1S(=O)(=O)N1Cc2ccccc2C2(CCC2)C1 88523,N1(C(=O)NCCc2c(C)ccc(Br)c2)CC(C2CCCCC2)CCC1C 88524,C(CC(=O)N1CCCC1C(N1CCCC1)=O)(C(N)=O)N(C)C(C)=O 88525,C1(CNC(COC)=O)CN(C(=O)COc2cccc(C#N)c2)C2(CCC2)C1 88526,C1(CC)(NC(c2cc(CNC(C3CC(C)(C)C3)=O)on2)=O)CCCC1 88527,c1(C(=O)NC(CNC(CC(C)OC)=O)(C)Cn2cccn2)cccc(N)n1 88528,c1(SC)c(C(=O)NC(C(=O)NOCC(C)(C)O)C2CCOCC2)cnn1C 88529,C(=O)(C(CC=C)CC(C)C)NC1(CC=C)CCN(C(c2cccnn2)=O)CC1 88530,NS(=O)(=O)c1ccc(C(=O)NC2CN(C(=O)C(O)C(F)F)C2)cc1F 88531,CCC(C)(CNC(C1COCC(C)O1)=O)C(=O)N(C1CCN(C)C1)C 88532,c1(OC)ccc(NC(=O)CCC2CCN(C(C3CC3F)=O)CC2)cc1C 88533,N1(C(C(COC)C)=O)CCN(C(c2nc(Cl)c(Cl)s2)=O)CC(C)(F)C1 88534,Cc1cc(C(N2CCC(c3ccncc3)CC2)C(=O)NC2CCC2)nc(Cl)c1Br 88535,C#CC1(O)CC(C(N2CCCC2CNC(c2ncccc2Br)=O)=O)C1 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88553,C(=O)(CCC(F)(F)CN=[N+]=[N-])N(CCNC(C1CCc2nn[nH]c2C1)=O)CC 88554,n1(CCCSCC)nnnc1C(C(C)(C)C)NCC(C)C1CCC1 88555,c1(C(N2CCC(NC(c3ccc(O)nn3)=O)CC2)=O)cc2cc(F)ccc2o1 88556,C1(C)(N(C(C=CCN(C)CC)=O)C2CC2)CN(C(=O)CCCF)C1 88557,C(=O)(CC(C)CC(=O)N(C(C)C(=O)NCC(F)C1CCC1)C)OC 88558,c1(C(N(C(C)CCNC(=O)CCc2cncc(O)c2)C)=O)cccn2nncc12 88559,C1(NC(C(c2ccnn2C)C)=O)CCCC1NC(=O)CCCn1cncn1 88560,n1(CCNC(=O)NCC(C)CN(C)C(=O)OC(C)(C)C)cccc1C=O 88561,c1(C(N2CCC(N(C(C3(C4CC4)CC3)=O)CC)C2)=O)cccn2c(C)cnc12 88562,N1(C(CC(C(CC)C)O)=O)CC2(CCN(C(=O)CC3CC(F)C3)CC2)C1 88563,Cc1cc(CNC(=O)NC2CCC(C(=O)O)CC2)c(F)cc1Br 88564,c1(C(C(=O)NCC2CCOC2)N(CCSC)CC)ccc(OC)c(C)n1 88565,CN1CC2(CC2)CC1C(=O)NOCC(N1CCC1C1CCC1)=O 88566,S(=O)(=O)(C1CCS(=O)(=O)C1)NC1CC(CNC(=O)NC2(F)CC23CCCCC3)C1 88567,C(CCC(=O)NCC(O)C(=O)NCC1(CF)CC1)OCC 88568,N1(C(c2nc(C)sc2C)=O)CCN(C(c2csc3nccn23)=O)CC(C)(F)C1 88569,C1(C(N(C2CN(C)CC2O)C)=O)CC(O)CCN1C(c1nccnc1N)=O 88570,N1(C(CN(C)C(N2CCOCC2)=O)=O)CCCC(C2(Cc3ccccc3)CC2)C1 88571,c1(CC)ccc(CN(C)Cc2nc(CO)n[nH]2)cc1 88572,N12CC(CC1(C)C)CC2=O.C(=O)(C(F)C(C)(F)F)NC1CC(N(C)CC)C1 88573,Cc1[nH]nc(C(=O)N(C(C)C(=O)N2CC(C(C)(C)O)C2)C)c1O 88574,C1(NC(C(C(C)C)c2cnn(C)c2)=O)CN(C(c2ns[nH]c2=O)=O)CC12CC2 88575,C(=O)(CCCC(C)(C)C)NC(C1CN(C(c2ccc(NC(CC)=O)cc2)=O)C1)C 88576,C(=O)(C1=CCCCC1)NC1CC(NC(=O)Cn2cc(Cl)cn2)C(O)C1 88577,CN1CC(C(N2CCC(C(=O)Nc3cncc(Cl)c3)(CO)C2)=O)NC1=O 88578,C1(CNC(c2cccc(CC)c2)=O)CC2(CO1)CN(C(=O)C(C1CCC1)OC)C2 88579,c1(N(C)CC2COC(=O)O2)nc(N2CC3CC2C3)c2cnn(C)c2n1 88580,C1(NC(c2c(C)nn[nH]2)=O)CN(C(c2ccc(-c3ccc(Cl)cc3)[nH]2)=O)CC1C 88581,CC(C)C(CCNC(C12CC(CN1C1CC1)C2)=O)NC(C1(C)CCCC1O)=O 88582,Cc1[nH]c(=N)ccc1C=CC(=O)NCCC(C)NC(C1CCCC12CC2)=O 88583,C1(CNC(C2CCC2(F)F)=O)CC2(CCN(C(c3cccc[n+]3[O-])=O)CC2)CO1 88584,C(=O)(C1=CCOC1)NC(C)CCCNC(c1cn(C2COC2)nn1)=O 88585,C12(C(N3CC(N(C)C)(C(N)=O)C3)=O)CCNCCCC1C2 88586,C#CCCCC(C)C(=O)N1CCN(C(c2cnoc2C)=O)CC1CCCC 88587,Cn1nc(Cn2c(N3CCCC(F)CC3)nnc2-c2ccccc2)c2c1CCC2 88588,c1(OC)ccccc1OCCC(=O)NCC1CC(NC(C2COCC(C)O2)=O)C1 88589,c1(NC(=O)NC2CCN(Cc3cccc(OCC)c3)C2)nc(C)c(Br)c(Cl)n1 88590,N1(C(C2C(C)C2)=O)CCCC(N(C(=O)CCC2CCCOC2)CC2CC2)C1 88591,c1(OC)ccc([N+](=O)[O-])cc1NC(=O)C(N1CCN(C)C(C)C1C)=O 88592,C1(C(N(C)CCC2CCCCN2C(c2cncc(Cl)c2)=O)=O)CCC(C)(C)CC1 88593,n1(CC(=O)OC)cccc(NC(C2CCC(O)(C(F)(F)F)CC2)=O)c1=O 88594,c1(CC(=O)NCC2N(C(C(N3CCC(O)CC3)C)=O)CC2)cccc(F)c1F 88595,CCCC(C)(CCC)C(=O)NCCC12CCC1CN(C(C1(C)CCSCC1)=O)C2 88596,C(c1ccsc1Br)=CC(=O)NC1CCC(CNC(c2ccoc2Cl)=O)C1 88597,N1(C(Cc2c(C(C)C)con2)=O)CCN(C(C)CNC(C2CCC(O)C2)=O)CC1 88598,N1(C(C(C(C)C)n2cnnc2)=O)CCN(C(c2cncc(F)n2)=O)C2(CCC2)C1 88599,C(C(C)(C)CC(=O)N(C1CCCN(C(c2cc(C#N)cs2)=O)C1)C)N(C)C 88600,c1(C(N2CCN(C(Cn3c(C)cc(C)n3)=O)CC2)=O)ccc(C(=O)O)c(F)c1 88601,C=C(C)CN=C(NCC1=CCCC1)NCC(N1CCN(C(C)=O)CC1)(C)C 88602,N1(C(c2cc(OC)ncc2)=O)CCN(C(C2CC(CCF)C2)=O)C(C2CC2)C1 88603,C(=O)(CC(CC)CC(F)(F)F)N1C(CN(C(CC(=O)NCC)=O)C)COCC1 88604,N1(C(CNC(c2n(C(C)C)ccc2)=O)=O)CCN(C(=O)CN(C)C(N)=O)CC1 88605,C12(NC(c3c(C)con3)=O)CCC(CN(C(C3(CO)CCOCC3)=O)C1)C2 88606,C12(C(N3CC(NC(CSC(C)C)=O)C(CC4CC4)C3)=O)CCCCCC1OCC2 88607,C(CC(CC)C(=O)NC1CCCN(C(c2ncccc2C(F)F)=O)C1)=CC 88608,C(C(=O)N1CCC(CN(C(=O)Cc2ccc(Br)s2)C)C1)(C(C)C)OC 88609,C1(OC)(CNC(=O)COCC2CCCO2)CCN(C(c2ccccn2)=O)C1 88610,N1(C(Cc2nc(CCP(C)(C)=O)sc2)=O)CC2(CCCN(C(=O)CC#N)C2)C1 88611,C1(C(N(CC#CC)C(C)C)=O)C2CC3C(C2NC(=O)CC2CC(SC)C2)C13 88612,C1(F)(C(N2CCC(NC(c3cc(CN4CCOCC4)on3)=O)C2)=O)CC=CCC1 88613,c1(NC2CC(NC(NCc3cncc(C)c3)=S)C2)ncnc2ncc(Br)cc12 88614,N1(Cc2cc(OC)c(C)cc2)CCCC(C2CCCN(C(c3cn[nH]c3)=O)C2)C1 88615,Fc1ccc(CNC2(c3nnnn3CC3CC3)CCOCC2F)c(F)c1C(F)F 88616,Cc1ccc(NC(=O)CC2CN(Cc3cc(F)c(O)c(Br)c3)CCO2)c(Cl)c1O 88617,CCC(CCN1CCCCC1)(c1nnnn1C1CC1)NCCC1CCCOC1 88618,O=C(C1=C(F)CN(C(C2CN(C3COC3)C2)=O)CC1)NCC(F)CO 88619,n1(CCCC)nccc1C(=O)NC(C1CCN(C(=O)C(O)C2CC2)C1)C 88620,N1(C(C2C(NC(C=CC=CC)=O)CCCCC2)=O)CCCN2CCCC2C1 88621,c1(C(N(C(C)CNC(C2SCCS2)=O)CC)=O)ccc(C)o1 88622,C1(CNC(c2cnc(SC)[nH]2)=O)CN(C(=O)Cc2nnc(S)n2C)CC12CC2 88623,C(C(C)(C)CC(=O)N1CCN(CCNC(C2(C3CCC(C)(C)C3)CC2)=O)CC1)OC 88624,CC(C)(O)C(F)(F)C(=O)N1CC2(CC(C(=O)NC(CC3CC3)C3CC3)CO2)C1 88625,N1(C(c2cnn(CCC)c2Cl)=O)CCN(C(=O)C(F)n2cccn2)C(CCO)C1 88626,N1(C(C)C(=O)NC(C)CNC(=O)CC(C)c2cnn(C)c2)CCC(O)CC1 88627,CCC(C)C(O)CC(=O)NCCN(C)C(c1ccn(-c2ccccc2OC)n1)=O 88628,CC1CC(NC(=O)CCC2CCC2)CN1C(c1cc(-c2ccoc2)ccn1)=O 88629,c1(C(C(=O)NC(CC)CNC(=O)C(C)O)(C)C)ccc(F)cc1 88630,C1(NC(c2c(OC)cc(I)cc2)=O)CC2CN(C(C3C=CC(=O)N=N3)=O)CC2C1 88631,Cc1ccc(CC(=O)NCC2CC3CN(C(C4CCSCC4)=O)CC23)c(Cl)n1 88632,c1(CSC)ccc(C(=O)NC(c2ccccc2)CNC(c2n[nH]cc2CO)=O)o1 88633,N1(C(c2cn(CC)nc2)=O)CC(C2CC2)(C(=O)NC(c2cccc(C)n2)C)C1 88634,Cc1cc(C)c(C=CC(=O)NCC2CCC2NC(c2cnc(Cl)[nH]2)=O)cc1C 88635,N1(c2c(C(=O)OCC)c[nH]n2)CCC2(CC1)CN(C(=O)C(C)SCC)CC2CO 88636,C1(CCC)CN(C(=O)CSC(C)(C)C)CCN1C(c1ncn(C(C)C)n1)=O 88637,C1(C(N2CC(NC(c3ccc(C(C)(C)C)[nH]3)=O)C2)=O)C2CCC(F)(F)C12 88638,c1(OCCC)ccc(C(N2CCC(CN(C(=O)Cc3ccon3)C)C2)=O)cc1 88639,N1(C(Cc2[nH]c(=N)sc2)=O)CC2CCN(C(=O)CC3CC4(C3)CC4F)CCC2C1 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88797,C(CO)(CCCCNC(=O)CCN1C(=O)CCC1=O)NC(C(C)(C)C1CC1)=O 88798,c1(C(=O)NCCN(C(CCCCC#C)=O)CCC)c(C)ccc2nsnc12 88799,c1(OC)cccc(Cl)c1CNC(=O)C(=O)NCC(c1ccc(Cl)c(Cl)c1)N(C)C 88800,Cc1c(C(N2CCSCC2C(=O)NCCc2ccncn2)=O)oc2ccccc12 88801,c1(C(=O)NC2C(C)CN(C(c3ncc(F)cn3)=O)CC2)cccc2c1ncn2C 88802,N1(C(C2COCCN(C(c3ccns3)=O)C2)=O)Cc2ccncc2C1 88803,c1(C(=O)NCC23CC(CN2C(C2CCC=CO2)=O)C3)cc2occc2s1 88804,C(CNC(=O)C=CC(F)(F)F)(C(C)C(C)C)NC(C(c1cc(C)sc1)(F)F)=O 88805,N1(CCCC(=O)NCCNC(c2c(C(C)(C)C)con2)=O)C(=O)CNC1=O 88806,N1(C(CN(C(C)=O)C)=O)CC(C(=O)NCC2(F)CCC2)CC(C)C1 88807,N1(C(C2(OC)CCC2)=O)CC2CC(NC(C3CC4(CCCC4)CO3)=O)CC(C2)C1 88808,Cc1cocc1C(N1CCCC1CNC(c1n[nH]c(C(C)(C)C)n1)=O)=O 88809,N1(C(CCCN(C(C)C)C)=O)CC2(CCC2NC(c2ccc(F)cc2C(F)F)=O)C1 88810,CC(CN=c1ncc2ccccc2[nH]1)N(C(=O)C1=CC2CCCC12)C 88811,c1(C(=O)NC(COC)(C)C)cnc2c(-c3cc(C)nnc3N)cccc2c1 88812,c1(C(N(CC(C)O)CCNC(=O)Cc2cc[nH]n2)=O)cccc2c1OCC(=O)N2 88813,C1(CNC(C(C2CCCCC2)OC)=O)CN(C(C2C=CC=CC=C2)=O)CCN1C 88814,C1(CNC(C(C)(C)C2CCOCC2)=O)CCCCN(C(=O)C(F)OC(F)(F)F)C1 88815,c1(CNC2C(C(N(C3CCOCC3)CC)=O)CCC2)ccc2ccc(Cl)cc2n1 88816,C1(N(C(Cc2c(C)cccn2)=O)C)CN(C(C2CC3CCC2CC3)=O)CCC1C 88817,N1(C(c2cc(OC)ns2)=O)CCCC(N(C(=O)CN2CCC2C)CCF)C1 88818,C1(C)(OC)CC(NC(c2ccc(CNC(=O)C(C)SC)nc2)=O)C1(C)C 88819,C(C(CO)C(C)(C)C)NC(CC1CC(NC(CCCN(C)C)=O)C1(C)C)=O 88820,c1(N(C(C2CCC(C(C)C)C2)=O)CC2CCN(C)CC2)ccc(F)c(F)c1 88821,C1(C(N2CCC(c3ccc(F)cc3)CC2)=O)CC2CC2N1C(=O)CN1CCCCC1 88822,C1(CC(=O)NCCC2(C(N3CC(O)(c4cc[nH]n4)C3)=O)CCCC2)COCC1O 88823,N1(C(c2c(CC)occ2)=O)CC2CCC1C(NC(=O)CCCC(N)=O)C2 88824,C(=O)(C(F)CC(C)(C)NC(=O)CN(C)C)NC(CC(C)O)C 88825,c1(C(=O)NC2CC(NC(C(COC)(C)C)=O)C2)cc(OC(F)F)cc(F)c1 88826,N1(C(CC(C)N(C(c2cncc(C)c2)=O)C)=O)CC(C(C)C)CCC1C 88827,C(CN=c1[nH]c(=NCC2(F)CCC2)c2c(F)cccc2[nH]1)NC(=O)NCC(C)C 88828,C1(CCOC)(NC(COCC(=C)C)=O)CCN(C(=O)C(CCSC)NC=O)C1 88829,C1(CC(=O)NC2C(C(N)=O)CC=C2)C2CN(C(c3ccnn3C3CC3)=O)CC12 88830,Cn1ncc2c(N3CC4CC3CN4c3ncncc3F)ncnc12 88831,C(C)(CCCCC#N)(N(C(C)CCCCCCO)C)C1CC1 88832,c1(CC(N2C(CNC(CCCC#CC)=O)COCC2)=O)c[nH]c2cccc(C)c12 88833,c1(-n2cc(CN)nn2)cccc(C(C)C)c1.N1(CC)CCOC(CC(=O)NC)C1 88834,C(c1ccccc1)=CC(=O)NCCOCC(=O)NCCCCN(C)C 88835,C1(NC(C(C#N)C2CC2)=O)CCCC12CN(C(c1sccc1OC(F)F)=O)C2 88836,Cc1nc2cccc(C(N3CC(N(C(=O)CCS(C)=O)C)C3)=O)c2[nH]1 88837,c1(C(C)(F)F)ccccc1C(=O)NC1CC(C)(NC(c2csc(=N)[nH]2)=O)C1 88838,n1(COC)nccc1C(=O)NC(C)CC(C)NC(=O)CC1CCCC1 88839,Cc1n[nH]c(C)c1CC(C)CNC(=O)C(CNC(=O)OC(C)(C)C)CO 88840,CC1CCc2[nH]nc(C(=O)NCC(C)N(C)C(c3cc(O)cs3)=O)c2C1 88841,C12(NC(C3N(C)CCCC3)=O)CCC(C(=O)NCC3CCC(O)CC3)(CC1)C2 88842,C1(C(N2CC(C)(CCC(=O)N(CC(CCC)O)C)C2)=O)CC12CCOC2 88843,N1(C(C2(C#N)CCCC2)=O)CCC2CCN(C(C3(CO)CC(F)(F)C3)=O)CC2C1 88844,c1(C(N2CC3C(CNC(=O)C=C4CCSCC4)(C3)C2)=O)cn2ccccc2n1 88845,N1(Cc2ccc(C)cn2)CCc2cccc(C(=O)NCc3ccccc3C)c2C1 88846,C1(C(=O)NC(c2nccn2C)CC)CCCN1C(=O)C=Cc1ccc[nH]1 88847,N1(C(CCC)=O)CCCC1Cc1cn(CCCNS(=O)(=O)C2CC2)nn1 88848,C1(C#N)(C(N(CCCCN(C(=O)CCCC(C)(C)C)C)C)=O)CC2CCC1C2 88849,C(=O)(C1=NOC2COCC12)N1C(CN(C(c2c(C(C)C)nns2)=O)C)COCC1 88850,C(CN=c1[nH]ccnc1F)(C1CC1)NC(c1cn(C(C)(C)C)nc1)=O 88851,CC1CN(C(C2C3CN(C(C4CC(O)C4)=O)CC23)=O)CC(C)O1 88852,N1(C(CC2CC(=C)C2)=O)CCN(C(C2(C)CC3CCC2C3)=O)CC(O)C1 88853,N1(C(C2(OC)CS(=O)(=O)C2)=O)CCCCC(CNC(c2cc[nH]n2)=O)C1 88854,C1(C(=O)NCCOCC2CC2c2ccccc2)CNC2(CCC2)C1 88855,c1(OCC(N2CCC(n3cc(CC=C)nn3)CC2)=O)c(F)cccc1Cl 88856,C1(NC(C(CN(C)C)N(C)C)=O)C(C)(C)C(NC(=O)C2=COCCC2)C1(C)C 88857,Cc1cccc(CC(N2CCCCC2C(C)(C)C)=O)c1F 88858,c1(OC)ccc(F)c(C(c2nnnn2C2CC2)NC2(C#N)CCOCC2)c1 88859,C(=O)(C=C1SCC(=O)N1C)NC1(CNC(c2ccc(C#C)cc2OC)=O)CCC1 88860,CC1(C)CN(C(c2cccc(N)c2F)=O)CC1NC(C1CCC2(CC2)C1)=O 88861,N1(C(CC(C)c2ccco2)=O)CCC2(CCC2)C(NC(=O)C(=O)NCC(F)F)C1 88862,C(C(=O)N=c1ccn(C)[nH]1)C1(C)N(C(CC(CCCC)CC)=O)CCC1 88863,C1(C(=O)NC(C2(C(=O)NC(Cc3ccco3)CO)CC2)C)CC(F)CN1C 88864,c1(C(=O)NCC(CC)(CC)NC(CC(CCC)O)=O)cc2cccnc2cc1F 88865,Cc1cc(Cl)ccc1CC(=O)NCC12COC(CNC(=O)Cc3ccco3)(C1)C2 88866,c1(C(N2C(COC)C=CCC2)C(=O)Nc2ccccc2)cc(Br)cnc1Br 88867,N1(C(c2cnc(CCC)s2)=O)CC(NC(C2CC2[N+](=O)[O-])=O)CC12CCCC2 88868,CC1(F)CN(C(C2CCCN2C(=O)C2CC2)=O)CCN(C(=O)C(O)CF)C1 88869,CCC(CN=c1[nH]c2c(c(=NCCCCN3CCCC3CO)[nH]1)CSC2)N(C)C 88870,N1(C(C2CCCC23CC3)=O)CC2(CCN(CC(O)COc3ccccc3F)C2)C1 88871,CC1ON=C(C(=O)N(C)CCC2CCN(C(=O)CCc3ccnn3C)CC2)C1C 88872,Cc1nc2cccnn2c1C(N1CC(N(C(=O)C(N2CCC(C)CC2)=O)C)C1)=O 88873,CC1(C)CN(C(C2CC3(CCC3)C2)=O)CCN(C(C2CC2(F)Cl)=O)C1 88874,C=C=C(C)CC(=O)NC(CNC(=O)C(c1ccccc1OC)OC)CC=C 88875,c1(CCC(=O)NC2CCN(C(Cc3c(C)noc3)=O)C2)cncc2ccccc12 88876,C(=O)(C#CC1CCCCC1)N1CCC2(CC(NC(CCCCCC=C)=O)C2)C1 88877,CCC(C)(CNC(=O)CCc1cscn1)NC(c1coc(C)n1)=O 88878,N1(C(C2CCCC(OC)C2)=O)CCCC2(C1)CN(C(=O)Cc1ccc(F)cn1)C2 88879,C1(NC(c2cccc(CO)c2)=O)CC12CCN(C(=O)C1=COCC1)C2 88880,c1(C(=O)NC(CNC(CCc2onc(C)n2)=O)C(C)(C)C)cc(C#N)ccc1N 88881,CCC(CC)C(=O)N1CCOC(C(=O)NC2CC(O)C(O)C2)C1 88882,N1(C(C(N2CC(C=CC)C2)=O)=O)CC(C)CC(C)C1 88883,CCC(C)C=CCOC(C1CC(Br)C1)=O 88884,C1(CNC(CC(=C)C)=O)COCCN(C(C2CCN(c3cccnc3)CC2)=O)C1 88885,c1(C(N2CCC(C(C)(C)NC(C3C(C)(CC)C3)=O)C2)=O)cnn(C)c1Cl 88886,C1(NC(C2CC(N=[N+]=[N-])C2)=O)C2CC(CN(C(=O)C=CC3CC3)C2)C1CO 88887,Cc1ccc(O)cc1C(N1CCCCCC1C(=O)NCC(c1cn(C)cn1)O)=O 88888,c1(CNC(N(C(C2CCCO2)C)C)=O)ccc2nccnc2c1 88889,C1(CN(C(C2C(C=C)C2)=O)C)CCCN(C(=O)C(C)(Cl)Cl)C1 88890,c1(C(=O)NC2CCN(C(=O)NC3(CC(=O)OC)CC3)C2)ccnc(C)n1 88891,C1(CN(C(C(C)=CC)=O)CC)CCN(C(C2(Sc3ccccc3)CC2)=O)CC1 88892,N1(C(C2(CNC(C3C(C)(C)CCCO3)=O)CC=CC2)=O)CCC2(C=CCO2)C1 88893,C1(C(=O)NC(c2csnn2)C)N(C(=O)C2=CCCC2)CCC1(C)C 88894,N1(C(CC=C)=O)CC2(CCC(NC(=O)CCOCC(F)(F)C(F)(F)F)CC2)C1 88895,c1(NC(C2C(NC(C=CC)=O)C2)=O)cc(Br)ccc1F 88896,c1(OC)ccc(F)c(C(=O)NCCOC2CN(C(=O)COC3(C)CCC3)C2)c1F 88897,Cc1nn(C)cc1NC(C1(NC(c2c[nH]c(C#N)c2)=O)CCSC1)=O 88898,c1(CCOC)ncc(CC(=O)NCC2(CNC(=O)CCC3CC3)CC2)[nH]1.C(=O)(N)N 88899,N1(C(C2CC3(CC(=O)C3)C2)=O)CCCC1C1CCCN1C(=O)Cn1nnnc1S 88900,C(C(C)C)(C(O)C(=O)N1CC(C)(C(=O)NCCC2CCCC(C)C2)C1)OC 88901,C1(CC)CN(C(=O)C=Cc2ccnn2C)CCN1C(=O)CC(C)N1CCCC1=O 88902,c1(N(C(=O)NC2C=CC2)CC)ccccc1 88903,c1(C(=O)NCC(CNC(c2ccc(C)nc2)=O)C)cc(Cl)ccc1O 88904,CC1CCC(C(=O)N(CCC(C)(C)O)C)CN1C(=O)CC1CCC(=O)N1 88905,C(=O)(C1=C(Cl)CCCC1)N1C(C(=O)NC2CC(CO)C2)(COC)C=CC1 88906,c1(CC)ccc(NC(=O)COC2CN(C(C=CC(=O)NC)=O)C2)c(C)n1.N(C)C 88907,c1(OCCC(=O)N(CC(C)O)CCNC(=O)Cn2cncn2)ccccc1F 88908,C(=O)(C1=CCC(F)(F)CC1)N1CCC(n2cc(-c3cncc(N)c3)nn2)C1 88909,c1(C(N2CCC3C(NC(C(CC)OCC)=O)C32)=O)cnn2cccc(Cl)c12 88910,O=C(CC1=CCCC1)NCc1cn(C2CCCN(C(C3CCCCS3)=O)C2)nn1 88911,C12(CNC(C=CC)=O)CCCC1N(C(c1ccc([N+](=O)[O-])cc1)=O)CCC2 88912,Cc1ncccc1CCC(N1CCCC(NC(c2ccncc2Cl)=O)C1)=O 88913,C(=O)(NNc1ccc(Br)cc1)Nc1nc(OC)cc(OC)c1 88914,c1(OC)cnncc1C(=O)OCc1cccc(NC2COC2)c1 88915,c1(CNC(c2n(C(CC)C)nnn2)(C)COC)cc(F)ccc1Cl 88916,c1(C(=O)NC)ccc(C(=O)NCCCCC(C)NC(=O)CCn2ccnn2)cn1 88917,C(=O)(N1CCC(C(=O)NCCCn2cnnn2)O1)c1cc(OCC)no1 88918,C1(C2CCN(C(c3cnoc3)=O)C2)(NC(C(CC)OC)=O)CC1 88919,c1(C(=O)NC2CC(F)(CNC(C(CC)(C)C#N)=O)C2)cc(F)cc2nn[nH]c12 88920,C1(C(N2CCC(CCCC)C2)=O)CCN(C(=O)CCCCC(C)=O)CC1(C)C 88921,Cc1cc(O)c(C(N2CCC(NC(=O)C(c3ccc(C)s3)C)C(O)C2)=O)nn1 88922,N(C1CCOc2ncccc21)C(=O)C(C1(O)CCCC1)F 88923,C1(CC)(NC(=O)CC(C)C(C)C)CCCN(C(c2csc(Br)c2C)=O)C1 88924,Cc1cc(CCC(=O)NCC2CC(C(=O)NC3(c4cccnc4)CC3)C2)no1 88925,c1(N(C2CCS(=O)(=O)C2)C(C)=O)ccc(CNC(=O)NC2CC2C)cc1 88926,CC1CC(c2ccsc2)CN1Cc1sc(Cl)cc1Br 88927,Cc1ccccc1COCC(C)N(C(=O)C(N1CCCC(n2ncnn2)C1)=O)C 88928,C(=O)(C#CC1CCOCC1)N1C(C)CCC(NC(c2cnc(OC)nc2C)=O)C1 88929,C1(NC(CC(CCC)C)=O)CCN(C(c2ccccc2CO)=O)CCC1(F)F 88930,c1(CNC(C2C(OCC)C2)=O)ccccc1CNC(c1coc(C#N)c1)=O 88931,CC(C)(C)CCC(F)C(=O)N1CC2COCC2(C(=O)NOC2CC3CCC2C3)C1 88932,C12(C(=O)NC3CN(C(Cc4ccc(C)cc4C)=O)C(C)C3)CCCN(CCC1)C2 88933,c1(C(=O)NC2CC(CNC(C(C)NC(c3ccoc3)=O)=O)C2)cccnc1O 88934,CC(O)C(C(=O)NC(CNC(=O)Cc1ccccc1SC(C)C)C1CC1)N(C)C 88935,C1(NC(C=CC(CC)=CC)=O)CCN(C(=O)COCc2nccn2C)C(C2CC2)C1 88936,C1(C(N2CC(OC(=O)NCC)C2)=O)(OC)CCN(C(C2CC(C)CCO2)=O)C1 88937,C(=O)(CC(CC)C(=O)OC(C)(C)C)NCC1OCCN(C(CCCCC)=O)C1 88938,C(C1CCC1)=CC(=O)NCC=CC(=O)N(C(C)CC1CC1)C 88939,CP(C)(=O)C1(C(=O)NC2CC(NC(=O)CC3CCC(=O)NC3)C(O)C2)CC1 88940,C1(NCC(CC)(C)Sc2ccccc2)CC2(c3ccccc3)CC1C2 88941,c1(NC(=O)NC2CCN(C)C2c2ccccc2)ccc(Cl)c(Cl)c1Cl 88942,c1(C(N2CCC(N(C)C(C3CC(F)C3)=O)C2)=O)ccc2nn(C)cc2c1 88943,C1(NC(CSc2cc(C)ns2)=O)CCCC(NC(c2cccc(CF)c2)=O)C1 88944,CCC(C)C(C)C(=O)NCC1(F)CC(CNC(c2c(Br)c(C)nn2C)=O)C1 88945,C(=O)(C#CC(C)(C)CNC(C1CC1CC)=O)NC(CC)C 88946,N1(C(C2CN(c3c(C)cccc3)C(=O)C2)=O)CCC2(CCOCC2)C1 88947,CCCC(C)N=c1[nH]c(=NC2CC(N3CCOCC3)C2)c2sccc2[nH]1 88948,C1(C(N(CCN(C)C)CCN)=O)COCCN(Cc2ccc(O)cc2F)C1 88949,c1(OCCCNC(c2n(CC=C)nnn2)C2(CC)CC2)cccc(C)c1C 88950,C(=O)(C(C)CC(C)CC(C)C)NC1CN(C(c2c(OCC)cccn2)=O)CC1(C)C 88951,CC#CCCCC(=O)N(C(CC(F)F)C(=O)N1CCC(C(C)CO)CC1)C 88952,C(CCC(CO)NC(C1CC1C1CCCO1)=O)NC(CCC=CC(C)C)=O 88953,CC(C)CCN=C(NCC(C)(C)F)N1CC2C(=O)NC(=O)C2C1 88954,Cc1cc(C)n2cnc(C(N3CC(N(C(=O)Cc4cccc(F)c4)C)C3)=O)c2n1 88955,O=C(CCCC#Cc1ccccc1)NCC1CCN(C(c2sc(F)cc2Cl)=O)C1 88956,CC1CCN(C(=O)C(CC(F)F)NC(C2CC3CC(=O)C2O3)=O)CC1(F)F 88957,Cc1c(C(=O)NC(C)CCCNC(=O)CC2(C)OCCO2)sc(Cl)c1Cl 88958,C(=O)(Nn1ccccc1=O)C1(CNC(C2C3CC(=O)C(C3)C2)=O)CCCO1 88959,Cc1scc(C(N2CC(NC(=O)Cn3nnnc3C3CC3)C(C)C2)=O)c1N 88960,N1(C(C=NOC)=O)CCC2C(CCCN2C(=O)CCc2nc3ccccc3[nH]2)C1 88961,c1(C(=O)NC2(C)CCN(C(=O)Cc3ccsc3Cl)C2)ccnc2ccccc12 88962,C1(CNC(c2nc(C(C)OC)sc2)=O)CN(C(c2cc(CC3CC3)on2)=O)CC1O 88963,CC1=CCCN(c2cc(N3CCN(C)CC3)ncn2)C1 88964,C1(n2cc(NCCN(C(C)(C)C)C(C)=O)nn2)CN(C(=O)CC2(C)CC2)CC1C 88965,C(=O)(C1=COCCO1)N1C(COC)(CNC(c2[nH]cc(C)c2C)=O)CCC1 88966,n1(CCCCNC(C(=O)NCCC(N2CCOCC2)C)=O)cc(Br)cn1 88967,C(C(C)(C)C(=O)NCC1(C2CCC2)CC1)N(C)C.C12CCCC1NC2=O 88968,CC(C)CC(C)(C)C(=O)NCC1CCCN1C(C12CC(CO1)C2)=O 88969,c1(N2CCC(C(C)NC(=O)CSCc3ccc(F)cc3)C2)nc(C)nc(C)c1F 88970,C(=O)(CCC(C)(C)c1ccccc1)NC(C(C)C)C(C)NC(=O)Cc1cn[nH]c1 88971,C(C)(N=c1[nH]c(N2CCOC(C(N)=O)C2)nc(=N)[nH]1)c1scc(C)n1 88972,c1(OC)cccc(CNC2CCC(C(N3CCOC4CC34)=O)C2)c1Cl 88973,C(=O)(C(COC)CC(C)C)N(CCC)CCNC(C1CCCCC1(F)F)=O 88974,C(c1ccc(OCCF)cc1)=CC(=O)NCC(C1CC1)NC(C12CCC1CC2)=O 88975,c1(C(N2CCC(CNC(c3n[nH]c4ncccc34)=O)C2)=O)c(F)ccc(O)c1F 88976,C12(C(=O)NCC3(NC(C(n4cc(C)nc4)(C)C)=O)CC(OC)C3)CCCCC1C2 88977,C1(C(N2CCCC(C)(OC)C2)=O)(OC)CCC(C)(C)C1.C12CCCCC1C(=O)N2 88978,C1(NC(=O)CC2CC2)CCOC12CCN(C(c1csc3c(Cl)cccc13)=O)CC2 88979,c1(C(=O)NCCCCCNC(C(C)C)=O)nc(C(F)(F)F)n2c1CCCC2 88980,C(CCC(=O)NC(C1CN(C(=O)CC2CNC(=O)O2)C1)C)OCC 88981,Fc1cc(OC(F)F)cc(-c2nc(-c3ccoc3)nn2CCN2CCC2)c1 88982,C(=O)(C1CCCc2nccn21)N1CCN(C(CNC(C2(C)CCOC2)=O)=O)CC1 88983,c1(C2C(CC(=O)NCCCN(C(c3cnsc3)=O)CC)C2)cccc(F)c1 88984,N1(Cc2[nH]ccc(=O)c2)CCCN(CCCc2ccccc2)CC1 88985,Cc1c(C(=O)NCC2CCC(NC(c3nocc3C(C)(C)C)=O)C2)cnn1C 88986,c1(C(=O)NCC(CC(C)C)NC(=O)CSC(F)F)cc(=N)[nH]c(Cl)n1 88987,CN1C2CCC1CC(C(=O)NCC1CCCN(C(C3CCC(C)(F)CC3)=O)C1)C2 88988,C1(CC)CCOC1C(N1CCCC1CNC(c1cnc(C(C)(C)C)[nH]1)=O)=O 88989,N1(C(C(F)=CC)=O)CC2CCC2(CNC(c2cc(Cl)c(Br)[nH]2)=O)C1 88990,c1(OCC(=O)NCCCCC(C)NC(CC2CC(SC)C2)=O)ccc(C)cc1F 88991,N1(C(CN(C(c2cccc(OC)n2)=O)CCO)=O)CCC(O)C(C)(C)C1 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89009,Cc1cc(C(=O)NC2CC(O)CN(C(c3cc(CO)cc(Cl)c3)=O)C2)ncc1F 89010,Cc1cc(N)c(C(N2CCN(C(c3cc(F)n[nH]3)=O)CC2C(C)C)=O)cc1C 89011,C(=O)(C1CCCc2ccccc21)N1CC(C)N(C(c2cccc(O)n2)=O)CCC1 89012,C1(NC(C(C(=O)OC)C)=O)CN(C(=O)CCN2CCCS2(=O)=O)CC12CC2 89013,N1(C(CCC=CC)=O)Cc2ccccc2C1C(=O)Nc1cncc(C(F)F)c1 89014,N1(C(CS(CC)=O)=O)CC2CCC1CN2C(=O)C(C(C)(C)C)c1ccc(C)cc1 89015,c1(-c2nc(NC(C3(C(=O)NC(C)C)CC3)=O)sc2)cccc(C#N)c1 89016,c1(NCC(N2CCC(C(C)NC(CN3CC(C)C3)=O)C2)=O)ccc(O)cc1 89017,C1(CNC(C(CC)(C)COC)=O)CC2(CCC2)CN1C(=O)C=C(C)c1cccs1 89018,c1(N2C(C)(CNC(C(C)(C)O)=O)CCC2)nc2c(F)cc(Cl)cc2s1 89019,c1(C(=O)NC2(CC=C)CN(C(C3(c4cc[nH]n4)CC3)=O)C2)cccc(C(N)=O)c1 89020,C(=O)(C(CC)CC(C)C)NCC1C(NC(CN(CCC#C)C)=O)C1 89021,CN1CC(C(=O)NC(CC2CCC2)C(=O)NCC2(C(C)(F)F)CC2)CCC1=O 89022,c1(C(=O)NCCN(CC(C)O)C(C2CCC2)=O)cc2sc(Br)cc2[nH]1 89023,N1(C(CCc2cc(OC)no2)=O)CC(CCNC(=O)C(C)N2CC(C)C2)C(C)C1 89024,C1(NC(CC2C(C)C2)=O)CC2(C1)CC(NC(c1ncoc1C1CC1)=O)C2 89025,C1(CC(=O)NCc2ccc(C(=O)NCC3(CO)CCOC3)o2)CC2(CC2)C1 89026,c1(C(=O)NCC(CN(C)C(c2cn(CC3CC3)nn2)=O)O)csc(C#N)c1 89027,C1(C(=O)NC2CC3(C(NC(CCc4ccn(C)n4)=O)C3)C2)CC2(CCOCC2)C1 89028,Cn1cc(Cl)c(C(=O)N(C2CC3CC2CN3)C2CCC(O)C2O)n1 89029,c1(CC(=O)N(CC(C)NC(C2C(C)(C)C2(C)C)=O)CC)ccc(OC)c(F)c1 89030,C1(CC(=O)NC2CCC(CC)CC2)C2CCCC2N1C(c1ncncc1OC)=O 89031,C12(CNC(C(C)N(C(=O)Cn3ccnc3C)CCC)=O)CCCC(CO1)C2 89032,C(=O)(N=c1cc(Cl)cn[nH]1)C1C(NC(c2cc(C)ncc2)=O)C1 89033,N1(C(c2ccc(SC)cc2)=O)CC2(C)CC1C2CNC(=O)Cc1ccc(C)nc1 89034,c1(OCC)cc(N2CCC(C(C)NC(=O)C(C)(C)O)C2)ncn1 89035,C1(C(N(C)CCN(C)C2CC2)=O)C2CC1N(C(C1CN(C3COC3)C1)=O)C2 89036,C(=O)(C(C)(N)C(F)(F)F)NCc1n(CC)nnc1C 89037,N1(C(C(C)n2cnnn2)=O)CC2(C1)CN(C(c1c[nH]cc1C1CC1)=O)CCO2 89038,C1(CNC(c2cc(C)ncc2C)=O)N(C(=O)C(F)=C2CCCC2)CCCC1(C)C 89039,c1(C(=O)NC2C(NC(C=C(C)C(F)F)=O)C2)oc(Br)nc1C 89040,C1(C(N2CCCN(C(Cc3ccc(C)s3)=O)CC2)=O)CCCCN(C)C1=O 89041,CS(=O)C=CC(=O)NCC1CC(NC(=O)Cn2cc(Br)cn2)C1 89042,C1(C#N)(CC(N2CC(C(C)NC(=O)NCCCl)C2)=O)CCOCC1 89043,N1(C(COCC(C)C)=O)CCC(O)(CN(C)C(C2CCCN2C(C)C)=O)C1 89044,c1(C(=O)NCCCC(C)NC(CCC)=O)cc2ncccc2[nH]1 89045,C1(C)(CC)CC(NC(c2c[nH]nc2OC)=O)CN1C(=O)Cc1ccnn1C 89046,C1(C(=O)NCC2(CNC(c3c(N(C)C)ccnc3)=O)CCC2)CCCCNC1=O 89047,c1(N(C)C)cncc(C(=O)NC2CC(NC(C3CC(n4ccnc4)C3)=O)C2)c1 89048,C1(C(C(=O)OC)N(C(C)C)CCOC)CC2OC(C)(C)OC2C1.C(CC1CC1)SC 89049,N1(C(C(CC2CCC2)OC)=O)CC2CC(C1)N2C(=O)Cc1ccc(Cl)cc1 89050,c1(C(=O)NC2C(NC(c3cc(SC)oc3C)=O)CC2)cc(O)nc(C2CC2)n1 89051,c1(NCC)ccc(F)c(C(=O)NCCN(C(=O)C(CC)NC(N)=O)CC(C)O)c1 89052,CCC(C)(CCC(C)C)C(=O)N1CC2CN(Cc3c(OC)cccc3Cl)C2C1 89053,C1(NC(C(C)OCC#C)=O)CCC(N(C(=O)C(F)CC2CCCCC2)C)CC1 89054,c1(C(=O)NCCCCC#C)ccc2c(c1)CN(C(C1CCN(C(=O)OC)C1)=O)C2 89055,c12cccc(c1)NC(=O)NC2CF.C1(C)(C(=O)OCC)CC(C(=O)OC)C1 89056,CC(CC(=O)NCC1CCN1C(=O)C(C)(C)C(N)=O)C(F)(F)F 89057,n1(CC)c(C(=O)N(C(c2ccccc2)CNC(C2(F)CC2C)=O)C)cnc1O 89058,C#CCC(CC(=O)Nc1cc(OC)cc(Cl)c1)NC(C1CCN(C)C1)=O 89059,CN1Cc2cc(NC(=O)NC3CCc4ncnn4C3)ccc2C1=O 89060,C(=O)(CCN=C(NCC1CCN(S(C)(=O)=O)C1)NC1CCOCC1F)NC 89061,c1(C(C)OC)nc(C(=O)NC2CC(CCNC(=O)C(c3ccccc3)O)C2)cs1 89062,c1(C(N2CCN(CC(O)C(C)(C)C)CC2)C(=O)NCC)nccc2ccccc12 89063,C1(CNC(CC(=O)NCC#C)=O)CCCN(C(C2CC(C)CCO2)=O)CC1 89064,C1(C(N2CC(O)(CN(C(CCOC)=O)C)C2)=O)CCC(C)(C)OC1 89065,c1(OCC(=O)NCC(CCNC(C2CC(C)(F)C2)=O)O)c(F)cccc1F 89066,N1(C(C(C=CC)O)=O)CCCC12CCN(C(C1CC(=O)CCO1)=O)C2 89067,c1(C(=O)NC23CN(C(Cn4c(C)cc(C(F)F)n4)=O)C(C2)C3)ccc(F)c(F)c1 89068,S(=O)(=O)(c1ccc(NCC2(C)CCC(=O)N2)c(F)c1)N1CCC(CC=C)C1 89069,C1(C(=O)NCc2ccc(C)s2)CC(N=[N+]=[N-])CN1C(=O)C(F)C1CCC1 89070,C#CC1(NC(=O)C(C)N(C(C2CCN(C)CC2)=O)CC)CCOC1 89071,N1(C(c2csc(CC3CC3)c2)C(=O)NC2CCC2)CC(O)CC(F)C1 89072,CC1(C)CC(C(=O)NC2CCCC2CNC(C2(Br)CC2(C)C)=O)=NO1 89073,C1(CC)CN(C(=O)CCc2cc(C)n(C)n2)CCN1C(=O)COc1ccncc1 89074,Cc1cc(C(=O)NC(C2CN(C(c3cnn(C)c3C3CC3)=O)C2)C)cc(N)c1O 89075,c1(C(=O)NCc2ccc(C(N3CC(O)(CO)C3)=O)cn2)n[nH]c2c1CCC2 89076,CCCCC(CNC(=O)CCOCc1ccccc1)NC(=O)C(O)CC 89077,c1(C(N(C2CC(NC(=O)CC3CCOC3C)C2)C)=O)n[nH]cc1NC=O.CCO 89078,C1(CNC(C(C(CC)O)C)=O)CCC2CN(C(c3nc(C)sc3C)=O)CC12 89079,C#Cc1cccc(C(=O)NCC2(O)CCN(C(C3CC3C3CC3)=O)CC2)c1F 89080,N1(C(=O)NCC)CCCC(C(=O)NCC2(OC)CN(C(C3(CC)COC3)=O)C2)C1 89081,C(CC#CC)(C(=O)NOCC(=O)N(C)C)NC(Cn1ncc(C#C)c1)=O 89082,CC(C)(CCF)C(=O)NC1CC(O)(CNC(C2CC(CC3CC3)C2)=O)C1 89083,c1(C(=O)NCC2COCCN2C(=O)Cc2cccnc2Cl)ccn2ccnc2n1 89084,N1(C(C2(F)CN(C(c3nc(COC)oc3)=O)C2)=O)CC(OC)C(O)C1 89085,O=C1OC2CC1N(C(=O)CCC1CCCCO1)C2 89086,c1(CC)nc(CNC(C2(NC(C3CC(=O)CS3)=O)CC(O)C2)=O)n[nH]1 89087,C1(C(C2CCN(C(C3CCCN3CCn3ccnc3)=O)CC2)=O)CCC2CCCC12 89088,C(CC1=CCN(C(C2CCc3ccnn3C2)=O)CC1)NC(C(C)(O)C1CC1)=O 89089,C(=O)(CCC(=O)NN(C)C)N1CC(C)N(C(=O)COc2cccnc2)CC1 89090,c1(C(=O)OC)ccc(F)c(C(N2CCN(C(c3cc(Cl)c[nH]3)=O)CC2CF)=O)c1 89091,c1(C(=O)NC2CC(NC(C3C4CC5C(C4=O)C35)=O)C2)ccc2c(n1)CCO2 89092,Cc1c(C(=O)NC(C(C)(C)N(CCO)CC)c2nnnn2C2CC2)cccc1Cl 89093,c1(-c2n(CC)c(N3CCC(CCCCS(C)(=O)=O)C3)nn2)cc(C)n(C)c(=O)c1 89094,N1(C(CC=C(C)C)=O)CCOC(CNC(=O)CC23COCC(C2)C3)C1 89095,Cc1cc(C)c(C(N2CC(N3CCN(C(C4CC(F)C4)=O)CC3)C2)=O)[nH]1 89096,N1(C(C2CN(C(C)=O)C2)=O)CCCC1(C)CNC(C1CC(=O)N(C2CC2)C1)=O 89097,C(=O)(CC(C)C(F)(F)F)NC(CCN(C(CCCCOC)=O)C)C 89098,C1(O)(C(=O)NC2CC(C(N3C(C)(C(=O)OCC)CCC3)=O)C2)CCOC1(C)C 89099,Cn1c(C(N2CC(CNC(C3CC(C)(C)CO3)=O)C2)=O)cc2sccc12 89100,C(=O)(C(CCNC(C1(C2CC2)CCCO1)=O)OC)NC1(COC)CC1 89101,c1(OC)nc(C)ccc1C(=O)N(CCCn1cc(C2(OC)COC2)nn1)C 89102,N1(C(CCc2c(C)nn(C)c2)=O)CC(NC(=O)CC=C(Cl)Cl)CCC1C 89103,C(c1c[nH]c2ccccc12)=CC(N1CCCC(C)CC1)=O.c12cccn1C(=O)S2 89104,C1(CC(=O)N(CC#C)CC=C)CCN(C(=O)C(C)C2CCC2)C1(C)C 89105,c1(C(C)C(=O)N(C2(CC(=O)C(C(C)COC)=O)CC2)C)cnn(C)c1.N(C)C 89106,C(=O)(C(C)(CC)OC)N1CC(CC=C)(C(=O)NCC2(COC)CC2)C1 89107,C1(NC(=O)CCc2nncs2)CC2(C1)CC(C(N1CCC(CO)C(O)C1)=O)C2 89108,N1(C(c2c(C)ncn2C)=O)CCC2(CCCN2C(c2cncc(Cl)n2)=O)C1 89109,CC1CN(C(=O)COc2ccccc2)CC(C)C1NC(=O)CCCN=[N+]=[N-] 89110,C1(C(N2CCC(CCNC(C3(CO)CC(F)(F)C3)=O)C2)=O)CC2CCCC(C1)C2 89111,c1(-c2cn(Cc3csc(C(CC)N4CC4)c3OC)nn2)ccc(F)c(C)c1C#N 89112,c1(NC(CCC)C)ncnc(NCCc2ncccc2C)c1C 89113,Cc1ncc(C(=O)NCC2CCCCN(C(c3cncs3)=O)C2)cc1N 89114,c1(C(=O)NC(CC)CN(C)C(C2CCCO2)=O)c[nH]c2c(Cl)cccc12 89115,N1(C(CC2ON=C(C(=O)OC)C2)=O)CCOCC(C)(CNC(C2(C)CCC2)=O)C1 89116,Cc1cc(NC(c2ccoc2CNC(C2(CO)CC(C)(C)C2)=O)=O)cnc1C 89117,C1(C(=O)NCC(CO)NC(C2(C=C)CCCCC2)=O)CNC(=O)CC12CCC2 89118,C1(NC(c2cnc(COC)s2)=O)CC2CC1CN2C(c1cn(C)c(C)n1)=O 89119,Cc1csc2ncc(C(=O)N(C)CC3CC(F)CN3C(=O)CC3(C)CC3)n12 89120,C=C=C(C)CC(=O)NC1CCC(N2CCN(C(=O)C(C)c3cc[nH]n3)CC2)CC1 89121,Cc1cc2c(C(N3CCSCC3CCNC(C34CC(C)C3C4)=O)=O)cccc2o1 89122,c1(NCC2CCCN(CC)C2)[nH]c(=NCCCC2CCCO2)nc2c1ncn2C 89123,Cc1nc(C)n(CCC(=O)NCC2(C(C)(C)O)CN(C(=O)CC(F)(F)F)C2)n1 89124,N1(C(C2CC3(C2)CC(F)C3)=O)CC2CCCC(C1)N2C(C1(O)CCCCCC1)=O 89125,n1(CC(=O)NC2ON=C(C(=O)OCC)C2)nnc2c(OC)ncnc12 89126,N1(C(C(COCC)(C)C)=O)CC2(CC)CC1(CNC(C1CC(C3CC3)C1)=O)C2 89127,C1(C(=O)NCC2(F)CC(NC(C3(CF)COC3)=O)C2)CCCCCC1 89128,c1(NC(C2(OC)CCN(C(C(CCCOC)C)=O)C2)=O)cn(C)c(=O)nc1O 89129,c1(OCCC)ccc(C(=O)NC2CC2NC(=O)C(CC)SCC)cc1 89130,N1(C(c2ccncc2O)=O)CCCC2C1CCN2Cc1ccc(F)c(F)c1Cl 89131,C(CCCC(=O)NC1(CN(C)C(C2(OC)CC2)=O)CC1)OCC 89132,C1(NS(CC(C)N(C)C)(=O)=O)CCC2COCCC2(C#N)C1 89133,CC1(C)CC(C(=O)NC2CCC2NC(=O)Cc2ccc(Cl)cc2)C(C)(C)O1 89134,CC(C)C(CNC(=O)CP(C)(C)=O)C(=O)NC(C)(CO)C(C)(C)O 89135,c1(CC)nn(C)c(Cl)c1C(N1CCC(O)(CNC(=O)C(F)(F)CN(C)C)C1)=O 89136,CC12CC(C(N3CC(=C(F)CNC(C4C5CCCC45)=O)C3)=O)(CCO1)C2 89137,c1(CC(=O)N(CCCCCNC(CN2CCC(C)CC2)=O)C)ccc(Cl)cc1F 89138,C1(CNC(C2(COC)CCCCC2)=O)CC2(CO1)CN(C(=O)C(C)COC)C2 89139,c1(OC)cc(CNC(=O)CC2(C)CN(Cc3cc(CO)ccc3O)C2)ccc1F 89140,c1(C(=O)NCC2C3CN(C(=O)CC4CC=CCC4)CC23)cc(O)ncn1 89141,Nc1cc(Cl)cc(Cl)c1C(=O)NCCC(O)CNC(c1cnc(C2CC2)[nH]1)=O 89142,c1(C(N2CCC(CNC(c3c(C)n(C)nc3)=O)C2)=O)cc(Br)cc2nc[nH]c12 89143,c1(OC)ccc(C(F)(F)F)c(SC)c1.c1(CN(CC=O)C(C)(C)C)occc1SC 89144,c1(C(=O)NCCN(C(COCCC#C)=O)CCCN(C)C)cnnc(O)c1 89145,C(=O)(CCCCCC(c1c[nH]c(C(=O)OC2(C)CC(CC)C2)c1)=O)NCC=CC 89146,C1(C(=O)NC2CC3COCC3C2)C2CC(C(O)C2O)S1(=O)=O 89147,CCC(C)N(OC)C(=O)C12CC(CN1C(C1CCCC(C#N)C1)=O)C2 89148,c1(C(C)C)nccn1CC(=O)NCC(O)CN(C)C(C1CC1C(C)(C)C)=O 89149,CC(C)C(C)C(CNC(=O)Cc1c(Cl)cnn1C)NC(=O)COCC1CCC1 89150,C(C(=O)NNC(=O)Cn1cccn1)(c1ccc(O)cc1)OCC 89151,CC(C)C(C)(CNC(=O)C(C)Oc1ccc(F)cc1)NC(=O)C=Cc1cocn1 89152,N1(C(=O)Cc2ccccc2)CC(C(F)(F)F)CCC1Cc1cn(CCCF)nn1 89153,Cc1cccc(CCCNC(c2nc[nH]n2)C)c1 89154,c1(C(=O)NC2(CO)CN(C(c3nccc(Cl)c3F)=O)C2)ccc2ocnc2n1 89155,C(=O)(C1=CCc2ccccc21)NC1C(NC(C(c2ccc(Cl)cc2)C)=O)C1 89156,c1(C(=O)NCC(CC)(C)NC(C2C=CCC2)=O)ccc(C#CC2CC2)cc1 89157,C1(S(N)(=O)=O)(C(=O)NC(C(C)NC(C2CCCC(=O)N2)=O)CO)CCC1 89158,C(=O)(CCCN1C(=O)C(=O)c2cccc(Cl)c21)N(CCCCNC(CCC)=O)C 89159,c1(OC)ccc(O)c(NC(=O)C(CCF)NC(=O)CCCCCN(C)C)c1 89160,C1(CC)CN(C(c2occc2CNC(=O)C(n2cc(C)cn2)C)=O)CC(=O)N1 89161,c1(C(=O)NC(C2CCCN(C(=O)C=CS(C)=O)C2)C)cc(C(C)(F)F)ccc1Cl 89162,C1(NC(=O)Cc2ccccn2)CCC2CN(C(=O)CCCCC(F)(F)F)CC2C1 89163,c1(C(=O)NC2(CC=C)CN(C(C3(OC)CCOCC3)=O)C2)cnc(S(C)(=O)=O)s1 89164,c1(C(F)F)n[nH]c(=NC2CCN(C3CN4CCC3CC4)CC2)s1 89165,N1(C(CSCC#C)=O)CC2(C(N3CCOC(CCF)C3)=O)CCC1CC2 89166,N1(C(c2cncc(C#C)c2)=O)CCC2CN(C(c3cccc(OC)n3)=O)CC12 89167,C1(n2cc(COCP(C)(C)=O)nn2)CCCN(C(=O)CN2CSCCSC2)C1 89168,N12CC(CC(O)C1)C2=O.n1(C2(C(=O)OCC)CCC2)cc(COC)nn1 89169,CC1C(NC(C2CC(O)C2)=O)CC2CCC1N2C(C1(CO)CCC1)=O 89170,Cc1c(NCCn2cc(Br)cn2)ncnc1N1CCCNC(=O)C1 89171,N1(C(CC2CC(OC)C2(C)C)=O)CC=C(C(=O)Nc2cnn(C(C)(C)C)c2)C1 89172,C1(NC(c2ccc(COC)o2)=O)CCCCC1NC(C1CCCC1C(F)(F)F)=O 89173,C(CC(C(C)(C)C)NC(c1cc(F)cs1)=O)N(C(c1c(CC)n(C)nc1)=O)C 89174,C1(CNC(Cc2cccc(OC)n2)=O)CCC2(CCC2)C1NC(=O)C1CC1 89175,N1(C(c2cc(F)ccc2F)=O)CC2CC(C1)CN(C(C1CC=CCO1)=O)C2 89176,C1(CC)CCC(F)(C(=O)OC)CC1.c1(CN2CC2OC)ccc(F)cc1 89177,c1(C(C)C)cc(C(=O)NCCOCCNC(C2COC(C)(C)CO2)=O)ccc1F 89178,C1(NC(C(CC)O)=O)C=CCCC1C(=O)NCC1CCCC12CC2 89179,c1(C(=O)NC23C(CCN(C(C4(CC)CC4)=O)CC2)C3)cc(O)nc2c1CCCC2 89180,CC(O)CC(=O)NCC1(C(=O)NCCCC2CCCC2O)CC1 89181,C1(N(C(C(C)C2CCCC2)=O)C)C2CN(C(=O)CCc3ccc(N)cn3)CC12 89182,Cc1cc(F)c(C(=O)NC2CC(C)(NC(c3ccnc4c3CCC4)=O)C2)cc1F 89183,C1(C(N(CC(=O)OCC)C)=O)CCN(C(=O)C(N2CCOC2=O)C)C1 89184,c1(C(=O)NC2C(NC(C3C(=C)C3)=O)C2)cncc(NC(C2(O)CC2)=O)c1 89185,N1(C(C2C(CC)CCC2)=O)CCC(C2(O)CN(C(c3c[nH]nc3CC)=O)C2)CC1 89186,c1(C(=O)NCC2CC(NC(C(C(C)O)N(C)C)=O)C2)ccc(C2CC2)c(F)c1 89187,c1(C(N2CC(C3(NC(C4CC(C)OCC4)=O)CC3)C2)=O)ccnc2c1ncn2C 89188,Cc1c(C(=O)NC2(C)CN(C(C3CCCN3C)=O)C2)cccc1Br 89189,c1(C(=O)NCCNC(Cc2c(C)ccc(F)c2)=O)cccc2c(C)ccnc12 89190,Cc1c[nH]cc(C(=O)NC(C(C)NC(c2cn(C)nc2C(F)F)=O)C(C)C)c1=O 89191,c1(C(N2C3CC(NC(c4n(CC)nnc4)=O)C3CC2)=O)cccc2c1ncn2C 89192,N1(C(CC(=O)OC)=O)CCC(CC(N)=O)(NC(=O)Cc2ccsn2)CC1 89193,C(=O)(C1CCc2cccc(F)c21)NCC(C1CC1)NC(c1c(C)noc1C)=O 89194,CCC(CCCC(=O)N(CC(O)(CC)CC)C)NC(=O)CC1CCCC(=O)C1 89195,N1(C(c2c(C)n(C)nn2)=O)CCC(F)(CNC(c2cc(C(F)F)[nH]n2)=O)CC1 89196,N1(C(c2n(CC)nc(C)c2)=O)CCC2CCC(NC(=O)C=CC3CCCN3C)C12 89197,N1(C(CS(=O)(=O)NC)=O)CCCC(C2CCN(CC(N)=O)CC2)C1 89198,N1(C(=O)OC(C)(C)C)CCC(C)(CC(O)C(=O)Nc2cccs2)C1 89199,N(C1CCCc2ccoc21)C(C1(NC(C(CC(C)(C)C)F)=O)CC1(C)C)=O 89200,Cc1cc(=NC(=O)N2CC(O)CCC2CO)[nH]n1-c1ccccc1 89201,c1(C(N2CCC(NC(C=CCC)=O)(CO)C2)=O)nc2ncccn2n1 89202,C1(C)(CNC(C(c2cn(CC)nc2)=O)=O)CCCN1C(=O)CCOCC(F)(F)F 89203,C1(CNC(C2(CCCC)CC2)=O)C=CC(NC(c2coc(Br)c2)=O)C1 89204,N1(CC2CCC(C)O2)CCc2cnccc21 89205,C1(C(=O)NC(C(C)NC(C=Cc2ccc(CC)cc2)=O)C)CCn2nnnc2C1 89206,N1(C(C(CC=C)CC)=O)CCCCC2C1CCCN2C(=O)Cc1cncnc1 89207,N1(C(=O)CCSC(F)(F)F)CCC(CNS(=O)(=O)CC2CCOC2)CC1 89208,c1(CCN2CCC(N)C2)ccc(OC(F)F)cc1F.CC(CCO)C1CCNC1 89209,N1(C(CCC(CC)OC)=O)CC2CCCC2(NC(c2c[nH]nc2Cl)=O)C1 89210,c12cc(ccn1)NC2=O.N1(CCN(CCC(=O)O)C)CCCCCC1 89211,c1(C(=O)NC2C(NC(=O)Cc3cccc(OC(F)F)c3)C2)c[nH]c2ncccc12 89212,C(=O)(CCC(C(C)C)NC(C1(C)CC(=O)C1)=O)Nc1ccc(C#C)nc1 89213,C1(CNC(C2CCC(OC)CC2)=O)CCN(C(=O)C(C)NC(=O)C2CC2)C12CC2 89214,C1(CC(=O)NCC2N(C(CCCN(C(=O)OCC)C)=O)CC2)CCCC1(F)F 89215,N1(C(c2[nH]n(C)c(=O)n2)=O)CCC(F)C(NC(C2CCCN(C(N)=O)C2)=O)C1 89216,c1(C(C)NC(=O)C(=O)N(C)CC2CCOC2C)cccc(Cl)n1 89217,N1(C(C2(C)CC=C(C)CC2)=O)CCN(C(C2(C#N)CCCOC2)=O)CC(O)C1 89218,c1(C(N(C2CCCC(NC(C3CC(=C)C3)=O)C2)C)=O)cnn2cc(C)cnc12 89219,O=CN1CCCC1C(N1CC2C(CNC(c3csnc3Cl)=O)C2C1)=O 89220,Cc1c(Cl)sc(Cl)c1C(N1CC2CC(NC(=O)CCc3ncc[nH]3)C1C2)=O 89221,C1(NC(C(C)Cc2cnn(C)c2)=O)CC2CCC1N2C(c1ccc(=O)n(C)c1)=O 89222,c1(C(=O)OC)c(N(C2CC2)Cc2cccc(C)c2)nc(SC)nc1C 89223,CCCCCCC(C)C(=O)NC(CNC(=O)COC(C)(C)C(F)(F)F)C(C)C 89224,N1(CC(=O)NCC2N(C(C(C)OCCN(C)C)=O)CC2)CCC(C)(C)C1 89225,CC1CCCn2c(C(N3CCCC(N4CC(O)C4)C3)=O)cnc21 89226,C1(NC(c2n(C)ccc2)=O)CCCCC1NC(c1ccncc1F)=O 89227,N1(C(C2C(CC)CCC2)=O)CC2CCCC(C1)N2C(c1ccc2cnsc2c1)=O 89228,C12(C(=O)NC3CCCN(C(c4ccc(NC)c(F)c4)=O)C3)CCCCN1CCC2 89229,N1(C(=O)NCCC(N2CCCCC2)=O)CC(O)CC(F)(F)C1 89230,C1(NC(C2(NC(c3nccc(C)c3N)=O)CCCC2C)=O)C2CCC3C(C2)CC13 89231,c1(C(C)OC)nc(NC2(CO)CCCN(C(=O)C(C)C(C)COC)C2)cc(Cl)n1 89232,N1(C(=O)Cn2cnnc2)CC2CCC(C1)N2C(=O)CCc1cncc(F)c1 89233,CC1CCN(C(C2CN(C)CCN(C)C2)=O)CCN1C(=O)Cn1ncccc1=O 89234,c1(C(C(=O)NC2CCCCN(C(CC(=O)NCC)=O)C2)C)cc2ccccc2o1 89235,CC1CN(C(=O)NCCCCc2ccc(F)cc2F)CC(C)S1(=O)=O 89236,C1(NC(c2c(Cl)cn(C)n2)=O)CN(C(C2CC(S(C)(=O)=O)C2)=O)CC2(CCC2)C1 89237,c1(C(N(C)CC2C3CN(C(CC(C=C)C)=O)CC32)=O)noc2ccc(F)cc12 89238,N1(C(C2=C(C)CC2)=O)CCCC1C1CCCN1C(C1CCc2nc[nH]c2C1)=O 89239,C1(COCC(=O)OC)CCCN(C(c2cc(N)cnn2)=O)C1 89240,Cn1cnc2cc(CC(=O)NC3CC4(C3)CC4NC(=O)CSS(C)(=O)=O)ccc12 89241,C1(NC(CCc2c(C)nn(C)c2)=O)COCCN(C(=O)C=CC2CCCC2)C1 89242,C(C#Cc1ccccc1)N1CC(C)C(NC(=O)CCCC(N)=O)C1 89243,C(=O)(C1=NNC(=O)CC1)N1CCN(C(C=Cc2cc(OC)ns2)=O)C2C1C2 89244,C1(C(N2CCC(CNC(c3onc(COC)n3)=O)C2)=O)CCCCNC1=O 89245,O=C(CC(C(F)F)NC(=O)CN1CCCC1)NC1CC2OC1C1CC21 89246,c1(C(=O)NC2CC(N(C(CC(C=C)C)=O)C)C2)cnc(O)n(C2CC2)c1=O 89247,C1(NC(C=COCC)=O)CN(C(=O)Cc2ccc(O)cc2)CC1N=[N+]=[N-] 89248,C1(C(=O)NC2CC(C)(NC(C(C(C)C)C)=O)C2)CC(F)(F)C1(C)C 89249,c1(C(=O)NC(CCN(C(c2nccc(C)c2O)=O)C)C)cc2cccc(F)c2o1 89250,C#CCC(O)C(=O)NC(C)(C)CNC(=O)C(=Cc1ccccc1)NC(C)=O 89251,C12(NC(C3C(C)=CCS3)=O)CCC(CC1)N(C(c1c(C3CC3)noc1C)=O)C2 89252,c1(C(N2C(CCOC)CN(C(C3SCC=C3C)=O)CC2)=O)cccc2nc[nH]c12 89253,CC(C(=O)NCCCN(C(=O)C(c1ccc(Br)s1)C)C)C(F)(F)F 89254,c1(CNC(c2[n+]([O-])ccc(OC)c2)=O)ccc2c(c1)CN(C(=O)C(C)C(C)O)C2 89255,C1(CC(=O)NC2C(C)N(C(=O)Cc3csc(=N)[nH]3)CCC2)SC2=NCCN2C1=O 89256,Cc1c(C(N2CCC(N3CC(F)(F)C3)CC2)=O)cc([N+](=O)[O-])cc1[N+](=O)[O-] 89257,C1(NC(CC(C)OC)=O)CC2CCC(C1C)N2C(c1ccc(C(=O)CF)cc1)=O 89258,c1(C(N2CCCC3(CNC(c4ccc(F)cc4)=O)C2C3)=O)cc(F)cc(F)c1O 89259,c1(OCC(=O)NC2CC2NC(c2ccnn2C2CCC2)=O)cccnc1 89260,N1(C(CCN(CCC)C(C)=O)=O)CCC(O)(CC)C1 89261,N1(C(c2cc(C3CCCC3)[nH]n2)C(=O)NC(CC)C)CCC(COCC)CC1 89262,C1(CC(N2CC(C)(CSC)C2)=O)CN(C(C2CCC(C)CC2)=O)CCO1 89263,n1(CC)cc(C(=O)N(CCCCCCNC(=O)OC(C)(C)C)C)c(OC)n1 89264,n1(CC(=O)NC(CC)CN(C)C(c2cnn(C)c2OC)=O)cc(C)ccc1=O 89265,C1(NC(C(C)(C)OC)=O)(COC)CCN(C(=O)C(c2cccc(Cl)c2)C)C1 89266,C1(C(=O)NCCC2CC(NC(C=C(C)Cl)=O)C2)C2CCCC12 89267,c1(C(=O)NC2(CCNC(C3CCOC3)=O)CCCC2)cnc(-n2cccn2)cn1 89268,C1(CC(N2CCOC(CCNC(=O)CN3CCC3C)C2)=O)(OC)CCCCC1 89269,c1(C(C(=O)Nc2c(COC)scc2)NC(C)C)ccc(Cl)c(Cl)c1 89270,C(CCC(C)NC(c1ccnn1CC1CC1)=O)NC(C=C(CCC)C)=O 89271,C1(C(N2CCN(CC3CCCO3)CC2)=O)(SC)CC2(CC(F)C2)C1 89272,c1(C(=O)NC(CC(C)NC(c2nnn(C)c2C(F)(F)F)=O)C)cc2n(c1)CCC2 89273,C1(CC(C)NC(C2CSCCS2)=O)CCN(C(=O)C(C)(C)N2CCCCC2)CC1 89274,C1(C2CC2)(C(=O)NCC2(CO)CCOC2)CN(C(c2ccon2)=O)C1 89275,C#Cc1cnn(C)c1C(N1CCOC(C(=O)NC(c2cn(C)nc2C)C)C1)=O 89276,C1(NC(c2cc(CNC(C34CCN(CC3)CC4)=O)[nH]n2)=O)COCC1C1CC1 89277,c1(N2CCCC(C)(N(C)C)C2)nc(NCC2(CCO)CCOC2)c2ncsc2n1 89278,c1(C(=O)NCCC(CNC(c2ccc(C)cc2Cl)=O)(C)C)ccn2nncc2c1 89279,c1(C(=O)NCC(CC=C)NC(=O)C(C)(CC)CCC)ccc(SC)c([N+](=O)[O-])c1 89280,c1(CC(N2CC(C(C)NC(c3cccc(OC)n3)=O)C2)=O)ccc(C)c(F)c1F 89281,c1(C(C(=O)NC(CN(C(C(n2ccc(C)n2)C)=O)C)(C)C)F)ccc(F)cc1 89282,C12(CNC(CC3CN(C(=O)C(C(C)C)n4cnnn4)C3)=O)COC(C(=O)OC)(C1)C2 89283,c1(-c2c(C)ccs2)csc(=Nc2cccc(C(N)=O)c2)n1Cc1ncoc1C(C)C 89284,C(=O)(C(C(C)O)NC(=O)CCCCN(C)C)NCCOCCC=C 89285,c1(C(C)=O)cc(C(=O)N(CC(C)CNC(=O)Cc2cnc(C)o2)C)co1 89286,CC1CCC(C)(C(N2CCC(=CCNC(=O)CC3(C)OCCO3)CC2)=O)C1 89287,C1(CNC(c2c(CC)noc2)=O)CN(C(=O)C(C)(C)S(=O)(=O)CC)CCC12CCC2 89288,Cc1cc([N+](=O)[O-])ccc1COC(c1nnn(C)c1C(F)F)=O 89289,C1(OC)CC(N=c2[nH]c(=NC(C)c3ccncc3F)c3ncccc3[nH]2)C1 89290,N1(C(C2=C(C)CCC2)=O)CCN(C(=O)C(C)C(C)(C)C)C2COCC12 89291,n1(CC)cc(Br)c(C(=O)N(CC(C)NC(=O)CCc2ccncc2)CC)n1 89292,c1(C(=O)NC2C(CNC(CSC)=O)CC2)ccc2c(c1)OCCCO2 89293,Cc1cc(C(N2CC(C(C)NC(C3CCC(C)(C)C3)=O)C2)=O)n(CC(F)(F)F)n1 89294,CC(C(=O)NCc1nc(C(=O)NC2(CC3CC3)CC2)co1)C(C)(C)C 89295,C1(C(C(=O)NCCC2(O)CN(C(C3(F)CCOC3)=O)C2)O)CCCCCCC1 89296,C1(C)(C(N2CC(C(C)OC)C2)=O)CCN(C(=O)C=C(C)C(C)C)C1 89297,N1(C(c2c[nH]c3ccncc23)=O)CCC2CCN(C(=O)CCOC3CC3)C2C1 89298,N1(CC)CC(C(=O)N(C2CCC(NC(c3nc(O)sc3C)=O)CC2)C)CCC1=O 89299,c1(C(=O)NCc2cn(C)nc2C(F)F)c(F)ccc(O)c1F 89300,c1(CCN2CC(NC(=O)NCCN(C)C)CC2=O)ccc2occc2c1 89301,CC1(C)CCCC(C(=O)NC2C3CC2N(C(=O)Cn2ccc(O)nc2=O)C3)C1 89302,C12(CNC(=O)CC3CCC(O)C3)CN(C(c3cnc(C4CC4)[nH]3)=O)CC(F)(C1)C2 89303,c1(C(N2C(C(N(CCCCO)CC)=O)CCC2)=O)ccc(C)cc1Cl 89304,C1(C(=O)NC(C2CC(NC(=O)C(C)Cc3cccnc3)C2)C)CCC(CO)CC1 89305,C(=O)(C(CCOCCOC)OC)NCc1ccc(C(C(=O)N)N(C)C(C)C)o1 89306,CC(C)C(CCC(=O)N(C)CCN(C)C(C)C)NC(=O)CSCc1nc[nH]n1 89307,N1(C(C(C)OCC#C)=O)CCOC(CC(=O)NCCc2ocnc2CO)C1 89308,c1(OC)c(C)ccc(C(N2CC3(C2)CN(C(C2CC(C(C)C)=NO2)=O)C3)=O)c1F 89309,c1(C(=O)NC(C2CCOC2)CNC(C=NOC)=O)c(N)cc(Cl)cc1F 89310,c1(C(=O)NCC2CN(C(CC(C=C)(C)C)=O)C(C)C2)cc(C)c(C)cc1N 89311,C1(NC(C23CCC(NC(C(COC)N(C)C)=O)(CC2)C3)=O)CC2(C1)CC(C#N)C2 89312,C1(CNC(=O)CC2CCNC2=O)CN(C(C2(O)CCCCC2)=O)CCO1 89313,N1(Cc2c(C)n[nH]c2)CCCC2(CCCN(C(c3ncsc3C)=O)C2)C1 89314,Cc1cccc(Br)c1C(N1CC(NC(=O)C(C(C)C)n2cncn2)C(O)C1)=O 89315,N1(C(C2(SCC)CC2)=O)CCCC1C1CCCCN1C(=O)C=CC1CCC1 89316,N1(C(C(CNC(CCc2n(C)ncc2)=O)O)=O)CCc2ncccc21 89317,N1(C(CN2C(C)CCC2)=O)CC(N(C(=O)Cn2ccc(O)nc2=O)C)C(C)(C)C1 89318,c1(C(=O)NC2CCCC2C(F)F)c(Cl)ccc2ccncc12 89319,N1(C(C=C2CCN(C(c3c(OC)ccs3)=O)CC2)=O)CCNC(=O)CC1 89320,Cc1c[nH]nc1C(=O)NCC1CCN(CC(=O)NC(C)C(C)C)C1 89321,C(=O)(C(C)C(O)C(C)C)NCc1c(C)nc(CC)o1.c12ccnc(c1)-n1cc-2nn1 89322,CC(CO)C(C)N=c1cc[nH]cc1S(=O)(=O)N1CCCC(C)(C)C1 89323,N1(C(c2c(C)scn2)=O)CCCC(C(N2CCCC2CNC(N)=O)=O)(C(C)C)C1 89324,N1(C(C2=NOC(C)C2)=O)CCCN(C(=O)C(C)Cc2ccncc2)C(C)C1 89325,CC(C)(O)C(CCO)NC(C1CC2(CC2)CN1C(c1cc(CCO)on1)=O)=O 89326,N1(C(C(C(C)C)C(C)NC(=O)C=CCF)=O)CCC(O)(C2CC2)CC1 89327,[N-]=[N+]=NC1CCCC1NC(C1(CCNC(C2CCS2(=O)=O)=O)CCC1)=O 89328,N(C(=NCC1CCC(=O)NC1)N1CCC(CCC#N)CC1)C(COC)C 89329,C1(c2n(CCSC)nnn2)(NC2CC(CO)C2)CCN2CCCC12 89330,c1(CN2CCC(NC(c3cn(CC=C)nc3)=O)C2)cc(Cl)cc(Cl)c1 89331,C1(CNC(c2ccn3ccnc3c2)=O)CC2COCC2N1C(c1cccnc1)=O 89332,N1(C(c2c(CC)ocn2)=O)CCC2CN(C(c3ccc(N)cc3O)=O)CCC2C1 89333,C(=O)(C1=CCCOCC1)NCC1(F)CCN(C(c2cncc(N)c2)=O)C1 89334,N1(C(c2nc(C(C)=O)sc2)=O)CC(NC(C2CCC(C)(C)O2)=O)C2(CC2)C1 89335,N1(C(C2CCN(Cc3c(C)nns3)CC2)=O)CCc2ccc([N+](=O)[O-])cc2C1 89336,c1(CC)ncc(C(=O)NC(C2CCN(C(C34CCC(CC3F)C4)=O)C2)C)c(C)n1 89337,Cc1nc(C(=O)N(C)CC2CCCN2C(=O)C(C2CCCO2)C2CC2)c(C)o1 89338,c1(C(=O)OC(COC)C(C)C)cc(O)nc(COC)n1 89339,C=CC1(CCNC(=O)NC2CC2C#N)CCCCC1 89340,S(=O)(=O)(c1cccc2c1OCCC2)N1CC(O)CC(OC(C)(C)C)C1 89341,N1(C(C(CN(C(=O)C=CCF)C)(C)C)=O)CCC2OCCCC2C1 89342,c1(C(N2C(C)CCC(NC(C(COC)C)=O)C2)=O)cc2c(OC)[nH]c(=N)nc2s1 89343,c1(C(=O)NCC2CN(C(CC(C)(C)OC)=O)CC2O)cc(=O)c2ccccc2o1 89344,c1(C(=O)NC2CCN(C(C(C(C)C)SC)=O)CC2(C)C)ccc(=O)n2c1CCC2 89345,N1(C(c2ccc(CC)cc2)=O)CCC2(C)CN(C(=O)CCOC(C)=O)CC12 89346,Cc1ccc(C(=O)N(CCCNC(C2CNC(=O)N2C)=O)C)cc1Cl 89347,N1(C(c2c(SCC=C)cccc2)=O)CC2(C1)CN(C(C1CCC3CC3C1)=O)C2 89348,N1(C(CCC)=O)CCN(C(=O)CCn2ccccc2=O)CC1CC 89349,C1(C(N2CCC(CC)C2)=O)CN(C(=O)C(C)COC)C(C)(C)C1 89350,CCC(CN(C)C)CC(=O)N1CC(F)CC1CC(=O)Nc1cncc(N(C)C)c1 89351,C(c1cnc(O)nc1O)=CC(N1CC(C)C(NC(=O)C(F)=CCCF)CC1)=O 89352,c1(C(=O)NCC2CCCC2NC(=O)CC(O)C2CCCC2)cc([N+](=O)[O-])cnc1O 89353,N1(C(C2(F)CC2)=O)CC2CC2(Cn2cc(CCCO)nn2)C1 89354,C1(OCC)CN(C)C(C)(C(N2CCC(CN(C)CCc3ccccc3)CC2)=O)C1 89355,C=C(CNC(=O)COc1cnn(C)c1)CCNC(=O)C(n1ccc(C2CC2)n1)C 89356,CCC1=C(C(=O)NCC2CN(C(C3CCCN3C(C)=O)=O)CCN2C)CCCO1 89357,N1(C(C(C)CF)=O)CCC2(CC1)CCN(C(c1cc(F)ccc1O)=O)CC2 89358,c1(CC(=O)NCc2ccc(NC(=O)Cn3ccnc3)s2)nc(O)n[nH]1.C1CSC1 89359,c1(C(=O)NC(C2CCN(C(C3(C)CC(=C)C3)=O)CC2)C)ccc(C)c(C)c1Cl 89360,Cc1cc(C(=O)NCCCCN(C(=O)Cc2ccnn2C)C)c2cnn(C)c2n1 89361,N1(c2cc(NCCCN(C(C)=O)C)nc(C)n2)CC(C2=NOCC2)C1 89362,n1(CC(N2C(CNC(COCCOCC#C)=O)CC2)=O)cc([N+](=O)[O-])cn1 89363,N1(C(C(=O)NCC)=O)CCC2OCCN(C(=O)CCOCc3ccccc3)C2C1 89364,N1(C(C(CO)NC(N)=O)=O)CC2CC1CN2C(c1cc(Cl)ccc1Cl)=O 89365,CCC(C)CC(=O)C(=O)NC(CO)C(=O)NCC1CCc2nccn21 89366,C(=O)(CC(CC)c1ccccc1)NCC(=O)N(C1CN(C(C(CC)C)=O)C1)C 89367,C1(NC(c2c(C)cns2)=O)CC2(C1)CC(NC(=O)Cc1cc(Cl)cnc1C)C2 89368,C#Cc1ccc(CNC(=O)C(O)CCNC(=O)CC2CC(C)C2)cc1 89369,C(CCCCC(=O)N1CC(N(C(=O)CN(C2CCC2)C)CC)C2(CC2)C1)OCC 89370,C#CCCC(C(=O)N1CCC(=C)CC1)NC(=O)CC1CCOC1C 89371,Cc1nc(C(F)(F)F)cc(=NCCC(C)(C)NC(=O)C(=O)N(C)C)[nH]1 89372,C(C(C)(C)C(=O)N1CC(F)CC1CNC(=O)C(C)Oc1ccc(Cl)cc1)OC 89373,C1(NC(CC=C)=O)CN(C(c2ccc(C(N)=O)o2)=O)CC1CO 89374,C1(NC(c2cn(CC)nc2)=O)(CO)CCN(C(=O)C(O)COC)C1 89375,N1(C(Cc2ncn(C)c2)=O)CC2CC1(CNC(C1CC13CCOC3)=O)C2 89376,c1(C(N(CC(C)NC(C(C=C)CC)=O)C)=O)ccn(C)c(=O)c1 89377,C1(O)(CN(CC#C)C(c2cccc(-c3ccccc3)c2)=O)CCN(C(=O)CO)CC1 89378,N1(C(C2C(=C)C2)=O)CCCC(N(C(=O)Cc2c(C)noc2Cl)C)CC1 89379,CC1(C)C(CNC(C2(c3cc[nH]n3)CC2)=O)CCN1C(C1CCNC1=O)=O 89380,c1(CNC(=O)NCCSCC(F)F)ccc2c(c1)CCO2 89381,N1(C(=O)OC(C)(C)C)CCC2CC(NCC3CCOC(C(F)F)C3)CCC12 89382,c1(OC)cnc(N2CC3C(C2)N3C(=O)C(c2ccccc2Cl)OC)nc1C 89383,C1(NC(c2cnc3sccc3c2)=O)CCC2CN(C(=O)C(=O)NC3CC3)CC2C1 89384,C(C1c2ccsc2CCN1C(c1nc(CC)oc1C)=O)SCC.C1CC(=O)N1 89385,Cc1cn(CC(=O)NC2CC23CCC(NC(=O)C(C)O)CC3)c2ccccc12 89386,C(C)(CO)(C(F)(F)F)NC(CC(CNC(c1cc(OC)n(C)n1)=O)C1CCC1)=O 89387,C1(OC(C)C)CCN(C(c2cc(CNC(=O)C=CC(F)(F)F)cs2)=O)C1 89388,C1(CC(N2CC(CCNC(CSCC#C)=O)C2)=O)CC2(CCCC2)CO1 89389,c1(C(CC)C)nccc(=NCC23CC(NC(c4[nH]ccc4COC)=O)(CO2)C3)[nH]1 89390,C1(C(C(=O)O)NC(c2ccc(CC)cc2)=O)CC(=O)N(C)C1c1cnn(C)c1C 89391,C(=O)(C1=CC2(CCOCC2)C1)NC1CC(C)N(C(c2cc(C(N)=O)cn2C)=O)C1 89392,N1(C(C(c2cccc(F)c2)C)=O)CCOC(CNC(C2(C#N)CC2)=O)C1 89393,C12(NC(=O)NCC(N3CCCC3)=O)CCCN(C(c3ccc(O)c(N)n3)=O)CC1C2 89394,N1(C(C(CC)CCOC)=O)CC2CCOC2(CNC(=O)Cc2sc(C)cc2C)C1 89395,Cc1c(C(N2CC(CF)OC(CF)C2)=O)oc2cc(Cl)ccc12 89396,CCS(=O)(=O)c1ccc(Cl)c(C(=O)NCC2CCN(C(=O)OC(C)(C)C)C2C)c1 89397,C1(CNC(C(Cc2ncn(C)c2)O)=O)CCC(NC(c2cnc(O)n2C)=O)CC1 89398,N1(C(COCP(C)(C)=O)=O)CCC2CCN(C(C3(CN(C)C)CC3)=O)C2C1 89399,c1(CNC2CCC(C(=O)NCC(C)O)C2)c(Cl)cc(F)cc1Cl 89400,Cc1cc(C(=O)N(CC(C)NC(C2CCOC(=O)N2)=O)C)c2c(n1)CCCC2=O 89401,N1(C(C(C)NC(C)=O)=O)CCN(C(=O)CCCc2nccs2)C(c2cn[nH]c2)C1 89402,N1(C(c2cccc(NC)n2)=O)CCC2(CCCCC2NC(=O)CC(C)C2CC2)C1 89403,S(=O)(=O)(c1ccc(Br)cn1)N1CC(CNC(c2ncccc2Cl)=O)OCC1 89404,C12(CC(=O)NC(CCN(C(C(CC)OC)=O)C)C)CC3CC(CC(C3)C1)C2 89405,c1(C(C(C)NC(c2n(CCSCC)nnn2)(C)COC(C)C)O)ccc(F)cc1 89406,C1(CNC(C(C)=C2CCC2)=O)CN(C(c2cccc(Br)c2)=O)CCC1(C)C 89407,Cc1c(C(N2CC(NC(c3cnc(CC(C)(C)C)o3)=O)C2)=O)nn(C)c1C1CC1 89408,c1(CN2C(C(N3CC4(COC4)C3)=O)CC3CC32)cc(O)ccc1Cl 89409,C(C(C)(C)C(=O)N(C)C1CC1)N(C(=O)C(C1CCOCC1)=O)C 89410,c1(C(=O)NCC2CC2NC(C2(Cl)CCC2)=O)ccc2c(n1)CCC2 89411,c1(C(N(CC(CC)NC(=O)C(CC)SC)C)=O)cc(C)c2c(O)n[nH]c2n1 89412,C(CC1=CCCCCC1)NCC1(C(=O)O)CCN(Cc2ccccc2)C1 89413,c1(C(=O)NCC(CO)NC(C=C(C)Cl)=O)cc2c(s1)-c1ccccc1OC2 89414,N1(C(C(CC=C)(C)O)=O)CC(C(N2CCC(C)(CCO)C2)=O)C2(CCC2)C1 89415,C(=O)(CC1=CCCC1)NCCO.C12CCN(CC1)CCn1cc(nn1)C2C(C)C 89416,CC1(C)CCC=C1C(=O)N1CCCN(C(=O)Cc2ccc(F)c(Cl)c2)CC1 89417,c1(C(=O)NCCN(C(C(=O)NC(CC)C)C)C2CC2)ccc2cccc(F)c2n1 89418,N1(C(C(N2CCCC(O)C2)C)=O)CCCC(C2CC2NC(=O)Cn2cnnn2)C1 89419,c1(C(N(C2CCN(C(=O)Cc3cn(CC)nn3)C2)CC)=O)ccn(C(C)(C)C)c1 89420,c1(C(N(CCNC(c2cccc(C3CC3)c2)=O)C2CC2)=O)c(O)cccc1Cl 89421,N1(C(CC(CNC(=O)C(=CC2CCCC2)C)OC)=O)CC2CC1CC2CF 89422,c1(C(=O)NC(CCNC(c2ccc(CC)[nH]2)=O)C)ccc2c(=O)n(C)cnc2c1 89423,Cn1ncc(C(N2CC(CNC(=O)CCOCC(F)(F)F)C(O)C2)=O)c1Cl 89424,c1(C(=O)NCC(C)NC(C2C(c3cccc(C)n3)C2)=O)cc(=O)n2nccc2[nH]1 89425,C(CCNC(C1(NC(C2C(C)(C)C2(C)C)=O)CC(O)C1)=O)(C(C)C)OC 89426,C(CC(=O)NC(c1cscn1)CO)(C(F)(F)F)NC(=O)CC1COCCOC1 89427,C1(c2nc(CNC(c3cscc3F)=O)[nH]n2)CCN(C(=O)Cc2cc[nH]n2)CC1 89428,Cc1ccnc(CN(C)C(c2n[nH]cc2CNC(c2cn(C)nn2)=O)=O)c1 89429,c1(NC2(C3CN(C(C4C5CCCC45)=O)C3)CC2)ccc2cnccc2c1[N+](=O)[O-] 89430,Cc1nnc2cnc(C(N3CC4CC3CCC4NC(=O)CC(C)(C)O)=O)cn12 89431,N1(C(C(CCCC)C)=O)CC2(CCCCN2C(=O)CCOCC(F)F)C1 89432,c1(C(N2CCC(N(C(=O)CC(F)F)C)C2)=O)ccc2c(c1)ncn2C 89433,N1(C(=O)Nc2c(Cl)cnc(SC)n2)CCCC2NC(=O)CCCC12 89434,C1(C)(CNC(C=CCCC)=O)CCCN(C(=O)C=Cc2nc(C)cs2)C1 89435,C(=O)(C(CC)C(C)(C)CC)NC(CC(=O)N(CCCCC)C)(C)C 89436,c1(CC)c(C(=O)NCCCCNC(=O)C(O)(CC)c2ccccc2)nnn1C 89437,c1(C(CNC(=O)CCC2CCCO2)=O)csc(CCc2ccco2)n1 89438,Cc1ccccc1NC(=O)C(N1CCOC(C(=O)N(C)C)C1)c1ccc(Cl)s1 89439,c1(-n2cc(C(C)(C)C)nn2)ccccc1CCC(N1CC(C(=O)O)C2CC12)=O 89440,c1(NC)ccc(C(=O)NC(CCn2cc(CC3(n4cncn4)CC3)nn2)=O)cc1 89441,Cc1cc(C=CC(=O)NC(C)C(C)NC(=O)C(C)(Cl)Cl)ccc1C(F)(F)F 89442,C1(NC(c2c(CC)noc2)=O)(CO)CCCN(C(c2cnc(C)cc2C)=O)C1 89443,c1(C(N(C(C(N)=O)C2CC2)CC)=O)cccc(S(=O)(=O)N(C(C)(C)C)C)c1 89444,N1(C(CCOC(C)=O)=O)CCC(F)(CNC(c2ccn(CC(F)F)n2)=O)C1 89445,CC(C)CC(CNC(=O)C=Cc1cncn1C)NC(C1CN(C)CCO1)=O 89446,c1(OC)ccc(C(=O)NCC(O)CN(C(=O)C2=CCCSC2)C)cc1OC 89447,C=CCC(C(=O)N1CC(O)CC1C(=O)NC1(C2CCCO2)CC1)OC 89448,CC1C(C=CC(N2CC(O)(CNC(c3cc(-c4ccoc4)on3)=O)C2)=O)C1(Cl)Cl 89449,C(CCNC(C1(CN)CC1)=O)N(C(C)C)C1CC1.C(C)(C)(C)O 89450,c1(C(=O)NC(CCN(C(c2c(C)con2)=O)C)C(C)C)c(Cl)ccnc1C 89451,CCC(CC)C(F)C(=O)NC(CCC(=O)N(C1CCC1C)C)C(C)C 89452,C1(CC(C)NC(=O)CC2CC(CC(C)(C)C)C2)CCN(C(=O)CC(Cl)Cl)CC1 89453,CCC(C)(CNC(C1CC1F)=O)NC(c1cc(CF)on1)=O 89454,c1(OC)ccc(CC(=O)NC2CCCC(C(=O)NCc3nc(C)no3)C2)c(F)c1 89455,c1(C(=O)NCC2(NC(C3CC3c3ccsc3)=O)CCC2)cccc2c1CCCN2 89456,c1(OC)cc(F)c(-c2nnc(N(C(C)CS(C)=O)C)n2CC2CCCO2)c(F)c1 89457,C1(CNC(CC(C)(C)O)=O)C2CCCCCC12.C12CCCCC1NC2=O 89458,C1(C)(CNC(CCC(=O)NC)=O)CCCS1(=O)=O.c12ccc(cc1)s2 89459,C1(C(=O)Nc2cccc(NC(=O)C(F)Cc3ccccc3)c2)CCCCCCC1 89460,N1(C(C(COC)C)=O)CCC(C(=O)NCC2CC23CCOC3)CC1C 89461,N1(C(C2(CSC)CC2)=O)CC(CO)(NC(C2CC(=O)N2)=O)C1 89462,C=C1Cn2c(C(=O)NC3(CO)CN(C(=O)Cn4cc(COC)nn4)C3)nnc2S1 89463,c1(NC(=O)CC2CCN(S(=O)(=O)C(F)(F)F)C2)ccc(Br)c2c1C(=O)NC2 89464,c1(CC)occc1C(=O)NCCN(CC(C)O)C(c1cc(CCOC)on1)=O 89465,c1(CC(=O)NCC(CNC(C2(C)N(C)CCC2)=O)O)cn2ccsc2n1 89466,CN1CCOCC2(COCCN2c2nnnn2CC2CCC3(CNC3)O2)C1 89467,C1(C(N2CC(NC(CSCC#C)=O)C(c3ccnn3C)C2)=O)COC2(CCC2)C1 89468,C1(C(=O)NCC2(C)CC2)CC(F)(F)CN1C(=O)CC1CC1 89469,c1(C(C)(C)C)ccc(N2CCN(C(C3(N)CCSC3)=O)CC2)cc1 89470,C1(C)(C(N2CC(OCCNC(C(c3cccnc3)OC)=O)C2)=O)C(C)(C)C1(C)C 89471,c1(C(=O)NCC2CC(c3ccccc3)CO2)ccc(Br)cc1 89472,N1(CCC(=O)NCCCN(C(c2cnc(C)o2)=O)C(C)C)CCCCC1=O 89473,C1(C(N2CCC(C(=O)NCc3c(C)nco3)C2)=O)CCC2(CC1)CC2 89474,C1(C(=O)NC2C(F)CCN(C(CC(C=C)(C)O)=O)C2)CN(CP(C)(C)=O)C1 89475,C(CC(C)CCNC1CCN(C(N2CCOCC2)=O)CC1)NC(C=CC(C)C)=O 89476,c1(OC)c(CNC(=O)NCc2cscc2C)cccc1C#N 89477,C1(C(=O)NC(CC=C)CO)CC(N=[N+]=[N-])CN1C(=O)C(O)CN(C)C 89478,C(=O)(C(CCSC)NC=O)NCCCCCN(C(CC)=O)C 89479,CCC(CC)CC(F)C(=O)NC(CNC(C1(C)CCOC1)=O)CCOC 89480,CN1CCCC1C=CC(N1CCOC(CCNC(=O)CSc2n[nH]c(O)n2)C1)=O 89481,C1(C(=O)NCC2(NC(CCSC)=O)CCCCC2)CN2CCN1CC2C 89482,c1(CC2(NCCN(C(CC(=O)OCCl)c3ccccc3)C)CC2)ccc(Br)cc1 89483,N1(C(c2c(OC)scc2)=O)CC2CN(C(=O)CN(C3CCC3)C)CC2(C)C1 89484,c1(C(=O)NCC2N(C(CCOCC#C)=O)CC(C)CC2)cccc2nonc12 89485,N1(CCCC)CCN(C(=O)CC2CCCCN2C(=O)Cn2cccn2)CC1 89486,C1(NC(=O)Nc2cccc(C)c2)COCCN(C(C2(CF)CC2)=O)C1 89487,C1(OC)CC2CCC(C1)N2C(C1CNCCN1c1ccncn1)=O 89488,c1(C(N2CCC(CO)CC23CC3)C(=O)NCCCF)cnc2n1CCOC2 89489,Cn1cc(C(=O)NCC2CCCC2NC(=O)CCCc2ncco2)c(C2CC2)n1 89490,Cc1c(C(=O)NCC(C)N(C(=O)CCC2CCCCN2C)C)c(Cl)nn1C 89491,c1(N2C(C)C(NC(c3ccc(CO)cn3)=O)CCC2)ncc(C#N)cc1Cl 89492,C(C)(CC(=O)NC1C2CC1N(C(c1ccc(CO)s1)=O)C2)(C(F)F)N(C)C 89493,c1(CC)ccc2cc(C(=O)NCC(C)CNC(C3(c4cc[nH]n4)CC3)=O)[nH]c2c1 89494,CC1(C)CN(C(C2CC=CC2)=O)C1C1CCN(C(C2CCC(F)(F)C2)=O)CC1 89495,C1(C(N2CCC(CF)C2)=O)CC12CCN(C(c1cn(C3CC3)nn1)=O)C2 89496,c1(CN(C(=O)Cc2cc(CO)on2)C)ccccc1CNC(C1CCC2CC12)=O 89497,C#Cc1ccc(C2CC2C(=O)NCCCCNC(=O)C=CC2CCCCC2)cc1 89498,C1(C(=O)NCC(C(C)C)NC(C2CCCCC2)=O)CCCCN1C 89499,CCCC(C)CCCC(=O)N(C1(C(=O)NC2(c3cc[nH]n3)CC2)CC1)C 89500,C1(CNC(CSCC#C)=O)Cc2ccccc2CN1C(c1cc(F)n(C)n1)=O 89501,c1(C(N2CC(CC=C)(NC(=O)Cc3ccsn3)C2)=O)c(C)cccc1[N+](=O)[O-] 89502,N1(C(C(C)OCC)=O)CC(NC(=O)CCCn2ccccc2=O)CC2(CC2)C1 89503,N1(C(C(C2CCC2)OCC)=O)CCc2ccc(C(=O)NC(CC)CO)nc2C1 89504,c1(CNC(C(CC)(C)C#N)=O)ccc2c(c1)CN(C(=O)Cc1ccns1)C2 89505,N1(C(C(CO)NC(c2ccoc2Cl)=O)=O)CC(F)(F)C(F)(F)C1 89506,Nc1cc(Cl)ccc1C(N1CC2CC(NC(c3ccc(F)s3)=O)C2C1)=O 89507,C1(NC(=O)C2=CCCCC2)CCCC12CN(C(c1ccn(CCO)c(=O)c1)=O)C2 89508,C(=O)(C#CC(C)(C)CNC(=O)Cc1ccoc1)N1CCOCC(C(C)C)C1 89509,c1(C(=O)NCC2N(C(Cn3ncc(C)c3)=O)CCN(C)C2)cccc2c1CCC2 89510,c1(C(=O)NC2CCN(C(c3c(OC)ccnc3)=O)CC2)cnc2cnccc2c1 89511,C1(C)(C(=O)OCC)CCN(C(C(=O)NC2CC2)C(C)C2CCCOC2)C1 89512,CC1(CNC(c2ncoc2Br)=O)CCCN1C(C1CC(F)C(=O)N1)=O 89513,C1(C(=O)N(C(C)C(=O)N(C(C)CN(C)C)C)C)(CC)CCNC1=O 89514,c1(SC)cccc(C(=O)NC2CCCC(C(=O)NCC3(C)CC3)C2)c1O 89515,c1cc(=NCCCC2CCCCC2)[nH]c(NC2CCC(C3CC3)C2)n1 89516,c1(C(N2CCC(F)(CF)CC2)C(=O)NCCCCCC)cccc(C2CC2)c1F 89517,CN1CC(O)(C(=O)NCCNC(=O)CC2(NC(=O)OC(C)(C)C)CC2)C1 89518,CC1CCN(C(=O)C(C)(C)N2CCCC2)CCN1C(C1CC2(CCCCC2)C1)=O 89519,N1(C(C(CC)N(C)C)=O)CCCC(c2n[nH]c(CNC(=O)CCNC(N)=O)n2)C1 89520,c1(C(N(CCCNC(C(CCOC)C)=O)C)=O)cnc2nc(O)nc(O)c2c1 89521,c1(C(=O)NC2C(OC)CN(C(c3conc3C(C)OC)=O)C2)cc(F)ccc1O 89522,C1(CNC(c2c(C)snc2)=O)CN(c2nc(C3CC3)ns2)CCC12CCOC2 89523,N1(C(CN(C2CC(C#N)C2)C(C2(C#C)CC2)=O)=O)CCC(CC)CC1 89524,c1(C(N(CC(CNC(C2(CC)CC2(F)F)=O)O)C)=O)nn(C)c2c(=O)[nH]cnc12 89525,c1(C(N2C(CN(C(C3CN(C4COC4)C3)=O)CC)CCC2)=O)cn2ccsc2n1 89526,c1(N2CCC(N(C(=O)CNC(=O)NC)CC)C2)nc(C#N)ncc1C 89527,C1(CNC(CCn2c(C)csc2=O)=O)CN(C)CCN1C(c1cccc[n+]1[O-])=O 89528,c1(CC)ccc(N)c(C(N2C3CCC2C(NC(C2(C)CCCC2(F)F)=O)C3)=O)c1 89529,c1(C(C(=O)NCC(=O)SCC)C)cccnc1.C1(=O)C(=O)NC(C)CN1.C(C)(C)(C)O 89530,Cc1nn(C)c(N2CCOCC2)c1CON1CCCN(CC2CCCN2C)CC1 89531,N1(C(CN2CCCC(CC)C2)=O)CC2(CCCC2NC(C2C=C2C)=O)C1 89532,N1(C(CC2C(C)C2)=O)CCC(OCCNC(C2CC2c2ccoc2)=O)CC1 89533,C(CC(C(C)(C)C)NC1(c2nnnn2-c2ccccc2C)CCC2(CC2)C1)SC 89534,C1(C(=O)NC(c2ccnn2C)C(N2CC(OC(C)C)C2)=O)C=CC=CC=C1 89535,CCC(C)(C)OCC(=O)NCC1CC1NC(=O)C=C(C)C(F)F 89536,Cn1cc(C(N2CCC(NC(C3CCC(c4cc[nH]n4)O3)=O)C2)=O)c(O)n1 89537,C1(C(=O)NC(COCCCNC(CCSC)=O)(C)C)OCCC1C 89538,N1(C(C2(OC)CCCOC2)=O)CC2CC(NC(=O)Cc3n[nH]c(C)n3)C(C2)C1 89539,Cc1ccc(CNC(C)CCc2ccc(Br)cc2)c(Br)c1 89540,C12(C(=O)NC(c3ccc([N+](=O)[O-])cc3)C(=O)O)CC=CCN1CCC2 89541,N1(C(c2ccnn2CC)=O)CCCC(CCC(=O)NC2C(OCCC)CCC2)C1 89542,N1(C(c2c(CNC(c3c(CC)noc3)=O)occ2)=O)CC2CCC2(OC)C1 89543,C1(C(=O)NC2C(NC(COc3cccc(CC)c3)=O)CCC2)C(F)(F)C12CCC2 89544,C1(CNC(c2n(C)ncc2)=O)CC(F)CN1C(c1ccnnc1)=O 89545,c1(C(=O)NC2CCN(C(c3cc(C(F)F)[nH]n3)=O)C2)cc(F)cc(F)c1 89546,C1(CNC(CCC=C)=O)CN(C(=O)C(C)CCO)CCC12CCOCC2 89547,c1(NC(CNC(c2c(CC)cno2)=O)=O)cccc(C#N)c1 89548,O=C(CCCn1cncn1)NC1C=CCCC1.n12cc(nn1)C(=O)N1CC2C1 89549,N1(C(c2ccc(CC)cc2)=O)CCC(NC(C2COCC2(C)C)=O)C(O)C1 89550,C1(C(=O)NCC2C(CC(=O)NC3(CO)CC(F)C3)C2)CCS1(=O)=O 89551,C1(C(=O)NC(CC)CCC(=O)N(CCCN(C)C(C)=O)C)CCCC(C)(C)CC1 89552,N1(C(CC)CO)CC(=O)N(CC(N)CF)C1 89553,c1(C(N2C(CCCNC(c3n(CC#C)cnn3)=O)CCC2)=O)cccc(CC)n1 89554,N1(C(C(C)OCOC)=O)CCOCC(NC(=O)CSCc2cscn2)C1 89555,N1(C(CC(=O)NC2(C)CC(NC(Cc3c(C)occ3)=O)C2)=O)C(C)CCCC1C 89556,C(=O)(C(O)CC(C)C)NCC1(CNC(COC(CC)(C)C)=O)CC1 89557,Cc1cc(C(=O)NCC2CC(F)(CNC(=O)CC(C)F)C2)ns1 89558,C1(C)(C(=O)NCCCOC)CCCN(C(=O)Cn2nc(C)cc2C)C1 89559,C1(NC(CSCCC)=O)CC(N=c2[nH]cnc3cnccc23)C1 89560,c1(C(=O)NC2CC(CNC(Cc3n(C)cnn3)=O)C2)ccc(F)cc1C(F)(F)F 89561,C12(CN3CCC(c4cccc(Br)n4)C3)CCCCCC1NCC2 89562,Cc1cncc(C)c1C(=O)NC1CN(C(c2cnc(O)o2)=O)CC1C 89563,C12(C(=O)NCC(=O)CCC3CC3(F)F)CCC(O1)c1ccccc12 89564,CCCC(O)CC(=O)NC(C)CNC(=O)COC(C)CC 89565,Cc1cc(CC(=O)NC23CC(C2)N(C(=O)CC(C)n2cccn2)C3)cc(C)c1 89566,c1(C(=O)NC(CCC)CCCOCCC(=O)O)ncc(Cl)c(N)c1Cl 89567,c1(-c2nn(C)c(C(=O)NCC(C)(O)C3CCC3)c2)cc(F)cc(F)c1 89568,C1(CC(=O)Nc2ncc(C)s2)CN(Cc2ccccc2OC(F)F)CCO1 89569,C(=O)(C1=CCSC1)NCc1c(C(=O)NCCC(CC)C)cco1 89570,C=CC(CC)CC(=O)NCC1CCN(C(=O)C(COC(C)(C)C)N(C)C)C1 89571,C(C)(C(O)C(F)F)NC(c1cn(CCNC(C(CC)O)=O)nn1)=O 89572,C1(n2cc(C3CCOCC3)nn2)(C(N(CCC2CC2)CC)=O)CCOCC1 89573,C1(CNC(C(C2CCOCC2)OC)=O)CC(C)N(C(=O)C=Cc2cncs2)C1 89574,C(=O)(C(C)C(C)(C)O)NC1C(NC(c2c(C)[nH]c(C(C)(C)C)c2)=O)COC1 89575,N1(C(CCCCSC)=O)CCC(NC(c2ccn(CC(F)(F)F)n2)=O)C(O)C1 89576,C(=O)(CCC(=O)N1CCCC1C1CCC1)Nc1nnc(CC(=O)OC)s1 89577,C#CC1(C(=O)N(CC(O)C2CCC2)C)CN(C(=O)C(c2ccn(C)n2)C)C1 89578,CC1(C(N2CCC(CF)(NC(c3coc4c3COC4)=O)C2)=O)CC2CCC1C2 89579,c1(C(C(=O)NCC(=O)OC)NC(=O)CCOCCOC(C)(C)C)cnn(C)c1 89580,c1(CCC(=O)NCC(=C2CN(C(c3cc(Cl)no3)=O)C2)F)nnc(O)nc1O 89581,N1(C(c2c(C)cc(C)[nH]2)=O)CCC(NC(c2cnc(C(F)(F)F)nc2)=O)C12CC2 89582,N1(C(CC)=O)CC(O)C(O)C1CNC(C1CC(c2cccc(Cl)c2)(O)C1)=O 89583,N1(C(CCc2onc(C)n2)=O)CCC(O)C(NC(=O)C(C)NS(C)(=O)=O)C1 89584,c1(C(=O)NCCC(C)NC(C=C(C)c2cccs2)=O)cnc(O)cc1C 89585,c1(C(=O)Nc2cc(OC)c(Br)cc2C)c(Cl)nc2cc(Cl)ccn12 89586,O=NN1CCCCC1C(=O)N(CCCNC(=O)C(F)C(F)(F)F)CCO 89587,C1(CC(=O)NC2(C)CC(NC(C(C)Cn3ccnc3)=O)C2)CCC(C)(C)C1 89588,N1(C(c2c(CC)cncc2)=O)CCC(C2CCCN(C(=O)CC34CC(C3)C4)C2)C1 89589,O=[N+]([O-])c1ccc(-c2cc(=NCc3ncccc3Cl)cc[nH]2)c(Cl)c1 89590,N1(C(C(C2CCN(C)CC2)C)=O)CCC(NC(c2cc(F)cc(Cl)c2)=O)C(F)C1 89591,C1(NC(=O)COC2COC2)CCC2CC1CN2C(C1CC1C(F)F)=O 89592,c1(CN(C(c2cccnc2)C(=O)OC)C)cc(Br)ccc1OC 89593,c1(C(=O)NCC(CO)NC(c2coc(C3CCC3)n2)=O)ccnc(C(F)(F)F)n1 89594,CCC(C)(COC)CNC(=NCc1ccccc1Cl)NC(C)C 89595,C(=O)(CC(F)F)NCCOCCCN(C(=O)CCc1ncccn1)C 89596,c1(CC)nc(C)ncc1C(=O)NC1CN(C(=O)CCC(C)SC)CC1F 89597,C(=O)(C1=CCN(C)C1)C(C1CC(F)(c2cn(CCC(=O)OC)nn2)C1)C 89598,Cc1ccc(=N)[nH]c1C(N1CC(NC(=O)CC2(C)CC2)C2(CC2)C1)=O 89599,Cc1ccc(C(F)(F)F)cc1C(N1CCC(C)(NC(c2ccccc2)=O)C1)=O 89600,c1(C(N2CCCCC(CNC(c3ccc[nH]3)=O)C2)=O)ccc2c(=O)ccoc2c1 89601,[N-]=[N+]=NCCCCC(=O)NC1(C(=O)NCC2CCCC2O)CCC1 89602,C#CC1(C(=O)NCc2nnc(CC)o2)CCN(C(=O)C(C)N=[N+]=[N-])C1 89603,C#CC1(CO)COCCN1Cc1csc(CN(C)C)c1 89604,c1(OC)ccc(CCC(=O)NC2CCC(NC(c3cnc(S)n3C)=O)C2)cc1F 89605,c1(OC)nc(=NC(Cc2cccs2)CC(=O)N2CCN(C)CC2)[nH]cc1C#N 89606,N1(C(C23CC(C2)C3)=O)CCC12CN(Cc1cccc(C(F)(F)F)c1O)C2 89607,Cc1noc(C)c1C(C)CC(=O)N1CCC(C(C)NC(C2(F)CC2)=O)C1 89608,C(C(=O)NN1CCCC1NC(c1ccccn1)=O)NC(C[SH]=N)=O 89609,C1(NC(=O)Nc2c(OC(C)C#N)cc(F)cc2)CCCC2OCCC12 89610,C1(NC(c2c(C)scn2)=O)C=CCN(C(c2ccnc(C3CC3)c2)=O)C1 89611,C#Cc1ccc(C(=O)NC(Cc2ccco2)C(=O)NCCN2CCOC2=O)o1 89612,CN1CCOC(N(C(C(=O)NCSC(C)(C)C)C(C2CC2)C2CC2)C)C1 89613,CC#CCC(C)N=c1[nH]c(=N)[nH]c(=NCC(c2cccs2)N(C)C)[nH]1 89614,c1(C(N2CC(CCNC(C3CCC3CF)=O)(OC)C2)=O)ccc(Cl)c(O)c1 89615,c1(CN=C(NCCOC)NCC2SCCc3ccccc32)ccc(S(N)(=O)=O)c(Cl)c1 89616,C1(CCC(=O)NCC(C)(C)F)CCN(C(c2cc(Cl)ncn2)=O)CC1 89617,CC1c2nnc(C3CC3)n2CCN1C(=O)N(C1CC1)Cc1cncc(Br)c1 89618,c1(CC(=O)NCC(CNC(=O)C(CO)C2CC2)OC)ccc(C(F)F)cc1 89619,Cc1ccc(SCC(=O)NC(C2CCCN2C(c2nccnc2Cl)=O)(C)C)cc1 89620,C(=O)(C(C)(C)CCCN=[N+]=[N-])N1CC2(CN(C(C3(F)C(C)(C)C3(C)C)=O)C2)C1 89621,CC1(C)COCCC1C(N1CC2CC2(NC(c2csc(-c3cnc[nH]3)n2)=O)C1)=O 89622,c1(CC(=O)NCCC(C)NC(C2CC3CCC2C3)=O)c[nH]c2ccccc2c1=O 89623,c1(C(C(F)F)NC(CCn2cc(CN(C(C)C)C)nn2)=O)c(F)cccc1F 89624,C1(C(N2C(CNC(CC=CCC)=O)CC(C)(C)C2)=O)Cc2cncn2C(=O)N1 89625,c1(OC)cc(C(F)(F)F)ccc1Br.c1(CC2CNC2=O)ccc(F)cc1F 89626,CCCCC(C)CCC(=O)N(CCCN(C(=O)CCc1c(F)cccc1F)C)C 89627,c1(C(N2CC(SC)C(NC(c3csc(Cl)c3)=O)C2)=O)ccc2cc[nH]c2c1 89628,Cc1coc(C2CC2)c1C(N1CCCCC1Cn1cc(Cn2ccnc2)nn1)=O 89629,Cn1c(CNC(C2CCC(CNC(c3nnsc3N)=O)C2)=O)nnc1O 89630,Cc1c(C(C(=O)NC2CCCC2)N(C)Cc2nc[nH]n2)cnn1C(C)C 89631,C1(C2CCCN(C(c3ccccc3)=O)C2)(NC(CC(CN(C)C)O)=O)CC1 89632,n1(CC)cnnc1CN(C(=O)CC(O)C1CC1)C 89633,N1(c2nnc(CC)s2)CCC(NC(=O)C(C)OCC(C)C)CC(C)(C)C1 89634,N1(C(C2C(CC(C)(C)C)C2)=O)CCN(C(C2CCC(O)C2)=O)C2CCCC2(C)C1 89635,N1(C(c2nncc(OC)c2)=O)C2CCC(C(=O)NOCC(N)=O)C1CC2 89636,c1(OC)noc(C)c1C(=O)NC(CNC(=O)C(C)(C)COCC(F)F)C1CCC1 89637,c1(C(=O)NCCC2N(C(C(C)OC3CCCC3)=O)CCOC2)csc2cncn12 89638,N1(CC)CCOCC1C(=O)NCc1cccc(CN2CCOCC2)c1 89639,N1(S(CCC)(=O)=O)CCC(CCNC(COC(c2ccccc2CC)=O)=O)CC1 89640,N1(Cc2cccc(C)n2)CCCC2CN(Cc3cccnc3)CCC12 89641,N1(C(=O)CC2CCN(C(C3(CC4CCC4)CC3)=O)C2)CCCN2CCCC2C1 89642,Cc1ccc2[nH]nc(C(=O)NC(CNC(C3CCC4CC3CO4)=O)C3CC3)c2c1 89643,CC1=C(c2ccccc2)CN(C(c2cccc(F)c2)C(=O)NCCC2CC2)CC1 89644,N1(C(C(CC)CC)=O)CC(NC(=O)CC2CC3CC3C2)C2(CCC2)C1 89645,N1(C(C(C)OCC#C)=O)CCC2(CC1)CCN(C(c1ccc(Cl)c(Cl)c1)C)CC2 89646,c1(NC(C2CCCN(C(CCCNC(=O)OCC)=O)C2)=O)ccc(F)c(C)c1F 89647,C12(C(N3CC(C=C)OCC3)=O)CCCC1CCN2C(c1cn(C2CC2)cn1)=O 89648,Cc1ncc(Cl)cc1C(N1CC(CO)(NC(=O)C(C)C(F)(F)F)C1)=O 89649,C1(NC(C2(C)CC(=C)C2)=O)CC2CC(NC(=O)C=Cc3c(C)coc3C)CC12 89650,c1(NC(c2ccnc(C)n2)C)ncc(Cl)cc1C(N)=O 89651,Cc1ccc(CC(=O)NC(C)(CNC(=O)C(c2ccccc2)C2CC2)CO)cc1 89652,N1(C(c2cc(Br)cs2)=O)CCC2(CC2C(N2CCOCC23CC3)=O)C1 89653,C(=O)(CC(O)C(C)C)NC(COCC)C(=O)NCc1[nH]cnc1C 89654,C(=O)(C(F)(F)CF)NCCOC1CN(C(C(C)N(CC)CC)=O)C1 89655,c1(C(=O)NC2CCC(NC(c3cn(CC)nc3C)=O)CC2)ccnc(C)c1Cl 89656,C(=O)(C1=C(F)CN(C(C2CC3(CSC3)C2)=O)CC1)N(C)CCC1CC1 89657,Cc1ccc(Br)cc1C(C)NC(N1CCCC(C)(C)C1C(F)(F)F)=O 89658,C(=O)(CCC(F)(F)C(F)F)N(C)CCC1CCN(C(=O)CC2CCOC2)CC1 89659,CCC(C)C(C(=O)N(C)CC1(O)CCCC1)N(C)C(C1CCCC(C)(C)C1)=O 89660,CN1CCN(C(C2CC3(CCO2)CC3)=O)C(C(N2CCCC(C#N)C2)=O)C1 89661,C(=O)(C(C)(C)C1=CCN(C(c2cnc(OC)nc2)=O)C1)N1CCCC(CCC)C1 89662,CCCC(C(=O)NCCN(C1CCCC1)C(c1ccsc1)=O)OC 89663,Cc1cnc2cc(C(N3CCN(C(C4CC=CC4)=O)C(CO)C3)=O)ccn12 89664,C#Cc1ccc(Br)c(C(=O)NC(C)CN(C)C(C2(C)C=CCCC2)=O)c1 89665,C1(C(=O)O)CN(C(c2cnco2)=O)CC12CN(C(c1ccccc1O)=O)C2 89666,c1(OCC(=O)NC2CN(C(=O)CO)C3COCC3O2)c(F)c(F)cc(F)c1F 89667,N1(C(C(C)CN(C)C)=O)CCN(C(C2(CC3CC3)CC2)=O)CCC1C 89668,c1(NC(=O)NCCCn2cnc(=N)[nH]2)ccc(N2CCOCC2)c(F)c1 89669,N1(C2C(=O)NN2C2COC2)CCC(CCOCc2cccs2)C1.CC(C)(C)OCCO 89670,c1(CNC(CC(C)(C(F)F)N(C)C)=O)cc2ccc(F)cc2cn1 89671,CCC(CC)(CCNC(c1ccon1)=O)NC(=O)C(Cc1ccccc1)N(C)C 89672,C1(NC(CC(C)C2CC2)=O)CN(C(c2ccc(O)nc2Cl)=O)CC12CC2 89673,c1(OC)ccc(-c2ncc(C(N3CC4CC4(CN(C)C)C3)=O)s2)cc1OC 89674,C1(N(C)CC=CC(=O)N(CC)Cc2c(C)cnn2C)CC(F)(F)C1.CCO 89675,CC(C(=O)N1CC(NC(=O)CNC=O)C(c2ccccc2)C1)C(F)F 89676,N1(C(C2CC3(CCC3)C2)=O)CCC2CCN(C(C3CCCCS3(=O)=O)=O)C2C1 89677,c1(OC)cccc(C=CC(=O)NC2CC2NC(=O)CC(C)(C)C)c1 89678,C1(c2ccc(C)cc2)CCCN1NC(=O)c1cnn(C2CCCCC2)c1C 89679,C(=O)(C(C)(C)c1cccs1)N(CCOCCNC(CSCC)=O)C 89680,C1(C(=O)NCCCCCCN(C(C=NOC)=O)C)CC12C1CC3CC(C1)CC2C3 89681,C1(COC)CN(C(c2cc(O)ncn2)=O)CCN1C(=O)C(C(C)C)n1cncn1 89682,CCC(COC)C(=O)N1CCCC(NC(=O)C=Cc2cncn2C)C1 89683,C1(CNC(=O)Cn2cncn2)CN(c2nncs2)CCC12CCC2 89684,C(=O)(C(O)CCC(C)C)N1CCN(C(CNC(C2(C#C)CC(=O)C2)=O)C)CC1 89685,c1(OC)cccc(OCCC(=O)N(C(C)CNC(c2cc(C)c(C)[nH]2)=O)C)c1 89686,c1(C(N(C(C)(C)CC(=O)Nc2cnccn2)C)=O)ccccc1O 89687,c1(N2CC(CNC(C3(C)CCNC3=O)=O)OCC2)cncc(C#N)n1 89688,c1(C(N(C)CCOCCCN(C)C(C2CCCC2O)=O)=O)cc2ccccn2c1 89689,C1(COC)CCCCN1C(=O)CC1CN(C(C2COCCO2)=O)C1 89690,N1(C(c2ccn(C(F)F)n2)=O)CCOC(C2CC2)C1 89691,c1(C(=O)OC)cccc(C(N2CC3(CC3)CC2CNC(=O)C=CSC)=O)c1C 89692,N1(C(c2cnn(CC)c2C)=O)CCCC(NC(=O)CC2(CO)CC2)C(F)C1 89693,c1(C(N2CCC(NC(c3c(C)ncnc3)=O)C2)=O)ccc(N)cc1C(C)(C)C 89694,N1(Cc2nc(OC)[nH]c2Br)CCCC12CCNC2=O 89695,N1(C(C2CSCCN2C(c2cccs2)=O)=O)CCc2ncncc2C1 89696,C(CN=c1cccc(S(=O)(=O)NCCC2COCC2O)[nH]1)c1ccc(C)cc1 89697,Cc1c(C(=O)NCC(C)CN(C(=O)CC2CCC2)C)c(-c2ccccc2)cn1C 89698,c1(C(=O)NCCCCCCNC(C2(C#N)C(C)(C)C2)=O)cc(O)cc(O)n1 89699,N1(CC)C(=O)NC(c2c(OC#N)ccnc2Cl)C(C(=O)Nc2ccccc2)=C1C 89700,C1(CN(C)C(C2CC(C(F)(F)F)C2)=O)CCCN(C(C2C3CC(=O)CC23)=O)C1 89701,C(=O)(C1CCCn2cncc21)NC(C)CCNC(c1c(Cl)ccc(O)c1N)=O 89702,C#CCC(C)(CC)C(=O)N1CC(C(=O)NC(c2ccc(F)cc2)C)C(C)(C)C1 89703,C1(CC(=O)NCC2CN(C(C(C3CC3)OC)=O)C2)Cc2ccc(Br)cc2C1 89704,N1(C(C2OCCN(C(CCCOC)=O)C2)=O)CCC(C2CCC2)C1 89705,Cc1c(CC(N2CCC(CCNC(=O)C(C3CC3)C3CC3)C2C)=O)cnn1C 89706,Cc1c(O)ccc(C(=O)NCC2CN(C(C3CC(C)CC(C)C3)=O)CCO2)c1C 89707,N1(C(c2n(C)ncc2C#N)=O)CCC2(CCCN2C(=O)CCS(N)(=O)=O)C1 89708,C(CN=c1[nH]c(N(CCC(C)C)C)nc2c1SCC2)(c1ccccc1F)OC 89709,O=C1CC(CC(=O)NCC2CC(O)(CNC(c3cccc(Cl)c3)=O)C2)C(=O)N1 89710,C1(CNC(c2c(C)cc(C)o2)=O)CN(C(=O)CNC(=O)CC(C)C)CCC1(F)F 89711,N1(C(C2CC23CCCCC3)C(=O)NCCCF)CCCC2(CCCNC2=O)C1 89712,c1(C(C)NCC(C)CF)ccc2nonc2c1 89713,c1(C(N(C2CCN(C(C3CC(O)C3)=O)C2)CC)=O)cnn(CC2CCCCC2)c1 89714,c1(C(=O)NC2C=CC(CNC(C=CCCC)=O)C2)c(C)cc(O)nc1C 89715,CC(O)(C(=O)NCC1CC2CN(C(=O)CCCc3ncco3)CC12)C(F)(F)F 89716,C1(C#N)(C(=O)NC2C(C)N(C(=O)CSc3cccnc3)CC2)CC12CCC2 89717,Cc1nn(C)c(Cl)c1C=CC(N1CCC(O)C(NC(C2CCNC(=O)C2)=O)C1)=O 89718,c1(C(N(C)CC2CN(C(=O)CC3COC(=O)N3)CCO2)=O)ccc2[nH]ccc2n1 89719,c1(C(=O)N(CC2N(C(C(C)=CC)=O)C3C(C2)C3)CC)cccc(Cl)c1F 89720,C#Cc1ccccc1CC(=O)NCc1nc(CNC(C2C=CC=CC=C2)=O)cs1 89721,C(CCCCNC(=O)COCC(C)C)N(C(C1C(C=C)C1)=O)C 89722,n1(CCNC(C2CC(n3ccnc3)C2)=O)cc2ccc(C(=O)O)cc2n1 89723,N1(C(=O)OC(C)(C)C)CCCCC(NC(=O)NC(CO)C2CC2)C1 89724,C1(CNC(C(F)=CC)=O)CCCN(C(C2CN(C(C)C)C2)=O)C1 89725,C(=O)(C1=CCC(NC(C2CSC2)=O)C1)N1CCCC(NC(C)=O)C1 89726,c1(C(N2CCCC2CN(C(C23C=CC(CC2)C3)=O)C2CC2)=O)cccc(O)c1F 89727,c1(C(N(CCNC(C2(CCOC)CCCC2)=O)C)=O)ccc(-n2ccnc2)cn1 89728,C1(C)(C(=O)NCCN(C(C(C)Cc2cccnc2)=O)CC(C)O)CCCN(C)C1 89729,N1(Cc2cc(OC)cc(C)c2)CCC2CN(c3nccc(C)n3)CC2C1 89730,c1(C(N2CCCC(C(C)C(=O)NC3CC(CO)C3)C2)=O)cncn(C)c1=O 89731,C(C)(CNC(=O)CC1CCSCC1)(CO)NC(C(C)=CC)=O 89732,C#Cc1cccc(C(N2CCC(O)(C(C)NC(=O)CCC3CCCOC3)C2)=O)c1 89733,Cn1cnnc1CC(N1CC(CO)(NC(c2ccc(C3CCOC3)s2)=O)C1)=O 89734,c1(NC(C2(C)N(C(c3c(C)nc4sccn43)=O)CC2)=O)cccc2nc(O)oc12 89735,C(=O)(C1=CCN(C(C2C=C(C)CS2)=O)C1)Nc1cn(CC=C)nc1 89736,N1(C(=O)CC2CC3(CC3)C2)CC(C2CN(C(C3C4(CC4)C34CC4)=O)C2)C1 89737,N1(C(CS(=O)(=O)NCC)=O)CCCC2(CNC(=O)CN3CC(C)C3)CCCC12 89738,C1(C(N(C2CCN(C(C3C(C(C)C)CCO3)=O)CC2)C)=O)CC2(CCCC2)CO1 89739,c1(CC)cnccc1C(=O)NC12CC(C(N3CCCCC3CCN(C)C)=O)(C1)C2 89740,C(=O)(N=c1ccnc(C(C)(C)C)[nH]1)C1CCN(Cc2n(C)cnc2)C1 89741,C1(C(N2C(C(=O)NCC3(O)CC3)(CC)CCC2)=O)C2CCC(C2)C1C 89742,CC(CN(C)C)CC(=O)N1CC(O)(CNC(=O)C(C)OC2CCCCCC2)C1 89743,C=CC1(C(=O)NC(CC)CC(F)(F)F)CCN(C(c2cc(C)cc(O)n2)=O)C1 89744,Nc1cc(C(N2CCCC2CNC(C2CCCC23CC3)=O)=O)cnc1Cl 89745,Cc1cnn(C)c1C(=O)NC(C)(C)CC1CCOC1 89746,c1(C(c2nnnn2Cc2cccs2)NCCC=C=C)ccnc(OC)c1 89747,CCCC(C(=O)NCC12CC(CN1C(=O)Cc1cnn(CC)c1)C2)NC(N)=O 89748,N1(C(CC2C(C)OCC2)=O)CCC(NC(=O)Cn2cncn2)C(C)(C)C1 89749,c1(OC(C)C(F)F)ccc(-n2cc(-c3cccc(C(=O)O)n3)nn2)cc1 89750,c1(CCNC(CC(C)SC)c2nnnn2C2CC2)n[nH]c2ccccc12 89751,C=C(C)c1ccnc(NC(=O)NCCc2ccc(F)c(F)c2)c1 89752,n1(CC)cc(Cl)c(C(=O)NC2(CNC(=O)CCCSC)CCCCC2)n1 89753,N12CCC3(CC1)CC3C2.N1(C(c2nc(SC)sc2)=O)CCCC(C(N)=O)C1 89754,c1(C(N2CC(C)(OCC(=O)Nc3cc(N)c(Cl)cn3)C2)=O)ccc(CO)nc1O 89755,O=C1NCC2CN(C(C3(CNC(=O)CC4CCCC4O)CCCC3)=O)CCC12 89756,c1(C(N(CC(=O)NC2CN(C)NC2=O)C)=O)ccc2c[nH]nc2c1 89757,C1(CC(N2CCC(CC(C)NC(=O)CSCCON)CC2)=O)CCC(C)(C)CO1 89758,O=C1Nc2cc(Br)cnc2N2CCN(Cc3ccc(-c4ccc(F)cc4)s3)CC12 89759,CN1C(=O)CN(CC(=O)NCCC2(NC(=O)Cc3ccsn3)CCC2)C1=O 89760,C1(C(N2CC(NC(c3c(Cl)cn(CCC)n3)=O)C2)=O)CC2CCCC(C1)C2 89761,c1(C(N2CC(C3(NC(c4c(SC)ccs4)=O)CC3)C2)=O)c(C)ccc(C)c1O 89762,n1(C(C)C)cc(C(=O)NCC2(F)CN(C(c3ccc(F)s3)=O)C2)c(O)nc1=O 89763,c1(N(C2CCN(C(c3c(OC)ccs3)=O)C2)CCO)nc(C)cc(C#N)n1 89764,c1(C(=O)NCCN(C(=O)C(C)(C)n2cnnn2)CC)cccc(S(C)(=O)=NC)c1 89765,C1(C#N)(C(=O)NC(C=CC(=O)N(CC#CC)CC#C)C)CC(=O)C1 89766,c1(CC)nc(C(C)C)ccc1C(N1CC(NC(=O)C(C)C2CC2)CC(F)C1)=O 89767,C1(CNC(c2cc(C)c(C)nc2C)=O)CN(C(=O)C(C)C(C)C)CCC12CCC2 89768,n1(-c2ccc(CC)cc2)cc(S(=O)(=O)N(c2cc(C)cc(=O)o2)c2cnsn2)cn1 89769,Cn1nc(C(=O)NC(CNC(c2ccoc2)=O)C2CCC2)cc1-c1ccccc1 89770,N1(C(CCC2N(C(C(C=C)OC)=O)CCCC2)=O)CCC(C)(N(C)C)CC1 89771,C1(N(C(C2N(C(C)=O)CSC2)=O)C)CCCN(C(=O)CCc2nc(C)c(C)[nH]2)C1 89772,C1(CNC(CNC(CC(C)(C)C)=O)=O)CN(C(=O)C(=O)NCC(F)F)CC(C)(C)C1 89773,C=CC1(CC(=O)NC(C2CCC2)C)CN(C(=O)C(C)NC(=O)OC)C1 89774,C1(CNC(C2C(C)OCC2)=O)CCCCN(C(=O)Cn2cnc(C(F)(F)F)n2)C1 89775,N1(C(C(N2C(CCC)CCSC2)=O)C)CCC(C)CC1 89776,CCCCC(C)(F)C(=O)NCCC1(C(=O)NC2CN3CCC2(F)CC3)CC1 89777,CCCC(C)C(=O)NCC1CC(COC)CN1C(c1n[nH]c(C)n1)=O 89778,CC1C2C(CCN2C(=O)CC2(O)CCOCC2)CN1C(=O)C=CCF 89779,c1(CC(N2C(CNC(=O)CC3CNC(=O)O3)CCC2)=O)c[nH]c2cccnc12 89780,N1(C(C(CCCC)CC)=O)CC2(C1)CN(C(=O)C(CC)CCOC)CCO2 89781,CC(O)(CC(=O)N1CC2CC1CC2NC(=O)C=Cc1ccco1)CC(=O)O 89782,c1(C(N(C(CCNC(CCC(CC)C)=O)C)C)=O)ccc(=NCCOC)[nH]c1 89783,Cc1cc(N(C(=O)CCCCCNC(c2cnc3n2CCC3)=O)C)cc(F)c1 89784,C1(C(NOC(C(=O)OC)C)=O)(CO)CCCN(C(C2(C#N)CCCOC2)=O)C1 89785,Cc1cc(Br)ccc1CC(N1CCOC(C(C)NC(=O)C2=C(Cl)CC2)C1)=O 89786,C(=O)(CCCC(=O)N(CC(C)NC(c1ccc(OC)c(Br)n1)=O)C)OC 89787,C1(C(=O)NC(C2CCCC2)CNC(CC2(C)OCCO2)=O)CC2CCC(C1)O2 89788,c1(C(=O)OCCN2CCC2C(N)=O)ccc2[nH]nc(C(N(C)C)=O)c2c1 89789,C(=O)(C1=C(Cl)CCOC1)NCC1CCC(NC(=O)Cn2nc(O)ccc2=O)CC1 89790,c1(NC(N2CCN(C(C(C)NC(CC)=O)=O)CC2)=O)ccc(Cl)c(F)c1O 89791,C1(C(N(C)CCNC(=O)C2=CCC2)=O)CC(C)(C)CCO1 89792,C12(CNC(c3cncc(C)n3)=O)CCC1CN(C(=O)CC1CNC(=O)C1)C2 89793,c1(CC)cc(C#N)c(NC(C2(F)CN(Cc3cnccn3)C2)=O)s1 89794,CCC(C(=O)N(C1CN(C(=O)Cc2sc(C)cc2C)CC1(C)C)C)C(C)C 89795,C(C(N=[N+]=[N-])C(=O)NCC1CC(C)N(C(=O)CCCc2ccccc2)C1)OCC 89796,O=C1Cc2ccc(C(N3CC4CCC4(NC(=O)CC4CCSCC4)C3)=O)cc2N1 89797,c1(C(CO)NC(C2CCN(Cc3cccnc3Br)C2)=O)cccc(O)c1 89798,N1(C(c2c(Br)ccc(N)c2)=O)CCC(NC(C2CC2F)=O)C2(CCC2)C1 89799,N1(C(C(CC)SC)=O)CCC(CNC(=O)C=Cc2cccc(OC)c2)C(C)C1 89800,CC1(CNC(=O)C2=COCCO2)CC(F)(F)CN1C(c1cn2ccnc2cn1)=O 89801,CS(=O)(=O)c1cc([N+](=O)[O-])ccc1NCC1CCCC1NC(C1(C(N)=O)CC1)=O 89802,N1(C(CCC2CCCC(=O)N2)=O)CC2CCC(C1)N2C(C1C(Cl)(Cl)C12CC2)=O 89803,CC1=C(C(=O)NC2(C(=O)NOCC(=O)N(C)C)CC2C)COCC1 89804,CC(C)(C)CCC(=O)N1CC(C)(C)CC1CNC(=O)Cn1ccc(C2CC2)n1 89805,N1(C(c2ncc(C(F)F)s2)=O)CCCN(C(C23CCC(CO2)C3)=O)CC1 89806,N1(C(c2ccc(OC)s2)=O)Cc2ccccc2C(NC(c2ccc(Cl)cc2)=O)C1 89807,N1(c2n(CCOCC=C)c(C3CC4(C3)OCCO4)nn2)CCc2c(Cl)cccc21 89808,N1(C(C2CCCN(C(C(C(=O)OC)(C)F)=O)CC2)=O)CCC(C)C(C)(C)C1 89809,c1(OC)ncc(C)cc1-c1ccc(CC(=O)Nc2cc(F)ccc2Br)cc1F 89810,CN1CCC(CC(=O)N(C)CC2CCCN(C(c3cccc(CO)c3)=O)C2)C1=O 89811,c1(C(=O)NC2CC(F)(CNC(CC3(C)CC3F)=O)C2)ncn2ccccc12 89812,N1(C(c2cn(C)c(O)n2)=O)CC2(CCC(NC(=O)CN3CCCNC3=O)CC2)C1 89813,N1(C(C2C(OC)(OC)CC2)=O)CC(C)(C(N2CC(F)CC2CO)=O)CC1(C)C 89814,Cc1cncc(C(N2CC(C(C)NC(=O)C(C3CC3)C3CC3)C2)=O)n1 89815,CC1CC2(CO1)CC(NC(=O)NC1CCCCC1C(C)(C)C)C2 89816,CCC(CC)=CC(=O)NC1(CC(=O)N(C(C)C(F)F)C)CCC1 89817,C#CC1CCCC(NC(C2CC2CCNC(c2cnn(C3CC3)c2)=O)=O)C1 89818,C(=O)(C(C)S(N)(=O)=O)NC1(CNC(c2cnc(OC)s2)=O)CCOC1 89819,C(CCC(C)(C)C(=O)NOCCC(C)C)NC(CC(C(C)C)C)=O 89820,C1(NC(=O)NC2(C)CCC(C(=O)NCC)CC2)C2CCC3C(C2)CC13 89821,Cc1nc(Cl)ncc1CN(CCC(N1CCCCCC1)=O)C 89822,N(C1CC2CCCc3cccc1c32)C(C=Cc1ccc(C(N(C)C)=O)cc1)=O 89823,C1(COC)CC2(CCN2C(C2CSCCN2C(c2cn(C)nn2)=O)=O)C1 89824,c1(C(=O)NC2C(C)CCN(C(C3CCC(=C)CC3)=O)C2)cnc2ccccc2c1 89825,c1(CNC2N(C(=O)NCc3ccc(C)cc3)C(C)CC2)cc(C)ccc1O 89826,C1(N(C(CC(C)O)=O)C)CCCCC1N(C)C(c1cc(CNC2CC2)ccn1)=O 89827,c1(C(=O)NCCCCNC(C2(C3CC3)CCC2)=O)cnc2cc[nH]c2c1 89828,c1(C(N(C2CCN(C(=O)COCCC(C)C)CC2)CC)=O)c(O)noc1C 89829,Cc1nscc1CC(=O)N(C(C)CNC(c1cn(C2CCOCC2)cn1)=O)C 89830,C=CC(C)(C)CC(=O)N1CCOCC1CN(C)C(C1(C)CCN(C(C)=O)C1)=O 89831,c1(COC)nc(=NC(C)CN(C)C(c2ccc(OCCO)cc2C)=O)s[nH]1 89832,c1(C(=O)NC2CN(C(Cc3c(C)ncs3)=O)C(C)C2)cc(N)ccc1C(F)(F)F 89833,C1(CC)C(C(=O)NCc2ccsc2C)CCN1C(=O)Cc1cc[nH]c1 89834,C(=O)(C(C)(C)C(=O)N1CCC(NC(=O)COC(F)(F)F)C(F)C1)NC 89835,c1(CC)ccc(C(N2CCC(C(=O)NC3C4CCC3CC4)C2)=O)cn1 89836,c1(-n2c(C(O)C(F)(F)F)nc(CC(C)OC)n2)cccc2nc[nH]c12 89837,CC1(CO)CCN(C(c2sccc2Nc2ncc3ccsc3n2)=O)CC1O 89838,C(=O)(CCCC(C)C)N(CCC1CCN(CC(=O)NC)CC1)CC 89839,c1(C(N2C(CNC(c3c(C)ccnc3C)=O)CC2)=O)cc2ncccc2cc1Cl 89840,CC1CN(C(c2n[nH]cc2Br)=O)CC(C)C1N=c1ccn2nccc2[nH]1 89841,c1(C(=O)NCC(C)N(C(C(C(C)C)NC(=O)OC)=O)C)cc(Cl)cc(Cl)c1 89842,c1(C(C)(C)C)cnn(C)c1C(=O)NCC=CCNC(=O)CSCc1cscn1 89843,C#CCC(O)C(=O)NC1CCC1NC(c1cnn(C)c1-n1cccc1)=O 89844,C1(CCNC(C2(C)CC(=C)C2)=O)CN(C(=O)Cc2cc[nH]n2)CCS1(=O)=O 89845,Cc1ncc2n1CCN(C(=O)C(C1CCCN(C(=O)CN(C)C(N)=O)C1)C)C2 89846,Cn1ncc(C(N2CCC(C(F)C(N)=O)CC2)C(=O)NCCCC2CC2)c1Br 89847,C1(C(N(CC(F)F)CCC)=O)CCCC2(CCC2)O1 89848,N1(C(C(N2C3CCC2CC3)=O)=O)CCC2CC(NC(c3cccs3)=O)C2C1 89849,C1(C(=O)NCC2CCC(NC(c3c(C)nns3)=O)C2)CC(c2ccncc2)=NO1 89850,c1(C(=O)NC2C3CN(C(C(CCCC)C)=O)C2CC3)cc(Cl)c2c(c1)OCCO2 89851,c1(OC)ncc(CN2CCCC(C(=O)N(C)CCSC)CC2)cc1Br 89852,C1(C(N(CCCCNC(=O)C(=O)Nc2ccccc2)C)=O)CC1C1CCCC1 89853,Cc1cc(C(=O)NCC2(C(=O)NC(c3nncn3C)C)CC2)nc(C)c1 89854,C(=O)(CC(C)CC(C)C)NC(CCC)CC(=O)NCC1(OC)CCCC1 89855,c1(C(=O)NC(CC)CN(C(=O)CNC(C2CCCCC2)=O)C)cccnc1N 89856,CC1CC(NC(=O)CC2CSCCS2)CN(C(=O)CCN(C2CCCCC2)C)C1 89857,c1(OC)ccc(F)c(C(N2CC(c3cn(CC(=O)NC(C)C)nn3)C2)=O)c1F 89858,C#CC1(C(=O)NC2(C=C)CCCC2)CN(C(C2CCCN2C=O)=O)C1 89859,c1(C(N2C(CNC(CCSC)=O)CC2)=O)ccc(NCc2nc[nH]n2)cc1 89860,C1(N(C(=O)Cn2ccnn2)CCOC)CCN(C(=O)C(F)C2CCCC2)CC1 89861,C1(C)(CNC(N2CCC(c3ccc(C)cc3)C2)=O)CCCS1(=O)=O 89862,C(=O)(CCCCCN(C(=O)CCc1ccco1)C)NCC(CC(C)C)O 89863,c1(C(c2cccc(Br)c2)C2CC2)c(Cl)ccc2c[nH]nc12.C12CCN(CC1)C2 89864,c1(C(=O)NC2CCC(N(C(=O)C3=C(Cl)CC3)C)C2)cc2n(n1)CCO2 89865,C1(CNC(C(C)(O)C2CCC2)=O)(NC(=O)CC2(O)CCCC2)CCC(F)(F)CC1 89866,c1(C(=O)NCCCCNC(C2CCN(C(CC)=O)C2)=O)nc(C)c(C)[nH]1 89867,c1(C(=O)NC2CCN(C(CCc3ncc(C)[nH]3)=O)C2)cn2ccn(C)c(=O)c2n1 89868,N1(C(CNC(N)=O)=O)CCCC2CCN(C(c3cn4c(n3)CCC4)=O)CC12 89869,C1(CC(=O)OC)CCCC2(CN(C(c3cc(-c4ccc(Cl)cc4)c[nH]3)=O)C2)O1 89870,Cc1cc(F)c2cc(C(=O)N(C(C)CNC(C3CC(C)(F)C3)=O)C)[nH]c2c1 89871,C(CN=c1cc[nH]cc1S(=O)(=O)N1CC2CC(C1)C(CO)O2)(C1CCCO1)OC 89872,c1(N2CC(SCC)C2)ccc(Br)c(S(=O)(=O)N(C(C)CC#N)C)n1 89873,c1(C(=O)NC2C=CC(CNC(c3n(C)ncc3Cl)=O)C2)ncn2c1CCCCC2 89874,C1(NC(c2c(COC)ncs2)=O)(CO)CCN(C(C2CCCC2)=O)C1 89875,CCCCC(O)C(=O)N1CCN(C(c2cc(I)ccc2Br)=O)CC1 89876,C(C(=O)NCCOC(C1CN(C(C)C)C1)=O)(C1CCCC1)NC(C)=O 89877,C=CCC(C)(C)CC(=O)N1CC(CNC(C2CCN(C)C2=O)=O)OC(C)(C)C1 89878,C1(CC(N2CCC(N(C(=O)CC=C(C)C)CCOC)CC2)=O)OCCCC1(C)C 89879,CCCCCC(O)CC(=O)NCC1CC1CNC(c1ccc(Cl)cc1O)=O 89880,CCC(C)CC(C(=O)NCC(C)(F)C(C)C)NC(=O)CCOCC1CC1 89881,Cc1cnc(C(=O)NCC(c2ccccc2)NC(C2COC(=O)O2)C2CC2)nc1 89882,N1(C(C2CC(F)(F)C2)=O)CCCC(C2(NC(C3(c4ncco4)CC3)=O)CC2)C1 89883,C1(C(=O)NCC(=O)NCC(F)F)CCN(C(=O)c2c[nH]c(=S)cn2)O1 89884,c1(C(NNC(=O)C2N(CC)CSC2)=O)nc2ccccc2[nH]1 89885,C1(C(=O)OC)CC2CCC(C1)N2C(CCSC)C(=O)NN1CC(C)(CC)OCC1 89886,c1(C(=O)NCC(CC(C)C)NC(=O)CCc2cnco2)cn2c(n1)CCC2 89887,C1(NC(c2c(CC)nns2)=O)CC2CN(C(=O)C(N3CSCSC3)C)CC2C1 89888,N1(C(COC)=O)CCC2(CC1)CC(NC(C13COCC1C3(F)F)=O)C2 89889,c12cnc(c(Br)c1)[nH]2.C(C(C)(C)C(=O)NCC1CCN1C(=O)OC(C)(C)C)OC 89890,C1(O)(CC#C)CC(C(=O)NCC2CCN(C(c3occc3C3CC3)=O)C2)C1 89891,C1(NC(CCCC(=C)C)=O)C(C)CN(C(c2cccc([N+](=O)[O-])c2)=O)CC1C 89892,c1(C(=O)NCCCc2cccc(OC)c2OC)c(C)ccn2ncnc12 89893,N1(C(C(C)OCC2CC2)=O)CCC(CNC(=O)Cn2cc(C3CCOC3)cn2)C1 89894,Cc1nc(C(=O)NC2CN(C(=O)CCc3ccoc3)CCC2C)c2ccccn12 89895,CCCCCCC(C)CC(=O)NCCN(C(C1CCC2CC2CC1)=O)CC1CC1 89896,c1(CNC(c2ccnc(Nc3ccccc3)c2)=O)cnc2ccc(F)cn12 89897,C=CCC(CC)C(=O)NC1(C)CCN(C(c2c(C)cccc2O)=O)C1 89898,c1(C(=O)NCCC2OCCN(C(C=Cc3occ(C)n3)=O)C2)cccc(C)c1N 89899,C1(C(=O)NC(CNC(c2nc(O)c(C)s2)=O)CO)(COC)CCCCO1 89900,C1(C(=O)NC2C(NC(C(C)(C)OC)=O)CCCC2)CC2C=CC1CCC2 89901,Cc1ccc(SCC(=O)NCC(C)(O)CNC(c2ccccc2CO)=O)c(C)c1 89902,c1(N(CCNC(C=Cc2cnc(C)s2)=O)CC2CC2)ncc([N+](=O)[O-])cc1Br 89903,C(=O)(CC(CC)C(=O)OC(C)(C)C)NCC(C(C)(C)C)NC(C(CC=C)(C)C)=O 89904,N1(C(C(C)(Cl)Cl)=O)CC2(C)CN(C(=O)C(O)C3CCCC3)CC2(C)C1 89905,O=C(C(O)CC(F)(F)F)OCCN(C(=O)CC(F)(F)F)Cc1ccccc1 89906,n1(CC)cc(CN(C(=O)C(CC2CCC2)NC(C2CCO2)=O)C)cn1 89907,c1(NC(=O)NC(c2ccccn2)C2CCCC2)ccc(Br)c(F)n1 89908,c1(C(=O)NC(C)CN(C(=O)CSC(F)(F)F)C)cccc(N2CCCC2)n1 89909,c1(OC)ccc(CN(C(=O)C(CC(C)C)N2CCCC2=O)C)c(OC)c1 89910,c1(C(=O)NCC(CC)NC(C(C(=O)OCC)(C)C)=O)cc2ccc(C)cn2c1 89911,C1(NC(C2CC=CCO2)=O)CCCN(C(c2ccc(Cl)s2)=O)C1 89912,C1(CCNC(c2[nH]cc(CC)n2)=O)CCCN(C(=O)CCCC#N)CC1 89913,C(C(C)(C)CNC(C1CC1C)=O)N(C(=O)CNC(=O)NC)CC 89914,Cc1cc(C(=O)NCC2(C)CCN(C(c3cc(Cl)c(C)cn3)=O)C2)c(C)nc1C 89915,c1(C(=O)NCC(C)(CO)NC(c2cc(CO)ccn2)=O)cncc(Cl)c1 89916,Cc1cc(CC(=O)NC(CNC(=O)C(F)(F)C(O)C2CC2)C2CCC2)ccc1O 89917,c1(C(=O)NC2CC(NC(C3C(CC)CCC3)=O)C2)cnn(C)c1Br 89918,c1(OC)ccnc(O)c1C(=O)NC1CC2(C1)CC2NC(C1C2CCCC12)=O 89919,C#CC1(C(=O)NCCC(C)(C)CC)CCN(C(C2CC3CCC3C2)=O)CC1 89920,n1(CC#C)cccc1C(c1nnnn1CCCF)N(c1cnccn1)C1CC1 89921,c1(CCCC(=O)NCC2CN(C(CC3(C)CC3(F)Cl)=O)C2)c[nH]c2ccccc12 89922,C(=O)(C(C)(C)CCCN(C(=O)COc1ccc(C(C)(C)C)cc1)C(C)C)OC 89923,c1(C(N2CC(C(=O)NC3(C)CC(C)(C)C3)C(O)C2)=O)ccnc2[nH]cnc12 89924,c1(CCCC(=O)N(C)CCNC(C2(C)CC2(F)F)=O)nc2ccccc2[nH]1 89925,Cn1ccc2sc(C(=O)NC3CC(NC(=O)C=CCN4CCCC4)C3)cc12 89926,N1(C(c2c(N(C)C)nccc2)=O)CC2(CCN2C(C2(C)CCCC2)=O)C1 89927,CCCCCCC(C)(CC)C(=O)NCC1CN(C(c2sccc2Cl)=O)CC1(C)C 89928,Cc1nc(CO)sc1C(=O)NC1COCC1CNC(C1CC(=O)N(C)C1)=O 89929,C1(NC(CC2(C=C)CCCCC2)=O)COC2(C1)CN(C(C1CCCC1(F)F)=O)C2 89930,N1(C(C2CCC(C)O2)=O)CCCC2CN(C(=O)CCc3ccn(C)c3)CCC12 89931,c1(N2CC3(CCN(C)C3)OCC2)nc2c(c(=NCC3CCCSC3)[nH]1)CCC2 89932,C(=O)(C1=CCCOCC1)NC(C1(O)CCN(C(c2c(OC)n[nH]c2)=O)C1)C 89933,C1(C(CNC(C2(CCOC)CCC2)=O)O)CCN(C(C2CC2C)=O)CC1 89934,N1(C(C2(CC(=O)OC)CC2)=O)CCC(O)(C(C)NC(=O)C(C2CCCCC2)F)C1 89935,c1(CC)nc(C#N)cc(=NCC2C(C)CCCN2C(c2cnnc(O)c2)=O)[nH]1 89936,C1(C(N2CC3(C2)C(=O)NC3)=O)CCCC(F)(F)C1.C1(C(N)=O)CCC(CO)CC1 89937,N1(C(C2(SC)CC2)=O)CC(NC(=O)C(CC)c2ccccc2)CC2(CC2)C1 89938,N1(C(C(=O)NC)C)CC(O)(C(C)NC(c2cn(CCC(C)C)nn2)=O)C1 89939,n1(CC)ccc(C(N2CCC(NC(=O)C(C)N3CC(C)C3)C2C)=O)c1C 89940,Cc1cc(C(C)C(N2CCC(Cn3cc(CCCO)nn3)C2)=O)c(C)o1 89941,CCCCC(CC)CC(=O)NCCCOCCNC(=O)C=Cc1cscn1 89942,C1(CC(=O)N(CCN(C(C(CC)(F)F)=O)C)C)Cc2ccc(Cl)cc2C1=O 89943,c1(OC)c(F)ccc(C)c1C(=O)NCCN(C(=O)Cc1cccs1)CCOCCO 89944,C12(CC(=O)NCCCCCC=C)CCC1CN(C(=O)Cn1ccc(C)c1)C2 89945,CCCCCCCC(=O)NC1CC(NC(=O)C(C)(C)C2CCCO2)CC1O 89946,CC1CC(=O)NC1C(=O)NCCCNC(C1CCC(C)CC1)=O 89947,CC(O)(C(=O)NCC1CCC(NC(=O)Cc2nccs2)C1)C1CC1 89948,N1(C(C23CC(CC(F)F)(C2)C3)=O)CCC2(CCCN(C(=O)C3=CCCC3)C2)CC1 89949,C1(C)(CNC(C2(CCN(C)C)CC2)=O)CN(C(=O)CC2CCCO2)CCO1 89950,c1(CC(N2C(CNC(Cc3c(C)n[nH]c3C)=O)COCC2)=O)ccc(C#N)cc1 89951,CN1CC=C(CC(=O)N2CC3(CCC3NC(c3csc(Cl)c3)=O)C2)CC1 89952,N1(CC(C(C)C)C)CC2CCC1C1CN(C(c3csc(C(C)C)n3)=O)CC21 89953,N1(C(c2c(CC)con2)=O)CCC2(CC(NC(=O)CS(=O)(=O)CCOC)CO2)C1 89954,n1(CC)cc(C(=O)NCC2CC(COC)CN2C(=O)CC2CCC(=O)C2)c(C)n1 89955,C1(NC(C(C)CN(C)C)=O)CC2CN(C(c3csc4nnsc34)=O)CC12 89956,C=C(C)CCCC(=O)N1CCCC(C(=O)NC2COC(C(C)C)C2)C1 89957,N1(C(C2C(C(=O)OC)C2)=O)CCC(NC(c2cn(C3CCC3)nn2)=O)C(O)C1 89958,C1(CC)(CC)CC(NC(=O)C(C)C(C)C)CN1C(c1cnc(OC(C)C)nc1)=O 89959,C=CC1(CC(=O)NC(C)(CNC(=O)Cc2cncs2)C2CC2)CC1 89960,Nc1cc(C(N2CCCC(F)(CNC(C3CCCCC3O)=O)C2)=O)c(F)cc1F 89961,c1(C(=O)NC(CNC(C(CC)(C)CO)=O)CO)ccc2c(c1)OCO2 89962,N1(C(C(C)NC(CC)=O)=O)CC(CNC(=O)CC(O)C(C)C)OC(C)(C)C1 89963,c1(C(=O)NCC(CO)NC(=O)CNC2CC3C=CC2O3)ccc2ccccc2c1 89964,Cc1cccc(Cl)c1CC(N1CCC(CO)C(C(F)(F)F)C1)=O 89965,C1(CNC(C(=O)N(CC=C(C)C)C(C)C)=O)CC(CO)CO1 89966,c1(CC)ccc(C(=O)NC(CNC(=O)CCc2cnn(C)c2)CC)cc1Cl 89967,c1(OC)cnccc1C(=O)NCCc1n[nH]cc1C(=O)NCC(C)(O)CCO 89968,c1(C(=O)NCCCC2OCCN(C(C(C)C(F)(F)F)=O)C2)noc2ccccc12 89969,N1(C(c2c(CC)c[nH]c2)=O)CC2CCCCC2(CNC(=O)CSCC(F)(F)F)C1 89970,C1(NC(c2csc(-c3cn[nH]c3)n2)=O)CN(C(c2cc(Cl)no2)=O)C2(CCC2)C1 89971,CC1CC(CC(=O)N(C)CC2CCCN2C(c2coc(Br)c2)=O)C(C)O1 89972,N1(C(C2C(OC)(OC)CC2)=O)CC(NC(=O)Cn2nnc(C3CC3)n2)C2(CC2)C1 89973,C1(C(N(CC(C)O)CCNC(c2cnsn2)=O)=O)CCn2c(O)nnc2C1 89974,C1(NC(c2n(C)ccn2)=O)CCN(C(C2OCC2(C)C)=O)C12CCC2 89975,CC(F)(F)CC(=O)NC1CC1NC(=O)COCc1ccncc1 89976,C1(NC(C(C)=C2CC2)=O)CCC(CNC(=O)C(C)Cc2cccnc2)C1 89977,c1(C(=O)NCC(CC)NC(C2C=CCC2)=O)c(Br)c(C)nn1C(C)(C)C 89978,C1(CC(=O)NCC(C)CNC(=O)COC2CCOCC2)CCC(=O)NC1 89979,C#CCC(C)(C(=O)NCCc1ccncn1)NC(C1CC(OCC)C1)=O 89980,N1(C(CCOCC(C)C)=O)CCCC(C2(NC(C3CCNC3=O)=O)CC2)C1 89981,S(=O)(=O)(c1ccc(=NCC2CCCCCC2(F)F)[nH]c1)N(C)Cc1cccnc1 89982,c1(C(N2CCC(C(=O)NCC(=C)C)CC2)=O)cc(C)ncc1C 89983,c1(C(N(CC(CC)NC(=O)C(F)=CC2CC2)CC)=O)c(C)cc(OC)cc1F 89984,N1(C(C(C)Sc2ccccc2)=O)CC(NC(c2cc(F)cc(Cl)c2)=O)CC(F)C1 89985,CCC(C(=O)N1CCOCC(C(=O)NC(C2CCOCC2)C)C1)C(F)(F)F 89986,c1(OC(=O)CCNCC2CCCN2CC2CCOC2)ccccc1Cl 89987,N1(C(c2c(C)nc(CO)s2)=O)CCC2CN(C(=O)Cn3ccccc3=O)CCC12 89988,CC1Cn2nc(C(N3CC(CNC(C4CCCC(F)(F)C4)=O)C3)=O)cc2C(=O)N1 89989,c1(C(C)C)cccc(CN2CC3(CC3C(=O)NC3(c4ncccn4)CC3)C2)c1O 89990,N1(C(C2(C)CCCN(S(CC(C)C)(=O)=O)C2)=O)C2CCC1CC(CO)C2 89991,N1(C(C(C)n2ccnn2)=O)C2CCC(C2)C1C(=O)NCC1(F)CCOCC1 89992,C(C(C(=O)NC1CC1)N1CCCC(c2ncc(C)s2)C1)(C1CC1)OC 89993,N1(C(c2c(CC)nccn2)=O)CCN(C(C23COC(CF)(C2)C3)=O)C2CC12 89994,N12CCN(Cc3ccc(I)cc3)CC1C2.N1(S(C)(=O)=O)CCN(CCC#N)CC1 89995,C1(NC(C=CC(C)C)=O)CCCN(C(=O)CC2(C)CC2(F)F)CC1 89996,N1(C(c2cc(CNC(c3[nH]cc(C)c3)=O)[nH]n2)=O)CCC(C)(N(C)C)C1 89997,C1(CNC(Cc2c(C)nsc2)=O)CC2(C1)CN(C(C1CCCN1C)=O)C2 89998,c1(C(N2CCC(C)(NC(C3CCC(CC)C3)=O)CC2)=O)[nH]nc2c1CCC2(C)C 89999,C1(NC(C)=O)Cc2ccccc2N1.c12ncc(o1)C(CC(C)C)N(C1CC1)C2 90000,c1(CN2CC(C#N)N(C(c3ccccc3S)=O)CC2)ccc(F)c2ccoc12 90001,C(=O)(C(O)CCCNC(=O)CC1CCOCC1)N1CCN(CC=C)CC1 90002,Cc1cscc1NC(C1CCC(CNC(=O)CCc2cnn(C)c2)C1)=O 90003,C1(NC(CC(C)c2ccncc2)=O)CN(C(=O)CSc2nncs2)CC1C 90004,N1(C(COCCC#C)=O)CCN(C(=O)C(O)CC(C)C)C(c2ccccc2Cl)C1 90005,c1(C(N2C(C(N(C3CC(C)(C)C3)C)=O)CSC2)=O)cc(C#N)cs1 90006,c1(C(CC)C)ccc(=NCCCOCCc2ccccc2)[nH]n1 90007,C(=O)(CCCC(CC)NC(=O)COCCC(C)C)N1CC2(CC(=C)C2)C1 90008,c1(C(N2C(CNC(C3(CCOC)CC3)=O)CC2)=O)cc(C)c2c(c1)CCC2 90009,CN1CCN(C(=O)CC2CCC3CC3C2)C(CNC(=O)Cc2cncnc2)C1 90010,Cc1cn2cc(C(=O)NCCOCCNC(c3ccn4ccnc4c3)=O)nc2s1 90011,N1(C(C(c2cccc(OC)c2)(C)C)=O)CC2(CC(NC(=O)CCC(C)OC)C2)C1 90012,c1(C(=O)OC)nc(NC2C3CC2CN(C(c2ccccc2)=O)C3)cnc1C 90013,N1(C(c2c(C)noc2)=O)CCCC(C(N2CC=CC2CN(C)C)=O)C1 90014,c1(OC)nn(C)cc1C(=O)NCC1(NC(=O)C=CS(C)=O)CCOC1 90015,Cc1c(CC(N2CCOCC(C)C2)=O)sc2ccccc12 90016,C1(C)(C(=O)NC2CC(C)(C(N3CC(NC(COC)=O)C3)=O)C2)CCCCCC1 90017,C(=O)(CC(C)CNC(C1CCS(=O)CC1)=O)N(C(C#C)C1CCC1)C 90018,c1(NCC2N(C(c3cc(C4CC4)ncn3)=O)CCC2)c(F)cccc1[N+](=O)[O-] 90019,Cc1ccc(C(=O)NCC(C)(CO)NC(=O)CC(C)c2ccncc2)n1C 90020,c1(C(=O)OC)cc(C(=O)NCC2CN(C(=O)C(C)(C)SC)CCC2C)cc(F)c1 90021,c1(C(N2CC3C(NC(C4CC(C)(O)C4)=O)C(CC3)C2)=O)csc2c(Cl)cccc12 90022,c1(NC(c2cccc(F)c2O)=O)ccc(-c2ccc(Cl)cc2C(=O)O)cc1F 90023,C(=O)(C1=NOC(C)(C)C1)NC1C(NC(c2c(C)nc[nH]2)=O)CCCC1 90024,C1(NC(C(CCC2CC2)NC(C(CC#C)O)=O)=O)CCc2n[nH]cc2C1 90025,N1(C(CC2C3CN(C(c4c(COC)cc[nH]4)=O)CC32)=O)CC=CC12CCOCC2 90026,C#CC1CCCCN1C(=O)CSCCNC(=O)C(=O)CC(C)C 90027,c1(C(N(CCN(C(C(C)N(C)C)=O)C)C(C)C)=O)cccc2c1OC(C)C2 90028,C(=O)(C#CC(C)(C)O)N1C(C(=O)NC(c2ccncc2F)C)CC(OC)C1 90029,N1(C2CC2)C(C=O)CC2CC12.c12cc(no1)C(=O)NC2.C(C)(COC(C)C)SC 90030,c1(C(=O)NC(C2CC=CCC2)C(N2CCC(=C)C2)=O)cnc(O)cc1C 90031,c1(CC)nc(C)c(CC(=O)NC(C)(C)CCNC(=O)Cc2csc(C)c2)c(C)n1 90032,C1(NC(CC(CCC)C)=O)CCSC12CN(C(c1ccc(N)cc1OCC)=O)C2 90033,N1(C(CCc2cccc(C)c2)=O)CCCC(C(=O)NCC2CSCCO2)CC1 90034,C=CCCC(C(=O)NCC1(C2CC2)CCC1)NC(=O)CC1COC(=O)C1 90035,c1(C2(C(N3CCC(NC(C(COC)C)=O)C3)=O)CC2(C)C)cccc(Cl)c1 90036,C1(CNC(Cc2c(C)noc2Cl)=O)CN(C(C2(C)CC(=O)N(C)C2)=O)CCCO1 90037,c1(C(=O)NCCC(C)(C)NC(C2CC2(Cl)Cl)=O)cnc2occc2c1 90038,N1(C(C(C(C)(C)C)OC)=O)CCC(C(=O)NCC(CC(C)C)N(C)C)C12CCC2 90039,C(C)(C(C)(C)C(=O)NC1CC2CCCC2C1)NC(C(C)C)=O 90040,Cc1cc(NC(=O)CCN2CCCC2)ccc1NC(C1CC(=C(F)F)C1)=O 90041,N1(C(c2cnc(Cl)s2)C(=O)NCCCC(=O)OCC)CCN(CC(C)O)C(C)C1 90042,CC(C)CC(C)CC(=O)N1CCCCC1C(=O)NC(c1cscn1)C 90043,C1(CNC(C#CC(C)C)=O)CCCC12CCN(C(=O)CC1OCCC1C)CC2 90044,C1(NC(C2(SC)CC(O)C2)=O)CN(C(c2ccc(F)cc2)=O)C2(CCC2)C1 90045,N1(C(C(CC)C)=O)CC(CO)C2(C1)CN(C(=O)C(c1cccc(Cl)c1F)(C)C)C2 90046,c1(-c2ccc(NCc3c(Br)ccc(C#N)c3)c(F)c2)cc2ccccc2cc1O 90047,CC(C)C(C(C)NC(=O)CCn1cncn1)NC(=O)Cc1ccc(O)cc1 90048,C1(C(N(CCC)C(C)C)=O)CN(C(=O)C(C)NC(C)(C)CC)CCO1 90049,CCC(C(=O)N(C(C)CCNC(c1ccc(S(N)(=O)=O)o1)=O)C)C(F)(F)F 90050,CN1CCC(O)C(NC(C2CC(NC(c3cnn4c3CCC4)=O)C2)=O)C1 90051,c1(C(N(CCCNC(C(C)c2cncs2)=O)C2CC2)=O)cc(N)c(Cl)c(O)n1 90052,C1(C(=O)NCCN(C(=O)C(O)CC(F)F)C)CC12CCCCCC2 90053,CN1CC(C(N2CCC(OCCONC(C(C)(C)CCF)=O)C2)=O)CCC1=O 90054,C1(C)(c2ccc(NC(c3c(C)non3)=O)cc2)NC(=O)NC1=O 90055,c1(NC(c2c(Nc3nc(C)cc(OC)n3)c[nH]n2)=O)cc(F)c(Cl)cc1Cl 90056,N1(C(Cc2ccnc(OC)n2)=O)CCN(Cc2ccccc2)C(C(F)(F)F)C1 90057,C1(NC(C2C(=C)CC2)=O)CN(C(c2cc3c(s2)CCC3)=O)CCC1C 90058,C1(C(=O)NCCCN(CCCNC(c2ccc(F)cn2)=O)C)Cc2nccn2C1 90059,C1(CCCC=C)CCCCN1S(=O)(=O)N=S(C)(=O)CCO 90060,c1(C(N(CCN(C(Cc2c(C)noc2)=O)C)C)=O)cc2c(F)c(F)c(F)cc2[nH]1 90061,CC1(C)CN(C(=O)CC2(O)CC2)C1C1CCN(C(C2CCS(=O)(=O)C2)=O)CC1 90062,c1(C(=O)NC(CCNC(C(CCC)C)=O)(C)C)cc([N+](=O)[O-])c[nH]1 90063,S(=O)(=O)(c1cc2c(cc1Cl)CCCC(=O)N2)N1C(C)(COC)CC(N)C1 90064,CC(C)(CS(C)(=O)=O)C(=O)NCC(C)(C)CNC(c1cnc(N)c([N+](=O)[O-])c1)=O 90065,Cc1cc(F)sc1C(=O)NC1CCC(CC(=O)NC2(C(=O)NC)CCCCC2)C1 90066,Cc1cccc(C(O)CN(c2cc(C#N)no2)Cc2ccccc2)c1 90067,Cc1cc(=NC(=O)C2CCCC(NCc3cnc(-c4ccccc4)s3)C2)[nH][nH]1 90068,c1(OC)cccc(NC(C2CN(C(=O)CC3CCCCN3C)CC2OC)=O)n1 90069,c1(OC)ccc(-c2ccccc2)cc1CN(CC(O)C1CCC1)C 90070,C=CCC(CC(F)F)NC(=O)COC1CCN(C(=O)C(C2(O)CCCC2)F)C1 90071,Cc1ccn2ncc(C(N3CCC4CC3CN4C(c3ccc(Cl)cc3)=O)=O)c2c1 90072,C(=O)(CCC(CF)CF)N1C(C)C(NC(=O)CN2CCOCC2=O)CCC1 90073,c1(CC)nc(Cl)[nH]c(=NC2CC(NC(=O)Cc3ccc(C)cc3C)C2)c1Cl 90074,C(C(CC(=O)NCCNC(N)=O)C1CCC1)NC(C(CC)OC)=O 90075,C12(C(N3CCC(OC)CC3)=O)CCC(NC(C3(C)CC=CCC3)=O)(CC1)CC2 90076,C1(OC(c2ccc(CS(=O)(=O)C(F)F)cc2)=O)CN2CCC1CC2 90077,Cc1cc(C(=O)N(C2CCN(C(c3ccc(C#N)cc3)=O)C2)CCO)ccc1Br 90078,C1(NC(c2cc(C3(C)CC3)on2)=O)CCCCC1CNC(C1(Cl)CCC1)=O 90079,N1(C(C2(CC)CCNC2=O)=O)CCn2c(CNC(c3cn(C)cn3)=O)nnc2C1 90080,N1(C(C=C(CCC)C)=O)CC(NC(=O)Cn2nnc3ccccc23)CC(C)(C)C1 90081,c1(C(=O)Nc2c(C)cc(C)nc2)cc2n(n1)CCCN(C(=O)C(C)O)C2 90082,CCC(C)C(C)C(=O)NCC1(F)CC(NC(=O)CCc2ncc(F)cn2)C1 90083,CC(C)CC(O)C(=O)NC(C1CN(C(=O)CCCn2ccccc2=O)C1)C 90084,C(=O)(CC(C(F)(F)F)NC(c1ccccc1F)=O)NC(c1n(CC)ncc1)C 90085,c1(C(N2CCC(O)(C(C)CNC(c3cccnc3)=O)C2)=O)csc2ccncc12 90086,N1(C(C=CCOCCOC)=O)CC=CC(NC(=O)CCCn2c(C)csc2=O)C1 90087,C1(C(=O)NC2C(CNC(C3(COC)CCCC3)=O)CC2)CCCS(=O)(=O)C1 90088,c1(C(=O)NC2CC(C)N(C(C3C4CC5C(C4=O)C35)=O)C2)ccc2c(c1)CCOC2 90089,C(=O)(C(C)(C)CCCOC)NCCONC(=O)COC(C)(C)CO.CCO 90090,c1(C(=O)NCC(C(C)(C)C)CO)cnc2cnc(Cl)cc2c1 90091,CC1(C)CN(C(=O)Cn2cccnc2=O)CC1NC(c1c[nH]cc(F)c1=O)=O 90092,c1(C=O)cccc(CF)c1.C1(C(CNC(CCC)=O)(C)C)CCCN1C(=O)CCC 90093,c1(N2C(CNC(CS(CCOC)(=O)=O)=O)CCC2)cc2c(cn1)C(=O)CCC2 90094,N1(C(CNC(C)=O)=O)CC(c2ccccc2)(N)C1.C1(C(=O)N)CC1Br 90095,c1(C(N(CC(C)NC(=O)C(C)(C)c2ccns2)CC)=O)ccc(Br)cn1 90096,N1(C(c2[nH]nc(OC)c2Cl)=O)CCCN(C(c2ccc(C(F)F)cc2)=O)C(C)C1 90097,CCC(C)(CCNC(=O)Cc1ccccc1F)NC(=O)CC1CCCCO1 90098,Cc1ncc(C(=O)NCC2(CNC(C3CNC(=O)C3)=O)CC2)c(C(C)C)n1 90099,C(=O)(C1=CCCC(C)(C)C1)NC(C1CCCN(C(c2ccc(SC)cc2)=O)C1)C 90100,N1(C(CCCC(=O)OC)=O)CC2CN(C(C3CCC(C)CC3)=O)CC2(C)C1 90101,c1(C(=O)NC(C)CC2CN(C(=O)CSC(F)F)C2)cccc(NS(C)(=O)=O)n1 90102,c1(C(N(CCNC(c2ccc(-n3ccnc3)nn2)=O)CC)=O)cc(Cl)nnc1O 90103,C1(NC(CCSC)=O)CCCN(C(c2ccc(C(F)(F)C(Cl)Cl)cc2)=O)C1 90104,c1(OCCC)cccc(-c2cccc(OCC3(C)CC3)c2)c1 90105,CC(C)(C(=O)NC1CCC(CNC(C2(CO)CCCO2)=O)C1)S(C)(=O)=O 90106,c1(C(C(=O)N(CCC)CCNC(=O)Cc2ccno2)N(C)C)ccccc1 90107,CC1(C(=O)NC2CC(CNC(=O)Cn3nnc(-c4ccccc4)n3)C2)CC(F)C1 90108,C1(N(C(CCC=CC)=O)C)CN(C(C2(COC)CC2)=O)CCC1O 90109,N1(C(CCCOCC)=O)CC2CC(NC(c3cnsc3C)=O)CC2C1 90110,N=c1nc(C(N2CC=CC(NC(C3CC(O)C3)=O)C2)=O)cc[nH]1 90111,C1(C2CCCN(C(=O)C3=CCC(C)CC3)C2)(NC(C2C(C3C(C)C3)C2)=O)CC1 90112,c1(C(=O)NCC2OCCN(C(CC3(C=C)CCC3)=O)C2)cc(C#N)c(O)nc1N 90113,Cc1cccc(NC(C23CC2CN(C(c2ccc(CO)cc2)=O)C3)=O)n1 90114,N1(C(C2(CC)CC(C)(C)C2)=O)CC(C)OC2(CCN(C(=O)CSC(C)C)CC2)C1 90115,C(=O)(C1=NOC(C)C1C)NCCC1(CNC(c2c(C)ccnn2)=O)CC1 90116,N1(C(c2ncncc2Cl)=O)CCN(C(c2nc(Cl)cs2)=O)CC(O)C1 90117,N1(C(C(C)SC(C)C)=O)CCc2ccccc2C1CNC(c1cnn(C)c1C)=O 90118,C(=O)(C(C)CC(F)(F)F)N(CCN(C(C)C)C(C1CC1C1CC1)=O)C 90119,C(C(C(=O)NCCC(C)CO)C(C)(C)C)NC(C(CC)(C)CC)=O 90120,C1(NC(CC(C=C)(C)O)=O)CC2CCC(C1F)N2C(c1ccccc1F)=O 90121,c1(C(N(CC(C)NC(=O)C=Cc2ccoc2)CC)=O)cnc2[nH]ncc2c1 90122,C1(NCCNC(C2CCCCC2)=O)COCC1F 90123,CCN=c1cc(-c2cn(CCCCNC(c3cccc(F)c3)=O)nn2)cc[nH]1 90124,N1(C(C(C)C2(O)CCC2)=O)CC2CCC(C1)N2C(C1CCC(C)(C)CC1)=O 90125,C1(CNc2c(OC(CC)C)cccn2)CCCC2(CC(C(=O)O)C2)O1 90126,C1(C(CNC(COCCOC)=O)NC(C2CN(C)C2)=O)CCCCC1 90127,C(=O)(C1Cc2ccccc21)NC(CCCC)CNC(c1cccc(C)c1CC)=O 90128,CCC(C)CCC(O)CC(=O)N(C1CCCN(C(=O)C2=CCOC2)C1)C 90129,Cc1nn(C)c2cc(NC(C3CC4CC4N3C(c3cc[nH]c3)=O)=O)ccc12 90130,C(Cc1cnc[nH]1)(C(=O)NCCN1CCC1)NC(=O)Cc1ccon1 90131,c1(C(=O)NCCCC(C)NC(CCC=C=C)=O)cc2c(nc1O)CCCC2 90132,C1(CC(=O)NC2(C)CN(C(C(C)CC3CC3)=O)C2)CCCC1(F)F 90133,Cc1cncc(C=CC(=O)NCCC2CCCCN2C(c2occc2C)=O)c1 90134,c1(C(N2CCCC(CNC(c3sccc3I)=O)C2)=O)cccc(F)c1I 90135,Cc1cc(C(=O)NCC(C)(C2CC2)NC(=O)CSC(F)F)cc(C)c1N 90136,N1(C(c2c(OC)c[nH]n2)=O)CC2CC(O)C1C2NC(c1ccc2nnnn2c1)=O 90137,c1(N2CCC=C(C)C2)[nH]c(=NCCc2cccs2)nc2c1ncn2C(C)C 90138,C1(CNC(c2n(C(CC)C)ncc2)=O)CN(C(c2snnc2C)=O)CCCO1 90139,c1(C(N2CC(C)C(CNC(=O)COc3cn[nH]c3)C2)=O)nc2ccc(Cl)nn2n1 90140,N1(C(C2CC3(CCN2C(=O)CC2(O)CCC2)CC3)=O)CCC2(CCC(O)C2)C1 90141,N1(C(C2N(C(C)C)CCC2)=O)CCC(C)(C)C(C(=O)N(C2CCOC(C)C2)C)C1 90142,N1(C(C(COC)O)=O)CCC(C2CCN(C(=O)C(C)(C)C(C)(F)F)C2)CC1 90143,CCCC(C)(C)CC(=O)N1CCC1CNC(=O)CCc1cn(C)nc1C 90144,c1(C(N2CC(C)CC(NC(CCCC=C)=O)C2)=O)c(C)[nH]c2ccc(Cl)cc12 90145,C1(C(=O)NC2(C3N(C(C(C(CC)C)C)=O)CCC3)CC2)CN2CCN1CC2C 90146,c1(C(=O)NCC(CCOC)NC(C2CC2(Cl)Cl)=O)ccc(CO)c(OC)c1 90147,c1(C(N(C)CCNC(=O)CCC2CCCOC2)=O)cccc(S(N)(=O)=O)c1 90148,N(C1CC(C)n2ncnc21)C(CC)CCc1ccccc1 90149,c1(NCC(C(C)C)(C)NC(=O)CCn2ncn(C)c2=O)ncc2c(n1)COC2 90150,C1(C(=O)NCC(CNC(=O)C(C)CN(C)C)OC)CC2CC1CC2(F)F 90151,c1(C(=O)NCCC(CCNC(C(C)N(C)C)=O)C)cnn2c1S(=O)(=O)NCC2 90152,c1(C(=O)NCC2OCCC(NC(C(C)(C(C)C)OC)=O)C2)cc(F)cc(N)c1F 90153,C1(NC(c2ccon2)=O)CCC2(CCCN(C(C3CCCO3)=O)C2)C1 90154,c1(NC(c2n(CCOC)nnn2)c2csc(Br)n2)ccc(C)c(O)c1C 90155,C1(NC(CCN(C(COCCC#C)=O)C)=O)CC2CC2C1 90156,c1(CC(=O)N(C2CC3CNC2C3)c2c(C)onc2)cccc(F)c1 90157,CCC(C#N)(CC)C(=O)NC(C)CCNC(C1CC2(C1)CC1(CC1)C2)=O 90158,C1(F)(C(=O)NC2C(NC(C3N(C)CCCC3)=O)COCC2)CCC(F)(F)CC1 90159,C=CCC(CC(C)C)C(=O)NCC1CCCC1NC(c1cc(COC)[nH]n1)=O 90160,C=CC(C)(C)CC(=O)N(C(C)CN(C(=O)CC1C(C)C1(F)F)C)C 90161,C12(C(=O)NC3C(NC(C4CC5(CCC5)C4)=O)CCC3)CC3CC(CC1C3)C2 90162,c1(C(N2C(CNC(CN=S(C)(C)=O)=O)CC2)=O)cc(Cl)ccc1[N+](=O)[O-] 90163,C#CC1CC2(CC2)CN1C(=O)C(C)N(C(c1cc(C(C)=O)c[nH]1)=O)CC 90164,C1(NC(CCCCC(CO)NC(=O)OC(C)(C)C)=O)CS(=O)(=O)CC12CC2 90165,c1(C(N(C(CNC(C2(SC)CC2)=O)C)C)=O)cc(Cl)nnc1Cl 90166,c1(CCC(=O)NC2CCC(NC(c3ccn(C4CCC4)n3)=O)C2)ccccc1Br 90167,N1(C(C2CCC(=C)CC2)=O)CC2CCOCC2(NC(=O)CCC(C)C)C1 90168,C1(N(C(C2CN(C(C)C)C2)=O)C)CN(C(=O)C(C)C2CC2)CC12CC2 90169,C=CC(CCC)CC(=O)N1CCCC1C=CC(=O)N(CC)OCC 90170,c1(C(=O)NCC(CNC(C2C(CC)CC2)=O)O)nccc(C)c1N 90171,c1(Cn2cc(C(C)NCc3ccc(-c4cccnc4)cc3)nn2)ccc(Br)cc1F 90172,N1(C(C=C(C)C(C)C)=O)CC(C(=O)NC(C)Cc2nc[nH]n2)C2(CC2)C1 90173,c1(C(=O)NCC2CC(NC(c3c(C)coc3)=O)C2(C)C)ccc(C)c(C(F)F)c1 90174,C=C(C)CCC(C)NC(=O)CC1CN(C(=O)CN2CCSCC2)CCO1 90175,c12cc(ncn1)CC1(CNCC1)C(=O)N2C1CC2CCC1C2.n1(CC)cc(Br)cn1 90176,CC(CN(C)C)C(=O)NCC(C1CCCC1)NC(C12CC(C1)C2)=O 90177,c1(OCC(N2CCC(Oc3ccc(C)cc3)C2)=O)c(F)cc(I)cc1F 90178,c1(NC(C2N(Cc3ccc(C)[nH]3)CCCC2)=O)nc(Cl)c(C)cc1[N+](=O)[O-] 90179,C1(NC(C2(CN(C)C)CC2)=O)CCC2(CC1)CN(C(C1CCCCS1)=O)CCO2 90180,CCCCC(C)C(=O)NC1CCCCCC1C(N1CC[Si](C)(C)CC1)=O 90181,N1(C(C(C)N2CCCC2)=O)CCCCC(CC(=O)NOC2CC23CCCCC3)C1 90182,S(=O)(=O)(c1cccc2ccccc12)N1CCOCC(NC(C(C=C)O)=O)C1 90183,C(CCC(CCC)NC(c1oc(SC)cc1C)=O)NC(CC(=C)C)=O 90184,N1(C(C(C(C)OC)O)=O)CC2(CCCCN2C(c2cnc3c(c2)CCCC3)=O)C1 90185,N1(C(CC(=O)NC)=O)CCCC(CC)C1C(N1CCCC(NC(C)=O)C1)=O 90186,N1(C(c2cc(C)c(C)nn2)C(=O)NCC2CCOCC2)CCC12CCSCC2 90187,c1(NC(C)=O)ccc(C(C(=O)NCCC#N)N(C)CC2CCCCC2O)cn1 90188,c1(C(N2CC3C(CNC(c4ccc(C#N)s4)=O)(C3)C2)=O)cnc2ccc(F)cn12 90189,C1(N(C)C(C2CC(F)(CF)C2)=O)CCCN(C(=O)COCCCF)C1 90190,c1(C(C(=O)NC(c2cnn(C)c2)C)O)ccc([N+](=O)[O-])cc1 90191,C(=O)(C(C)C1OCCc2sccc21)N1C(C(=O)OC)CC1.C12CC(C1)C2 90192,C1(CC)CN(C(C2(OC)CCOCC2)=O)CCN1C(c1occ2c1CCC2)=O 90193,CC1(NC(=O)CCc2cc(Cl)cc(Cl)c2)CCC(NC(C2CC(C)(O)C2)=O)CC1 90194,c1(CC(=O)NC2CC(NC(=O)Cc3cnc[nH]3)C2)csc2ccc(Cl)cc12 90195,c1(C(=O)NC2(C)CC(NC(=O)C(F)n3ccnc3)C2)nc(Cl)ccc1N 90196,Cc1c(C(=O)NCC2(C(C)NC(C3CCCN(C)C3)=O)CC2)nnn1C(C)C 90197,Cc1c(C(=O)NC(C)C(C)NC(c2ccc(Br)o2)=O)cncc1Br 90198,N1(C(c2c(C)nc(-c3ccccn3)s2)=O)CCC(C)C(NC(=O)C=CC2CC2)C1 90199,c1(NC(=O)C(=O)NCC(CC)C(=O)OCC)ccc2c(c1)CCCS2(=O)=O 90200,C(C1CCCCC1)=CC(=O)NC(CNC(CC(C)OC)=O)C1CCC1 90201,C1(CNC(c2c(C)cncc2)=O)N(C(c2nc(=O)n(C)[nH]2)=O)CCC1(C)C 90202,c1(NC2CN(C(=O)NCc3cccc(C)c3)CC(F)C2)ccc(Cl)c(C)c1F 90203,c1(C(=O)NC(CCCNC(C(C(C)C)OC)=O)(C)C)ncn2c1COCC2 90204,C1(CC(N2C(CC(=O)N(C3CCCOCC3)C)CCC2)=O)CCN(C)CC1 90205,C12(C(=O)NCCCCC3(NC(CCCC)=O)CC3)CCC(CC)(C1)OC2 90206,C(C1=NOC2OCCC12)NC(=O)NCc1cc(Cl)ccn1 90207,C#CCC(C)(C(=O)N(CCCSC)C)NC(=O)C1=C(C)CCC1 90208,C1(NC(C(CC)N(C)C)=O)CCCCC12CCN(C(C1(C#N)CCCC1)=O)CC2 90209,C1(C(=O)NCCCCCCC2CC2)COCCN(C(=O)CNc2ccccn2)C1 90210,c1(C(=O)NCC2(F)CCC(NC(CS(C)(=O)=O)=O)C2)ccc(F)c(Cl)c1N 90211,N1(C(C)=O)CC2(CCCC(CNC(c3cnsc3)=O)O2)C1 90212,c1(Nc2ccc(OC)cc2)ccnc(CO)c1F.C12(CC1)C(=O)O2 90213,c1(N(C(c2ccc(COC)c(F)c2)=O)CC2(C)CNCCO2)ncc2ccsc2n1 90214,C1(CN(C(C2(C)CC(C(=O)OC)C2)=O)CC2CC2)C(C)(C)C1(C)C 90215,CCC(CC(=O)NCC1(CC(=O)NC2CN3CCCC2C3)CC1)C(C)(C)C 90216,CC1(C)COC(CC(=O)NC2CC3C(NC(=O)CC4CC5CC5C4)C3C2)C1 90217,c1(CC(=O)NCC2C3CN(C(C=C(C)C(F)F)=O)CC32)ccc([N+](=O)[O-])cc1F 90218,N1(C(c2c(C)cc(F)s2)=O)CC2CCC2(NC(c2nnn(C(C)C)c2C)=O)C1 90219,c1(CC)nocc1C(=O)NCc1cc(C(=O)NC2CC(C)(CO)C2)on1 90220,CCCS(=O)(=O)CC(=O)NCC1(F)CCN(C(C2Cc3nc(C)cn3C2)=O)C1 90221,c1(OC)cccc(CC(=O)NC(C2(O)CCN(C(=O)CP(C)(C)=O)C2)C)c1Cl 90222,C(=O)(CCC(C)(C)C#N)NC1CC(C)N(C(=O)CSCc2ccccc2)C1 90223,C#CCC(C(=O)NN1CCCC1C(=O)N(CC)Cc1cn[nH]c1)OC 90224,N1(Cc2c(N)cccn2)CCc2c(Cl)cccc21 90225,N1(C(CCN2C(C)CCCC2)=O)CCC2CCC12CNC(c1coc(Cl)n1)=O 90226,c1(CC)cccc(C(=O)NCC2=CCN(C(=O)C(N3CCC(C)C3)=O)CC2)c1F 90227,c1(C(=O)OC)cnc(N2CCC(C(C)C(N3CCC(O)C3)=O)CC2)nc1 90228,Cc1cc2c(cc1Cl)C(NC(=O)COCCn1cc(Cn3cccn3)nn1)CO2 90229,C1(CC(=O)NCC2CC(OC)C2)CCN(C(c2cn(CCO)nn2)=O)C1(C)C 90230,Cc1ccc(C(=O)NC2CCCC(N(C(=O)Cn3cc(CO)nn3)C)C2)n1C 90231,C1(NC(=O)CCN2CCOCC2)CN(C(C2(c3cc[nH]n3)CCC2)=O)CC1O 90232,C1(C(=O)NCCCN(C(c2cnc(S)[nH]2)=O)C2CC2)(CO)CC(F)(F)C1 90233,Cc1nc(C(C)C)ncc1C(=O)N(C(C)CCNC(=O)C(F)=CCCF)C 90234,c1(C(N(CC(CC)NC(=O)Cc2sccc2Cl)C)=O)cnc(OC)cn1 90235,c1(NC(C(c2ccc(Cl)s2)N(CC(=O)OCC)C(C)C)=O)ccc(OC)cc1 90236,C1(CC)(CC)CC(NC(=O)CC2CCC(=O)N2C)CN1C(=O)CCC1CCCC1 90237,S(=O)(=O)(c1cccc(=NCc2ncccc2N)[nH]1)NC(CC)C1CC1 90238,CC1C(NC(=O)CCn2ccccc2=O)CCCN1C(c1ccc(C#N)s1)=O 90239,N1(C(C(C)NC(CC)=O)=O)CCN(C(C2CC3(C2)CC3(F)F)=O)CC1C 90240,Fc1ccc2scc(CNC3CCCCC3c3cccc(Cl)c3)c2c1 90241,C1(NC(C2CCN(C)C2)=O)CC2CC(C1)N(C(C1SCCS1)=O)C2 90242,N1(C(c2cc(CC(C)C)on2)=O)CCCCC1CNC(=O)CCN1CCCC1 90243,c1(OC)cc(C(N2CC(CNC(C34COCC3C4)=O)(OC)C2)=O)ncn1 90244,CC#CCCC(=O)N1CCC(C(N2CC(C)C(F)C2)=O)CC1 90245,CC(C)CC(C)CNCC12CC(N(C)C)(C1)C2 90246,N1(c2n(CCC#C)c(C(CC)NC(=O)OC)nn2)CCC2(CCOCC2)C1 90247,N1(C(CCCC2C(C)C2)=O)CCC(CNC(=O)C(CCO)N(C)C)CO1 90248,c1(CC)ccc(F)c(C(N2CC(NC(c3cn(C)nc3COC)=O)C2)=O)c1 90249,c1(C(=O)NC2CC(NC(C3(C(N)=O)CC(F)(F)C3)=O)C2)cc2cnc(Cl)cc2s1 90250,C1(NC(=O)CSCc2ccc(Cl)cc2)CC2CC1N(C(c1cnco1)=O)C2 90251,c1(C(N2CC(O)(CCNC(c3nc(C#C)sc3)=O)C2)=O)nc(O)nc(O)c1N 90252,C1(C(=O)NCC2CCCCC2NC(=O)CCC2OCCO2)(OC)CCCCC1 90253,N1(C(=O)OC(C)(C)C)CCN(CN2CC(NC(C)(C)C)C(CO)C2)CC1 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90307,C1(C(=O)NC2C(CC(C)(C)C)C2)CCCN(C(C23CCC(CC2)C3)=O)C1 90308,N1(C(C)=O)CCC2CCC(NC(c3cccc(CCN4CCOCC4)c3)=O)C1C2 90309,C1(C(=O)NC(C(C)C)(C)CNC(c2cnc[nH]2)=O)CCC2(CCC2)CC1 90310,c1(CCC)ncoc1C(=O)NC(C(=O)N1CC(O)C1)C1(C)CC1 90311,Cc1cccnc1CC(=O)NC1(CC=CC(=O)NCCC2CCC3CC23)CCC1 90312,c1(CCC(N2CCCN(C(C(C)C)=O)CC2CO)=O)ccc2c(c1)COCC2 90313,CC1(C)C=C(C(=O)N2CC(CNC(C3(c4cc[nH]n4)CCC3)=O)CC2(C)C)C1 90314,c1(N2CCC(n3ncc(C)c3)C2)nc(NCc2cc(C)on2)nc2c1CCCC2 90315,C1(C)(c2cn(CCC=C)nn2)CCCN(c2ccc(C(=O)NC)nn2)C1 90316,C1(O)(CNC(=O)C(=O)NC2CC2)CCN(C(=O)C=CC(c2ccc(F)cc2)=O)C1 90317,Cc1cc(=O)ccn1CC(N1CC(F)CC1CNC(=O)COc1ccon1)=O 90318,Cc1cc(C(N2CC(CC(C)NC(=O)Cn3cc[n+](C)c3)C2)=O)[nH]c1C 90319,C(CC(C)(C)CNC(c1ccc(-n2cncn2)nc1)=O)NC(c1c(C)csc1)=O 90320,C1(C)(C2CC(CNC(=O)NC3N(C(C)(C)C)CC3)C2)NC(=O)NC1=O 90321,C(CC)(CCCC(=O)N(C)CC1CCCN(C)C1)NC(CCCCCOCC)=O 90322,c1(C(N)=O)cc(=NCC2CCCCC2NC(C2CCCO2)=O)[nH]c(Cl)n1 90323,N1(C(C=COCC)=O)CC2CC(O)C1C2NC(=O)COc1c(Cl)cccc1Cl 90324,C1(C(N2CC(C)(CCC(N3CC(C)C(C)C3)=O)C2)=O)Cc2ccccc2C1 90325,N1(C(CCNC(=O)NC)=O)CC(CNC(=O)CSC)CC1(C)C 90326,CCC(C)(O)C(=O)N1CC(CN2CCN(C(C3(S(N)(=O)=O)CC3)=O)CC2)C1 90327,N1(C(CCCCCC)=O)CC2(C1)CN(C(C1CCC1OC)=O)CC2C(=O)O 90328,CCC(C)CC(C)C(=O)NCCN(C)C(c1ccc(CN(C)C)nc1)=O 90329,N1(C(COCC=C)=O)CC(NC(C2CC2CF)=O)C(C)C1 90330,N1(C(C(C)OC2COC2)=O)CCC(C)(C)C(CNC(c2ccc(=O)n(C)n2)=O)C1 90331,O=[N+]([O-])c1cccc2[nH]nc(CNc3nc4c(s3)CC(C(F)(F)F)CC4)c12 90332,c1(N2CCOCC(NC(CCOCC#C)=O)C2)ncc([N+](=O)[O-])cc1Br 90333,N1(C(C2(C#N)CCCC2)=O)CC(C2CN(C(C34CC(C(F)F)(CO3)C4)=O)C2)C1 90334,c1(C(=O)NCCC2(NC(C(CCSC)O)=O)CC2)c(C)ncnc1C 90335,N1(CC(=O)N(CC(C)O)CCNC(C2CN(CC)C(=O)N2)=O)C(=O)CN(C)C1=O 90336,c1(-c2nc(C(CC)C)nn2C2CC(OC(C)(C)C)C2)ccn2c1CSCC2 90337,C1(C(=O)NCC(c2cn(C)cn2)O)(NC(C(C)c2cc[nH]n2)=O)CC1(C)C 90338,C1(C)(COC)CC(NC(c2c(Cl)cccc2Cl)=O)CN1C(=O)CCC(C)C 90339,C1(OC)CC(CNC(=O)Cc2cncs2)(NC(=O)CC23CC(C2)C3)C1 90340,n1(CC(=O)NC(CC(C)C)CNC(=O)CCCN(C)C)nnc2c1CCCC2 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90359,C1(C(N2C(CCCNC(C3CCC(CC)O3)=O)CCC2)=O)CCOC(C)(C)C1 90360,c1(C(=O)NCCC(=C)CNC(=O)C(F)=C(C)C2CC2)c[nH]c2cccnc2c1=O 90361,c1(NCCC(C)S(C)=O)cc(=NCc2nc(O)n[nH]2)[nH]cn1 90362,C(=O)(CCC1=CCCCC1)N1CCC(C)(NC(=O)CC2CCC(=O)N2)CC1 90363,N1(C(CCN(C(C)C)C(C2CC(=O)CS2)=O)=O)CCCC(C(=O)OC)C1.N(C)C 90364,C1(NC(CCCC#C)=O)CCN(C(=O)Cc2ccc(Br)nc2)C(C)C1 90365,CN1CC2CCC(C1)N2C(C1CC(F)CN1C(=O)CC1CSCCO1)=O 90366,CP(C)(=O)c1cccc(C(=O)N=S2(=O)CCCCCC2)c1 90367,C1(NC(CC2N(C(C)C)CCC2)=O)(CO)CCN(C(=O)CCC2CC2(Cl)Cl)CC1 90368,c1(C(=O)NCC(CC=C)NC(=O)CCC(C)CC)nccc2[nH]nc(C(C)C)c12 90369,N1(C(C(CC)(C)CO)=O)CC23CCCC2(C1)CN(C(c1c[nH]cc(C)c1=O)=O)C3 90370,c1(CC)cc(C(=O)NCC(O)CN(C)C(c2cnc(S)nc2)=O)nn1CCO 90371,C(=O)(C1=CCc2ccccc21)N1C(CNC(C2=CC(C)(C)C2)=O)C(C2CC2)CC1 90372,N1(C(C2CN(C(C)C)C2)=O)CCC(C)(C)C1C(=O)NCc1nc(C)co1 90373,C1(=CC(=O)NC2CC(F)(CNC(C3CCC(OC)C3)=O)C2)CCCCCC1(C)C 90374,N1(C(C(CCC)CC)=O)CC2(CCN(C(=O)C(c3cn(C)nc3C)C)C2)C1 90375,n12nc(C)c([N+](=O)[O-])c1N2CC.C1(C)CC(OC)C1.C(=O)(COC)OC 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90411,C1(C2CCCN(C(=O)Cc3nncn3C)C2)(NC(C(C)OC2COC2)=O)CC1 90412,C(C1=CCCN(C(c2ccsc2C)=O)C1)NC(Cc1cn(CC)nn1)=O 90413,c1(OC)ncccc1C(=O)NCCCCC1CCN(C(=O)Cn2ncnn2)CC1 90414,C1(NC(Cc2n(C)nnc2)=O)CC2CN(C(C3(O)CCCC3)=O)CC12 90415,c1(OC)ccc(CN2CCC(O)(C(=O)NCC3CCC3)C2)c(Br)c1 90416,Cc1cc(=NCCCOc2ccccc2F)[nH]c(=NCc2cc(Br)cnc2O)[nH]1 90417,c1(C(N(CC(CC)NC(C2(S(C)(=O)=O)CCC2)=O)C)=O)cnc(O)n(C)c1=O 90418,C1(C(=O)NC(C#C)CC(C)C)C2CCN(C(=O)C(OCC)OCC)CC12 90419,S(=O)(=O)(c1ccc(NCc2c[nH]c(=N)s2)c(Cl)c1)NC(C(CCC)C)C 90420,N1(C(C=C(C=C)C)=O)CCC(NC(=O)Cn2c(C)csc2=O)CC(O)C1 90421,N1(C(C2C(=C)C2)=O)CCCC(COC)(NC(=O)COCC(C)(C)C)C1 90422,CC1(C)CCCCC1NC(=O)CCOCCCNC(=O)Cc1nc(=N)[nH][nH]1 90423,c1(NC(=O)CC(C(F)F)NC(c2cn(C3CC3)nn2)=O)cccc2c1OCC2 90424,c1(C(=O)NC2C(CC)N(C(=O)CC3CC=CC3)CC2)cc2ccccc2c(=O)o1 90425,N1(CC)CC(NC(=O)CCN(C)C(C2(C)CCC2)=O)C(C)(C)C1 90426,C(N=c1cc(F)nc[nH]1)C1(CNC(C(c2ccc(OC)c(F)c2)C)=O)CC1 90427,c1(-c2cccc(NC(C)=O)c2)ccc2c(C(=O)NC3CCC(F)(F)C3)n[nH]c2c1 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90677,CC(CN(C)C)CN=c1nc(N2CCCC(C(F)F)C2)c2cccc(F)c2[nH]1 90678,N1(C(CCNC(=O)OC)=O)CC(C)(C)CC1CNC(=O)C(C)Cc1cnn(C)c1 90679,C(=O)(C(O)CC[S+](C)C)N1CC(C(C)NC(C(C2CCCCC2)OC)=O)C1 90680,c1(CNC(Cc2cccc(CCCCC)c2)=O)noc2c1COCC2 90681,C(=O)(C#CC1CCCO1)NC1C(NC(c2cc(-c3cn(C)nc3)[nH]n2)=O)COC1 90682,Cc1cc(C(=O)Nc2cccc(NC(=O)CCN(C)C)c2)c2ccc(F)cc2n1 90683,C1(C(=O)NC2(CC)CCCN(C(=O)Cc3ccco3)C2)CCc2nccn2CC1 90684,c1(C(=O)NC(CCCCNC(C(C)OCCOC)=O)C)c(OC)ccnc1O 90685,C1(CNC(N(C2CCC23CCC3)C)=O)CCc2cn(C)nc2C1 90686,c1(C(=O)NC(C2CN(C(C=C(CCC)C)=O)C2)C)ccc2nncn2c1 90687,C1(C)(CNC(c2nc(CC(C)C)sc2)=O)CN(C(=O)C(O)CC2CC2)CCO1 90688,CC(C)CC(O)C(C)C(=O)N1CCC(C)CC1CN 90689,C(=O)(C(C)CC(N)=O)N1C(CNC(c2cnc(C)n2C)=O)CCC1 90690,c1(C(=O)NC(C(=O)NC(C)CCCCO)CC2CC2)ccc(=O)n(C)c1 90691,C1(CN(C(COCCC)=O)CC)CCCCN1C(c1csc(C)c1OC)=O 90692,C1(CNC(Cc2cc(C)on2)=O)CC(NC(=O)CN2C(=O)CNC2=O)C12CCC2 90693,c1(C(=O)NCC(C)CNC(C2COC(=O)N2)=O)cc(Cl)c(F)cc1Cl 90694,c1(CCC(=O)NCCCN(C2CCN(CC)C2)CCC)ccccc1F 90695,CN=c1nc(N2CCN3C(CCS3(=O)=O)C2)[nH]c(=NC2CC2C(C)C)[nH]1 90696,C1(C(=O)NC(C#C)CC)CSCCN1C(c1cccc[n+]1[O-])=O 90697,C(C(C)(C)CNC(=O)CC1CCNC1=O)N(C(C1(C)CC1(C)C)=O)CC 90698,C#CC(C(C)C)NC(=O)CCN(C(=O)CCC1CC1)CC 90699,CC(C)CC(C(C)C)NC(=O)NCC(c1cccc(Cl)c1)(C)C 90700,C1(CN(C(c2c(OC)nsc2)=O)C)COCCN1C(=O)Cc1ccccc1F 90701,CC(C)CCCCCC(=O)N1CC(N(C)C(C2CC3CCC2C3)=O)C1 90702,Cc1cc(O)n2ncc(C(N3CC(C)(C)CC3CNC(=O)C(N)=O)=O)c2n1 90703,C=CCC(CNC(=O)Cn1cc(C2CCC2)nn1)NC(C1CCCN1C)=O 90704,CCCCCS(=O)(=O)CC(=O)N1CC2CC1CC2NC(c1nnn(C)c1CC)=O 90705,N1(C(C2C(NC(C3(C#N)CC(C)C3)=O)COC2)=O)CC2CCC2(CO)C1 90706,C1(C(=O)NC(c2ccc(Cl)s2)C)CCCN1C12CC(C1)C2 90707,CC(N=c1[nH]c(=NCC2CCOCC2)[nH]c2c1SCC2)c1nc(O)n[nH]1 90708,Cc1nc2ccccn2c1C(=O)NC(C1(O)CCOCC1)C 90709,C12(CCC1)C(=O)NC2.C(=O)(C(F)F)NC1(C(=O)OC)CC1 90710,CCCCCC(O)C(=O)NC(C(=O)NCC(C)(C)C(C)(C)C)c1cccs1 90711,c1(C(N(CC(CC)NC(=O)CC2(O)CCOC2)C)=O)c[nH]nc1OC 90712,C(=O)(C1=COCCO1)NC(C)CCCNC(C12CC(CCO1)C2)=O 90713,c1(C(C(=O)NC2CCOC2)N(CC(COC)C)C)cc(S(C)(=O)=O)co1 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90803,c1(C2C(NC(CC3(OC)CCC3)=O)C2)c(Cl)cccc1Cl.C12CCC1CNC2=O 90804,N1(C(Cn2c(C)cc(C)n2)=O)CCC(CC(=O)N(CC(C)O)C)C1(C)C 90805,C1(CNC(c2ccno2)=O)CCCC2(CN(C(=O)Cn3ncc(O)nc3=O)C2)O1 90806,N1(C(C2(C(=O)OCC)CC2)=O)CCCOC(CNC(=O)CC2(C)CCCCC2)C1 90807,Cc1cccc(C(=O)NC(CNC(c2cnc(OC(C)C)c(Cl)c2)=O)CO)c1N 90808,C1(NC(c2cc(CNC(=O)CCOCC3CC3)no2)=O)CCCC1C1CC1 90809,C(c1cccnc1)=CC(C)NC(=O)CCCc1ncco1 90810,O=S(=O)(c1ccc(N2CCN3CCCC3C2)c(F)c1)NC1CCc2ccccc21 90811,c1(C(N2CCC3(C(N4CC5(CCC5)C4)=O)CC3C2)=O)cc2cccc(Br)c2[nH]1 90812,CC1CC(N(C)C(c2ccc(CN3CCCC3CNC(N)=O)nc2)=O)CCN1C 90813,N1(C(c2csc(C3CC3)c2)C(=O)NC2(C)CC2)Cc2ccc(Br)cc2CC1C 90814,C1(OC)CC(CNC(c2scc(C)c2C)=O)N(C(C2COCCN2C)=O)C1 90815,C(C(C)(CC(C)C)Cc1ccccc1Br)NC(=O)C(F)=CCCF.CCC=O.C 90816,N1(C(C(C)(C2(C)CC2)OC)=O)CC(CO)C2(C1)CN(C(c1conc1C)=O)C2 90817,C(CCCNC(=O)CC1CCC1C)N(C(COCCOCC)=O)C 90818,C=CCCC(C)(C)CNCc1ccccc1C(C)(C)C#N 90819,C1(C(=O)NC2(CNC(C(c3ccc(CC)cc3)=O)=O)CC2)SC2C=CC1CC2 90820,c1(C(N2CC(NC(C3CC3C(N)=O)=O)CC(C)C2)=O)c(F)ccc2c1OCO2 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91012,c1(OC)ccnc(C(=O)N(CCCNC(c2c[nH]c(=N)o2)=O)C)c1C 91013,Cc1cc(OC2CN(C(=O)NCc3ccc(I)cc3C)C2)cc(C)c1 91014,c1(NC2(CC(=O)OC)CCOC2)ccc(C2(C(=O)O)CC2)cc1 91015,C1(NC(C2C(C)OCCC2)=O)CC2CCC1CN(C(c1cnccc1Cl)=O)C2 91016,C(C(C)(O)C1=CCC2CC1C2(C)C)NC(C(Cc1cn(C(CC)C)nn1)O)=O 91017,C(=O)(CCCCC(N)=O)N1C2CC(CNC(COCCCC(C)C)=O)C1CC2 91018,c1(OC)cc(F)ccc1C(=O)NCCC1CN(C(c2nc(C3CC3)oc2C)=O)C1 91019,N1(C(CC2C(C)CCN(C(=O)CCCn3cncn3)C2)=O)C2CCCC1COC2 91020,C1(C(=O)NCC2=CCN(C(C(C=C)O)=O)CC2)Cc2cc(C)ccc2S1 91021,Cc1ccc(C(C(N2CCN(CCO)CC2)=O)NC2CC2C2CC2)cc1 91022,N1(C(c2ccc(CNC(C(C=CC)O)=O)o2)=O)CCN(C)C(CO)C1 91023,CCC(C)CC(=O)C(=O)NCC(c1ccccc1)CNC(=O)CCc1ncc[nH]1 91024,C1(NC(CCc2cc(C)on2)=O)CC2CC(NC(=O)C=CCCC(C)C)CC2C1 91025,c1(C(=O)NCCN(C(CC2CC(=C)C2)=O)Cc2ccccc2)ccc(N)cc1C 91026,C1(C(=O)NCC(C(=O)NCCNC(=O)NC)N(C)C)COCC1(C)C 91027,c1(C(=O)NCC(N2C(C(=O)OC)CCC2)=O)ncccc1NCc1nnc(C)s1 91028,Cc1cc(OCC(=O)NCCC(C)CCNC(C2CC(C)(O)C2)=O)cc(C)c1 91029,C1(CC)CC(C(=O)Nc2cccc(C(F)(F)Br)n2)CCC1=O 91030,c1(C(N2C(CCNC(C3(CC=C)CCC3)=O)COCC2)=O)ncnc2c1CCC2 91031,c1(C(=O)NCCCCCCC(C)C)cc(F)ccc1S(C)(=O)=O 91032,CCCC(C(=O)NCC1CCCCN1C(=O)CC(C)(C)F)N(C)C 91033,c1(OC)ccccc1OCC(=O)NCCC1(NC(c2ccc(SC)s2)=O)CCC1 91034,C#CCCCC(C)C(=O)NC(C1(O)CN(C(c2ccsc2C)=O)C1)C 91035,C1(COC)(NC(=O)CCn2ccc(C)n2)CCN(C(C2CC(C#N)C2)=O)C1 91036,C1(C(=O)NCCNC(C2CCN(C3CC3)C2=O)=O)CCCc2ccccc2C1 91037,N#Cc1cc(F)c(C(N2CC(F)(F)CC2C(=O)Nc2cc(Br)ccn2)=O)c(Cl)c1 91038,CCC(F)C(=O)NC1CCC1NC(=O)Cn1cc(C(=O)N(C)C)nn1 91039,N1(C(C=CC)=O)CCC2(CC1)CC(NC(=O)CC1CC3(C1)CC31CCC1)CCO2 91040,C1(CC(N2C(C)(C)CCC(C(=O)OCC)C2)=O)CCc2ncc(Br)n2C1 91041,C1(C(N2CC3CC2CN3C(=O)OC(C)(C)C)C(=O)NC)CC2OC(C)(C)OC2C1 91042,c1(C(=O)NCC(Cl)Cl)cc(CNC(c2cnn[nH]2)=O)cs1 91043,C1(C(=O)NCC2N(C(c3nc(CC)oc3)=O)C3C(C2)C3)CCC(C)(F)CC1 91044,C1(CC(=O)NC2CN(C(C3CC34CCOC4)=O)C2)CCc2ccccc2C1 91045,N1(C(Cc2cccc(C)c2)=O)CC(CO)C2(C1)CN(c1nnc(C(F)F)s1)C2 91046,C1(OCCOCC(=O)Nc2ccccc2)CN(C(c2sccc2F)=O)C2CC12 91047,C1(C)(COC)CCCN(C(=O)C(CCCOC)NC(=O)C(CCF)OC)C1 91048,N1(Cc2c(C)cc(Br)cc2)CCc2nn(C)c(C(=O)NCc3sccc3Cl)c2C1 91049,N1(C(CC2CCN(C)C2)=O)CC2CN(C(=O)CCC3CCC(=O)NC3)CC2C1 91050,C1CC(O)C(=O)N1.c1(C(c2nnnn2C(C)C)NCCOC)cnnn1C 91051,C1(C(=O)NC2CC(CNC(c3csc(C4CCCO4)n3)=O)C2)(COC)CCCO1 91052,N1(C(C2C(C)=CCS2)=O)CCCC(C)(C(=O)NC2CCCC2F)C1 91053,c1(C(=O)NC(C)CC2CN(C(=O)Cc3ncc(Cl)s3)C2)ccc(OC(F)(F)F)cc1 91054,Cn1cc(C(=O)NCC23CCC(C)(CC2)CC3)c(O)nc1=O 91055,N1(C(C(C2CCOCC2)C)=O)CCN(C(C2C(C)C2C)=O)CC12CCC2 91056,N1(C(=O)C(F)CC2CCOC2)C2CCCC1CN(C(C13CCC(CC1F)C3)=O)C2 91057,C1(C(=O)NC2(C)CN(C(C(C)C(=O)OC(C)(C)C)=O)C2)CCS(=O)(=O)N1C 91058,N1(C(c2ccc(COC)cc2Cl)C(=O)NCCOCC)CCCC(N=[N+]=[N-])C1 91059,CCC(C)C(C)C(=O)N1CCC(C)C(c2ccccc2)C1 91060,N1(C(c2c(C)noc2)=O)CCCC(NC(c2nnc(C(F)(F)F)s2)=O)C1C 91061,c1(NCCCC(C)NC(CN(CC)Cc2ccccc2)=O)cccnc1F 91062,C1(NC(=O)Cn2ccnn2)CCC(CCNC(C2(CCF)CCC2)=O)C1 91063,c1(C(=O)NC2CCC(C(=O)NCC3CCCC34CC4)CC2)cc(F)cc(F)c1 91064,C(=O)(CCN=C(NCC1(CCO)CCCCC1)NC1CC(O)C12CCC2)NC 91065,C(c1cccnc1)=C(C)C(=O)NC1CC1CNC(c1ccc(F)cc1)=O 91066,C1(C(=O)NC(CC=C)CNC(c2sc(F)cc2C)=O)CCC2CC2CC1 91067,CC1=C(C(=O)N2CCC2CNC(c2cc(Cl)cnc2O)=O)CCC1 91068,CC1(C)C(O)CCN1C(C1CCOCC1)C(=O)NCCC#N 91069,C#Cc1cccc(NNC(=O)Nc2cn3nc(Cl)cc(I)c3n2)c1 91070,N1(C(C2N(CC)CCCC2)=O)CCN(C(c2c(N)cc(Cl)cc2F)=O)CC(O)C1 91071,C(=O)(CCCS(C)(=O)=O)N1CCC(NC(c2c(C)n[nH]c2)=O)CC1C1CC1 91072,C1(NC(=O)Cc2cn[nH]c2)CN(C(c2ns[nH]c2=O)=O)CC(F)(F)C1 91073,N1(C(C(C)NC(CC)=O)=O)CCCC(CNC(=O)CSc2nncs2)C1 91074,N1(C(c2c(C(C)C)nn(C)c2)=O)CC(NC(C2CC2C(F)F)=O)CC2(CC2)C1 91075,c1(OC)cnc2[nH]c(C(=O)NCC(C)N(C)C(c3ccnn3C3CC3)=O)cc2c1 91076,C1(NC(C2CC=C(C)CC2)=O)CN(c2snc(C)c2C#N)C2(CCOCC2)C1 91077,c1(C(N(C2CN(c3cc(C)nn3C)C2)CCC)=O)cncc(-n2cccn2)n1 91078,C1(C)(CNC(C(CC)n2ccnc2)=O)CCN(C(C2CC3C=CC2C3)=O)CC1 91079,c1(C(N2CC(CCOC)N(C(=O)C3=C(C)CCC3)CC2)=O)c(C)cc(C)oc1=O 91080,c1(C(C)C)ncc(NC(=O)C(C2CCCC2)NC(=O)CN=[N+]=[N-])cn1 91081,C1(NC(CC2(NC(CCc3ncn(C)c3)=O)CC2)=O)CCS(=O)(=O)C1 91082,c1(C(C)=O)cccc(OCC(=O)NCC2(NC(C3CCCN3C)=O)CC2)c1 91083,C1(OC)CC(CCNC(=O)Cc2ccc(O)cc2)N(C(c2snc(O)c2Cl)=O)C1 91084,c1(C(CSCCC)(C)NCC2CC(SCC)C2)nnnn1C(C)C 91085,C1(NC(C=CCNC(=O)CCOCC2CC2)=O)CC2(CCC2)C1O 91086,c1(CCC(N2CC(CN(C(CCCC)=O)C)OCC2)=O)nc2cc(Cl)ccc2s1 91087,Cc1ncc(C(N2CC3C(NC(C4COCC4(C)C)=O)C3C2)=O)n1C 91088,c1(OC)cc(OC)cc(N2CC(NC(N3CC4CC(C3)O4)=O)CC2=O)c1 91089,NS(=O)(=O)c1ccc(CC(=O)NC2(CO)CCCN(C(=O)C3CC3)C2)cc1 91090,N1(C(C2C(=C)C2)=O)CCC(CC)C1CNC(=O)COc1ccc(OC)cc1 91091,C1(O)(CN(C)C)CN(C(c2coc(CNC(c3cc(Cl)c[nH]3)=O)c2)=O)C1 91092,c1(CCNC(c2ncc(CCNC(C3C(C)C3)=O)s2)=O)c(F)cccc1Cl 91093,c1(SC)nc2c[nH]c(=NCc3cnc4n3CCS4)nc2s1 91094,N1(C(c2c(C)nc(C)[nH]2)=O)CC2CC(NC(C3CCCCS3)=O)CC2C1 91095,c1(C(C)(C)C)cc(CN2CC(C(=O)NCC(F)CO)CC(F)C2)ccc1O 91096,C1(NC(C2CC(Cl)(Cl)C2)=O)CCN(C(=O)CN2CC3CC3C2)CC1O 91097,c1(C(N2C(CNC(C(CC)c3ccccc3)=O)CC2)=O)noc(C)c1[N+](=O)[O-] 91098,C12(C(=O)NC(C)Cc3cn[nH]c3)CC(C)(CN1C(=O)CC1(O)CCN(C)CC1)C2 91099,Cc1ccnc(C(C)NC(=O)CC2(CNC(=O)CCn3cc(C)cn3)CC2)n1 91100,c1(C(N2CCN(C(C(Cc3ccccc3)OC)=O)CC2)=O)ccc(N)c(C)c1Cl 91101,c1(C(=O)NC2C(NC(C3(O)C(C)(C)C3)=O)CCC2)cccn2ncc(Br)c12 91102,C1(C(C)C)CCC(C(=O)NCC#CC2CC2)N1C(=O)CC1OCCO1 91103,N1(C(C2C(C(C)C)CCO2)=O)CCCC(C)(C)C1CNC(=O)C1=NOCC1 91104,C1(CNC(C(C)OC2CCCC2)=O)CCN(C(=O)CCc2ccc(F)nc2)CC1 91105,C1(C(=O)NCCC2(C)CCN(C(C3(C)CCC(=O)NC3)=O)C2)SC2C=CC1CC2 91106,c1(C(C)C)conc1C(=O)NCCC(C)NC(C1CCOC1C1CC1)=O 91107,c1(NC(C(c2cccc(Cl)c2)NC)=O)nc2cccc(Br)c2[nH]1 91108,C(=O)(CCCC(C)CC)NC(CC)C(=O)NCC1(C)CCC(C)CC1 91109,Cc1[nH]c2ccnn2c(=O)c1CC(=O)NC1CN(C(=O)C2=CCOC2)CC12CC2 91110,C(c1ccc2occc2c1)=CCC(N1C(C)CN(C(=O)OC(C)(C)C)C(C)C1)=O 91111,c1(OC)ccc(COCCOC(=O)COc2ccc(O)cc2I)c(Cl)c1 91112,c1(OC)cncc(C=CC(N2CCC(NC(=O)Cc3ccon3)C2(C)C)=O)c1 91113,c1(CC)ccc(C(=O)NCC2CCC2NC(=O)C=CSc2ccccc2)c(O)c1 91114,c1(C(=O)NCCc2c[nH]c(=NCc3cc(Cl)ccn3)s2)[nH]nc2ncccc12 91115,N1(C(C(C)N(C)C)=O)CC2(CCNC(c3cn4c(n3)SCC4)=O)CCC1C2 91116,CC(C)(CCC#N)C(=O)NCCC1CCC(NC(=O)Cc2ccoc2)C1 91117,Cc1coc(C)c1C(N1CC(CNC(=O)CCNC(=O)CO)C2CC12)=O 91118,c1(CN(C(C(C)n2ccnc2)=O)C)cc(Cl)ccc1O 91119,N#Cc1ccc(CCC(N2CCC(Nc3ccccc3F)C2)=O)cc1 91120,Cc1cc(C)c(C(N2CCOC(C)(CNC(c3cnsn3)=O)C2)=O)c(C)n1 91121,N1(C(c2cncc(Cl)c2Cl)=O)CCC2(CC(NC(C3(O)CC3)=O)CO2)C1 91122,c1(SCCCC(=O)N(C2CCCCC2=O)C)ccc(Br)cc1 91123,C1(NC(C2C(C)C2C)=O)CCN(C(c2cn(C)[nH]c2=N)=O)CC12CCC2 91124,N1(C(CN(CCOC)C)=O)CCCCC(C2CN(C(C3CCCN(C)C3)=O)C2)C1 91125,N1(C(C=CCOC)=O)CCC2(C1)CN(C(=O)CC(C)CN(C)C)C2 91126,CC1(C)CN(C(=O)CCNC(=O)CO)CCC1C(N1CC2CCCCC2C1)=O 91127,Cc1cc(C(=O)NCCCNC(c2cc(C(F)F)ccc2F)=O)cc(N)c1O 91128,N#Cc1ccc(C2(C(=O)NC3(C(=O)NCC(C4CC4)N(C)C)CCOC3)CC2)cc1 91129,c1(CC)nc(C(=O)NCC2CC(O)CN2C(=O)C(O)CC)c(N)s1 91130,CC(C)CC(CNC(c1ccncc1)=O)NC(c1ncoc1C1CCCO1)=O 91131,N1(C(Cn2c(C)ccn2)=O)CCCC12CCC(NC(=O)C=Cc1cnc[nH]1)CC2 91132,CC1CCC(C(N2C3CCC2C(CNC(=O)CC2COC(C)(C)C2)C3)=O)CC1C 91133,C1(NC(=O)Cc2cnoc2)CCCN(C(=O)C(O)Cc2cnc[nH]2)C1 91134,C(=O)(C(C)(C)C(F)F)N.N1(C(C)(C)C2CC2)CCCCC(C(NOC(C)CO)=O)C1 91135,c1(CC)occ(C)c1C(=O)NCC1CC1NC(=O)C=CCc1ccsc1 91136,c1(N(C)C)cc(C(N2C3CCC2(CNC(c2ccns2)=O)CC3)=O)ccc1[N+](=O)[O-] 91137,N1(C(C)=O)CCc2cc(C(=O)N(C3CN(C(C4(C)CC(C)=NO4)=O)C3)C)ccc21 91138,c1(C(N2C(CNC(=O)CCCn3ccnn3)CC(OC)C2)=O)cncc(O)c1Cl 91139,C1(NC(n2ncccc2=O)=O)CN(C(=O)CSC(F)F)C2(CCCOC2)C1 91140,c1(C(N2C(C)CCC2)=O)cn2c(n1)CN(C(c1c(Cl)cnn1C)=O)CC2 91141,c1(C(N(CCCNC(C2COCC(C)O2)=O)CCO)=O)cc2cccn2c(O)n1 91142,c1(CNC(N2CCC(NS(=O)(=O)C3CC3)CC2)=O)ccc2nonc2c1 91143,c1(C(N2CC(C)C(CNC(=O)CN(C)CCO)CC2)=O)c[nH]c2c(F)cccc12 91144,C1(NC(c2c(C)sc(Cl)n2)=O)CCN(C(=O)COCC2CCCOC2)CC1F 91145,c1(OC)cc(C)cc(C(=O)N(C2CC(NC(=O)CN(C)C3CC3)C2)C)c1N 91146,CCCCCCC(C)CC(=O)NC1CCN(CCOc2cccc(F)c2)CC1 91147,C1(CNCc2cc(OC)c(OC3CC3)cc2)(COC)CCCNS1(=O)=O 91148,C(=O)(CS(=O)(=O)CCO)N(CCn1cc(C2(N(C)C)CCCCC2C)nn1)CC 91149,CN1C(=O)CN(CC(=O)NCC2(F)CN(C(C3(c4cccs4)CC3)=O)C2)C1=O 91150,c1(CC(N2CCC(N(C(=O)CC3CSCCO3)CC)C2)=O)ccc(F)cc1 91151,CCCCC(C(=O)NC1CCCC1NC(c1cccn1C1CC1)=O)C(C)C 91152,c1(OC)ccc(CC(O)C(=O)NC(CNC(c2cnc(O)o2)=O)C(C)(C)C)cc1 91153,C1(c2[nH]nc(Sc3ccc[nH]3)n2)CC(=O)CC12CCC2.C12CN(C(=O)C(F)(F)F)CCN1C2=O 91154,c1(-c2cc(C)no2)ccc(S(=O)(=O)N2CCCN(C(=O)CNS(C)(=O)=O)CC2)s1 91155,C1(C(=O)OC)CN(C(=O)C(N2CCOC(CSC)C2)=O)CCN1C 91156,c1(C(N(C)CC2CCCN(C(C3CC4(CC(=O)C4)C3)=O)C2)=O)ccc(Cl)c(Cl)c1 91157,C1(NC(C(C)O)=O)CCCC(NC(c2ccc(N3CCCCC3)cc2)=O)CC1 91158,CC(C)CC(CNC(C1(c2ccccc2F)CC1)=O)NC(C1CCS1(=O)=O)=O 91159,N1(C(CC2CC=C(C)CC2)=O)CCC(C(=O)N(c2cc(F)ccc2C)C)C(O)C1 91160,CC(C(=O)N1CCC(CN(C)C(c2cc(C(C)(C)C)nn2C)=O)C1)C(F)(F)F 91161,C#Cc1cncc(NC(C2(CNC(c3cc(C4CC4)no3)=O)CC=CC2)=O)c1 91162,N1(C(C(CC)NC(N)=O)=O)CC2CCC1C(CNC(C1(F)CC=CC1)=O)C2 91163,O(C1CCc2c1cccc2[N+](=O)[O-])C(C1=NOC(C)C1)=O 91164,c1(C(C(=O)NC2CCN(CCSC(C)C)CC2)OCC)ccc(F)cc1C 91165,Cc1cc(C)n(CC(=O)OCC2CCCCC2)c(=O)n1.C1CCNC(=O)N1 91166,c1(OC)cccn2ncc(C(=O)NCC3(OC)CCN(C(c4ccsc4)=O)C3)c12 91167,N1(C(C2C(C)(C)OCC2)=O)CCC(F)CC1C(N1CC(CF)C1)=O 91168,C1(CC=C)(C(=O)N(C)Cc2nc(C)ns2)CCCN1C(C1CC1C(C)(C)C)=O 91169,Cc1ccc(C#N)cc1C(=O)N(C1CC(NC(=O)C(c2ccccc2)F)C1)C 91170,C1(C(=O)NCCCNC(c2ccn(C3CCC3)n2)=O)CC2(CCCO2)C1 91171,c1(C(=O)NC(c2c(F)cccc2Cl)C(=O)OC)cc(Cl)ccc1Cl 91172,Cc1cccc(C)c1C(=O)N(CCC(C)NC(=O)C(C)SC(C)C)C 91173,C1(NC(c2c(SC)scc2)=O)CCN(C(c2[nH]nnc2C)=O)C(C)C1 91174,C1(NC(C2C(=C)CC2)=O)CN(C(c2ccccc2N2CCOCC2)=O)CC1(C)C 91175,c1(C(=O)NCC2N(C(CSCC)=O)C3C(C2)CCC3)ccc(S(=O)C(C)C)cc1 91176,Cc1ccncc1C(N1CC(N(C)C)C(CNC(C2C=CCCC2)=O)C1)=O 91177,O=C(C1=C(c2ccccc2)CCC1)NC1(C2CN(C(C3CCOC3=O)=O)C2)CC1 91178,N1(C(c2cc(Br)cs2)C(=O)NC(CC)C)CC2CCC(C)(C1)C2(C)C 91179,Cc1cccc(C(=O)NCCCNC(c2cnn(CCN(C)C)c2)=O)n1 91180,C1(NC(=O)Cc2cc[nH]n2)CCCC(NC(=O)Cc2nc(C3CC3)cs2)C1 91181,C1(OC)CN(C(=O)C(C)SC)CC1NC(=O)OC(C)(C)C 91182,C1(C(=O)O)(CC)CCN(C(=O)Cc2csc(C3CC3)n2)CC1 91183,c1(-c2occ(C)c2CN(CC(C(C)(C)C)C2CC2)C=O)c(F)c(F)cc(F)c1F 91184,C1(N(C(Cn2cc(C(C)=O)nn2)=O)C)CC12CCN(C(C1CCCC1O)=O)CC2 91185,O=C(CC1CC2(C1)CN(C(=O)CC1CCOC1=O)C2)Nn1cnnc1 91186,C1(NC(C2COCCO2)=O)CCN(C(c2ncc(Cl)cc2Cl)=O)CC1O 91187,C1(CC)CCC(O)(C(=O)NCCNC(C2CN(C3(CC(=O)NC)CC3)C2)=O)C1 91188,c1(C(C)(C)C)ccc(NNC(=O)NCc2ccc(NC3CCOCC3)cc2)cc1 91189,C(CC1CCC1)(C(=O)N(C(C)C(=O)NCC(C)(C)O)C)OC 91190,c1(C(C)C(=O)N2CCCC2)ccc(S(=O)(=O)NC2C3CCC(C3)C2(C)C)cc1 91191,N1(C(CONC(=O)C2C(C(=O)OC)C2)=O)CCC(C2(C)CC2)C1 91192,N1(C(c2nnc(C(C)C)s2)=O)CCC(NC(=O)CCC2CC2(C)C)C(CO)CC1 91193,C1(C(C)NC(=O)C(C)(O)c2ccccn2)CCN(C(c2cccnc2)=O)CC1 91194,Cc1c(C(=O)NCC2CN(C(C3CCCO3)=O)C2)cccc1N 91195,Cc1[nH]c(=N)ccc1C=CC(N1CC(O)(CCNC(C2(C)CCCC2O)=O)C1)=O 91196,c1(C(=O)Nc2cnc(Br)c(F)c2)cnc2c(C3=CCCCO3)cccc2c1 91197,C(=O)(CCC(=O)OC1CC(C)OC1=O)c1ccc(C)s1.C123CC(C1)(C2)CNC3=O 91198,Cc1cc(C(=O)NCCSCC(N2CCC(c3ncco3)C2)=O)nc(O)c1 91199,C(c1cncn1C)=CC(=O)NCC1(NC(c2ccc(COC)o2)=O)CC1 91200,N1(C(CNC(CCCN(C(C)C)C)=O)=O)CCCCC1C(C)O 91201,Cn1cccc1CC(=O)NCC1(C(C)(C)O)CN(C(c2csnn2)=O)C1 91202,Cc1ccc(C(N2CCC(C(C)(C)NC(C3CCC(C(N)=O)CC3)=O)C2)=O)n1C 91203,c1(C(N(CC(CC)NC(=O)COC(c2ccn(C)c2)C)C)=O)ccc(OC)nc1 91204,C12(C(=O)NC3C(OC)CCC3)CC(CN(C(c3ccc(C4CC4)o3)=O)C1)C2 91205,c1(C(=O)NC2CC(C)N(C(=O)CCc3cnoc3)CC2)cccc2ccncc12 91206,C1(C2CCCN(c3nc(C)cc(C#N)n3)C2)(NC(C(CC(C)C)OC)=O)CC1 91207,N1(CC(=O)NC2CCC(N(C)C(c3cnn(CC(F)F)n3)=O)C2)C(=O)CNC1=O 91208,N1(Cc2c(C)ncs2)CCC(c2ccccc2)(C(=O)NCc2cnn(C)c2F)C1 91209,N1(C(C)C)CC(NC(=O)C=CC2CCCN2C(c2cn(C3CC3)cn2)=O)C(C)C1 91210,C#Cc1ccc(C(=O)NC(C(=O)N(C(C)C(=O)OC)C)C(C)(C)C)cc1 91211,C1(NC(C=CC(C)C)=O)CC2CC(C1)N(C(=O)Cc1cc(F)ccc1Cl)C2 91212,Cc1sc(=O)n(CC(=O)NCC(C2CC2)NC(=O)CC2CCCS(=O)(=O)C2)c1C 91213,Cn1c(CC(=O)NCC2(F)CN(C(=O)CNC(=O)NC3CC3)C2)nnc1S 91214,c1(OCC(=O)NCC2CC(OC)CN2C(=O)C2CC2)c(F)c(F)cc(F)c1F 91215,C1(NC(c2nn(CC)c(O)c2)=O)CC(NC(=O)Cn2nc(C)nc2C)C12CCC2 91216,C(=O)(CCC(=O)c1ccccc1)N1CCC(CCNC(c2ccc(Cl)nc2)=O)C1 91217,N1(C(C(Cn2cccn2)NC(c2ccccc2F)=O)=O)CCCC2(CCCC2)C1 91218,c1(OCOC)cc(-c2nc(C(=O)Nc3cncc(C#N)n3)ccc2F)ccc1C 91219,Cc1cc(C(=O)NC(c2ccsc2)CO)nc(Br)c1 91220,N1(C(=O)NCCOC(C(=C)C)=O)CCC2(CCN(Cc3cc(Br)ccc3C)C2)C1 91221,N1(C(c2ccnc(C)c2C)=O)CCC(C(=O)NCc2nnnn2C)=C(F)C1 91222,Cc1cn2c(C(N3CCC(CNC(c4sc(F)cc4C)=O)C(C)C3)=O)cnc2s1 91223,CC1CN(C(=O)CCc2nccn2C)CC1NC(c1cnncc1C(F)(F)F)=O 91224,c1(C(N(C2CCCCN(C(C(CCSC)O)=O)C2)C)=O)cc2n(c(=O)c1)CCS2 91225,C(N=c1cc(Cl)nc(C)[nH]1)C1N(C(C=CC=CC)=O)CCCC1 91226,N1(C(CCCC=C)=O)CC2CC(C1)C(CO)C2NC(=O)C(CCC)=CCC 91227,C1(CC(=O)NCC2CC(NC(CC=CC)=O)C2)CCn2cncc2C1 91228,C1(C(=O)NCc2c(C(=O)NC(COC)C3(C)CC3)n[nH]c2)CC2(CCC2=O)C1 91229,C(=O)(CC(C)(C)C(=O)N1CC(OC)C(NC(=O)C(C)CC)C1)OCC 91230,Cc1nc(NC(=O)NC(C)CF)sc1Cc1ccnn1Cc1ccc(Br)cc1 91231,C1(=CC(=O)OCc2nnc(CC(C)C)o2)CCN(C)CC1 91232,C1(NC(COCc2nc(C)on2)=O)CN(C(=O)CCn2cnc(=N)[nH]2)CC1O 91233,CCC(C#N)(CC)C(=O)NCC1CN(C(=O)C(C2CCOCC2)O)C(C)(C)C1 91234,C1(C(=O)N(C2(C(=O)NC)CC2)C)(NC(COCC=C)=O)CC(O)C1 91235,CP(C)(=O)CCC(=O)NN(C1CC(=O)N(CCO)C1)C(C1C(CC)C1)=O 91236,C1(NC(Cc2n(C)ccc2)=O)CCC(C)(CNC(=O)CC2CC(=O)NC2=O)CC1 91237,N1(C(C2CC(NC(C3CC(C(C)C)C3)=O)C(O)C2)=O)CC2CC2C2CC12 91238,N1(C(c2c(C(C)C)noc2)=O)CC(C(=O)NCC2(C)CCCC2O)C(F)(F)C1 91239,c1(C(N2CCC(CN(C(=O)C=CC3CC3)C)C2)=O)ccc(Br)cn1 91240,N1(C(c2c(C)oc(C(C)C)n2)=O)CC(CNC(=O)C(=O)NCCC#N)CCC1C 91241,c1(N(C)CC2CC2(F)F)ncccc1S(=O)(=O)NC12CCC(C(F)(F)F)(CC1)CC2 91242,C(=O)(C(F)CC(C)(C)NC(=O)CCC1CC1(C)C)NCCSCC#C 91243,N1(C(C(CC)N(C)C)=O)CCC(O)(CCNC(c2[nH]c(C)nc2C)=O)C1 91244,C(CC(=O)N1CCC(N(C)C(c2ccccc2O)=O)C1)(C(F)(F)F)OC 91245,c1(OC)ccc2c(C(N3CC(NC(=O)CC4CCOC4C)C3)=O)csc2c1 91246,CCC(C)C(C(=O)N(O)Cc1cn(-c2nccs2)nn1)Oc1ccc(F)cc1F 91247,C(=O)(CC(O)C(Cl)(Cl)Cl)NC(c1ccc(OC)cc1)CCCC 91248,c1(NC(C2(C)CCN(C(c3ccc(F)nc3F)=O)C2)=O)c[nH]c2ccc(Cl)cc12 91249,S(=O)(=O)(CC(=O)NCCCOCCNC(C1OCCCO1)=O)N(C)C 91250,CC1CC(NC(C2CCC(N(C)C)C2)=O)CN1C(c1ccc(OC2CC2)cc1)=O 91251,C1(C(N2CC(=C)C2)=O)CC(C)N1C(=O)CC1(COC)CC1 91252,CCC(O)(CC(=O)NCC1CC1NC(c1cncc(Cl)c1Cl)=O)c1ccccc1 91253,C#CC1(C(=O)NC2CCC(CO)C2)CCN(C(C2CC3(CCC3O)C2)=O)C1 91254,c1(OCC)ccc(C(=O)NCC(CC)NC(c2nc(Cl)c(Cl)s2)=O)cc1 91255,c1(CNC(C(C2CCC2)N(C)CCO)=O)cccc(C(N2CCNC(=O)C2)=O)n1 91256,Cc1sc(S(N)(=O)=O)cc1C(=O)NC1CCC1NC(C12COC(CCO1)C2)=O 91257,C1(C)(NC(c2cc(SC)oc2)=O)CCN(C(=O)C(n2cnc(C#N)n2)C)CC1 91258,N1(C(c2ccc(CC)[nH]2)=O)CCC2(CC1)CN(C(=O)CC1CCC3CC13)CCO2 91259,c1(OC)ccc2c(c1)CC(OC)CN2C(=O)Nc1c(F)c(C)nn1C 91260,N1(C(c2c(C)ncnc2O)=O)CC(C2CN(C(C3CCOC3C)=O)C2)C1 91261,C(c1ccccc1)=C(CC)C(=O)NC1CCC(CCNC(C2(C)CC2(F)F)=O)C1 91262,Cn1cnc(C=CC(=O)NC2COCC2NC(=O)COC2CCOC2)c1 91263,C(=O)(C1Cc2ccccc21)NCC1N(C(c2cn(C3CC3)cn2)=O)CCC(C)C1 91264,CCCCCC(C)(C)CNC(c1nnnn1C1COC1)(C1CCOC1)C 91265,N1(C(C(CC)OCC)=O)CC(F)(F)CC1CNC(c1ccn(C2CC2)c1C)=O 91266,N1(C(CSCCOC)=O)CCC(C)(CNC(=O)CN(c2ccccc2)C)C1 91267,c1(C(=O)NCC(CNC(C(C2CCCCCC2)C)=O)(C)C)cn(C)c(O)n1 91268,C#Cc1ccc(CC(=O)NC(CNC(c2cncc(C)n2)=O)CCCC)cc1 91269,N1(C(c2cc(CC)no2)=O)CCC(NC(=O)CC(F)F)C(CC)C1 91270,C(=O)(C(CCO)N(C)C)NC1CCC(NC(CC(=O)NCC)=O)C1 91271,C1(CC)CN(C(=O)CSCC(=O)N(C)C)C(C)CO1 91272,c1(C(=O)NC2CCN(C(CC(CC)C)=O)CC2O)nc2ccccc2cc1Br 91273,C(=O)(CS(=O)(=O)C1CCCC1)N1CC(NC(C(C(CC)C)O)=O)C(OC)C1 91274,C(CC(C)C)(C(F)(F)F)NC(C(N1CCC(CNC(CCCC)=O)CC1)=O)=O 91275,C(=O)(CCCCCF)NCCNC(C1(SC)CCC1)=O 91276,c1(OC(C)C)cnc(C(N2CC(CC(C)NC(C3C=CCCC3)=O)C2)=O)cn1 91277,N1(C(c2nc(CC)oc2)=O)CCN(C(C2(C)C=CCC2)=O)C2(CCC2)C1 91278,C1(NC(c2ccncc2O)=O)COC2(CCN(C(c3cc[nH]c3)=O)C2)C1 91279,C1(CNC(C(C=C)O)=O)CCCCN(C(c2cc(=O)n(-c3ccccc3)[nH]2)=O)C1 91280,c1(CC)cc(C(=O)NCC(C)NC(=O)C=Cc2c(C)coc2C)c2c(c1)CCO2 91281,N1(C(CNC(=O)OCC)=O)CCN(C(c2cccc(Cl)c2OC)=O)C(CCO)C1 91282,c1(CCC(=O)NC2CC3(C(NC(C(F)OC)=O)C3)C2)c(C)nc(O)nc1O 91283,c12cnc(nc1)CC1CCCN(C1)C2=O.n1(Cn2cccc2)cc(CCCO)nn1 91284,N1(OCCOCCOCCOCC=C)CC=CC1C.N1(C=O)CCC(C2CC2)C1 91285,C1(NC(C(COC)C)=O)CCN(C(=O)Cc2ccc(OC)c(OC)c2)CC1O 91286,N1(C(c2c(C(=O)OC)c(C)[nH]n2)=O)CCCC(C)(NC(C2CC2(C)C)=O)C1 91287,CC(C)C1=CCC(C(N2C3CCC2CC(CCNC(=O)CSC2CC2)C3)=O)CC1 91288,N1(C(c2c(CC)occ2)=O)CCC2(CCC2NC(C2COCC(C)(C)O2)=O)CC1 91289,Cc1nccn1C(C)C(=O)NC1CCCC1NC(=O)CSCC(N)=O 91290,CN1CCn2ncc(C(=O)NCC3CN(C(=O)C(C)(C)C(F)F)CC(C)(C)C3)c21 91291,c1(C(N2C(CNC(C(CC#C)C)=O)COCC2)=O)ccc(OCCCC)cc1Cl 91292,c1(C(N(C(C(=O)NC(CC=C)C(=O)OC)C)C2CC2)=O)c(C)[nH]c(C)c1C 91293,S(=O)(=O)(c1cncc(Br)c1)N1C(NC(c2cc(Br)nc(Br)c2)=O)COCC1 91294,C1(NC(c2ccc(C(C)=O)cc2)=O)(CO)CCCN(C(C2CC(O)C2)=O)C1 91295,Cn1nc(C(=O)NC2CCCN(C(C3(Sc4ccncc4)CC3)=O)C2)cc1Cl 91296,c1(C(N2CC(OCCNC(C3C(OCC)C3C)=O)C2)=O)cnnc(C)c1 91297,C1(C(=O)NCc2ncccn2)CC(F)CCN1C(c1cncc(Cl)c1)=O 91298,n1(CC(=O)NOCC(N2CCC2c2ccccc2Cl)=O)cnc(C(=O)O)cc1=O 91299,c1(OC)cc(S(N)(=O)=O)ccc1NC(C1CSCCN1Cc1nc(C)cs1)=O 91300,c1(C(=O)NC(C(=O)NCCC(C)O)C2CCOC2)c[nH]c2ccccc12 91301,c1(CNC(CN2CCN(C(C(CCC)NC(C)=O)=O)CC2)=O)ccc(Cl)c(Cl)c1 91302,C(=O)(C(C)C(C)NC(c1cnc(OC)s1)=O)N(CCCOCC)CCO 91303,CC(C)C(CC(=O)NC1(C(N)=O)CCCCC1)NC(C1CCC2(CCC2)C1)=O 91304,N1(C(c2c(CC)cno2)=O)CCC(C)(C(=O)N(CC(C)C(F)(F)F)C)C1 91305,c1(CCn2cc(C3(F)CN(C(C4(C)CCOC4)=O)C3)nn2)ccc(F)cc1 91306,N1(C(C2(CC#C)CCC2)=O)CCC(CO)(NC(=O)CCc2ccc(Cl)s2)C1 91307,CC1CN(C(C23CCC(CC2)OC3)=O)CCC1NC(=O)CC1CC=CCN1C 91308,C1(C(=O)Nc2ccnc(Cl)c2Br)Cc2cc(O)ccc2CN1Cc1cnc(Br)s1 91309,C(=O)(C#CC1CCCCC1)NC1C(NC(C(CCCC)CC)=O)COC1 91310,C1(C(N(CC(COCC)O)C)=O)C2CN(C(C3(F)CC=CCC3)=O)CC12 91311,N1(C(C2(N(C)C)CCC2)=O)CCCC(C)(C(=O)NCCc2ccccn2)C1 91312,N1(C(CC(C)F)=O)C(CNC(c2cc(C3CCCC3)no2)=O)CC2CCCCC12 91313,N1(C(C2C(C)C2C)=O)CCC(C(C)C(=O)NCCCC2(O)CC2)C1 91314,c1(C(N2C(CNC(c3c(C)cno3)=O)CCCC2)=O)c(O)nnc2c1CCCC2 91315,Cc1ccc(CCCC(=O)NCC(C)NC(c2ccc(O)nc2C)=O)cc1C 91316,C1(CNC(C2(C)C=CCCC2)=O)CN(C(c2cc(O)ncn2)=O)C2CCCCC12 91317,N1(C(COCCCCC)=O)CC2CCN(C(c3ccc(F)c(F)c3N)=O)C(C2)C1 91318,Cc1cc(=O)n(C)cc1C(=O)NCC1C(CNC(=O)C=CC2CCCN2C)C1(F)F 91319,c1(NC(C(C2CCN(C(C3C(C)(C)C3(C)C)=O)C2)F)=O)ccc(O)cc1F 91320,c1(NCC(N2CCN(CC)CC2)(C)C)ccc(S(=O)(=O)NC2CC(F)C2)cc1C#N 91321,c1(C(=O)NC(CNC(c2c(C)nc(CC(C)C)s2)=O)C2CC2)cn2c(n1)CCC2 91322,c1(CNC(=O)NC(c2cc(Cl)ccc2O)C)nnc2n1CCS2 91323,Cn1ncc(C(=O)NCc2occc2C(=O)NCC2CCCSC2)c1N 91324,c1(CN2CC(NC(=O)C=Cc3ccsc3)C2)cccc(C(=O)O)c1F 91325,C(=O)(C(C)CCCC(C)=O)NCC(C)=CC(=O)NC(C)Cn1cnnc1 91326,c1(C(=O)NCC(CC)NC(=O)C(c2ccc(F)c(C)c2)=O)nc2ncccn2n1 91327,C(=O)(C1=CCCCC1C)NCc1ccc(C(N2CC=C(C)C2)=O)cn1 91328,C1(NC(C(c2n(C)ccc2)=O)=O)CCCC(NC(c2cnsn2)=O)C1 91329,C1(C(N2CC(NC(=O)C=CSC)C2)=O)(NC(CNC(C)=O)=O)CCC(C)(C)C1 91330,Cc1cc(Br)ccc1CN1CC2(CC2C(=O)N(C2CCOCC2)C(C)C)C1 91331,C(=O)(N=c1nc2ccc(I)cn2[nH]1)Nc1c(C)c(O)ccc1 91332,N1(C(=O)Cc2cccnc2)CCCC(C2CN(C(C34CCC(CC3)OC4)=O)C2)C1 91333,CC1CCC(c2nnnn2CCOC(C)(C)C)(NC(C)Cc2cnccn2)C1 91334,C(=O)(C1Cc2ccccc21)NCC(CCNC(C1CC2(CC(=O)C2)C1)=O)O 91335,C1(CCC)(NC(C2CC3(CCC3)C2)=O)CCCN(C(C2CS(=O)C2)=O)C1 91336,N1(C(C(C2CC3CCC2O3)NC(C)(C)C)=O)CC23CCCC2(C1)C(=O)NC3=O 91337,c1(CNC2C(CC=C)CCCC2)cc2cccc(OC)c2o1 91338,CC(C)C(C(=O)N1CCC(CO)C(NC(=O)CSCC(F)(F)F)C1)C(C)C 91339,c1(C(=O)NC2CCN(C(C3C(C=C)CC3)=O)CC2CO)cccc2c1CCC2 91340,C=C1CC(C)(C(=O)NC2CCCC2NC(=O)CCC2CCC(C(N)=O)O2)C1 91341,c1(C(=O)OC)cc2c(Cl)c(-c3ccc(C)c(C)c3)ccc2s1 91342,C1(C(N2CCCC(O)(CNc3ncc(F)cn3)C2)=O)CC2CCC1CC2 91343,C1(C(=O)NC(C)CNC(=O)Cc2cn(C)nc2Cl)CCc2nnc(O)cc2C1 91344,C1(CNC(c2ccc(CC(C)(C)O)s2)=O)CCCCN(C(C2CC=CCC2)=O)C1 91345,c1(NC(C(C)(O)C2CCCCC2)=O)cc[n+]([O-])cc1 91346,O=C1CCc2cc(OCC(=O)Nn3cncn3)ccc2N1.C(C1CC1)C1CC1 91347,Cc1nc(C(=O)NCC(C)C2CC2)ccc1C#N 91348,N1(C(c2c(C)cc(C3CC3)nc2)=O)CC2(CCC(NC(=O)CN(C)C)CC2)C1 91349,C1(NC(c2cccnn2)=O)CCC2CN(C(=O)C=CC=C(Cl)Cl)CC2C1 91350,N1(CC)CCCC1C(=O)NCCCSc1cc(C)no1 91351,C1(C)(CN(C(CCCC)=O)C)CCCC1NC(=O)CC1CCCOC1 91352,Cc1cc(NC(C2CCN(C(c3cnn4cc[nH]c34)=O)C2)C)ncc1[N+](=O)[O-] 91353,C#CC1(C(=O)N(C)CC2CCCC2(C)C)CCN(C(=O)C(O)CC(C)(C)C)CC1 91354,c1(OC)cccc(C(N2CCCC2C(C)NC(=O)C2CC2)=O)n1 91355,c1(CN2C(CNCC3(O)CCNCC3)CC(OC)C2)cnc(N(C)C)cc1Cl 91356,N1(C(C2CCCCO2)=O)CCNC(C(N2CCCC(F)C2)=O)C1 91357,N1(C(C2CCC(F)(F)C2)C(=O)NC2CCC2)CCc2ncc(C(F)(F)F)cc2C1 91358,C1(NC(c2on(C)c(=O)c2)=O)CCCCC12CCN(C(C1OCCC1(C)C)=O)C2 91359,c1(C(N2CCOC(C(N3CC(F)(F)C(F)(F)C3)=O)C2)=O)cc2cc(F)ccc2[nH]1 91360,C1(C(N(C(C)(C)CC(N2CCC(F)CC2)=O)C)=O)CCCCC(=O)N1 91361,c1(NC(CNC(CC=CC=C)=O)C2CCC2)nc2c(C(=O)OCC)cccc2o1 91362,CN(C)N=Nc1ccccc1C(=O)NC1CCC(NC(=O)CC2CCCO2)CC1 91363,c1(C(=O)NC(C(CO)NC(c2c(CC)scc2)=O)C)cc(F)cc2cc[nH]c12 91364,C(=O)(C(CC(C)C)C(C)C)NC(C(=O)N(C1CC(C)C1)C)CCN(C)C 91365,c1(C(N(C)CC2OCCN(C(C3(C=C)CCC3)=O)C2)=O)cnn2cccc(Cl)c12 91366,C(=O)(CCCCCF)NC1(C(N2CCC(C(C)OC)CC2)=O)CCN(C)C1 91367,N1(Cc2c(C(=O)OC)c(Br)c(Br)s2)CCC(C2=NOCC2)C1 91368,c1(C(=O)NC(CC=C)CNC(=O)C(C)CC2CC2)cnn2ccnc(C)c12 91369,C12(C(=O)OC(CCCCCC)N=[N+]=[N-])CCCC1N(C(C)=O)CC2 91370,C12(CNC(C(CC#C)C)=O)CC(CO1)N(C(=O)CC(C)(C)C#N)C2 91371,c1(OC)cccc(C)c1C(=O)NC(C)C(c1ccccc1)NC(C12CCC1C2)=O 91372,CCN=C(NCCc1cc(OC)cc(OC)c1)N1CCC(CNN2CCOCC2)C1 91373,C1(CNC(CCC=CC)=O)CCN(C(c2cnc(C(F)(F)F)s2)=O)CC1C 91374,N1(C(c2coc(C(F)F)n2)C(=O)NCCCSC)CCC2C(O)CCCC2C1 91375,Cc1ccc(Cl)cc1C(=O)NCC(C)CNC(C12COC(C1)C2)=O 91376,c1(C(N2CCC(NC(C(CC)O)=O)CC2)=O)c(Br)sc(C)c1C 91377,n1(CC)ccc(=NC(=O)C(CCOC)NC(c2coc(C(F)F)c2)=O)[nH]1 91378,N1(C(COCCCC)=O)CCCC(NC(=O)C(C)N2CCC2)C1 91379,C1(C(=O)NC(c2nncs2)C)CC12CCN(C(c1ccc(O)cn1)=O)C2 91380,C(CCC(C)C)(C(=O)NC1CCCN(C(=O)C(F)n2ccnc2)C1)NC(C)=O 91381,c1(C(=O)NC2CN(C(Cn3nc(C)oc3=O)=O)CC2(C)C)ccc2c(c1)CCC2 91382,C(=O)(C(CC(C)C)ONC(=O)CC1CC(F)C1)N(CC)CC1(O)CCC1 91383,C12(NC(COCC(=C)C)=O)CCCC1N(C(c1ccc(O)cn1)=O)CC2 91384,CCC(C)(COC)C(=O)N1CC(CNC(c2ncc(Br)cc2OC)=O)C1 91385,c1(C(=O)OC)ccc2c(c1)OC(CNC(=O)CCC1CC(F)(F)C1)C2 91386,C(c1ccc(C(F)(F)F)c(O)c1)=CC(=O)Nc1[nH]c(=NCC)sc1 91387,N1(C(c2c(SC)cccn2)=O)CC(NC(c2csc(C)c2)=O)CCC1C 91388,c1(CC)cc(C)c(C(=O)NC2CCCC2CC(=O)N(C2CC2)Cn2cccn2)o1 91389,c1(C(=O)NC2CCC2NC(C2CCCC2)=O)cnc2[nH]nnc2c1 91390,CCCCCCC(CC)C(=O)NCC1CN(C(C2(CCO)CC2)=O)CCC1(F)F 91391,c1(N(CCN(C(c2c(OCC)nc(C)cc2)=O)CC)CC)c([N+](=O)[O-])cnn1C 91392,CCCC(C#N)C(=O)NCC1(NC(=O)C=Cc2ccc(C(=O)NC)cc2)CC1 91393,C1(C2CC2)(C(=O)NC(COC)C2CC2)CN(C(=O)C=Cc2ccoc2)C1 91394,Cc1ccc(CN(C)C(C2C3CN(CCSc4nc(C)c(C)[nH]4)CC23)=O)cc1 91395,c1(C(N2C(C(N(CC#C)CC#C)=O)CC2C)=O)coc2c1COC2 91396,C1(NC(=O)C=CCO)CC2CC1CN(C(c1coc(Sc3ncccn3)n1)=O)C2 91397,c1(C(=O)NC2C3CN(C(c4c(C)cc(C)[nH]4)=O)CC32)cc2c(ccn2C)s1 91398,N1(C(C(C)n2cccn2)=O)C(CC(N2CC(O)(C(F)(F)F)C2)=O)C2CCCC12 91399,CCC(CC1CCCC1)C(=O)NC(C)CC1CN(C(c2c(C)[nH][nH]c2=N)=O)C1 91400,c1(C(N2CC(C)N(C(c3ccc(Cl)[nH]3)=O)CC2)=O)ccc2c(c1)NC(=O)C2 91401,N1(c2onc(C)n2)CC(C(N2CC(NC(=O)CNS(C)(=O)=O)C(C)C2)=O)CC1=O 91402,N1(C(c2cc(-c3cccnc3)[nH]n2)=O)CCC2C1CCCN2C(c1nc[nH]n1)=O 91403,c1(CN(CCn2ncc(Br)n2)CC)ccc(Br)c(Oc2ccccc2)c1 91404,CC(C)CCCNC(=O)C(C)CC1CCCO1.N12CC(O)(C1)C(C)(C)CCC2=O 91405,N1(C(COC2CC2(F)F)=O)CCN(C(c2ccc(O)cc2)=O)CC(C)(F)C1.CSC 91406,Cc1csc2ccc(C(=O)NCCC(C)(C)NC(C3CCC4CC34)=O)cc12 91407,C1(NC(c2c(C)cno2)=O)CCC2(C1)CN(C(C1(C)CC1)=O)C2 91408,C1(C(=O)NCc2ccsc2)CC12CCN(CCC1(F)CC1)CC2 91409,N1(C(CC2C(C)CC2)=O)CC(NC(C2CC3(CCC3O)C2)=O)CC12CCCCC2 91410,C1(NC(c2nc(OCC)oc2)=O)CN(C(=O)C(C)c2cccs2)CCC1F 91411,CS(=O)c1ccccc1C(=O)NCC1(O)CN(C(=O)C=CC2CCCO2)C1 91412,CC(C)CC(CNC(=O)C(C)(C)CO)C(=O)NCC(C)CCCO 91413,c1(C(=O)NCCC(C)C)n[nH]c2ccc(-c3ccc(-c4cncs4)cc3)cc12 91414,C1(C(N2CCN(C)CC2CO)=O)CC2(CCC2)CN1C(=O)CN1CCNC1=N 91415,c1(CC(=O)NC(C2CCN(C(=O)C(C)(C)CC3CC3)C2)C)ccc(C#N)cc1 91416,CCCCCC(O)C(=O)NC(C)(CNC(c1cc(C)ccc1C(C)C)=O)C1CC1 91417,N1(CCNC(=O)Cc2cncs2)CCN(C(C2(CO)CCOCC2)=O)CC1 91418,Cc1nc(C)c(C(N2CCC(C)(CCNC(C3(CF)COC3)=O)C2)=O)nc1C 91419,C1(C(N2CC3C(NC(c4cc(C)cc(O)c4)=O)C3C2)=O)(OC)CCC(C)(C)C1 91420,Cc1nn(C)cc1C(O)C(=O)NC1CCN(C(=O)C(=Cc2cccnc2)F)C1C 91421,c1(NC(c2c(Nc3nccc(OCC)n3)ccs2)=O)cc(C(N)=O)cc(F)c1 91422,c1(CCC(=O)NC(CNC(=O)COC2CCCOC2)C2CC2)ccc(F)c(F)c1 91423,c1(CN2CCCC(C(=O)OC)C2)cccc([N+](=O)[O-])c1.C12CC(CN1C)NC2=O 91424,C1(F)(CNC(CN(c2ccccc2)CC)=O)CC(NC(C2C3COCC23)=O)C1 91425,C(=O)(C(F)C(F)(F)C(F)(F)F)N(c1c(OC)c(Cl)ccc1)C 91426,c1(C(=O)NCC2(C(=O)NCC(C(C)C)(C)F)CC(C)(C)C2)cc(O)cc(F)c1 91427,Cc1cc(C)n(CC(=O)N(CC(CO)(CO)NC(c2cn[nH]c2)=O)C)n1 91428,Cc1cc(NCC=CBr)ncc1S(=O)(=O)N1CCN(C=O)CC1 91429,CN1CCN(CC(N2CCCC(NC(c3cccc(N)n3)=O)CC2)=O)CC1=O 91430,C1(NC(c2cnc(S)nc2)=O)CC(C(N2CCN(C3CC3)C(=O)C2)=O)C12CCC2 91431,C1(NC(=O)COc2ccc(Cl)cc2)CCN(C(C2CCOCC2)=O)CCC1CO 91432,C1(C(N(CCN(C(=O)CCOCC2CCCO2)C(C)C)C)=O)CCCCS1 91433,C(=O)(C1=CCCSC1)NC(C(C(=O)NCCN1CC=C(C)CC1)C)C 91434,C1(C)(C(=O)NCC=CC(C)N)CC=CCC1 91435,C1(NC(c2ccnn2CCF)=O)CC2CCC(C1)N2C(=O)CC1CCCC(=O)N1 91436,c1(CC)c(C(=O)NC2CC2CNC(=O)Cn2nnnc2C2CC2)ccn1C 91437,c1(C(C#C)NC(=O)N(c2cnn(C)c2)CC#C)cccc(Br)c1 91438,CCC(C(=O)Nn1ccnn1)NC(=O)C#CC(C)(C)C 91439,c1(CCCCC)nc(C(N2CCC2CNC(C2CCC2C(F)F)=O)=O)cs1 91440,c1(C(=O)NCC(N(C(CCOC)=O)C)C2CC2)ccc(S(C)=O)cc1 91441,CCCCC(C)C(=O)NC1CN(c2ncccc2Br)C1 91442,c1(OC)cc(NCC2CC(NC(c3cncc(C)c3)=O)C2)nc(C(F)(F)F)n1 91443,C(CNC(c1cnn(CC2CC2)c1)=O)(CC(F)(F)F)NC(C1(C#C)CC1)=O 91444,N1(C(=O)NC2CC2)CCC2(COC(C(=O)OCCCNC(c3nc[nH]n3)C)C2)C1 91445,c1(OC)ncc(C(=O)NC2CC(C)(NC(=O)CCC3CC3C)C2)c(C)n1 91446,Cc1cn2c(C(=O)NC(C)C(CO)NC(C3(F)CCOCC3)=O)c(Cl)nc2s1 91447,C(=O)(C1=CC2C=CC(C1)C2)NCC(CCNC(CC1CCN(C)C1=O)=O)(C)C 91448,c1(C(=O)OCC)ccnc(NC(CNC(C2CC2F)=O)C(C)C)c1[N+](=O)[O-] 91449,c1(SC)ncc(C)c(N2CCN(CC(=O)Nc3cccc(C(F)F)c3Cl)CC2)n1 91450,C(=O)(CCC(C)(C)C#N)NC(CCCNC(CCc1ccc(OC)c(C)c1)=O)C 91451,C(=O)(CCCCCN=[N+]=[N-])N(C)CC.C(=O)(CCC1CCC1)N(C)CCOC(F)F 91452,c1(C(=O)NC2C(C)(C)CCN(C(C3CCCCS3)=O)C2)cnc2ccc(F)cn12 91453,N1(C(C2ON=C(C)C2)=O)CCN(C(=O)CC#N)CC1C(C)C 91454,C=CC(C)(CC)C(=O)NCCC1CSCCN1C(c1cc(=N)[nH]n1C)=O 91455,N1(C(c2cc(CC)n(C)n2)=O)CCC(CNC(c2cnn(C)c2)=O)C(F)(F)CC1 91456,N1(C(c2nc(CC)sc2N)=O)CCC(C2(NC(=O)C(O)C3CC3)CC2)CC1 91457,c1cnc2ccc(-n3nc(C4CCCO4)nc3CC3CC3)cc2c1 91458,N1(C(c2cnc(CC(C)C)s2)=O)CC(CNC(C2(CC(C)C)CCC2)=O)C2CC12 91459,C1(C(N(C)CC2CCN(C(=O)CN(S(C)(=O)=O)C)C2)=O)CCCC(F)(F)C1 91460,N1(C(C)C)CC2CCC1CN2N1CC(C(=O)O)C2CCCC12 91461,c1(C(=O)NCC(N(C(=O)CN2CCOCC2)C)C2CC2)cc(F)cnc1Cl 91462,c1(C(C(=O)NC(CC)(C)C)N(C)Cc2cncnc2)ccc(C)c(C)c1F 91463,C=CCCCCCCCC(=O)NC1COCC1CNC(C1CCSC1)=O 91464,C12(C(N3CC4C(CNC(c5cccc(F)c5O)=O)C4C3)=O)CC3CC1C2C3O 91465,C#CCC(C)(C)C(=O)N(CCC(C)NC(c1ccccc1OCC#N)=O)C 91466,c1(CC)nn(C)cc1C(=O)NCC(C1CCC1)NC(C1(OC)CCSC1)=O 91467,C(=O)(C(C)(C)CN(C)C)NCc1nc(OCC)oc1 91468,CC1(C)CN(C(=O)CSC(F)F)CC1NC(C1(F)CCCC1)=O 91469,N1(C(C2C3CC(C)(C3)OC2)=O)CC(NC(c2cccnc2)=O)CC12CCOCC2 91470,N1(C(C(C)NC(=O)OC)=O)C(C)CC2CN(C(c3ccc4c(c3)CCO4)=O)CC12 91471,c1(CCC(=O)N(CC(C)NC(C2CC2(C)C)=O)C)ccccc1[N+](=O)[O-] 91472,C1(CNC(C(CN(C)C)NC(C2CC2C(C)(C)C)=O)=O)CCCC12CC2 91473,Cc1c(NCC2(c3ccccc3)CC2(C)C)ncnc1NC1CC(F)(F)C1 91474,C1(NC(Cc2c(C(=O)OC)csc2)=O)CC2CC(NC(=O)CCc3nccs3)CC12 91475,N1(C(C(C)N(C(C)=O)C)=O)CC(C2(NC(C3CN(S(C)(=O)=O)C3)=O)CC2)C1 91476,c1(CC)ocnc1C(=O)NC(CNC(c1ncc(C(F)F)s1)=O)C1CC1 91477,Cc1nc(C)c(C(N2CCC(CNC(=O)C(F)C3CCC3)C(F)(F)C2)=O)nc1C 91478,c1(C(=O)NCC(CO)NC(c2n(CC)ccn2)=O)cccc(C2CC2)c1 91479,CN1CCN(C)CC(C(=O)N(CCCNC(C2(n3cncn3)CC2)=O)C2CC2)C1 91480,CC(=O)CCN=C(NCC(=O)NCCOC1CCC1)NC1CSC1(C)C 91481,N1(C(C(C2(O)CCC2)NC(C(COC)OC)=O)=O)CCC(CO)=C(F)C1 91482,C(c1cncc(C)c1)=CC(N1CCC(C(=O)NCC(=O)OC)CC1)=O 91483,C1(CNC(CC(C)(C)C)=O)CCN(C(C2CCN(c3ccccc3)C2)=O)C12CC2 91484,c1(CNC2CN(C(c3n(C)cnc3)=O)CC2F)cc2c(Br)cccc2s1 91485,CC1=CCC(C(=O)NCCCC2CCCN2C(c2csc(C(N)=O)n2)=O)CC1 91486,N1(C(C(C)CN(C)C)=O)CCCOC(CCNC(c2ccc(Br)cc2)=O)C1 91487,C1(C)(C(=O)NCC(CC)NC(=O)Cc2ccsc2Br)CCCC1(F)F 91488,N1(C(CSCCN(C)C)=O)CCCC2(CCC(NC(C3CC4CCC3C4)=O)C2)C1 91489,c1(C(=O)NCC(C)N(C)C(C23CC2C3)=O)ccc(N)c(N)c1 91490,CCCCS(=O)(=O)CC(=O)N1CCCC2CN(C(c3cc[nH]c3C3CC3)=O)CC12 91491,CCS(=O)(=O)c1cccnc1C(=O)NCCCN(C)C(C12COCC(C1)OC2)=O 91492,c1(CSC(C)C(=O)NC(C)(CNC(c2nnsc2C)=O)CO)ccccc1Cl 91493,C1(CC(=O)NC2C(CC(C)(C)C)C2)C2CCCC2N1C(c1ccc(C(N)=O)o1)=O 91494,N1(C(CNC(C)=O)=O)CCCC2(NC(=O)COc3ccc(C#N)cc3)CCCC12 91495,C1(CNC(C2(CC=C)CCOCC2)=O)CC(C)(C)CN1C(c1cnccn1)=O 91496,c1(C(N2CC(CC)N(C(=O)CO)CC2)=O)c(C(F)F)nc2n1CCCC2 91497,N1(C(C=CCOC)=O)CC(NC(C2CCN(C(=O)OC(C)(C)C)C2)=O)C(O)C1 91498,C#CC1(C(=O)NCCOCCOCCOC)CN(C(=O)C(O)CCN(C)C)C1 91499,Cc1cc(C)c(C(=O)N(S(=O)(=O)CC2CCCC(C(F)(F)F)O2)C2CC2)o1 91500,C(=O)(C(CC(C)(C)C#N)N1CCN(C)C(=O)C1)NCCCCC 91501,CC(C)(C)CCC(F)C(=O)NCC1CN(C(=O)C2=NNC(=O)CC2)CCC1(F)F 91502,C1(NC(C2C(C(C)C)C2)=O)CN(C(=O)C2=CC(C)C2)C2CCCC12 91503,c1(CNC(C2(OCC)CCC2)=O)cc(C(=O)NCCSCCO)no1 91504,C1(CNC(=O)C=CCN2CCCC2)CCCCN1C(C1(Br)CC1)=O 91505,CC1CCN(C(c2cc3ccsc3[nH]2)=O)CCN1C(=O)C=C1CCSCC1 91506,c1(C(=O)NC2(C)CCN(C(c3n[nH]cc3Cl)=O)CC2)cc(F)cc(N)c1F 91507,c1(C(N(C2CCN(C(C3CC3COC)=O)CC2)CC#C)=O)cccc2sccc12 91508,c1(OC)c(C(=O)N(C2CC(NC(C3CCCC3O)=O)C2)C)cc([N+](=O)[O-])cc1Cl 91509,c1(OC)ccccc1C=CC(=O)NC1CCCCC1N(C(=O)CSC(F)F)C 91510,CCC(CC)C(C)C(=O)N1CCC(O)(CN(C(=O)CC23CCCN2CCC3)C)C1 91511,Cc1ccc2c(C(=O)N(C(C)CCNC(=O)C(CN(C)C)C(C)C)C)csc2c1 91512,C1(NC(C2(C(N)=O)CC2)=O)CCCC(C(=O)N(CCCOCC#N)CCO)C1 91513,CCCC(CCCNC(C1(C)CC1C)=O)NC(C1CCN(CC(F)F)CC1)=O 91514,Cc1ccc2[nH]c(=NCC3(O)CN(C(C4CCCC5(C4)CC5(F)F)=O)C3)sc2n1 91515,C#CC1CN(C(=O)COC(C)CC)CCN1C(=O)Cc1n[nH]c(=N)s1 91516,N1(c2cc(C)nc(CO)n2)C2CCC1CC(CNC(c1cc3c([nH]1)CCC3)=O)C2 91517,CCCC(C(=O)NC1CCCC(NC(c2ccc(N)c(SC)c2)=O)C1)S(N)(=O)=O 91518,C=C=CC(C)C(=O)NC(c1ccc(F)cc1)CNC(c1ccn(C2CCC2)n1)=O 91519,C1(NC(C(C2CCCCCC2)C)=O)C2CC1N(C(=O)COC1(C)CCC1)C2 91520,CCCCCCC(F)C(=O)N1CCC(CN(C(=O)CC2(O)CCOC2)C)CC1 91521,N1(Cc2cn(CCNC(=O)CC3CC4(CCC4)C3)nn2)CCCCCC1=O 91522,c1(NC(C(CC)C)c2nnnn2CC2CCCO2)ccc(C#N)c(F)c1 91523,c1(C(=O)NCC(CNC(CCC(C)N(C)C)=O)O)cc(Cl)cc(Br)c1 91524,c1(CC)ccc(Br)cc1C(=O)NCC=Cc1nnn(C)n1 91525,CCC(C)CCC(O)CC(=O)NC1CCN(C(=O)CCS(N)(=O)=O)CC12CCC2 91526,C12(CNC(Cc3cccc(C)c3)=O)CCC(C1)N(C(C1CCCCCCC1)=O)C2 91527,Cc1nnc2ccc(C(=O)NC3CCCC(NC(C4CC(F)C4)=O)C3)cn12 91528,C(=O)(CC1C(=O)Nc2ccccc21)NC1CCN(C(c2ccc(C)[nH]2)=O)C1(C)C 91529,Cc1ccc(C(C)NC(=O)CN(C(=O)CCN2CCCCC2)C2CCC2)nc1 91530,c1(NCC=C)[nH]c(=NCC2C(F)(F)C23CCC3)nc2c1ncn2C 91531,CS(=O)(=O)CCC(=O)NCC1CC(CNC(c2cn3ccnc3s2)=O)CO1 91532,N1(C(CC2CC(C)C2)=O)CCc2nc(CNC(=O)C(C)(C)C(C)(C)C)sc2C1 91533,N(C(=NCCC(C)C)N1CCN(c2ccc(C)cc2)C(=O)C1)CCC(=O)NC 91534,C12(NC(c3cccnc3F)=O)CCCN(C(c3cc4cccnc4s3)=O)CC1C2 91535,C(=O)(CCC(C)(C)C#N)NCC1CC(NC(c2ccc(SC)o2)=O)C1(C)C 91536,N1(C(c2c(CN(C)C)cco2)=O)CCCC2(CCCN2C(=O)Cc2ccon2)C1 91537,C(=O)(CCCCCc1ccccc1)N1CC(NC(C(CC)=CC)=O)C(OC)C1 91538,N1(C(CCc2nc(C)sc2)=O)CCCC12CCN(C(C1CCC1(F)F)=O)C2 91539,N1(C(C2(C)CC(C)(C)C2)=O)C(C(=O)N(CC2CC2)CC2CC2)C2CC(O)C1C2 91540,C(=O)(C1=CC2CCCCCCC12)N1C(C)(C)C(CNC(=O)CCF)CC1 91541,N1(C(COC2(C#C)COC2)=O)CCN(C(=O)C(C)CC=C)C2COCC12 91542,c1(C(=O)NC(CC)CNC(c2ncn(C)c2C)=O)cnc2ncnn2c1C 91543,c1(C(CNC(CCOC)=O)NC(C2(F)CCOCC2)=O)ccccc1F 91544,C1(CN2CCN(C(=O)Cn3ccnn3)CC2)CCCC2(CCC2)O1 91545,c1(CC)c(C(=O)NCCNC(C2CCCN2C(C)C)=O)cnc2ncnn12 91546,C=CCN=c1[nH]cc(C(=O)NC2CN(C(=O)CCC3CCC(=O)N3)CC23CC3)s1 91547,c1(C(N(CCCNC(=O)C(C(C)O)N(C)C)CC)=O)ccc(S(=O)(=O)CF)nc1 91548,Cc1nc(C=CC(=O)NCC(C)CNC(=O)C=Cc2nnn(C)n2)cs1 91549,Cc1cnn(C(C)C(=O)NCC2CC(F)(CNC(c3cnn(CCO)c3)=O)C2)c1 91550,N1(C(C2C(C#N)C2)=O)CCC(N(C(=O)C2CC2)Cc2ccccc2)CC1 91551,C1(CN(C(c2c(OCC=C)cccc2)=O)C)CN(C(=O)C=CCOC)CC12CC2 91552,c1(OC)c(O)cc(C(=O)NCC2CC(F)CN2C(=O)C(C)OC)cc1C#N 91553,c1(N2CC(C(=O)Nc3nc(C(F)(F)F)cs3)SCC2)ccn2ncc(I)c2n1 91554,CCC(CC)(CCNC(=O)C(C)(CC)OC)NC(=O)CSC(F)(F)F 91555,C(=O)(C(C)(C(C)C)OC)N(CC(C)N(C(CCN(CCOC)C)=O)C)C 91556,C(=O)(C(F)C(C)(C)O)NCCOC1CCN(C(CC2(C(=C)F)CCC2)=O)CC1 91557,C1(C)(CC)CCC(N=c2[nH]c(=NCc3ccncn3)[nH]c3c2CCCC3)CC1 91558,N1(C(c2cc(OC)c(OC)nc2)=O)CCN(C(=O)CS(=O)(=O)N(C)C)C2CCC12 91559,CC1CN(C(C2(C)CCCN2C(=O)Cc2cncnc2)=O)CC1N=[N+]=[N-] 91560,C1(NC(C(C2CC2)Sc2c(OC)cccc2)=O)CCN(CC)C(C2CC2)C1 91561,Cc1nn(CC(=O)NCC2(O)CN(C(=O)CSCc3ncc[nH]3)C2)c(=O)n1C 91562,C1(C(=O)NC(CC)C2CC2)(NC(=O)CC(C)F)CC(F)C1 91563,C1(C(=O)NC(CNC(CCCC)=O)C(C)C)(OC)CCC(F)(F)CC1 91564,N1(C(N(c2cccc(S(C)(=O)=O)c2)C)=O)CCCC2(CC1)CNC(=O)N2 91565,N1(C(CC(C)(C)C)=O)CCN(C(c2cnn(C(C)(C)C)c2)=O)C(CS(C)(=O)=O)C1 91566,Cn1nc(C(F)F)cc1C(=O)NCC(c1ccccc1)NC(C1CC2CC1CO2)=O 91567,C(=O)(CCC[N+](=O)[O-])NC1(C)CCN(C(=O)CC2CC(F)(F)C2)C1 91568,c1(C(=O)NCCOCC(=O)NC(CC#C)C)cnn(C)c1C1CC1 91569,c1(C(C)C(=O)N(c2cn(C)nc2Cl)CC2CCOCC2)ncc2ccccn12 91570,c1(N2C(CNC(CC(C)C3CC3)=O)CCCC2)ncnc2sccc12 91571,N1(C(C(C(C)C)N(C)C)=O)CCC2(CCN(C(C3CCCC3O)=O)C2)C1 91572,c1(NC(c2ncn(C)n2)C)ccc(S(=O)(=O)NCC2CSCCO2)cc1Cl 91573,C(=O)(C1=CCCSC1)NC(c1c(CC)cccc1)CNC(=O)C(F)OC(F)(F)F 91574,c1(NC(C2N(c3nc(C)c(F)cn3)C3C(C2)C3)=O)cc(F)c(C)c(Br)c1 91575,c1(C(=O)NC2C3(CN(C(CC(=O)NCC)=O)C3)CC2)cccc2c1OC(F)(F)O2 91576,CC1CCN(C(=O)CCC2(C)CC2(F)F)CC1NC(C1CC=CCC1)=O 91577,N1(C(c2n(C(C)C)ncn2)=O)CCC(CF)(NC(c2ccc(C(F)F)nc2)=O)C1 91578,C(=O)(C(C)(C)C(C)NC(C1CCO1)=O)NCC(C(F)(F)F)OC 91579,c1(C(N2CC(NC(C3(C)N(C(C)=O)CCC3)=O)C2)=O)ccc(P(C)(C)=O)cc1 91580,C1(C(=O)NCc2cnc(C)[nH]2)C2CC3C(C2NC(=O)CC2CNC(=O)O2)C13 91581,C=CC(C)(C)CC(=O)N(C1CCN(C(c2oc(Br)cc2C)=O)CC1C)C 91582,c1(-n2cc(NS(CC)(=O)=O)nn2)ccc(OCCN(C)C)cc1 91583,c1(C(=O)NC2CC2)nccnc1N.c12cc(cs1)CN(C)C(=O)CCNC2=O 91584,c1(-c2n(CCOC)c(N3CC4CC3(C)C4)nn2)ccc2cn(C(C)C)nc2c1 91585,CC(C)(C)C1=NOC(C(=O)NC2CC(NC(=O)Cn3cnnc3O)CC2O)C1 91586,CCCCC(C(=O)N1CC2CC2(C(=O)OC)C1)NC(=O)CCCCCF 91587,N1(C(CCCCOC)=O)CC(F)(F)CC1C(N1CCN(CCF)CC1)=O 91588,C(CC(O)CC(=O)N1CCCC(NC(C2(C)CCOCC2)=O)C1)SC 91589,C1(C)(C(N2CC(CNC(CNC(CC)=O)=O)C2)=O)CCOC(C)C1 91590,C1(CNC(c2c(SCC)cccc2)=O)CCCCN(C(C2CC2(C)C)=O)C1 91591,C1(O)(CC)CCCN(C(C2(OC)CCN(C(=O)C#CC(C)(C)O)C2)=O)CC1 91592,c1(C(N2CC=CC(NC(C(C)(CO)OC)=O)C2)=O)cccc(C)c1C#N 91593,C1(CC(=O)N(CC(CNC(CSCC(C)C)=O)C)C)CCC(=O)C1 91594,C1(CN)CC(C(=O)NC(C)CC(=O)NC)=NO1.CCCCCC(=O)C(C)=O 91595,C1(NC(CC(CC)SC)=O)CN(C(=O)CCc2ncco2)CCC1O 91596,C(=O)(C1=NOC(CC(N2CCC(O)(CNC(C3C4CCCC34)=O)CC2)=O)C1)OC 91597,c1(C(=O)NC(C(C)NC(CCOC)=O)CO)cc(C)c(OC)c(Cl)c1 91598,N1(C(c2c(C(C)C)[nH]cc2)=O)CC(CNC(=O)CC(C)N(C)C)CC(C)(C)C1 91599,c1(N2CCC(N3C(C)(C(=O)OC)CCC3)CC2)nc(C(C)C)nc(C)c1Br 91600,C1(NC(C=C(C)C(F)F)=O)CC1C1CCCN(C(c2ccc3nc[nH]c3c2)=O)C1 91601,c1(N2C(CN3CCN(C)CC3)CCC2)nc(=NC2CC2F)[nH]c2cccc(F)c12 91602,C1(NC(C(N2C(=O)CCC2=O)C)=O)C2CC1N(C)C2.C1(N(CC(=O)N)C)CCCC1 91603,C1(C(=O)NCCCCN(C(=O)Cc2cc(Cl)ccc2O)C)CC(C2CC2)=NO1 91604,N1(C(C)C)CCN(C(=NCC2CCCCC2C)NCc2ccc(F)cc2)CC1=O 91605,N1(C(C(CC)C(C)C)=O)Cc2n[nH]cc2C1C(=O)N(CCCO)OC 91606,N1(C(CSCCCC)=O)CC(N(C(=O)C(C)CC)C)C(C)(C)C1 91607,N1(C(C2C(C)OC(=O)N2)=O)CC(NC(=O)CCc2ccccc2Cl)CC(C)C1 91608,CCC(O)CC(=O)NCC(C)C(=O)NCCc1ncccc1C 91609,c1(C(=O)NCC2CCN(C(=O)COC3CCOCC3)C2)cnc2[nH]cnc2c1 91610,N1(C(Cc2cnn(C)n2)=O)CCC(F)(CNC(C23CCCC(C2)OC3)=O)CC1 91611,C(=O)(CCCC(=O)OC(C)(C)C)N(C)CCN(C)C(C1CC(F)(NC2CC2)C1)=O 91612,c1(C(N)=O)ccc(C(=O)NCCC2CCN(C(C3CC=CCC3)=O)C2)cn1 91613,c1(C(=O)NC2CCCC(CNC(=O)Cc3csnn3)C2)cc2cc(F)ccc2[nH]1 91614,Cc1cc(CC(=O)NCC(C)(C2CCC2)NC(=O)CN2CC=CC2)c(C)s1 91615,C12(C(=O)NCC(C)(C)NC(c3c(C)c(O)ccc3)=O)CCCN1CC(O)C2 91616,N1(C(CCC2(NC(C(CC)C(=O)OC)=O)CCC2)=O)CCC(F)(F)C(C)C1 91617,c1(N2C(C)CC(=O)NCC2)c(C#N)cnc2c(Cl)n(C)cc12 91618,N1(Cc2c(OC)cccc2Br)CCOC2(CCS(=O)(=O)C2)C1 91619,Cc1cc(C(=O)NCC2CCCN(C(C3CCC3(C)C)=O)C2)cc(O)c1 91620,c1(C(N2CC(CCCCNC(COC(C)C)=O)C2)=O)ccc2ncnc(O)c2c1 91621,Cc1cc(=O)c(C(=O)NC2(C3CCCN3C(C3CCCC34CCC4)=O)CC2)c[nH]1 91622,N1(C(C(C(C)O)C)=O)CCC(C2(O)CN(C(C3CCC4(CCC4)CC3)=O)C2)CC1 91623,C1(C(=O)NCC(CC)C)CN(C(=O)CCCC(=O)OC)CC(C)(C)C1 91624,N1(C(CCC(C)C)=O)CCCC2CN(Cc3cc(Cl)ccc3F)CCC12 91625,c1(C(=O)OC)ccccc1C(N1CCCC(C(C)(O)CNC(=O)COC)C1)=O 91626,c1(C(=O)NC(C(C)NC(C(C(=O)NC)(C)C)=O)C)[nH]c2ccc(OC)cc2c1C 91627,N1(C(=O)NC(CCCC=C)C(=O)NC)CCc2c(cnn2C)C1C(=O)OC 91628,C1(NC(C2C(C(C)O)C2)=O)CCCN(C(=O)CC2(C(F)(F)F)CCC2)CC1 91629,C1(NC(C2(OC)CCC2)=O)CCN(Cc2ccc(-c3ccccc3)s2)CC1F 91630,c1(C(N(C2CN(C(C3C(OC)CCC3)=O)CC23CC3)C)=O)cc2sc(C)cc2[nH]1 91631,C(=O)(C(F)C(C)(F)F)NC(C(C)C)CCN(C)C(c1ocnc1C1CC1)=O 91632,C(=O)(C1=CC2CCCCCC12)NCCCC(C)NC(c1cc(C(C)C)on1)=O 91633,N1(C(CCCNC(C)=O)=O)CCCC(C2CN(C(=O)CCc3ccc[nH]3)C2)C1 91634,c1(C(=O)NC2CC2CNC(C2CC3CCC2O3)=O)cc2n(n1)CCOC2 91635,C1(CNC(NC(c2cccs2)C)=NCCc2cn(C)nn2)Cc2ccccc2O1 91636,c1(C(N2CC(NC(C(C=C)O)=O)C(O)CC2)=O)nccn2ccnc12 91637,N1(C(C2(OCC)CCOCC2)=O)CC2(CC(CNC(C3CC(C)(C)CO3)=O)C2)C1 91638,N1(C(C=C(C)C(F)F)=O)CCC(NC(=O)CNC(C2CCCN2C)=O)C1 91639,C(C)(C(C)(C)C(=O)NCCC(O)C(F)(F)F)NC(CC1(CC)CCC1)=O 91640,N1(C(C2=NNC(=O)C2)=O)CC2CCCC(NC(c3noc4c3CCCC4)=O)C2C1 91641,Cc1ncnc(C)c1C(=O)NCC=CCNC(C1CC(c2ccccc2)CO1)=O 91642,N#Cc1c(F)cc(C(=O)NCc2ccc(CNC(=O)CCC(F)F)cc2)cc1F 91643,C1(COC)CC(CNC(=O)CC2CC(=O)NC2=O)N(C(c2cc(Cl)c[nH]2)=O)C1 91644,N1(C(C(CC(C)C)F)=O)CCN(C(c2ncc(F)cc2F)=O)CCC1C 91645,C1(C#N)(OC)CC(C(=O)NCC#CC(=O)NCC2CC=CCC2)C1 91646,C(=O)(C(F)CCC(C)(C)C)NC(C(N1CCCC(C)C1)=O)CO 91647,N1(C(c2c(OCC)scc2)=O)CCN(C(c2cn(C)c(=O)n2C)=O)C2COCC12 91648,N1(C(CN)=O)CCC2(CC1)CC2NC(c1cc2ncccc2[nH]1)=O 91649,CC1(C)CC(CO)CN1C(=O)C1=NOC(CNC(=O)C=CC2CCCCC2)C1 91650,N1(C(C=C(C)C(C)C)=O)CC2C(NC(c3c[nH]nc3F)=O)CS(=O)(=O)C2C1 91651,CC(C)(C)C(=O)N1CCCC1C(=O)NC1(CNC(=O)C=C2CCC2)CC1 91652,C(C(=O)N1CC(N(C)C(c2ccc(Cn3cc(Cl)cn3)s2)=O)C1)(C(C)C)OCC 91653,c1(C(=O)N(CC(=O)Nc2cccnc2)CCO)ccc2nonc2c1 91654,c1(C(N2CCOCC(NC(C(Br)=C(C)C)=O)C2)=O)nc2cnccc2s1 91655,CC1(C(=O)NCCC2CCN(C(=O)Cc3nncs3)C2)COc2ccccc2O1 91656,O(NC(=O)C(Cn1cccn1)NC(C1CC(=O)NC(=O)C1)=O)CC1CC(=C)C1 91657,O=[N+]([O-])c1cccc2c(N3CCN(CCCO)CC3)nc(Cl)cc12 91658,C1(O)(CNC(C(c2cccc(OC)c2)C)=O)CCCN(C(C2(SC)CC2)=O)CC1 91659,c1(C(=O)OCC=CC(CC)C)ccc(S(=O)(=O)C(C)C)cc1 91660,C=CC(C)(CCOC)C(=O)N1CCCN(C(c2cc(CF)on2)=O)C(COC)C1 91661,N1(C(CSCCCC)=O)CCC2(NC(=O)Cc3cnc(C)[nH]3)CCCC12 91662,c1(C(=O)NCC(C23CCC(CC2)C3)O)ccccc1Br 91663,N1(C(C2C(OC)CCC2)=O)CC(C2CN(C(c3cnc(=N)[nH]c3)=O)C2)C1 91664,N1(C(C2C(C(C)C)C2)=O)CCCN(C(c2ccc(CCF)cc2)=O)CC1 91665,c1(C(N)=O)ccc(C=CC(=O)NC2CCC(NC(C3(F)CCOC3)=O)C2)cc1 91666,C12(C(=O)NCC3C(COCC)C3)CCC1CN(C(c1cn(CCO)nn1)=O)C2 91667,c1(OC)cc(OC)c(C(=O)NC2CCC2CNC(=O)Cc2ccoc2C)c(N)c1 91668,CC1(C)C(NC(c2cncnc2)=O)C(C)(C)C1NC(c1ccc(F)s1)=O 91669,C#CC1(C(=O)Nc2cnccc2CO)CN(C(c2cc(C)on2)=O)C1 91670,c1(CC)cc(N)ccc1C(=O)N(C1CCC(NC(=O)C=CS(C)=O)CC1)C 91671,N1(C(C(C)C)=O)CCC(CC(C)NC(C2CCCN2C)=O)CC1 91672,N1(C(C=CC(=O)N(C)C)=O)CCCC1C(=O)NCCc1ccncn1 91673,C1(NC(CC2C(C)(C)N(C(=O)Cn3cncn3)CC2)=O)CCC(C2CC2)CC1 91674,C1(C(=O)NCC(=O)OCC#C)CC1C1CN(C(=O)CCCOCCC)C1 91675,c1(CN(C(=O)Nc2ncc(F)cc2Cl)CC)ccc(F)c(F)c1 91676,c1(CNCC(c2ccccc2Cl)(C)O)cc(Cl)cc(Cl)c1 91677,c1(C(=O)NCC2OCC(CNC(=O)C=Cc3ccccn3)C2)cc(=O)c(O)c[nH]1 91678,C(C)(CNC(=O)Cn1cc(CO)nn1)(CC(C)C)NC(C(CCOC)OC)=O 91679,CC1CC(NC(C2CCC(C#N)CC2)=O)CCN1C(=O)Cc1ccsc1Cl 91680,C1(C)(C(=O)NCc2c(C(N3CC(C(N)=O)(OC)C3)=O)c[nH]n2)CCN(C)CC1 91681,Cc1cc(O)nc(C)c1C(N1CCC2(C1)CN(C(C1(C)CCCOC1)=O)C2)=O 91682,C=C(CC)CN=c1nc(N2CCCN(C(=O)C3CC3)CC2)c2c([nH]1)CCC2 91683,CC1CCc2[nH]nc(C(N3CCC(NC(=O)C4=CCSC4)C3C3CC3)=O)c2C1 91684,C1(NC(C2CC(C(C)C)C2)=O)CCOC(CNC(c2cccc(C(F)F)n2)=O)C1 91685,c1(C(N2CCC(NC(C3N(CC)CCOC3)=O)(CO)C2)=O)ccc(F)cc1F 91686,C1(C(=O)NC(CC)CO)CN(C(=O)C(C)NC(=O)Cn2cnnn2)CCC1O 91687,CCS(=O)CC(=O)NC1(C(=O)NCCOCC(F)(F)F)CCSC1 91688,c1(OCC(=O)NCC2C(NC(COCC)=O)C2)cccc(C(N)=O)c1 91689,c1(N(C2CS(=O)(=O)C2)C2(c3n(C(CC)C)nnn3)CCC2)ccc(F)c(Cl)c1Cl 91690,C1(NC=O)CCCC(NC(=O)CCCC#N)CC1.c1(C(=O)OC)ncccc1CCC 91691,C(c1ccccn1)=C(C(N1CCC(N(C(C2CC(C)(O)C2)=O)CC)C1)=O)C 91692,Cc1cnc(C=CC(=O)N(C)CC2CCN(C(C3CCN3C3CCCC3)=O)C2)[nH]1 91693,C12(NC(C(C(C)C)SCC)=O)CCCC(NC(c3ccc(C)cc3N)=O)(C1)C2 91694,C(CC(C)(C)C(=O)NC(CNC(c1ccccc1NC(N)=O)=O)CO)OC 91695,N1(C(C(C(C)O)C)=O)CCCC2CN(C)CC12.C(=O)(C=CC(=O)NCC)C(C)=O 91696,C1(N(C(=O)CCC2CC(F)(F)C2)CC)CCCN(C(=O)C(CO)NC(N)=O)C1 91697,N1(C(=O)NCC)CCCC(C(=O)NC2(NC(=O)Cc3csc(CC)n3)CCC2)C1 91698,C1(NC(CC(=C=C)C)=O)COC2(CCCN(C(c3cc(NC)ccc3Cl)=O)C2)C1 91699,N1(C(C(CC)n2cncn2)=O)CCC2(CCCC2C(N2CCC3OCCCC3C2)=O)C1 91700,N(C(=NCCCc1ccnn1C)NC(c1ccc(F)c(F)c1)C)C(C#C)CCC 91701,N1(CC)CCN(C(C2CCN(C(=O)C3=CCCC3C)CCO2)=O)CC1(C)C 91702,C1(C)(NC(CCCC)=O)CCN(C(=O)C(O)C(C)CC)CC1 91703,c1(C(N(CC(C)O)CCNC(C2CC(N(C)C)C2)=O)=O)nnn2c1CCCCC2 91704,c1(OC)ccc(Br)c(F)c1CN1CCOC(C)CC1 91705,c1(-c2onc(-c3ccc(-c4ccc(C)cc4)nc3)n2)ccc2ncccc2c1 91706,C1(C(C)C(=O)NCC=CCl)CCN(C(=O)C(C)(C)N2CCCC2)C1 91707,C(C)(CO)(C(=O)NCC1(F)CC(NC(c2cc(Cl)n(C)n2)=O)C1)NC(C)=O 91708,CC1CN(C(=O)NC2CCOCC2)CCN1C(c1ccncc1Cl)=O 91709,Cc1cc(Cl)cc2cc(C(=O)N(CC(O)CNC(C3CS(=O)(=O)C3)=O)C)[nH]c12 91710,C(=O)(C1=CCCOCC1)N1CC(C)CC(NC(c2c(CCC)occ2)=O)C1 91711,N1(C(C(C2CC2)OC)=O)CC(C)(OCC(=O)N(CCCF)C)C1 91712,CC(C)C(C)CC(=O)NC1(CNC(C2CC3CCCC23)=O)CCOCC1 91713,N1(C(c2c(NC(C)=O)c[nH]c2C)=O)CC(NC(=O)C2=CCOC2)C2(CCC2)C1 91714,N1(C(C(C(=O)OCC)CC)=O)CCC2(CC(C(N3CCC(O)C(O)C3)=O)C2)C1 91715,C=CC(C)(O)CC(=O)N1CCC(CC(C)NC(=O)C(n2cc(Cl)cn2)C)CC1 91716,C1(C(=O)OC(C)(C)C)CCN(C(c2ccc(SCc3nncs3)cc2)=O)C1(C)C 91717,c1(SC)ccc(CCCC(N2CC(N(C(=O)C=CCN(C)C)C)C(F)C2)=O)cc1 91718,N1(CCn2c(C)cc(C)n2)CCC(C2CCN(C(=O)CC(C)C(C)C)CC2)C1 91719,C=CCCCCCCC(=O)NCC(=C)CCNC(C1CCCCC12CCC2)=O 91720,c1(CC(=O)NC(C)CNC(c2ccc(C(=S)C3CC3)s2)=O)ccc(Cl)nc1 91721,c1(NC(C(C(C)NC(=O)C(C)(Cl)Cl)C)=O)cc(O)cc(F)c1 91722,N1(C(c2cc(C)nn2C)=O)CCCC2(CCCN2C(c2nc(C)sc2C)=O)C1 91723,c1(CCC)ccc(S(=O)(=O)N2CC3CCC(C2)N(C(c2nnc(C)o2)=O)C3)cc1 91724,c1(C(=O)NCCN(C2CCCC2)C(C=Cc2ncc(C)[nH]2)=O)ccc(Cl)cc1O 91725,c1(C(=O)NC2CCC(N(C(c3nccc(OC)c3)=O)C)C2)ccc(C)c(C)c1O 91726,C(=O)(C1CCCc2scnc21)N1CCC(N(C(=O)CC2C=CCCC2)CC)CC1 91727,c1(CC(=O)NCCC(C)N(C(=O)C(C)Oc2cccnc2)C)ccc(Cl)s1 91728,C1(Sc2c(C(=O)OCC)c(=O)cc[nH]2)CCC2(CCOCC2)CO1 91729,C1(CNC(CCC(N)=O)=O)CN(C(=O)Cc2cccs2)CC12CC2 91730,c1(CNC(c2cc(C)on2)=O)ccnc(C(N2CCC(C(C)O)C2)=O)c1 91731,C#CCCCC(=O)N1CC(NC(C2(c3cncc(Br)c3)CC2)=O)C(F)C1 91732,Cn1nc2c(c1NC(C13CCC(NC(=O)C(C)(C)C#N)(CC1)CC3)=O)CCC2 91733,S(=O)(=O)(c1cccc(=NCc2c(Br)nnn2C)[nH]1)NCC1CCC(C)(CC)O1 91734,N1(C(c2snc(CC)n2)=O)CC2CCC2(C(=O)OC)C1 91735,Nc1cc(C(N2CC(CNC(=O)Cc3cc(O)nnc3O)C2)=O)cc(O)c1Cl 91736,C1(C(=O)NCC(C)(CO)NC(c2cc(F)n[nH]2)=O)CC2CCCC(C1)C2 91737,C(=O)(C1=CC2(CCOC2)C1)N(CC(=O)NCC1(C)CC2CCC1C2)C(C)C 91738,CC1(C)CCCC(CNC(=O)CC2CCCC(NC(c3scnc3Cl)=O)C2)O1 91739,C1(OC)CCCC(CC(=O)Nc2cccc(C(=O)C(F)(F)F)c2)C1 91740,c1(NC(C2(F)CN(C(CCn3ncc(C)c3)=O)C2)=O)cccc(Cl)c1C 91741,C=C(Br)CC(C)(C)C(=O)NCCC1CCC(NC(c2cnnn2CC)=O)C1 91742,CC(C)(O)C(C)(C)CNC(C1C=CC(NC(=O)CCc2cccnc2)C1)=O 91743,N1(C(CC(C)=C(C)C)=O)CCC2(CC1)CC(CNC(c1ncn(C)n1)=O)C2 91744,C1(OC)(CNC(=NCC2CCCCN2C(C)C)NC2CC2(C)C)CCSCC1 91745,C(=O)(CCCCC(C)CC)NCC(CCC)C(=O)NCc1nn(C)c(=O)n1C 91746,c1(C(=O)NCCOC)ccc(NC(=O)C(=O)N(C2CCCCC2SC)C)cc1 91747,CCCCC(O)C(C)C(=O)N1CCCCC1CC(=O)NC1CC(OC(C)C)C1 91748,c1(C(N2CCC(NC(CNC(C)=O)=O)C(CO)C2)=O)cc2nc(Cl)ccc2o1 91749,C1(CNC(=O)Cc2csc(S)n2)C2CN(C(=O)Cc3nncs3)CC12 91750,C(C)(C)(CC(F)C(=O)NCCC1CCOCC1)NC(C(NOC)=O)=O 91751,c1(C(=O)NCC(C)N(C(c2cccc[n+]2[O-])=O)CC)cnc2c(cnn2C)c1N 91752,N1(C(CCc2n(C)ncc2)=O)CC2CC2C1C(=O)NCc1nc(N(C)C)no1 91753,Cc1nc2ncc(-c3nc(-c4ncnc5c4c(Br)cn5C)no3)c(=O)n2[nH]1 91754,N1(C(c2c(C)n[nH]c2)=O)CCc2nc(O)cc(C(N3CCCC(F)CC3)=O)c2C1 91755,C1(CS(=O)(=O)NC(C2(CC=C)CCCCN2)=O)CCCC2(CCC2)O1 91756,c1(CCC(=O)NCCC2CN(C(C3CC4CCC4C3)=O)CCO2)cccc(O)c1 91757,C(CC(C(=O)N1CC(O)C1)NC(C1C(C)C1C)=O)=CC 91758,c1(C(=O)NC2C(CNC(c3cn(C(C)C)nn3)=O)CCC2)ccc([N+](=O)[O-])[nH]1 91759,C=CCC(C)C(=O)NOCC(=O)NCC1CCCN1C 91760,CC1(NC(=O)C#CC2CC2)CCCN(C(c2csc3nccn23)=O)C1 91761,C12(NC(c3c(SC)cccc3)=O)CCN(C(C34CC(C)(C3)C4)=O)CC1C2 91762,C=CCCC(C)(C)NC(=O)CC1(NC(=O)CC2CCCOCC2)CCC1 91763,CC1(C)C(C(=O)NC(C2CCCCC2)C(N2CCC(F)(F)C2)=O)C1(F)F 91764,S(=O)(=O)(c1ccc(Br)cc1NCc1ccc(-c2nc[nH]n2)cn1)NCCC 91765,N1(C(C(=CC2CCCC2)C)=O)CC2CCOC2(CNC(c2cncc(C)n2)=O)C1 91766,N1(C(C=CCOC)=O)CCOCC(NC(=O)C(F)(F)CN(C)C)C1 91767,Cc1ccc(F)c(CNC(C2CCC(CNC(C3CC4CCC4C3)=O)O2)=O)c1 91768,c1(CC)ccc(C(=O)NCC2(C)CC(NC(=O)C(C)(C)n3cccn3)C2)nc1 91769,CCCC(CCC)C(=O)NC1CC(O)CN(C(=O)C(C2CCOCC2)F)C1 91770,N1(C(C2N(C(c3ccn(C(F)F)n3)=O)CC2)=O)CCC2(SC)CCCC12 91771,C(=O)(C(CC(F)F)C1CCC1)N(CC(CNC(C(=Cc1cccs1)C)=O)O)C 91772,N1(C(C(C)=CC2CC2)=O)CCC(C)(C)C1C(=O)NCc1nc(C(N)=O)no1 91773,CC(C)C(F)C(=O)NC1CCCC(NC(c2cn(CC(=O)OC(C)(C)C)nn2)=O)C1 91774,C1(C(=O)NC2(C(NOCCCOC)=O)CC2C)CC(=O)CCO1 91775,C1(N(C(=O)CC2CSCCS2)CC)CC2CCC(C1)N2C(=O)Cc1ccsc1 91776,N1(C(C2CC(CCNC(=O)COCC3CCC3)C2)=O)CCOCC2(CC2)C1 91777,c1(C(N2CCC(O)(C(=O)OC)CC2)C(=O)NCCOCC)nc(Br)c(C)cc1Cl 91778,C#CCCN=C(NCC(C)Cc1cccs1)NC1CC(CNC(=O)OC(C)(C)C)C1 91779,C1(CC(=O)N(C2CN(C(C3CCN(C4CCCCC4)C3)=O)C2)C)CCCOCC1 91780,Cc1cc(C(=O)O)cc(C)c1NC(=O)C(=O)NC1N(CC(C)O)CCCC1 91781,c1(C(C)C)ccc(C#N)c(NC2CCN(C(c3c(F)ccnc3Cl)=O)CC2C)n1 91782,CCN=c1[nH]c(C)c(C(N2CCCCC2CNC(C2CCNC2=O)=O)=O)s1 91783,c1(C(N2CC(C)N(C(c3cnn4ccsc34)=O)CC2)=O)cccc2ccsc12 91784,CC1CC(CNC(=O)C(F)(F)C2(O)CCC2)CN1C(=O)COc1ccccc1Cl 91785,Cc1cc(=NC(C)CC2CCOC2)[nH]c(=NCc2nnc3n2CCOC3)[nH]1 91786,Cc1ccc(C)c(SCC(=O)NCCCC(C)NC(c2c[nH]c(Br)c2)=O)c1 91787,C1(C(N2CCC(N(C(CN(C(C)=O)C)=O)C)C2)=O)COCCN1C 91788,N1(C(C=C(CCC)C)=O)CCC(NC(c2csc(CC(F)(F)F)n2)=O)CC1C 91789,C=CC(CCC)CC(=O)N1CCN(C(=O)CNC(=O)C(C)(C)C)CC1 91790,n1(CC)cc(Br)c(C(=O)NCC(C)(CO)NC(c2[nH]c(C)nc2C)=O)n1 91791,c1(CC)nc(C)c(C(=O)NCCC2CCC(NC(=O)Cc3cccn3C)C2)s1 91792,N1(C(Cn2ccc(C)n2)=O)CC2CN(C(c3ccc4ncnn4c3)=O)CC2C1 91793,c1(C(=O)NCCCNC(C2CC(O)C(F)C2)=O)cncc2c1CCCC2 91794,c1(C(N2CC(CNC(=O)CC3COC4CC3C4)OCC2)=O)c[nH]cc(Br)c1=O 91795,N1(C(c2nc(COC)sc2)C(=O)NC(C)CC)CC(NC(C)=O)C(C(N)=O)C1 91796,C(CCC(=O)N(CCC)CC=C)OCC1C(NC(COCCOCC#C)=O)C1 91797,Cc1cccc(C=CC(=O)NC2CC(C)(C)C2OCc2ccccc2)c1 91798,C(=O)(C1CC=Cc2ccccc21)NCC(C)(CO)NC(=O)Cn1cccc1 91799,N1(C(C(COC)C)=O)CC(NC(=O)C2=CSCCO2)CC12CCC2 91800,C(=O)(C1=CCCCC1C)N1CC(O)(CN(C(CCCOC)=O)C)C1 91801,C1(CNC(c2c(COC)cco2)=O)CCCN(C(=O)C(F)(F)c2csc(Cl)c2)C1 91802,c1(CN(CCN(C(C(CCCC)ON=C(C)C)=O)C)C)nc(C)cc(C)c1C#N 91803,N1(C(=O)Nc2c(C(=O)NC)n(C)nc2)CCC2NC(=O)NCC2C1 91804,N1(C(C(CC)C(C)(F)F)=O)C2CCCC1CN(C(=O)C(C)(C)S(C)(=O)=O)CC2 91805,C1(CNC(COCCC)=O)CC2COCC2N1C(c1c(F)ccnc1F)=O 91806,c1(C(N2CC3CC2CC3O)C(=O)NCCCC)ccc(C)c(Cl)c1 91807,C(=O)(C(O)C1=CCCCC1)N1CC(NC(CC2CC(CC)OCC2)=O)C1 91808,C1(NC(C2(CC)CCCCC2)=O)CN(C(=O)CC2CCN(C)C2)CC1N=[N+]=[N-] 91809,N1(C(C(C(CC)O)C)=O)CC=C(CCNC(c2ccnn2CC2CC2)=O)CC1 91810,CC1(C)CCN(C(=O)CC2CCC(=O)NC2)C1C(=O)NC1(CF)CCC1 91811,CC(O)(CC(=O)NC1CCCC1C(=O)NCc1cc(F)c(Cl)cc1Cl)CC(=O)O 91812,C(=O)(CC(C(C)CC)NC(C1(CO)CCOC1)=O)NC(C=C)CO 91813,C1(NC(=O)Cc2cccs2)(COC)CCN(C(=O)CSc2ccncc2)CC1 91814,Cn1ncc2ncnc(NCC3CC(C(=O)NCCNS(C)(=O)=O)CO3)c12 91815,c1(C(C(=O)Nc2cccc(OC3CC3)c2)O)cc(F)c(F)c(F)c1 91816,C1(OC)(OC)CCC1C(=O)NC1CCCC1CNC(=O)C(c1ccccc1)OC 91817,c1cc2[nH]c(=NCCCOc3ccncc3)[nH]c(=NCC3CCCS3)c2s1 91818,n1(-c2cn(C)nc2)nccc1S(=O)(=O)Oc1ccc(F)cc1 91819,C1(C(N2CC3CC(NC(CN(C4CCC4)C)=O)C3C2)=O)Cc2ccccc2N1 91820,CC(C)(C)CC(O)CC(=O)N1CC=CC(C(=O)NCc2ccncc2)C1 91821,C1(O)(C(N(CC(C)NC(c2ccc(C(=O)CF)cc2)=O)C)=O)CC(C)(C)C1 91822,CCC(C)(CC)C(=O)NCCC(CNC(c1[nH]ccc1C)=O)OC 91823,CCCC(O)C(CO)NC(c1cnn(CCNC(=O)CSCCC(C)C)c1)=O.C(C)=O 91824,c1(CC(=O)NCCC2CCN(C(C(CSC)OC)=O)C2)ccc(C(C)(C)C)cc1 91825,N1(CC(N2C(CNC(Cc3cc(C)ns3)=O)C=CC2)=O)CCNC(=O)C1 91826,Cc1ccc(C#N)c(NC(C2C3CC2N(S(=O)(=O)c2ccncc2)C3)=O)c1 91827,c1(OC)cc(S(=O)(=O)NC2(CO)CN(C(=O)C(c3ccccc3)C)C2)ccc1Br 91828,Cc1c(F)cccc1S(=O)(=O)N1CC(O)CC1C(=O)NC1CCN(C(C)C)C1 91829,N1(C(COC2CCCC(C)C2)=O)CCN(C(=O)Cc2ccc(F)nc2)CCC1C 91830,n1(CCC(N2C3C(NC(C(C)(C)F)=O)CC(C3)C2)=O)ccc2ccccc12 91831,c1(NC(C2C(NC(c3ccc(C)[nH]c3=O)=O)C2)=O)sc2ccccc2c1C#N 91832,C1(NC(c2cnc(CC)s2)=O)CN(C(c2cc(C)nc(Cl)c2)=O)CCC1C 91833,c1(C2OCCN(C(=O)NCC3(n4ccnn4)CCOCC3)C2)c(Cl)cccc1Cl 91834,C=CC(C)(CC)C(=O)N1CCN(CC(N2CCCN(C(N)=O)CC2)=O)CC1 91835,c1(C(=O)NC2CCN(C(CN(C(C)=O)C)=O)C2(C)C)nn(C)c2c1CCC2 91836,C(=O)(C(O)CC(C)(C)C)N1C2CC(C(N(C3CCCC3)C)=O)C1CC2 91837,N1(C(c2c(C)[nH]c(=N)s2)=O)CCCN(C(C2CC23CCCCC3)=O)CC1 91838,c1(CN2CCC(NS(CCC)(=O)=O)C2)ccc(OC)c(F)c1 91839,N1(C(CC=C)=O)CC(CNC(=O)C(C2CC2)SC)CC12CCC2 91840,c1(OCCOC)cc(C(=O)NC2CCCC2CF)ccn1.c1(C(=O)N)nc(C)no1 91841,C1(C(N(C2(C(N(CC(CC)C)C)=O)CCC2)C2CC2)=O)C2CCC(F)C12 91842,C#CC1CN(C(C2(C=C)CCN(C(=O)CNc3ccccn3)C2)=O)CCN1C 91843,C1(OCC)CC2(C1)CC2C(N1CCC(C(C)NC(c2nocc2C2CC2)=O)C1)=O 91844,C(=O)(C(CC)CCCC)N(C(C1CC=CCC1)C(=O)Nc1cccc(CC)c1)CC 91845,C12(CNC(c3c(C)coc3)=O)CCC(CC1)N2C(c1cc2scnc2[nH]1)=O 91846,C=Cn1cc(C(c2nnnn2Cc2ccccc2OCC)NC2CC2CF)cn1 91847,C1(OC)CC2CC1CN(C(=O)CC1(N(C)C(c3cnncc3C)=O)CC1)C2 91848,c1(C(N2CC(OCCNC(CCC3CCC(C)O3)=O)C2)=O)cccc(Cl)c1 91849,C(C(C)N=c1[nH]c(=NC2CC(CO)C2)[nH]c2c1CC(C)CC2)OC 91850,c1(NCC(CC(=O)NC)C)[nH]c(=NC(C)c2nncs2)nc2ncn(C)c12 91851,c1(CC(=O)NCC(C)N(C)C(C2CN3CCC2CC3)=O)ccc(Br)cc1F 91852,c1(C(CNC(c2cnnn2C2CC2)=O)NC(C2CCCCC2)=O)ccccc1F 91853,C1(NC(C2C(C)C2)=O)CN(Cc2cc(Cl)cc(Cl)n2)CC1C#N 91854,C(=O)(C(C)(C)C(=O)N1CC(N(C)C(C2C3CN(C)CC23)=O)C(F)C1)OCC 91855,c1(C(=O)NCC(CC=C)NC(=O)C(C)(C2CC2)OC)n[nH]c(C)c1[N+](=O)[O-] 91856,Cc1cc(O)ncc1C(=O)N(C1CCCN(C(=O)Cc2ccc(O)c(Cl)c2)C1)C 91857,C1(C(N2CCC(NC(c3c(OC)nccc3)=O)C2)=O)CC12CCCCC2 91858,N1(C(c2cc(C)sc2)=O)C2CCC1CN(C(=O)CN1CCC(N(C)C)CC1)C2 91859,N1(C(CC(=C)C)=O)CCC2(C1)CN(C(c1ccnn1C(F)F)=O)C2 91860,Cc1nsc2ncc(C(N3CCCC4(C3)CN(C(C3CCCOC3)=O)C4)=O)cc12 91861,c1(CC)ccc(C(=O)N(CC(C)NC(=O)COCCCC(C)C)C)c(OC)c1 91862,CC1CCC(C)(C(=O)NC2CC(CNC(c3cnc(S)[nH]3)=O)C2)C1 91863,c1(NC(C2CC(O)CN2Cc2ccc(Br)nc2)=O)c(F)cc(F)cc1[N+](=O)[O-] 91864,c1(-c2cn(C3CC(C)(O)C3)nn2)ccc(N)cc1 91865,c1(C(=O)NC(CNC(c2cc(OC)nn2C)=O)C(C)C)sc2cccnc2c1Cl 91866,C(CC(=O)NC12CC1CN(C(c1nc(Cl)sc1C)=O)C2)(C(C)C)OCC 91867,C(CCCCCn1cc(CC2CC(O)CN2CCO)nn1)NC(C1CCOC1)=O 91868,c1(C(N2C(CC)CN(C(=O)CC3=CCCCC3)CC2)=O)cc2cc(Cl)cnc2[nH]1 91869,c1(CC)ncncc1C(N1CCC(CNC(C23COC(CC)(C2)C3)=O)C1)=O 91870,c1(C(c2nnnn2C(C)C)NCC(CC=C)(C)C)c(F)cnc(Cl)c1C 91871,N1(C(c2cc(C)[nH]c2)=O)CC23CCCC2(C1)CN(C(=O)CCc1ncccn1)C3 91872,CN1CCc2cc(C(=O)N(C3CC(NC(C4CCCC(C#N)C4)=O)C3)C)ccc21 91873,c1(C(=O)NC(CC)(C)CNC(C2CCC(=O)N2C(C)C)=O)csc2cncn12 91874,C(N=c1[nH]c2cc(Br)ccc2o1)C1C(C)CN(C(C2CCOC2)=O)C1 91875,c1(NCc2ccc(C)cc2)ncnc(N2CCC(O)C(F)C2)c1C 91876,N1(C(c2c(C)cc(Cl)cc2)=O)CCCC(C2CCN(C(=O)C(O)C(C)C)CC2)C1 91877,N1(C(c2ccc(CO)s2)=O)CC2CCC(C1)N(C(c1scnc1C(F)(F)F)=O)C2 91878,c1(C(N(CC(c2ccccc2)CC)CC)=O)ccc(C(F)(F)F)s1 91879,N1(C(CC(C)O)=O)CCOCC1C(=O)NC(C)(CO)CCF 91880,CCC(C(=O)N1CC(C)C(C)(C(=O)NCC=Cc2cccnc2)C1)C(F)(F)F 91881,C1(NC(C2C(CCOC)C2)=O)CC2(C1)CN(C(c1cc([N+](=O)[O-])c[nH]1)=O)C2 91882,C1(NC(c2cc(C)[nH]n2)=O)CC(O)CN(C(=O)CC2(c3ccccc3)CC2)C1 91883,c1(NCCOCC=C)cc(=NC2CCOc3ccccc3C2)[nH]c(COC)n1 91884,C1(CCNC(C(C)C2CC2)=O)CCC(NC(=O)CN2CCOC2=O)C1 91885,c1(C(C)NC(=O)NC2C(c3n(CC)ccn3)OCC2)c(Cl)ccc(F)c1Cl 91886,c1(OC)c(C(=O)NCC(C)N(C(=O)COC2CCOC2)C)cc(Br)cc1F 91887,CN1CCOCC1CC(=O)NC12CC1CN(C(c1cn(-c3ccccc3)cn1)=O)C2 91888,C1(CCOCCN(C(COC2CN(C(C)=O)C2)=O)C)CC(F)(NC=O)C1 91889,c1(C(=O)NC(CCNC(c2cc(C(C)C)no2)=O)(C)C)cc2c(ccn2C)[nH]1 91890,C1(C(N2CCCC(N(C(Cc3c(C)cco3)=O)CCF)C2)=O)CCCCC1(F)F 91891,C1(C(=O)NCC(CC)(C)Cl)COCCN1C(c1cc(=O)cc[nH]1)=O 91892,C=CCC(C)(C)CC(=O)N1CC=CC1CNC(c1ncnc(C)c1C)=O 91893,C1(NC(CCOCCN(C)C)=O)CN(C(=O)C=CC2CCOCC2)CC2CC12 91894,N1(C(=O)CN2CCN(C)CC2)CCN(C(=O)N)CC1.C12(CC1)C(=O)N2C.COC 91895,CC1=NOC2(C1)CC(C(N1CC(NC(C3CCS(=O)CC3)=O)C(C(F)F)C1)=O)C2 91896,C1(C(=O)NC(C(C)C)C2CCC2)(CC)CCN(C(c2c[nH]nc2Cl)=O)CC1 91897,N1(C(C(CCC)O)=O)CC2(C1)SCCC2NC(=O)CCc1cncc(OC)c1 91898,c1(CNC(C2CC(CCNc3cc(OC)ncn3)C2)=O)ccc(C)c(Cl)c1F 91899,C1(NC(C2(CC#C)CCCC2)=O)CCC(C)(NC(c2cc(Cl)ncc2O)=O)CC1 91900,Cc1noc(C)c1CCC(=O)NC1(C)CC(NC(C2CC23CC3(F)F)=O)C1 91901,N1(C(CC2CCN(C(=O)OC(C)C)CC2)=O)CCC2(CC1)OCCc1ccccc12 91902,c1(NC(CCC)CCCNC(=O)CCC(N)=O)ccc(S(C)(=O)=O)cc1[N+](=O)[O-] 91903,C1(N(C(C2CC2OC(C)=O)=O)C(c2sccc2C(C)(C)C)=O)CCc2ccnn2C1 91904,Cc1ccc2[nH]c(C(N3CC(O)(C(C)(C)CNC(=O)C#CC4CC4)C3)=O)cc2c1 91905,n1(CC)cc(Br)c(C(=O)N(C)CCN(C)C(C2CCS(=O)(=O)N2)=O)n1 91906,C1(c2n(CC=C)nnn2)(OCC2(CNCC)CCCCO2)CCCCCCCC1 91907,CC(C)CC(C(=O)N(C(C)(C)C)C)ONC(=O)C1CC(N2CCC2)C1 91908,C1(F)(C(=O)OCC)CN(C(=O)Oc2cccc(C#N)c2)CC12CCOCC2 91909,O=C1NCC2(CO1)COC(CF)CN2C(C1C2CC=CCC12)C(=O)OC 91910,C1(NC(C2CCCNS2(=O)=O)=O)CCN(C(C2CCCSC2)=O)CC12CCC2 91911,CC(C(F)C(=O)N1CCC(NC(C2(CC3CCC3)CC2)=O)C(O)C1)C(F)(F)F 91912,C=CCC(CNC(C1CCCO1)=O)NC(c1cc(COc2ccccc2)on1)=O 91913,C1(NC(COCCCC)=O)CN(C(=O)CC2CC2CC)CCC1OC 91914,c1(C(N(CC(O)CNC(=O)CNS(C)(=O)=O)C)=O)c[nH]cc1Br 91915,c1(NC(N2CCC(n3cc(CO)nn3)C2)=O)cc(Cl)cc2nccnc12 91916,N1(C(c2cc(F)cc(F)c2Br)C(=O)NCC)CCc2nc(C)n(C)c2C1 91917,N1(C(C2(CCC)CCC2)=O)CCC2C(C(=O)NCC(F)(CC)CC)C2C1 91918,CCCCCCCC(O)C(F)(F)C(=O)NCCN(C(=O)CC1CCCCCC1)C 91919,c1(N2CC(C)(COC)OCC2)ccc(S(=O)(=O)NC2CCCCCC2F)cc1Br 91920,C12=C(Cl)N=CNC1=NCCN1CCN2CC(OC)C1c1cnn2cccc2c1.CO 91921,c1(C2(F)CC(C(=O)NC(C)CCN(C)C(C3CC3C)=O)C2)cccc(F)c1 91922,Cc1cccc(C(N2CCC(C(N3CCCCC(C)(F)C3)=O)CC2C)=O)c1C#N 91923,N1(C(C(CSC)O)=O)CCC2(C1)CN(C(c1n[nH]c3c1CSCC3)=O)CCO2 91924,C(=O)(C(C)(C)CCC(C)=O)NCc1c(OC)ccc(F)c1 91925,c1(OC)cccc2cc(C(=O)NC3CCN(C(=O)C(F)=C(C)C)C3)oc12 91926,C1(CN(C(CNC(=O)OC)=O)C)CCN(C(=O)CC2CC2(Cl)Cl)CC1 91927,N1(C(COCCCC)=O)CC(C)CCC1CNC(=O)C=Cc1ccnn1C 91928,c1(C(=O)NC(C(C)C)CNC(=O)C(c2ccnn2C)O)ccnc(C2CC2)n1 91929,c1(OC)cccc(C)c1NC(C1(CNC(c2cccn2C)=O)CCCO1)=O 91930,C1(C(=O)NC2C=CC(C(=O)NC)C2)(CC)CCN(C(c2ccn(CCF)n2)=O)C1 91931,CC1CN(C(c2cc[nH]n2)=O)CC1NC(c1ccc(-c2ncon2)cc1)=O 91932,c1(C(=O)NC(C(=O)NC2(C)CC(O)(CO)C2)C2CC2)cccc2occc12 91933,C(=O)(C(=O)CC(C)C)NC(C(=O)NCC(CC)C#N)(C)CO 91934,C12(C(CNC(=O)C(Cl)=CCl)NC(=O)CNC(c3ncc[nH]3)=O)CCC(CC1)C2 91935,N1(C(C=CC=CCCCCC)=O)CCCC(N(C(c2cc(C)sc2C)=O)CC)C1 91936,C1(CC(=O)NCCOC(C)=O)CCCN(C(=O)Cc2cn(C)nn2)C1 91937,c1(C(=O)NC(C)Cn2cc(COC(=N)O)nn2)coc2ccc(Br)cc12 91938,Cc1cc(NC(C2CC(C)(C)CN2C(c2cccc(CC#N)c2)=O)=O)cnc1Cl 91939,c1(C(N2CCC3(CC(NC(c4occ(C)c4)=O)C3)C2)=O)ccc(C)c2c1CCC2 91940,c1(C(C)NC(C2(F)CN(C(C3CCC(CC)O3)=O)C2)=O)c(C)noc1C 91941,C1(C(=O)NCCC(CNC(=O)C(C)(C)n2cncn2)OC)CCc2c[nH]nc2C1 91942,C1(C(=O)NCC(C(=O)OC)OC)CCCN(C(=O)C(OC)OC)CC1 91943,N1(C(C)=O)CCCC(O)(C(=O)NC(C)(CNC(=O)CCn2cccc2)C(C)C)C1 91944,N1(C(C2N(CCCC)CCCC2)=O)CCCCC(NC(C2(CC(C)C)CC2)=O)C1 91945,C(=O)(C(C(C)(F)F)NC(=O)CCc1ccc(F)c(CN)c1)OC 91946,c1(C(C)C)ccc(CC(=O)NCCCNC(=O)C(C)Cc2ccc(Cl)cc2)cc1 91947,C1(NC(C2(C)CC(C)C2)=O)CN(C(C2C=CCS2)=O)C2(CCCC2)C1 91948,c1(C(=O)NCC(C)CO)c(Cl)nn(C)c1Cl 91949,c1(CC)cc(C(=O)NCC(N2CCN(C(=O)C(O)COC)CC2)C)ccc1F 91950,C(=O)(C(C)NC(C)=O)N(C1CCCC1)CCNC(CSCC#C)=O 91951,CCC1=NOC(CC(=O)NC(C2CCN(C(C3C(Cl)(Cl)C34CC4)=O)C2)(C)C)C1 91952,c1(C(C)C)ccc(N2CC(C(N3CCCC(CNC(=O)CO)C3)=O)CC2=O)cc1 91953,c1(C(=O)NC2CN(C(C(COCC)C)=O)CC2N=[N+]=[N-])cnc2c(c1)ncn2C 91954,Nc1cccc(C(=O)NCC2CCC2NC(c2ccnnc2O)=O)n1 91955,c1(NC(CC2N(C(C=CCOC)=O)CCC2)=O)c(Cl)nc(Cl)nc1Cl 91956,Cc1ccc(C(CNC(=O)CC(C)(F)F)NC(c2ccn(C3CC3)n2)=O)cc1 91957,C1(CN(CCCNC(c2c(C)onc2)=O)C2CC2)CCC(C)(C)CC1 91958,N1(C(C=Cc2ccc(OC(C)C)cc2)=O)CCN(C(=O)CCCF)CCC1C 91959,C1(C(N2CCCC(C(C)C(=O)NCc3cc(Cl)no3)C2)=O)CN(C)CCN1C 91960,C(CCCCC(=O)NCC(O)C(F)(F)F)NC(c1c(C)snn1)=O 91961,C1(C(N2CCC(O)(CN(C(CCCC(=C)C)=O)C)C2)=O)Cc2ccc(F)cc2O1 91962,CC(C)C(C(=O)N1CCCC1CNC(c1ccc(-c2cnn[nH]2)cc1)=O)C(C)C 91963,c1(C(N2CC(C)C(CNC(=O)C(C)C(C)(C)O)C2)=O)ccc(F)c(F)c1 91964,N1(C(C(=O)NC2CCCN(c3cc(O)ncn3)C2)=O)CCOC2(CCCC2)C1 91965,N1(C(C(CC=C)C(C)C)=O)CC2N(C(=O)C(C)C3CCC3)CCC2(C)C1 91966,n1(Cc2cn(CC3N(CCS(C)=O)CCC3)nn2)nc(Cl)c(C#N)c1N 91967,Cc1ccc2cc(C(=O)NCCCNC(=O)C(F)C3CC3)c(C)nc2c1 91968,N12CCN(C3CC13)C(=O)C=CC2=O.c1(OCc2cccnc2)ccc(F)cc1 91969,C#Cc1cccc(C(=O)NCc2cccc(CNC(C3CCCC3C)=O)c2)c1F 91970,C(=O)(CC(C)C(C)C)NC1(C(=O)NCc2ncc(CC)s2)CCCCC1 91971,Cn1cc(C#N)cc1C(=O)NC(CC1CCOCC1)C(=O)NCc1nnc(O)o1 91972,C1(CNC(CCN(C(C)C)C(C2CC3CC(=O)C2O3)=O)=O)CCCC2(CC2)C1 91973,CC(C(=O)NCC(O)CNC(c1cncc(F)c1)=O)C(=O)N1CCOCC1 91974,N1(C(CCOC(CC(C)C)C)=O)CCCC1(C)CNC(C1CN(C)C(=O)N1)=O 91975,c1(C(N2CCCCC2CC(F)(F)F)C(=O)NCCC)ccc(C2CCCC2)cc1 91976,c1(CC(=O)NCC(CC)NC(C2(OC)CC2)=O)c(C)nc(C)nc1O 91977,c1(C(N2CC3CCCCC3C2)=O)ccc2c(-c3ccc(CO)o3)cccc2n1 91978,C1(C(=O)NC(CN(C(=O)C(C)SC(F)(F)F)CC)C)CC2CCC(C1)S2(=O)=O 91979,N1(C(C2CC(CCC)C2)=O)CCOCC(NC(c2cccc(O)c2Cl)=O)C1 91980,C12(NC(C3CN(C)C3)=O)CCCN(C(=O)Cc3cc(F)cc(Cl)c3)CC1C2 91981,n1(CC)ncn(NC(=O)C(CCNC(=O)CNC(=O)C(C)CC)C2CCC2)c1=O 91982,c1(C(=O)NCC(CNC(c2c(C)nc(O)[nH]2)=O)(C)O)ccc2ccccc2n1 91983,c1(C(N2CCC(CNC(C3(C=C)CCCCC3)=O)C2)=O)nnn2ccccc12 91984,C(CC(C)P(C)(C)=O)C(=O)NC(c1nccc(=N)[nH]1)C 91985,C#CC1(F)CN(C(c2ccoc2CNC(C2CC2(C)C(F)F)=O)=O)C1 91986,Cc1c(NCC2(C)CCCCO2)ncnc1N1CCC(C(O)C(N)=O)CC1 91987,CC1C(C)N(C(=O)Cc2cnccn2)CCN1C(c1cnc(F)c(F)c1)=O 91988,N1(CC(=O)N(c2nc(-c3ccc(Br)cc3)cs2)C)CCOC(C#N)C1 91989,C=C(C)C1OCCC1C(=O)NC(C)(C)C=CC(=O)NCC12CCC(CO1)C2 91990,N1(C(CCC(C)OC)=O)CCC(C2(NC(c3ccccc3C#N)=O)CCC2)CC1 91991,C(CNC(=O)CC(=O)Nc1nccs1)(CC(=O)NCC1(C)CC(C)C1)OC 91992,c1(C(=O)NCC2CCCN(C(CCC)=O)CC2)cc(S(=O)(=O)NC)cs1 91993,c1(C(=O)NC2C(OC)CN(C(c3c(OC)ccnc3)=O)C2)cc2n(n1)CCO2 91994,C1(C)(C(=O)NCCCCN(C(C(CC)NC(C)=O)=O)C)CCCCC1 91995,C1(CNC(CN(CC(=O)NC(C)C)C)=O)CCCN(C(C2CC(N(C)C)C2)=O)C1 91996,C1(NC(=O)C(F)C2CCOC2)(CNC(C23CCC(C2)C3)=O)CCCC1 91997,C1(C(C)NC(=O)CC2CC3(CCO2)CC3)CCC2CN(C(c3ccsn3)=O)CC12 91998,S(=O)(=O)(CCCN=c1nc2scnc2c(NCCC2(CSCC)CC2)[nH]1)NCC 91999,C1(C(N2CCCC(N(C(=O)CC3CCCS3(=O)=O)C)C2)=O)CCCCC1(F)F 92000,c1(C(=O)NCC2(CNC(c3ccc(C)cc3O)=O)CCC2)cc2cn[nH]c2cn1 92001,c1(C(=O)NC2C(C)CN(C(=O)C(O)C3CCCC3)C2)cc2ccc(F)cc2[nH]1 92002,c1(CN2CCC(C(=O)Nc3n(C)cc(Br)n3)CC2)ccn2ccnc2c1 92003,N1(C(c2c(CCC)n(CC)nn2)=O)CCN(C(C2CSC2)=O)C(CC(C)(C)C)C1 92004,Cc1cnc(N(C2CCNCC2F)C(c2ncccc2C)=O)nc1 92005,C1(C(=O)NCCOCCSC)(C2CC2)CCCN1C(=O)C(C)NC=O 92006,N1(C(CC(CN(C)C)(C)C)=O)CCN(C(=O)CCOCC2CCCO2)C2CCCC12 92007,c1(CCCC(=O)NCC2(F)CCC(NC(C3CC3(F)F)=O)C2)cc(Cl)ccc1Cl 92008,N1(C(C2(COC)CC2)=O)CCC2(CC2C(N2CC(C#N)(COC)C2)=O)C1 92009,c1(C(=O)NCCCNC(C2(S(N)(=O)=O)CC2)=O)ccc(=O)n(CC2CCCO2)n1 92010,C1(NC(c2cc(COC)on2)=O)CCCN(CC(O)Cn2nc(C)nc2C)C1C 92011,Nc1nn2ccccc2c1C(=O)NC1CCC(F)(F)C1O 92012,C1(C)(CC)CC(C(=O)NCc2cc(C(=O)NC(C)Cc3cnccn3)no2)C1 92013,C(=O)(CC(C)CC(C)(C)C)NC(CC1CC2N(C(CC=CC=C)=O)C(CC2)C1)C 92014,c1(CC(=O)NCC2=CCN(C(COC(C)=O)=O)CC2)c(C)[nH]c2ccnn2c1=O 92015,CN1CCC(CNC(C2CC(C)(NC(=O)C(C3CCCCC3)=O)C2)=O)C1 92016,Cc1cc(N)c(F)c(C(N2CCCC(F)(CNC(C3(O)CC3)=O)C2)=O)c1F 92017,C1(C#N)(C(=O)NCC(CNC(C(C)=C(CC)C)=O)OC)CCCC(=O)C1 92018,C1(NC(c2c(Cl)cc(C)s2)=O)COC2CN(C(=O)CCNS(C)(=O)=O)CC12 92019,c1(C(=O)NCC2(C)CC(NC(C(C3CCCCO3)OC)=O)C2)ccc(Cl)cc1 92020,C(c1ccc(F)c(F)c1)=CC(=O)NC(C)CCCNC(C1CCC1C)=O 92021,C1(NC(C=Cc2c(C)cccn2)=O)CCN(C(=O)CSC(F)F)CCC1CO 92022,C12(NC(C3CCC(C(N)=O)CC3)=O)CCC1CN(C(=O)CC1CCCS1(=O)=O)C2 92023,Cc1cc(=O)n(CCC(N2CC(NC(c3cn(C4CC4)nn3)=O)C(O)C2)=O)cn1 92024,Cc1ccc(C(N2CCN(C(=O)C(C)n3cncn3)CC2C2CCC2)=O)c(N)n1 92025,c1(C(N2CC(OCCNC(CCCCOC)=O)C2)=O)ccnc2c1nnn2C 92026,C(c1csc(Br)c1)=CC(=O)NC1CCCC(NC(=O)CC2CCC2)C1 92027,N1(C(C2(C)CCCCC2)=O)CC(CO)C2(C1)CN(C(c1ccc(C#N)o1)=O)C2 92028,c1(C(C)C)cc(C(N2CCN(C(=O)C=CCF)CC2CO)=O)cc(O)n1 92029,c1(C(=O)NCCN(C(=O)C(C2CCCCCC2)C)CC)cncc(C2CC2)c1 92030,c1(C(=O)NCc2[nH]nc(C(C)(C)O)n2)ncn2c1COc1ccccc1-2 92031,c1(C(=O)O)ccc(CC(=O)OCc2nccn2Cc2ccccc2)cc1Cl 92032,CC1CC(NC(C2(C(F)(F)F)CC(F)(F)C2)=O)CN1C(c1cncc(O)c1)=O 92033,N1(C(CC2CC(OCC)C2)=O)CCN(C(=O)C=Cc2nccs2)CC1C1CC1 92034,C(=O)(C1=CCC(C)(C)CC1)N(CCN(C(c1ccc(OC)cc1Cl)=O)C)C 92035,CC1C2CC(C2NC(=O)CN2CCOCC2)N1C(c1cccc(O)c1F)=O 92036,C1(C(=O)NC2(CCNC(CCc3onc(COC)n3)=O)CCC2)OC2CCC1C2 92037,N1(C(c2cc(OCC)n[nH]2)=O)CCN(C2CN(C(c3cn(C)c(O)n3)=O)C2)CC1 92038,Cc1nc(N(C)C)sc1C(N1CCCC1C1CCCN(C(C2CCCC2)=O)C1)=O 92039,N1(C(c2cc(-c3ccc(C)o3)[nH]n2)=O)CCCC1(C)CNC(c1cncs1)=O 92040,Cc1cc(C(N2CCCC2CNC(C2CCCC(N(C)C)C2)=O)=O)ncc1F 92041,c1(C(N2CC(Cc3cn(CCC(C)=O)nn3)OCC2)=O)cc2sccc2cn1 92042,CC1COCC(CSCC2CCC(C3CC3)O2)O1 92043,c1(C(=O)NCC(CC)NC(c2cnc(OCC)s2)=O)noc(C)c1[N+](=O)[O-] 92044,N1(C(C#CC(C)C)=O)CC(C(=O)NC2CCCN(c3ncccn3)C2)C(C)(C)C1 92045,N1(C(C2(COC)C=CCN2C(=O)CCc2cncs2)=O)CC2(CCOC(=O)N2)C1 92046,N#CC1CN(C(c2cc(O)ccc2Br)=O)CCN1C(c1ccsn1)=O 92047,C1(C2CCCN(C(=O)CCN3CCC3)C2)(NC(C2C(C(C)(F)F)C2)=O)CC1 92048,N1(C(c2c(C)nc(C)[nH]2)=O)CC2CCN(C(c3c[nH]cc3C(C)(C)C)=O)CC2C1 92049,c1(SC)cncc(C(=O)N(C(C)CNC(=O)CCc2ccc(C(C)C)cc2)C)c1 92050,CC(C(=O)N1CC(OCC(F)F)C1)C(C)NC(=O)CC1(O)CCCC1 92051,CC1(C)CC(NC(C2(CO)CCCCC2)=O)CN(C(c2ncc(F)cc2N)=O)C1 92052,N1(C(c2n(C)nc(Cl)c2)=O)CCC=C(C(=O)N2CCCCC2)C1 92053,c1(C(=O)NCC(C)NC(c2cc3n(n2)CCCC3)=O)cc2nc(Cl)ccc2s1 92054,C12(C(=O)NCC3CCCOC3)CCC(C(=O)Nc3cc4ccoc4s3)(CC1)C2 92055,c1(CNC(C2(C3CCCN3C(C3CCCS3)=O)CC2)=O)ccc(O)nn1 92056,C1(CS(=O)(=O)OC)CN(N2CC(O)(CC#N)C2)CC1C(F)F 92057,C1(NC(CCCNC(C=Cc2ncn(C)c2)=O)=O)CC2(CCOC2)C1 92058,N1(CC)CC(C(=O)NC2CN(C(c3ccccc3C(F)(F)F)=O)CC2C)CC1=O 92059,N1(C(C2(COC)CC(F)(F)C2)=O)CC(CNC(C2(F)CC=CC2)=O)C(F)(F)C1 92060,N1(C(COCCC(=O)OC)=O)CCc2ccccc2C(NC(=O)C(C)(F)F)C1 92061,c1(C(=O)NC(COC)C)cnn2cccc(-c3c[nH]c4ncccc34)c12 92062,C=CCC(CC=C)c1nc(-c2cccc(F)c2)nn1CCCc1ccccc1 92063,Cc1nc(C(N2C(C(=O)NCC(O)CF)CC3CC23)=O)cc(O)n1 92064,C1(C)(CNC(C=C(C)C(C)C)=O)CCN(C(C2(C)CC2(Cl)Cl)=O)C1 92065,C(=O)(CCc1nccs1)NCCN(C(CNC(C)=O)=O)C 92066,C1(C(=O)Nc2cn(CC(C)C)nc2)CN(C(c2ccc(C(F)F)o2)=O)CCN1C 92067,C(=O)(C(O)(C(F)(F)F)C1CC1)NCC1CN(C(c2c(SC)cccn2)=O)C1 92068,Cn1cc2ccc(NC(C3CC34CCN(C(=O)CCC3CCC3)CC4)=O)cc2n1 92069,c1(NC(C(C)OC(c2cncc(C(F)(F)F)c2)=O)=O)c[nH]c2ccc(F)cc12 92070,c1(OC)ccc2ncccc2c1C(N1CCC(O)(CNC(=O)C(C)(F)F)CC1)=O 92071,CC1CCC(CNS(=O)(=O)c2ccccc2OC(F)(F)F)Cc2ccccc21 92072,c1(C2(C(=O)NCC3(F)CC(NC(c4c[nH]cc4Br)=O)C3)CC2)ccc(Cl)nc1 92073,N1(C(CCc2ccc(C)cc2)=O)CC(N(C)C(c2ccnnc2O)=O)C2(CC2)C1 92074,C(=O)(C1=COCCO1)NCC(C(C)C)NC(C(CC=CC)C)=O 92075,C(N=c1ccc(C#N)n[nH]1)C1N(C(=O)Oc2c(C)ccc(OC(F)F)c2)CCC1 92076,C1(CN(C(C2(CC)CC2)=O)C)CCCCN1C(c1cncc(N)c1)=O 92077,C1(NC(CSCC=C)=O)CC(C(=O)N(C)CC2CC(F)(F)C2)CC1O 92078,N1(C(C(C)SCC)=O)CCC(C(O)CNC(=O)CC2(N(C)C)CC2)CC1 92079,Cc1nc(O)nc(C)c1C(=O)NC1CC(NC(=O)COc2cccc(F)c2F)C1 92080,CCC(CCOC)C(=O)N1CCSCC1CCNC(c1cnccc1C)=O 92081,CC1CC=C(C(=O)NC(C(=O)NC2CC2(C)C(F)F)C(C)(C)O)CC1 92082,C1(NC(C2CCN(C)CC2)=O)C2CC3CN(C(=O)CC4CSCCS4)C1C3C2 92083,C1(C(=O)NC(CC)(C)C)CCCN(C(c2cnncc2C)=O)C1 92084,Cc1cccc(C2(C(N3CCC(CC(=O)N(C)C)C3)=O)CC2)c1 92085,c1(C(C)=O)ccc(Br)cc1NC(C1CCN(C(c2cc(C)n(C)n2)=O)CC1O)=O 92086,c1(C(N2C(C)(C)C(NC(c3nc(Cl)c(Cl)s3)=O)CC2)=O)cn2c(n1)CCCC2 92087,CC1(C)CN(C(=O)COCc2cccc(Cl)c2)CCC1NC(C1CC12CCC2)=O 92088,CCC(F)(F)C(=O)NCC1(OC)CN(C(C2CC2(Cl)C(=O)OCC)=O)C1 92089,c1(C(=O)NCC2(CNC(C(C(=C)Cl)(C)C)=O)CC23CCC3)nnn2c1CCCC2 92090,c1(C(N2CCC(N(C(CN(c3ccccc3)C)=O)C)C2)=O)cc(O)c(F)cc1N 92091,c1(C(=O)NC23C(CN(C(c4cc(OC)ns4)=O)C2)C3)c(C)cccc1C 92092,C(CC1c2ccccc2CCN1C(c1cc(C)cs1)=O)NC(COCCSC)=O 92093,CN=c1ccc(C(=O)NCCC2CN(C(=O)CN(C)S(N)(=O)=O)C2)c[nH]1 92094,C(C(C)CC(F)(F)F)NC(C(=O)N(C(c1ccc(C)cc1)c1cnn(C)c1)C)=O 92095,CON(CC1CC1)C(=O)CC(C(F)F)NC(c1cnnn1C1CC1)=O 92096,N1(C(C(CSC)OC)=O)CCC(C(=O)NCC2CCSC2)=C(F)C1 92097,CCCC(C)(CC)C(=O)NCCN1CCCN(C(C2CC3(CC(OC)C3)C2)=O)CC1 92098,N1(C(CCCCOC)=O)CC2CN(C(=O)CC(C)(C(F)F)N(C)C)CCC12 92099,c1(C(N(C)CC2(NC(C(CCOC)C)=O)CC2)=O)ccc(Cl)c2occc12 92100,C(CO)(C(=O)NCC1CCC(CNC(=O)CCN(c2ccccc2)C)C1)N(C)C 92101,C1(CC#C)CCN(C(c2cn(C(C)C)nc2Br)C(=O)NC2COC2)CC1 92102,c1(CCC(=O)NCC2C(NC(CC3C(C)(C)C3)=O)C2)c(F)cccc1F 92103,c1(C(N2CC(CC=C)(NC(c3cc(Cl)c(C)cn3)=O)C2)=O)ccc(C)c(F)c1N 92104,c1(C2(C(=O)NC(CNC(C(COCCOC)F)=O)C(C)C)CC2)ccnc(Cl)c1 92105,Cc1cccc2c(C(=O)NCC(CC(F)(F)F)NC(C3CC3F)=O)nccc12 92106,c1(CNC(C2(CCC(=O)O)CC2)=O)cc(O)nc(NC(C2(CCN(C)C)CC2)=O)n1 92107,N1(C(C(CC#C)CC#C)=O)CC(C)OC2(CCN(C(=O)C(C)(C)C#C)C2)C1 92108,C1(C(=O)NCC(CN(C)C(C2(C(F)(F)F)CCC2)=O)O)CC(C)(F)C1 92109,C1(CCNC(C2(C)CC2)=O)CN(C(C2CC(Cc3ccccc3)=NO2)=O)CCO1 92110,C1(C)(CC)CC(NC(C2(CO)COC2)=O)CN1C(c1cc(OC)cc(Cl)c1)=O 92111,C1(C)(C(N(CC(CNC(c2n(CC)ncc2)=O)(C)C)C)=O)CC(C)OC(C)C1 92112,c1(CC)nnc(C)cc1C(N1CCN(C(=O)CCNCCCCOC)CC1C)=O 92113,c1(C(=O)NC2CCCCN(C(c3cc(C)nnc3)=O)C2)ccc2c(C)[nH]nc2c1 92114,C(=O)(C(C(C)(C)OC)c1ccccc1)NC(CC)C(F)F 92115,CC(C)CC(O)C(C)C(=O)NCn1ccc(C(=O)NCCC2CC2)c1 92116,CCC(Cc1ccccc1)CC(=O)NC1CN(C(=O)CS(C)(=O)=O)C(C)(C)C1 92117,C1(NC(COCCC)=O)CC(NC(C2CC2[N+](=O)[O-])=O)C(O)C1 92118,C(=O)(C1=CCCOC1)NC(C(=O)NCc1c(C)scc1)CC1CCC1 92119,c1(OCC(=O)NCC(C)(O)CNc2cc(SC)ncc2)cc(C)cc(C)c1 92120,C(CCCC(C)NC(=O)C(C)Oc1ccccc1)NC(C1(COC)CCCC1)=O 92121,c1(OCC)ccc(C(=O)NC2CCC(NC(=O)CS(C)(=O)=O)CC2)cc1 92122,C(=O)(C1CCc2c(Cl)cccc21)NCC1(C(F)F)CCN(C(C=COCC)=O)C1 92123,c1(CNC(C2(C)CCN2C(C2CCO2)=O)=O)cncc(O)c1 92124,C#CC1(C(=O)NCc2cccs2)CN(C(C2CCSC(C)C2)=O)C1 92125,C1(C)(C(N2CC(OC)(CNC(=O)CNC(c3ccncc3)=O)C2)=O)CCCCC1 92126,c1(C(N(CCC(C)NC(C2CCOC2)=O)C)=O)cn(C(F)(F)F)cn1 92127,c1(C(=O)NCC2CCCN2C(C2CC2[N+](=O)[O-])=O)cnc2ccc(Cl)cn2c1=O 92128,Cc1csc2ccc(C(=O)NC3CC(CNC(C4CC5CC4C5)=O)C3)cc12 92129,c1(SCC)cc(CNC(c2ccc(C(N3CCN(C(C)=O)CC3)=O)s2)=O)ccn1 92130,C1(N(C(CN2C(C)CC2)=O)C)CCCN(C(c2sccc2CO)=O)CC1 92131,Cn1nc2c(c1C(=O)NC1CCN(C(C3CCC3F)=O)CC1)CS(=O)(=O)CC2 92132,C1(CNC(c2cc(F)cc(F)c2Br)=O)CCN(C(c2cn[nH]c2)=O)CC1(F)F 92133,N1(C(C2C(=C)CC2)=O)CC(=O)Nc2ccc(C(F)(F)F)cc21 92134,N1(C(CC(C=C)CC)=O)CC2CCC1C(CNC(=O)C=Cc1csc(C)n1)C2 92135,CC1(CCNC(C2(C#N)CC3CC3C2)=O)CCN(C(=O)COC(F)F)CC1 92136,N1(C(c2ccc(C)c(C)c2C)C(=O)NC)CC=C(c2ccc(Cl)cc2)CC1 92137,N1(c2cc(N3CCCC(C(C)C)CC3)ncn2)CCc2nncn2CC1 92138,c1(C(=O)NCc2cn(CCCN(C)C(C3CC3(F)F)=O)nn2)cn(C)nc1C(F)F 92139,C1(C)(C(=O)NCC(CNC(C(CC)F)=O)O)CNC(=O)C1 92140,C1(O)(CC)CCN(C(c2nnnn2NC(=O)C(F)(F)F)c2cccs2)CC1 92141,Cn1nnc2c1C(C(=O)NCC#CCNC(C1CCOCC1(C)C)=O)CCC2 92142,CC1(C)CCC(n2cc(C3CCOC3)nn2)CN1C(c1ccn2cncc2c1)=O 92143,N1(CC(COCC(c2ccccc2)OC(C)=O)O)CCCC(NC(C)=O)C1 92144,N#Cc1ccc2c(c1)N(C(C1CCC(CNC(=O)CCC3CCCO3)CC1)=O)CC2 92145,c1(OC)cccc(C(=O)NCC(C)N(C(=O)CC2(O)CCCOC2)C)c1OC 92146,N1(C(C(C)NC(=O)C(C)(C)C)=O)CC2CC(C1)CN(C(C1CC1C(N)=O)=O)C2 92147,c1(CC)ncncc1C(N1CCCC1C(C)(C)NC(=O)C(C)Cn1ccnc1)=O 92148,c1(C(=O)NCCN(C(=O)CCCCC(N)=O)C(C)C)ccc2[nH]cc(C#N)c2c1 92149,c1(C(=O)N(C(C(C)NC(CN(CCCCCC)C)=O)C)CC)cnc(OC)nc1 92150,CC1(C(=O)NCCc2ccsc2)CCCN(C(c2c[nH]c(=N)o2)=O)C1 92151,N1(C(C(N2CC(C)C2)C)=O)CCN(C(c2ccncn2)=O)CC1c1nccn1C 92152,Cc1cc(CN2CCN(c3ccc(C4CC4)c(C)n3)CC2)ccc1F 92153,C1(C(N(C(CCNC(CCC#C)=O)C)C)=O)CCOC1C=C 92154,N1(C(C2CCCO2)=O)CC2(C(=O)NC(CO)C(F)(F)F)CC1CO2 92155,C1(CC=C)(NC(=O)C(O)C=CCCC)CCCN(C(C2(CCF)CC2)=O)C1 92156,N1(C(c2cnc(C)[nH]2)=O)CCCC(N(CCF)C(=O)C2CC2)C1 92157,C(=O)(CCCS(C)(=O)=O)NCC1(CNC(C(C)Cc2cnco2)=O)CC12CCC2 92158,C=CC(C)(C)CC(=O)NCCOC1CN(C(C2CCC(C)S2)=O)C1 92159,C(C)(C)(CC(F)C(=O)N(C)CC1COC(=O)N1)NC(c1c(C)c[nH]n1)=O 92160,C(=O)(C(C)(C)C(C)O)N(CC=CC(N1CCC(C)(NC(C)=O)C1)=O)C 92161,C(N=c1nnc(C)c(C)[nH]1)C1(C)CCN(C(CNc2cc(C(=O)OC)on2)=O)C1 92162,c1(OC)cc(F)c(Cl)cc1C(=O)NC1CN(C(C2CCCC(=O)O2)=O)CCC1O 92163,c1(C(=O)NC(CC=CC)C(=O)Nc2cncnc2OC)c[nH]c(=N)c(C)c1 92164,N1(c2cc(NCc3n(C(C)C)cnc3)ncn2)CCCOC(C(C)C)C1 92165,CC(C)C(C(=O)NC1CC(C)(C)C12CC2)C(C)NC(=O)CCCn1ccnc1 92166,C1(C(=O)Nc2cn(CC(C)C)nc2)CC(C)CN(C(=O)CCn2cncn2)C1 92167,N(C(=NCC1CCC1)N1CCC2(CCOC2)C1)CC1(C)CC2C=CC1C2 92168,c1(C2C(C(=O)NC3C=CC(CNC(c4c(C)ccs4)=O)C3)C2)ccccc1Cl 92169,c1(C(=O)NCC(C(C)(C)C)NC(C2C(CC(C)(C)C)C2)=O)cc(C#N)ccc1N 92170,C1(C(N(C2CCN(C(CCC#CC)=O)C2)C)=O)CC2(CCCC2)C1 92171,c1(OCC(=O)N(C(CN(C(c2c(C(C)C)nco2)=O)C)C)C)ccccc1C#N 92172,Cc1cccc(C(C(C)C)NC(N2CCC(c3cc(O)n[nH]3)C2)=O)c1 92173,C1(CC(N2CC3C(CNC(Cc4nc(C)c(C)s4)=O)C3C2)=O)CC2(CCC2)CO1 92174,C1(CNC(c2scc(C(N)=O)c2)=O)C(O)C(O)CN1C(C1CCCCC(=O)N1)=O 92175,C(C(O)C(C)(C)C)N(C(C(C)N(C(Cc1c(C)ocn1)=O)C)=O)C 92176,N1(C(c2c3c([nH]n2)C(C)CC3)=O)CCOC2(C1)CN(Cc1ccc(O)cc1F)C2 92177,C=C(C)CCNC(=O)NCC(C)NC 92178,CC1CCn2ncc(C(=O)NC(CNC(c3ccncc3O)=O)C(C)(C)C)c2C1 92179,Fc1cc(Cl)cc(Br)c1CN(c1ncc2cn[nH]c2n1)C1CNCC1F 92180,N1(C(C(=O)N(CC(CC)C)C)=O)CCCC2(CCCN(C)C2)C1 92181,c1(CC)cc(C(=O)NCC(O)CCNC(C2CCSC2)=O)cc(C)c1 92182,C(=O)(CC1=CCCCC1)NC1C(C)(CN(C(CC2(OCC)CCC2)=O)C)CCC1 92183,C1(OC)CC2(CCCN(c3ncc(Br)cc3NC(=O)OC(C)(C)C)C2)C1 92184,C#Cc1cc(NC(C2(C)CCCN2C(=O)CC(C)SC)=O)ccc1C 92185,C1(CCCNC(C(C2CC(C)(C)C2)OC)=O)CCCCN1C(=O)C=CCO 92186,C12(c3nc(CO)nn3-c3nn(-c4ccc(F)cc4)ccc3=O)CNCC1COC2 92187,c1(-n2cc(Sc3cncnc3)nn2)ccc([N+](=O)[O-])cc1F.N12CC3CC1(C3)C2=O 92188,c1(C(=O)NC(CCCNC(C(C)O)=O)c2ccccc2)c[nH]c(C#N)c1 92189,N1(C(C=CC(C)(C)C)=O)CCc2c(CNC(=O)CC34CCCC3C4)cccc2C1 92190,C(=O)(C(CN(C)C)CC)NCc1c(C(=O)NC(C(=O)NC(CC)C)C)[nH]cc1 92191,C(=O)(C(C)S(C)(=O)=O)NCc1c(C(=O)NC(c2ncc[nH]2)CC)n[nH]c1 92192,N1(C(CC2C(C)C2)=O)CCCC1C1CCN(C(=O)CO)C1 92193,C1(C2CC2)(CNC(C2(OC)CCC2)=O)CCN(C(c2c(Br)nnn2C)=O)C1 92194,Cc1nc(C(N2CC(F)CC2CNC(C2C(C(F)F)C2(C)C)=O)=O)cn1C 92195,CC(C)CC(F)C(=O)NCCC1CCCCN1C(c1ccnn1C(C)C)=O 92196,c1(CNC(=O)COCCNC(C2CCCS2)=O)ccncn1 92197,N1(C(C=CC=CC)=O)CC(NC(=O)C(C)SCC)CC1(C)C 92198,C#CC1(O)CN(C(=O)CSCCNC(C2(CF)CC2)=O)C1 92199,CC#CCCC(=O)N1CC(OCC)C(NC(=O)CCCN(C)C(C)C)C1 92200,C1(O)(CN(C(=O)CCC2CCC(=O)N2)C)CN(C(=O)CCc2cn[nH]c2)C1 92201,c1(CC)ccc(C(=O)NC2CC(N(C(=O)C=CC3CCOCC3)C)C2)cn1 92202,C1(CC(=O)NCC(C)(CO)NC(C(C)=C2CCCC2)=O)COC(C)(C)C1 92203,N1(C(CNC(C(C)(C)C)=O)=O)CCOC(C)(CNC(C2CC2(Cl)Cl)=O)C1 92204,C1(NC(C(COC)(F)F)=O)COC2(CNC(=O)CCN3CCCC3)CC1C2 92205,C#CCC(CC(F)F)C(=O)N1CCCC1CCC(=O)Nc1ccc(C)cc1CO 92206,CCC(CC)CC(F)C(=O)N1CCC2(CC1)CC2C(N1CCC1C1CCC1)=O 92207,N1(C(c2ccc(CC)cn2)=O)CC2(C)CC1(C(N1CC3CCC3(CO)C1)=O)C2 92208,c1(C(N(CC(C)N(C(CN(CCC)C)=O)C)C)=O)ccc(N2CCOCC2)cc1 92209,C(C1=CCN(Cc2cc(Cl)ccc2Br)CC1)NC(c1cccc(F)c1Cl)=O 92210,C1(CC(=O)NCC(CNC(CCCN(CC)CC)=O)F)CC(OCC)C1(C)C 92211,N1(C(C(C)OCC=C)=O)CC(C(N2CCCC(C(C)(C)O)C2)=O)C(C)(C)C1 92212,N1(C(C2(N(C(c3n(C(C)C)ccn3)=O)C3CC3)CCC2)=O)CC2(CC(CO)CO2)C1 92213,C=CCCCCCCC(=O)N1CCN(C)C(C(=O)NC2CCCC2CN(C)C)C1 92214,c1(OC)c(NC(C2CC(C)CN2C(c2ccccc2S)=O)=O)cc(F)cc1F 92215,C1(S(C)(=O)=O)(C(=O)NC(C)CC(C)NC(c2ccncc2F)=O)CCC1 92216,c1(C(=O)NCC(CNC(C2(c3ncco3)CC2)=O)OC)cc(F)c(F)cc1F 92217,C(=O)(CC(C)C(=O)NC1(C)CN(C(=O)CCn2cc(Cl)cn2)C1)OC 92218,Cc1nc(C2CC2)[nH]c1C(=O)NCC1(CCNC(C2(C)CCCC2C)=O)CC1 92219,N1(C(C2CC=C(C)CC2)=O)CCCC2CN(C(=O)CC3CC=CCC3)CC12 92220,N1(C(CC2CN(C)C2)=O)CCN(C(c2cccc3c2CCC3)=O)C2CCCCCC12 92221,Cc1ccc(CC(N2CC(CNC(=O)CNS(N)(=O)=O)C(O)C2)=O)c(F)c1 92222,CCC(CCC(=O)N1CC(n2cccn2)C1)NC(=O)CC(C)C1CC1 92223,CC1CCN(C(=O)C(=O)NCC(F)F)C1CNC(c1c(Br)ncn1C)=O 92224,C(=O)(C(C)S(=O)(=O)C(C)C)NC(CC(C)C)CNC(=O)CCc1cnn[nH]1 92225,N1(C(C(C)=CC)=O)CC(CNC(=O)CCC(CC)CCC)OC2(CCC2)C1 92226,c1(N(C)Cc2ccccc2[N+](=O)[O-])ccc(S(=O)(=O)NCC2CCCCS2)cn1 92227,C(CCCC(=O)NCCCCCO)N(C(C1C(C(C)C)OCC1)=O)C 92228,C1(CC(=O)N(C2CCN(C(=O)COCCF)CC2)C)COC(C)(C)CO1 92229,N1(C(C=CC(=O)N(C)C)=O)CCOC2c3ccccc3OCC12 92230,C1(NC(C(c2cccc(Cl)c2)CC)=O)CCC(NC(C2CCSC2)=O)CC1 92231,O1NC(=O)C(F)C2(O)CN(C(=O)C1(C)C)C2.c1(OC)ccc(=N)[nH]n1 92232,CC1CN(C(C2(C(F)F)CCCC2)=O)CCN1C(C1CCC(=O)NC1)=O 92233,C1(NC(Cc2c(C)cc(C)s2)=O)CN(C(c2cccc(N)c2)=O)C2(CCC2)C1 92234,C1(CC(=O)N(C)CC2N(C(C3CC(OCC)C3)=O)CCOC2)COCC(C)(C)O1 92235,N1(C(COCCCC)=O)CCN(C(C2(C)CCC(OC)C2)=O)CC12CCC2 92236,C1(OC)(OC)CCN(c2nnc(-c3cnn(C)c3)n2CCC#N)C1.C1(C)CC1 92237,C1(C(C)NC(C2CCCCC2)=O)CCCN(C(c2c(C(F)(F)F)cnn2C)=O)C1 92238,C1(CNC(C2C(C=C)C2)=O)COCCN1C(=O)CC1CCSCC1 92239,c1(C(=O)NC2(c3cccc(Cl)c3)CC2)cnn2ccc(-c3ccsc3CO)cc12 92240,O=C(C=CC(N1CCOCC1)=O)NN1CCCC1C(=O)N=c1ccn(CCO)[nH]1 92241,C1(NC(C2CC(SC)C2)=O)CC2COCC(C1)C2NC(c1cnn[nH]1)=O 92242,C1(C(=O)NCCCN(C(C)C)C(C23CSCC2C3)=O)CC2CC(=O)C1C2 92243,c1(C(N(C2CCCCC2)C)=O)c[nH]c2cccnc12.C12CC(C1)C(=O)N2 92244,Cc1nc(CO)ncc1NC(=O)C=CC1CCN(C(=O)C(C)CC#N)CC1 92245,C1(CC)CCN(C(=O)CCOC2CC2)C1CNC(=O)C(CCSC)OC 92246,C1(CNC(C(c2cccc(O)c2)C)=O)CCN(C(=O)C=CC2CCCC2)CC1 92247,CCC(C)(CC)C(=O)NC(C1CCN(C(=O)C(C)Oc2cccnc2)C1)C 92248,c1(C(=O)NC(CN(C(c2cc(CN(C)C)c[nH]2)=O)CC)C)c(Cl)cnn1C 92249,c1(CCC(=O)NCC(F)CNC(C2(CO)CC2)=O)ccc(F)c(Br)c1 92250,c1(C(C)C(=O)NC(C2(O)CN(C(c3ncccc3Cl)=O)C2)C)c(F)cccc1F 92251,C(=O)(C(CCF)NC(=O)C(CCC)NC(N)=O)N(C(C=C)C)C 92252,c1(C(=O)OC)coc(C=CC(=O)N(CC(C)NC(=O)Cc2ccon2)C)c1 92253,N1(C(c2scc(C(C)=O)c2)=O)CCN(C(C2CC2(F)Cl)=O)CC(C)(C)C1 92254,c1(C(=O)NC2CC(NC(C3(C)CNC(=O)C3)=O)C2)ccc2nc(C3CC3)[nH]c2c1 92255,C1(C(=O)NCC(=O)N(C(c2ccncc2)C)CC)CCC(OC)CC1 92256,C1(CNC(C2CCCC3CC23)=O)CCCC12CCN(C(C1CCCC1O)=O)CC2 92257,c1(OC)n[nH]c(C(=O)NCC2CCC(NC(c3ccc(Cl)o3)=O)C2)c1Cl 92258,N1(CCN=C(NCC(CC)CO)NC2CCC2)CCc2ccccc21 92259,C1(CN(C(C(C=C)O)=O)C)CC(F)CN1C(C1CNC(=O)N1)=O 92260,C(=O)(CC1=CCN(C(c2c(F)cccc2F)=O)CC1)Nc1ccc(C)nc1C 92261,c1(C(N2CC=CC(NC(C3(CC=C)CCOCC3)=O)C2)=O)onc2ccccc12 92262,c1(C(C)N(C(=O)C(C)(C2CC2)N(C(=O)CN(C)C)C)C)ccccn1 92263,N1(C(C(n2cnc(C#N)n2)CC)=O)CC(CNC(=O)CC(C)C)C(C(F)(F)F)C1 92264,C(=O)(CCCCC(C)CC)NC(CCCC)CNC(c1ncoc1C1CCC1)=O 92265,C1(NC(CCCN(C)C)=O)CCC2CN(C(c3nc(Cl)cs3)=O)CC2C1 92266,C(CC(F)CN=[N+]=[N-])NC(c1cc(CNC(C(C)NC(CC)=O)=O)ncc1)=O 92267,Cc1nn(CC(N2CCCC(NC(c3ccc[nH]3)=O)C2C)=O)c(C)c1C 92268,C1(C(N(C(CC)C2CC2)C)=O)COCCC1NC(c1cc(C)sn1)=O 92269,c1(N(C)Cc2cnn(CC)c2C)ncnc(NC2CC3CC(O)C2C3)c1C 92270,c1(C(=O)NC2CC3(C(NC(=O)CC4CCCS4(=O)=O)C3)C2)nc2cnccc2s1 92271,Cc1ccc(Cl)cc1NC(=O)CCCCCNC(=O)Cn1cnnc1O 92272,CCCC(CCCNC(C1CC1c1ccccc1)=O)NC(C1CC1(Cl)Cl)=O 92273,c1(OC)ccc(C(N2CC(CNC(=O)CC3CCOCC3)CC2(C)C)=O)c(F)c1 92274,CCC(O)CC(=O)NCCC1(CNC(=O)CCc2nc(-c3ccco3)no2)CC1 92275,CC1(C)CC(NC(c2cc(C#N)c[nH]2)=O)CCN(C(C2(C)CCCC2(F)F)=O)C1 92276,C1(CNC(C(N2CCOCC2)C)=O)CCN(C(C2CNC(=O)C2)=O)CC1 92277,c1(N(CCNC(C23CCCCC2OCC3)=O)CC)ncnc2c1nnn2C 92278,Cc1c[nH]c(C(=O)NC2CC(CNC(c3cc(N)c(F)cn3)=O)C2)cc1=O 92279,C(CCC(C)C)(C(=O)N(C)CCOCC1CC1)NC(CC(CC)SC)=O 92280,c1(C(c2n(CCOCC)nnn2)NCc2sc(Br)nc2C)cncc(Br)c1C 92281,C1(CC(C)NC(CCC(C)C)=O)CC2CCC(C1)N2C(=O)COCC(F)F 92282,c1(C(=O)NCC2CC(NC(C(c3n(C)ncc3)O)=O)C2)ccc2c(c1)COC2 92283,c1(C(=O)NC(C2(C(=O)NC3CCCC3(F)F)CC2)C)ccc([N+](=O)[O-])o1 92284,C=CC1CN(C(c2cccc[n+]2[O-])=O)CC1NC(c1ccc(C(C)C)c(F)c1)=O 92285,c1(C(=O)NC(C(C)NC(Cc2ccc(OC)cc2)=O)C(C)C)c(F)cccc1F 92286,C1(CCC(=O)NCC(C2CC2)SC)CCCN1C(=O)CCn1cccn1 92287,c1(CC(=O)CN2CCN(C3CC(F)(F)C3)CC2)ccc(Cl)cc1 92288,CCC(C)(CN(C(=O)C(C1CC1)NC(=O)NC)C)NC(c1coc(CSC)c1)=O 92289,C1(O)(CC(C)C)CCN(C(C2CC=CCC2C)C(=O)NCc2cccs2)C1 92290,c1(OC)cccc(Br)c1CN1CC2C(C1)N2C(c1ccc(C2CC2)cc1)=O 92291,c1(C(=O)NCC(C)(O)CNC(C2CC2(Cl)Cl)=O)cn2ccccc2n1 92292,c1(NC(C)CN(C(C(C(C)C)SC)=O)C)c(F)cccc1[N+](=O)[O-] 92293,c1(C(=O)NCC(C2CCCCC2)NC(C(C)OCCOC)=O)ncc(Cl)cc1Cl 92294,c1(OC)ccc(Cl)c(F)c1C(=O)NCC(C(C)C)NC(=O)CSc1ccncc1 92295,c1(OC)ccnc(NCC(=O)NCC(C)CNC(C2(C)CCCC2C)=O)n1 92296,C1(C(F)F)(OC)CCCN(C(c2nc(Br)nn2C)C(=O)NC(C)(C)C)C1 92297,N1(C(C(C(C)C)C)=O)CCn2ncc(CN(C)C(C3C4CCCC34)=O)c2C1 92298,C1(NC(CC(CC)C(C)C)=O)CN(C(C2(CC3CC3)CC2)=O)Cc2ccnn2C1 92299,c1(C(=O)Nc2ccc(-n3c(C)cc(C)n3)nc2)cc(F)c2nc(C)cn2c1 92300,CCCCC(O)C(=O)NCC1(C)CCN(C(c2cccnc2OC)=O)C1 92301,c1(NC(CSC(C)=O)CC(C)C)ccc(F)cc1C 92302,C(CO)(CC(C)(C)C)NC(C1C(CNC(Cc2nc(C)[nH]n2)=O)C1(C)C)=O 92303,C1(NC(c2cnc(SC)[nH]2)=O)C2CC(NC(=O)C=Cc3cscn3)CC12 92304,C1(N(C(c2scc(CC)n2)=O)C(C2CCOCC2)C)C(C)OCC12CCNCC2 92305,c1(C(N2CC(O)(C(C)NC(=O)CCN(C)CCO)C2)=O)cc(Cl)c(Cl)[nH]c1=N 92306,C=C=CCC(=O)N1CCC(C(C)(C)NC(=O)Cc2cc(CC)no2)C1 92307,C(C(C)(C)CC(=O)NCC1(CNC(c2oncc2C)=O)CC12CCC2)OC 92308,N1(C(c2coc3c2COC3)=O)CCN(C(=O)C(F)(F)C(F)(F)F)CC2(CC2)C1 92309,CC(C)CCC(=O)C(=O)N1CC(C2CC2C(N2CCC(CCCO)C2)=O)C1 92310,C1(O)(CNC(Cn2cc(CNC(CCC=CCC=C)=O)nn2)=O)CCC(C)C1 92311,C#CCC(C)C(=O)N1CCN(CCCNC(c2cc(CN(C)C)on2)=O)CC1 92312,c1(OCC(C(=O)NC(CNC(COC)=O)(C)CO)C)ccccc1Cl 92313,CC(CC(=O)N1CCC(O)(CCNC(=O)C(F)CC2CCOC2)C1)C(F)(F)F 92314,c1(C(C)C)cc(C(N2CC(CO)(NC(c3cccc(F)c3F)=O)C2)=O)ccc1F 92315,C(C1CCCO1)=CC(=O)NCCC(C)N(C(=O)CCC1CCC1)C 92316,C(=O)(CCCN=[N+]=[N-])NCCCCC(C)NC(C1(COC)CC1)=O 92317,CCC(C(=O)NCCCCC1(NC(=O)Cc2csc(Cl)n2)CC1)C(F)(F)F 92318,CC(C)(C#N)CCCC(=O)NCCC1CN(C(=O)CNc2c(F)cccc2F)C1 92319,C1(NC(c2csc(C(F)F)n2)=O)CC2CN(C(C3(C(F)(F)F)CCCC3)=O)CC12 92320,C12(CNC(COCCOCC)=O)CC1CCN2C(=O)CN1CSCC1=O 92321,c1(C(=O)NC2(C)CN(C(CN(C(COC)=O)C)=O)C2)cc(C(F)F)ccn1 92322,C1(CNC(c2n(CC=C)ccc2)=O)C(C)CCCN1C(c1cc([N+](=O)[O-])n[nH]1)=O 92323,Cc1cc(C(N2CCC2C(=O)N(CC(F)F)C)=O)oc1C 92324,N1(C(C2CC(C)N2C(C2CC3CCC(C2)O3)=O)=O)CCc2ccccc21 92325,N1(C(COC2C(CC)CCCC2)=O)CCC2(CCCN2C(C2CC3(CC3)C2)=O)C1 92326,c1(C(N2CCC(C(CO)NC(c3c(C)onc3)=O)CC2)=O)ccc2nonc2c1 92327,C1(NC(C2(COC)CCC2)=O)CN(C(=O)COc2cccc(F)c2)CC2(CC2)C1 92328,C1(NC(c2cccc(C#C)c2)=O)CN(C(=O)CCC2CC2)CC1C1CC1 92329,c1(C(N2CCCC(N3CCCC3=O)C2)C(=O)NCC(C)C)cnn(C(C)C)c1I 92330,C1(C(=O)NC(c2ccc(C)nc2)C)CCN(C(c2ccccc2F)=O)C(C)(C)C1 92331,C(=O)(C1=CCc2ccccc21)NC(C)CC(C)NC(c1cnc(Cl)n1C)=O 92332,c1(C(C(=O)NC2C(CC(=O)NCC(c3cccs3)C)C2)O)cccnc1 92333,C1(NC(CCC(N)=O)=O)CCC2CCN(C(=O)C(C3CC(F)(F)C3)O)C1C2 92334,N1(C(C(CC(C)C)=O)=O)CCC2CN(C(C3(C4CC4)CCC3)=O)CC2CC1 92335,n1(C(C)C)cnc2c(N(C)Cc3nc[nH]n3)[nH]c(=NCc3nncs3)nc12 92336,N1(C(C(c2ccccc2)OC)=O)CCCOC(CNC(C2(SC)CC2)=O)C1 92337,c1(C(=O)NCCCN(C(C2CC(C)(F)C2)=O)CC)cc2n(n1)CCCNC2=O 92338,n1(CCNC(N(CCCC=C)C)=O)cc(NC(=O)OC(C)(C)C)nn1 92339,N1(C(C2C(C)(C)CO2)=O)C2CCC1CN(C(C1CC3C=CC1C3)=O)C2 92340,C1(N(C(C(CCC)CC)=O)C)CC2CCC(C1)N2C(=O)C(F)(F)C(O)CC 92341,c1(N(CCC)CCNC(C2(C#N)CCC2)=O)cc(N2CCNC2=O)c(F)cc1F 92342,c1(C(N2CC(OC)C(NC(=O)CC(C)N(C)C)C2)=O)ccc(F)c(C(C)C)c1 92343,C1(O)(C(N(CCNC(Cc2ccn(CC)n2)=O)C2CC2)=O)CCC(C)(C)CC1 92344,Cc1ncc(CCNC(=O)CCN(C(=O)C=CC2CCOC2)C(C)C)[nH]1 92345,N1(C(C(CC)(F)F)=O)CC2CCN(C(=O)CCOCC3CCCC3)CCC2C1 92346,c1(C(C(N2C(C)(CNC(C(C3CC3)OCC)=O)CCC2)=O)=O)ccc(Cl)cc1O 92347,c1(C(N2CCN(C(c3cccc(F)c3)=O)CC2)=O)coc2c1C(O)CCC2 92348,c1(OC)cc(F)ccc1NC(=O)CN1CCCN(C(c2cccc(Cl)c2)=O)CC1 92349,CC1CN(C(=O)Cc2cc(O)nc(O)n2)CCN1C(c1coc(Cl)c1)=O 92350,c1(NC(C(=O)NCC2N(C(=O)OC(C)(C)C)CCCCC2)=O)cnc2n1CCCC2 92351,c1(C(=O)NCC2CN(C(CC3(C=C)CC3)=O)CC2O)nc2n(c1Cl)CCCC2 92352,c1(C(C)=O)cccnc1Oc1ccc(Br)cc1.c12cnc(s1)CN(C=O)C2 92353,N1(C(C)=O)CCCC2(C1)C(NC(=O)Cc1cc(F)c(F)cc1F)CCN2C 92354,c1(C(=O)NCC(CC)(C)NC(c2csc(-c3cnn(C)c3)n2)=O)nc(O)sc1C 92355,N1(C(CN(CCC#C)C)=O)CCCC(C(=O)N(C2(C(COC)O)CC2)CC#C)C1 92356,c1(C(N2CCN(C(C3CC34CCC4)=O)CC2CCO)=O)ccc([N+](=O)[O-])c(Cl)c1 92357,C1(C(=O)NC(CC)(C)C(F)(F)F)CCN(C(=O)CN(C)C2CC2)C12CCC2 92358,C1(C(=O)NC2C(CNC(CNS(NC)(=O)=O)=O)CCC2)COC(C)(C)CO1 92359,Cc1cccn2c(CC(=O)NC(C)C(=O)NC(c3ccccc3)C(=O)O)cnc12 92360,c1(NC)cc(Cl)ccc1C(N1CCC(CO)C(NC(C2(C)CCCCO2)=O)C1)=O 92361,C(c1ccccc1F)=CC(=O)NC1(C)CCN(C(CN2C(C)CCC2)=O)C1 92362,C1(C(=O)NCCCOC(=O)NC)CSC(CCC(C)C)C(=O)N1 92363,CCC(=O)CCC(=O)N1CCCN(CCNC(=O)C(F)C2CCOC2)CC1 92364,N1(COC)CCN(C(c2ccc3c(c2)CC3)C(=O)NCC2CC2)CC1=O 92365,c1(C(=O)NCCC2CC(C(=O)NCC3(C)CCCO3)C2)cnn2c1OCC2 92366,C1(C(=O)NC2C(CNC(c3nc(N(C)C)oc3)=O)CC2)CCCCC1(F)F 92367,Cc1cc(C(=O)NC2CCC2CNC(=O)Cn2ccc(C3CC3)n2)ccn1 92368,c1(C(=O)NCC2N(C(c3c(C)nns3)=O)CC=C2)cnc2nc(O)ccc2c1 92369,N1(C(CC2CCC(C)C2)=O)CC23CCCC2(C1)CN(C(c1coc(CO)c1)=O)C3 92370,c1(C(C(N2C(C(=O)OCc3ccccc3)CSC2)=O)O)cc(F)c(F)cc1F 92371,C1(C(=O)NCc2ccn(CCC)n2)CCCC(NC(c2c[nH][nH]c2=N)=O)C1 92372,c1(CCNC(C(C2(C)CC2)NC(C(C)=CCC)=O)=O)ccn(C)n1 92373,CN1CCN(C(=O)C(F)(F)c2cnccn2)CC1CNC(C1(C)CC=CCO1)=O 92374,c1(CNC(C(=O)NCc2ccc(SC)cc2)=O)ccc2c(c1)CCO2 92375,Cc1cc(C(=O)NCCC2CC(NC(=O)Cc3ccsn3)C2)n2nc(C)cc2n1 92376,N1(C(CC2CC(=O)C2)=O)CC(NC(=O)C=CC2CCC2)C2CC12 92377,CC1(C#CC(=O)NC2CN(C(=O)C3=CCCCC3)CC23CC3)CC1 92378,Cc1onc(CC(=O)N(CC(C)CNC(=O)C(O)CC2CCCCC2)C)c1C#N 92379,CN1CCC(CN(C)C(C2CC(NC(C3(C)CC3)=O)C2)=O)CC1 92380,N1(C(CC2CCCN(C)C2)=O)CCC2(CCC2CNC(=O)CCC2CC2)CC1 92381,C1(NC(Cn2c(C)ncc2)=O)CN(C(C2(Cl)CC2(C)C)=O)CC(C)(C)C1 92382,C(F)(F)(C(=O)NNC(=O)CSCCCC1CC1)c1cccc(C)n1 92383,N1(C(c2cc(C(F)F)cs2)C(=O)NCC(C)C)CCCC2CC(C)CCC12 92384,N1(C(C(C)(C)C2CCCO2)=O)CC2(C=C(C(=O)NOCCN3CCCC3=O)CO2)C1 92385,C1(C(=O)NCCCC(CO)NC(=O)CN(C)C)(OC)CCS(=O)(=O)C1 92386,c1(C(=O)NCc2cc(C(=O)NCC(CC)(C)Cl)n(C)n2)cc(C)nnc1O 92387,C1(CNC(c2ccc(Cn3cc(CC4CCOC4)nn3)o2)=O)CCCOCC1 92388,C1(CNC(C2(C)CCN(C)C2)=O)CC2(CC(NC(=O)CC3CC4(CCC4)C3)C2)C1 92389,C1(SC)CN(C(=O)CSc2nncs2)CC1NC(=O)CCc1ccsc1 92390,C1(NC(C=Cc2ncc(C)[nH]2)=O)CN(C(=O)C(C2CC2)C2CC2)CC1C1CC1 92391,N1(C(C23CN(C(C(CCC)Cl)=O)C(C2)CO3)=O)C2CCC1CC(CO)C2 92392,c1(N(C(CCNC(C2(OC)CCS(=O)(=O)C2)=O)C)C)ccc([N+](=O)[O-])cc1Cl 92393,N=c1nc2c(c[nH]1)CC(C(=O)NCCCCNC(=O)CC13CCCC1C3)CC2 92394,C1(C(N(CCNC(CCC=C=C)=O)CCOC)=O)CCC2(CCC2)CO1 92395,C1(C(=O)NCC2(O)CN(C(C(CCC#C)O)=O)C2)CC(c2cn(C)nc2C)=NO1 92396,C1(NC(C(N2C(CC)CCC2)=O)=O)CCCCN(C(=O)CSc2ccccn2)C1 92397,CC1(C)NC(=O)N(CC(=O)NC2CC(NC(=O)C(CO)NC(N)=O)C2)C1=O 92398,C1(CNC(=O)C(=O)Nc2nnc(-c3ccccn3)s2)CCCN2CCCC12 92399,c1(C(N(C)CC2CN(C(C34CC(F)(C3)C4)=O)C2)=O)cc2n(n1)CCNS2(=O)=O 92400,c1(C(N2CCC(C)(NC(C(CC(C)C)NC(N)=O)=O)C2)=O)cnn2c1NCCC2 92401,C1(NC(Cc2c(C)con2)=O)CCCCN(C(=O)C(F)C(C)(F)F)C1 92402,c1(C(=O)OC)cnn(C)c1S(=O)(=O)NCC1OC(=O)CC12CCC2 92403,Cn1ncc(Cl)c1C(=O)NCC1(CO)CCN(C(=O)C=CC(C)(C)C)C1 92404,N#Cc1c(NCCNC(C2(c3ccc(Br)o3)CC2)=O)cccc1F 92405,C1(NC(c2c(C)onc2CO)=O)CCC2CN(C(=O)CCCN(C)C)CC2C1 92406,C#CC1(C(=O)NC(c2ccc(O)nc2)C)CCN(C(C2C=C(C)CS2)=O)C1 92407,C1(NC(c2c(C)nc(C)o2)=O)CC(NC(=O)Cc2ncc(F)cc2F)C12CCC2 92408,C(C(C)(C)C(=O)NCc1ccc(C(N2CC(OCCO)C2)=O)nc1)SC 92409,Cc1cc(F)cnc1C(=O)NC(CC1CC1)C(=O)NCC1CC2(CCC2O)C1 92410,N1(C(C=C(C)C)=O)CCC(N(CCO)C(c2cnco2)=O)C1 92411,C1(OC)CN(C(=O)COC2(C)CCCC2)CC1CNC(C1CCCN1N=O)=O 92412,C(N=c1cc(C)nc(C)[nH]1)C1CN(C(c2cc(C)ncc2)=O)C(C)C1 92413,C1(C(N2CC(CC)(NC(=O)Cc3cccnc3O)C2)=O)CCC2CC1C2(C)C 92414,C(CC1CCc2ccccc21)NC(N1CCCC1Cc1cc(F)ccc1Cl)=O 92415,C1(NC(C2N(C(CCC)=O)CCCC2)=O)CCN(C(=O)CCCC(F)F)C1(C)C 92416,c1(C(N(CCCNC(=O)CC(C)(C)F)C(C)C)=O)cc(Cl)cc(F)c1N 92417,C1(CC)CC(C)CN(C(=O)CCC2CCC(NC(C3CCC(CC)CC3)=O)C2)C1 92418,C=C=CC(C)C(=O)NC1CCN(CCNC(=O)C(C)CC=C)CC1 92419,c1(C(=O)NCc2cn(CCOC(C)=O)nn2)ccc(-n2cc(Br)cn2)cc1 92420,C=CCC(CC)C(=O)N1CC(CNC(=O)CC(C)(C)OC)CC1(C)C 92421,c1(C(=O)NCC(C)NC(C2CC2(F)F)=O)ccc2c(c1)B(O)OC2 92422,c1(C(=O)NCC(CC(C)C)NC(c2ccn(C)c2)=O)cc2ccc(Cl)c(F)c2[nH]1 92423,N1(C(C(C2CCCO2)OC)=O)CC2(CCN(C(c3cc(N)c(F)cc3C)=O)C2)C1 92424,N1(C(CC(=O)OC)=O)CCN(C(=O)CNS(=O)(=O)N(C)C)C(CO)C1 92425,c1(C(N(CCNC(c2ccc(OCCF)cn2)=O)CC)=O)nccn2nccc12 92426,C(=O)(CC1OCCc2ccccc21)N1CCC(C)(NC(=O)CC2(O)CCC2)CC1 92427,C(=O)(C(COC(C)=O)C(F)(F)F)NC1C2(NC(C(CCCC)C)=O)CCC(C1)C2 92428,Cn1ncc(C(=O)NC2CCC(n3cc(C4CCOCC4)nn3)CC2)c1C1CC1 92429,N1(C(C2C(NC(c3ccc(OC)s3)=O)C3C=CC2C3)=O)CCC2(CCOC2)C1 92430,c1(CC)ccc([N+](=O)[O-])cc1C(=O)NC1CCN(C(C2CSCC(=O)N2)=O)CC1 92431,CC(CC(=O)NC1(C)CCN(C(c2ncccc2O)=O)C1)C(F)(F)C(F)(F)F 92432,N1(C(C2CN(CC)C(=O)C2)=O)CC2(CCN(C(c3ccc(Cl)o3)=O)CC2)C1 92433,N1(Cc2ccc(C#C)s2)CC2(CN(C(=O)Nc3ccccc3F)CCO2)C1 92434,c1(OCC(=O)NC2C(NC(c3c(Br)ccc(C)c3)=O)C2)ccc([N+](=O)[O-])cc1 92435,c1(C(N2C(C)C(C)N(C(c3cncnc3)=O)CC2)=O)ccc(S(=O)(=O)CF)cc1 92436,CC1C2CC(C2OC(C2CN3CCN2CC3)=O)N1Cc1ccccc1 92437,C1(CN(C(c2c(C)cns2)=O)C)CN(C(=O)CCc2cccc(O)n2)CCO1 92438,c1(OC)cc(F)c(NC(=O)COC2CN(C(=O)C=CC3CCOCC3)C2)c(F)c1 92439,c1(CSCCC(=O)N(C(C)CNC(=O)CC2CC2)CC)ccc(F)cc1 92440,N1(C(=O)Cc2cncnc2)CCOC2(C1)CN(C(c1cc3c(s1)COCC3)=O)C2 92441,C(=O)(C1CNCc2c(-c3ccccc3)cccc21)N1CCC(c2onc(C)n2)C1 92442,C(=O)(CC(C)(O)C(F)(F)F)N1CCN(C(C2C(OC)(OC)CC2)=O)CC1 92443,N1(Cc2cn(C3(SC)CC3)nn2)CC(C)N(C(C2C3CCC(=O)C23)=O)C(C)C1C 92444,C1(NC(C2(CC)COC2)=O)CCC12CCN(C(=O)CCc1cc(Br)no1)CC2 92445,C1(C(F)(F)F)(C(=O)NC2CN(C(C3C(C)(C(C)C)C3)=O)C2)CC2CCC1CC2 92446,c1(CCC)cc(C(N2CC(N(C(=O)CSc3nccn3C)C)C2)=O)n(C)n1 92447,c1(C(=O)NCC(CC)NC(=O)CN(C)C(C)=O)csnc1C 92448,c1(OC)cc(Cl)ncc1NC(C1CC1C(=O)NC(c1ccc(C#N)cc1)CO)=O 92449,N1(C(C=Cc2c(C)ccs2)=O)CCC2CN(C(C3CC34CCSCC4)=O)CCC12 92450,C#Cc1cn(C)nc1C(=O)NCC1CN(C(c2cnoc2C2CCC2)=O)CC1C 92451,c1(CNC(C2N(C(C3CC(OCC)C3)=O)CCC2)=O)ccc(O)c(C)c1 92452,c1(C(C)NC(=O)NC2CC(C)(COC)C2)cccc(SC)c1 92453,C1(C(=O)NC2C(C)(C)CN(C(=O)Cc3ccsc3)C2)CCc2nccn2CC1 92454,C#Cc1ccc(C(=O)NCCC(C)NC(C2CC(C#N)C2)=O)c(F)c1 92455,C(c1ccccc1[N+](=O)[O-])=CC(=O)NC1CCN(C(C2CCCCC2)=O)CC1F 92456,N1(C(C2(CC)CC2)=O)CCN(C(c2ccc(C3CC3)c(F)c2)=O)CC12CCC2 92457,CCC(C)C(O)C(=O)N(c1ccnc(C)c1)C(C1CCC(C(=O)OC)O1)=O 92458,CC1(CC(=O)NCC2CN(C(=O)Cn3nccn3)C3CC23)CCOCC1 92459,c1(C(=O)OC)cccc(CNC2(F)CC(NC=O)C2)c1OC.C12CN(C1)C2=O 92460,c12cc(C)ccc1CN2C1CC(N)C1.c1(SC)ccccc1 92461,NC1CCN(C(c2csc(-c3ccco3)n2)=O)C(CO)C1 92462,N1(C(C2CCN(CC)CC2)=O)CCN(C(C2CCSCC2)=O)C(CC#N)C1 92463,N1(C(C(C(C)C)SCC)=O)CCOC2(CCN(C(=O)CCCc3cncs3)C2)C1 92464,C(C(C)(C)CC(=O)N1CCC(N(CCO)C(c2cnnc(C)c2)=O)C1)OC 92465,C1(NC(c2nc(C)n(C)n2)=O)CC2CC(NC(=O)C3=CCOCC3)CC2C1 92466,Cc1cn(CCC#N)[nH]c1=NC(=O)c1csc(Nc2ncncc2F)n1 92467,C1(Cc2scc(C(=O)OC)n2)CCN(C(=O)NCC2(C)CCCS2)C1 92468,CC1Oc2c(C(=O)NC(CNC(=O)C(C)(F)F)C3CC3)cccc2NC1=O 92469,CC1(C)CCC2(CC1)CC2C(=O)NCC1CCN(C(C2CCOCC2)=O)C1(C)C 92470,N1(C(CCc2c(C)ncs2)=O)CCN(C(C2CCS(=O)(=O)N2C)=O)CC(O)C1 92471,C1(C(N2CCC(N(C(=O)C=CSC)CCC)C2)=O)CCc2nc(C)ncc2C1 92472,c1(OC)ccc(N(C(=O)C(C)N(C)Cc2ccc(Br)s2)Cc2ccco2)cc1 92473,CN1CC2C(C(=O)NC3CC(NC(=O)NC(=O)NC(C)(C)C)C3)C2C1.C1(=O)CN1 92474,Cc1cc(CNC(=O)NC(Cc2cccc(Br)c2)C(=O)O)ncn1 92475,C(C(C)(C)CN=c1[nH]c(=N)[nH]c(=NC(Cc2ccccc2)c2cncs2)[nH]1)SC 92476,c1(C(N2CC=CC(NC(C3(OC)CCCOC3)=O)C2)=O)cnc(Cl)cc1N 92477,c1(C(=O)OC)cc(S(=O)(=O)N(C(c2ccccc2)CF)C)ccc1F 92478,C1(N(C)C)CCC(CN2CCCC(C(O)C(F)(F)F)C2)CC1 92479,C=C(C)C(C)(O)C(=O)NNC(=S)NCCCC1CCCN1C(=O)OC(C)(C)C 92480,Cc1ncnc(C(=O)NC(C)CC(C)NC(=O)CCC(=O)c2ccc(Cl)s2)c1C 92481,c1(C(C(N2CC(C)OC(C)C2)=O)(C)C)ccc(Cl)cc1[N+](=O)[O-] 92482,C(=O)(C(CC(C)C)N(C1CC1)CC1CC1)OC.c1(C2C(=O)N2)ccccc1Br 92483,CC1CN(C(=O)C(C)(CO)NC(c2ccc(CC#N)cc2)=O)Cc2nncn21 92484,N1(C(C(C(C)C)N2CCCC2=O)=O)CC2CCCN(C(c3cc(O)no3)=O)C2C1 92485,N1(C(C(CO)OC)=O)CCC(O)(CCNC(=O)COC2CC(F)(F)C2)CC1 92486,c1(C(=O)NCC(=CC(=O)NC(C(CCC)C)CO)C)ccc2cc[nH]c2n1 92487,c1(C(=O)NCC2CCN(C(CC(C)(C)C#N)=O)C23CC3)nccc2n[nH]cc12 92488,c1(CC(N2C(CNC(C=CCC)=O)CN(C)CC2)=O)ccc2c(c1)COC2 92489,Cc1cccc(C(=O)C(=O)Nc2cccc(CNC(=O)CC(C)C)c2)c1 92490,c1(CC(C)(C)C)cn(CC(C)C(=O)NC)nn1.C(CC)OCCOCCOCC 92491,CP(C)(=O)c1ccc(C(=O)NC2C3CN(C(C45CCCC(C4)OC5)=O)CC23)nc1 92492,N1(C(=O)CCCC(F)F)CCC2(CCN(C(=O)C3=CCCC3)C2)C1 92493,N1(C(c2ncnc(C)c2C)=O)CCCC2(CCN(C(=O)COCC(F)(F)F)C2)C1 92494,c1(C(N2CCC(CN(C(C(F)OC)=O)C)C2)=O)cccc2ccc(O)nc12 92495,C1(C(=O)Oc2ccccc2)CCCN1Cc1conc1-c1ccccc1 92496,C1(C(=O)NCC2(CNC(C3(OC)CC3)=O)CC2)CCCC2(CCOC2)O1 92497,c1(CCC(N2CCC(OCCNC(c3c(CC)cco3)=O)C2)=O)c(C)noc1Cl 92498,Nc1ncnc2c1ncn2CCCCC(=O)Nc1cccc2c1ncn2C 92499,c1(CCC)nc(C)c(C(=O)NC2CC(NC(=O)C(=CC3CCCC3)C)C2)o1 92500,c1(CC(=O)NC(C)CCCNC(C2(C)CC2C)=O)ccccc1Br 92501,c1(C(=O)NC2C(C(=O)NCCn3ncc(C)c3)COC2)cncc(F)c1 92502,C(=O)(C(C)C(C)NC(=O)CCN(CCCO)C(c1cnns1)=O)OC 92503,CC(C(=O)N(C(C)CCNC(c1ccc(C2CCOC2)cc1)=O)C)C(C)(F)F 92504,C1(C(=O)NCC)CCCN1C(c1ccc(CNC(=O)CCCNC(N)=O)s1)=O 92505,C1(C)(CNC(c2ccn(CC(C)C)n2)=O)CCCN1C(=O)COC1CCCCC1C 92506,n1(CC)ccc(C(=O)N(C)CC2CCN(C(=O)C(C)COC)C2)c1C 92507,C1(C(=O)NCC2C(NC(CCN(C)CC)=O)CCCC2)CCC2CCCCN12 92508,C#CCCCCC(=O)N1CCN(C(=O)CC(C)c2ccccc2)CC1CCO 92509,C(CC(CC)C(=O)NC(C1CC=CCC1)C(=O)NC1CCCC(CO)C1)=CC 92510,S(=O)(=O)(c1c[nH]c(C(N2CC(CCNC(=O)C(O)C(C)(C)C)(OC)C2)=O)c1)NC 92511,N1(C(C(CC)(C)F)=O)CC(NC(c2ccc(CO)nc2)=O)C(N=[N+]=[N-])C1 92512,C1(C(=O)NC2CC(F)(CNC(c3ccc(CF)cc3)=O)C2)(OC)CCC(C)(C)C1 92513,Cc1cc(C(=O)NCc2ccc(C(=O)NCC3CCCCC3(C)C)s2)nc(C)c1 92514,N1(C(C(CC)=CC)=O)CCCC(CNC(C2CCCCC2C)=O)C1 92515,C(=O)(C1=CC2(CCN(C(c3ccc(C(C)C)o3)=O)C2)C1)NCc1ccc(SC)o1 92516,c1(NC)cncc(C(N2CCCC(CN(C(=O)Cc3ccnc(C)c3)C)C2)=O)c1 92517,c1(NCC2(F)CCN(C(=O)C=C3CCSCC3)CC2)ccc(Br)cc1[N+](=O)[O-] 92518,c1(C(=O)NC2C(CNC(C=CC(=O)OCC)=O)CCCC2)cc(OC)cc[n+]1[O-] 92519,C1(NC(CN(c2ccccc2)C(C)=O)=O)COCC1CNC(c1ccsc1)=O 92520,C1(NC(c2c(C)snc2)=O)CCCC(C(=O)NCCOCC(O)CO)CC1 92521,c1(CC)nn(C)c(OC)c1CN=C(NCc1n[nH]cc1C1CC1)NC1CC1 92522,N1(C(C2N(C(C3(CC)CC(C)(C)C3)=O)CCCC2)=O)CC(C2CCCCC2)C1 92523,c1(C(N2CCC(N(C(c3cnc(O)n3C)=O)CC)C2)=O)cccc2nccnc12 92524,c1(NCC(CC)(C)C)ncccc1S(=O)(=O)NCCC(F)(F)CC 92525,N1(C(C(CC)=CCCC)=O)CC(NC(C2(COC)CCCC2)=O)C(COC)C1 92526,N1(C(CS(CC)=O)=O)C2CCC1C(CNC(c1c[nH]cc(Cl)c1=O)=O)C2 92527,N1(C(C=CC=CC)=O)CCC(CC(=O)NC(CN2CCCC2)CC)C1 92528,N1(C(CCCCCC)=O)CC2CCCC2(NC(c2nnccc2C)=O)C1 92529,CCC(C)C(=O)N1CCC(N(C(c2occc2Cl)=O)CC)C1 92530,c1(CC2C(NC(COCCN(C)C)=O)CCC2)c(Cl)csc1Cl 92531,C=CCCN=C(NCC(C)C(F)(F)F)NCCc1ccc(C2CCCCC2)cc1 92532,C1(C(=O)NCC2CCCN(C(=O)C3=CCCCO3)C2)CC2CC1CC2(F)F 92533,CCC(C)(C(=O)N1CCC(F)(C(=O)NC(C)C(C)(C)C#N)C1)OC 92534,c1(C(N2CCN(C(C(C)=C(CC)C)=O)C(C)C2)=O)cc(C#N)ccc1Cl 92535,C1(C(=O)NC(CCN(C(=O)Cc2cccnc2)C)(C)C)OCCOC12CCC2 92536,Cc1ncc(C(F)(F)F)cc1C(=O)NCC1CCC1NC(c1ccon1)=O 92537,C1(NC(=O)C=CC2CCCO2)CCCCCN(C(C2(C3CCCCC3)CC2)=O)C1 92538,c1(C(=O)NCC(CN(C(=O)C2=CCOCC2)C)O)cnc2c(Br)cccn12 92539,N1(C(C(c2cn(CC)nc2)=O)=O)CCOCC(NC(C2CCC3CC23)=O)C1 92540,C(=O)(CCCC(=O)N(CC(C)NC(=O)C(O)CC1CCOCC1)C)N(CC)CC 92541,c1(C(c2nnnn2C)NCc2c(C(=O)OC)cc(Br)o2)cc(F)cc2c1OCC2 92542,N1(CC(=O)NCC2CCC(NC(C=C(C)C)=O)CC2)CCCCC(O)C1=O 92543,N1(C(C=NOC)=O)CC(NC(c2cnc(C)c(CC(C)C)c2)=O)CC(O)C1 92544,C1(CC(=O)NCCN(C(C)C)C(C23CC4CC2C3C4)=O)CCCN(C)C1 92545,CCC(C)(C)N(CC(C)NC(=O)CC1(OC)CCC1)C(=O)CC1(N(C)C)CC1 92546,C1(CC)C(C(=O)N(C)Cc2cnn[nH]2)CCCN1C(C1CC2(CC2)CO1)=O 92547,n1(CC(=O)N(C)CC2N(C(C(C)N(C)C)=O)CCC2)ccc2ccccc12 92548,Cn1cnc2c1CCC(C(=O)NCC1CC(NC(c3ccc(O)c(F)c3)=O)C1)C2 92549,C12(CC3(C(N4CCN(CCCC#C)CC4)=O)CC3)CC(C)(C1)OC2C 92550,C1(C(=O)NCCCNC(=O)OC)C2CCC(C2)N1C(C1CC2CC2C1)=O 92551,C1(C(N2CC(O)(CN(C(C3C(C(=O)OC)C3)=O)C)C2)=O)C(C)(C)C1(C)C 92552,N1(C(C(=O)NC(C)CN2CCOCC2)=O)CC2CCC1C1CNCC21 92553,C1(C)(CCC)CCN(C(=O)C(C)Cn2cccn2)C1.C1(=O)CC2(CC2)N1C 92554,Cc1ccccc1C(C)CC(=O)N1CC(O)(C(C)NC(c2nn[nH]c2Cl)=O)C1 92555,Cc1cccc2c1CCOC2C(=O)Nc1ccc(F)c(C#N)c1Cl 92556,CC1CC(CNC(C2CCC(F)CC2)=O)CN(C(=O)Cc2cncnc2O)C1 92557,c1(CC(=O)NC(CCNC(C(CCO)N(C)C)=O)C)cccc2c1CCC2 92558,CC1CN(C(C2CCC=CCC2)=O)CC1C(N1CCCC(CCO)C1)=O 92559,c1(OC)cc(NC(C2CC2NC(c2cccc(O)c2O)=O)=O)ccc1C 92560,CC(CCCCN=c1c(C#N)c[nH]c2ccccc12)NC(C1CC1C)=O 92561,Cc1cc(F)ccc1C(O)C(N1CCN(C)CC1CNC(=O)C=CC1CCC1)=O 92562,C1(C(=O)NCc2c(C(=O)NCCC3CCN(C)C3)scc2)CCC(=O)NC1 92563,Cc1c(C=CC(=O)NCCCCC(C)NC(C23CCC(CC2)CO3)=O)cnn1C 92564,C(C(C)(CC(C)C)NC(C1CCOCC1(C)C)=O)NC(c1cccc(C)n1)=O 92565,N1(C(CCSC)=O)CC2CCCC(CNC(=O)CN3CCn4nccc43)C2C1 92566,C(C)(C)(CC(=O)N1C(C(=O)NCC2CCC2(F)F)CCC1C(C)C)OC 92567,S(=O)(=O)(c1c[nH]ccc1=NCCC1CC1F)NCCCCN(C)C 92568,N1(C(C2C(C)CC=CC2)=O)CCN(C(=O)CCn2ccccc2=O)CC1CCO 92569,n1(CC)ccc(=NC(=O)C2(C(C)C)CCN(C(c3ncc[nH]3)=O)C2)[nH]1 92570,N1(C(CCN(C(c2c(CC)cco2)=O)C)=O)Cc2n[nH]cc2C1CO 92571,c1(C(=O)NCCC(=C)CNC(=O)C=CC=CC)[nH]c(O)nc1C 92572,Cc1nc2sccn2c1C(=O)NCC(O)CNC(C1C2CCC1CC2)=O 92573,C12(NC(C3CN(C(C)=O)C3)=O)CC(CNC(C3CCOC3=O)=O)(C1)OC2C 92574,C1(CCn2cc(COC)nn2)CCN(C(=O)C(=O)NCCC(N)=O)CC1 92575,N1(C(c2ccc(C=C)cc2)C(=O)NC2CCCCC2)CCC2(CCCO2)CC1 92576,C1(C(N2CCC(C)(CNC(=O)C3=NNC(=O)C3)C2)=O)CCc2nccn2C1 92577,c1(C(=O)NCCN(CCC)C(c2c(C)nsc2C)=O)cc2c(C)c(C)ccc2[nH]1 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92596,C1(CNC(CN(CC(C)C)C(C2CC2(C)C(F)F)=O)=O)CNC(=O)CO1 92597,CC1CCCC=C1C(=O)NCC(C)(C)C#CC(=O)N1CCC(N(C)C)CC1 92598,N1(C(C2CN(C)C2)=O)CC2COCC(C1)C2NC(C1CCC2(CCOCC2)O1)=O 92599,N1(CCC)CC2(CN(C(c3c[nH]cc3C)=O)C2)C1 92600,C12(C(=O)NC(CC#C)CC)CC1CCN2C(c1c[nH]c(C)c1)=O 92601,C(=O)(CCC(CC)(CC)[N+](=O)[O-])NCC1(SC)CN(C(C2CCN(CC)C2)=O)C1 92602,C1(C)(C(=O)NCCN(CC=C)C)CCN(C(C2CC2[N+](=O)[O-])=O)C1 92603,c1(C(N(c2ncc(C3CC3)s2)CC)=O)c(C)cc(C)cc1C 92604,C(c1ccccc1F)=CCC(=O)NC(C1N(C(C(CCOC)C)=O)CCC1)C 92605,CN1CCC(CC(=O)NC2(C)CCN(C(C3CCOC3)=O)C2)C1=O 92606,N1(CCOC)CC(C(N2CCC(NC(=O)CCSCC(C)C)C2)=O)CCC1=O 92607,CC1OCCOC1C(=O)NC1C=CC(CC(=O)NCc2ccsc2)C1 92608,C1(CC(=O)NCCC(CNC(=O)CCOc2ccccc2)O)CCCC(=O)N1 92609,C1(CCCC)CCN(C(=O)NCC2(C)CCN2C(=O)OC(C)(C)C)CC1 92610,c1(C(=O)NCC(CNC(c2c(CC)sc(=N)[nH]2)=O)(C)O)cnc2ncnn2c1C 92611,C1(CC(=O)OCC)CN(C(C)C(N2CCC(N3CCCCC3)CC2)=O)CCO1 92612,N1(C(N(CCCC)CCCC)=O)CCCC(c2nc(O)n[nH]2)C1 92613,CC(C)(C#N)CCC(=O)NC1CN(C(c2cc(F)c(F)c(F)c2)=O)CC12CC2 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92631,N1(C(COCCC)=O)CCC(O)(C(C)NC(c2cnc(N(C)C)c(Cl)c2)=O)CC1 92632,c1(CC)ccc(C(=O)NC(CC2CCOCC2)CO)nc1C 92633,c1(C(N2C(C)C(NC(=O)Cc3csnn3)C(C)CC2)=O)ccc2ncccc2n1 92634,Nc1ccc2ccccc2c1-c1ccccc1Cl 92635,c1(OC)cc(C)ccc1NC(=O)C(=O)NC1(CO)CC(C)C1 92636,c1(CNC(c2c(OC)cc(Br)cc2)CO)n[nH]c2c1CCCCC2 92637,N1(C(c2[nH]cc(CC)c2)=O)CCN(C(c2nc(Cl)c(Cl)s2)=O)C2COCC12 92638,CC1CN(C(=O)CSc2nnc(S)s2)CC(C)C1NC(c1cccc(=O)o1)=O 92639,c1(OC)cc(CC(N2CC3(CCN3C(c3csnn3)=O)C2)=O)ccc1C 92640,C(=O)(CC(F)(F)C(F)(F)Br)NCC(C)NC(c1ncc[nH]1)=O 92641,C1(C(N(CC(C)CNC(c2ccc(CCO)cc2)=O)C)=O)C(C2CC2)C1(F)F 92642,N1(C(C(C)C)=O)CCOC(CNC(C2CCOC(=O)N2)=O)C1 92643,CCCC(O)C(=O)N1CC(O)CC1CNC(=O)CCC1OCCO1 92644,c1(OCCC(C)C)cc(=NC(=O)c2ccn(C3CC3(F)F)n2)[nH]o1 92645,Cc1cc(C(F)(F)C(=O)NCCN(C2CCCC2)C(=O)CC2(O)CCCC2)cs1 92646,C12(C(N3CC(C#C)(N(C)C)C3)=O)CCC(CN(C(=O)C(C)CCOC)C1)C2 92647,N1(C(C=NOC)=O)CC2(NC(=O)COCC3CCCCO3)CCCC2(F)C1 92648,N1(C(C2C(C=C)C2)=O)CC(CNC(c2cc(C(C)(C)C)n[nH]2)=O)C2(CC2)C1 92649,C(=O)(C1=NOC(CN(C(=O)C(C#N)C(C)C)CCCO)C1)OCC 92650,c1(OCC)ccc(C(N2CC(c3cc(OC)ccc3O)C2)=O)cc1Cl 92651,C1(OC)CC(NC(C2(Br)CC2)=O)CN(C(c2ccccc2C2CCOC2)=O)C1 92652,CCCC(CCCNC(C1CCN1CC)=O)NC(c1cccc(Cl)c1N)=O 92653,CCCC(C(O)C(=O)NCc1nnc(CC)s1)NC(=O)CCN(C)C 92654,O(NC(=O)CCN(C(=O)C(C(C)C)OCC)CCO)CCCC#C 92655,C(N=c1cc(NCc2ccnnc2)nc[nH]1)C1(OC)CCSC1 92656,c1(CC(N2C(CCNC(=O)C(O)c3ccsc3)COCC2)=O)cn2ccsc2n1 92657,C=Cn1nncc1C(=O)NC(CN(C)C(c1occc1COC)=O)(CO)CO 92658,c1(OC)ccc(N2CCN(C(C)C(=O)NC(C3CCC3)C)CC2)c(F)c1 92659,N1(C(=O)NCCC(=O)OC(C)C)CC2CCCCC2(CCC(=O)O)C1 92660,N1(C(CNC(CC)=O)=O)CCCC(N(C(=O)C(CO)NC(N)=O)CC)C1 92661,Cc1sc(C(F)(F)F)nc1C(=O)NC1CN(C(C2CCCOC2)=O)CC1C 92662,c1(C(=O)NC2CCN(C(C3CCN(C(C)=O)C3)=O)CC2)ccc(O)nc1C 92663,C1(CNC(CCNC(N)=O)=O)CC2CN(C(c3cc([N+](=O)[O-])c[nH]3)=O)CC12 92664,N1(CCCN2CCCC(C(=O)OC)C2)CCCc2c1ccc([N+](=O)[O-])c2F 92665,C1(NC(C2CCCN(CCC)C2)=O)CCCCN(C(c2ccco2)=O)CC1 92666,C1(NC(C(CC=C)c2ccccc2)=O)CCCN(C(C2CCC(=O)N2)=O)C1C 92667,Cc1ccc(CC(=O)NC23CC(CNC(=O)CC4CC(C(F)F)C4)(C2)C3)c(Cl)n1 92668,CC1(C(N2CCOC(CCNC(=O)COc3cccnc3)C2)=O)CNC(=O)C1 92669,C(=O)(C(C)(C)CCCO)N1C(CN(C(C2CN(CC)C(=O)C2)=O)C2CC2)CCC1 92670,CC1CN(C(C2CC3CC3C2)=O)CC1(C)C(=O)N(C1CCC2(CC1)CC2)C 92671,CCC(CC(=O)N1CC(C)(NC(C2CC(CC(F)F)C2)=O)C1)CC(F)(F)F 92672,CCCCCC(C)(C)C(=O)NCC1CCC(C(N2CCOC(C(=O)OC)C2)=O)C1 92673,c1(C(=O)NCC23C(CN(c4ccnc(N(C)C)n4)C2)C3)c(Cl)cccc1[N+](=O)[O-] 92674,CCC(CNC(=O)C(c1cccs1)NC(=O)C(C)C1(O)CCC1)CC 92675,C1(CCCNC(C(C)C)=O)CCCCN1C(c1cn(C2CCOC2)nn1)=O 92676,c1(OC)ccc(OCCNC(c2nnnn2CCCSC)c2ccns2)cc1 92677,C1(CNC(c2ccc(C)o2)=O)CC(NC(=O)CN=S(C)(C)=O)C12CCC2 92678,CC(CC(=O)N1CC(CNC(=O)CCNC(=O)CO)C(F)(CO)C1)C(C)(C)C 92679,CCC(CC)(C(=O)OC(C)(C)C)C(=O)N1CCN(C(c2nccn2C)=O)C2CC12 92680,CC(CC(=O)O)(c1ccc(F)cc1)n1cc(C2(COC)CC2)nn1 92681,c1(N(C)C)cc(C(=O)NC2CCC2CNC(=O)CCCc2ccsc2)ccc1Cl 92682,C1(NC(CCC=C)=O)CCN(C)C12CCCN(C(=O)CC1CC(=O)NC1=O)C2 92683,c1(C(=O)NCCN(CCOC)C(c2c(C)nn(C)c2C)=O)c(C)nc(C)nc1C 92684,C1(NC(C(=O)Nc2nnc(SCCOC)s2)=O)CN=C(C(F)(F)F)O1 92685,N1(C(Cc2cn(CC(C)NC(C(=O)NCC)=O)nn2)=O)CCCC(C(=O)OC)C1 92686,c1(C(=O)NC(C(C)C)CNC(=O)CCCc2cncs2)cnc2[nH]cncc1-2 92687,C1(C(C)(F)F)(NC(C(C)Sc2ccccc2)=O)CCCCC1 92688,c1(C(=O)NC2(C(=O)NC(C(=O)OC)C3CCC3)CCCC2C)cncc(C=C)c1 92689,CC(C)CC(CNC(=O)C(C)(C)C1(C)CC1(F)F)NC(=O)COC1CCC1 92690,c1(OC)cccc(NC(=O)C(c2ccc(Br)nc2)N(CCC#N)CCC#N)c1 92691,CC(CC(C)(C)C)C(=O)NC1(CCO)CN(C(=O)CC2NC(=O)NC2=O)C1 92692,C1(C(=O)NC(c2nc(C)[nH]n2)CO)CN(C(c2nonc2N)=O)CC1(F)F 92693,Cc1nn(C)cc1CC(N1CCC(CN(C(=O)COCCc2cccs2)C)C1)=O 92694,N1(C(C2C(CC)C2)=O)CC2CCC(NC(C3(CCOC)CC3)=O)CC2C1 92695,C1(C(N(C)CC2N(C(C(C)OC3COC3)=O)CCC2)=O)CCS(=O)(=O)C1(C)C 92696,C1(CNC(C2(CC(C)C)CCNC2=O)=O)COCCN(C(C2(F)CC2)=O)C1 92697,C1(NC(c2[nH]cc(CC)c2)=O)C(C)CCN(C(=O)CC2CCCC(C)C2)C1C 92698,c1(NCC(=O)NC2(CO)CN(C(c3ccc(OC)cn3)=O)C2)ccc(F)cc1F 92699,N1(C(C23C(C)(C)OC(CO)(C2)C3)=O)CC2(CCC(NC(=O)C(F)C3CCC3)CC2)C1 92700,c1(-n2c(C(C3CC4CCC3O4)NCCCCC)nnn2)ccc(OC(F)F)cc1 92701,Cc1ncncc1C(N1CC(O)(C(C)(C)CNC(C2(C)CCN(C)C2)=O)C1)=O 92702,c1(CC=C)cccc(C(=O)NCC2(COC)CN(C(=O)C(O)CSCOC)C2)c1 92703,Cc1cc(Cn2ccnc2-c2cccnc2-c2n[nH]c(C)n2)cc(C)c1 92704,Cc1nccc(C(=O)NC2CCC2NC(c2ccn(C3CC3)c2C)=O)c1O 92705,C1(NC(C(COC)(C)OC)=O)CC2(C1)CN(C(=O)C(C)n1cccn1)C2 92706,N1(C(C2CC(O)(CC#C)C2)=O)CC2(CNC(=O)C(=O)N(C)C)CC1CCO2 92707,C1(C(N(C)Cc2nccs2)=O)CCC(n2cc(-c3cnccn3)nn2)CC1 92708,N1(C(CCC(C)c2ccccc2)=O)CC2(C1)CN(C(C13CC(CO1)C3)=O)C2 92709,C1(NC(C2CC(OC)C2)=O)(CO)CCCN(C(=O)COCCCN(C)C)C1 92710,N1(C(C(C)NS(CC)(=O)=O)=O)CCCC(C2(NC(=O)C(F)C(C)C)CC2)C1 92711,c1(SC)nccc(N2CCC(CF)(NC(c3cc(Cl)n(C)n3)=O)C2)n1 92712,CC(C)C(O)CCN=c1nc2c(cnn2C)c(NCCc2ccc(N)cc2)[nH]1 92713,C1(CNC(c2[nH]ccc2CNC(C23CCCC2C3)=O)=O)CCC2(CC1)CC2 92714,Nc1c(F)ccc(Cl)c1C(=O)NC1CN(C(c2cc(Cl)c(F)cc2F)=O)CC1O 92715,C=CCCC(CC(C)C)C(=O)NCC(C)(C)OCC(=O)NCCC(CCC)SC 92716,C1(NC(CCSCC(C)C)=O)CCCN(C(C2CCCC2O)=O)CC1 92717,N1(C(c2ccc(C(F)(F)F)cc2)=O)CCc2cc(-c3cc(F)ncc3F)ccc2C1 92718,C#Cc1ccc(CC(=O)NC2CCCC2NC(=O)C(C)CCCOC)cc1 92719,C(c1ccccc1)=CCC(=O)N(C)C(N(CC(N1CCCC1CCCO)=O)C)=O 92720,C1(C(=O)NC(CC)C(F)(F)F)CCCCN(C(=O)Cc2csnc2C)C1 92721,C#CC1(NC(=O)CSCCNC(=O)Cc2cc[nH]n2)CCCOC1 92722,C(=O)(CCCCCCC)N1CCC(CC#C)(C(=O)N(CC(O)C(C)(C)C)C)C1 92723,C1(NC(c2c(C)nccn2)=O)CC2(NC(C3CC(O)C3)=O)COC1C2 92724,CC(CCO)C(=O)N1CCC(CNC(c2ccc(SC(C)C(N)=O)cc2)=O)CC1 92725,CCCC(C(O)C(=O)NCC(C)(C)CC(C)O)NC(=O)CCS(N)(=O)=O 92726,N1(C(CCc2ccc(C)nc2)=O)CC(O)CC1(C)CNC(=O)C=CC(C)(C)C 92727,C1(C)(C(N(CCC)CCOC)=O)CC12CCN(C(=O)CCCC(=O)C1CC1)CC2 92728,N1(C(=O)CN2CC=CC2)CC(NC(C23COCC(C2)C3)=O)CC(O)C1 92729,O=S1(=O)CC2CC(N=c3ccn(CCCSc4ccccn4)[nH]3)CC2C1 92730,C(=O)(C1=NOC2COCC12)NCC(C(=O)N(CC)Cc1cnccn1)(F)C(C)C 92731,C1(C2(O)CN(C(=O)C=C3CCOCC3)C2)(CNC(C2CN(C)C(=O)CC2)=O)CC1 92732,CCC(C)C(C)(O)CNC(=O)CN(C1CC(C#N)C1)C(c1ccnc(O)c1)=O 92733,c1(C(N(CC(CNC(CC(C)SC)=O)C)C)=O)cc(Br)ccc1N 92734,C1(C(N2CCc3sc(-c4ccnc(F)c4F)nc3C2)=O)Cc2ccccc2CN1 92735,N1(C(=O)CCC2CC(F)(F)C2)CCN2CCN(C(=O)C(F)C(F)(F)F)CC2C1 92736,c1(C(N(CCNC(c2cc(CN(C)C)on2)=O)CC2CC2)=O)cn(C)ccc1=O 92737,CC(CCNC(C1(C)CC1)=O)CCNC(=O)C(C)(C)Cc1cnn[nH]1 92738,c1(C(N2CCC(NC(C(c3cc(C)cc(F)c3)C)=O)C2)=O)cnn2c1OCCC2 92739,c1(N(C)Cc2ccn(CC)n2)ccc(S(=O)(=O)NC(C2CCN(C)CC2)C)cn1 92740,Cc1cc(CCCCO)ccc1NC(=O)CC(C(C)C)c1ccccc1 92741,Cc1c(C(=O)NCC2CN(C(C3CCC4CC4C3)=O)CCCO2)cncc1Cl 92742,C12(NC(c3c(C)cc(C)[nH]3)=O)CCN(C(=O)Cc3cncnc3O)CC1C2 92743,C(CCCC(C)C)NC(C(C1CN(C(c2scc(OC)c2)=O)C1)O)=O 92744,c12ccc(cc1)NS(=O)(=O)C2.O(NC(=O)COC)CC 92745,C1(CNC(=O)CCOC2(CNC(CCOCCOC)=O)CC2)CCCOC1 92746,C(=O)(C(C)(C)C(=O)OC(C)C(=O)Nc1c(CC)cccc1C(C)C)OCC 92747,c1(CNC(C(=O)Nc2c(C(=O)OCC)cccn2)=O)n[nH]c2c1CONC2=O 92748,c1(C(N2C(CNC(C(CCCC)O)=O)CC(F)(F)C2)=O)cc2c(=O)[nH]ccn2c1 92749,N1(C(c2n(CC)ncc2)=O)CCN(C(=O)C(c2cccc(Cl)c2)SC)CC12CC2 92750,C1(NC(C2(NC(C=CCOC)=O)CC2C)=O)CC12CC(O)C2 92751,c1(NC)scnc1C(N1CCC(C(C)C(=O)NC)C1)=O.C1C(C)N1C(C)C 92752,CC(C(=O)NC1CC(c2ccccc2)(NC(C2COC(=O)N2C)=O)C1)C(F)F 92753,N1(C(c2n(C(CC)C)ncc2)=O)CCCN(C(C2(CC3CC3)CC2)=O)C(C)C1 92754,c1(OCC)ccc(C(N2CCC3C(C2)N3C(c2ccc(Br)nc2)=O)=O)cc1OC 92755,N1(C(C(CC)O)=O)C2CCC1CC(NC(c1cccc(N)c1C)=O)C2 92756,N1(CCSc2cn(CC(=O)N(C(C(N)=O)C3CC3)C)nn2)CCCC(CCO)C1 92757,c1(C(N2CC(NC(c3cc(CC)on3)=O)C2)=O)c(Cl)cc(C)cc1Cl 92758,N1(Cc2nc(CCOC)on2)CCC2(NC(=O)CC3CCCC(=O)N3)CCCC12 92759,CN=c1nc(N2CCCC(C)CC2)[nH]c(=NCCS(=O)(=O)C(C)C)[nH]1 92760,c1(OC)ccc(Br)c(C(=O)NCC2CCN(C(C3CNC(=O)C3)=O)CC2)c1 92761,c1(N(CCOCC)C)nnc(C2CCC(=O)N2)n1Cc1sccc1C 92762,C1(NC(C2(COC)CC2(F)F)=O)CCCCC1NC(=O)C(CCO)N(C)C 92763,N1(C(C2C(C(C)C)CCO2)=O)CC=CC(C(N2CCCC2CC(C)(C)C)=O)C1 92764,CCC(C)C(C(=O)N1CC=CC1(C)C(=O)NC(c1cn[nH]c1)C)N(C)C 92765,C(=O)(CCCCCCOC)N1CCC(COC)(NC(c2csc3nccn23)=O)C1 92766,c1(C(=O)NCCN(C(=O)Cc2csc(Cl)c2)CC)ccc(-c2cc[nH]n2)s1 92767,N1(C(=O)CCOc2cc(F)ccc2F)CCC2(CCN(c3cnc(F)cn3)C2)C1 92768,c1(C(=O)NCC2CC(C)N(C(C3CCCC(C)C3)=O)C2)cccc(=O)n1O 92769,Cc1sc(Cl)nc1C(N1CC(C(C)NC(=O)C(C)Cc2cccnc2)C1)=O 92770,N1(C(c2c(C)cns2)=O)CCC2CCC12CNC(C1(N2CCCC2)CCC1)=O 92771,C1(NC(C(C)(Cl)Cl)=O)COC2(CCN(C(C3CCn4ccnc4C3)=O)CC2)C1 92772,C1(C)(NC(C(C2CCOCC2)C)=O)CCN(CCOc2cccnc2)C1 92773,c1(CN2C(C(=O)Nc3cccc(C4(C(=O)O)CC4)c3)CC2)ccc(Cl)c(Cl)c1 92774,C1(C(=O)NCC=CCNC(c2cnc(O)s2)=O)(C(F)F)CC(F)(F)C1 92775,Cn1cccc1CCC(=O)NCCCCCNC(=O)C(C1CCOCC1)F 92776,C(=O)(C(C)(C)C(C)C)NCCCCC1(NC(CC(=O)NCC)=O)CC1 92777,CC1(C)C(C(c2nnnn2C2CC2)NCCn2ccnn2)C1(C)C 92778,CCN=C(NCC1CCCO1)NCCNC(c1ccc(Br)cc1)=O 92779,c1(C(=O)NC(C)(C)CCNC(=O)OC(C)(C)C)ccc(C(=O)O)cc1C#N 92780,C1(C2CC2)(C(N2C(CC(N)=O)CCC2)=O)CN(C(c2ncn3c2CCC3)=O)C1 92781,c1(C(N2CC(C(N)=O)(CNC(C3(F)C(C)OCC3)=O)C2)=O)scc2c1CCCC2 92782,O=S(=O)(c1c[nH]ccc1=NC1CCCCCC1CCO)NCCN1CCSCC1 92783,C1(CNC(=O)Cc2sccc2F)COCCN(C(=O)CCCc2cccnc2)C1 92784,C1(NC(C(c2cn(C)nc2)O)=O)CCCC2CN(C(c3cc(F)n(C)n3)=O)CC12 92785,c1(C(=O)NC2C(NC(c3nn(C)c(Br)c3)=O)C2)ccn2ccsc12 92786,C12(C(N3CCC(O)(CNC(C=C(CC)C)=O)C3)=O)CCC(C1)C(C)(C)O2 92787,c1(N2CCN(C(C)=O)CC2)nc2c(F)cc(F)cc2c(=NC(C)c2nc[nH]n2)[nH]1 92788,C(CNC(C1CC2CC2C1)=O)(CC(F)(F)F)NC(CSc1n[nH]c(=N)s1)=O 92789,N1(Cc2cccc(OC)c2C)CC2CN(C(c3ccc(N(C)C)nc3)=O)CC2C1 92790,C12(C(=O)NCC3(CNC(=O)C=Cc4cncs4)CCCC3)OCCCC1C2(F)F 92791,C1(NC(c2n(C)c(Cl)cn2)=O)CCN(C(c2c(F)cccc2Cl)=O)CC12CCC2 92792,c1(NC(=O)NC)ccc(F)c(Nc2cc(C(=O)OC)nc(C3CC3)n2)c1 92793,N1(C(=O)CCc2ccccc2)CCCC(CO)C1.c12cnn(c1)C1CN(C1)C2=O 92794,C(c1ccccn1)=CC(=O)NCCC(=C)CNC(=O)CC(C)c1ccncc1 92795,C12(C(=O)NCC(CNC(c3c(C(C)C)n(C)nc3)=O)(C)O)CCC(C1)OC2C 92796,c1(NC(c2scc(CC)n2)=O)ncnc2c1ncn2C1CC(O)C(O)CC1OC 92797,N1(C(CNC(CC)=O)=O)C2CCC1CC(CNC(=O)CC13CNC(=O)C(C1)C3)C2 92798,Cc1[nH]nc2c1CCC(C(=O)NCCc1coc3ccccc13)C2 92799,c1(C(N2CCCC(NC(C3(CC=C)CC3)=O)C2)=O)c[nH]c2cc(Br)ccc12 92800,CC1=CCCC2CN(c3ncc(Br)cc3OCCO)CC12 92801,CCC1=NOC(C(N2CCC(C(C)(C)C(=O)NCCCc3nccs3)C2)=O)C1 92802,c1(C(C)OCC)nc(C(=O)NC(C)CC2CN(C(c3cc(Cl)cs3)=O)C2)cs1 92803,N1(C(C(C)N2CCCC2)=O)CC2C=CC1C(C(=O)NCCc1cn(C)cn1)C2 92804,O=C(C1=CCCOCC1)NC(CO)C(=O)NCCCc1cnn[nH]1 92805,N1(C(C(C2CC2)SC)=O)CCN(C(c2cc(C)nc(C)c2)=O)C(C2CC2)C1 92806,C(=O)(CC(C)CNC(=O)C(C)(C)CC1CC1)NC(c1ncc(C)o1)C 92807,N1(C(=O)NC2CC2c2ccc3c(c2)CCC3)C2CCC1CC(C(=O)NC1CC1)C2 92808,C1(C)(NC(C2(C(C)=O)CC2)=O)CCN(C(=O)C(C)(C)NC(c2ccccc2)=O)C1 92809,N1(C(CCCCCC#C)=O)CC2CCCC(NC(C3CCNC3=O)=O)C2C1 92810,c1(CC(=O)NC2CC2NC(c2cc3scnc3[nH]2)=O)cccc(F)c1Cl 92811,c1(CC(=O)NCCOC2CCN(C(c3cc(C)no3)=O)C2)ccccc1S(C)=O 92812,c1(C(C(F)(F)F)NCC(c2n(C)cnc2)O)cccc(C(F)F)c1 92813,c1(NC(C=Cc2c(C)n(C)nc2)=O)ccc2c(c1)C1(CCCCC1)C(=O)N2 92814,c1(N(C2CN(C(c3cc[nH]c3C3CC3)=O)C2)C)cc(O)nc(O)n1 92815,c1(CNC(c2ccc(CN(C(=O)CC(F)(F)F)C)o2)=O)ccc2c(c1)sc(=O)n2C 92816,c1(N2CCC(N(C)C(C3(C)CCC(=O)N3)=O)CC2)ncc([N+](=O)[O-])c(=N)[nH]1 92817,C(=O)(CCC(C)C#N)NCC1CC(NC(c2c(CC)nn(C)c2)=O)C1 92818,C1(C)(C(=O)NCC(CNC(C2CC(CC)(CC)C2)=O)C)CCC(C)C1 92819,C(=O)(CCC(C)(C)NC(=O)C1=C(Cl)CCC1)NCC1CC(CC)C1 92820,Cc1ccc(O)nc1CNC(=O)CC(C)(C)CNC(C1OCCC1C(C)C)=O 92821,C(C(CC(F)(F)F)C(=O)O)n1cc(-c2ccc(F)cc2OC(F)F)nn1.CC=O 92822,CC(C)C(C(=O)NCC1(F)CN(C(c2nc(=O)n(C)[nH]2)=O)C1)NC(N)=O 92823,Cc1cc(C)c(C(N2CCCCCC2CNC(c2nccnc2N)=O)=O)cc1N 92824,c1(C(=O)NCC2CC(OC)CN2C(C2CCCCC2)=O)cc(Cl)cc([N+](=O)[O-])c1 92825,c1(C(=O)NCC(CC)(CC)NC(=O)C(C(C)(C)C)NC(N)=O)cc(C)nnc1O 92826,c1(OC)cc(N)c(F)cc1CSc1ccc(OCC2Sc3ccccc3O2)cc1 92827,C(=O)(C(C)(C(C)C)OC)N1CCC(CCNC(CC(C)SC)=O)CC1 92828,c1(C(N2CCN(C(C(CC3CCC3)C(=O)OC)=O)CC2)=O)ccnc2ccsc12 92829,C1(NC(C(CC)CO)=O)CC2(CCN(C(C3C=C3C)=O)C2)C1 92830,C1(CNC(Cn2c(CCC)nnc2S)=O)CCN(C(=O)C2=CC(C)(C)C2)C12CC2 92831,c1(C(=O)NC(C2(O)CCN(C(Cc3nc(C)[nH]n3)=O)C2)C)cccc2cncn12 92832,C(=O)(C(C)(C)CS(C)(=O)=O)N1CC(O)(CNC(c2c(CC)cccc2)=O)C1 92833,c1(NC(C2CC3CC3N2Cc2cocn2)=O)ccnc2cc(Br)ccc12 92834,Cn1nc(C(F)(F)F)cc1C(N1CCC1CNC(=O)CC1CCCS1(=O)=O)=O 92835,CC1CN(C(C2(CO)CCOCC2)=O)CC(C)N(C(=O)CCc2cc(Cl)no2)C1 92836,c1(C(=O)NCC2C(NC(C3(C(N)=O)CCC3)=O)C2)cccc(F)c1F 92837,C=CCCCCC(=O)NC(C)C(C)NC(c1cc(C2CCCCC2)on1)=O 92838,c1(OC)ccccc1C1CC1C(=O)NCCC(C)(C)NC(C1C(Cl)(Cl)C12CC2)=O 92839,N1(C(C(CC)F)=O)CCN(C(C2CC(N(C)C)C2)=O)CC1c1cnn(C)c1 92840,c1(CNC2CCC(C)CN2C(=O)OC(C)(C)C)nnc2n1CCOC2 92841,Cc1cc(CNC(c2[nH]ccc2C2CC2)=O)oc1C(=O)NCC(C)(O)C1CC1 92842,C1(C(C)C)N(C(C2(CO)CCN(C(c3ccc[n+]([O-])c3)=O)C2)=O)CC1(C)C 92843,N1(CCNC(c2n(CC)ccn2)=O)CCCN(C(c2nn(C)cc2Br)=O)CC1 92844,C(=O)(C(CC(C)(C)C)OC)NC1CC2(CC(NC(CN(C(=O)OC)C)=O)C2)C1 92845,C1(CC(C)C)CC(NC(=O)C(N2CC(c3ccccc3)C2(C)C)=O)CCO1 92846,C1(NC(=O)NC2CCN(Cc3ccccn3)C2)CC2(CCC2)CO1 92847,c1(SCC#C)cccc(C(=O)NC(C)CCCNC(=O)C(C)OCC(C)C)c1 92848,N1(C(c2n(C)ncc2)=O)CCC(C2(NC(c3coc(C(F)(F)F)c3)=O)CC2)CC1 92849,CC1=CCN(C(C2CC(N(C)C(c3ccoc3C)=O)C2)=O)CC1 92850,c1(C(=O)NC2(CC(=O)NC3CC(C)(COC)C3)CCCCC2)n[nH]c2c1CCC2 92851,C1(CC(=O)NCC2CN(C(C3C(C=C)C3)=O)C2)CC2(CC2)C1 92852,Cc1cnc(F)c(CNC(=O)C(CCC(C)C)NC(=O)C2=CCCCC2)c1 92853,N1(C(CN(C2CCC2)C)=O)CCCCC12CN(C(C1(c3ccno3)CC1)=O)C2 92854,c1(NC)cnc(Cl)cc1C(=O)NC(C1CCN(C(C2CCCC(=O)N2)=O)C1)C 92855,c1(SC)nc2nc(C)c(CC(=O)NCCC3COCCN3C(=O)CO)c(C)n2n1 92856,C1(C(=O)NC(C#C)CC2CCCC2)C2CC3C(C2NC(c2cc(CO)[nH]n2)=O)C13 92857,N1(C(C(C)OCC)=O)CCc2ccccc2C1CNC(=O)Cc1ccsc1Cl 92858,c1(NC(=O)NC(CC)COCC(F)(F)F)cc(OC)c(Br)cn1.c1cccc(C)c1 92859,c1(C2(C(=O)NC(C(C)NC(C3CN(C(C)=O)C3)=O)C)CCC2)cccnc1 92860,Cc1cc(C(N2CCC(NC(c3cc(-c4ccccc4)co3)=O)C2)=O)cs1 92861,N1(C(C2CCC(NC(C3CC(C)(F)C3)=O)C2)=O)CC(CO)C(CO)C1 92862,N1(C(COc2cc(C)cc(C)c2)=O)CCN(C(=O)C=Cc2cocn2)C(C)C1C 92863,C=CCCCCC(=O)N1CCCOC(CCNC(=O)CC(C)NC(N)=O)C1 92864,c1(C(=O)NC2CCC(OC)C2)cnc2ccsc2c1 92865,N1(C(=O)OC)CCC2(CC1)CC(C(=O)N1C3CCC1COC3)c1ccccc12 92866,C1(O)(CNC(C(CO)N(C)C)=O)CCN(C(c2nn(C)cc2C(F)(F)F)=O)C1 92867,C1(CN(C(COCCCC(C)C)=O)C)CN(C(C2CCCCS2)=O)CCO1 92868,Cc1nnc2cc(N3CCN(C(C4CCCC(C)(C)C4)=O)CC(O)C3)ncn12 92869,c1(OC)cncc(C(C(=O)NC2CC2)N(c2c(C)cccc2Cl)CC2CC2)c1C 92870,c1(C(=O)NCC(CC)NC(C2N(CCC)C(=O)CC2)=O)ccc(F)c(C)c1Cl 92871,c1(C(N(CCN(C)Cc2nnc(CO)s2)C)=O)cc(Br)c[nH]1 92872,CC1CCN(C(=O)C=CBr)C1CNC(=O)C=CC1CCOC1 92873,c1(NCC2(CC)CCCCC2)nc(N(C)CC2CCCO2)cc(C)n1 92874,Cc1ccc(C(=O)NC(C(=O)NCC2CC(F)C2)c2cccs2)[nH]1 92875,C1(NC(CC2C(NC(C=CC(C)C)=O)CCC2)=O)CC(O)C12CCC2 92876,C1(C2CCN(C)CC2)(C(=O)NC(CC)CNC(=O)CCC2CC2(F)F)CC1 92877,C(=O)(C1=C(Cl)CCCC1)NCC1C2CN(C(CCNC(=O)NC)=O)C1C2 92878,O=S(=O)(c1cccc(=NCC2=NOCC2)[nH]1)NC1COCC1N1CCCCC1 92879,CC(C)CC(C)C(=O)NC1C=CCN(C(c2ccnc(Cl)c2O)=O)C1 92880,c1(C(=O)NC(CC=C)CNC(=O)CCc2nncs2)c(Cl)cccc1Cl 92881,C(=O)(C(C)(O)C(C)(C)C)NCC(CN(C(=O)CSc1ccccc1[N+](=O)[O-])C)O 92882,Cc1cc(C(=O)NC2CN(C(c3cncnc3C(C)C)=O)CC2O)c(C)s1 92883,n1(CCC(=O)OCc2cccc(OC)n2)nc(C)c(C)c1C 92884,N1(C(C(CNC(C2(C)CCCO2)=O)O)=O)CCCc2occc2C1 92885,N1(C(C2(COC)CCOCC2)=O)CCC(CNC(=O)CCF)(COC)CC1 92886,c1(C(C(=O)NCC2CN(C(C(c3ccc(F)cc3)OC)=O)C2)C)cccc(F)c1 92887,c1(C(=O)NCC2CN(C(C3(Cl)CCC3)=O)CC2(F)F)cnn2c1CCC2 92888,N1(C(Cn2ncn(C)c2=O)=O)CCCC1C1CCCN1C(=O)OC(C)(C)C 92889,c1(C(=O)NCC2C(CC(=O)NCC(CC3CC3)OC)C2)ccn(CC)c1C 92890,C1(NC(c2cnc(OCC)s2)=O)CN(C(c2ccn(CCF)n2)=O)CCC1CO 92891,C12(C(N3CC(C(C)NC(=O)CCCN(C)C)C3)=O)CCCCC1C2 92892,Cc1c(CNC(=O)C=CCC(C)(C)NC(=O)Cc2cccnc2O)nnn1C 92893,C1(NC(c2ccc(C(C)C)s2)=O)CCC(NC(=O)CCC2CCCCN2C)CC1 92894,N1(c2nccc(N3CCC(C)CC3)n2)CC(NC(C2C=CCCC2)=O)CCC1C 92895,N1(C(CC2(C)CCCO2)=O)CC2CCCC2(NC(c2cc[nH]c2)=O)C1 92896,N#Cc1cccnc1CN(c1ncc(Br)s1)CCc1ccccc1 92897,c1(-c2ccc(C(=O)OC)s2)ccc(-c2cc(CN(C)C)ccc2OC)cc1F 92898,C1(CC)CCC(C(=O)NCC(c2ccccc2)NC(=O)Cc2ccncn2)CC1 92899,c1(OC)csc(C(c2nnnn2C)NCC2CCO2)c1OC 92900,C1(C(C)C)CN(C(c2ccsc2C#N)=O)CC1C(N1CCOC(C2CC2)C1)=O 92901,C1(C(=O)NCC(C)(C)NC(c2nnc(C)s2)=O)CCCC(F)(F)CC1 92902,C(=O)(C(C)(F)C(F)(F)F)NCC(C(C)C)NC(c1cc(N)ccn1)=O 92903,c1(C(N2C(CCCNC(C3(C)CC3(Cl)Cl)=O)CCC2)=O)ncc(F)cn1 92904,C1(CC)CN(C(C23CCC(F)(CC2)C3)=O)CCN1C(c1cnn(C(C)C)n1)=O 92905,c1(OC)cc(O)c(NC(c2ccnn2CC2(C)COC2)=O)cc1C 92906,N12CCN(CC13CC3)Cc1ccc(o1)C2.c1(N(C(C)=O)CCO)ccc(Cl)o1 92907,c1(C(N2C(CN(C(=O)C3=CCCCC3)CC)CCCC2)=O)nc[nH]c2ncnc1-2 92908,c1(C(N2CC(O)CC(NC(C3(C=C)CC3)=O)C2)=O)ccc2c(OC)ncnc2c1 92909,c1(C(=O)NCCN(C(C(C(C)OC)O)=O)C)c2c(c[nH]c1=N)CCC2 92910,C1(NC(c2ccc(C(F)F)c(F)c2)c2n(CCCF)nnn2)Cc2cscc2C1 92911,N1(C(=O)CC2(CO)CC2)CCCC2(C1)CN(C(c1cc(C(=O)O)cs1)=O)C2 92912,C=CCC(C(=O)NCCCNC(c1cnn(C)c1Br)=O)NC(C)=O 92913,C1(CN(C(=O)NCC)C)(CNCC2CC(F)C2)CCOCC1 92914,C12(C(=O)NC(CC)CNC(=O)CNC(C3CCCC3)=O)CCCC1C2Br 92915,C1(C(=O)NCC(CO)NC(c2cnc(Cl)n2C)=O)(OCC)CCCCCC1 92916,C(CCCCC(=O)N1CCC(NC(c2cn(C)c(C)n2)=O)CC1C1CC1)SC 92917,N1(C(C(C)C(C)O)=O)CCC2(CC1)CC(NC(=O)Cn1ncccc1=O)C2 92918,c1(C(N2CCN(C(CCC)=O)CC23CC3)=O)nccc2ncccc12 92919,c1(OC)c(C(N2CCN(CC3CN(C(=O)CC4CSC4)C3)CC2)=O)c(C)nn1C 92920,C1(C(=O)NC(CNC(COc2cc(C)c(Cl)cc2)=O)C)CCCC(F)(F)CC1 92921,c1(C(N(CCN(C(CN2CC(C)C2)=O)C)C)=O)cc(=O)c(Br)c[nH]1 92922,C1(N(C(=O)CNC=O)C(C)C)CS(=O)(=O)CC1O.Cc1ccccc1CCCSCC 92923,C(=O)(CC1=CCOCC1)NCC(CC(C)C)(C)NC(=O)Cn1ncnn1 92924,CC1(NC(=O)C(Cl)Cl)CCCCC1C(=O)NCC1CN(C2CCC2)C1 92925,c1(CCC(=O)NC(CN(C(C(CC)NC(N)=O)=O)C)C)cccc(OC(F)F)c1 92926,N#Cc1ccc(C(=O)N(CCCNC(c2cccn(O)c2=O)=O)C2CC2)cc1 92927,c1(C(=O)NC2COCCN(C(c3c(OC)csc3)=O)C2)cc(F)cc2ccoc12 92928,N1(C(C=Cc2c(C)ccnc2)=O)CC2CCC1CC2NC(C1CC12CCOC2)=O 92929,C1(C(=O)NC(CCOC)CNC(=O)CSC(F)F)CCN(C(C)=O)CC1 92930,c1(COC)ccc(C(N2CC(NC(C3(C4CCCCO4)CC3)=O)C(O)C2)=O)cc1 92931,Cc1ncc(C=CC(=O)NCC2(F)CC(NC(=O)CC(=O)N(C)C)C2)c(O)n1 92932,N1(C(CC2C(=O)NCCC2)=O)Cc2occ(C(N3CCC3C3CCC3)=O)c2C1 92933,C1(OC)(OC)CC(OC)CN(N2CCCC2C2CCCCC2O)C1 92934,C1(C(=O)NCCC2(C(=O)NCc3cc(Cl)ccc3F)CC2)CNc2ccnn2C1 92935,CCCCC(CC(=O)NCC1(C(C)C)CC1)NC(C1(C2(C)CC2)CC1)=O 92936,C(=O)(C(C)(C)CCCNC(C1CCCN(C)C1)=O)NCc1ccc(CC)o1 92937,c1cc(CN2CCCC2)c2c(c1)CN(c1ncnc3c1CCC3)CC2 92938,Cc1c(C(N2CCC(CNC(=O)C(C3CCOCC3)C)CC2)=O)cccc1O 92939,CON1CCC(C(=O)NCC2CC3CN(C(C45CCCC4C5)=O)CC23)CC1 92940,C1(C(=O)NCC(CC)NC(=O)Cn2cc(Cl)c(C)n2)CC(=O)N(CC)C1 92941,c1(C(=O)NC(C2CCN(C(C3(OC)CCSCC3)=O)C2)C)ccc2cnoc2c1 92942,c1(C(=O)NCC(CCNC(C2(OC)CCCOC2)=O)O)cnc(C(F)F)c(C)c1 92943,Cn1cnc2c1CN(C(=O)COC(C)(C)CNC(c1ccc(N)c(F)n1)=O)CC2 92944,c1(CC(=O)N(CC(CNC(C2CC(=C)C2)=O)O)C)ccccc1OC(C)C 92945,N1(C(C(C(=C)Cl)(C)C)=O)CC2CC(NC(c3ccc4nnnn4c3)=O)CC2C1 92946,c1(CC(=O)NC2(C)CC(NC(CCSCC)=O)C2)ccc(F)cc1F 92947,C1(C#C)(C(N(CCN(CC#C)C)CC)=O)CCN(C(C2CC2F)=O)CC1 92948,c1(NC(c2ccc(Nc3cc(N(C)C)ncn3)nc2)=O)cccc(O)c1Cl 92949,C(c1cnn(C)c1)=CC(=O)NC1(C2N(C(CCOCC#C)=O)CCC2)CC1 92950,c1(SC)cccnc1C(=O)N(C(C)CNCc1cccc(OCCO)c1)C 92951,CC(C)(C(=O)NCC=CCNC(C1CNC(=O)C1)=O)c1ncco1 92952,c1(-c2nc(CCC)on2)cccc(N(c2ncc(Br)cn2)C2(CO)CNC2)c1 92953,c1(CNC(=O)NC23CCC(C(=O)OC)(C2)CO3)cccc2c(Br)ccnc12 92954,CC(CF)CC(=O)NCC1(CCCNC(=O)C(C)N(C)C)CCCC1 92955,C(=O)(C1CCCc2nc[nH]c21)N1CCCC(NC(c2cccc(F)c2)=O)C1 92956,CCC(CC)C(=O)N1CCC(C)(C(=O)NCc2ccccc2OC)C1 92957,C(CC(C(C)(C)C)NC(C1CC(=O)CC(=O)N1)=O)N(C(=O)C=Cc1ccsc1)C 92958,C(=O)(C#CC1CCOCC1)N1C(CNC(C=Cc2cn(C)nn2)=O)CC(F)(F)C1 92959,c1(SC)ccc(S(=O)(=O)NC2CC3(CNC(=O)O3)C2)c(Cl)c1 92960,c1(C(N(CCN(C(c2ccn(CCN(C)C)n2)=O)C)C)=O)cc(Cl)c(Cl)[nH]1 92961,C(N=c1[nH]c(C)c(C(N2CCOCC2C(C)C)=O)s1)c1ccc(C)c(Cl)c1 92962,CC1C(NC(c2ccn(CCF)n2)=O)CCN1C(C1C=CCS1)=O 92963,C12(C(=O)NC3C(SC)CN(C(=O)CC4=CCCC4)C3)CCCC(C)(C1)OC2 92964,N1(CC(=O)NCC(=C)Br)CCCC(CNC(c2cc(OC)no2)=O)C1 92965,C(=O)(CCCC(C)NC(c1[nH]ccc1C1CC1)=O)NCC(C)NC(=O)OC 92966,CC1CCC(NC(C2CC(C)(C)C2C(F)(F)F)=O)CN1C(c1cc2occc2s1)=O 92967,C(=O)(C(CC(F)F)C1CCC1)NC(CNC(=O)COc1cccc(F)c1F)CO 92968,C1(NC(CC2C(C)C2)=O)C2CC1N(C(=O)CCOc1ccccc1O)C2 92969,C12(NC(c3snc(O)c3Cl)=O)CCC1CN(C(=O)CCOc1cccnc1)C2 92970,N#Cc1ccc(CCC(=O)NCCc2cccc3sccc23)c(F)c1 92971,CC1=NOC(C)(CNC(=O)C(c2ccoc2)NC(=O)C(C2CCCCC2)F)C1 92972,N1(C(c2ccnc(Cl)c2)C(=O)NCC2CC2)CCC2(CC1)OCc1ccncc12 92973,N1(C(c2c(OC)cc(F)c(F)c2)=O)CCCC2C1CCN2C(C1CC(F)C1)=O 92974,c1(C(N2C3(CNC(CC(C=C)C)=O)CCCC(C2)C3)=O)ccc2oc(C)nc2c1 92975,C(=O)(CS(=O)(=O)CC(C)C)NC(C1(O)CCN(C(C(CC)CC)=O)CC1)C 92976,S(=O)(=O)(c1cnc2ccccn12)NCC1(CC)CCOCC1 92977,N1(C(c2cnc(CC)[nH]2)=O)CC(C)N(C(=O)Cc2coc3ccccc23)CC1C 92978,Cc1noc(C)c1CSCCC(=O)NCC1(F)CN(C(=O)CC2CC2C)C1 92979,N1(C(C(C=CCCC)O)=O)C2CCC1CN(C(c1cc(SC)ccc1Cl)=O)C2 92980,c1(C(=O)NCC(CC)NC(=O)C(C)Oc2ccc(C(C)C)cc2)csc(C#N)c1 92981,C1(NC(C2CC(=C)C2)=O)CS(=O)(=O)C2CN(C(c3nnn(C(C)C)c3C)=O)CC12 92982,CC1(C)CCC12CN(C(=O)C1=CCN(C(C3CC34CCOC4)=O)C1)C2 92983,C(CN=c1ccn(CC=O)[nH]1)c1cc(OC)c(O)c(Cl)c1.N1(CCO)CCCCC1 92984,N1(C(C(CC#C)C2CC2)=O)C2CCC1CN(C(=O)C(C)C1CCC1)C2 92985,CCCC(O)C(=O)NC(C(N1CCC(CSC)C1)=O)C1(C)CC1 92986,N1(C(C(C=C)OC)=O)CCN(C(c2c(CC)cccc2F)=O)CC1COC 92987,c1(OC)ccc(CN2CCC(CC(N3CCCC3C(N)=O)=O)C2)c(Br)c1 92988,C1(CC(=O)N(C(C=CC(C)=O)=O)CC)CCN(C(=O)Cn2cnnn2)C1(C)C.CCCCO 92989,c1(C(=O)NC2(CO)CN(C(C3C(SC)CCC3)=O)C2)cc(F)cc(Br)c1 92990,CCC(O)C(C)(C)C(=O)N1CCC(C(n2cc(CO)nn2)NC(=O)CCCN=[N+]=[N-])C1 92991,S(=O)(=O)(CC(=O)N1CCCC(N(C(=O)CC2CCCC(OC)C2)C)C1)NCC 92992,CC1(C(N2CCC(CNC(C3(CF)CCOCC3)=O)C2)=O)CC=CCO1 92993,c1(CC)csc(NC(=O)CC(CNC(=O)Cc2ccccc2)OC)c1C 92994,Cc1ncc(Br)cc1C(N1CC(N(C(=O)CC2CCC(C)(C)C2)C)C1)=O 92995,c1(CNC2CC(C(N3CCN(CC#C)CC3)=O)C2)cccc2nc[nH]c12 92996,Cc1cc(N)cc(C(N2CC(CO)(NC(c3ccccc3F)=O)C2)=O)c1F 92997,c1(C(C)C)cccc(C(N2CCCCC2CNC(=O)C(C)(C)c2cscn2)=O)c1 92998,C(CN=c1[nH]c(=NCC2CCCN(CC)C2)[nH]c2c1COC2)OCC(=C)C 92999,c1(C(N2CC(NC(c3n(C(C)C)ncn3)=O)C2)=O)cccc(OCC(F)F)c1 93000,N1(C(C2CCCC2)=O)CCN(C(=O)C=CC2CCCCC2)C(c2ccncc2)C1 93001,c1(C(=O)NC2CN(C(C3(C#C)CCCC3)=O)CC2O)ccc(Cl)c(C)c1Cl 93002,N1(C(CCOCCC)=O)CC(CNC(=O)C(C)Sc2ccc(C)cc2)C(F)(F)C1 93003,C1(C(=O)NC2C(CNC(=O)Cn3cnc([N+](=O)[O-])n3)C2)CCC2(CCCCC2)C1 93004,c1(OC)ccc(O)c(C(=O)NC2CC(CCNC(C3CC3Br)=O)C2)c1 93005,c1(C(N2C(CNC(c3cc(C)[nH]c3C)=O)CCCC2)=O)c(C)cc(O)nc1C 93006,N1(C(c2c(C)noc2)=O)C2CCC1CN(C(=O)C(C)CC1CCC1)C2 93007,O(NC(=O)CC(C)NC(C1CCCN(C(C)C)C1)=O)CCOC(C)C 93008,N1(C(c2ccsn2)=O)CCCN(C(c2cnn3c2NCCC3)=O)C(CO)C1 93009,C1(NC(c2csc(C)c2N)=O)CC2(C1)CC(NC(=O)C(C)NC(=O)C(C)(C)C)C2 93010,C=C(C)C(CC(=O)N1CCCC(CC(=O)N(C)CCN(C)C2CC2)C1)OCC 93011,c1(C(=O)NCC2(C)CC(NC(c3ncc(CC)cn3)=O)C2)c[nH]cc(C)c1=O 93012,CCC(CCOC)C(=O)N1CCOC(C)(CNC(=O)CCNC(=O)COC)C1 93013,c12nc(C)ccc1C(=O)N2.c1(OC)cc(C(=O)N(C2CCCCC2)C(C)C)sn1 93014,Nc1nonc1C(=O)NCC=CC(N1CC(C2CCCO2)C1)=O.n1(CC)ccnn1 93015,N1(C(c2cc(C)cc(C)c2)=O)CCCC2(NC(c3ccnnc3C)=O)CC2C1 93016,CC1OCCN(C(C2CCN(C(c3ccco3)=O)C23CC3)=O)C1C 93017,N1(C(CCSCCCC)=O)CC2CCCN(C(c3ncoc3C)=O)C2C1 93018,C1(NC(CC2C(C)(C)C2)=O)CC2(CCCN(C(c3c(Cl)csc3Cl)=O)C2)C1 93019,c1(N(CC)CC)ccc(CN=C(NC2(C)CCC2)NC2CC2C)cn1 93020,c1(C(=O)NCC2(NC(c3cn(C)c(=O)n3C)=O)CC2)ccn2c(O)nnc2c1 93021,Cc1cccc2[nH]cc(C(N3CC(C)(NC(C4CCC(C5CC5)C4)=O)C3)=O)c12 93022,N1(C(C(CCC)NC(C)=O)=O)CCCC(F)(CNC(C2SCCCS2)=O)C1 93023,c1(CC)ccc(F)c(C(=O)NCC2COCCN(C(=O)CC(C)C(F)F)C2)c1F 93024,N1(C(C2C(C)CCC2)=O)CCN2CCN(C(=O)CN3CCC(=O)CC3)CC2C1 93025,C1(CNC(C2(C)CC3CC3C2)=O)CC(C(F)(F)F)CCN1C(=O)CCCN=[N+]=[N-] 93026,C(=O)(C1=NN(C2CC2)C(=O)CC1)N1CCC(O)(CNC(C2C(C(N)=O)C2)=O)CC1 93027,C(C(C(=O)N(C)Cc1nccn1CC)C(C)(C)C)NC(c1oc(CC)c(C)c1)=O 93028,N1(C(C=CCCC=C(C)C)=O)CCC(NC(c2ccc(Cl)cc2C)=O)C(CO)C1 93029,CC(C)(C(=O)N1CCC1NC(=O)CN1C(=O)NC(C2CC2)(CCO)C1=O)C(F)F 93030,C(=O)(C(C)CCCC(C)C)NC(CC=C)CNC(=O)C=CC(=O)N(C)C 93031,N1(C(CCc2cccc(OC)c2)=O)CCC(C)(NC(C2(O)CCCCC2)=O)CC1 93032,c1(C(N2C(C(C)Nc3cc(OCC)ncn3)CCCC2)=O)ccc(C#N)nc1C 93033,N1(C(c2cnc(C)nc2C)=O)CCCC2(CCN2C(=O)C(c2ccccc2)O)C1 93034,CCC(O)C(C)(C)C(=O)NCCN(C(=O)CCN(C1CCCCCC1)C)CC 93035,c1(C(=O)NCC(CCNC(c2ccc(C#C)cc2)=O)O)c(C)cc(C)cc1C 93036,c1(OCC(=O)NC)cccc(CC(=O)NCC#CCNC(=O)CC=C(C)C)c1 93037,C1(CCOC(C)(C)C)(NC(C(C)N(C)C)=O)CCN(C(=O)Cc2cscn2)CC1 93038,N1(C(c2nc(C)nn2C)=O)CCC2OCCN(C(=O)Cc3sc(C)nc3C)C2C1 93039,Cc1cccnc1C(=O)NCCC1N(C(C2CCCN2C2CCCC2)=O)CCC1 93040,c1(OCCC(=O)NC(CNC(C(C)CO)=O)C(C)(C)C)ccccc1C(N)=O 93041,CCCCC(O)C(=O)N1CCCC1(C)CNC(=O)CSc1n[nH]c(O)n1 93042,c1(CN(C2CCCC2c2ccccc2)C)cc(F)cc(F)c1O 93043,N1(C(c2c(C)cc(C)o2)=O)CCC(NC(=O)C(C)CN2CCOCC2)C12CC2 93044,C1(NC(c2cc(CSCC)on2)=O)CN(C(=O)C(C(C)(C)C)OCC)CCC1(C)C 93045,c1(NC2(CNC(C(C=C)O)=O)CC2)cnc(C#N)c(C#N)n1 93046,S(=O)(=O)(c1ccc(C=CC(=O)N(C2CCNCC23CC3)CC2CC2)cc1)NC 93047,C(=O)(CCCC(=O)NC(C)C(CO)NC(C1NC(=O)OC1C)=O)NCCC 93048,c1(CC)nn(C)cc1C(=O)NCC(n1cc(CC2CCCCC2)nn1)C 93049,Nc1cccc(C(=O)NCC2CCCCN2C(C2CCC2(F)F)=O)n1 93050,c1(C(N2C3CC(NC(C4CCS(=O)(=O)CC4)=O)C2CC3)=O)ccc2nnnn2c1 93051,C1(CS(=O)(=O)CCCn2cc(CCCCCCC)nn2)C(F)(F)C12CCOCC2 93052,c1(C(=O)NCC2(COC)CN(C(C3CN(C)C3)=O)C2)cc(Cl)cnc1OC 93053,c1(C(=O)NC(CC)CNC(=O)C(C)C(O)CC)ccccc1N=[N+]=[N-] 93054,C1(CC(=O)OC)CC(NC(=O)CC(=O)NCC#N)CCO1 93055,C(=O)(CCC(C)(F)F)N1CCC(CN2CCN(C(C3C(C)OCC3)=O)CC2)CC1 93056,c1(C(N2CCC(N(C(=O)CSC(F)F)C)C2)=O)cc2cscc2s1 93057,c1(C(=O)NCC2N(C(=O)C#CC3(C)CC3)CCN(C)C2)cc2ccc(Cl)cc2s1 93058,C1(C2CCCC2)(NC(C2C3CN(C(C(CCC)F)=O)CC32)=O)CCC1 93059,N1(Cc2nccc(C)c2)CCC2(CCN(C(c3ccc(C)c(C)n3)=O)C2)C1 93060,c1(C(N2CCOCC(CNC(C(C)(O)C3CC3)=O)C2)=O)cccc2scnc12 93061,N1(C(Cc2cc(C)[nH]n2)=O)CCC2CCN(C(c3c(C)[nH]c(C)c3C)=O)CC2C1 93062,C1(C2CC2)(COC(C(CC=C)(C)N(C)C)=O)CCN(C(C)=O)CC1 93063,C(=O)(CC(C)(C)CNC(C1(C)CC(=O)C1)=O)NC(C(=O)N(CC)CC)C 93064,CC1OC2(C)CC1(C(=O)NC1CCN(CCOCC(F)(F)F)CC1)C2 93065,c1(CC)nnc(=NCC2C3CN(C(=O)C(C)(C)C4CC4)CC23)[nH]c1CC 93066,n1(CC(N2CC(C)NCCC2)=O)ncc2ncccc12.N12CC3C(C3C1)C2=O 93067,Cc1ncc(NC(=O)CCC2CCN2CC(=Cc2ccccc2)N)cc1Cl 93068,C(=O)(C(C)(C)Cc1ccccc1)NC1CC(N(C(=O)CSCc2ncc[nH]2)C)C1 93069,Cc1ccc(C(=O)NCC2(C(C)(C)O)CN(C(C3CCOC3)=O)C2)nc1F 93070,c1(C(=O)NCC2N(C(C(C)CC3CCC3)=O)CCOC2)cc(Cl)nnc1O 93071,c1(SCC)cncc(C(N2CC(CCNC(c3cn(CC)nc3C)=O)C2)=O)n1 93072,C(=O)(CC1=CCN(C(=O)CN2CCCC2)CC1)NCCc1nccc(C)n1 93073,N1(C(CNC(c2c(C)ccs2)=O)=O)CC(CO)CC1C 93074,N1(C(c2c(C)cccc2C)=O)CC2CCC1C(CNC(C1(C(F)F)CCC1)=O)C2 93075,C#Cc1ccccc1CN(C(C(=O)NCC(c1ccc(Cl)c(Cl)c1)OC)=O)C 93076,C=C=CCC(=O)NC1CCC(C(=O)NC(C)Cc2cnc[nH]2)C1 93077,C(=O)(CC(CC=C)c1ccccc1)NCC1(NC(CCCC=C)=O)CCOC1 93078,c1(OC(C(N2C(C(C)NC(C(C)(C)OCC)=O)CCC2)=O)C)ccc(Cl)cc1 93079,c1(C(=O)NC2(COC)CCN(C(C3CC(C)C3)=O)C2)ccc2c(c1)COC2(C)C 93080,c1(C(N2CCN(C(c3c(OC)c[nH]n3)=O)C(C)C2)=O)cn2nc(OC)ccc2n1 93081,CC1CCc2ncc(C(N3CC4CCC3CN4C(=O)C(C)C(C)(C)O)=O)n2C1 93082,C(=O)(CS(=O)(=O)c1ccc(Cl)cc1)NC(CC)CNC(=O)CCOC(C)C 93083,N1(C(Cc2c(C)cnn2C)=O)CCCN(C(c2ccc(OC(F)F)cc2)=O)CC1 93084,C(=O)(NNC(=O)COc1ccccc1Cl)N(C)CCN(C1N(C(C)=O)CCC1)C 93085,c1(OCC)nccc(C(=O)NCC2CC(C)N(C(c3c(C)noc3C)=O)C2)c1F 93086,CCC(CC)(CC)C(=O)N1CC(OC)C(NC(c2cc(=O)n(-c3ccccc3)[nH]2)=O)C1 93087,c1(C(c2n(C(C(=O)OC)C)nnn2)NCCn2cnnn2)ccc(C#N)cc1F 93088,c1(C(C(=O)NC2CCCN(C(C=CC=CCC)=O)C2)O)cccc([N+](=O)[O-])c1 93089,C1(C(N2C(COC(C3(CO)CCCC3)=O)CCCC2)=O)CCc2[nH]nc(O)c2C1 93090,CCC(F)(F)CCNC(=O)NC1CC(=O)N(CC2CC2)C1 93091,C1(NC(C(N2CCCCCC2)C)=O)CC2CCC1N(C(=O)CCC(N)=O)C2 93092,C#CC1CCCN(C(c2ccccc2C2CCN(c3ccnc(SC)n3)CC2)=O)C1 93093,c1(C(=O)NCC2(F)CCN(C(C(n3c(C)cc(C)n3)C)=O)C2)cc(C)c(C)nn1 93094,C(c1cccc(O)c1)=CC(=O)NC1CN(C(CCCNC(C)=O)=O)C2C1C2 93095,c1(COC)ncncc1NCc1cccc(-c2cccc(N(C)C)n2)c1 93096,CC1OC2CCC1(C(=O)N(CCCN(C(=O)COCC1(F)CC1)C)C)C2 93097,N1(C(Cn2c(=N)nc[nH]2)=O)CC(NC(=O)C2=CCCSC2)CC12CCOC2 93098,N1(C(c2cn(C)c(Br)c2)=O)CC2CC(CNC(=O)C(F)=C3CCCC3)C2C1 93099,c1(N2CC=C(CNC(C(C)(C)C(F)F)=O)CC2)ncnc2c1CCCC2 93100,C(=O)(C(=O)CC(C)CC)N(C(CNC(C(CCCC)O)=O)CC)C 93101,N1(C(c2c(CC)n(C)nc2)=O)CCC2CCN(C(c3cscc3SC)=O)CC12 93102,N1(CC)CCOC(C(=O)NCC=CC(=O)NOCC2CCC2)C1 93103,N1(C(c2cn(C3CCC3)nn2)C(=O)N(C2(C)CC2)C2CC2)CCN(CCC#N)CC1 93104,c1(-c2cn(CC(CCSC)(C)O)nn2)ncc([N+](=O)[O-])cc1Br 93105,S(=O)(=O)(c1ccc(C(=O)NC2CCC(CNC(c3cncc(N)n3)=O)C2)o1)NC 93106,N1(C(c2ccc(C)cn2)C(=O)NCCSC)CCC(O)C(C)(O)C1 93107,C(=O)(C(CN(C)C)CC)NC1C=CC(CC(=O)NCCCSCC)C1 93108,CC(C)(CNC(=O)C=CC1CC1)CC1CN(C(c2cc(CC3CC3)on2)=O)C1 93109,C1(NC(C(F)=CC)=O)CC(CNC(c2ocnc2C2CC2)=O)C1(C)C 93110,CC1(O)CCCN(C(=O)C(Cc2cnc[nH]2)NC(=O)CCN2CCCC2=O)C1 93111,C1(C(NOCCCC)=O)CN(C(C2CN(C(=O)NC)C2)=O)CC12CCC2 93112,N1(C(c2cnc(OC)s2)=O)CCCN(C(=O)CN2CCOCC2)CC1C 93113,C1(N(C(=O)CC2COC(=O)C2)C)CCCCN(C(C2CS(=O)(=O)C2)=O)C1 93114,c1(NCCCNC(=O)OC)ccc(S(=O)(=O)N(C(C)CS(C)(=O)=O)C)cc1Cl 93115,c1(OC)cnnc(C(=O)NCC(C2CC2)NC(C2(OC)CCOC2)=O)c1 93116,C1(C(N2CC(C)C(CNC(c3csc(S)n3)=O)C2)=O)CCc2nnc(O)n2C1 93117,c1(C(=O)NCC(C(C)C)NC(C2CC3(C2)CC3(F)F)=O)cccc(C(N)=O)c1N 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93136,CC1(C)CC(O)C(O)CN(C(=O)CC2CCN(C(=O)Nc3cc[nH]c(=N)n3)C2)C1 93137,CC1CCC(NC(C2CC23CCSCC3)=O)CN1C(=O)CCN1CCCCC1 93138,c1(SCC2CC(CC)CN(C(=O)OC(C)(C)C)C2)cc(Cl)ncc1Cl 93139,c1(C(=O)NCCN2CCN(C(=O)COC3CCOC3)CC2)cnc2sccn12 93140,C1(NC(Cc2cn(CC)nn2)=O)COCCN(C(=O)C=Cc2ccc(CC)o2)C1 93141,c1(CCNC(N(CCCO)C)=O)csc2ccc(Br)cc12 93142,N1(C(C2C(C)(C)C2)=O)CCC(O)(C2(NC(c3cc(C(N)=O)ccn3)=O)CC2)CC1 93143,C1(CNC(COCC)=O)CCN(C(=O)CCCCCOCC)CCC1(F)F 93144,C1(C(=O)N(C)Cc2cnco2)(COC)C=CCN1C(=O)CN1CCCC1 93145,c1(N(C(CNC(c2cc(CCC)[nH]n2)=O)C)C)ncnc(Cl)c1Br 93146,CONc1cccc(NC(=O)NCCCCCCOc2c(Br)cccc2Br)n1.CCO 93147,C=C(C)C1OCCCC1C(=O)NCC1C=CCN1C(c1ccnn1CC)=O 93148,C1(C(=O)NC(CC)CNC(c2snc(C)c2Br)=O)CC2(CCOCC2)C1 93149,c1(N(C)C)nc2ncnc(N(CCOCCO)C3CC3)c2s1.C1(C)CCCC1 93150,Cc1cnc(O)c(CNC(=O)CC(C)N(C)C(C2CCCC(=O)CC2)=O)c1 93151,C1(O)(CN(C(CC(C)(C)OC)=O)C)CCCN(C(c2nnn3c2CCC3)=O)C1 93152,c1(C(N2C(C)CC(NC(C=C(C)C)=O)C2)=O)ncnc2c1c(Br)cn2C 93153,N1(C(CCOc2ccc(C)c(Cl)c2)=O)CC2CCCN(C(C3CC3C)=O)C2C1 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93380,C1(Nc2cc(OCC)nc(OC)n2)CC2CCCC(C1)N2C(=O)C(OC)OC 93381,CS(=O)(=O)c1ccsc1C(=O)Nc1ccc(-c2cccnc2)nc1 93382,C=CCC(C)C(=O)NC(C)(CO)C(=O)NCC1(CC2CC2)CCC1 93383,c1(NCC(NC(CCNC(CC(C)C)=O)=O)C2CC2)ncnc(-c2ccccc2)n1 93384,C(=O)(CCCCC#N)NC(C(C)NC(=O)Cc1ccccc1Br)(C)C 93385,C1(NC(COCCCOC)=O)CC(F)CN(C(=O)C(C)(F)CC2CCCC2)C1 93386,Oc1cccc2c1CN(c1nc(=NCC3CC4C(C3)C4(F)F)[nH]c3c1COC3)C2 93387,CCCC(C)(CCC)C(=O)NCC1CC2(CO1)CN(C(=O)CCC#N)C2 93388,C1(NC(C(CCC)NC(N)=O)=O)CC2CC1N(C(c1cnc(OC)c(C)c1)=O)C2 93389,c1(N(CC(=O)O)C)ccc(-c2nscc2O)cc1O 93390,C1(CNC(C2(C)CS(=O)(=O)C2)=O)CCC2(CN(C(C3CCC(C)CC3)=O)C2)O1 93391,c1(C(N2CCC(O)(CNC(c3n(CC)nnc3)=O)C2)=O)c(Cl)ccc(Cl)c1Cl 93392,CCC(O)CC(=O)NC(C(=O)NCc1nc[nH]n1)c1ccoc1 93393,N1(C(=O)NC(C)C(C)(C)C(F)F)CCCC1C1CCCCO1 93394,C#CC(CC(C)C)NC(C1CCN(C(=O)CCc2csnn2)C1C(C)C)=O 93395,N1(C(c2cnc(CC)s2)=O)C2CCC1CN(C(c1cnnc(C)c1)=O)CC2 93396,CCC(O)C(C)C(=O)NC1CC(CNC(=O)CC(c2ccccc2)NC(N)=O)C1 93397,CC(C)C#CC(=O)NC(C)(CNC(=O)C(C)NC(C1CCCC1)=O)CO 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93416,c1(C(=O)NCC2(CN(C)C(C3C(C(F)F)C3(C)C)=O)CC2)cc(N)cc(F)c1 93417,c1(C(=O)NCC(CNC(C(C(C)O)N(C)C)=O)C(F)(F)F)ncc2n1CCCC2 93418,C1(c2nnnn2C2CC2)(CCC(F)F)CCCC(C)(C)C1 93419,Cc1oc(C(N2CCN(C(=O)CC3CC(=O)NC3=O)CC2)=O)cc1S(C)(=O)=O 93420,N#Cc1ccc(=NCC2CCC(NC(c3cnc(Cl)[nH]3)=O)C2)[nH]c1 93421,c1(C(=O)NC(CC(C)NC(c2ccc(CCC)cc2)=O)C)ccc(OC)cc1F 93422,C1(C(=O)NCCCOCCOC)CCCCC1NC(=O)CN1CCCC1C 93423,C1(NC(CCNC(C(C)(C)C)=O)=O)CCCC(NC(c2csc(C#N)c2)=O)C1 93424,Cc1nc(N2CC(C)(C)CC2CNC(C2(F)CCS(=O)(=O)C2)=O)c2c[nH]nc2n1 93425,c1(OC)cccc(C(CNC(c2sccc2C)=O)NC(=O)CCNC(C)=O)c1 93426,c1(CCC(=O)NC2C(CNC(C(COCC)C)=O)C2)ccc(F)cc1 93427,C(=O)(C(C(=O)OC)C1CC1)NC(CCNC(COCC)=O)C 93428,CP(C)(=O)C1CCCC1C(=O)NCC1CCN(C(c2ccc3c(c2)NCC3)=O)C1 93429,C1(C(N(CCOC)CCNC(=O)C=Cc2ccoc2)=O)CCCC(C)CC1 93430,c1(CC)ccnc(C(=O)NC(C2CCN(C(c3cnn(C)c3F)=O)CC2)C)c1 93431,C12(NC(c3cc4ccccn4n3)=O)COCCC1CN(C(=O)Cc1cc[nH]n1)C2 93432,C1(CNC(c2n(CC(=C)C)nnn2)c2cnoc2)Cc2ccccc2C1 93433,N1(C(c2c(C)nccn2)=O)CCCC2C(NC(C3CCCC3C)=O)C(C)(C)C12 93434,C1(C(N(C)Cc2nncn2C2CC2)=O)C=CCN(C(=O)CSC2CC2)C1 93435,N1(C(CC(CC)C)=O)CC2(C1)C(NC(=O)Cc1ccc(C)cc1)CCS2(=O)=O 93436,CC(C)CCC(=O)N1CCCC1CCC1CCN(C(=O)Cn2cc(Br)cn2)CC1 93437,c1(C(N2CC3C(CC(=O)NC(C)(C)C#N)(CC3)C2)=O)ccc2c(c1)COC2 93438,N1(C(C(CCC)C)=O)CC2CC1CC2NC(c1ccc(NS(C)(=O)=O)cc1)=O 93439,CCCCC(O)CC(=O)N1CC2C(CC(=O)NC(c3ccccc3O)C)C2C1 93440,CN=c1[nH]c(C(N2CCN(CCCNC(=O)CCC3CCOC3)CC2)=O)cs1 93441,C1(C(=O)NC(CC(C)C)C)CC(C)(C)CN1C(c1cnc(Cl)n1C)=O 93442,N1(C(CC2(OC)CC2)=O)CCCC2CN(C(c3ncccc3F)=O)CCC12 93443,C1(CNC(CN(C)CCO)=O)CCCCN(C(=O)C2=CCOCC2)C1 93444,CC(C)(F)CCC(=O)NCc1cc(C(=O)NCCc2ccon2)co1 93445,c1(CC)n[nH]c(CC)c1CC(N1CC(CN(C)C(C2CCCOC2C)=O)C1)=O 93446,C1(C#N)(C(N(C)CC2CC(F)CN2C(C2CC(C)(F)C2)=O)=O)CC2CCC1CC2 93447,O=C1CN(C(C2CC3(CC3)CN2C(c2cc(O)no2)=O)=O)CCCN1 93448,CC1CN(C(c2cnns2)=O)CC(C)N1C(C1CC(=O)NC1(C)C)=O 93449,CC1(C(N2CCC2CNC(c2cccc(C(F)F)n2)=O)=O)COCCO1 93450,N1(C(C(C)Cn2cccn2)=O)CCn2c(CNC(=O)CC3CCOC3)nnc2C1 93451,N1(C(c2cnc(C)n2C)=O)CC2(C(=O)NCC(F)Br)CC1CCO2 93452,N1(C(COc2c(C)cccc2)=O)CCC(N(C(=O)Cc2csnc2C)C)C(C)C1 93453,N1(C(c2csc(-c3ccoc3)n2)=O)CC2CCC(C1CO)N2C(c1cscn1)=O 93454,C1(O)(CC)CCN(C(=O)C(C)NC(C)(C)CC)CC1.C12(CC1)C(=O)NC2 93455,CCCC(CCC)C(=O)NC(CC1CC1)C(=O)NCC(F)(F)CC1CC1 93456,c1(CC)ccc(C(=O)NC2CCC(N(C)C(c3cc4scnc4[nH]3)=O)C2)c(C)n1 93457,N1(C(C)=O)CSCC1C(=O)NC(C)CCCNC(C1(c2ccccc2)CCC1)=O 93458,N1(C(C(CC2CC2)NC(c2cc(COC)[nH]n2)=O)=O)CC(C)OCC(C)(C)C1 93459,N1(C(C(C(C)O)NC(=O)C=CC(=O)NC2CC2)=O)CCN(C)C(CO)C1 93460,C(c1cn[nH]c1)=C(C)C(=O)N(C1(CC(=O)NC(C2CCN(C)C2)C)CC1)C 93461,C(=O)(C1Cc2c(Cl)cccc21)N1CCC(NC(C(CCC)C)=O)C(F)C1 93462,C1(NC(C(C(C)C)NC(c2c(C)cc(F)cc2)=O)=O)CCC(=O)N(C)C1=O 93463,N1(C(CCP(C)(C)=O)=O)CCC2(CCC2)C(NC(=O)COc2cccnc2)C1 93464,C1(S(N)(=O)=O)(C(N2CCCC(NC(CNC(CC(C)(C)C)=O)=O)C2)=O)CCC1 93465,N1(C(CCOCC(C)C)=O)CCCN(C(=O)C(C)Cc2ccco2)CC1 93466,CC1=C(C(=O)N2CC(NC(c3ccc(O)nc3Cl)=O)CC(C)C2)C(C)(C)CCC1 93467,CC1(C)CN(C2CCCNC2=O)CC(CNC(C2(F)CCS(=O)(=O)C2)=O)O1 93468,C1(CC(=O)NC(c2nc(C(=O)O)n[nH]2)CC)CCc2ccccc2N1 93469,N1(C(C(CC)O)=O)CCN(C(c2ccccc2Oc2ccccc2)=O)CC(O)C1 93470,CCC(CC)CCCC(=O)NCC1(COC)CN(C(c2cnc(Cl)s2)=O)C1 93471,N1(C(c2nc(OC)oc2)=O)CCCC2CN(C(=O)CN(C)CCOC(C)=O)CC12 93472,C(C(C(C)(C)C)NC(=O)C(C)CCN1CCCC1)N(C(C)=O)CC.c1(O)ccccc1 93473,C(=O)(CCCCCS(N)(=O)=O)N1C(CC)CCC1.c12nc(cc(C)n1)CN2C 93474,C=CC1(NC(c2cn(CC)cn2)=O)CCCCC1 93475,[N-]=[N+]=NCCCC(=O)NC1CC(C(=O)NCC(=O)NCC2CCC2)C1 93476,Cc1cc(C)nc(CN2CC(F)CC2CN=[N+]=[N-])n1 93477,C1(CNC(=O)Cc2cccc(Cl)c2)CC2(CO1)CN(C(C1(CO)COC1)=O)C2 93478,C#Cc1cn(C)nc1C(N1CCC(CNC(c2ncc(F)cc2C)=O)C1)=O 93479,C1(NC(c2ccnc(F)c2)=O)CCCN(C(C2CCN(C(=O)C3CC3)CC2)=O)C1 93480,c1(OC)cc(N)ccc1C(N1CC(NC(c2c[nH]cc2Br)=O)C(C)C1)=O 93481,C(=O)(CCCN(C)N=O)N1CC(C)C(C)(CNC(C2(C)COC(=O)OC2)=O)C1 93482,c1(NC(C2CCC(C)N2C(C2CSCC(=O)N2)=O)=O)ccc(=O)n(CCO)c1 93483,C1(CNC(=O)CSc2nc[nH]n2)CCN(Cc2ccccc2F)CC1(F)F 93484,c1(OC)ccccc1N.c1(C2C(=O)CC(O)CN2C)cccc(Br)c1 93485,C1(CC=C)(NC(=O)C(O)Cc2ccco2)CCN(C(=O)Cc2ccc(Cl)cc2)C1 93486,CC(C)(O)CCC(=O)NCC1CN(C(=O)Cc2cnccn2)CC1C(F)(F)F 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93821,c1(CNC(C2(c3ccc(-c4ccnc(F)c4)cc3)CC2)=O)cc(F)c(Br)cc1Cl 93822,C1(C(N(CC(C)(C)NC(C2COCCO2)=O)C)=O)CCCCC1C(N)=O 93823,CC1CN(C(C2(n3cncn3)CC2)=O)CCC1N(C(=O)CC1(C)CCC1)C 93824,c1(C(N2CC(C)C(NC(c3cc(Cl)ccn3)=O)CC2)=O)cc(N)c(F)cc1F 93825,C1(C(=O)OC)CCC(C2CCCCC2)CN1C(=O)C(=O)NCC1(OC)CCOCC1 93826,C12(COC)CC(NC(C3CSCCS3)=O)(CN1C(c1cc(Cl)n(C)n1)=O)C2 93827,C=CC(CCC)CC(=O)NC1CCN(C(=O)CC2CCC(OCC)CC2)C1(C)C 93828,CC(C)C(F)(CNC(C1CNC(=O)N1)=O)C(=O)NC1CC2C=CC1C2 93829,N1(C(C=CC2(C)COC2)=O)CCCN(C(=O)Cn2cnc(Br)n2)CC1 93830,Cc1ccc(C(=O)CN(CCNC(=O)CN2CCC2C)C2CC2)s1 93831,c1(-n2nnc(C(=O)NCCCNC(C(C=CC)O)=O)c2C)ccc([N+](=O)[O-])cc1 93832,N1(C(c2cnc(CC)[nH]2)=O)CCC(NC(c2cc(N)c(Cl)cn2)=O)C2(CCC2)C1 93833,C(=O)(C1=CC2CCCCCCC12)N(CCCCCCNC(c1ccc(F)s1)=O)C 93834,C1(CNC(CSC)=O)CC(C(=O)N(CC(O)C(C)(C)C)C)=NO1 93835,CC(CC(=O)N1CCC(C(=O)NCCCCC(N)=O)O1)n1cccc1 93836,C1(NC(CC2(C)CCCO2)=O)CCC2(CCCN2C(c2ccoc2Cl)=O)CC1 93837,C1(CC=C)(NC(=O)CCCC2CC2)CCN(C(=O)CC2CCC(C)CO2)C1 93838,c1(CC(=O)NC2COCCC2NC(C2(F)CC=CCC2)=O)ccnc(Cl)c1F 93839,C1(C(=O)NC(CCOC)CNC(C2CCC2)=O)CCN(c2nc(C)cs2)CC1 93840,c1(CC(=O)NC2C(NC(C3N(C(CCC)=O)CCC3)=O)CC2)cccc(O)c1F 93841,C1(CN(c2nc(OC)c(Br)cn2)C)CC2CCC(C1)N2C(=O)C1=C(C)OCC1 93842,N1(CC(=O)NCCN(C)C(c2ncsc2C2CC2)=O)CCCC(N(C)C)C1 93843,c1(CN2CCCC(NC(C3CCCC(C)C3)=O)C2)c(Br)cc(F)cc1Br 93844,N1(CC(=O)NC2(CC)CCC(C)CC2)C(=O)CCC(N)C1=O 93845,N1(c2cc(C)ncn2)CCC2(CCN(C(C3Cc4cccc(C)c4O3)=O)C2)C1 93846,C1(C)(CC)CCCN(C(=O)COCCNC(c2csnc2Cl)=O)C1 93847,c1(C(N(CCNC(C2CC2C)=O)CC)=O)c(O)cnc2ccccc12 93848,C1(OC)CC(CNC(C2(C#N)CCC2)=O)N(C(c2c(C)n[nH]c2C)=O)C1 93849,N1(C(C2(F)CCCN(C(COCC(=O)OC)=O)C2)=O)CCn2cnnc2C1C 93850,c1(NC2C(C3CCN(C(C(=O)OCC)=O)CC3)OCCC2)cccc2[nH]ncc12 93851,c1(CC(=O)N2C(C)CNC(=O)CO2)cncc(F)c1.C1(CC)CCCO1 93852,c1(OC)cnc(F)c(C(=O)NCCCC(CO)NC(C2(C)COCCO2)=O)c1 93853,c1(C(=O)NCCN(C(c2sccc2CN(C)C)=O)CC)ccc2nsnc2c1 93854,N1(C(c2c(C)[nH]nc2Cl)=O)CCN(C(C2CC2F)=O)C(c2cc(F)cc(F)c2)C1 93855,N1(C(=O)OC2CCCN(C(N(C)C)=O)C2=O)CCOC(C2CCCO2)C1 93856,c1(C(=O)NCC2(O)CCN(C(c3csc(C)c3C)=O)CC2)cc2ccccn2c1 93857,N#Cc1cc(C(N2CCN(C(C3(Cl)CC34CCOCC4)=O)CC2)=O)ccc1F 93858,c1(C(=O)NCCC2(O)CCN(C(CC(C(C)C)O)=O)C2)cc2c(Cl)ccnc2s1 93859,Nc1nccnc1C(N1CCC1CNC(c1c(Br)n[nH]c1Br)=O)=O 93860,N1(C(C2=C(C)CCOC2)=O)CC(C2CCCN(C(C3CCCCCN3C)=O)C2)C1 93861,C1(NC(=O)Cn2cnnn2)CCC2(CC1)CC2NC(C12CC3CC1C2C3O)=O 93862,N1(C(c2n(CC)nnc2)=O)CC2CCCC1C2CNC(c1cnc(Cl)s1)=O 93863,c12ccc(o1)S(=O)(=O)N2.N1(N(C)C(c2ccccc2)=O)CC(CO)CC1=O 93864,C1(NC(=O)NCC)CCN(N(C(CC(=O)OCC)=O)Cc2ccc(O)cc2)CC1 93865,c1(C(N2C(C(N3CCC(CF)CC3)=O)CCC2C2CC2)=O)cccc(O)c1F 93866,N1(C(CCCOC)=O)CC(OC)C(NC(=O)CCCc2nccs2)C1 93867,CCC(C(=O)NC(=O)CCSC)OCCN(CC1CC1)CC1CC1 93868,C1(COC)CN(C(c2cc(C)n(C(C)C)c2)=O)CCN1C(C1CC(F)CN1C)=O 93869,CC(CC(=O)NC1CCCN(C(=O)CCCC2CCCCC2)CC1)C(F)F 93870,c1(C(N2C(CNC(C(C)Cn3ccnc3)=O)CC2)=O)ccc2cc[nH]c2n1 93871,C=CCC(C(=O)NCC1CCC(NC(c2cc(C3CC3)sn2)=O)CC1)C(C)C 93872,C(=O)(C(CCN(C)C)NC(=O)CCOC)NCC(C1CCCC1)OC 93873,C1(C(C)(C)NC(=O)CCN2CCC2)CCN(C(c2ccc(OCCF)cc2)=O)CC1 93874,c1(NC(c2c(C)cc(C)cc2C)C)nccc(=NC(C)c2n[nH]c(=N)s2)[nH]1 93875,N1(C(C(CCC)NC(=O)CC2(OC)CCC2)=O)CCC(C)(C#N)CC1 93876,C(CCN=c1nc(N2CCOC(CF)C2)c2sccc2[nH]1)N1CCP(C)(=O)CC1 93877,C1(CC)CC(OC)CN(CC(=O)NNC(=O)c2cccnc2)C1 93878,Cc1cc(CC(=O)NCC(CC(C)C)NC(=O)Cn2ccccc2=O)n(C)n1 93879,c1(C(N2CC(F)CC(C(=O)NC3CCCN(C)C3)C2)=O)ccc2cn(C)nc2c1 93880,N1(C(C2C(OCC)CC2)=O)CCCC(CO)(NC(=O)CC(CC)C2CCC2)C1 93881,c1(C(N2CC(C)CC(NC(c3n(CC)c(O)nc3)=O)C2)=O)c(F)ccc(F)c1O 93882,c1(SC)cccc(CCNC(=O)NCc2nn(C)cc2Br)c1 93883,N1(C(C(C(C)C)NC(C)=O)=O)CC2CCCN(C(=O)C(CC(C)C)C(N)=O)C2C1 93884,c1(C(N2CCC(CNC(c3ccccc3NCCO)=O)C2)=O)ccc[n+]([O-])c1 93885,c1(C(N2CCCC2)CNC2CC2)ccc(Cl)c(F)c1.CN1CC(CN2C(=O)N2)C1 93886,C(N=c1[nH]c(=NC(C)C(C)F)[nH]c2cccnc12)c1cc(OC)nn1C 93887,C1(n2cc(SCC(=O)NCC(C(C)C)CN3CCC(C)C3)nn2)CCCCNC1 93888,c1(CC(=O)NC(CN(C(=O)C=C(C)c2ccsc2)CC)C)cc[nH]c(=N)c1 93889,c1(OC)cc(CCNC(C2C3CCCC3CN2C)=O)cc(OC)c1OC 93890,Cc1ccc(C=CC(=O)N(CC(O)CNC(C2(C)CNC(=O)C2)=O)C)cc1Cl 93891,N1(C(C(n2ncc(C)c2)C)=O)CC=CC(C(=O)NCCN2CCC(C)C2)C1 93892,N1(C(c2ncc(I)s2)C(=O)NCCCCCC)Cc2ncsc2C1 93893,N1(C(CNc2ccn(C)n2)=O)CCCCC1CCCNC(=O)CSC(F)F 93894,CC(CC(=O)NCCC(C)NC(=O)Cc1csc(-c2ncccn2)n1)C(C)(C)C 93895,C(=O)(CC(C)(C)C(=O)N1CC2CC(NC(c3ccnnc3Cl)=O)C2C1)OCC 93896,N=c1[nH]nc(CC(=O)NC2CCC(NC(=O)CCN3CCC(F)C3)C2)s1 93897,C1(NC(c2ccc(F)cn2)=O)(CNC(=O)C(O)Cc2ccccn2)CCOCC1 93898,C(CCCCCC=C)NC(C(CN(C(c1c(C#C)c[nH]n1)=O)C)C)=O 93899,N1(C(C2C(C)(C)NC(=O)C2)=O)CCOC2(CCN(C(=O)CCCCO)CC2)C1 93900,C1(CC)CCN(C(=O)Nc2cccc(C3COC3)c2)C(CC)C1 93901,C(C1c2ccsc2CCN1C(c1ccc(F)cc1)=O)NC(CN(C)C)=O 93902,C1(CNC(Cc2c(C)noc2C)=O)C2CCC(C2)N1C(c1[nH]nnc1C1CC1)=O 93903,C1(OC)CCCC(C(=O)C(C#N)C(=O)N(C)CCOc2cc(C)ccc2C)CC1 93904,c1(OC)ccc(C(N2CCC(NC(C3CC34CC4)=O)C2(C)C)=O)cc1CC1CC1 93905,N1(Cc2c(OC)ccc(O)c2)CCC2CN(C(=O)CSc3nc[nH]n3)CCC12 93906,C#CCCS(C)(=O)=NC(=O)Cc1cc(F)cc(Br)c1 93907,C1(C)(C(=O)NCC2(OC)CN(C(=O)CCc3cccc(C)c3)C2)CCC(C)C1 93908,C12(C(=O)NCC3(NC(=O)CCc4cncs4)CCOCC3)CCCCC1C2(F)F 93909,C1(NC(CCn2ncc(C)c2)=O)CCN(C(=O)C(F)C(C)C)CC1(C)C 93910,Cc1nc(C(=O)N(C)C)ccc1C(N1CC(C2(N(C(=O)CO)C(C)C)CC2)C1)=O 93911,N1(C(c2cc[nH]n2)=O)CCC2(CCN(C(C3CCC4(CCC4)CO3)=O)CC2)C1 93912,C1(C(=O)NCCc2ccc(C)cn2)CCC2(CC2)N1C(c1ccco1)=O 93913,N1(C(C(C)n2cccc2)=O)CCCC(C(=O)NC2CCCC(O)C2)CC1 93914,C1(COC)(CNC(=O)C(C)(C)N(C)C)CCCN1C(C1CC(=O)C1C(C)(C)C)=O 93915,Fc1c(Cl)c(CC(c2ccccc2)NCc2ccc3occc3n2)ccc1Cl 93916,c1(C(=O)OC)ncc(Br)cc1NC(C1CCN(C(=O)C(=O)c2ccco2)C1)=O 93917,c1(C(=O)NC(C)CCNC(=O)C(C)c2cccs2)ccn2c1CSCC2 93918,c1(C(N2CCCC(CN(C)C(C3CC4(C3)CC4F)=O)C2)=O)c(F)cc(O)cc1F 93919,C1(S(=O)(=O)NC(=O)CN(c2ccccc2)C)(OC)CC1 93920,c1(C(N(C2CN(C(c3ncccc3Cl)=O)CC2F)C)=O)scc2c1OCCO2 93921,C(=O)(C(C)(C)C(N)=O)N(C1CCN(CC(=O)N(CC#C)CC)C1)CC#C 93922,N1(C(CNC(N)=O)=O)CCCCC1C1CCN(C(C23CC(CF)(C2)C3)=O)CC1 93923,c1(NC(=O)NCCCC(C)c2ccccc2)ccc2c(c1)nc(C(=O)N(C)C)n2C 93924,c1(C(CCC)NC(c2sccc2Br)C)cccc(C(F)(F)F)c1 93925,Cc1cc(C(=O)NC2CCCC(CNC(=O)Cc3ccnc(F)c3)C2)nc(C)n1 93926,c1(C(=O)NC(C)CN(C)C)ccc(SC2CC2Cl)cc1F 93927,c1(NC(C2CCCN(C(CCNC(=O)OC(C)(C)C)=O)C2)=O)ccc(C#N)c(Cl)c1 93928,CC1OCCOC1C(=O)NC1(CO)CCN(C(c2cnn(C)c2Cl)=O)C1 93929,CCC(C(=O)NCC1CC1NC(c1cn2ccnc2cn1)=O)C(F)(F)F 93930,C=Cn1nncc1C(=O)NCC(CC(=O)NCC(C)C(F)(F)F)OC 93931,c1(CC(=O)NC2(CCNC(C3(C(=O)NC)CC3)=O)CCC2)cccc(F)c1Cl 93932,C1(CNC(c2scc(OC)c2)=O)CN(C(=O)C=C2CCSCC2)CCN1C 93933,c1(OC)ccc2c(c1)OC(C)(C)CN(C(C1CN(C)CCO1)=O)C2 93934,c1(C(=O)NC(C(CO)NC(C(c2cccc(C(F)F)c2)C)=O)C)ccc(F)cc1F 93935,c1(C(=O)NCC(CNC(C2CCOC2)=O)OCC)cccn(CC(F)(F)F)c1=O 93936,c1(CN2CCCC(C(N3CCC(CCOC)CC3)=O)C2)ccc(I)cc1F 93937,C1(CC)CC(O)CCN1C(C1COCC1NC(c1coc(C)c1)=O)=O 93938,N1(C(C2(CO)CC(C)(C)C2)=O)CCCC(F)(C(=O)N(C2CCOCC2)CCO)C1 93939,n1(CCCC(=O)NC(C)C(c2ccccc2)NC(=O)C2=CCC2)ccccc1=O 93940,C1(C(N2C(CNC(=O)CCCC3CC3)CC3(CC3)C2)=O)CCc2nncn2CC1 93941,c1(N(C)C)sc(COCCNC2CCN(CC=C)C2)nc1C.C1CCC(=O)O1 93942,c1(C(=O)NC2C(CNC(C3(C(C)C)CCC3)=O)C2)cnn(C)c1-n1cccc1 93943,CCS(=O)(=O)CC(=O)NC(CCC1CC1)C(=O)NC1(CSC)CC1 93944,N1(C(C(C)OCC2CC2)=O)CCC(CNC(c2cc(O)n(C)n2)=O)C(O)C1 93945,C1(CCCCCNC(CCC#C)=O)CCN(C(c2ncn(C)c2C)=O)CC1 93946,N1(C(COCc2cc(C)no2)=O)CC(CNC(=O)C=C2CCSCC2)CCC1C 93947,c1(C(C)(C)OC)ccccc1C(N1CCC(N(C)C(C2CCCC2(F)F)=O)C1)=O 93948,n1(C(CC)CCO)cnc2c(N(C3CCOCC3)CCF)ncnc12 93949,C12(NC(C3CC(OC)C3)=O)CCCC1N(C(c1csc3nccn13)=O)CC2 93950,C1(NC(C(C)=CC2CC2)=O)CC1C1CCN(C(c2nccc3n[nH]cc23)=O)CC1 93951,c1(CN(C)C)ccc(C(=O)NC2(C)CCN(c3nnc(C4CC4)o3)C2)cc1 93952,C1(C(=O)NC(CC)(C)C2CC2)CC12CCN(C(=O)C(O)CC(F)(F)F)CC2 93953,Cc1ccc(C(F)F)cc1C(=O)NC1CC(C)(NC(=O)CC2CC=CCC2)C1 93954,c1(C(N2CCC(C(C)C)C2)C(=O)NCCC)c(C)nn(-c2ccc(F)cc2)c1Cl 93955,S(=O)(=O)(c1cccs1)N1CCC(C(N2CCC2C(F)(F)F)=O)CC1 93956,C1(CC(=O)NCC(CSCC)(F)F)CCC2(CC1)COC2 93957,C1(CNC(CCC2CCC(C)O2)=O)CCC2(CN(c3ccnc(C#N)n3)C2)O1 93958,CC1CCN(C(C2(C)CCOC(C)C2)=O)CC1CNC(c1nccnc1Cl)=O 93959,C(C(C)CN=c1ccnc(N2CCCC(COC)(OC)C2)[nH]1)OC 93960,C1(C)(C(N2CCC(NC(C3(COC)CC(=O)C3)=O)CC2)=O)CCN(C)C1=O 93961,CCC(CNC(C12CC(CC(F)F)(C1)C2)=O)(CC)NC(c1cn(CCO)nn1)=O 93962,c1(C(=O)OC)sccc1S(=O)(=O)Nc1cc(C(=O)O)cc(C(C)C)c1 93963,C1(NC(C=NOC)=O)(CNC(=O)C(C2CC2)OCC)CCCCC1 93964,CCC(C)(C#N)C(=O)N1CC(NC(c2ocnc2C2CC2)=O)C(C)C1 93965,Cc1ncc(C(N2CCC(CCNC(=O)Cc3csc(C)c3)C2)=O)c(C)n1 93966,c1(CC(N2C(CNC(C(CC)C(C)C)=O)COCC2)=O)c[nH]c2cnc(Cl)cc12 93967,c1(SCC)cc(CC(N2CC(C(=O)OC)C2)=O)cs1 93968,c1(C(=O)NCC2(OC)CCN(C(C3CC4CCC3O4)=O)C2)cnc2ncccn12 93969,C(=O)(C(CCC(C)(C)C)OC(c1cc(O)ccc1Br)=O)OC 93970,N1(C(c2ccc(COC)[nH]2)=O)CC(C)CCC1CNC(c1nccc(C)n1)=O 93971,C1(CNC(c2ccc(C(C)(C)C)s2)=O)CN(C(=O)C2CC2)CC1C(F)(F)F 93972,C1(CCC)CN(C(=O)C(CC)Oc2ccccc2)CCN1C(c1cc[nH]c1)=O 93973,C(=O)(C(O)CCCNC(c1c(C)ccnc1O)=O)N1CC(CC)OCC1 93974,N1(C(c2c(CC)cc(N)cc2)=O)CCCC2(NC(c3ccc(OC)s3)=O)CC2C1 93975,c1(NC(C)=O)ccc(CC(=O)NCC2CCC(NC(c3ccsc3C)=O)C2)cc1 93976,C1(C(=O)NC(CSC)(C)C(=O)Nc2cccc(N(C)C)c2)CCCCNC1=O 93977,CCCC(O)CNC(=O)C(=O)NCc1cn(C2CCCNC2)nn1 93978,C1(NC(C2(C)CC(F)C2)=O)CCCCC1NC(=O)CSc1ccccc1Cl 93979,C1(C(=O)NCCC(C)NC(C(C)Cc2cccc(F)c2)=O)CC(C(C)(C)C)=NO1 93980,c1(NC(c2c(CNC(C(C3CCC3)OCC)=O)ocn2)=O)ccc(O)c(C)c1 93981,N1(C(c2cc(OC)ncn2)=O)CCOC(C)(CNC(=O)Cc2cccnc2C)C1 93982,CN1CCC(N(C(c2cc(Br)cs2)C(=O)NC(C)(C)C)C)C1 93983,CC1(C)CC(CNC(=O)CCc2nc[nH]n2)CCN1 93984,c1(CC)cc(N)ccc1C(=O)NCC1CCCCN1C(=O)CCc1cnc(O)[nH]1 93985,c1(NC(=O)NC(CSC)C)cc2cccc(F)c2cn1 93986,c1(-c2cncc(NC(C3(c4cccc(Br)c4F)CC3)=O)n2)ccc([N+](=O)[O-])cc1 93987,c1(C(=O)OC)cnc(C)[nH]c1=NCCC(C)NC(=O)C1CCCc2n[nH]cc21 93988,CCCC(CNC(C1CC(C(=O)OC)C1)=O)C(=O)N(CCCC(O)CO)C 93989,C1(NC(C2N(C(c3ccc(CSC)o3)=O)CCOC2)=O)CC2(C1)CN(C(C)=O)C2 93990,C1(NC(C2CCS(=O)CC2)=O)CCCN(C(=O)CCC2CCCCC2)CC1 93991,N1(C(N)=O)CC(CO)C1.C1(=O)CN1.C12(CC1)C(C)NC(=O)N(C)C2 93992,Cc1cc(F)c(C(N2CCCC2CN(C)C(C2CC=CC2)=O)=O)cc1F 93993,n1(CC)cc(CNC(C2CN(C(c3ccc[nH]3)=O)CCO2)=O)c(C)n1 93994,c1(OC)ccc(NC(=O)C2CC2)cc1NC(=O)NCc1ccccc1CCCl 93995,c1(OC)ccc(C(N2CC3CCC2C3NC(=O)C#CC(=O)N(C)C)=O)c(N)c1F 93996,N1(Cc2cc(COC)no2)CCC(=O)N(CCC(C(F)(F)F)OC)C1=O 93997,C1(NC(=O)C=Cc2cscn2)CC2CCC1(CNC(c1cc(Cl)c[nH]1)=O)C2 93998,c1(C(=O)NC(CNC(C2(COC)CCCO2)=O)C)ccc(Cl)c(N)c1 93999,N1(C(c2nc(CC)sc2)=O)C2CCC1C(NC(c1cnc(C(F)(F)F)nc1)=O)C2 94000,C(CCNC(=O)CN)(C(N)=O)NC(COC(CC)CC)=O 94001,c12ncc(F)c(n1)OCC(=O)N2.C1(CCCCNC(C)=O)CCN(C(C)=O)CC1 94002,Cc1oc(C#N)cc1C(N1CC(O)(C(F)C(N2CCCC(C)(O)C2)=O)C1)=O 94003,Cc1nc2ccc(C(N3CCCN(C(C45CC6CC4C5C6)=O)C(C)C3)=O)cc2[nH]1.O(F)C 94004,CC1CSc2ccc(Br)cc2C1NC(c1c(N)sc2c1CCC2)=O 94005,c1(C(N2CCCCC(CNC(C3(C4CCC4)CC3)=O)C2)=O)cccn2cnnc12 94006,N(C(=NCc1ccn(CCOCCSC)n1)NCC)C(c1cnc(CC)o1)C 94007,CC(CCc1ccccc1)CC(=O)N(C1CCN(CC2CCCO2)CC1)CCO 94008,n1(C(CC)C)nccc1NC(=O)CNC(c1ccc(C)s1)=O 94009,C(=O)(CN=c1cc[nH]cc1)NCC1CCN(C(c2c(CC)noc2)=O)C1(C)C 94010,c1(CC(N2C(CNC(c3ccsn3)=O)CC3CC32)=O)cc2ccccc2o1 94011,c1(C(N(C2CCC(NC(CCOCCOC)=O)C2)C)=O)csc2cccnc12 94012,C1(C(N2CC3C(CNC(c4c(C)ccs4)=O)(C3)C2)=O)C(O)C(=O)N(C)C1C 94013,CC(C)(O)CC(=O)NC1CC1NC(C1(c2ccc(O)nc2)CCC1)=O 94014,c1(CC)ccc(C(=O)NCC2CCCCCN2C(C2CCC(=O)C2)=O)cc1Cl 94015,Cc1snnc1C(N1CC(c2ccccc2)(NC(c2cc(CO)on2)=O)C1)=O 94016,C(=O)(CS(=O)(=O)c1ccccc1Cl)NC(CNC(C1N2CC(C)N(CC2)C1)=O)C 94017,CCC(CCC(=O)NCCCC(C)NC(=O)CNS(N)(=O)=O)OC 94018,N1(CCC(=O)OC(CN(C(C)=O)C(C)C)OC)c2ccccc2Sc2ccccc21 94019,Cc1nc(O)nc(C)c1C(=O)NCC(C)(O)CNC(C1CC=CCO1)=O 94020,C1(C(=O)NCCC(C)(C)NC(COC(CC)C)=O)CCc2ccc(F)cc2O1 94021,Nc1ccc(C(=O)NC2CC(CCC(=O)NCC(F)CO)C2)nc1F 94022,C1(CNc2nc(C)cc(CCNC(CSC)=O)n2)CC2CCC1N(C(C)=O)C2 94023,N1(C(CSC2C(=O)OCC2)=O)C2CCC1CC(NC(c1ccc(O)nn1)=O)C2 94024,c1(CC(N2CC(CNC(CCOC(C)=O)=O)C2)=O)ccc2c(c1)COC2 94025,N1(C(c2cc(C)cc(F)c2)=O)CC(NC(c2cccc(C)n2)=O)C2CCCC12 94026,C1(NC(C2CC(OC)C2)=O)C2CC(NC(=O)CCC3NC(=O)NC3=O)CC12 94027,c1(C(=O)NC2(CNC(C(C(C)C)F)=O)CC(F)(F)C2)nccc2n[nH]cc12 94028,c1(C2(C(C)(C)O)CC2)cn(CC(N2CCC(N3CCC3)C2)=O)nn1 94029,N1(C(c2ccn(CCC)n2)=O)CC2CC1(C(=O)N(CC(C)CO)C)C2 94030,CCC(C)(C)C(=O)N1CCCC(CCNC(=O)C(C)COc2ccccc2)C1 94031,c1(C(=O)NC2CCCN(C(C(C)N(C(C)=O)C)=O)CC2)cc2ccc(F)cc2[nH]1 94032,CN1CC(C)(C(=O)NC2CC(NC(c3cccc(OC(F)F)n3)=O)C2)CC1=O 94033,C1(C(=O)NC2(CSC)CCC2)CN(C(C2(C)CC(F)(F)C2)=O)CC1F 94034,c1(SC)cccc(C(=O)NC(C)(C)CCCNC(=O)Cn2cnnn2)n1 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94053,C=CCC(C(=O)N1CCC(CN(C(=O)C(CC)NC(N)=O)C)CC1)C(C)C 94054,C1(CCNC(CCOCC)=O)CCCN(C(C2CC(C)(C)C2)=O)CC1 94055,C1(C(=O)NCc2noc(C3CC3)n2)CC(=O)CN1C(=O)CC(O)C1CCCC1 94056,C1(C(C)(C)C)CC(N=c2[nH]c(=NCC=CC3CC3)[nH]c3cccnc23)CCO1 94057,C1(O)(C(N2CC3(C(=O)OCC)C(C2)CCO3)=O)CCc2ccccc2C1 94058,N1(C(c2cc(C(C)C)nc(O)c2)=O)CC2CCC1CN2C(=O)C=CC1CCOC1 94059,C1(NC(=O)CO)CC2CC1CN(C(=O)CCc1nc(O)n[nH]1)C2 94060,C1(NC(CC2CC(=O)OC2)=O)CCOCC1C(N1CC=CC1)=O 94061,Cc1ccccc1OCCNC(C1CCCCN1C(C1(F)CCCCC1)=O)=O 94062,c1(OCCC)ccc(CNc2ccc(OCC)cc2)nn1.C1CO1 94063,Cc1cccc(CNC(=O)C(CNC(C2(C)CCC3CC3C2)=O)C(C)C)c1C 94064,C1(NC(c2c(OC)cccc2)=O)CN(C(C2CC(C)(C)C2)=O)CC2(CCC2)C1 94065,C(C(CC(C)C)C(=O)N1CCC1CNC(c1cc(Cl)cc(Cl)c1OC)=O)OC 94066,C1(NC(c2cnsn2)=O)CC2CC(NC(c3ccnn3CCF)=O)C2C1 94067,N(C)(C1CCc2c(Cl)cccc21)C(c1ncc(C)s1)C(=O)NC(C)(C)C 94068,C1(CNC(C2CN(C)C2)=O)CC2CCC1N2C(C1(c2ccccc2)CCOCC1)=O 94069,CCC(C(=O)N(CC(C)NC(c1cnn[nH]1)=O)C)OC 94070,c1(C(=O)NCC2C=CC(NC(=O)CCSC(F)(F)F)C2)sc([N+](=O)[O-])cc1Cl 94071,N1(C(C(c2n(C)ncc2)O)=O)CCC2(CC1)CC(NC(C1(C)CCC1)=O)C2 94072,CC1CN(C(=O)COCCOCCO)CC1CNC(=O)Cc1ccnn1C 94073,N1(C(c2n(C)ncc2)=O)CCC(C(=O)NCC2C=CCC2)CC1 94074,c1(C(=O)NCCN(C(c2ccc(OC)c(Cl)n2)=O)C2CC2)c[nH]nc1S(N)(=O)=O 94075,O=C1NCCn2nc(C(=O)NC3CS(=O)(=O)CC3Nc3ncc(Cl)cn3)cc21 94076,CC1(C)OC2C3CC(C2O1)N(C(C1CCC(=O)C1)c1ccccc1)C3 94077,N1(C(c2c(OC)cc(C)s2)=O)CCCOC(CCNC(C2CC2[N+](=O)[O-])=O)C1 94078,C1(C(N2CC3CCC2CC3)=O)(N(C(=O)OC(C)(C)C)C2CC2)CC2CCC1C2 94079,C(=O)(C(CC)CC(C)C)NCCCOCCNC(CCCC(=C)Br)=O 94080,C1(NC(C2CC(=C)C2)=O)CCC2CCN(C(c3ccc(-n4cnnc4)c(N)c3)=O)C12 94081,c1(C(=O)NCCN(C(=O)CC(C)(C)CCOC)CC)cc(C)c(C)c2ncsc12 94082,N1(C(C(CCC)C#N)=O)CCC(C)(C)CC1C(=O)NC(c1ncc(C)cn1)C 94083,N1(C(c2cc3ccccn3c2)=O)CCC2OCCN(C(C3CC4CC4C3)=O)C2C1 94084,C1(COC)CN(C(c2ccsc2Cl)=O)CCN1C(=O)C#CC1(C)CC1 94085,C1(C(=O)NC2CC(NC(c3ncnc(C)c3C)=O)CC2O)CCN2CCCC2C1 94086,CC1CN(C(c2csc(Br)c2)=O)CC1NC(C1(C)CC2(CC2)C1)=O 94087,C1(O)(C(=O)NCc2cn(CC(C)NC(c3cc[n+]([O-])cc3)=O)nn2)CCSCC1 94088,N1(C(CN(C(C(C)C)=O)C)=O)CCOC(CNC(=O)CCC2CCCC(=O)N2)C1 94089,N1(C(=O)CCN2CCC(O)CC2)CC2OCC(NC(C34CC(CO3)C4)=O)C2C1 94090,C1(C(N2CCC(NC(C3(CO)CC3)=O)C(O)C2)=O)CN2CCCC2CO1 94091,C(C(=O)NC1CCCCC1NC(=O)CCOC1CCC1)(C(C)C)OCC 94092,C1(C(=O)OC)C(C(=O)OC)C2CCC1N2Cc1ccccc1Br 94093,C(=O)(C(C)CC(F)(F)F)NC1COCCN(C(CC(COC)C)=O)C1 94094,N1(C(C(CC(C)C)C(N)=O)=O)CC(NC(=O)C2=CCCCO2)CC12CCCCC2 94095,C12(C(=O)NCC(CNC(c3coc(C4CC4)n3)=O)F)CCC(CO)(CC1)C2 94096,Cc1c(NCC(c2cccc(F)c2)(C)C)ncnc1N1CCC(C)(CO)CC1 94097,C(=O)(CCCCC(C)=O)NCC1CCN(C(c2ncc(CC)cn2)=O)CC1C 94098,c1(OC)cccnc1C(=O)NCCC1(OC)CN(C(C2CC(CC)=NO2)=O)C1 94099,c1(OCC(C2CCOC2=O)=O)cc(N2CCCC2=O)ccc1O 94100,c1(OC)c(F)ccc(C(=O)NCC2CCC2NC(c2ccsn2)=O)c1F 94101,c1(CCC(=O)NCCC(CNC(C2(COC)CCC2)=O)O)cc2ccccc2o1 94102,C1(C(=O)NC(C=C)C)OCCC1CNC(C1(OC)CCC1)=O 94103,Cc1c(CNC(C2COCCN(C(c3cnsn3)=O)C2)=O)cccc1O 94104,C1(C#N)(C(N2CC(COC)(NC(=O)CC3CCC4CC34)C2)=O)CCCCC1 94105,C1(C(N2CC(O)C(O)C2)=O)(CC)CCCN(C(c2ncccc2N)=O)C1 94106,CNS(=O)(=O)N1CCC(C(N2CCCC2CCNC(=O)CC(C)COC)=O)CC1 94107,c1(C(N(C2(C3CCCN3C(=O)CCc3cnn(C)n3)CC2)C)=O)cc(F)cc(F)c1 94108,Cc1[nH]c(C#N)cc1C(=O)NC1CN(C(=O)C2=CC(C)(C)C2)CC1C(F)F 94109,CCCCC(C(=O)NC1CC(=O)N(C2CN(c3ccc(Br)cc3F)C2)C1)NC(N)=O 94110,c1(OCCC(=O)NCCC(F)Cn2cc(C3CCCCO3)nn2)ccccc1Cl 94111,C1(NC(c2nn(CC)c(O)c2)=O)CN(C(=O)Cc2ccccc2O)CC2(CC2)C1 94112,c1(OC)ccn2cc(C(=O)NC3(C)CN(C(=O)C4=CCCCC4)C3)nc2c1 94113,n1(CCC)cccc1C(N1CC(CCO)(NC(=O)C(CSC)OC)C1)=O 94114,C12(C(=O)NC3CCN(CC)C3)C(NC(c3cnc(S)nc3)=O)C3CC1C2C3 94115,C1(C(=O)NCC2(C)CCN(C(c3nc(NC(C)=O)sc3)=O)C2)COC(C)(C)CO1 94116,CCCC(C)(C)CC(=O)NCc1cc(C(=O)NC2CCCC(CC)CC2)ccn1 94117,c1(C(=O)NCCC(=C)CNC(c2ccc(C(C)C)nc2O)=O)ccc(Br)cc1C 94118,C1(CC)(CNC(CN2CC(CNC(=O)CSC(C)C)C2)=O)CCCC1 94119,C1(NC(COC(C)C)=O)CCCCN(C(C2(Cl)CC2(F)F)=O)CC1 94120,c1(CC(=O)NCCN(C)CCF)n[nH]c2cc(Cl)ccc12 94121,N1(C(C(C)(C2CC2)OC)=O)CCC2(CCCCC2NC(=O)CCC2CC2)C1 94122,C12(CC(=O)N(C)CCNC(=O)C=CC3COC(C)(C)O3)CCCCC1C2(F)F 94123,N1(C(C=CCC(C)(C)NC(c2n(C)cnc2)=O)=O)CCOCC(C(N)=O)C1 94124,c1(CN(c2ccnc(Br)n2)C(=O)CSC2CCCN2)ccc(Cl)cc1 94125,C(c1ccc(Br)o1)=C(C)C(=O)NCC1CC1CNC(c1ccc(=N)[nH]n1)=O 94126,N1(C(c2cc(OC)no2)=O)CCN(C(c2ccccc2)=O)C2CCCC12 94127,C(C)(C)(C#CCCCC)NC(C1(N(C(COC2(C#C)COC2)=O)C2CC2)CCC1)=O 94128,C1(CC)CN(C(=O)CN(C)C)CCC1NC(=O)C(c1cccc(C)c1)(F)F 94129,CCC(C(=O)NC1CC(CO)N(C(C2CNC(=O)O2)=O)C1)C(C)C 94130,N#CC1(Cc2cc([N+](=O)[O-])cs2)CCN(Cc2ccc(NC(=N)N)cc2O)C1 94131,c1(CNc2ccc(NC(C3CC(=O)NCC3)=O)nc2)cn2ccccc2n1 94132,CC(C)CC(CNC(c1cnn(C(C)C)c1)=O)C(=O)NC1CCSCC1 94133,N1(CC)C2CCC1CN(C(C1(NC(C3CCC(C)=C(C)C3)=O)CCOCC1)=O)C2 94134,Cc1cccc(C2CCCCN2C(=O)C(=O)NC2COCCC2n2cccn2)c1 94135,C1(OC)CC(CNC(c2cncc(C(F)F)c2)=O)N(C(=O)COCC(F)(F)F)C1 94136,Cc1cc(Cl)ccc1OC(C)C(=O)NCCC1=CCN(C(=O)COC(F)F)CC1 94137,c1(C(N(CCCCCNC(C2(F)C(C)C2)=O)C)=O)cccc2c1NC(=O)CC2 94138,C1(C(=O)NC(C)(C)C(N2CCOCC(O)C2)=O)CC(=O)CC12CCC2 94139,c1(C(C(N2CC(O)(CCNC(CC3C(C)(C)C3)=O)C2)=O)C)nc(F)ccc1Cl 94140,CC1C(C)N(C(C2CCCS2)=O)CCN1C(c1cc(C2CCOCC2)[nH]n1)=O 94141,c1(Nc2ccccc2C(N(C)Cc2c(C)n[nH]c2)=O)cn(C)nc1N(C)C 94142,C(=O)(C(CCC1CC1)NC(=O)CSCC(F)F)NC(C=C)CO 94143,CC(C(=O)N1CCC(CC2CCC2)C1)S(C)(=O)=O 94144,C1(F)(CNC(CC)=O)CCC(CNC(C2CCC(C3CC3)C2)=O)CC1 94145,CC1CN(C(=O)C=Cc2cc(Br)cs2)CC1NC(C1(Cl)CC1)=O 94146,CCCCCCCCCCN(CCC)Cc1csc(C)n1 94147,N1(Cc2cccc(C(N)=O)c2)CCCC2(C1)CN(c1ncnc3n[nH]c(Br)c13)C2 94148,c1(C(N2CCC3(C(C(=O)NCCCCCO)C3)C2)=O)cccc2[nH]ccc12 94149,C(=O)(C(C)C(F)(F)F)NC(CCC)C(=O)NCC1(F)CC1 94150,c1(C(N(CCC)CCNC(=O)CC2CC=CC2)=O)coc2c(OC)cccc12 94151,c1(C(=O)NC2C(NC(c3n(CC)ccn3)=O)COC2)ccc(C)cc1Br 94152,Cc1ncc(N)cc1C(=O)NCCOCCNC(C12CCC(O)C1CC2)=O 94153,c1(C(N2CCCC2C)C(=O)NCCCSC)cc(C(F)(F)F)ccc1C 94154,N1(C(c2c(C)c(CO)ccc2)=O)CC2CC(NC(c3n[nH]cc3Cl)=O)C(C2)C1 94155,c1(SCC(=O)N(CC(CNC(C(c2ccccc2)OC)=O)O)C)cnn(C)c1 94156,c1(C(c2nc(-c3cccnc3C)no2)OC)ccc(C)c(F)c1 94157,c1(C2C(C(=O)OCC)C2C(C)C)ccc([N+](=O)[O-])c(N)c1 94158,Cc1cnccc1CN1CCC(NC(=O)N(c2ccccc2Br)C)CC1 94159,C1(C(N2CCC(CC(C)NC(=O)C3CC3)CC2)=O)CCCCC1(C)C 94160,Fc1ccc(N2CCN(CCCC3CC3)CC2)cc1 94161,Oc1ncccc1CN(Cc1ccccc1)CC1CC1C1CC1 94162,Cc1cc(C(=O)NC(C)CNC(C2(c3c(C)cccc3C)CC2)=O)c(N)c(C)c1 94163,Cc1cccc(-c2nc(C(=O)NC3CC(CNC(=O)C4=CCC4)CC3O)cs2)c1 94164,c1(C(=O)NC)cccc(C(N2CC(CNC(=O)C(C)c3ccsn3)C2)=O)n1 94165,Cc1cc(N2CCC(C(=O)OCCCCCOc3ccccc3)C2=O)ccc1F 94166,c1(NCC)ncc(C(=O)NC2(CCNC(C3CNC(=O)C3)=O)CC2)cc1Cl 94167,C(=O)(CC(O)CNC1CCS(=O)(=O)C1)N(CC)CC 94168,N1(C(CC2(OCC)CCC2)=O)CCCCC1CCNC(C1CC(N=[N+]=[N-])C1)=O 94169,Cc1oc(C(=O)NC2C3CN(C(c4cnc(O)n4C)=O)CC23)cc1S(C)(=O)=O 94170,N1(C(C(CC=CC)NC(c2ccn(C)c2)=O)=O)Cc2nc(C)sc2C1 94171,n1(CC(=O)NC(CNC(C2(OC)CCCOC2)=O)(C)C(C)C)ncc(O)nc1=O 94172,c1(C(=O)OC)sc(Cl)cc1S(=O)(=O)NC1COCCN(C(=O)CC(F)(F)F)C1 94173,S(=O)(=O)(c1ccc(N2CCC(CC3CC(NC)C3)C2)c(Cl)c1)NC(CC)CCO 94174,C=C1CCN(C(c2ccc(F)cn2)=O)C(C(=O)NCCN(C(C)C)C2CC2)C1 94175,c1(C(N2CCC(OCCNC(C3CCC3)=O)C2)=O)cnc(C2CC2)nc1 94176,C1(NC(c2cc(C)[nH]c2C)=O)CC(O)CN(C(C2CCC(C)O2)=O)C1 94177,n1(CC)nc(C)c(C(=O)NCC2CC(F)CN2C(=O)CC2C=CCCC2)c1Cl 94178,N1(C(CC2CCN(C(c3ccc(OC)cc3)=O)C2)=O)CCCN(S(C)(=O)=O)CC1 94179,C1(C2CN(C(c3cnc(C(F)(F)F)cn3)=O)C2)(NC(c2ccsc2)=O)CC1 94180,c1(C(C)(C)C)ccc(C(=O)NCC(C)(CO)NC(C23CCC2CC3)=O)nc1 94181,N1(C(COc2ccc(C#C)cc2)=O)CC(C)CN(C(C2(C)CC=CC2)=O)CC1C 94182,C1(OC)CC(CNC(c2cc(F)n(C)n2)=O)N(C(c2ccc(C#N)o2)=O)C1 94183,C(=O)(CCS(=O)(=O)C(F)(F)F)NC1C(NC(CC(C)(C)C#N)=O)COC1 94184,C1(C(=O)NCCCN(CC)CC)(CC)CCCN1C(c1n[nH]cc1C)=O 94185,CC1(C(=O)NCC2(NC(C3CCS3(=O)=O)=O)CCCC2)CCC(O)CC1 94186,C1(NC(C(COCC)C)=O)CN(C(c2cc(C)c(Br)o2)=O)CC1SC 94187,CC1(C)CC(C(=O)NCC2CN(C(=O)CCc3ccoc3)C(C)(C)C2)CNC1=O 94188,N1(C(CCSCC)=O)CC(NC(C2Cc3nnc(C)n3C2)=O)CC12CCOCC2 94189,C1(CNC(c2c(C)ncnc2)=O)CN(c2nc3ccccc3s2)CC2(CCC2)O1 94190,C1(OC)CC(CNC(c2cccnn2)=O)N(C(C2CC2OC(C)(C)C)=O)C1 94191,N1(C(Cc2c(OC)cccc2Cl)=O)CCCC2(CCc3ccccc32)C1 94192,C1(C(=O)NC(CCC)C(=O)NCC)CCN(C(=O)OC(C)(C)C)C12CC2 94193,C1(F)(CNC(C(C=C)O)=O)CCCN(C(c2ccc(C)cc2Br)=O)C1 94194,Cc1ccc(C(C)CC(=O)NCC2CCN2C(=O)C(C)(C)C23CC(C2)C3)cc1 94195,c1(C(N2C3(CNC(CNc4c(C)n[nH]c4C)=O)CC(C2)C3)=O)c(Cl)cccc1Cl 94196,N1(C(C(=O)NCCCSC)c2ccns2)CCOCC(CNS(C)(=O)=O)C1 94197,c1(OC)cncc(NC(c2ccnc(SC(c3ccc(C)cc3)=O)c2)=O)n1 94198,c1(C(N2CCCCC2C2CCCCC2)C(=O)NCCC)nn(CC)cc1Cl 94199,N1(C(c2c(C(C)C)cco2)=O)CC(CNC(C2CC2C)=O)OC(C)(C)C1 94200,C(=O)(CC(C)CCC=C(C)C)N1CC2(CN(CCC)C2)C1.c12ccc(c(O)c1)CN2 94201,c1(OC)ccc(C(=O)NC23CC(NC(C4CC45CCOC5)=O)(C2)C3)cc1O 94202,C1(CN(C(=O)CCCn2cncn2)CC)CCN(C(=O)Cc2cn(C)cn2)CC1 94203,c1(C(N(C2CCN(C(=O)C(C)CSC)C2)C(CSCC)=O)=O)ccccc1NC 94204,C[Si]1(C)CCN(C(=O)C(Cn2cncn2)NC(=O)Cc2cn[nH]c2)CC1 94205,c12cccc(c1)NC(=O)C2.c1(CCOCCOCC)ocnc1C(=O)O 94206,c1(C(N(C(C)CCNC(C2OCC2(C)C)=O)C)=O)cc(C2CC2)oc1C1CC1 94207,CCCCC(CC)CC(=O)NC1CCC(C(=O)NCC2(OC)CC2)C1 94208,N1(C(Cc2c(C)n(C)cn2)=O)CCN(C(c2ncc(N)cc2Cl)=O)CC1C 94209,c1(SCC(N2CCC(CC=C)(NC(=O)CC3(C)CC3)C2)=O)ccc2c(c1)CCC2 94210,C1(C(N2CCC2(C)C)=O)(OC)CCN(C(C2CCC(=O)O2)=O)C1 94211,c1(CN(C2CCOC2C)C(C)C)ccc(C(F)Cl)cc1 94212,C(=O)(C(C)(CC)CC)NC(C(=O)N1CCC(CCCC)C1)CCF 94213,C1(CC(=O)N(CCN=[N+]=[N-])C)C=CC(NC(=O)CCc2cccs2)C1 94214,C1(CC(=O)NCC(C)(C)N(F)F)CC(C)(C)CN1C(C1CC(=C2CC2)C1)=O 94215,N1(C(C2N(C(c3c[nH]nc3Cl)=O)CC23CCCC3)=O)CCCC(C2CC2)CC1 94216,c1(C(N2C(C)(CNC(C3=C(C)CCC3)=O)CCC2)=O)cc(Cl)c2ccccc2n1 94217,n1(CCC)ncc(C(N2CCOC(CNC(c3ccccc3Br)=O)C2)=O)c1C 94218,c1(C(=O)NCCCN(C(C2(COC)CCCO2)=O)CC)ccc2n[nH]cc2c1 94219,C1(NC(c2cc(OC)n(C)n2)=O)CCN(Cc2sc(Cl)nc2Cl)CC1OC 94220,c1(C(=O)NC2C(NC(CCCCC(C)C)=O)COC2)cc(F)cc2cnccc12 94221,CCC(CC(C)C)C(=O)NC1CCC1NC(C1(OC)CCCC1)=O 94222,N1(C(C2C(OC)C2)=O)CCN(C(=O)Cc2csc(Br)n2)CC(O)C1 94223,N1(C(c2cnc(C(C)O)s2)=O)Cc2c[nH]nc2C(C)(C)C1 94224,Cc1cc(C(=O)NC2CCCC(C(=O)NOCC3CCCCC3)C2)nc(C)c1 94225,CCC(C)(CCC(C)C)C(=O)N1CC2OCCN(C(=O)C=CC(C)(C)C)C2C1 94226,c1(CNC(C2CCN(C(C3CCC(N(C)C)C3)=O)CC2)=O)cc(=O)n2ncsc2n1 94227,c1(COC)cc(CN2CCOCC2C#N)ccc1OC 94228,C1(CNC(=O)C(F)=CCCF)C=CC(NC(c2cnc(C3CC3)s2)=O)C1 94229,N1(C(CCN(CC)CC)=O)CCC2(NC(=O)CCOCC(C)(C)C)CCCCC12 94230,C1(COC)(CNC(=O)CCC(C)(C)F)CCN(Cc2c(C)nsc2C)CC1 94231,c1(CC)cc(C(N2CCC(O)(CNC(c3cnc(CC(C)C)[nH]3)=O)C2)=O)c(C)o1 94232,CC(C)(CCCC(=O)N1CC2(CCCCC2)C1)NC(=O)Cn1cccn1 94233,C1(CNC(c2nc(-c3ccc(Br)cc3)ns2)=O)CCCN(c2ncccn2)C1 94234,c1(C(N(C)CC2N(C(C(C)C3CC3)=O)CCOC2)=O)cnn2c1CCC2 94235,CCC(C#N)(CC)C(=O)N(C)CC1CN(C(=O)CCN2CCC(F)C2)CC12CC2 94236,c1(CCCC(=O)NCCNC(C2COCCO2)=O)c[nH]c2ccccc12 94237,C1(CC)CN(C(c2ccc(NC(C)=O)cc2Cl)C(=O)NCCC2CC2)CCN1C 94238,N1(CC)CC(C(N2CCC(CCNC(=O)CC(C)F)CC2)=O)CCC1=O 94239,c1(C(N2CCC(O)(CN(C(=O)CN3CC4CC4C3)C)C2)=O)ccc(F)c(O)c1F 94240,c1(-c2c(C(N(C)CC3CCN(C(C(CSC)C)=O)C3)=O)occ2)ccc(F)cc1 94241,c1(NC(C(=O)NC2(CN(C(CC(C)C)=O)C)CC2)=O)ccc(C#N)c(Cl)c1 94242,N1(C(c2cc(C)oc2)=O)CCC(NC(c2cnn(C)c2)C)C(C)C1 94243,c1(OCCCC(=O)NC(CNC(CC=CC)=O)COC)ccc2c(c1)CCC2 94244,c1(-c2c(NC(c3cc[nH]n3)=O)ccc(C)c2)cc(CO)c2cc[nH]c2c1 94245,C1(NC(Cn2c(C)cnc2)=O)CCCC2CN(C(c3ccc(=O)n(C)c3)=O)CC12 94246,C1(NC(CSCC#C)=O)CC2CN(C(=O)C(C)CC3CCCC3)CC2C1 94247,C1(C(=O)OC)CCN(C(=O)CSc2cc(Cl)ncc2OC)CCC1(F)F 94248,c1(CN2CC(CNC(c3cocn3)=O)C2)cccnc1O 94249,C12(C(N(N3CC(CC4(Oc5ccccc5)CC4)C3)C)=O)CC(C(F)F)(C1)C2.COC 94250,O=C1C=C2CN(C(C34CC(C(=O)NC(c5cnccc5Cl)=O)(C3)C4)=O)CCC2S1 94251,c1(C(N(C(C)CNC(c2cccc(Cl)c2OC)=O)CC)=O)cc(Cl)cc(C)c1N 94252,c1(C(N(C(=O)C(C)c2nccs2)CC)C2CC2)cccc(Br)c1 94253,N1(CCCNC(N2CC=CC2CF)=O)CCOCC1 94254,Cc1ncsc1CCC(=O)NC1CC(CCNC(C2(CO)CCC2)=O)C1 94255,C1(C2CCCN(C(=O)C(O)C3CC3)C2)(NC(CSC(C)C)=O)CC1 94256,CC(C)S(=O)(=O)CC(=O)NC1CC(CCNC(c2ccc(N(C)C)cc2Cl)=O)C1 94257,C1(C(=O)Nc2c(OC)nccc2)CC2(CC(NC(=O)C(C)S)C2)C1 94258,C(C)(C(=O)NNC(=O)NC12CCCC1C2)c1ccc(OC)c(F)c1 94259,O=C(CCC=CBr)NCC1CCCC(NC(c2ccnc(C3CC3)c2)=O)C1 94260,N1(C(c2cc(C)on2)=O)CCN(C(C2COC3COCC3O2)=O)CC(O)C1 94261,N1(C(c2ccc(C(C)=O)cc2)=O)C2CCC1CC(NC(c1cc(Cl)cnn1)=O)C2 94262,C1(NC(C2CC(OC)C2)=O)CCCC2CN(C(=O)CCn3c(C)csc3=O)CC12 94263,c1(C(=O)NCC2(O)CN(C(=O)CC3CCC(O)C3)C2)cnc2c(c1)COCC2 94264,C(=O)(CCCCCN(C(=O)C(C)SCC)C)N1C(C#C)CC1 94265,C1(NC(C2C(CC)C2)=O)CC2(CCCCN2C(c2cn3cccc(Cl)c3n2)=O)C1 94266,C1(C(=O)NCc2cscn2)CC2(C1)CN(C(=O)C(c1ccccc1)O)C2 94267,Cn1ncc2c(NCC3COCC4(CCC4)O3)[nH]c(=NCC3(S(C)=O)CC3)nc12 94268,C12(c3cc(NC(CCSCCCCCCCC)=O)[nH]n3)CC3CC(CC(C3)C1)C2 94269,c1(C(=O)NC2C(NC(C3C(=C)C3)=O)CCC2)cn(C)[nH]c1=N 94270,N1(C(C2CCC(SCC)CC2)=O)CC2CCC(NC(C3CC4C=CC3C4)=O)C2C1 94271,c1(SC)ncc(C)c(N2CCCC(C(N3C(CO)CCC3C)=O)C2)n1 94272,C1(C(=O)NCC2(CCNC(c3cc(-c4ccoc4)[nH]n3)=O)CC2)CCCCS1 94273,c1(CC(=O)Oc2cc(C(C)=O)c(Cl)cc2)cccc2sccc12 94274,c1(C(=O)NC(CCCC)CNC(C2C(C)C2C)=O)cccn2ncnc12 94275,CCCCCCCC(=O)N1CCC1C(=O)Nc1ccc(C(=O)NC)nc1 94276,c1(N2CCC(C(C(=O)OC)F)CC2)nnc(C2CCc3c[nH]nc32)n1CC(C)C 94277,c1(Sc2c(-n3cc(CNC(CCCCSC)=O)nn3)cccc2)cc(C)cnc1F 94278,C(CC(O)C(F)(F)F)NC(C=CCN(C(CCCOCC=C)=O)C)=O 94279,C1(C)(CNC(C(C)SC)=O)CCN(C(c2cncc(CO)c2)=O)C1.C(N)=O 94280,CC(c1ccco1)=CC(=O)N(C1(CC(=O)NC(c2nc(C)no2)CO)CC1)C 94281,C1(C2(NC(C3(C#N)CCN(C)CC3)=O)CCC2)(C(=O)NCC)CCC1 94282,N1(C(C)C(=O)NCC(c2ccccc2)NC(=O)CC2CCC2)CCC(O)CC1 94283,c1(NC(=O)NC2CCN(C(=O)C=Cc3ccccc3)C2)ccc2cccnc2n1 94284,N1(C(=O)OC(C)(C)C)CCCC1CNC(C1CC(N2CCCC2)C1)=O 94285,c1(C(N(CC(C)NC(=O)CCc2ccc(F)c(F)c2)C)=O)ccc(Cl)c(F)c1 94286,c1(NC(N2CC3CN(S(=O)(=O)CCCl)C3C2)=O)cnc2[nH]ccc2c1 94287,N1(C(C(F)OC)=O)CC(NC(=O)CCc2nc3cccnc3[nH]2)CC12CCOCC2 94288,c1(OC)ccc(C(C)(C)C)cc1NC(=O)C(=O)N(C)CC1CC(=O)C12CCC2 94289,c1(OC)nn(C)cc1C(=O)NC(C)C(C)C(=O)NCCCCC1CCCC1 94290,C1(C(N(CCF)CC)=O)CC(NC(C2CC(F)(CF)C2)=O)CCO1 94291,n1(CCC)ncc(C(=O)NCC23CC(NC(c4ncn(C(C)C)n4)=O)(C2)C3)c1C 94292,C1(C(=O)NCC(C(=O)NCC2(C#N)CCC2)N(C)C)COCC1(C)C 94293,c1(C(=O)NCC(N(C(c2c(C)snc2)=O)C)C2CC2)cnn(C)c1Cl 94294,C(=O)(CC(C)C(C)C(C)C)NC(CC)(CC)CCNC(c1cn(C)ccc1=O)=O 94295,C=CCCC(O)CNC(C12CC1CN(C(=O)COC)C2)=O 94296,C(CCCCC(=O)NC1(CF)CCN(C(=O)CC(=O)OCCC(C)C)C1)SC 94297,c1(OC(CC)C#N)cc(NC(=O)C(N2CCC(CN(C)C)CC2)=O)ccc1OC 94298,Cc1ccc(S(=O)(=O)CC(=O)Nc2cn(C)c(=O)cc2Br)cc1C 94299,CC1CCN(c2ncc(C(=O)NCC(C3CC3)N(C(=O)C=CCO)C)s2)CC1 94300,Cc1cncc(C(N2CCC(CCNC(=O)C=CS(C)=O)C2)=O)n1 94301,N1(C(C2CN(C(CCOCC#C)=O)CC2C(C)C)=O)CCCC(C)(F)C1 94302,C(C(C)(C)CC(=O)NC1CCC1CNC(=O)CSC(F)F)OC 94303,CC(C)C#CC(=O)NC1CCC(NC(C2CCCOC2c2ccnn2C)=O)CC1 94304,C(=O)(C(C)(C)C(=O)N1CCC(C)C(N(C(=O)Cc2ccccc2Cl)C)C1)OCC 94305,N1(C(C)CNC(c2cnccn2)=O)CCN(C(=O)CN2CCC(C)(C)C2)CC1 94306,C1(CCC)(CNC(=O)CCCN(C)C)CCN(C(C2(CCOC)CCC2)=O)CC1 94307,C=CC(C)CC(=O)NCC#CC(=O)N(C(C)C(C)(C)O)C 94308,N1(C(C23C(CN(C(C4C(C)CCOC4)=O)C2)CCC3)=O)CC(C)(C)OC(C)(C)C1 94309,C(=O)(CCC1CCc2ccccc21)NC1C(NC(=O)Cc2coc(C(F)F)n2)C1 94310,c1(OC)cccc(C(=O)NC(C)CCN(C(=O)C(C)(C)C2CCCC2)C)n1 94311,CCCC(CC)C(=O)NCC1CCCN(C(c2cncc(CO)c2)=O)CC1 94312,C#Cc1ccc(C(=O)NCC2CCCN2C(=O)C(C)CN2CCOCC2)cc1F 94313,CC1CNC(=O)CC(NCc2ccc(Cl)c(Cl)c2)C1 94314,c1(C(N2CCCC(CCNC(CNC(C)=O)=O)C2)=O)cccc2c1CCN2 94315,C1(CC(=O)NC(CO)C(=O)NCC2(c3ccon3)CC2)CCCC(COC)C1 94316,Cc1cc(C(=O)NCC2CC3(C2)CN(C(c2cc(C)sn2)=O)C3)c(O)c(C)n1 94317,C1(NC(C2(C)C=CCC2)=O)C=CCN(C(=O)Cc2ccnc(Br)c2)C1 94318,Cc1ccc(CSCC(N2CC(NC(C3CCCC3(C)C)=O)C(C)C2)=O)cc1 94319,C1(OC)CCC2(C(N3CC(NC(=O)C(C)OC4CCCC4)C(C)C3)=O)CC12 94320,C12(NC(c3cncc(OC)c3)=O)CCCN(C(=O)Cc3ccsc3)CC1C2 94321,c1(C(=O)NC(CN(C(=O)CC2CC=CCC2)CC)C)ccc(Cl)c(N)c1 94322,N1(C(c2ccc(SC)cc2)=O)CC2CC1CCN2C(=O)C=Cc1nc(C)cs1 94323,C#Cc1cncc(C(=O)NC(C)C(c2c(F)cccc2F)O)c1 94324,C(c1ccc(F)cc1)=CC(N1CC2CN(C(C3CCCS3)=O)C2C1)=O 94325,N1(C(C2N(C(c3cc(OCC)n[nH]3)=O)CCC2)=O)CC2CCOC2C1 94326,C(=O)(C1=C(C#N)CCC1)N1CCC(C=C)(C(=O)NCC(C)N(C)C)C1 94327,C(=O)(C(C)(C)CC(F)(F)F)NC(CNC(c1n(C)cnc1)=O)C1CC1 94328,c1(NC(=O)NC2(CNC(=O)Cc3cnoc3)CC2)ncnc2ccsc12 94329,Cc1cc(F)cc(C(=O)NC2CCC(NC(=O)C(C)c3cc[nH]n3)CC2)c1C 94330,Cc1cc(F)c(NC(=O)NCCC2CCCN(C)C2)cc1Cl 94331,CC(C)(O)CCNC(=O)CC1(NC2CCN(Cc3ccccc3)C2)CCC1 94332,N1(C(c2nn(CC)c(C)c2)=O)CCCC(C)(C(=O)Nc2c(Cl)cnnc2Cl)C1 94333,N1(C(C=C(C)C(C)(C)C)=O)CC2CC1C2C(=O)N(C1CCCC(O)C1)C 94334,C1(C)(CNC(C=NOC)=O)CN(C(C2(OC)CCSC2)=O)C(C)(C)C1 94335,C1(CN(C(CC(=O)NCC)=O)C)CN(C(=O)C(C)(CC2CCC2)OC)CC12CC2 94336,N1(C(C2(OC)CS(=O)(=O)C2)=O)CC(NC(C2CCCC2C(C)C)=O)CCC1C 94337,C1(NC(Cc2cnc(C)s2)=O)CC2CCC(C1)N2C(C1(C#N)CC2CC2C1)=O 94338,C#Cc1ccc(NC(=O)CC2(c3ccc(OC)cc3)CCC2)cn1 94339,C(C(C)(C)C(=O)NC(c1ccccc1F)CNC(C1CCCO1)=O)N(C)C 94340,S(=O)(=O)(c1ccccc1-c1cnc(F)cc1)NC(c1nccc(C)n1)C 94341,C1(NC(c2c(C)cc(F)s2)=O)CC2CCC(C1C)N2C(c1ccc(CF)cc1)=O 94342,C1(NC(COCC(=C)C)=O)C=CC(CC(=O)NCCOC2(C)CCC2)C1 94343,C1(NC(CCC(C)=O)=O)CCN(C(c2ccc(C(F)(F)F)nn2)=O)C(C)C1 94344,c1(C(=O)NCC2(C)CCC(NC(c3cccc(C)n3)=O)C2)cc(F)c(F)cc1F 94345,C12(CNC(C(COC)(F)F)=O)CCCC1N(C(c1c[nH]c(=N)s1)=O)CC2 94346,C#CCC(CC(F)F)C(=O)NCc1ccc(CCNC(=O)CCCOCC)cc1 94347,c1(C(=O)NCC(CC(C)C)NC(=O)C(C#N)=CC2CC2)cccc([N+](=O)[O-])c1 94348,C1(OCCCCC)CCCC(OC(=O)Cn2nnnc2C)C1 94349,c1(C(=O)N)c[nH]c2ccccc12.c1(SC)nccc(NC(C)(C)CN(C)C=O)n1 94350,CC1CCCN(C(C23CCC(NC(=O)CC4CCOC4(C)C)(CC2)C3)=O)C1CO 94351,c1(C(C)NCC(CCCC)CC)nc2ccccc2c2ccccc12 94352,c1(C(=O)NC(C2CCOC2)CNC(c2cnc(OC)s2)=O)cccc2c1CCO2 94353,c1(C(=O)OCC)c(C)o[nH]c1=NC(=O)NC(c1nncn1CC)C(C)C 94354,c1(C(=O)NCC2C(C)CN(C(=O)Cc3ccccc3Cl)C2)ccnc2[nH]cnc12 94355,N1(C(CCCC)=O)CC(NC(=O)CNC(c2ccc(C)s2)=O)C(C)C1 94356,C1(C(N2CCC(C(=O)NCc3ccccc3)CC2)=O)(OC)CC(O)C12CCC2 94357,N1(C(c2cn(CCC3CC3)nn2)=O)CCCN(C(C2CC23CC(O)C3)=O)C(CO)C1 94358,C12CCN(CC1)CCN2C1CC1.c1(NC(C2(C(=O)NC)COC2)=O)ccc(Br)o1 94359,c1(C(=O)NCC2CCN(C(=O)CC3CCCO3)CC2)cccc2c1CCCC2=O 94360,c1(C(C)NC(C2(F)CN(C(C(C)SC)=O)C2)=O)cncc(F)c1 94361,C(=O)(C1=COCCC1)NC(CC(=O)NCC(CC(C)O)C)(C)C 94362,C1(C(C)C)CC(C(=O)NCCC2CCCCN2C(=O)C(C)CF)CCO1 94363,c1(N(CCC(O)C(C)(C)C)C)nc(=N)[nH]c(=NC2CC2c2cccc(F)c2)[nH]1 94364,CC1(C)CCOC1CC(N1C(CNC(C2OCCC2(C)C)=O)CC2CC12)=O 94365,C(=O)(C1=CC2CCCCC12)NC(c1ccccc1)CNC(C(=C(C)C1CC1)F)=O 94366,c1(C(N2C(CNC(C(C)(O)C3CC3)=O)CCCC2)=O)cnc(Cl)cc1Cl 94367,C1(NC(c2nc(C(C)OC)oc2)=O)CCC(NC(C2CC2F)=O)CC1 94368,c1(C(=O)NC2CC2NC(C2CC(=O)N(C3CCCC3)C2)=O)csc2c1CCCC2 94369,c1(N2CC(C(=O)NC)OCC2)nc2c(c(=NCCC3CC3)[nH]1)CCC2 94370,N1(C(C(C(CC)C)OC)=O)CCC(N=c2nc(C(F)(F)F)[nH]s2)C2(CCC2)C1 94371,CC#CCC(C(=O)NCC1=CCN(C)CC1)NC(=O)Cc1ccc(O)cn1 94372,N1(C(CNS(CC)(=O)=O)=O)CCCC(CCNC(C2CCCO2)=O)CC1 94373,c1(OC)ccc2cc(C(N3CCC4CN(S(=O)(=O)CC(C)C)CC34)=O)ccc2c1 94374,c1(OC)nc(C)ccc1C(N1CC(NC(=O)Cc2nnc(C)o2)C(C#N)C1)=O 94375,Cn1cnc2c[nH]c(=NC3CC(C4CC4)C3)nc12 94376,N1(C(C(=O)NC2CCCCC2)=O)CC2CN(C(=O)CC3CC4(CC4)C3)CC2C1 94377,C(=O)(CCCCCCCSC)NC(CNC(c1c(COC)ccs1)=O)C 94378,N1(C(C2C(=C)C2)=O)CCCC2(C1)C(NC(=O)C(C(F)(F)F)C(F)(F)F)CCN2C 94379,C1(CC)CCCN(C(=O)CC(C)(C)C2CC2)C1C(=O)NC1CN(C)C(C)(C)C1 94380,CC1CCCC=C1C(=O)NC1CC(C(C)NC(c2cc3cccnn3c2)=O)C1 94381,CC(C)(C(=O)NCC(C1CCCCC1)NC(=O)CCOC1CCCOC1)C(N)=O 94382,N1(C(C23C(CN(C(CC4CCCC(C)O4)=O)C2)C3)=O)CCN(C)C(=O)C1 94383,Cc1cc(SCC(=O)NCC(C)(CO)NC(C2CC(C)CCO2)=O)cc(C)c1 94384,c1(C(=O)OC)cc(OC)cc(OC(F)(F)F)c1CN1CC2CCOC2(CN)C1 94385,CCC(CC(=O)NC1CC1CNC(=O)CSCC#N)C(C)C 94386,c1(NCC(C)SC)cc(=NC(C)CCc2cnn(C)c2)[nH]c(C)n1 94387,C(=O)(C(C)CCCOC=O)N(C(CCNC(COCCCC)=O)C(C)C)C 94388,c1(C(=O)NC(CC)(C)CNC(c2ccc(C(F)F)o2)=O)c(C)cc(C#N)cc1C 94389,n1(CC)nc(C)c(C(=O)NCC(C)N(C)C(c2sccc2C#N)=O)c1C(F)F 94390,N1(C(c2ccc(C(=O)OC)nc2)=O)CCN(C(C2CC(C)(C)C2)=O)CC1CF 94391,c1(COC(C)C)ccc(CNC(=O)N(C)Cc2cscc2Br)cc1 94392,C1(C(=O)NCC2CN(C(Cn3nc(C)oc3=O)=O)C2)Cc2ccccc2C(=O)O1 94393,[N-]=[N+]=NC1CC(C(=O)NCC(CC2CC2)CO)N(C(=O)C2=CCCOCC2)C1 94394,N1(C(CC(CNC(CC=C=C)=O)(C)C)=O)CC(=O)N(C)CC1CC 94395,CC1CN(C(c2cccc3[nH]c(=N)oc23)=O)Cc2ccccc2O1 94396,c1(C(=O)NC(C(C)C)Cc2ccc(F)cc2)ccc(N2CCCC2=O)c(Cl)c1 94397,Cc1ccc(-n2nc(C(C)C)nc2C2CC(=O)N(c3c(C)noc3C)C2)c(C)c1 94398,CC1(C(=O)NCC2OCCC2C(=O)NCCOCC2CCC2)CC(C#N)C1 94399,Cc1cccc(Br)c1C(C(=O)N(CC(C)C(C)(C)C)C)NC(c1c[nH][nH]c1=N)=O 94400,C=CC(CC)CC(=O)NC12CC(C1)N(C(=O)C(C1CC1)OC)C2 94401,C=CCCCCCC(C)(c1nnnn1CC=C)NC(C)CCC(=O)OC 94402,C(C)(C)(CN=c1[nH]c2ccccc2s1)C1CCN(C(C(C)OC2COC2)=O)CC1 94403,C1(C(=O)NC(C)CNC(=O)CCc2cncc(F)c2)Cc2nn(C)cc2C(=O)N1 94404,C12(C(N3C4(CNC(c5c(C)scn5)=O)CC(C3)C4)=O)CC(C)(C1)OC21CCC1 94405,CCC1=NOC(C(=O)NC(CNC(c2cnn(CC)c2C2CC2)=O)CC)C1 94406,C1(C(=O)NC2CC(NC(c3c[nH]c(=NC)s3)=O)C2)CCc2c[nH]nc2C1 94407,Cc1cc(C(F)F)oc1C(N1CC(NC(C2CCC(F)(F)C2)=O)C(O)C1)=O 94408,CN1CCOC(C(=O)N(C)CC2COCCN2C(c2csc(Cl)c2)=O)C1=O 94409,C1(CC(=O)N(CCCNC(C2CCC2C)=O)CCC)COCCN1CC 94410,Cc1csc(C(N2CCCC(C(C)NC(C34CC(CCO3)C4)=O)C2)=O)c1C 94411,C1(C(N2C(C(=O)NC(CC)CCCO)C=CC2)=O)CCOC(=O)CC1 94412,c1(OC)ccc(C(C)(C)C(=O)N(O)Cc2cn(C(C)C(C)O)nn2)cc1OC 94413,C1(NC(C2CC(C)(C)OCC2)=O)CC2(CCCN(C(c3cnc(O)o3)=O)C2)C1 94414,C1(CCC)CN(C(=O)CC(C)CC)CCN1C(=O)CN1CCC(C)CC1 94415,C1(CCC)(NC(=O)CCC2CC2C)CCN(C(C2CC3CCC3C2)=O)CC1 94416,c1(C(N(C(C)CNC(C2CC2(C)C)=O)CC)=O)cc(OC)c(O)c(OC)c1 94417,N1(C(C2(CCCC)CCC2)=O)CC2C(C(=O)NCCn3nncc3C)C2C1 94418,CCCC(CC)C(=O)NC1(CO)CCCN(C(c2cc(C(CC)CC)no2)=O)C1 94419,N1(C(C2CCC(C)CC2)=O)CCCC2(NC(C3CCC(C(C)C)CC3)=O)CC2C1 94420,C(=O)(CCC(F)(F)F)N(CC(C)NC(=O)C(C)CC1CC1)CC 94421,C1(C(=O)NC(C(N2CC(C#C)C2)=O)Cc2cn[nH]c2)CC12CCCC2 94422,C1(NC(C2(OCC)CCC2)=O)C2CCC(C2)C1C(=O)N(CC(O)CC)CC 94423,c1(CN)ccccc1-c1cn(CCC(=O)NC2CC3CC3C2)nn1 94424,C1(C(=O)NC(CNC(CC2(CC(=O)OC)CCCC2)=O)C)CCn2nnnc2C1 94425,n1(-c2cccc(C(=O)O)c2)cccc(NC(=O)C2=CC(N)C2)c1=O 94426,c1(C(N2CC3CC2CCC3NC(=O)C(F)(F)CC2CC2)=O)cccn2ccnc12 94427,N1(C(C(C)(C)NC(=O)OC)=O)CCC(C2CC2)(CNC(=O)C=CC(N)=O)C1 94428,C1(CCNC(c2[nH]cc(C(C)=O)c2)=O)CN(C(c2sccc2CC#N)=O)CC1C 94429,O=C(C1CCCOc2ccccc21)NC1COCC1n1cc(-c2ccsc2)nn1 94430,c1(CNC(c2c(C)cnnc2)=O)ccc2c(c1)CCC2NC(=O)CSC(F)(F)F 94431,c1(C(=O)NC(C2(CNC(C3CC(SC)C3)=O)CC2)C)cc2ccncc2c(O)n1 94432,N1(C(c2c(CC)ocn2)=O)CC2CC2(C(=O)NC2(C)CCCC2)C1 94433,C1(CN(C)C)CCN(C(c2cncnc2)=O)CC1.C12(CC1COC)N(CC)C2=O 94434,N1(C(c2nn(C)c(F)c2)=O)CCCCCC1CNC(C1C2CCCCC12)=O 94435,c1(OC)nc(NC(C2C3CN(C(=O)CCSC)CC23)=O)ncc1Br 94436,C1(C(=O)NC(C(C)OC)C)CCC(O)(Cc2ccccc2)CC1 94437,c1(C(=O)NC2(c3ccccc3)CN(C(c3cnn(C4CC4)c3)=O)C2)n[nH]c(O)n1 94438,c1(C(=O)NC2CC3(C(NC(CC4ON=C(C)C4)=O)C3)C2)ccnc2[nH]c(O)nc12 94439,n1(C(C)C)[nH]cnc1=NC(=O)c1ccccc1.c12ccc(cc1)CN(C)C2 94440,C1(C(=O)NCCCCCNC(CC(C)OC)=O)CC(=O)N(c2cnn(C)c2)C1 94441,CCCCC(CC)C(=O)NC(C)CCNC(c1sccc1SC)=O 94442,Cc1cc(C(N2CCNC(C(=O)NC3CC(O)C3)C2)=O)cc(C#N)c1 94443,c1(C(N(C2CCCCC2)CCNC(C(CSC)O)=O)=O)sc2cncn2c1C 94444,c1(C(C(=O)NCC2CCCO2)N(CCC(C)(C)C)C)ccc(F)c2[nH]ncc12 94445,N1(C(C(CCF)NC(c2cc(C)ns2)=O)=O)CCCC(C)(O)C1 94446,C1(CC(=O)NC(CC)CO)CCCC12CN(C(c1ccc(F)c(F)c1)=O)C2 94447,c1(NC(C)=O)cccc(F)c1-c1cnc(F)c(C(N2CC3C(C2)C3(C)C)=O)c1 94448,c1(C(=O)NC(c2cccc(N)n2)C)cnc2n1CCOCC2 94449,C(=O)(C(C)(C)CC(F)(F)F)N(CC(CNC(c1c(OC)n(C)nc1)=O)C)C 94450,CCC(C)(O)C(=O)NC1C=CCN(C(c2cn(C)nc2C)=O)C1 94451,c1(CN(C(CCN(C(CCCN(C)C)=O)CCO)=O)C)ccc(O)cc1 94452,CCC(CC)C(F)C(=O)NC(CC1CCCC1)C(=O)N(C1CCC(F)(F)C1)C 94453,C1(C(=O)NC(CN(C(=O)CCCCSC)CC)C)COCCN1C 94454,C12(C(=O)NCC3(CNC(Cc4c(C)ncs4)=O)CCCC3)CC(C)(CO1)C2 94455,C(CN=c1[nH]c2c(c(=NCC(C)(C)SC)[nH]1)CSC2)c1ccc(OC)c(Cl)c1 94456,Cc1cc2ncc(C(=O)NCC(C)NC(=O)CN3CCCC3C)cc2[nH]1 94457,N1(C(CCC=C)=O)CCC(CO)(NC(c2csc(-c3nc[nH]n3)n2)=O)C1 94458,c1(CNC2(c3n(C)nnn3)CSCSC2)cc(Br)c(C#N)cc1F 94459,C1(CNC(=O)C(O)CN2CCCC2)CCN(C(c2cc(CF)on2)=O)CC1 94460,N1(C(C(C)N(C(C)=O)C)=O)CCC(CO)(CNC(=O)CCCc2cccnc2)C1 94461,c1(CNc2ccc(OC)cc2F)cnc2c(c1)c(C)nn2C 94462,C(=O)(C(C1CN(C(C2(C(C)C)CC2)=O)C1)OCC1CC1)N(CC(=O)SC)CCC 94463,C1(CNC(C(C(CC)C)C)=O)CC2COCC2N1c1nnc(-c2ccccc2)o1 94464,c1(CN(CCCN(C(=O)OCC)C)C)cccn1Cc1ccccc1 94465,c1(N(C)C)cccc(C(=O)NCC23CC2CN(C(=O)CCC2CCCC2)C3)c1 94466,C1(NC(C(C)NC(C)=O)=O)COC2(C1)CN(C(c1cnc(C(C)(C)C)o1)=O)C2 94467,N1(C(C2CN(C)C2)=O)CCCC1C(=O)N(C)Cc1nnc(O)o1 94468,c1(C(=O)NCC2(O)CN(C(C(C)Sc3nncn3C)=O)C2)nn(C)cc1N 94469,c1(OC)ncc(C(=O)NCCOC2CN(C(=O)C(c3cccnc3)=O)C2)s1 94470,c1(CNC(=O)CC2CC(N)C2)ccc(F)cc1[N+](=O)[O-].Cc1c(OCCO)cncc1Br 94471,c1(NC(C)CC(C)NC(C2CCC3CC3CC2)=O)c([N+](=O)[O-])cnn1C 94472,c1(C2(NC(CSc3cnc(CCCC)[nH]3)=O)CC2)ccc(F)c(F)c1 94473,n1(CC)nncc1C(=O)N(CCN(C)C(C1(N(C)C)CCC1)=O)C(C)C 94474,C1(CCNC(C(COC)C)=O)CN(C(=O)C(F)=C(C)C)CCCO1 94475,c1(OC)cccn2ncc(C(=O)N(C3CN(C(=O)CN4CCC4C)CC3O)C)c12 94476,c1(OC)cc(CC(=O)NCCC2(CNC(=O)CC(C)(F)F)CC2)cc(F)c1.C1CC1 94477,c1(C(N2CCC3CN(C(C4CCN(C)C4=O)=O)C3C2)=O)ccc2c(c1)OCCC2 94478,c1(C(C(=O)NCCCNC(C(CCSC)OC)=O)=O)cc(F)ccc1F 94479,C12(CNC(c3cn(CCC)nc3)=O)CC1CN(C(=O)CC1CCC1(F)F)C2 94480,C1(C(N2CCN(C(CNC(=O)CC(F)(F)F)=O)CC2)=O)CCc2nc(O)[nH]c2C1 94481,Cc1c(C(=O)NCC2(CC(N3CCCC3C(N)=O)=O)CC2)[nH]ccc1=O 94482,Cc1noc(C)c1C(=O)Nc1ccsc1C(=O)NC1CC1(F)F 94483,c1(N2C(CNC(Cc3c(C)ccs3)=O)CCCC2)ncc(Br)c(C)n1 94484,CC1(C(N2CC(CO)C(c3ccccc3)C2)=O)Oc2ccccc2NC1=O 94485,N1(c2nnn(C)n2)CC2C3CCC(C2C1)N(C(c1cc[n+]([O-])cc1)=O)C3 94486,c1(NC(C2COCCN2C(C2CC2C2CC2)=O)=O)cc(F)ccc1Br 94487,N(C(=NCCc1cnccn1)NCCN1CCOCC1)CC1(C)CCCCO1 94488,C1(O)(C(=O)NC(C)CCNC(=O)CC2(C)CCOC2)CC2CCC1C2 94489,C1(CCNC(C(C2CCCN(C(C3C4CN(C)CC34)=O)C2)C)=O)CCCC2CC12 94490,C1(C(=O)NC2C(NC(Cc3c(C)cco3)=O)CCCC2)CN2CCN1C(C)C2 94491,C1(CCC)CN(C(c2nc(C)oc2OCC)=O)CCN1C(c1cc(=O)cc[nH]1)=O 94492,c1(C(=O)NC(C)(CNC(c2cn[nH]c2)=O)Cn2cccn2)cccc2scnc12 94493,c1(C(=O)NC2(C3CN(C(=O)CCCF)C3)CC2)cc2cc(Br)ccc2s1 94494,c1(C(COC)NC(=O)CCc2cccs2)ccc(F)c(F)c1 94495,c1(C(=O)NCC(=C)CCNC(=O)Cc2occc2C)ccccc1SCC 94496,C1(C(=O)NCC(CCC)NC(c2c[nH]nc2C2CCOC2)=O)(CC)CC(C)(C)C1 94497,N(C1CN(c2nc3ccccc3s2)CCc2ccccc21)C(CC(C)C(F)F)=O 94498,C(=O)(C(C)(C)C(=O)N1CC2C(OC)C2C1)NCCOc1c(OC)cccc1 94499,c1(C(C(=O)NCC(C2CCC2)NC(CSC(C)C)=O)(F)F)ncc(Cl)n1C 94500,c1(COC)ccc(C(=O)NC2CN(C(=O)CCCN(C)C(=O)OC)CC2O)cn1 94501,c1(C(=O)NC(CC)(CNC(=O)C(F)(F)COC)CC)ccc2cccnc2n1 94502,c12nc(ncc1Br)C2=O.N1(Nc2ccc(N3CCN(C(C)=O)CC3)cc2)CCCC2CC12C 94503,C(C)(C)(CCNC(=O)Cc1cc(C(C)C)no1)NC(COCC(=O)NC)=O 94504,CCCC1=C(C(=O)OC)C(c2cc(CN)nn2C)NC(=O)N1CCOC 94505,C1(NC(CNC(CCC)=O)=O)CN(C(c2cc(-c3cccs3)on2)=O)C2CC12 94506,c1(C(=O)NC2CC(CNC(CCCOC)=O)OCC2)cc2cccc(F)c2s1 94507,C(C(C(=O)NOCCCC)NC(c1ccc(C)nn1)=O)SCC 94508,c1(C(N2C(C(=O)OCC3(C)CC(C)(C)C3)CCC2)=O)c(Cl)cncc1Cl 94509,N1(C(CC(C(=O)OCC)(C)C)=O)CC2(C1)CN(C(=O)C(C)(C)C(C)C)CC2CO 94510,Cc1cc(C(N2CC3CCC2C(NC(=O)C(F)C2CCOC2)C3)=O)c(Cl)cc1F 94511,c1(C(C)C)ccc(C2(C(N3CCC(N(C)C(=O)C4CC4)C3)=O)CCCC2)cc1 94512,Cc1cc(F)ccc1COCCOCCN.C1CO1.C(CNC(=O)O)OC(=O)N 94513,c1(C(N2CCC(c3ccco3)C2)C(=O)NCCCSC)cccc(CO)n1 94514,Cc1ccc(C(=O)NCC=CCC(N2CC(CO)CC2C)=O)cn1 94515,c1(CC)cc(NCC2(CC3CCCCC3)CCOC2)cc(Cl)c1C#N 94516,c1(C(N2CCCC(C3N(C(CC=C)=O)CCC3)C2)=O)ccc(CC)cc1Cl 94517,CCCCC(O)CC(=O)NC(CCC1CCC1)C(N1CCC2(CCCO2)C1)=O 94518,c1(C(=O)OC)ccc(NC(C2CC(O)CN2Cc2ccsc2Br)=O)cc1Cl 94519,c1(C(=O)NC23CCN(C(c4c(C)cc(C)o4)=O)CC2C3)ccc2occ(C)c2c1 94520,N1(C(c2c(OCC)cccc2)=O)CCCC2C1CCN2c1ncc(Br)c(OC)n1 94521,C(=O)(C1=CCSC1)N(C(C)(C)CC(=O)NC1(C)CCOCC1)C 94522,C1(C(=O)NCCCn2cc(CC3CCNC3=O)nn2)C2Cc3cc(Cl)ccc3C12 94523,c1(C(N(C)CC2CCCN(C(c3c(C)cn(C)n3)=O)C2)=O)cc2cccnc2s1 94524,N1(C(c2cncc(OC)c2)=O)CCCC(C)(C(N2C(C)CCC2(C)C)=O)C1 94525,C1(NC(C2C(OC)CC2)=O)CCCC(NC(c2nc(OC)c(C)s2)=O)C1 94526,C=CC(C)(O)C(=O)N1CC(NC(=O)CCOCC)C(C(F)(F)F)C1 94527,CN1CCN(C(=O)C(C)(C)n2cnnn2)CC1CNC(=O)C(F)(F)C1(O)CCC1 94528,C=C(C)CC(C(=O)NC(c1cccc(F)c1)C)NC(=O)C(=O)NCC(F)F 94529,c1(C(=O)NC2C(CNC(c3ccn(CCOCC)n3)=O)C2)ccc(F)c(Cl)c1 94530,c1(CCOC)nc(=NC2(C(C)(C)NC(C3CCNC3=O)=O)COC2)s[nH]1 94531,C1(OC)(CNC(C2CC2C)=O)CCN(C(c2sccc2CC#N)=O)C1 94532,c1(C(N(C(CNC(C2CCN(C(CC)=O)C2)=O)C)C)=O)cc([N+](=O)[O-])cc(C)n1 94533,C1(NC(c2ccc(OC)nc2)=O)CN(C(C2CC(=C3CCC3)C2)=O)CC1C(F)F 94534,c1(N2CC(CN(C)C(c3c[nH]cc3Br)=O)C2)nc(Cl)nc2c1ncn2C 94535,c1(NCCC(CCC)C)ccc(S(=O)(=O)NC(COC)C(C)(C)C)cn1 94536,c1(CNC(c2c(C)n(-c3ccc(F)cc3)nn2)=O)cn2cc(F)ccc2n1 94537,CC1SCCN(C(=O)C(C)(C)C2CCN(C(=O)C#CC3CC3)C2)C1C 94538,CC1=C(C(=O)NCC(C)(F)CNC(C2(C(C)C)CNC(=O)C2)=O)C(C)(C)CCC1 94539,c1(C(N2CCN(C(C(CC)CC)=O)C(C(C)(C)C)C2)=O)ccc2c(c1)COCO2 94540,C(=O)(CCC(=O)NCCC)N(C1CCN(C(CSC2CC2)=O)C1)CCC 94541,Cc1cc(N)c(C)nc1C(=O)NC1CCN(C(=O)Cc2ccc(F)cn2)C1 94542,CN1CCN(C(=O)CC2CCCCO2)C(CNC(C2C(C)(C)C2(C)C)=O)C1 94543,c1(C(=O)NCC=C2CCN(C(c3cnc(C)n3C)=O)CC2)cnn2c1N(C)CC2 94544,n1(CC(=O)N(C2CCCN(C(C(COC)(C)OC)=O)C2)C)nnc2ccccc12 94545,N1(C(c2ccc(C)c(F)n2)=O)CC2(CCCC2NC(C23CC2COC3(C)C)=O)C1 94546,c1(C(=O)NC(C(=O)OC)Cc2cn(-c3cnn(C)c3)nn2)cccc2nccn12 94547,C1(CNC(=O)CC2C=CCCC2)CN(CC=Cc2cccc(CO)c2)CCCO1 94548,C(CCCCCN(C)C(C1CC1CN(C)C)=O)NC(CSCC)=O 94549,c1(C(=O)NCc2c(C)c(Cl)ncc2)n[nH]c2c1CN(C(C1CC1C)=O)CC2 94550,c1(C(N(CCN(C(CCCN(C(C)C)C)=O)C)C)=O)cc(O)c2ccsc2c1 94551,c1(N(CCCC)C)ncnc2c1ncn2CC(C)(Cc1ccccc1)CO 94552,C1(CNC(C2CCCO2)=O)CC2CC2N1C(=O)CC1CC(n2cnnc2)C1 94553,C(=O)(CC(C)CC(C)C)N1C(C(=O)NCC2(CC)CC2)CSCC1 94554,N1(C(C(OC)OC)=O)CCN(C(=O)CCCSC)CC(CO)C1 94555,C(=O)(C(CNC(C1CC1C#N)=O)C(C)(C)C)NCC(C(=O)OC)C 94556,C=C1CC(C(N2CC(C(N)=O)C2)=O)(CNC(C2CCOC2)=O)C1 94557,O=C1CCOC(C(=O)NCC2CC(F)(CNC(=O)C(F)n3ccnc3)C2)C1 94558,N1(C(C(=O)NC(C(=O)OC)C)C(C)C2CCCC2)CCC2(CCCCO2)C1 94559,CCC(CCC(=O)N(C)CC1(CO)CC1)NC(c1cn(CC)nc1C)=O 94560,C1(NC(c2csc3nc[nH]c(=O)c23)=O)CC(CO)C12CCOCC2 94561,c1(C(N(CC(C)(C)NC(C2CCC=CCC2)=O)C)=O)ccc2scnc2c1 94562,N1(CC(=O)NCC2(O)CC(NC(c3ccc(CC)o3)=O)C2)CCCCCC1=O 94563,Cc1nc(N(C2(CN)COC2)Cc2ccnc(C)n2)cc(O)n1 94564,N1(C(Cn2c(CCC)nnc2S)=O)CCCC(C)C1.N(C)C 94565,Cc1nccc(C(=O)NC(CCC2CC2)C(=O)NCC2(CO)CCCO2)c1C 94566,c1(OCC(=O)NC2(CC=C)CCOC2)cc(C)cc(C)c1 94567,CC1CCN(C(=O)CCC2CCCOC2)CC1CC(=O)NC(C)(C)CF 94568,N1(C(CC=CC=C)=O)CCC(OCC(=O)N(CC(C)OC)C(C)C)C1 94569,c1(OC)n[nH]c(NC(C2CC23CCN(Cc2cnc(O)c(Cl)c2)C3)=O)c1C#N 94570,CN1CCN(CC2CC2)C(C(=O)NOC2CCCC2)C1.C1(=O)CN1 94571,c1(C(N2CC(NC(C(C)C3CCOC3)=O)(CO)C2)=O)coc2c1CS(=O)(=O)C2 94572,N1(c2ncc(C(=O)OCC)s2)CCOC(C)(CNC(=O)CCN2CCC(F)C2)C1 94573,N1(C2CN(C(=O)CC3CC3(Cl)Cl)C2)CCN(C(c2ccc(CF)cc2)=O)CC1 94574,C(=O)(C1CCCn2cnnc21)NC1C(C)CN(C(c2c(Cl)cncc2Cl)=O)C1 94575,c1(OCC=C)ccc([N+](=O)[O-])c(C(=O)OCC(C(=O)O)C2CCOCC2)c1 94576,c1(C(c2n(CCOC)nnn2)NCC2(Br)CC2)nc(Br)cn1C 94577,c1(C(=O)NCC2C(CNC(C3CC(CC)OCC3)=O)C2)nc(N(C)C)nc(=N)[nH]1 94578,c1(C(=O)NC(COCC)C(=O)N2CCC(O)C2)ccc([N+](=O)[O-])[nH]1 94579,N1(C(C(C)(C2CC2)OC)=O)CCC2(CC1)CC(NC(=O)C=CC1CC1)CCO2 94580,C1(F)(C(N2CCCC(CC(C)C)C2)=O)CCN(C(C2CCCC(=O)C2)=O)CC1 94581,C(=O)(CCCCCF)NC(CC)CNC(=O)C=Cc1nnc(C(C)C)o1 94582,c1(C(=O)NCC(C)(C2CC2)NC(CC(CC)C)=O)cccc(-c2ccccc2)c1O 94583,C1(NC(C2=CC(C)C2)=O)CCC12CCN(C(=O)Cc1cnnn1C)CC2 94584,N1(C(C2(C)CCC(C)C2)=O)CC(C2CN(C(c3nn[nH]c3C(F)(F)F)=O)C2)C1 94585,C1(C(=O)O)(NC(Cn2cc(C(=O)OC)nn2)=O)CC2CCC12 94586,c1(OCC)cccc(CC(=O)NC(C)CNC(=O)CC2COC3CC2C3)n1 94587,C(CCC(C)(C)NC(=O)C(c1ccc(C)s1)C)NC(C(C)NC(COC)=O)=O 94588,C(=O)(C1=C(Cl)CCC1)NCC(C)(C(=O)O)OC 94589,N1(C(C(c2ccc(Cl)s2)C)=O)CC2(NC(=O)C(C)n3cccc3)CC1C2 94590,c1(C(=O)NCC(CC)(CC)NC(=O)CCCC#N)sc2nccc(C)c2c1C 94591,C1(C(N2CC=CC(NC(C3N(C)C(=O)CC3)=O)C2)=O)CC2(C1)OCCO2 94592,N1(C(C(C)N=[N+]=[N-])=O)CC2(CO)CC1(C(N1CCCC3(C1)N=N3)=O)C2 94593,CCC(CN=c1ccnc(N2CCC(c3cnccn3)CC2)[nH]1)N1CCCC1 94594,c1(OC)cc([N+](=O)[O-])ccc1C(=O)NC1CC1CNC(c1sccc1CC#N)=O 94595,C1(CC(=O)Nc2cn[nH]c2)CCN(Cc2cnn(-c3ccccc3)c2)C1 94596,C(=O)(C(C)C(F)(F)F)N1CC(NC(C(c2c(OC)cccc2)O)=O)C(SC)C1 94597,CC1CC(NC(c2cccc(-c3cc[nH]n3)c2)=O)CN(C(=O)C#CC2CCC2)C1 94598,CC1(C#N)CN(C(=O)C(N2CCCCC2c2nc3ccccc3o2)=O)CCO1 94599,C(=O)(C#CC1CCCCO1)N1C(CCNC(C(CCCC)O)=O)CCCC1 94600,C1(C(=O)OC(C)(C)C)CC(=O)CC12CCC2.C1(CC2C(=O)N2)CCS(=O)(=O)C1 94601,C(=O)(C(C)(CC)CC)N1CCC(N(C(C=CC)=O)CCC)CC1 94602,c1(OC)ccnc(CNC(C2(CNC(=O)CC3(C#N)CC3)CCCCC2)=O)c1 94603,C1(C(N2CC(F)(CNC(c3nc[nH]c4ncnc3-4)=O)C2)=O)CN=C2N=CNN2C1 94604,N1(C(c2c[nH]c(=NC)o2)=O)CCCCC(CNC(C2CC3C=CC2C3)=O)C1 94605,CC(CF)CC(=O)N1CCCC(NC(c2conc2C2(C)COC2)=O)C1 94606,N1(NC(C2(CCO)CCCC2)=O)CC(F)(F)C(F)(F)C1.C12CC(C1)C(=O)NC2 94607,CC1(C)CC2(CC(C(=O)NCC3CCCN3C(=O)Cc3cccc(F)c3F)C2)C1 94608,c1(OCC)nc(C)ccc1C(N1CC(NC(c2cnc(CC)s2)=O)C(O)C1)=O 94609,N1(C(c2ncnn2-c2ccccc2)=O)CCC2C(C1)C2(F)F 94610,c1(C(=O)Nc2c(C)nc(C(C)C)s2)cnn2ccc(CN)cc12 94611,CS(=O)(=O)CCCC(=O)NCC1(F)CCC(NC(C2CN(S(C)(=O)=O)C2)=O)C1 94612,C1(C(=O)NCC2C(C)(C)CN(C(=O)COCC(F)F)C2)COc2ccccc2O1 94613,C1(NC(C(C)OCOC)=O)CCN(C(c2csc(CO)n2)=O)CC1 94614,c1(C2(C(N(C3CN(C(C(=O)NC(C)C)=O)C3)C)=O)CCC2)ccccc1.C1CC1 94615,c1(C(=O)NCC(C2CCCCN2C(C2CC2(F)F)=O)(C)C)cccc(N)c1 94616,C1(C(=O)NCc2ccc(C)cn2)CN(C(=O)C2=COCCC2)CC1(F)F 94617,C(=O)(C1=C(C)CCC1)N1C(C(N2CC3CCC3C2)=O)(CC)CCC1 94618,C1(CNC(C(N2CCSCC2)C)=O)CCC(CNC(=O)Cc2cn[nH]c2)CC1 94619,C1(NC(c2cc(C(F)F)no2)=O)CC2CN(C(=O)Cn3nccn3)CCN2C1=O 94620,CCCCCCC(F)C(=O)NCC(CC)NC(c1nc(C)sc1C)=O 94621,CC(CC(C)(C)C)C(=O)N(CCCN(C)C(c1cc(C(F)F)no1)=O)C 94622,N1(c2snc(COC)n2)CCC2(CCOC2)C(CNC(C2CC3CC3CO2)=O)C1 94623,N1(C(CCNC(=O)NC)=O)CC2(COC(CNC(c3cc(Br)no3)=O)C2)C1 94624,C(=O)(C(CP(C)(C)=O)C(F)(F)F)Nc1c(CC)noc1 94625,O=C1NCc2ccc(-c3ccc(N4CCN(c5cccc(Cl)c5)CC4)cc3)cc21 94626,N1(C(C(C)OCC(F)(F)F)=O)C2CCC1C(CNC(c1ccccc1)=O)C2 94627,c1(C(=O)NCCC2(OC)CN(C(c3scc(OC)c3)=O)C2)cc(C)cc(O)n1 94628,C1(C)(C(=O)NCCCCC)CCCN(C(c2cccc(OC)c2O)=O)C1 94629,C1(CNC(=O)Cc2cnoc2)CCCC1C(=O)NC1C2CCCC12 94630,c1(OCC(=O)OC)cccc(CC(C)NC(c2ccccc2-n2cccc2)=O)c1 94631,c1(C(=O)NCC2C(NC(CC(=O)NCC#C)=O)CCC2)nnn2c1COCC2 94632,N1(C(C(C)OCC)=O)CCC2(CC1)COC(C(=O)NCc1cncc(C)c1)C2 94633,C1(C2CC2)(CNC(C2(C(C)C)CCCC2)=O)CCN(C(C2CCS(=O)(=O)C2)=O)C1 94634,C1(CC)CCN(C(C2CCS(=O)(=O)C2)=O)C1CNC(c1cscn1)=O 94635,O=C(CC1OCc2ccccc21)NC1CCCN(C(c2ccncn2)=O)CC1 94636,c1(OCC)ccc(O)cc1NC(=O)C(C)C(C)NC(C1(CO)CCCO1)=O 94637,c1(C(C)O)ccccc1C(=O)N(CCC(C(C)C)NC(=O)CC1CCCC1)C 94638,c1(NCCC2CCC(NC(C(C(C)(C)O)F)=O)C2)nnc2c(c1C#N)CCCC2 94639,c1(C(=O)NCC(CCCC)NC(c2cc(O)n(CC)n2)=O)cc[nH]c(=NCC)c1 94640,C1(NC(CCCOCC)=O)COC2C(NC(c3cnn(C(C)C)c3C)=O)COC12 94641,c1(C(=O)NC2CCN(C(C(n3ncc(C)c3)C)=O)C2)ccccc1CO 94642,N1(C(CN2CC(=O)NCC2)=O)CCC2(CCCC2NC(c2ccccc2)=O)CC1 94643,Cc1nc(O)c(Br)cc1C(=O)NC1(CO)CN(C(=O)C(Cl)=CCl)C1 94644,c1(OCC(=O)NC(CCNC(c2nc(CCC)oc2)=O)(C)C)cc(Cl)cc(Cl)c1 94645,c1(OCC#C)ccccc1OCCC(=O)NC12CCCC(C1)O2 94646,C(CCCC)(CC(=O)NC(CO)C(C)(C)CO)NC(CCCC#C)=O 94647,C1(N(CC(=O)NCc2cocn2)C(=O)C2CC2)CCCC12CCNCC2 94648,c1(C(N2CCC(C3CC3NC(C3(CF)CC3)=O)CC2)=O)ccc([N+](=O)[O-])cc1Cl 94649,C(C(=O)N1CCC(C(=O)NCc2cc(C)[nH]n2)O1)OCCOC 94650,C12(C(N(C3CCN(C(=O)Cc4cc(Cl)cs4)C3)C)=O)CC3CC(C1)CC(O)(C3)C2 94651,Cc1nc2c(C(N3CC(NC(c4cc(CO)[nH]n4)=O)CC3C)=O)ccnc2[nH]1 94652,c1(OC)cnc(F)cc1C(N1CC(NC(=O)Cc2cc(C)no2)C(C)(C)C1)=O 94653,N1(C(C(CCC#C)O)=O)CC2CCN(C(c3cccc(CC)c3)=O)CC2C1 94654,c1(C(N2CCC(COC)C2)=O)cnc(CNC(=O)C=CC2CCCN2C)nc1 94655,C1(C)(C(=O)NC2CN(Cc3ccc(C)cc3)C2)CCCCC1C 94656,CC(C)C(CNC(=O)C(c1cncnc1)C)C(=O)NCc1ccc(C#N)cc1 94657,c1(CC(=O)N(CC(CC)NC(C2COC3(C)CC2C3)=O)CC)c(C)cccc1C 94658,C1(NC(c2n(C(C)C)ncc2F)=O)CC(O)CN(C(C2CCN(C)CC2)=O)C1 94659,c1(C(N2CC(OC)C(NC(c3occc3C)=O)C2)=O)ccnc2cc(F)cnc12 94660,CN1CCCC2CN(Cc3cc(N4CCOCC4)nc(F)c3)CCC12 94661,c1(C(N2CC(n3cc(C(CC(C)C)O)nn3)C2)=O)ccc(Cl)c(F)c1 94662,N1(C(c2c(C)cns2)=O)CCC2CCC(NC(c3cc4ncccc4s3)=O)C1C2 94663,CC(C)C(F)C(=O)NCC1(F)CC(Nc2ncccc2C(=O)C(F)(F)F)C1 94664,c1(C(N(C2CCN(C(C34CC(C)(CCO3)C4)=O)CC2)CC)=O)cc(=O)cc(C)[nH]1 94665,c1(CN(C(=O)Cc2cc[nH]n2)C)cnn2c1CN(C(C1CCC(C)(C)C1)=O)CC2 94666,c1(C(N(C2CCN(C(c3ccc(COC)o3)=O)C2)CCC)=O)cc(C(C)C)no1 94667,N1(C(Cc2ccc(C)cc2C)=O)CC(O)(C2(CNC(=O)C=C3CCCC3)CC2)C1 94668,c1(SC)cc(C(=O)NCC(O)CNC(c2cnc(C)n2C(F)F)=O)cc(Cl)c1 94669,C1(C(N(C)CC2COCCN2C(C2CSCCS2)=O)=O)CC2CCC1C21CC1 94670,c1(C(=O)NC(C2CCN(C(=O)CC3CCC3)C2)C)cscc1S(C)(=O)=O 94671,Cc1onc(C(=O)NC(CNC(=O)CC2CC(F)C2)CC(C)C)c1[N+](=O)[O-] 94672,N(C(=NCCc1ccc(Br)cc1)NCCc1cnc(C)cn1)C(CC)C(F)F 94673,C(=O)(C(C(C)(C)C)NC(C)=O)N1CC(c2cn(CCC=C)nn2)C(O)C1 94674,N1(C(C=CC)=O)CCC(NC(c2ccc(N3CCCC3)nn2)=O)C(CC)C1 94675,C1(CNC(C2(CC#N)COC2)=O)CN(C(c2ccc(C3CC3)o2)=O)CCO1 94676,c1(C(=O)NCC2(C(C)NC(C3N(CC)CCOC3)=O)CC2)ccc([N+](=O)[O-])cc1 94677,CN1CC(CCNC(C2CCCC2CNC(=O)C=Cc2cocn2)=O)CC1=O 94678,c1(NC(CCN(C(=O)C(F)C2CCOC2)C)=O)cccc2ccccc12 94679,c1(C(NOCC(=O)N(C)Cc2cccnc2O)=O)cccc2[nH]ccc12 94680,C1(C(N(CC(=O)OCC)C2CC2)=O)CC(NC(=O)CC2CC(OC)C2)C1(C)C 94681,c1(C(N(CCC(C(C)C)NC(COC(C)C)=O)C)=O)cc2n(n1)CCCC2 94682,c1(C(=O)NC2C(CNC(C3(CC=C)CC3)=O)C2)c[nH]c2ccc(Cl)cc12 94683,CC1CC(O)CN1C(=O)NC(C1CC(F)(F)C1)C(F)F 94684,N1(C(CCC=C=C)=O)CC2(CO)CC1(C(=O)NCCc1ccccc1F)C2 94685,c1(CNC(C(Cc2cc(C)c(O)cc2)N)=O)cnn2c1CCCC2 94686,Cc1ccc2cccc(C(=O)N(C3CN(C(c4cnc(Cl)cn4)=O)C3)C)c2n1 94687,Cc1sc2ncc(C(=O)NC(C)(C)CNC(=O)CC34CCCC3C4)c(=O)n2c1C 94688,CS(=O)(=O)c1ccnc(NC2C3CN(C(c4cc(Cl)on4)=O)CC23)n1 94689,C(=O)(C1=CCOCC1)NCCC(C)(C)NC(c1cccn(C2CCC2)c1=O)=O 94690,N1(C(c2c(C)ncn2C)=O)CC=C(CNC(=O)COCCCF)CC1 94691,C(=O)(C(C(=O)N1CC2CC1C2NC(=O)C(F)C(C)(C)O)C(C)C)OCC 94692,C(=O)(C1=C(Cl)CC1)NC1CCN(CCCNC(C2(C)CC=CC2)=O)C1 94693,CC1CCCC1N(C)C(C1(CCNC(=O)Cc2ccsc2)CCC1)=O 94694,C1(NC(C(COC)(C)OC)=O)CCCCCN(C(c2ccccc2Cl)=O)C1 94695,C(CCC(C)C)(C(=O)Nc1ccc(N(C)C)cc1)NC(C(CCC)CC)=O 94696,N1(S(CC)(=O)=O)CCC2(CC1)CC(C)N(C(C1CC1(C(=O)OCC)C(C)C)=O)C2 94697,N1(C(c2nc(SC)sc2)=O)CCC2(CCC2)C(NC(=O)C(C)n2cccn2)C1 94698,C(C(C)C(=O)NN(C)C(C1C=CC1C(=O)OC)=O)OC.C12(CC1)CC2 94699,N1(C(C(CCCNC(c2n(C=C)ncc2)=O)(C)C)=O)CC(C)OCC(C)(C)C1 94700,N1(C(c2c(C)nns2)=O)C2CCC1C(c1cn(CC(c3ccccc3)O)nn1)C2 94701,Cc1cc(C(=O)NCC(C)(C)CNC(c2ccc(F)c(C)c2)=O)c(C)c(O)c1 94702,c1(SC)ccc(C(=O)NC(C)(C)CNC(=O)CO)cc1.C1(CN)CC1 94703,c1(C(=O)NCCN(C(=O)C(C(C)C)n2cc(Br)cn2)CC)cn(C)nc1Cl 94704,c1(-c2cn(CC(=O)NC3CCC4CC34)nn2)cc(OCC(F)F)ccn1 94705,N1(C(C2(F)CCN(C(c3scc(OC)c3)=O)CC2)=O)CCCC2(CCC2)C1 94706,C(=O)(C(C)CC(C)(F)F)N(C(c1c(OC)n(C)nc1C)=O)C(C)C 94707,C1(NC(CSC)=O)CCC2(CC1)CN(C(=O)C=Cc1ccncc1)CCO2 94708,c1(C(N2CCCCC2C2CCCC2)C(=O)NCCCF)nc(F)ccc1F 94709,C1(SC)CCN(C(=NCCc2ccc3c(c2)COCC3)NC2CCS(=O)(=O)C2)C1 94710,C=Cn1nccc1C(=O)NCC(CC(=O)NCCN(CCCF)C)C1CCC1 94711,c1(C(=O)NCCC(CNC(CC2N(CC)CCC2)=O)O)cc(O)n(CC)n1 94712,c1(C(=O)NC(CC=C)CNC(c2c(C)cccc2C)=O)n[nH]c2c1CC1CC21 94713,C(=O)(C(C)CN(C)C)NCCC(=O)NC1(C(=O)NCCC)CC1 94714,c1(N2CCC(C)(N(C)C)CC2)cc(=NC2CCSC2C)[nH]c(C(F)(F)F)n1 94715,CCC(C)(C#N)C(=O)NCC12CC(NC(=O)CCc3cnccn3)(CO1)C2 94716,c1(C(=O)NCCC(C)N(C)C(c2ncc(Cl)cc2Cl)=O)cnn2c1OCC2 94717,N1(C(C(CC)n2ccnc2)=O)CC2CCCC2(CNC(=O)CC#N)C1 94718,CC1CN2CCN1CC2C(=O)NC1CC(C)(NC(c2ccncc2N)=O)C1 94719,c1(-c2ccc(C3NC(=O)OC3)cc2)cccc2c1CCN(S(=O)(=O)CCCCCl)C2 94720,C1(C(=O)NCC(C)(C)NC(C(C)SC)=O)CCC(=O)N(C)C1 94721,CC1CCC(CNC(C2CC(CC(C)C)C2)=O)N(C(=O)Cn2ncnn2)C1 94722,CC1CN(C(C2C3CCC(C3)N2Cc2cc(Cl)cc(Cl)c2)=O)CC(=O)N1C 94723,C(=O)(CC(C(C)(C)C)NC(=O)CC1CC2CC2C1)NCC12N(C)CC(C1)C2 94724,c1(CCNC(C(C)NC(c2ccc(Cl)cc2)=O)=O)c[nH]c2cnc(Cl)cc12 94725,C(c1ccccc1)=CC(=O)NCCCOCCNC(C(OC)OC)=O 94726,C1(C(N(C2(CC(=O)N(CC(C3CCCC3)O)C3CC3)CC2)C)=O)CCC2(CC2)C1 94727,C(=O)(C(C)CC(=O)N1CCC(n2cc(-c3cc(CO)ccc3C)nn2)C1)OC 94728,C(=O)(C(C#N)C(C)(C)C)N(CCCN(C)C(C1CCCC1F)=O)C 94729,C1(C(=O)NCC2OCC(C(=O)NCc3cc(C)n(C)n3)C2)CCCC1C1CC1 94730,CC(C)(C#CC(=O)NCC1CCC12CCCCC2)CNC(=O)OC(C)(C)C 94731,C1(C2CC2)(CNC(CCCCCC)=O)CCN(C(=O)C(C)(C)C(O)CC)C1 94732,c1(C(C(=O)NCC(C)CNC(C2(C)CC=CC2)=O)=O)c[nH]c2ccccc12 94733,Cc1cccc(C(N2CCC(NC(C3CCC(C)(C)CO3)=O)C2)=O)c1C(F)(F)F 94734,CC1(NC(=O)C(O)CC(F)F)CCN(C(=O)Cn2ccc(C3CC3)n2)CC1 94735,O=C(CCc1ccccc1)C(=O)NCC1CCCN1C(=O)Cc1nccs1 94736,c1(OCC)nc(NCc2c(C(=O)NC(C)(C)C)cccc2)ncc1Br 94737,CCCC(C)(C)C(=O)NC(Cc1ccccc1)CCNC(c1ccc(Cl)nc1O)=O 94738,C(=O)(CCCC(C)C)N1C(C2CCN(C(CCn3ncc(C)c3)=O)C2)CCCC1 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94931,c1(C(C)N(C)CC2CCCC2C(F)(F)F)ccc(S(C)(=O)=O)cc1 94932,c1(C(N(CCCN(C(C(Br)=C(C)C)=O)C)C)=O)cocc1C 94933,C1(C(=O)NC2CC(C)(C(N3CCC(C(C)CO)CC3)=O)C2)CC2(CCC2)CO1 94934,N1(C(C(CC)OC)=O)CCCN(C(=O)Cc2cccc(NC(C)=O)c2)C(CO)C1 94935,C(CC(=O)N1CC(NC(C)=O)C1)(C(F)(F)F)NC(c1c(CC)ocn1)=O 94936,C1(NC(C2(CC=C)CCCC2)=O)CCN(C(=O)COCC(=C)C)CC1CO 94937,c1(C(N2CC(CNC(C3C(C)CCCC3)=O)C2)=O)cc(O)c(O)c(O)c1 94938,C1(CNC(CC)=O)CN(C(C2CCN(CC)C2)=O)CCCO1 94939,c1(C(=O)NC2C(NC(CN(C(=O)OCC)C)=O)CCC2)c[nH]nc1S(N)(=O)=O 94940,C1(CC(=O)NC2C(NC(CC)=O)CC2)CCCCC(=O)N1 94941,CC(C)(CCNC(=O)Cc1csc(C2CC2)n1)NC(=O)C(F)Cc1ccccc1 94942,N1(C(CN(C(=O)OC)C)=O)CCC2(C=C(C(=O)N(CCN=[N+]=[N-])C)C2)C1 94943,Cc1cc(O)c(Cl)cc1C(=O)N(C)CC1CCCN1C(c1cccc(F)c1F)=O 94944,CC1CC2CN(C(=O)CC(C)(C)N(C)C(C3COCC3(C)C)=O)CCN2C1 94945,N1(C(C2N(C(C(N3CCNC3=O)C)=O)C(C)CC2)=O)CCc2c[nH]nc2C1 94946,N1(C(C(=Cc2cnc[nH]2)C)=O)CCCC(NC(=O)Cn2cc(Br)c(C)n2)C1 94947,C1(N(C(C=C(CC)C)=O)CCNC(=O)CCc2ccccn2)CCCCCC1 94948,O=C(CCCn1ccnc1)NC1(CC2OCC(C(N3CCC4CC34)=O)C2)CCC1 94949,N1(C(C(F)OC)=O)CCC2(CC1)COCC(CNC(c1ncc[nH]c1=O)=O)O2 94950,N1(C(c2cc(OCC)no2)=O)CC2CC2(NC(=O)CC(c2cccc(F)c2)O)C1 94951,C1(C(N(CC(=O)OC)C)=O)COCCN(C(=O)CC=C(Cl)Cl)C1 94952,C1(NC(C=CCC)=O)CN(C(=O)C(c2c(F)cccc2F)OC)CCC1O 94953,Cc1ccc(N2CCC2CNC(=O)CN2CC(C)C2)cc1.C12CCC(O1)NC2=O 94954,N1(C(C2OCCC(C)(C)C2)=O)CC(NC(c2cn(CCO)nn2)=O)C2(CCC2)C1 94955,C1(OC)COc2cc(C(N3CC(c4ccsc4)OC(C)C3)=O)nn2C1 94956,CC1CN(C(=O)NC(c2c(F)cccc2Cl)CO)CC1(F)F 94957,n1(CC)ncc(NC(C2CC(NC(c3cccnc3O)=O)C2(C)C)=O)c1C 94958,C1(CN(C)C(c2csc(-c3ccccn3)n2)=O)CCCN(C(=O)CCF)C1 94959,C(C(=O)NCC1(C(=O)NC2CC(N(C)C)C2)CCC1)(C(C)C)OCC(C)C 94960,CN1CCCC(F)(C(=O)NC(C2CCCC2)CNC(c2cscc2Cl)=O)C1 94961,C(CCCCC(=O)NC(c1csc(C)n1)C)N(C(CNC(=O)OCC=C)=O)C 94962,C1(NC(CCNC(N)=O)=O)CCSC12CN(C(C1(NC(C)=O)CCOCC1)=O)C2 94963,C1(C(=O)NCC2C3CN(C(CCc4c(C)cccc4)=O)CC32)CC12CCOCC2 94964,N1(C(C2(CNC(c3nc(C)n(C)c3)=O)CC3(CC3)C2)=O)CCC2(CCOC2=O)C1 94965,S(=O)(=O)(c1ccc(NCC(C)O)c(F)c1)N(CC(C)N(C)C)C 94966,c1(C(=O)NC2CCCC(NC(c3n(C)cc(Cl)c3)=O)C2)cc(F)ccc1F 94967,N1(C(COc2ccc(CC)cc2)=O)CCCN(C(c2ccc(C(N)=O)[nH]2)=O)CC1 94968,c1(C(N2CC(C(C(=O)NC(C)CC3(O)CCC3)O)C2)=O)cnnn1C1CC1 94969,C(=O)(C(O)CC(C)(C)C)N1CCN(CCN(C(CC(C(=C)C)O)=O)C)CC1 94970,N1(C(=O)OC(C)(C)C)CC(O)CC1CNC(=O)NCc1conc1C(F)(F)F 94971,N1(C(CC(C)O)=O)CC(C(=O)NCCCCC(C)(C)C)CC1(C)C 94972,c1(C(=O)NC2CCN(C(c3n(CC)c(O)nc3)=O)CC2)cccc(C(F)F)c1F 94973,C1(C2CCN(C(c3cc(C)n(C)n3)=O)CC2)(NC(C(CC)CN(C)C)=O)CC1 94974,Cc1nc(O)ccc1C(=O)NCC1CN(C(=O)CC2CCC(=O)N2C)CC1(F)F 94975,c1(C(=O)NCc2c(C(=O)NC(C(=O)OC)C)nco2)ccncc1O 94976,c1(OC)cc2cc(c1)-c1csc(c1)C(=O)N2.C(C(C)OC(C)C)NC(C)=O 94977,C1(C(c2cc(Cl)ccn2)OC)CCCCC1C(=O)NCC1(CC#C)CCCO1 94978,c1(CN2CCC(C(C)NC(C3(NC(N)=O)CC3)=O)C2)cnc2ccccn2c1=O 94979,CC1CN(C(=O)CC2CC=CC2)C1C(=O)NC1(CCCCO)CC1 94980,C1(C(=O)OC)CCN(C(=O)N(CC(c2ncccn2)(C)C)CC2CC2)CC1 94981,N1(C(C(C)OC)=O)CCCC1C=CC(=O)NCc1oc(C)nc1C 94982,c1(C(C)C)ccc(C(=O)NCC2CCC(C)N(C(c3ncn(C)n3)=O)C2)c(F)c1 94983,c1(OCCC(=O)NCC(C(C)C)NC(=O)C2=COCC2)cccc(Br)c1 94984,C1(CC)C(NC(=O)CN2CCCNC2=O)CCCN1C(C1CCC(=O)NC1)=O 94985,C1(CC(=O)NCCOc2cccnc2)CCCN(C(=O)CSCCCCl)CC1 94986,C(C(C)C)(C(O)C(=O)NCCN(C(=O)COc1ccc(C(C)C)nc1)CC)OC 94987,n1(CC)c(=O)n(CC(N2CC(CC(C)NC(C3(F)CC3)=O)C2)=O)c2ccccc12 94988,C1(CC)(CO)CCCN1C(c1ccc(CNC(C2CCCC2C)=O)s1)=O 94989,CC1CN(C(C2(Cl)CCC2)=O)CC(C(=O)NCCN=S(C)(C)=O)O1 94990,C=CC1(C(=O)NOCC(=O)NCC(=O)NCC(C)C)CCC1 94991,c1(C(=O)NC(C2CCCN(C(C3CCCCCC3)=O)C2)C)cnn2c1OCCC2 94992,c12ccc(c(O)c1)Cc1nnc(s1)NC2=O.CC(C)(C)OC(=O)NCC(N)=O 94993,CS(=O)(=O)CCC(=O)NCC(CO)NC(=O)Cc1csc2nccn12 94994,C(C(C)(C)CC(=O)NCCCOC1CCN(C(=O)C(O)C(C)C)CC1)OC 94995,c1(OC)cccc(CNC(N2CC(CN(C3CCC(C)O3)C)C2)=O)c1 94996,c1(C(=O)NC(C)CC(=O)c2ccco2)cc(P(C)(C)=O)ccn1 94997,c1(-n2cc(C(C)NC(=O)Cn3cc(Cl)c(O)nc3=O)nn2)ccc2nc[nH]c2c1 94998,Cc1cc(F)c(C(=O)NCC2CCCN2C(c2cc3c(o2)CCCC3)=O)cc1F 94999,N1(C(C2CCN(C(C)=O)C2)=O)C2CCC1C(CO)N(C(c1ccc(C)s1)=O)C2 95000,Cc1[nH]c2ncccc2c1C(=O)NCC(CO)NC(C1CCCC(O)C1)=O 95001,C1(NC(C=C(C)Cl)=O)CC2CC(NC(c3nc(-c4cccs4)oc3C)=O)CC12 95002,CC1CN(C(c2nc(Cl)sc2Cl)C(=O)NC2COC2)CC1O 95003,C1(NC(CC2(COC)CC2)=O)CCCC(NC(=O)CC2CCCCO2)C1 95004,C1(C)(NC(C2OCCC(NC(Cn3ncn(C)c3=O)=O)C2)=O)CCCCCC1 95005,Cc1ccc(NC(C2CC(F)CN2Cc2cc3sccc3s2)=O)c(C#N)c1 95006,C12(C(=O)NCC(C)C)CC1CN(C(c1ccc(SC(F)(F)F)cc1)=O)C2 95007,c1(OCC)cccc(C(C(=O)N2CC(CNC(=O)CC3CNC(=O)C3)C2)OC)c1 95008,CN1CCC(C)(NN2CC3CC2CS3)C1 95009,c1(C(=O)NC2CCC(CNC(C3=C(C)CCC3)=O)C2)cccc2c1OCCCO2 95010,N1(C(C(C)n2cccc2)=O)CC2(CCC(CNC(C3CN(C)C3)=O)O2)C1 95011,C1(NC(C2(CCCC)CC2)=O)CN(C(c2csc(COC)c2)=O)C2(CCOC2)C1 95012,N1(C(c2ncc(C(C)(C)C)[nH]2)=O)CC2(C1)CN(C(C1CC3CCC1O3)=O)C2 95013,C1(c2cn(C3COCC3O)nn2)(NC(C(C)C(C)(F)F)=O)CC2(CCCC2)C1 95014,C1(F)(CNC(=O)CCC2CCCC2)CCN(C(c2cc(Cl)c[nH]2)=O)CC1 95015,c1(COC)nn[nH]c1C(N1CCC(C(N2CCCC2CC2CC2)=O)C1)=O 95016,C1(CC)(CNC(c2ccoc2Cl)=O)CCN(C(C2CCC(N(C)C)C2)=O)C1 95017,c1(C(=O)NCc2c(C(N(C(C)COC)CC)=O)[nH]cc2)cc2ccccn2c1 95018,Cc1ccc2c(C(=O)NCCC(C)NC(=O)CC3CN(C)CC3O)n[nH]c2c1 95019,C12CCCN(C1)C(=O)NCc1noc2n1.C(C(C)N(C)C(=O)OC(C)(C)C)SC 95020,S(=O)(=O)(c1cncc(Br)c1Cl)NCCCCCCC(=O)O 95021,C1(CCNC(CN(C(CSCC=C)=O)CC2CC2)=O)CCCCC1C 95022,C1(CNC(CNC(=O)OC)=O)CC(NC(=O)C(N2CCCCC2=O)C)CCO1 95023,N1(C(C)=O)CC2CC(O)C1C2NC(=O)CCCc1ccc(C)cc1 95024,c1(C(N(CCCNC(c2cc(C3CC3)ns2)=O)CC)=O)cccc(N(C)C)c1 95025,C1(C2CCC2)(C(=O)NC(C)CCCNC(=O)CNC(c2cccnc2)=O)CC1 95026,N1(C(CCC#N)=O)CC2(CCOCC2)CC1CNC(C1(C(N)=O)CCC1)=O 95027,N1(C(c2c(C)noc2)=O)CCC(N(C(=O)C=CC=C(Cl)Cl)C)C(C)C1 95028,CC(O)CC(C)(C)CNC(C1(CCNC(=O)CC2CCCCO2)CC1)=O 95029,Cn1cnc2c(C(=O)Nc3cccc(NC(C4CC(C(N)=O)C4)=O)c3)ccnc12 95030,Cc1ccc(SC(C)C(=O)N(C2CCCN(C(c3nc(O)c(C)s3)=O)C2)C)cc1 95031,C1(NC(c2ccc(CC)cc2)=O)CC2CC1CC2C(N1CCC1CC(=O)NC)=O 95032,N1(C(C(CC)(C)C)=O)CCC(NC(=O)Cc2ccc3n[nH]cc3c2)CC(C)(C)C1 95033,C(C(C)C(=O)N1C(C(=O)NCCOCCN(C)C)CC1C)SC 95034,C12(NC(=O)Cc3ccccc3)CCCC1CN(C(=O)COCC1CCOC1)C2 95035,Cc1cc(C(N2CCC(C(N3CCC(N(C)C)CC3)=O)C2)=O)cc(C)c1C#N 95036,c1(CNC(=O)NC(C#C)CC2CCCO2)ccc(C(F)F)c(F)c1 95037,C12(NC(C3(F)CCN(C(c4csc(Cl)c4)=O)CC3)=O)CCCCC1OCC2 95038,N1(C(Cc2ccc(C)o2)=O)CCC2CCC(NC(=O)Cc3ccc(Cl)s3)C1C2 95039,C#CC1(C(=O)NCC23CC(NC(=O)CC(C=C)c4cccs4)(C2)C3)CCCCC1 95040,C1(C)(NC(c2ccc(Cn3cc(C(C)(C)N(C)C)nn3)cc2)=O)CCCC1(F)F 95041,C=CCCCC(=O)N1CCCC1C=CC(=O)NCCN(C)C1CC1 95042,N1(C(CN(C(CNC(CC)=O)=O)C2CCC2)=O)CCC2(CCOCC2)C1 95043,C1(N(C(c2c(CNC(Cn3ccc(C)c3)=O)cc[nH]2)=O)C)CCC(CO)CC1 95044,n1(CCNC(c2cc(NC(C)=O)n[nH]2)=O)cnc(C(=O)NCC(C)OC)c1 95045,N1(C(c2c(CC)nn[nH]2)=O)CC2CCN(C(c3coc(Br)n3)=O)CCC2C1 95046,c1(CC)c(C(N2CCC(CNC(c3cccc(CO)c3)=O)CC2)=O)cnn1CC 95047,CN(Cc1ccccc1N1CCCC1)N1CCC2(CNC(=O)N2)C1 95048,C1(C(C)C)CN(C(=O)CN2CCOCC2)CCC1NC(C1(C2CCC2)CC1)=O 95049,c1(C(N(CC(=O)NCC(C)C)CC(C)C)=O)ccn2ccnc2c1 95050,C1(CNC(C(COC)(C)O)=O)CC(F)(F)CN1c1nccc(C#N)n1 95051,c1(NC(c2c(NC(c3c(C)ccc(O)c3)=O)c[nH]n2)=O)ncnc2sccc12 95052,CCCCCC(O)CC(=O)NC1CN(C(c2ccc(OC(F)F)cc2)=O)CC1F 95053,c1(C(=O)NC(CNC(C2OCCN(C(C)=O)C2)=O)C)ccc2c(c1)NC(=O)CO2 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95123,c1(C(=O)NC2CN(C(C3(C)CC(=C)C3)=O)CC2F)csc2c1CCCC2 95124,c1(NC)ccc(C(=O)NCC(C)(C(C)C)NC(=O)Cc2ccc(O)nc2)cc1F 95125,C1(C(N2CC(CC)(OC)C2)=O)CCCCCN1C(C1C2CCCCC12)=O 95126,C1(N(C(C(C)OCCOC)=O)C)CCCN(C(c2ccc(C#N)o2)=O)CC1 95127,N1(C(c2c(Cl)cc(C)nc2)=O)CCC2CCN(C(=O)CC3CC3(C)C)C2C1 95128,c1(NC(c2cccc(Cl)c2I)=O)ccc2c(c1)CN(c1nccc(C(F)F)n1)C2 95129,c1(C(N2CCCC2)=O)ccc(Cn2cc(-c3ccc(C(F)F)nc3)nn2)cc1F 95130,c1(C(N2CCC(C)(CNC(C(C)N3CCC3)=O)CC2)=O)c2c(nn1C)CCOC2 95131,CCC(F)(F)C(C)(C)C(=O)N1CCC1CNC(=O)CNS(=O)(=O)c1ccccc1 95132,N1(C(c2cc(OC)ncn2)=O)CCCC(CO)(NC(=O)CN(C)C(=O)C2CC2)C1 95133,c1(C(=O)NCCCCCC(=O)N(C2CCCC2C#N)C)cc2ccccc2[nH]1 95134,c1(C(N2C(C(=O)NC(CC)C(C)O)CC(F)C2)=O)ccc2cc[nH]c2c1Br 95135,n1(CCCN(CC(=O)OCC)C(=O)C2CC2)cc(-c2cnsc2)nn1 95136,C1(C(N2CCOCC2)=O)(N(C(C(F)=CCC)=O)C2CC2)CCSC1 95137,Cc1nn(C)c(Cl)c1CN1CCCC(N(C)C(=O)NCc2ccccn2)C1 95138,N1(C(CC(C(=O)OC)(C)C)=O)CCCC2C1CCCN2C(c1ncn(CC)n1)=O 95139,C12(C(=O)NCC3CN(CC)C(=O)O3)C(NC(=O)C(OC)OC)C3CC1C2C3 95140,N1(C(c2cc(C)c(C)[nH]2)=O)CC(CNC(C2OCCN(C)C2=O)=O)CC(C)C1 95141,C1(C(=O)NC(CCC)C)CCC2(CC2)CN1C(=O)OC(C)(C)C 95142,N1(C(CC2CCCN(CC)C2)=O)CCCC2CN(C(=O)CCC3CCCO3)CC12 95143,N1(C(C(COC)C)=O)C(C(=O)Nc2c(-c3ccccc3)nnn2C)CCC1C 95144,C1(NC(c2n[nH]c3c2COC3)=O)CN(C(c2cc(O)ncc2F)=O)C2CCCC12 95145,c1(C(C)S(N)(=O)=O)ccc(C(=O)OCCP(C)(C)=O)cc1 95146,N1(C(C2(CCN(C)C)CC2)=O)CCN(C(=O)C(C)(O)CC(F)(F)F)CC12CCC2 95147,c1(C(N(CCC(C(C)(C)C)NC(C(C)CO)=O)C)=O)cc2cc(Cl)sc2[nH]1 95148,c1(CNC(=O)CCOC2CCCC2)ncc(C(=O)NCC2CCSC2)cn1 95149,C1(C#N)(NCCCC(CN(C(C)(C)C)C(c2cccc(C(=O)OC)c2)=O)C)CCCCC1 95150,c1(C(=O)Nc2c(C)ncc(Br)c2)cc2oc(C)cc2[nH]1 95151,c1(CC)c(NC(C2CCC(C(C)C)N2C(c2ccncc2N)=O)=O)cnn1C 95152,C(=O)(C(C)C(C)(C)O)NC1C(CNC(c2nn(C(CC)C)c(C)c2)=O)C1 95153,N1(C(C(=O)N(CC(F)F)C)=O)CCCC1c1ncc(-c2ccccc2)[nH]1 95154,Cc1cnn(CC(N2CCC3(CC3NC(=O)C3=CCCCO3)C2)=O)c(=O)c1 95155,c1(CC(=O)N(C2C(NC(CC=CC)=O)CCCC2)C)ccc(C)c(Cl)c1 95156,C1(CNC(=O)C=CC2CC2)CCCN(C(c2cc(C3CCOCC3)no2)=O)C1 95157,c1(-c2nnc(C)o2)ccc(C(=O)NCC(CO)NC(=O)CCC=CC(C)C)cc1 95158,c1(CN(C(=O)C(=O)NC(c2cc[nH]c2)=O)CC(C)C)ccc(Cl)c(C(F)(F)F)c1 95159,O=C1NCCC12CCN(N1CCC(O)(c3ccccc3Br)C1)CC2 95160,C1(NC(C=C(C)CN2CCOCC2)=O)CC2CC1N(C(=O)CC1CC3CC3C1)C2 95161,n1(CCCOC)nnnc1C(c1nncn1C(C)C)NC(COC)C(C)C 95162,C1(CC(=O)NCC(CCNC(C(CC)=CCCC)=O)O)CCCOCC1 95163,C1(NC(Cc2scc(C)n2)=O)COC2(C1)CN(C(C1CC1F)=O)C2 95164,Cc1cc(C(=O)NC(CNC(=O)C(C)Cc2ccc(F)cc2)C(C)C)nc(O)c1 95165,c1(NCc2ccc(C)nc2Cl)ccc(S(=O)(=O)NC2COC(C3CC3)C2)cc1Cl 95166,c1(CC(=O)NC2C(NC(C(C3CCC3)OC)=O)C2)sccc1Cl 95167,C1(CNC(C(C=CC)O)=O)CCN(C(c2csnc2C2CC2)=O)CC1O 95168,Cc1cocc1C(N(CC(=O)NC1CCOC1)CCN(C)C)=O 95169,n1(CC(N2C(C)CCCCC2)=O)c(=O)nc(C(F)(F)F)n(C)c1=O 95170,C(c1cncnc1O)=CC(=O)NC(CCC)CNC(=O)CC1CN(C)C1 95171,C(CCCCCO)c1cn(CC(=O)NCCSCC2C(C)C2)nn1 95172,N1(C(c2cc(C)sc2C)=O)CCCC(NC(=O)C=Cc2cccnc2)C1C 95173,C1(CC(=O)N(C2CCCCC2)C)C2CN(C(=O)CC(F)F)CC12 95174,O=C(C1CCCn2nccc21)NC1(CO)CN(C(c2cc(F)c(F)cc2Cl)=O)C1 95175,c1(C(=O)NCCC2CCN(C(C=CC(=O)OC)=O)C2)cc(C)ccc1OC(F)F 95176,c1(NC2C(SC)CCC2)nc2ccccc2nc1NCC(C)C(C)C 95177,c1(C2(C(=O)NC3C(NC(=O)CO)CCC3)CCC2)ccc(Br)cc1 95178,c1(C(N(CCC(=O)N(CCCO)C)CC=C)=O)nn(C)cc1Cl 95179,C1(CN(C(C(C)OCC)=O)C)CN(C(c2c(Cl)n[nH]c2CC)=O)CCO1 95180,C(=O)(C1=C(F)CN(C(c2ccc3occc3c2)=O)CC1)N(C(C)C(C)(C)O)C 95181,N1(C(C(CCSC)N(C)C)=O)CCCC(CNC(=O)C=CC2CC2)CC1 95182,Cn1ncc2c(N)c(C(=O)NC(CNC(=O)CC3CC(=O)C3)CO)cnc12 95183,N1(C(C=CCC)=O)CC(C2CN(C(c3cc(C)c(OCCOC)c(C)c3)=O)C2)C1 95184,N1(C(CCc2nc(C)c(C)o2)=O)CC(CO)C2(C1)CN(C(C1CC(F)(F)C1)=O)C2 95185,C1(OC)CN(C(=O)CC2OCCO2)CC1NC(=O)CC1(O)CC1 95186,c1(CC(=O)N(CCNC(=O)C(C)(CC)OC)CC)ccc([N+](=O)[O-])cc1Br 95187,Cc1ccc(CC(C)C(=O)NC(C)C(CO)NC(=O)CCC2CCCCC2)cc1 95188,C(=O)(C(=O)N1CCC(C(N2CCCC(C#N)C2)=O)O1)N(C)C 95189,c1(OC)ccc(CN2CC3CC3(C(=O)Nc3c[nH]nc3C)C2)nc1Br 95190,C1(C(=O)NCCCCCNC(c2[nH]n(C)c(=O)n2)=O)CCCC12NC(=O)NC2=O 95191,N1(C(C2CCC(COC)C2)=O)CC2(CCN(C(c3cc(C)sn3)=O)C2)C1 95192,C1(C(=O)NCCN2CCC(NC(C3C4CCCC34)=O)CC2)CCCCC1(F)F 95193,C1(CNC(C(C(C)C)F)=O)CC(C)CN(C(c2sccc2CO)=O)C1 95194,C1(C(N2CCC(C(C)NC(=O)Cn3cnnc3)CC2)=O)Cc2nccnc2C1 95195,N1(C(=O)Cc2ccn(C(F)F)n2)CCCC(C2CN(C(=O)CO)C2)C1 95196,C(C)(CCC(=O)NCCN1CCC(NC(C2(C)CC2Br)=O)CC1)SC 95197,N1(C(C(C(C)OC)NC(c2c[nH]c(=S)cn2)=O)=O)CC2(C1)CC2(F)F 95198,C1(NC(CCSC)=O)CN(C(=O)COCC=Cc2ccccc2)CC12CC2 95199,Cc1ccc(F)c(C(N2CCC(O)(C(C)NC(=O)C=C3CCOCC3)C2)=O)c1Cl 95200,c1(CNC(C2(C)CCCS2)=O)cccc(CNC(C2(C(F)F)CCCC2)=O)c1 95201,C(=O)(C1CCc2cccnc21)NCC(C(C)C)NC(c1ncc(Br)cn1)=O 95202,C1(NC(C(C2CCCC2)NC(C(COC)C)=O)=O)CC2CCC1O2 95203,C=CCN=C(NCC=CC1CC1)NCC1C(C)(C)C1(F)F 95204,C1(NC(CN(CCC)C)=O)CCSC12CN(C(=O)C(C(C)C)n1cncn1)C2 95205,C(=O)(CC1=CCCCC1)NC1CN(C(C2CC3(CC(C)C3)C2)=O)CC12CC2 95206,C1(C(=O)NCC2N(C(c3c(SC)ccs3)=O)CCC2C)CC2(CCCO2)C1 95207,c1(C(=O)NCCC2N(C(CSCCC)=O)CCOC2)c(C)nc(O)nc1C 95208,C(c1nc2ccccc2s1)=CC(=O)NCC(N=c1nc(C2CCCC2)[nH]s1)C1CC1 95209,Cc1ccc(C2CCCC2N(C)CC2CC=CCC2CC2CCN(C)CC2)cc1 95210,C12(C)CC(OC)CN1C(=O)C1(CC1)NC2=O.c1(C(=O)OCC)cncn1C.CSC 95211,CC1(C)CCC(NC(=O)CCC2(NC(=O)C=CC3(C)COC3)CC2)C(CCO)C1 95212,N1(C(c2ccc(NC)cc2)=O)CC2(C1)C(NC(=O)C(C)CC1CC1)CCS2(=O)=O 95213,Nc1ccc(Cl)cc1C(=O)NCC1(F)CC(NC(=O)CC2CCOCC2)C1 95214,C1(NC(CCCC(=O)NC(C)C)=O)COC2(CCN(C(C)C)C2)C1 95215,CC1(C)CCN(C(C2OCCC2(C)C)=O)CC1C(=O)NC1(CC(N)=O)CC1 95216,CN=C(NCCCn1cccn1)NC1CC(OC(C)(C)C)C1 95217,c1(C(N2C3(CNC(c4cnc(OC)nc4)=O)CC(C2)C3)=O)cnc2cccnn12 95218,C1(C(N2CCN(CC(N3C(CO)CC(OC)C3)=O)CC2)=O)CC2(C1)CC21CC1 95219,CC1(C)CCCC(O)(C(=O)NCC2(C)CCN(C(C3CC=CCO3)=O)C2)CC1 95220,Cc1c(CC(=O)NCC=C2CCN(C(=O)CCCCN(C)C)CC2)cnn1C 95221,CC1CCC(C(=O)NC2CC2CNC(c2ccnnc2O)=O)CC1 95222,c1(C(=O)NC2CCN(CCCNC(CSCC#C)=O)C2)c[nH]c2ccncc12 95223,Cc1cc(N2CC(CN(C(=O)CC(C)c3cnn(C)c3)C)C2)c(Br)cc1[N+](=O)[O-] 95224,Nc1cc(C(=O)Nc2nc(-c3ccc(Cl)s3)cs2)c(F)c(F)c1F 95225,c1(C(N2CCCC(C)(NC(=O)CCC3CC3CC3CC3)C2)=O)ccc([N+](=O)[O-])cc1 95226,N1(C(C(C)(C)NS(C)(=O)=O)=O)CC2CCN(C(c3cc(F)cc(Cl)c3N)=O)C2C1 95227,c1(C(=O)NC2CCC(NC(c3c(SC)cccc3)=O)CC2)cnc(O)c(F)c1 95228,C(=O)(C(F)(F)CC(C)C)N1CC(CNC(c2c(CC)cns2)=O)C1 95229,Cc1cnc(C(=O)NC2CCN(C(=O)C=CC3COC(C)(C)O3)C2)cc1Br 95230,c1(CCC(=O)NCC2N(C(c3occ(C)c3C)=O)CC2)c(Cl)cncc1Cl 95231,C1(NC(CSCC#C)=O)C2CC3CN(C(=O)CC(n4nc(C)cc4C)C)C1C3C2 95232,c1(C(=O)NCC2(CNC(c3cnc(C(F)F)cn3)=O)CC2)c(F)cccc1F 95233,c1(C(=O)NCCCOCCN(C)C(C2CC23CCOC3)=O)cn2cccnc2n1 95234,c1(C(N(C(C(=O)NC(C(=O)OCCC)(C)C)C)CCC)=O)ccc(CC)c(F)c1 95235,CCCC(C(O)C(=O)N1CCC(N(C)CC)C1)NC(=O)CCn1cnc(=N)[nH]1 95236,CC(C)(F)C(C)(F)C(=O)N1CCCN(C(C2CCC(O)CC2)=O)CCC1 95237,C(=O)(C1=CCCN(C(C2C=CC=CC=C2)=O)C1)NCC=CCCC 95238,CC1CCCc2c(C(=O)NC3(CNC(=O)CCN4CCCC4=O)CC3)cnn21 95239,CC1C(c2ccccc2)NCCN1C(C1CCC2CC2CC1)=O 95240,C12(C(N3C4C(NC(CC5(OCC)CC5)=O)CC(C4)C3)=O)CCC(CO)(CC1)CC2 95241,n1(CC)c(O)nc2cc(C(=O)NCC3CCC3NC(=O)CSC)ccc12 95242,C1(CC)COC(C)CN1C(c1nc(F)ccc1Br)C(=O)NC1CC(F)(F)C1 95243,C12(NC(C=CC(=O)N(C)C)=O)CCCCC1N(C(=O)Cc1csc(=N)[nH]1)CC2 95244,N1(CC(=O)NCC(CNC(CCOC(C)=O)=O)C)CCCCC1C 95245,CC1OCCCC1C(=O)NC1CCC(NC(c2csc(Cl)c2Cl)=O)C1 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95511,c1(NCCCCNC(c2cnn(C3CCCC3)c2)=O)ncnc(Cl)c1CO 95512,N1(CC(=O)NCC2CN(C(C(OC)OC)=O)C(C)CC2)C(=O)CC(C)(C)C1=O 95513,c1(CC)cc(C(=O)NC(C)CC2CN(C(=O)Cc3cc(C)on3)C2)sc1C 95514,N1(C(CNC(=O)OCC)=O)CCOCC(C)(CNC(=O)C(C)C2CCCO2)C1 95515,C1(C(=O)NC2(CNC(C3(C4CCC4)CC3)=O)CCC2)CC(c2ccccn2)=NO1 95516,C=CCC(C)(C)C(=O)NCC1(NC(c2cnc(CSC)s2)=O)CCC1 95517,CCC(C(=O)NCC(C)NC(c1ccc2nccn2c1)=O)C(C)(F)F 95518,c1(CC(=O)NC2C(NC(C(C)OC(C)(C)C)=O)C(O)C2)cncnc1O 95519,c1(-n2cc(CCCC(=O)N(C(C)(C)C)C3COC3)nn2)cncc(NC2CCC2)c1 95520,C1(C(=O)Nc2cccc(C3(C)CC3)c2)CC2CCCCN2C1=O 95521,c1(C(=O)NCCCCC(C)NC(C2CCC3CC3C2)=O)ccc2c(c1)CCOC2 95522,c1(OCC)ccccc1-c1cn(CC2CCCN2C(C2CC2Cl)=O)nn1 95523,C(=O)(C(F)(F)c1ccccn1)NCC(C)(C1CC1)NC(=O)C(O)CN1CCCC1 95524,CCCC(C)CC(=O)N1CC(NC(c2ccnc(Cl)c2O)=O)C(C)C1 95525,Nc1ccccc1-c1cn(CCCC(=O)NCCc2csc(O)n2)nn1 95526,c1(-c2ccc(NCCC)s2)cccc(CN(c2cc(C)no2)C(C)=O)c1 95527,C(CCSC)(C(=O)N1CCC1C(=O)NOCCO)OC.c1(N)cnn(C(F)F)c1 95528,c1(C(=O)NCC(C)NC(=O)C(C2CC2)N(C)C)cc(-c2cccnc2)on1 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95841,N1(C(c2c(C)csc2)=O)CC2CC(C1)CN(C(C1CC(C)(C)C(C)(C)C1)=O)C2 95842,c1(C(N2CCOCC(NC(C(COC)(F)F)=O)C2)=O)cc2ccc(F)cc2cn1 95843,c1(C(N2CCC(N(C(c3c(C)nn[nH]3)=O)CC3CC3)CC2)=O)ccc(F)c(F)c1 95844,C1(NC(c2cc(C(C)C)no2)=O)CCCC(NC(C2(CN(C)C)CCOC2)=O)C1 95845,c1(C(=O)NCC(CC)(C)NC(C2CNC(=O)N2)=O)nc2ncccn2n1 95846,Cc1cccc(F)c1CNC(=O)CN(C(=O)CC1CCSC1)C 95847,N=c1cc[nH]cc1CNC(C1CCN(c2ccc(OC(F)(F)F)cc2)CC1)=O 95848,C1(C(=O)NCC(C)NC(COc2cccc(C(C)=O)c2)=O)CN2CCC1CC2 95849,CN(CCCC(=O)N1CCC(c2n[nH]cc2CNC(=O)C(O)C(F)(F)F)C1)N=O 95850,c1(CC)cccc(C(=O)NC2CN(C(=O)CCC(C)SC)CC2C(F)F)c1O 95851,O=C1CCC(C(=O)N2CC3(NC(C4CCCCS4(=O)=O)=O)CCC2CC3)=NN1 95852,Cc1onc(C(N2CCCC(NC(c3cc(Br)no3)=O)C2)=O)c1[N+](=O)[O-] 95853,c1(CC)ccnc(C(=O)NC2CC(NC(C3(n4cccn4)CCC3)=O)C2)c1 95854,c1(N2CC(C)(C)OCC2)nc2cccnc2c(=NC2CCC(CC(N)=O)C2)[nH]1 95855,N1(C(C(CC#C)(C)C)=O)CC(CNC(=O)C(C)n2cccn2)C2(CCOCC2)C1 95856,C1(CC(=O)NC(CNC(c2ccc(CNC(C)=O)s2)=O)CO)(OC)CCCCC1 95857,C12(CC(=O)N(C)Cc3cnccn3)CC(CCO1)N(C(=O)CC1COC(=O)C1)C2 95858,c1(CNC(N(C(C)C(=O)O)CCC)=O)cccc(-c2nnco2)c1 95859,N1(C(C(CC(C)C)ONC(C2CCOCC2(C)C)=O)=O)CCc2c(nnn2C)C1 95860,c1(C(=O)Oc2cccc(CN=c3nnn(C)[nH]3)c2)oc2ccccc2c1CO 95861,C1(C(N2CC3C(NC(C(C)N(C(C)=O)C)=O)C3C2)=O)CCC([N+](=O)[O-])CC1 95862,c1(CNC(C23CCCCC2C3)=O)ccc(CNC(c2cc(Cl)ncn2)=O)cc1 95863,C(CC(=O)N1CC2CCC(C1)N2C(=O)C=Cc1ncc[nH]1)(C(F)(F)F)OC 95864,C1(C(=O)NC(C(=O)NC)CC2CC2)CCC(C2CC2)N1C(C1CC(F)CN1C)=O 95865,N1(C(c2cnc(COC)s2)=O)CC2(CCC2NC(=O)C=C(C)Cl)C1 95866,c1(CC(=O)NCC(C)(C)NC(C2C(C)C2)=O)ccc(O)c(Cl)c1 95867,N1(C(C2(C)COC2)=O)CCCC2(CCCCC2NC(C2CC3CC3C2)=O)C1 95868,Cc1cc(C(=O)N(C2CC(C#N)C2)CC(N2CCC(CCO)CC2)=O)cc(C)n1 95869,N1(C(C(C)NC(COC)=O)=O)CC2C(NC(=O)CCN3CCC(O)CC3)C2C1 95870,N1(C(CCC(C)(C)NC(CCCOCCOC)=O)=O)CC2CCCCCC2C1 95871,Cn1nc(C(=O)N(c2nc(CSc3ccccn3)cs2)CCO)c2cc(Br)ccc12 95872,C(=O)(CC(C)(C)C)N(CCNC(C1CCC(OC)C1)=O)CC 95873,CC(C)(C)CC(O)C(=O)N1CC=CC1CNC(c1ncc2[nH]ncc2n1)=O 95874,N1(C(C2(C3CCCO3)CC2)=O)CCCCC1C(=O)N(C)CC1(CC)CC1 95875,C(CC(C(=O)N1CCOC(CCCNC(=O)C(Br)=C(C)C)C1)OC)OC 95876,c1(C(N(C(C)C(N2CCCC(C)(C)C2C)=O)CC)=O)ccc2[nH]ccc2c1 95877,CCC(CC(=O)NC1CN(C(c2[nH]cc(C)c2C)=O)CC(C)(C)C1)CC(F)(F)F 95878,c1(C(N2C3(CNC(CC4(C)CC4(Cl)Cl)=O)CC(C2)C3)=O)cccc2c[nH]nc12 95879,N1(C(c2c(COC)ccs2)=O)CCN(C(=O)C=Cc2cscn2)C(CC(F)F)C1 95880,c1(Oc2scc(NC(=O)Nc3cc(C(=O)OC)n(C)c3)n2)cc(F)ccc1Br 95881,Cc1nc(NC2CC2)sc1C(=O)NC(C)CN(C)C(C1CC2CC2C1)=O 95882,C(CC(C)(C)C)(C(=O)NOCc1ccc(F)cc1)NC(CC=C(C)C)=O 95883,c1(OC)ccc2c(c1)C(C(=O)NCC1CCCN1c1ccc(N)cc1)CC2 95884,c1(CC)cc(C(N2CCCC2(C)CNC(c2cc(F)cc(F)c2)=O)=O)ccc1C 95885,c1(C(=O)NC2C(C)CN(C(=O)CCCN(C)N=O)C2)noc2c1CC(C)(C)CC2 95886,C#CCC(C)(C)C(=O)NC1CC(N(C(=O)CCC=CC(C)C)C)C1 95887,c1(OC)cnnc(C(=O)NCC2(CN(C)C(C3CC4CCC3O4)=O)CC2)c1 95888,O=C(CN1C(=O)C(F)(F)Oc2ccccc21)OC(C(F)(F)F)c1nccs1 95889,C1(C(=O)NCCN(C(c2ccn(C)n2)=O)CC)CCN(S(=O)(=O)NC)CC1 95890,CC(CC(N)=O)C(=O)NCC(N=c1[nH]nc(-c2ccccc2)o1)c1ccccc1 95891,C1(CNC(C2CC(F)(CO)C2)=O)C2CN(C(=O)CSc3ccc(F)cc3)CC12 95892,C(=O)(NNc1cc(Cl)nc2ncccc12)NCC1(O)CCC(C)C1 95893,n1(CCCOC)nc(-c2ccc(N)cn2)nc1CCn1cnccc1=O 95894,C1(C2C(OCCC(=O)NC3CC3)C2)CCCN(C(c2cncc(C3CC3)c2)=O)C1 95895,N1(C(CN(C(=O)C(CC)CCCC)CC#C)=O)CCCNC(=O)C1CCOC 95896,C1(NC(CC(C)F)=O)CN(C(=O)CCOc2cccnc2)C2(CCCC2)C1 95897,C(CCC(O)CO)NC(C1CC(CNC(C2(CO)CCCO2)=O)OC1)=O 95898,C1(NC(c2cc(OC)c(Cl)cc2)=O)CCC2CN(Cc3nncn3C)CC2C1 95899,c1(C(=O)NC2CCC(C)(CNC(c3c(C)nn(C)c3)=O)C2)cccc([N+](=O)[O-])c1 95900,c1(SC)ccc(Cl)c(C(N2CCN(CCc3cn(C(C)C)nn3)CC2)=O)c1 95901,CC(C)C(C)CC(=O)N1CC(O)CC1CNC(=O)COc1ccon1 95902,C1(OC)CN(C(=O)C(C)N(C)C(C)=O)CCC1NC(C1CCCCO1)=O 95903,N1(C(Cc2nc(CC)sc2)=O)CC2CN(C(c3cccc(OC)c3N)=O)CC12 95904,C1(NC(C2CC(CC)(CC)C2)=O)C=CCN(C(=O)C(N2CCOCC2)C)C1 95905,c1(C(N2C(CC(=O)Nc3c(OC)cccc3)CCC2)=O)ccc(S(C)(=O)=O)c(F)c1 95906,Cc1c(C(N2CC3(NC(=O)CSc4cnn(C)c4)CC2C3)=O)cccc1C1CC1 95907,N1(C(C(C)(C)OCC)=O)CCCC(C(=O)NCc2nc(CO)n[nH]2)C1 95908,C(C)(CNC(c1ccc(-c2cccs2)o1)=O)(CO)NC(C=C(CCC)C)=O 95909,c1(OC(C)C)cc(C(=O)N(CCCN(C)C)CCO)ccn1.C12CCN(C1)C2=O 95910,c1(C(c2nnnn2C(C)C)NCC2(CCCC)CC2)ccc(-c2csc(C)n2)s1 95911,c1(C(N(C2CCN(C(c3cc(C(C)=O)on3)=O)C2)C)=O)cncc(C)n1 95912,c1(NC(C(C)n2ccnn2)=O)cccc(CNC(c2ccoc2Br)=O)c1 95913,c1(OCCC)c(F)cc(NCCCC(F)F)cc1F 95914,C1(NC(CCOC2CN(C(C3(CC=C)CC=CC3)=O)C2)=O)CC1C1CCCC1 95915,N1(C(c2c(C)ccs2)=O)CCN(C(C2CCN(CC(F)(F)F)C2)=O)CC2(CC2)C1 95916,C1(C(=O)NCC2(C(N(C3(CN(C)C)CCC3)C)=O)CC2)CCC(C)(C)C1 95917,C(=O)(CC(C)(C)CC(F)F)NC1CC(C)N(C(C2CC(N(C)C)C2)=O)C1 95918,Cc1cccc(C(=O)NCC2(C)CCC(NC(c3cnccn3)=O)C2)c1 95919,C1(C#N)(C(=O)NCC2CC(OC)CN2C(C2CCC2(C)C)=O)CCOCC1 95920,C1(C(=O)NCCSCCC=C)CCC(O)CN1C(c1cccc(OC)n1)=O 95921,C12(NC(CN(CCC)C)=O)CC(CNC(=O)CCC(C)(C)OC)(C1)OC21CCC1 95922,c1(C(N(C(CCC)C)C)=O)ccn(CCNC(=O)CC2(C)CCCO2)c1 95923,N#Cc1cc(Br)ccc1CN1CC2CN(c3ncc(C4CC4)cn3)CC2C1 95924,N1(C(C2(C)C(C)C2)=O)CCOCC(CNC(c2ccc(Cl)c(Cl)c2)=O)C1 95925,n1(CC(C)C)ccc(OCC(C)C)n1 95926,N1(CC(=O)NCC(CC)NC(=O)C(C2CC2)N(C)C)C(=O)NC2(CCCC2)C1=O 95927,N1(C(COc2c(COC(C)(C)C)ccc(C)c2)=O)CC2C3C=CC(C3)C2C1 95928,C(C(=O)N=c1ccn(C(C)C)[nH]1)(c1cccs1)NC(c1c(C)cns1)=O 95929,c1(-c2cccc(CO)c2F)ccc2nccn2n1 95930,CN=c1[nH]c(=NCCCN2CCOC2=O)[nH]c(=NC2CC(=O)N(C)C2)[nH]1 95931,C#CC(C(C)(C)C)NC(=O)COCCNC(c1cccc(CC)n1)=O 95932,C(=O)(C(C)Cc1cccnc1)N(C(c1cn(Cc2ncoc2C(F)F)nn1)C)CCS 95933,C(CC1C(=O)Nc2ccccc21)NC(=NCCCC)NC(C)CCC(F)F 95934,C1(C(N(CC(=O)OC)CCC)=O)COC2(C1)CN(C(=O)C(N1CCCCC1)C)C2 95935,C1(CCC)CN(C(C2CCCCN2CCC)=O)CCN1C(=O)C1=CCC1 95936,C(=O)(C1=NOC2(CCN(C(c3ccc(I)cc3F)=O)C2)C1)NC(C)C(C)(C)C 95937,c1(N2C(CNC(C3(OC)CCC3)=O)C(C)CC2)nc(O)c2ccc(Cl)cc2n1 95938,c1(NC)cnccc1C(=O)Nc1cnn(CCO)c1.C12(CCCCC1)C(=O)NC2 95939,c1(C(C(C)NC(=O)CCc2cnc[nH]2)NC(=O)CSc2nncs2)ccccc1 95940,C1(CNC(CCC(CC)C)=O)CC2(CO1)CN(C(=O)CC1CCCCC1)C2 95941,N1(C(c2c(C(C)C)ccs2)=O)CC(CO)C2(C1)CN(c1cc(Cl)ncn1)C2 95942,C=CCN(OC)C(=O)C(C)N(C(=O)CCC(CC)OC)C1CC1 95943,c1(C(N2CCCC2C(C)(C)OC)C(=O)NC(CC)(C)C)cnc(OC)c(F)c1 95944,C(=O)(C#Cc1ccccc1)NC1CCCN(Cc2c(C)c[nH]n2)CC1 95945,C1(NC(C2N(C(CSc3cccc(C)c3)=O)CC=C2)=O)CC2CC1CC2CO 95946,N1(C(C2C(c3ccc(C(C)C)cc3)C2)=O)CCC(C2(NC(=O)CO)CC2)CC1 95947,C#CCCCCC(=O)NCC12CC(NC(C3CCCC3(F)F)=O)(C1)C2 95948,C1(C2CCOC2)(C(N(CCN(C(C(C2CC2)OC)=O)C)C)=O)CCOCC1 95949,c1(C(=O)NC2CCN(CCCNC(C(C=C)OC)=O)C2)cc(O)cc(=O)o1 95950,C(=O)(CCOCCC#N)NCCN(C(COCCC)=O)CCCN(C)C 95951,c1(CC=CC(=O)NCC2CN(C(C3(F)CCOC3)=O)CCO2)ccc(F)cc1 95952,CC1CCN(C(c2cc[nH]n2)=O)CCN1C(C1(c2ccccc2)CC(O)C1)=O 95953,N1(C(C2(C(F)F)CCCC2)=O)CC(Nc2ncnc3scnc23)CC2(CCC2)C1 95954,c1(C(=O)Nc2c(C#N)nc(C)o2)cn2c(n1)CN(C(c1ccccc1I)=O)CC2 95955,CC(=O)CCCC(=O)N1CCCC1CN(C(=O)C(c1cccc(Br)c1)(C)C)C 95956,C1(C(N2CC(NC(=O)CCCCCO)C(C(F)(F)F)C2)=O)Cc2ccncc2C1 95957,Cc1nc2c(s1)CCCC2NC(=O)NNC(=O)C1CC1c1cccc(Br)c1F 95958,c1(C(N2CCCC(CNC(c3cncs3)=O)CC2)=O)c(F)ccc2c1OCO2 95959,N1(C(C(c2ccccc2F)C)=O)CCC2C(NC(=O)CSc3ccc(Cl)cc3)C12 95960,c1(C(=O)NCC=CCNC(c2cc(C)nn2CC(F)F)=O)c(Cl)ccc(C)c1O 95961,C1(C(=O)NCC(C)(CNC(c2ncc(C)cc2F)=O)OC)CC(=O)CC(=O)N1 95962,c1(C(=O)OC)ccc(C(=O)NC(CNC(c2ccn(CCOC)n2)=O)CO)s1 95963,N1(C(c2c(C)c[nH]n2)C(=O)NCCC#N)CCN(c2ccccc2)CC1 95964,C1(O)(C(C)NC(=O)CC2CCOC2)CCN(C(C2COC3COCC23)=O)CC1 95965,c1(C(=O)NC2CCN(C(C(CSC)C)=O)C(C)C2)cn2cnnc2cn1 95966,C1(C(N(OC)C)=O)CC(O)CN1C(C)=O.C(C)(C)C 95967,CC(C(C)(C)CO)NC(c1n[nH]c(C(C)C)n1)c1nnnn1-c1ccccc1 95968,N1(C(C(C)CC(N)=O)=O)C2CCC1CC(N(C)C(c1cccc(C(N)=O)c1)=O)C2 95969,c1(C(N(c2ccc(-c3nn[nH]n3)cc2)C(C)CC(=O)O)=O)ccc2c(c1)C(=O)OC2 95970,C1(NC(C2CCN(c3ccccc3)C2)=O)CCN(C(=O)Cn2cc(Cl)cn2)C1 95971,C1(C(=O)NC(C2N(c3snc(CCSC)n3)CCC2)(C)C)CCSC(C)C1 95972,N1(C(=O)Cn2cc(C3CC3)nn2)CCC2CN(C(=O)C(O)c3ccco3)CC2C1 95973,C1(C(C)Cc2cc[nH]c2)CCN(NC(c2cc(C(C)(C)C)n[nH]2)=O)CCC1(F)F 95974,c1(CNC(c2ccc(NC(c3cc(CC)n(C)n3)=O)nc2)=O)nc(Cl)ccc1F 95975,c12ccc(cc1)OCCO2.C(C)(C)(CC(=O)OC)NC(=O)Nc1ncn(NC)n1 95976,c1(C(N(CCN(C)CCC2CCCC2)C)=O)cc(-c2ccoc2)on1 95977,Cc1cnc(C(=O)NCC2CCCCC2NC(c2c(O)cccc2F)=O)c(C)c1 95978,c1(C(=O)NC(C(CO)NC(CN(CC)CC)=O)C)ccc(F)cn1 95979,CC(C)C(C(C)NC(c1cscc1Br)=O)NC(c1ccc(CO)o1)=O 95980,C=CCCC(C)NC(=O)C(C)CN(C)C(c1csnc1OC)=O 95981,c1(NC)ccc(Cl)c(C(=O)NCC(C(C)(C)C)NC(=O)C(C)c2ccon2)c1 95982,C1(C(=O)NCc2cncnc2)CN(Cc2cnc(Cl)c(Cl)c2)CCC1(F)F 95983,CCCS(=O)(=O)CC(=O)NC(C)CNC(=O)CCCNC(=O)OCC 95984,C1(CC(=O)NC(C#C)(C)C2CC2)C2CCC(C2)N1C(C1CCOC1C(=C)C)=O 95985,C1(N(C)C(C2CCCS2)=O)CCCC2CN(C(=O)CC3CCS(=O)(=O)CC3)CC12 95986,C=CCC(CC(=O)NCc1cccc(C#N)n1)NC(=O)Cc1cccnc1OC 95987,N#Cc1cc(NC(C2COCCN2C(C2CC2C2CC2)=O)=O)cc(Cl)c1 95988,C=CCC(C)(CNC(=O)C1=CCC(NC(=O)CCOC2CCCC2)C1)CO 95989,c1(OC)cc(OC)c(C(N2CC(NC(=O)C(C)O)CC3(CC3)C2)=O)c(N)c1 95990,c1(C(=O)NC2C(C)CCN(C(=O)CCOC3COC3)C2)cc2cccc(Cl)c2[nH]1 95991,c1(C(N(CC(C)O)CCNC(=O)Cc2cc(C3CC3)no2)=O)cnc2c[nH]nc2c1 95992,N1(CC)CC2(CN(C(c3ncoc3CNC(=O)CNC(N)=O)=O)C2)C1 95993,C1(CC)(CO)CCN(C(=O)C(CO)NC(c2cc(Cl)no2)=O)C1 95994,C1(CC#C)(C(=O)NC(C)CC(C)NC(C2CCOCC2)=O)CCCC1 95995,Cc1cc(C(C)(C(=O)NCCC(C)CO)NC(=O)OC(C)(C)C)ccc1Cl 95996,c1(OC)ccc2[nH]nc(C(=O)NC(C)CNC(c3c(F)cc(C)cc3F)=O)c2c1 95997,C=Cc1cccc(CN2CCN(CC(N3CCC(C)CC3)=O)CC2)c1 95998,CC1CN(C(c2cccn3ncnc23)=O)C(C)CN1C(c1ccc(O)nc1Cl)=O 95999,CCCC(CCC)CC(=O)NCC1(F)CC(CNC(=O)CC(CC)OC)C1 96000,C(CO)(CCCCNC(C1(CF)CCC1)=O)NC(=O)COc1ccccc1 96001,c1(C(N2C3CC(NC(C=C4CCC(C)CC4)=O)C2CC3)=O)cccc2nc[nH]c12 96002,C(=O)(C(C)CS(C)=O)NCC(C12CCC(CC1)C2)NC(c1sc(C)c(O)n1)=O 96003,c1(C(=O)NCC#CCNC(c2nncc(OC)c2)=O)cc2ccc(Cl)c(F)c2o1 96004,c1(C(=O)NC2C3N(C(c4ccc(C)o4)=O)CC(CC3)C2)ccc2ncccc2c1 96005,C12COCCC1CC(=O)N2.CS(=O)(=O)SC1CC1c1ccco1 96006,C1(NC(C(CCC)O)=O)CCCN(C(=O)CCc2ccc(F)nc2)CC1 96007,C1(C(=O)NC2CC(NC(C=CC3C(C)C3(Cl)Cl)=O)C2)C2CC3C(C2=O)C13 96008,C(CC(=O)NC1CCn2ccnc2C1)(C(C)(C)C)NC(C=Cc1n(C)ncc1)=O 96009,c1(-c2c(C)occ2)nc(CC2CCC(O)C2)n(C2COC(C)(C)C2)n1 96010,c1(C(=O)NC(CC=CC)C(=O)NCC(O)CCO)cnc2ccccn12 96011,C(=O)(C1=CCOCC1)NCC1(C)CCN(C(=O)C=CI)C1 96012,N1(C(C2C(C(N)=O)C2)=O)CC2CCC(C1)N2C(c1ccc(F)c(N)c1)=O 96013,CC1COCC(CC(=O)NC(c2cccnc2)C(=O)N2CC(O)C2)O1 96014,c1(NC(CC)CNc2ccccc2)nccc(=NC(C)c2cccnc2)[nH]1 96015,c1(OC)ccc(C(N2CC(NC(C3CCOCC3)=O)C3CC3C2)=O)cc1[N+](=O)[O-] 96016,c1(CCC(=O)NC2CC3CCC2N3C(C2CC3(CC3)CO2)=O)ccc(O)c(F)c1 96017,CC(C)C(C(=O)NC1(C(N)=O)CC1)n1cc(C(C)(C)O)nn1 96018,C1(N(C(Cc2cc(C)sc2C)=O)C)CCCCN(C(C2CC2C(F)(F)F)=O)C1 96019,c1(C(N2CCC(CCCc3cn(CC)nn3)CC2)=O)ccc(C)cc1C(F)F 96020,N1(C(C2CCN(C(c3cscc3Br)=O)C2)=O)CCC(O)(c2ccccc2)CC1 96021,CCC(CN(C)C)CC(=O)NC1CC(CNC(=O)C(=O)Nc2ccccc2)C1 96022,c1(NC(c2c(C)n(-c3cc(F)ccc3F)nn2)=O)ccc2c(F)n[nH]c2c1 96023,C(=O)(CC(C)P(C)(C)=O)NCC(C(C)(C)C)NC(c1scc(OC)c1)=O 96024,C1(N(CC(=O)OC)CC)(C(=O)N)CC(F)C1.C(CC(=O)OC)(C1CC1)OC(=O)C1CC1 96025,C1(CNC(=O)N(C)C)CCC(C2COCCN2C(=O)CCCCCOC)O1 96026,N1(C(C(C=C)O)=O)Cc2ccccc2CC1CNC(c1cc(C2(C)CC2)on1)=O 96027,c1(C(=O)NC(C2CCN(C(CS(CC)=O)=O)C2)(C)C)cc(F)cc(C)c1C 96028,C1(CC)CN(C(c2cc(C)n(C)c2)=O)CCC1CNC(C1CC1[N+](=O)[O-])=O 96029,N1(C(c2n[nH]c(C)c2O)=O)CC(=O)NCC1C(=O)NC1CCOC1(C)C 96030,C1(C(C)NC(=O)C(C)(F)F)CN(C(c2ccc(Cn3ccnc3)[nH]2)=O)CCO1 96031,CC(C)(C#N)CC(=O)N1CCCC1CCC1CCN(C(C2CC(=C3CC3)C2)=O)CC1 96032,C(=O)(CC(C)c1ccco1)N(C1CCCCC1)CCNC(CSCC#C)=O 96033,Cc1sc(Cl)c(C(=O)NCC(=O)NC2CC(NC(C)CCCC(C)C)C2)c1C 96034,C(=O)(C(C(C)C)C(C)C)N1CC2C(CN(C(COCc3cc(C)on3)=O)C)C2C1 96035,C1(CN(C(=O)Cc2ccoc2C)CC)CCCN1C(C1CCCCO1)=O 96036,N1(C(C2CCC(C)CC2)=O)C(CC(N2CCCC2CC(N)=O)=O)C2CCCC12 96037,C1(NC(c2c(SCC)cccn2)=O)CC2CC1CN(C(=O)CC1CC3CC3C1)C2 96038,C1(C(C)NC(CC(=O)NCC#C)=O)CN(C(c2ncsc2CC)=O)CCO1 96039,c1(C(=O)NCCN(CC(C)O)C(=O)CSc2nnnn2C)cccc2nsnc12 96040,c1(OC(C(=O)NCC=CCNC(CCC)=O)(C)C)ccc([N+](=O)[O-])cc1 96041,c1(CN(C(c2c(C)cc(CC)o2)=O)Cc2cccnc2F)ccc(Cl)c(Cl)c1 96042,C1(NC(C(C)c2cccs2)=O)CCN(C(c2c[nH]c(C(F)(F)F)c2)=O)CC1F 96043,c1(C(=O)NCCC2OCCN(C(CC(=C)C)=O)C2)ccc(O)cc1[N+](=O)[O-] 96044,C1(CCC(=O)NC(C2(C(N(CCCOC)C)=O)CC2)C)CCC(=O)C1 96045,c1(C(N(C)CC)=O)cc2ccc(OCCN(C(COC(CC)C)=O)C)nc2[nH]1 96046,N1(C(C)=O)CCC(F)(F)C(NC2(c3nnnn3C)CCN3CCCC23)C1 96047,C1(NC(C2(COC)CC=CC2)=O)COC2(C1)CN(C(=O)Cc1ccoc1)C2 96048,N1(C(c2ccnc(C(=O)OC)n2)C(=O)NCCCSC)CCC(S(N)(=O)=O)CC1 96049,N1(C(CSCC#C)=O)CC(CNC(=O)C(CC)OCC)C(C)C1 96050,C1(C)(C(=O)NC2(CCCC(=O)NC(c3cnsc3)C)CCC2)CC(=O)N(C)C1 96051,C1(C(N(CC(O)CNC(c2coc(CO)c2)=O)C)=O)CC12CC(C)(C)C2 96052,N1(C(C2(CNC(c3c(C)snn3)=O)CC3(CC3)C2)=O)CC2CCC(C1)C2C#N 96053,c1(C(N2CCC(OC(F)F)CC(C)(C)C2)=O)cnc2ccccc2c1 96054,C1(C)(CC)CC(NC(C23CC(CO)(C2)OC3C)=O)CN1C(=O)CSC(F)F 96055,C1(NC(c2cnc(S)nc2)=O)CN(C(C2CC2F)=O)CC2(CCC2)C1 96056,C1(n2cc(C3CN(C(=O)CCC4CC45CCC5)C3)nn2)CCOCC1O 96057,c1(C(=O)NC2CC(NC(CCCOCCC)=O)C2)ccc(C(C)C)cc1O 96058,C1(C)(C(=O)NCC(C)OCc2ccco2)CCCN(C(c2cccc(I)c2)=O)C1 96059,N1(C(c2ncccc2Cl)=O)CCCC2(CC(NC(=O)C(F)(F)C3CC3)CO2)C1 96060,c1(C(=O)NCC2N(C(c3c(COC)cc[nH]3)=O)CCC2)nc(C)n2c1CCCC2 96061,C(C(CCO)C(C)(C)C)N(C(=O)NC1C(C)CCC1)CC1CC1 96062,N1(CC(N2CCCN(c3c(C)c(O)c(Br)cn3)CC2)=O)CC2(COC(C)(C)C2)C1 96063,c1(NCCSc2ccc(C)cc2)nc[nH]c(=NCC2CC23CC3(F)F)c1C 96064,Cn1cc(Cl)c(C(=O)NC2CC2CNC(c2cnc(-c3ncccn3)s2)=O)n1 96065,C1(N(C)C(C2CC2F)=O)CCN(C(C2CC(c3ccccc3)CO2)=O)CC1 96066,C1(C(C)CNC(C2C=CCS2)=O)CCN(C(c2cnc(O)o2)=O)CC1 96067,c1(OC)nccc(C(N2CCCCC2CCC(=O)N(C)CCn2ccnc2)=O)n1 96068,N1(C(CC(CCCC)O)=O)CC2(CCN(C(c3cc(C)nc(C)c3)=O)CC2)C1 96069,C1(C)(CC(=O)OC)CCN(C(c2csc(CNC(C3C4CCC(F)C34)=O)c2)=O)C1 96070,C1(F)(C(=O)NCC2N(C(c3c(CC)nco3)=O)CC=C2)CCCN(C)C1 96071,c1(-c2nc(C(C3CC3)OC)nn2-c2nc(Br)nn2C)cnn2c(C)ccnc12 96072,Cn1cc(C(N2CCC(F)(CNC(=O)C(O)C(F)F)C2)=O)c(Cl)n1 96073,N1(C(C2N(Cc3c(C)cc(Br)cn3)CC3(CC3)C2)=O)CCC(C)(CO)C(O)C1 96074,C#CCCC(O)CCNC(c1cccnc1CNC(=O)C(C)C1(O)CCC1)=O 96075,C1(C(N2CC(SC)C(n3cc(C(C)(C)CO)nn3)C2)=O)CCCCN1N=O 96076,Cc1cnc2nccc(C(N3CC(CNC(c4cscn4)=O)CCC3C)=O)c2c1 96077,c1(NC(C2C(NCc3ccc(OCC)c(C#N)c3)C2)=O)nccc2scc(Br)c12 96078,N1(C(Cc2cc(C)[nH]n2)=O)CCC2CN(C(c3coc4c3COC4)=O)CC2C1 96079,N1(C(C)(C)CO)CCN(C(=NC2CC2)NCC(c2ccccc2F)O)CC1 96080,C(=O)(C(O)P(C)(C)=O)N1CC2C(C(N3C(C)(C(=O)NC)CC3)=O)C2C1 96081,C1(N(C(c2c(NC)scn2)=O)C)CCCN(C(=O)C(C)CC(C)C)CC1 96082,c1(C(N2CCC(C(=O)NCCCSC)(CC)C2)=O)cc(C#N)[nH]c1C 96083,C1(C(=O)NC(c2cnn[nH]2)C)CC(O)CN1C(C1CN(C(N)=O)C1)=O 96084,c1(CC(=O)NC(CNC(c2ncn(C)c2)=O)C2CC2)cccc(Br)c1 96085,c1(CC)ccc(CC(=O)NC2CCC(C)N(C(c3[nH]c(C)cc3C)=O)C2)cc1F 96086,C(=O)(C1=NOCC1)N(C1CCCC(N(C)C(c2cncc(N)n2)=O)C1)C 96087,C(=O)(C#CC1CCCOC1)N1CC(C(C)NC(=O)Cc2cscn2)OCC1 96088,Cc1ccc(C(=O)NC(C(=O)Nc2c[nH]c(=S)cn2)c2ccoc2)cc1 96089,c1(C(=O)OCC)cc(C(N2CCCC2CCNC(=O)C(C)C2CCC2)=O)[nH]c1C 96090,C1(NC(C(F)OC)=O)CN(C(=O)Cc2cncn2C2CC2)CC1O 96091,c1(C(=O)NC2C(CNC(C3(C(C)C)CCOCC3)=O)CC2)cc(C#N)ccc1F 96092,c1(Cc2nnc(CNC(N(CCC#N)C)=O)o2)ccc(-c2ccccn2)cc1 96093,N1(C(C(C)(C)F)=O)CC2CCC(CNC(=O)CCc3cccc(F)c3)(C2)C1 96094,Cc1ccc(C(=O)N(C2CCN(C(c3cc(Cl)no3)=O)CC2C)C)nc1O 96095,CCC(F)(C(=O)OC)C(=O)NC(C)CCNC(C1(n2ccnn2)CC1)=O 96096,CC1CN(C(=O)C=Cc2cnccn2)CC(C)CN1C(C1COC1)=O 96097,Cn1ccc(C(=O)NC2CCC2C(=O)Nc2ccc(C(F)(F)F)cc2F)cc1=O 96098,C1(CCC)CCCN(C(=O)C(CNC(=O)C=NOC)CCC)CC1 96099,C12(CNC(C3CC(CC)(CC)C3)=O)CCCC(CN1C(c1cncc(C)c1)=O)C2 96100,c1(NC(C2CCCC(C(=O)OC)C2)=O)nn(C)c2ccccc12 96101,c1(OC)ccc(NC(=O)NC2CN3CCC2(C(F)(F)F)C3)c(OC)c1 96102,C1(CNC(C2CCCN2C=O)=O)CCN(C(C23CCCC2CCC3)=O)C12CC2 96103,C1(CCC=C)(C(=O)NCC(N2CCOCC2)C)CN(C(C2CCCO2)=O)C1 96104,C1(CC(=O)NCC(C(C)C)NC(C2CCC(C(=O)OC)C2)=O)CCCC(C)(C)O1 96105,C(CC(=O)N1CC2(CCOC2=O)C1)(C(C)(C)C)NC(C(CCC)(C)O)=O 96106,C=CCC(F)(F)C(=O)NC1CN(C(c2cc(CC)ccn2)=O)CC1OC 96107,N1(C(c2ccn(CC)n2)=O)CCCCC(NC(c2c(NC(C)=O)c[nH]c2C)=O)C1 96108,CC1CN(C(c2ccnn2CCF)=O)CCC1CNC(C1CC2(CCOC2)C1)=O 96109,CC1CN(CC(=O)NC2CC2)CCC1NC(c1cn(CC2(O)CC2)nn1)=O 96110,Cn1ccc2ccc(C(=O)NC(C)(CNC(C3CC(O)C3)=O)C3CC3)cc12 96111,c1(C(C(=O)NCCC)N(CCC(C)OCC)C)ccc(C)c(OC)n1 96112,N1(CC(c2cccc(C)c2)=O)CC(S(=O)(=O)C2CCCCC2)C1 96113,N1(C(C2N(CC)CCOC2)=O)CCCC(O)(CCNC(=O)Cc2ncoc2C)C1 96114,Cc1nn(-c2ccccc2)nc1CNC(=O)Cn1cc(C2CC2CO)nn1 96115,C(C(C)C(F)C(=O)NC(C)(C)CN(C)C)NC(Cc1ccc(C)s1)=O 96116,c1(C(N2CCC(CC(N3CCC(CC(=O)OC)CC3)=O)C2)=O)ccc(C#N)c(Cl)c1 96117,C(CCC(C)CC(=O)NC1(CF)CCN(C(=O)CN(C)CCO)C1)=C(C)C 96118,n1(CC(=O)NC2C(CNC(CCSCCC)=O)C2)nc2n(c(=O)c1=O)CCC2 96119,CC(C)CCC(=O)N(CC(O)CN(C(=O)CNS(=O)(=O)Cc1ccon1)C)C 96120,C1(NC(C2CCC(C(F)F)CC2)=O)COC2(C1)CN(C(C1(F)CCCC1)=O)C2 96121,N=c1c(C(=O)NCCCCC2CCCO2)c[nH]n1Cc1ccccc1 96122,N1(C(Cn2c(C)nnn2)=O)C2CCC1C1CC1(NC(C1CCOCC1(C)C)=O)C2 96123,C(=O)(C(C)(C)C(=O)N1CCCCC1Cc1cn(-c2cccnc2)nn1)OC 96124,Cc1ccc(CC(N2CCC(C(F)F)(CNC(C3CCC3(C)C)=O)C2)=O)c(C)c1 96125,C(=O)(CC(F)(F)F)NCC(=O)N(C)CC1N(C(c2nnc(CC)s2)=O)CCC1 96126,c1(C(N2CCCCC(CNC(C3C(C)C3)=O)C2)=O)ccc2nn[nH]c2c1 96127,Cc1ncc(Br)c(C(N2CC3CC2(CO)CO3)=O)n1 96128,CC(C)(CCNC(c1csc(-c2ccccc2)c1)=O)C1CC1 96129,C(=O)(C1=CCCN(C(C2CC(O)C2)=O)C1)N(CC(C)O)CC(C)O 96130,CC1SCCCN1C(N1CCCC1c1ccn(C)n1)=O 96131,C1(C(N(CCC(=O)NCC2C3COCC23)C)=O)OC2CCC1C2 96132,CC1CC(NC(c2ncccc2C(F)F)=O)CN1C(=O)CCc1ccon1 96133,N1(C(COC(C)C)=O)CCCC(NC(c2ccn(C)c(=O)c2)=O)C(F)C1 96134,N1(C(c2n(C(CC)C)ncc2)=O)CC2CCN(C(C3CCC(=O)N3)=O)CCC2C1 96135,c1(OCC)ccc(CCC(=O)NC(C)(C)C(C)NC(=O)C=Cc2ncco2)cc1 96136,C1(C(=O)OC)(NC(c2cc(C3CCCN3C)[nH]n2)=O)CCCNC1 96137,N1(C(c2c(C)cno2)=O)CCN(c2nc(C(C)C)ns2)C(CCO)C1 96138,c1(CN=C(NC(COC)C)NCCc2c(C)cccc2C)cc(F)c(C)cc1F 96139,C1(C)(C(=O)NCCCN(C(C)=O)C)CCN(C(C2CC(=C3CC3)C2)=O)CC1 96140,C1(C(C)(C)C)CCC1C(N1CC(C(O)C(=O)NCc2cnc[nH]2)C1)=O 96141,N1(C(=O)Cc2ccc(C)o2)CCC(NC(C2(C(=O)OCC)CC2)=O)C(C)C1 96142,N1(C(C2(CC=C)CC2)=O)CCCC(C2(NC(c3cnc(Cl)c(F)c3N)=O)CC2)C1 96143,c1(NC2CCN(C(=O)NC)CC2)nc(C(F)(F)F)ccc1I 96144,c1(OC)ccncc1C(=O)NCc1nocc1C(=O)NCCC(F)(F)F 96145,CC(C)CC(C)(O)C(=O)N1C2CCC(C(=O)NCc3cnns3)C1CC2 96146,N1(C(Cc2cc(C)ns2)=O)CCC2(NC(=O)CCn3cccn3)CCCCC12 96147,c1(OCC)cc(C=CCNCc2ccc(Cl)s2)ccc1OC 96148,N1(C(CC(COC)(C)C)=O)CCC(N=[N+]=[N-])(C(=O)NOCC(N)=O)C1 96149,Cn1ccc2[nH]c(C(N3CCC(NC(C4(n5cccn5)CC4)=O)C3)=O)cc12 96150,c1(CNC(CCC2N(C)CCC2)=O)ccc(C(=O)NCC(N2CCCC2)C)nc1 96151,C(C(=O)N=c1cc(C)n(C2CC2)[nH]1)=CC1CN(C(C2C(CC)CCCC2)=O)C1 96152,N1(C(CCC)=O)CCC2(CCCN2C(=O)CCc2ccc(OC)cc2)C1 96153,Cc1cccnc1CC(N1CCC(C(F)F)(CNC(c2cc(CF)on2)=O)C1)=O 96154,c1(C(N2CC3C(CNC(C=COCC)=O)(C3)C2)=O)cc(Cl)cc(Cl)c1OC(F)F 96155,CC1(C(=O)NCC2CN(C(C3C=CCS3)=O)CC2O)CCCC1O 96156,c1(C(=O)NC(CNC(=O)C=CCn2cncn2)CO)ccc(C2CCOC2)nc1 96157,CN1CCC(C(N2CCCC2C(=O)NC(C)(C)CCCC)=O)C1=O 96158,c1(NC(C(C)NC(=O)NC)=O)cc(NC2CCCC2)c(F)cc1F 96159,Cc1nc(NCc2cc(CO)on2)cc(=NC(C)c2ccc(Cl)c3c2CCC3)[nH]1 96160,c1(NC(C2CC2NCc2cscn2)=O)cccc(Cl)c1I 96161,c1(-c2c(OC)cccc2F)nc2c(s1)C(NCCC1CC1)CCC2 96162,N1(C(COCCOC)=O)CCC2(CNC(=O)C3=NNC(=O)CC3)CCCCC12 96163,c1(NCC(C)CNC(=O)CC2CC(O)C23CCC3)ncnc(N(C)C)c1[N+](=O)[O-] 96164,c1(CN2CCCC(C(N3CCOC4CC34)=O)C2)cnc(Cl)cc1Cl 96165,c1(C(=O)NC2(CN(C)C(c3ccc(CO)cc3)=O)CC2)cccc(N(C)C)n1 96166,Cc1c(C(N2CC(C)(NC(C3OC4CCC3C4)=O)C2)=O)[nH]c2c(Cl)cccc12 96167,c1(C(=O)NCC2CN(C(C3(CC(C)=O)CC3)=O)CC2C)cccc(Cl)c1F 96168,N1(C(CC2(C=C)CCC2)=O)CCC(C2(NC(=O)C(C)O)CC2)C1 96169,c1(CO)cc(-c2ccc(Cl)c(C(F)(F)F)c2)ccc1O 96170,c1(COC)nn(C)cc1C(N1CCCC1(C)CNC(c1ccc(C)nc1)=O)=O 96171,N1(C(c2cnn(C)c2C2CC2)=O)CCC2(CCN(C(=O)CC3(C)CC3(Cl)Cl)C2)C1 96172,c1(C(=O)NCC(CN(C(c2c(O)ccc(CC)c2)=O)C)C)cc(S(N)(=O)=O)co1 96173,c1(OC)cc(C(=O)CN2CCC(S(N)(=O)=O)C2)cc(Br)c1OC 96174,C1(OC)CCC(C(=O)NCC2CCCCC2NC(=O)CSC2CC2)CC1 96175,Cc1ccc(Cl)c(N)c1C(N1CCC(CNC(=O)C(C)(F)F)C(F)(F)C1)=O 96176,C=CCCC(C(=O)N(CCNC(=O)CC(=C)Br)CCOCCO)c1ccccc1 96177,C1(CNC(C(C)(C)C#N)=O)CCCCN(C(=O)CC2SC(=N)NC2=O)C1 96178,c1(C(=O)OC(c2ccc(F)cc2F)C(=O)OC)cccc2nsnc12 96179,C1(CNC(CNC(CC)=O)=O)(NC(C23CCCC2CC3)=O)CC2CCC1CC2 96180,CCC(C)(C(=O)N1CCCN(CCNC(=O)C(C)(C)C2CCCC2)CC1)C(F)F 96181,C1(NC(c2cnn(C)c2Cl)=O)CCC2CC1CN2C(c1cc([N+](=O)[O-])c[nH]1)=O 96182,c1(C(=O)NCC(=O)NCCNC(C2ON=C(CC)C2)=O)n[nH]c2ccc(Cl)cc12 96183,Cc1cc(NC(C2CCCCCN2C(c2cccs2)=O)=O)ccc1O 96184,CCCCCCCCN(C(=O)C(CC1CC1)NC(=O)C(C)O)CC.OCC 96185,C1(C(N2CC(CCC)N(C(=O)C=C(C)Cl)CC2)=O)COc2cc(F)ccc2C1 96186,N1(C(c2c(OC)c(Br)ccc2)=O)CCn2cnc(C3=CCSCC3)c2C1 96187,Cc1cc(C(=O)NCCN2CCN(C(C3CCNC3=O)=O)CC2)cnc1O 96188,N1(C(C(C=CC)O)=O)CCCC2(CCN(C(=O)C=CSc3ccccc3)CC2)C1 96189,CCC(C)(CC)C(=O)N(CCCCCNC(C1CCCC(C)CC1)=O)C 96190,C(=O)(C(F)(F)C(O)C1CC1)NC(C)C(CO)NC(c1cc(Cl)ccc1F)=O 96191,C1(C)(CC)C=C(C(=O)N2CC3(CNC(c4n[nH]cc4OC)=O)CC2CO3)C1 96192,CC(C)CN=C(NCC1(CN(C)C)CCC1)N1CC(C)S(=O)(=O)C(C)C1 96193,CCC(CC(C)C)C(=O)NCC1CC2(CC2)CN1C(c1cn(CCOC)nn1)=O 96194,CS(=O)(=O)c1ccc(C(N2CCC(N(CCO)C(C3CCNC3=O)=O)C2)=O)cc1 96195,C1(CNC(CC(C)N(C)C)=O)CN(C(c2n[nH]c3c2COCC3)=O)CC(C)(C)O1 96196,CCCC(C(C(=O)NC)N1CC(O)C2(CCC2)C1)OC 96197,c1(CC(N2CC(=C(CNC(C(CC)n3ccnc3)=O)F)C2)=O)ccc(F)cc1C 96198,C(=O)(C(F)(F)C(F)(F)F)NCC1CN(C(Cc2ccc(C)c(Cl)c2)=O)CC(C)O1 96199,N1(C(C=CC(CC)C)=O)CC(O)(C(F)C(=O)N2CC(OC(=O)N(C)C)C2)C1 96200,N1(C(C2(C)CC=CC2)=O)CC2(CCCC2NC(C2(C3CCC3)CC2(F)F)=O)C1 96201,c1(NC(c2nc(C(N3CCC34CCCCC4)=O)cs2)=O)c(F)cc(F)cc1Cl 96202,C1(CN(C(=O)C(C)(O)COC)CC)CCN(C(c2cnn(C)c2SC)=O)CC1 96203,N1(C(C2(C)CC(=C)C2)=O)CCN(C(c2cnc(C)o2)=O)C(c2cn[nH]c2)C1 96204,CC(C(=O)N1CCC(n2cc(-c3ccccc3O)nn2)CC1)C(F)F 96205,N1(C(=O)Cn2nnc(=O)[nH]2)CC2(CCN(C(c3ccc(Br)cc3F)=O)CC2)C1 96206,N1(C(C(Cn2ccc(C)n2)C)=O)CC2CN(C(c3ccc(C)c(O)c3)=O)CCC12 96207,N1(C(CC(COC)(C)C)=O)CCCC2(NC(C3CC3F)=O)CCCC12 96208,c1(C(N2CC=CC(NC(COCC(C)C)=O)C2)=O)cn2ccncc2n1 96209,N1(c2nc(C)c(Br)cn2)CCC2(CC(C(=O)N(C)CC#N)C2)C1 96210,c1(OCC(=O)N(CC(C)O)CCNC(=O)CNC=O)ccc(Cl)cc1 96211,c1(C(=O)NC2C(C(N(C(CC(C)C)CO)C)=O)OCC2)ccc([N+](=O)[O-])[nH]1 96212,c1(C(=O)NC(CN2CC(C)CC(C)C2)C)nc(Cl)c(Br)cc1[N+](=O)[O-] 96213,c1(C(N2CCC(COC)C2(C)C)=O)n[nH]c2c1CN(C(=O)C(=O)C(C)(C)C)C2 96214,N#Cc1ccc(F)cc1CNC1CCN(c2ncccn2)C1 96215,CC1C(NC(=O)CC2=CCN(C)CC2)CC2CCC1N2C(C1CCCOC1C)=O 96216,C12(CNC(c3cccc(C)n3)=O)CCCCC1N(C(c1ccc(O)cc1)=O)CC2 96217,c1(C(=O)OC)cc(Cl)ccc1S(=O)(=O)Nc1ccc(CC(C)O)cc1 96218,C(N=c1[nH]c(=N)[nH]c(=NCC(CSC)N2CCN(CC)CC2)[nH]1)C1(OC)CCC1 96219,c1(OC)ccccc1CC(=O)C(=O)NCC1CCCN1C(C1CCOCC1)=O 96220,CCCS(=O)(=O)CC(=O)NC1CCC(NC(=O)CC2OCCC2(C)C)CC1 96221,C1(N(C)C(c2cc(C(C)(C)C)on2)=O)CCC(NC(=O)CCCC#N)CC1 96222,c1(C(=O)NC(CNC(c2c(C(C)C)c[nH]n2)=O)(C)C)ccc2c(c1)C(C)C(C)O2 96223,C1(CNC(CC2(CSC)CC2)=O)CC12CCN(C(c1c(C)nsc1Cl)=O)CC2 96224,CN1CCOCC1CNC(C1(NC(C2CCCOCC2)=O)CCCCC1)=O 96225,C1(C(=O)NCC(C)NC(c2cnoc2CC(C)(C)C)=O)CCCCC1O 96226,N(C(=NCCOC)NCC(Cc1ccccc1)CO)CC(CC)C 96227,c1(C(=O)NNC(=O)C2CC(O)CN2Cc2ccccc2)cc(F)cnc1Br 96228,C1(C(=O)NCC(C)NC(c2c(CCC)n[nH]c2)=O)CC12CCC1(CC1)CC2 96229,Cc1cc(C(N2CC(F)(C(N3CCCC(CC(C)C)C3)=O)C2)=O)nc(C)n1 96230,c1(C(=O)NC(CCOC)CNC(=O)C(C)NC(=O)C(C)(C)C)ccc(N)c(F)c1 96231,CC(F)(CC1CCCC1)C(=O)NCC1CCN1C(c1cc(Cl)cs1)=O 96232,N(C[Si](C)(C)C)C(C1(C(C)NC(C2CC2(C)C(F)F)=O)CC1)=O 96233,C1(CNC(C(CCN(C)C)NC(c2c(OC)nccn2)=O)=O)C2CCCCCC12 96234,C1(CC(N2CC(NC(C(C)Cc3cnn(C)c3)=O)(CO)C2)=O)CCC(=O)C1C 96235,CC(CC=Cc1ccccc1)C(=O)NCCCCC1CCCN(C(=O)CNC=O)C1 96236,N1(C(C(C)O)=O)CCN(C(=O)C=Cc2ccc(C(F)F)cc2)C(CC(C)(C)C)C1 96237,c1(N2CCC(N(C)C(C3CC4C=CC3C4)=O)C2)nccc(C#N)c1[N+](=O)[O-] 96238,C1(c2cn(CC3N(C(C(c4cn(C)nc4)O)=O)CC3)nn2)CC2C=CC1C2 96239,C1(C(=O)Nc2c(COC)nn(C)c2)N(C(C2CC=C(C)CC2)=O)CCC1(C)C 96240,N1(C(CCN(C)CC)=O)CCC2(CCN(C(=O)CC3CCCN3C)CC2)C(C)C1 96241,c1(NCCc2ccc(OC)nc2)ccc(S(=O)(=O)N2CCCC(C)C2C)c(Cl)c1 96242,c1(C(N2CCN(c3nc(C)nc(Cl)c3)CC2)=O)cc(Br)cc(Cl)c1C 96243,C1(C)(C(N2CC=CC(C(=O)NC(CCC(C)C)C)C2)=O)CCC2CC2C1 96244,c1(N(C(C2COCCN2C(=O)CC2CCOC2)=O)CCO)cccc(Br)c1 96245,N1(C(C2N3CC(C)N(CC3)C2)=O)CCCC2(CCCN2C(=O)CC2CC23CC3)C1 96246,c1(CN2C(C(=O)Nc3cncc(O)c3)CNCC2)c(F)cccc1I 96247,C1(C(=O)NC2C(NC(C3=C(C)OCC3)=O)COCC2)CN2CCN1CC2C 96248,N1(C(CCC(=O)NC)=O)CC(C)CN(C(c2cnccn2)=O)C(C)C1 96249,C(c1csc(C)n1)=CC(=O)NC(CCNC(c1n(CC)cnn1)=O)C 96250,c1(NC(C(CNC(=O)Cc2cncs2)O)=O)cnccc1C1CC1 96251,c1(C(C(=O)NCC2C(NC(C3(COCC)CC3)=O)C2)O)cc(Cl)sc1Cl 96252,c1(N(C)C)ccc(CCC(N2CC3C(CNC(=O)COCCCF)C3C2)=O)cc1 96253,N1(C(CNC(CCC)=O)=O)CC(N=[N+]=[N-])CC1C(=O)NC(c1cnn[nH]1)C 96254,C1(CCNC(c2c(CC)ccs2)=O)CN(C(C2CC(F)C(=O)N2)=O)CC1C 96255,c1(C(=O)NC2CCCN(C(c3ccc(CC)o3)=O)C2)c(C)ccc(C)c1N 96256,c1(C(=O)NC(CNC(CSCC#C)=O)CCOC)cnc2c(C)cccc2c1 96257,CC(CCNCCc1ccnc(Cl)c1F)P(C)(C)=O 96258,N1(C(C2C(CC)CCC2)=O)CC(C)(C)OC2(C1)CN(C(=O)C1=CCS(=O)(=O)C1)C2 96259,C1(C)(C(N(CC(C)O)CCNC(=O)Cc2ccno2)=O)CCC(=O)N1 96260,c1(CC)nc(CCNC(C2CC(C)N2C(c2ccnn2CCF)=O)=O)n[nH]1 96261,N1(C(=O)CCSC2CCCC2)CC2(CCN2C(c2ccccc2C(F)F)=O)C1 96262,N1(C(c2ccc(CC)nc2C)=O)CC2CC(C)N(C(C3CCN3C)=O)C2C1 96263,c1(C(=O)NC2C(NC(c3cc(Cl)cs3)=O)COCC2)ccc(F)c2c1CCC2 96264,C(=O)(CC1=CCOCC1)N1CCC(O)(C(C)NC(=O)Cc2c[nH]nc2O)C1 96265,Nc1ccc(C(=O)NCC2CCN(C(C3CC(F)C(=O)N3)=O)C2)cc1F 96266,C1(C(=O)Nc2cccc(NC(C3(C)CC3)=O)c2)SC2C=CC1CC2 96267,C(=O)(C(C)CCCC(C)=O)NCC(CC)N(C)C(c1ccnn1C(F)F)=O 96268,CC1CC=C(C(=O)NC(C2CCCC2)CNC(=O)CSC(C)(C)C)CC1 96269,Cc1ncc2cc(C(N3CCC(c4nc(C5CC5)no4)CC3)=O)c(O)nc2n1 96270,c1(COC)nn[nH]c1C(=O)N(C1(C(=O)NCCC(C)SC)CC1)C 96271,CCC(C)CCC(O)CC(=O)N1CCC(c2nnnn2C2CCCC2)(NCC)C1 96272,N1(c2snc(C(C)(C)OC)n2)CCOC(C(C)NC(C2CC(=O)N2)=O)C1 96273,c1(CC(N2C(CNC(C3OC4CCC3C4)=O)CC(F)C2)=O)nc([N+](=O)[O-])n[nH]1 96274,C1(C(=O)NCC2CC(NC(COC(CC)(C)C)=O)C2)OCC2COCCC12 96275,Cc1nc(C(C)C)nc(O)c1C(=O)NC1CCC(NC(c2cnc[nH]2)=O)C1 96276,C1(CN(C(COCCSC)=O)C)CN(C(=O)Cc2cncnc2)CCO1 96277,C1(NC(CCCN(C(=O)CCC(F)(F)F)C)=O)CC2CCC(C1)N2C 96278,C1(C2CCOCC2)(C(N2CC3(CN(C(C4CC4F)=O)C3)OCC2)=O)CCOCC1 96279,CC1CCc2onc(C(=O)N(CC(C)NC(c3ccc(Cl)cn3)=O)C)c2C1 96280,C(C(N=[N+]=[N-])C(=O)NCc1cc(C(=O)NC23CC(C(=O)OCC)(C2)C3)no1)OCC 96281,c1(CN(CCC)CCO)cncc(-c2ccc(CN(C)C)cc2)c1 96282,C=CCCC(O)CN(C(=O)C(c1ccco1)NC(c1cnc(O)o1)=O)C 96283,C#CCC(C)(C)C(=O)N1CC(C(N2CC(C(F)(F)F)C2)=O)C2(CC2)C1 96284,C1(CC=C)(NC(COCCC=C)=O)CN(C(c2cc(Br)cs2)=O)C1 96285,C(C(C)N(C)N1CCCC1C1CCCCN1C)c1cccc(C)c1 96286,O(N=c1cc[nH]cc1S(=O)(=O)NC1CC2(CCC2)C1)C1CC(C)S(=O)(=O)CC1 96287,c1(OC)ccc(F)c(C(=O)N(CCNC(C2CC(N(C)CCO)C2)=O)CC)c1F 96288,c1(NC(C)CCNC(C2CC2(F)F)=O)nnccc1C#N 96289,N1(C(CCCN(C(C)C)C)=O)CC(C)C(C)(CNC(c2ncc(CO)[nH]2)=O)C1 96290,c1(C(=O)NC2CC(NC(CCc3c(OC)cccc3)=O)C2)nc(Cl)ccc1N 96291,N1(C(=O)CCOc2cccc(Cl)c2)CC2CC(C1)N(C(=O)C(O)CC(F)F)C2 96292,N1(C(C2CC3(CC(NC(C(C(C(C)C)OC)O)=O)C3)C2)=O)CCCC2(CCCC2)C1 96293,C1(C(=O)NC2CC(C(C)C)OC2)CN(C(C2(C)CC(=O)C2)=O)CC1F 96294,C1(CC2C(C(=O)NC34CC(NC(C(C)c5ccco5)=O)(C3)C4)C2)CN2CCN1CC2 96295,Cc1nc2ccc(C(=O)NC(C)C(C(C)C)NC(=O)CC(C)C)cc2c(=O)n1C 96296,C1(C(N2CCC(C)(C(N3CC(CC(C)C)OCC3)=O)C2)=O)CC2CC(=O)C1O2 96297,O=C(NNC(=O)C12CCC1C2)C1CCC1 96298,CC(C)CCCC(C)C(=O)NCC1CN(C(c2ccc(CO)o2)=O)CCCO1 96299,N1(C(c2c(C)ccs2)=O)CC2CN(C(=O)CC3COCCN3C)CC2(C)C1 96300,c1(C(N2CCCC(C)(NC(c3cc(C(N)=O)[nH]n3)=O)C2)=O)cc(F)c(F)c(F)c1 96301,C12(NC(C3CCS3(=O)=O)=O)CCCN(C(c3cc4ccsc4s3)=O)CC1C2 96302,c1(C(N2CCC(C(C)NC(=O)C3=CSCS3)C2)=O)nc2ccccn2n1 96303,C1(NC(C2(COC)CC2)=O)CC(O)CN(C(c2c(OC)ccnc2O)=O)C1 96304,CCCC(C(=O)N1CCC1CNC(=O)C(=Cc1cccc(F)c1)F)S(N)(=O)=O 96305,C(=O)(CC(C)C(C)C)N1CC(CCCCNC(CCc2cnc(C)o2)=O)C1 96306,C(CC(C)C)(C(N)=O)NC(c1n(CC=C)nnn1)c1cnc(-c2ccccc2)s1 96307,CC(C)CC(CC(=O)NC(C(N)=O)C1CC1)NC(C1COCCC1C)=O 96308,C(=O)(CCC(=O)c1cccnc1)NCC(C)(C)CNC(c1ccsc1)=O 96309,CC(C)(C#N)C(=O)NCCCOCCCNC(C1CC(O)(c2ccccc2)C1)=O 96310,N1(C(CCCC(=C)C)=O)CC2(CCN(C(=O)C(C(C)(C)C)N(C)C)CC2)CC1C 96311,C1(F)(CNC(CSCC)=O)CCN(C(c2ccc(Oc3cccnc3)cc2)=O)C1 96312,C1(CNC(CCCN(C)C)=O)CCCCN(C(=O)CC2(C3CC3)CC2)C1 96313,N1(C(CCCN(C(C)=O)C)=O)CCOC(CNC(C2COCCN2C(C)=O)=O)C1 96314,C1(N(C(CCC(C)C)=O)C)CN(C(C2CCCN(C(N)=O)C2)=O)CCC1C 96315,c1(C(=O)NCC2(NC(=O)C=CI)CCCCC2)ccc2nc(O)[nH]c2c1 96316,c1(C(N2CCC(OC)(CNC(c3ccc(C)nc3O)=O)C2)=O)ccc(N)c(O)c1 96317,C1(NC(CCCOC(C)C)=O)CCCC(CNC(=O)CC(=O)NCC2CC2)C1 96318,C(=O)(C1CCc2c(Cl)cccc21)N1CCC(NC(c2sccc2Cl)=O)C(F)C1 96319,C(=O)(NNC(=O)C1CCS(=O)(=O)C1)N(N1CCOCC1)Cc1cnc(CC)s1 96320,N1(C(c2nccc(C)n2)=O)C2CCC1CN(C(=O)COCC1CCCO1)C2 96321,N1(C(C(CC)(C)F)=O)CC(CNC(=O)CNC(=O)CNC(C)=O)OC(C)(C)C1 96322,C1(N(C)C(C2CCC(=O)C2)=O)CCCN(C(=O)CCCN2C(=O)CNC2=O)CC1 96323,C1(CNC(C(C)(C)NC(C=COC)=O)=O)CC(C)CN(C(=O)C(C)CC(F)F)C1 96324,C1(C2CCC2)(C(=O)NCC2C(NC(c3cccc(C(F)F)n3)=O)CC2)CC1 96325,c1(C(=O)NC2CC(CCNC(C(C=C)(C)C)=O)C2)sc2cccc(F)c2c1Cl 96326,C1(Nc2ncc(C3C(CNC(N4CC(C(CC)CC)C4)=O)C3)s2)(CO)CCCC1 96327,c1(OC)ccc(F)cc1C(=O)NC1CC(C)N(C(c2ncccc2CSC)=O)C1 96328,Cc1cccc2[nH]c(C(=O)NC(C3CCCCN3C(C3OCCCO3)=O)C)cc12 96329,C1(NC(C2C=CCC2)=O)CC2CC(C1)N(c1nccc(CO)n1)C2 96330,C(c1nc2ccccc2s1)=CC(=O)OCC(c1cc(OC)c(O)cc1)=O 96331,C1(C(N(C)Cc2c(C)nn(C)c2)=O)CCN(C(=O)C(C)n2cncn2)C12CCC2 96332,N1(CC2C(C)(C)C(OC)(OC)C2(C)C)CCOc2ccccc2C1C(=O)OC 96333,Cc1nn2c(c1C(=O)NCCNC(=O)C1Cc3ccc(Cl)cc31)CCCC2C 96334,N1(C(c2ccc(OC)c(C)c2)C(=O)NC2CCCC2)CCC2(CC(=O)N(C)C2)C1 96335,c1(OC)ccc(CC(N2CCCC2CC(N2CCC(F)C2)=O)=O)c(OC)c1 96336,Cc1cc(NC(=O)CC2(NC(c3cnccc3C)=O)CCC2)c(F)c(Br)c1 96337,N1(C(c2[nH]cc(C)c2C)=O)CC(NC(=O)CC2CC2(C)C)CC1(C)C 96338,CC1CCC(C(C)(O)CNC(C2(NC(=O)Cc3cnnn3C)CCC2)=O)CC1 96339,c1(C(N2CCC(NC(c3cc(Cl)cc(F)c3F)=O)C2)=O)cccc2cc[nH]c12 96340,CC1=C(C(=O)NC(C)CN(C(=O)C(C)N(CC(F)(F)F)C)C)S(=O)(=O)CCO1 96341,C1(CN(C)C(N)=O)CCCN(C(C2CCCN2C(C2C3(CC3)C23CC3)=O)=O)C1 96342,C1(OC)CCC2(C(=O)NCC(C3CCCC3)NC(c3scnc3Cl)=O)CCC12 96343,C(=O)(C1COc2ccc(F)cc21)OCc1c2nnc(C)n2cc(Cl)c1 96344,c1(C(=O)NC(c2cccc3cc[nH]c23)c2ccccc2)nc2c(s1)CCCCC2 96345,S(=O)(=O)(c1cccnc1NCC1CCC(C2CC2)O1)N1CCCC(C=C)C1 96346,c1(C(N(C2CN(C(C3(C)CCCCO3)=O)C2)C)=O)coc(S(C)(=O)=O)c1 96347,N1(C(c2c(OC)nsc2)=O)CCN(C(=O)CC(C)N(C)C)C(c2cccnc2)C1 96348,c1(C(=O)NCCC(C)NC(C(Br)=C(C)C)=O)cccc2cccc(C)c12 96349,c1(C(C(=O)NCC2CC(NC(CSCC(N)=O)=O)C2)=O)ccc(Cl)cc1Cl 96350,C1(CC(=O)NCCOC(C)=O)C=CC(NC(=O)C=Cc2ccsc2)C1 96351,c1(CC)cc(OC)ccc1C(=O)NC1CCN(C(=O)C(C)C(C)C)C1.C(C)(=O)O 96352,C#Cc1cccc(C(=O)NCC(N2CCN(C(C3CC3C(C)(F)F)=O)CC2)=O)c1C 96353,c1nccnc1CN.c1(CN(C)C)csc(C(=O)Oc2ccccc2)n1 96354,Cc1ccc(C)c(CC(=O)NC2C3CC2N(C(C24CC(CO)(C2)OC4C)=O)C3)c1 96355,C#CCC(C(=O)NC(C1CCCC1)CNC(C1CN(C(=O)N(C)C)C1)=O)C1CC1 96356,C1(C(=O)NCC)(OC)CCN(C(=O)C(=O)NC(C)CS(=O)(=O)N(C)C)CC1 96357,C1(COC)(CNC(=O)CC(C)OC)CCN(C(=O)C(C)CC(C)C)CC1 96358,CC1(C)CC(NC(C2CC=CCO2)=O)CN1C(=O)CCC(=O)NCC1CCCC1 96359,c1(NC(C2(OC)CCCN(C(=O)OC(C)(C)C)C2)=O)ccc2ccc(O)cc2c1O 96360,c1(OC)ccc(C(N2CCCC(CNC(=O)CCc3ccoc3)C2)=O)c(Br)c1 96361,c1(CC(=O)NCCC(=O)N(c2ccccc2)C)ccncc1Cl 96362,N1(C(C23OC(C)C(C2)C3)=O)CCCN(C(c2cc(C(N)=O)ccn2)=O)CC1 96363,c1(C(=O)NC2CC(CNC(=O)COCCc3ccccc3)C2)cnn(CCF)c1 96364,CC1(C)OC(=O)CC1C(N1CCC12CN(C(c1ccc(Br)cc1)=O)C2)=O 96365,C1(C(=O)OCC)CCN(C(C2CC(NCc3ccnnc3)C2)=O)CC1 96366,c1(CC)oc(C)cc1C(N1CC2CC2(CNC(c2sc(C)cc2OC)=O)C1)=O 96367,C1(NC(c2cccn2CC(F)F)=O)CCCC1n1cc(CCn2cncn2)nn1 96368,C1(CNCC(CNC(C)=O)C)C2CC3CC(C2)CC1C3 96369,c1(C(=O)NC2(C)CC(NC(c3ccc(CO)o3)=O)C2)cnc2scnc2c1 96370,CC(CC(F)F)C(=O)NCCCOCCN(C(=O)Cc1sc(O)nc1O)C 96371,C(=O)(CCCCC(N)=O)NCC(S(C)(=O)=O)CNC(C1CC1C#N)=O 96372,Cc1cccc2ncc(C(N3CCC(C)CC3CNC(c3c[nH][nH]c3=N)=O)=O)n12 96373,C1(CNC(CC(=C)C)=O)CCC2(CO1)CC(NC(=O)C=CC1CCC1)C2 96374,N1(C(=O)OC(C)(C)C)CC(C(=O)Nc2ccc(Cc3cncs3)cc2)C2CC12 96375,CCCC(C)(CC)NC(C1(NC(=O)CNC(=O)CC(C)C)CCN(C)C1)=O 96376,C(C(F)(C(=O)NCC1CN(C(N)=O)C1)C(C)C)NC(C(CC)(C)C#N)=O 96377,C(=O)(C1CCCc2c[nH]nc21)N1CC(CCC)C(CNC(=O)C(C)C(C)(C)C)C1 96378,Cn1nc(C(=O)NC2CC3(CCCN(c4nnnn4C)C3)C2)c2cc(F)ccc12 96379,C1(NC(=O)C=Cc2cnc[nH]2)CC2(C1)CC(C(=O)NCC1CCC(F)(F)C1)C2 96380,c1(C(=O)NCC(CNC(c2c(CC)nc(C)[nH]2)=O)F)cc(O)cc(F)c1 96381,c1(CCCNC(C2C(OC)CCCCC2)=O)cn(C)[nH]c1=NC(=O)OC(C)(C)C 96382,N1(C(C2CCN(C(=O)COc3ccccc3)C2)=O)CC2COC(=O)C2C1 96383,N1(C(=O)C2=CCCSC2)CCC(C2CC2)C1CNC(C1(C2CCOCC2)CC1)=O 96384,N1(C(c2noc(CC)c2C)=O)Cc2occ(C(=O)NCCC3CC(F)(F)C3)c2C1 96385,Cc1cc(F)c2nc(O)cc(C(=O)NC3CCCN(CC(F)F)C3)c2c1 96386,c1(C(=O)NC2C(F)CCN(C(CCC(C)=O)=O)C2)ccc(Cl)c(C)c1F 96387,C(=O)(NN1CCCN(C)CC1)NC(c1c(C)ccnc1)C1CCC1 96388,c1(C(=O)NC2CC(C)N(C(=O)COCC3CCCOC3)C2)csc2nccn12 96389,c1(C(=O)NC2CC(NC(C3CCCOC3)=O)C(O)C2)cnc2c(F)cccn12 96390,N1(C(Cc2cc(CC)no2)=O)CCC(C2CC2)C1CNC(=O)C(=O)NCC(F)F 96391,c1(C(N2CCCCC(C(N3CC(CC)N(C)CC3)=O)C2)=O)cccc2[nH]ncc12 96392,C1(NC(NNC(=O)Cc2ccccn2)=O)C2CC3CC1CC(O)(C3)C2 96393,C1(NC(C(C)CO)=O)CC2C(NC(C3CC=CCC3C)=O)C2C1 96394,C(C(C)(C)C(=O)N1CCC(C)C1)NC(C1(CC(=O)OCC)CC1)=O 96395,c1(CC2CCCN2CC=CCNC(C2N(CC)C(=O)CC2)=O)cccc([N+](=O)[O-])c1 96396,c1(C(=O)NCC2CN(C(CC(C)NC(N)=O)=O)CC2O)onc2c1CCCC2 96397,c1(NC(C2C(NC(c3ccccn3)=O)C2)=O)ncc(F)cc1Br 96398,N1(C(CCC=C)=O)CCn2cc(C(N3CCC4(CCCO4)C3)=O)nc2C1 96399,N1(C(=O)NCc2nc(C3OCCO3)cs2)CCOc2c(F)cccc21 96400,N1(C(CN(C(C(C)Cc2ccccc2)=O)CO)=O)CCN(C2CCNC2=O)CC1 96401,C1(O)(CCNC(C(=O)NC(C)C)=O)CN(C(=O)C(C)CC2CCCCC2)C1 96402,N1(C(c2c(Cl)cnc(C)n2)=O)CC2(CCC2)CC1CNC(=O)CCc1ccon1 96403,C1(NC(c2cnccn2)=O)CCC2(CC1)CN(C(c1ccoc1Cl)=O)CCO2 96404,c1(CNC(Cn2cc(C3(C)CC(OC)(OC)C3)nn2)=O)ccc2nsnc2c1 96405,n1(CC(=O)N(CCCNC(C2C(COC)CC2)=O)C)ncccc1=O 96406,C1(SC)CN(C(=O)Cn2cnc(=N)[nH]2)CC1NC(C1(C)CCCO1)=O 96407,C12(CNC(CSCC=C)=O)CC1CN(C(c1cc(C3CC3)nn1CC)=O)C2 96408,N1(C(C2CCC(OCC)CC2)C(=O)NC2COC2)CC2C3C=CC(C3)C2C1 96409,C#CCCCC(=O)NCCN(C(=O)CNC(=O)COCC=C)C(C)C 96410,C1(NC(c2n(C(C)(C)C)ncc2)=O)CCC2CC1CN2C(C1(C)CCOCC1)=O 96411,c1(C(N2C(CNC(=O)C=C(Cl)Cl)CC3(CC3)C2)=O)cc(O)nc2cnccc12 96412,C(=O)(CC(O)C(Cl)(Cl)Cl)NC(c1cnn(C)c1)C(=O)N(CC)CC 96413,C1(CC(=O)NCCCCCCN(C(=O)C=Cc2cnccn2)C)CCC(=O)NC1=O 96414,O=C1CN(C(=O)CCc2nc(O)n[nH]2)C(C(=O)NC2CCC3(CC3)C2)CN1 96415,C(=O)(C1CSc2ccccc21)NC1C(NC(c2cccc(S(C)=O)c2)=O)CCC1 96416,C1(C(=O)OC)(OC)CN(S(=O)(=O)CCc2ccsc2)C1 96417,c1(OC)ccc(F)c(C(=O)NC2CC2CNC(=O)CCOC(C)CC(C)C)c1Cl 96418,C1(C(=O)OC)CCC(CC(=O)NCCCNC(c2cccn2C)=O)CC1 96419,CC1(C(=O)NCCC2(O)CCN(C(=O)CC3CSC3)C2)CCC(F)(F)CC1 96420,C1(C)(CC(=O)NC2(CC(=O)NC3CC(OC)C3)CCC2)CCCCC1 96421,C1(C(=O)NCCCCC(C)NC(CN(CCOC)C)=O)CCC2(CC1)CC2(F)F 96422,c1(-n2cc(C(C)N(C)C)nn2)ccccc1C(=O)N(C(C)CCO)C 96423,CCC(C(=O)OC)C(=O)N1CCCCC1CCNC(=O)CSc1n[nH]c(C)n1 96424,C(C)(c1ccc(F)cc1F)=CC(=O)NCCN(C(=O)CC1CCN(C)C1=O)CC 96425,C#CCCCCC(=O)NCc1ccc(C(=O)NC(CCC)C(F)(F)F)nc1 96426,C12(C(N3CC(C)C(CCNC(C4CCCO4)=O)C3)=O)CCC(CC1)OC2 96427,C1(OC)CC(C(C2(n3cc(CO)nn3)CC2)=O)N(C(=O)CCc2cn[nH]c2)C1 96428,c1(OC)cc(F)c(Br)cc1S(=O)(=O)Nc1cc(C)ccc1S(N)(=O)=O 96429,N1(C(C2CC(C)=C(C)CC2)=O)CCC(C)(C)CC1C(=O)NCc1ccnc(O)c1 96430,C1(NC(C)=O)CC(NC(c2ccc(OC(F)F)cn2)=O)C1(C)C 96431,c1(C(=O)NC2C(NC(C3(C#N)CCCO3)=O)COC2)cc2ccncc2s1 96432,S(=O)(=O)(CCCCF)NC1CCCN(C(=O)Nc2ccc(F)cc2)C1 96433,CC#CCC(C(=O)NC1CC1)NC(=O)OC(C)(C)C.C(C)(C)(CCCO)N 96434,c1(NC(=O)NCc2ccc3nonc3c2)cc2cccnc2c(Br)n1 96435,N1(C(C2CC3CC2C2CC32)=O)CC2CCC1CN2C(C1CCCS1)=O 96436,C1(C(N(CCO)CC)=O)C2CCCC2CN1C(c1cnn2cccc2c1)=O 96437,N1(CCC(=O)NC(CC(C)NC(Cc2ccn(CC)n2)=O)C)CCN(C)CC1 96438,N1(C(c2n(CC)ncc2Cl)=O)CCC(C2CCN(C(=O)C=C3CC3)C2)C1 96439,Cc1coc(C(C)C)c1C(=O)NCC1CN(C(=O)C(C)OCCC(C)C)CCO1 96440,N1(C(C2C(OC)CC2)=O)C2CCC1C(F)C(NC(=O)Cc1cnccn1)C2 96441,CC1C(=O)CCC(C(=O)NC2(CF)CCN(C(c3cscn3)=O)C2)C1(C)C 96442,c1(CNC(c2cc(F)ccc2F)=O)ccc2c(c1)OCO2 96443,CC1(C)CN(C(=O)CCn2cccn2)CC1NC(C1CCCC(C(F)(F)F)C1)=O 96444,Cc1ccc(C(=O)NCC(c2ccccc2)NC(=O)C(F)C2CCC2)c(F)c1F 96445,c1(C(C)CNC(=O)NCc2sncc2Br)cccc(C(F)(F)F)c1 96446,C(c1cnc[nH]1)=CC(=O)NCC(c1ccccc1)CNC(C12CC(CO1)C2)=O 96447,C(C(C)C(=O)NC1CCC1NC(=O)C(C)(C)C)OCC 96448,N1(C(C2CN(C(N)=O)C2)=O)CC(O)(CNC(=O)COC2CCOC2)C1 96449,Cc1ccc(C)n1-c1cn(C(C)C(=O)NC(c2ccc(F)cc2)CF)nn1 96450,c1(C(=O)NC(CC(C)C)CNC(C2CC2C#N)=O)c[nH]c2c(F)cccc12 96451,N1(C(CC=CCNC(=O)Cc2cccc(O)c2)=O)Cc2cccnc2C1 96452,N1(CC(=O)NCC(CNC(CC(C)CN(C)C)=O)(C)C)CCn2nccc21 96453,C#CCCCC(=O)NC1CCC(CCNC(c2ccc(Cl)cc2)=O)C1 96454,c1(OCC)cc(C(=O)N(C2CCN(C(=O)C=CCF)C2)CCO)ncn1 96455,C1(NC(C(CC)N(C)C)=O)CN(C(c2nc(C)c(C)s2)=O)CC(F)(F)C1 96456,C1(OC)CC(NC(=O)CN2CCP(C)(=O)CC2)CN(C(C2CSCCS2)=O)C1 96457,C(=O)(C1CCc2cc(Cl)ccc21)NC1C2CN(C(COC(CC)C)=O)C1C2 96458,CS(=O)(=O)C(CNC(=O)Cc1cc[nH]c1)CNC(C1(F)CCOC1)=O 96459,O=C(CCCOc1cccnc1)NCC1CN(C(c2csc(CO)n2)=O)C1.CCO 96460,c1(C(=O)NCC(CNC(c2c(C)ccn2C)=O)C)cccc2[nH]cc(Cl)c12 96461,CC1(C)CC(CC(=O)NCC(=C2CN(C(C3(C4CC4)CC3)=O)C2)F)CO1 96462,Cc1cc(C(=O)NCCC2CCC(NC(c3ccc(Cl)c(F)c3)=O)C2)cc(O)n1 96463,N1(C(Cn2c(C)cnc2)=O)CCN(C(=O)CCCCC#N)CC1C 96464,C1(CNC(C2C(CC)OCC2)=O)C2CN(C(c3c(N)cnn3C)=O)CC12 96465,c1(C(=O)NCCCN(C(C2CC(C(C)C)OCC2)=O)C)c(F)cc(O)cc1F 96466,C(=O)(C(C)(C)CN(C)C)NC1C=CC(CC(=O)N(CC(CC)(C)OC)C)C1 96467,N1(C(c2csnn2)C)CCC(C2(NC(=O)CCC(C)(C)C)CC2)CC1 96468,C1(C(N(CCCOCCNC(c2ccc(C)cc2)=O)C)=O)CCC2(CCC2)C1 96469,n1(C)[nH]cc(C(=O)OC)c1=N.C1(COCC)CC(NC(=O)C=CC(=O)OC)CCO1 96470,C1(CC2CC(C)CN2)CN(C(=O)C2=C(Cl)CCC2)CCN1C.N12CCNCC1C2 96471,C12(CNC(COCC)=O)CC1CN(C(=O)Cn1cc(I)cn1)C2 96472,Cn1cnc2c(N(CCCC3CC3)CCO)[nH]c(=NCc3cc(C(N)=O)co3)nc12 96473,C(=O)(C(C)CC(F)(F)F)N1CC(C)(C(=O)NCCCc2cc(C)no2)C(C)C1 96474,CC1(C)CC(C(N2CC3CCC3(CNC(=O)CSc3cn[nH]c3)C2)=O)C(C)(C)O1 96475,CCCC(C)CC(=O)NC(C)(C)CNC(C1SCCS1)=O 96476,N1(C(C(C(CC)CC)C)=O)CC(CNC(c2csc(C)n2)=O)OC2(CCC2)C1 96477,C1(C(=O)NC(C(C)C)CNC(C2(S(N)(=O)=O)CCC2)=O)CC2(CCCCC2)CO1 96478,n1(C(C)(C)C)cnc(C(N2CC(O)(CCNC(=O)C(F)=C3CCCC3)C2)=O)c1 96479,c1(-c2nc(Cc3cc(C)nc(C)n3)nn2CCCN(C)C)nc2nc(C)ccn2n1 96480,N1(C(CN(CCCCC)C)=O)CC(NC(=O)COCCCCC)CCC1C 96481,C1(CNC(CCC=CC)=O)CCCN(C(c2cn(C)nc2C(F)(F)F)=O)C1 96482,N1(C(c2cc(COC)sc2)=O)CC2CC1CN2C(=O)CC1CC2(CC2)C1 96483,CC1CCc2[nH]c(C(=O)NCCNC(C3(CCO)CC3)=O)cc2C1 96484,C(C(=O)N(OC)C(C)CC)C12C(CN(C(c3cncc(C=C)c3)=O)C1)CC2 96485,C1(CNC(C2(CC#C)CC2)=O)(OC)CCN(C(c2ccc(CC)cc2O)=O)CC1 96486,c1(C(CC)NC(=O)COC(C)(C)CNC(c2cc(C)no2)=O)ccccn1 96487,c1(C(N2C(CNC(C(C)(C)CF)=O)CC2)=O)ccc(Cl)c2ccccc12 96488,C(=O)(C(C(C)C)c1cnc(C)s1)NC(CC(C)NC(C=CC)=O)C 96489,Cc1c[nH]cc(C(=O)NC23CC2CN(C(=O)C(F)C(C)C)C3)c1=O 96490,c1(SC)c(C(=O)N(C)CCN(C(C2CC2C2CCC2)=O)C(C)C)cccc1F 96491,CC1(C)C(CO)CN1C(=O)C(C1(O)CCC1)NC(=O)C(O)CN1CCCC1 96492,CCCCC(C(=O)NC1(C(=O)OC)CCC1)NC(C1CC1C(N)=O)=O 96493,N1(C(CCCC(C)=O)=O)CCCC2(C1)C(NC(c1ccc(CO)o1)=O)CCN2C 96494,CCCCN=C(NCc1cc(Br)ccc1Cl)N(C)Cc1cc(C)on1 96495,c1(C(N2CC3C(CNC(c4cc(CC)nn4C)=O)C3C2)=O)cc2ccccc2o1 96496,CC(C)CC(C)(CNC(C1CC(CCO)C1)=O)NC(=O)CN1CCCCCC1 96497,C1(C(N(CC(=C)C)CC)=O)CC(CNC(=O)CCc2cn[nH]c2)C1 96498,N1(C(C=CC(=O)OC(C)(C)C)=O)CCN(C(=O)C2=CCCS2)C(CCO)C1 96499,c1(C(=O)NC(CNc2nccc(OCC)n2)C2CC2)[nH]c2ccc(F)cc2c1C 96500,c1(NC(CC(=O)NCC2CC2CNC(C2(F)CCC2)=O)=O)ccccc1O 96501,C1(NC(C(CCF)NC(C=CC(=O)N(C)C)=O)=O)CCCCC12CC2 96502,C#CCC(CC#C)C(=O)NC(C)(CC)CCNC(c1ccc(Br)c(C)n1)=O 96503,C(CCC(=O)NC(CNC(C1(NC(c2ccccc2)=O)CC1)=O)CO)OCC 96504,CCCC(C)(C)C(=O)N1CC2CCCC2C1.c12ccccc1C(=O)N1CCCC21 96505,C(=O)(C(O)C(C(C)C)OC)N1C(C(=O)NC2CCN(C(CC)=O)C2)CC(F)(F)C1 96506,C(CO)(C(C)(C)CO)NC(C(C)CNC(=O)CCn1cccc1)=O 96507,N1(C(=O)CSc2nncs2)CCCC(NC(C2CC2(F)F)=O)CC1 96508,C1(C(=O)NCCCC(CCC)NC(=O)C(=O)NCC)COC2COCC2O1 96509,c1(C(C(CO)NC(c2ccc(OCCO)cc2)=O)O)c(F)ccc(Cl)c1F 96510,C1(C(=O)Nc2ccc(C)c(C)c2)(COC)CCN(C(=O)CC2CNC(=O)O2)CC1 96511,C1(CC(=O)NC2C=CCN(C(c3c(C#N)scc3)=O)C2)CCn2cncc2C1 96512,C1(F)(C(=O)NCC2C3CN(C(c4cc(C)n(C)n4)=O)CC32)CCN(C)CC1 96513,c1(C(=O)NCC2N(C(CC(C=C)C)=O)CC(F)C2)c[nH]c2cc(C)ccc12 96514,N1(C(CC2CC(=O)NC2=O)=O)CC(NC(=O)COCCCN(C)C)C2CCCC12 96515,c1(C2CCN(C(=O)NCCC(=O)N(C)C)C2)cc2ccccc2[nH]1 96516,c1(OC)ncc(Br)cc1C(=O)NCC1(C)CN(Cc2csc(C)n2)C1 96517,Cc1ccccc1CCNC(=O)CCN(CCCO)C(=O)CC1CC2CC2C1 96518,C1(NC(C(CC)N(C)C)=O)CCN(CCC2CCOCC2)CC1O 96519,c1(COC)nc(NC(CNC(=O)C(C)C(C)COC)C2CC2)cc(O)n1 96520,c1(NCC(C2CCC2)OCC)ncccc1S(=O)(=O)N1CCC(C(F)F)C1 96521,C12(NC(CS(=O)(=O)NC)=O)CCCCCC1N(C(=O)CCc1ccc(C)o1)CC2 96522,C1(C(=O)NCC2C(C)CCN2C(c2cc(C(F)F)nn2C)=O)CNC(=O)CC1C 96523,C1(CNC(=O)NC2CCOC2=O)CCN(Cc2ccc(CCO)cc2)CC1 96524,c1(CN(C)C)ccc(S(=O)(=O)NC(c2ccccn2)CNCCS(C)(=O)=O)cc1Br 96525,C(C(C)(F)C(C)(C)F)NC(CC1CC(C)N(C(=O)CCNC(=O)CO)C1)=O 96526,CC1CC(NC(C2CC(F)(F)C2)=O)CCN1C(c1cc(CO)ccn1)=O 96527,N1(c2ncnc(OC)c2C)CC2CN(c3c(OC)cccc3)CC2C1 96528,N1(C(=O)NC2C(C)NCCC2)CCOC2(CCS(=O)(=O)C2)C1 96529,CCC(C)(CNC(=O)C(C1CCCCC1)C)C(=O)NCC1COCCN1C 96530,c1(C(N2C(CNC(CC=C)=O)CC2)=O)cn(CC(c2ccccc2)O)nn1 96531,C1(CNC(Cc2cc(C)sc2)=O)(NC(=O)CC2CCCN(C)C2)CCN(C)C1 96532,c1(C(N(CC(C)O)CCC(C(=O)NC(C)C)=O)=O)cnc(-c2ccccc2)[nH]1 96533,C1(C(C)(F)F)CCCCN1C(=S)Nc1ccc([N+](=O)[O-])cc1 96534,c1(C(=O)NCCC(C)N(C(CC(CC)O)=O)C)[nH]nc2ncnc(O)c12 96535,N1(C(COCCOC)=O)CCCCC1CC(=O)NC(C)C 96536,N1(Cc2ccc(C)nc2C)CCn2cnc(-c3cc(F)cc(F)c3F)c2C1 96537,CC(CC(=O)N1CCCCC1C1(NC(=O)C(=Cc2c[nH]cn2)F)CC1)C(C)(C)C 96538,c1(N2CCC(C)C(F)(F)CC2)nc(=NCC2COCC2(C)C)[nH]c2c1CCCC2 96539,C(Cc1ccoc1)(C(=O)NCc1ccns1)NC(CSC)=O 96540,CC(C)CC(=O)NC(c1ccnn1C)C(=O)NC(C)CC(N)=O 96541,NC(=O)CC(O)C(=O)N1CCC(CO)(NC(C2CCCCC(=O)N2)=O)C1 96542,CC1CCn2ncc(C(N3CCC(C)C(CNC(=O)C(C)(F)F)C3)=O)c2C1 96543,C(=O)(C(F)(F)C1(O)CCC1)N(CC(CN(C(C(N1CC(C)C1)C)=O)C)O)C 96544,c1(C(=O)NCC(=C2CN(C(C3COCCO3)=O)C2)F)cnc2[nH]cnc2c1 96545,C=Cc1ccc(C(=O)NC2(C(=O)NC(C)Cn3cccn3)CC(F)C2)cc1 96546,N1(C(CC(CC)C)=O)CC2CC(NC(=O)CC3CC(F)(F)C3)CC2C1 96547,c1(C(N(C(COC)(C)COC)C)=O)cc(Cl)c(Br)c(Cl)c1.C(C)(C)(C)O 96548,C(N=c1nc2c(ncn2C)c(N(C)CCOC)[nH]1)C1CC(OC)C1(C)C 96549,N1(C(CC2C(C)OC(C)C2)=O)CC2(CCCCN(C(c3cn[nH]c3)=O)C2)C1 96550,c1(N2C(CNC(c3cc4ncc(C)n4cc3)=O)CC2)cc(C)c([N+](=O)[O-])cc1Br 96551,CC(CN=c1[nH]c(N2CCC(Cn3cccn3)C2)nc2ccc(Cl)cc12)C(N)=O 96552,c1(C(N(CC(CNC(C2(CC)CCNC2=O)=O)O)C)=O)ccc2ncncc2c1 96553,c1(CN(CCC)C(=O)NC2(CC(F)F)CCCO2)c(C)noc1C 96554,c1(CCC)c(C(N2CC(NC(C3CN(C(C)=O)CCO3)=O)C(C)C2)=O)cnn1C 96555,Cc1cnc2ccc(C(N3CCC(C)C(CNC(C4(CCF)CC4)=O)C3)=O)cn12 96556,C1(NC(CCN(C)CC)=O)CN(C(=O)CCC=CC(C)C)C2(CCOC2)C1 96557,N1(C(c2c(C)n(C)nc2)=O)CCC2(CC1)CC(NC(=O)C1CCc3nccn31)C2 96558,C(=O)(C#CC1CCOCC1)N1CC(OC)C(CC2CC2)C1.C12(CCC1)C(=O)N2 96559,C1(NC(CC(C)=C(C)C)=O)CC2CN(C(=O)CCn3cnc(=N)[nH]3)CC2C1 96560,N#Cc1ccc(Cl)c(C(N2CCC(OCCCNC(C3CCCS3)=O)CC2)=O)c1 96561,Cc1[nH]cc(C(=O)NCC23CC2CN(C(c2cc(C(C)C)on2)=O)C3)c(=O)c1Cl 96562,C12(C(N3CC4C(C(=O)OC)C4C3)=O)CC(CO1)N(C(c1cc(C)cs1)=O)C2 96563,Cc1ccc(C(C)(C)C(=O)NCC2(c3ccc(Cl)cc3)CC2(C)C)cn1 96564,CC1CCCCN1CC(=O)NC(CC1CCCC1)C(=O)N1CC(C)(C(F)(F)F)C1 96565,C(CN=c1nc(Cl)[nH]c(C)c1C#N)N(C(c1ccc(OC)cn1)=O)C 96566,N1(C(c2c(C)cn(C)c2)=O)CCCCC12CC(NC(C1CCCCS1)=O)C2 96567,Cc1cn2cc(C(=O)NCC3CN(C(C4OCCC4C(C)C)=O)C3)sc2n1 96568,C(=O)(C(C)(C)CC(=O)NC1CCCC1(C)CN(C(=O)C(C(C)C)SC)C)OC 96569,CCC(CC)(CO)C(=O)NCCOC(C)(C)CNC(c1cn(C)ccc1=O)=O 96570,C1(CC)COC(C)CN1C(c1cc(CNC(C2CCS(=O)CC2)=O)on1)=O 96571,c1(Cc2scc(C(=O)NC(CN(C3CCS3(=O)=O)CC)(C)C)n2)ccccc1F 96572,N1(C(C(=O)NCCOCC)C2CCSC2)CCCC(C(=O)OC)C1C 96573,c1(C(=O)Nc2ncc(C#N)s2)cnc2[nH]nc(-c3ccc4c(c3)CCO4)c2c1 96574,N1(C(C=C(CC)CC)=O)CC2CCCN(C(=O)CCc3c(C)nn(C)c3C)C2C1 96575,N1(C(C2(C=C)CCN(C(=O)CC(=O)OC)C2)=O)CCc2nc(O)[nH]c2C1 96576,C(=O)(C1=CCCOC1)N1C(CCNC(C2CC2(Cl)Cl)=O)CSCC1 96577,C1(C(=O)OCC(c2ccccc2)=O)CCCCC12CCC2 96578,c1(NC(C2CCC3(CN(C(CSC)=O)C3)O2)=O)cc(F)cc2[nH]ccc12 96579,N1(C(C2=CC(C)(C)C2)=O)CCN(C(=O)CCCCN2CCCCC2)C2COCC12 96580,Cc1cc(=NCC2(C)CCCCCCC2)[nH]c(=NCCN2C(C)CCCC2C)[nH]1 96581,c1(-c2cn(C3CCN(C(C4CCN(CC(C)C)C4)=O)C3)nn2)cc(F)ccc1F 96582,CN1CCC(C(=O)NCCCN2CCN(C(C3(C)CC3(F)F)=O)CC2)C1=O 96583,C1(NC(Cc2ccc(OCC)cc2)=O)CC(C)CN(C(c2cscc2C#N)=O)C1 96584,C1(C(N2CCC(C3C(NC(=O)C(F)F)CCCO3)CC2)=O)COCC2(CCC2)O1 96585,N1(C(C(C)NC(=O)NC)=O)CCC(CNC(c2ccc(C(N)=O)cc2)=O)C(C)C1 96586,C1(C(=O)NCC2CCN(C(C(F)(F)SC)=O)C2)CCCN(C(=O)N(C)C)C1 96587,c1(CC(=O)NC(CC)CN(C(=O)CSC(F)(F)F)C2CC2)cccc2c1OCO2 96588,C(=O)(C1=CCCC1C)NC1CCC(C(=O)NCC2CC(C(=O)OC)C2)C1 96589,c1(C(N2CCC(CCNC(C=COCC)=O)CC2)=O)oc2c(c1C)C(=O)CCC2 96590,n1(CCOCC=C)c(N2CCC(C)(C(=O)OC)C2)nnc1CO 96591,C1(C(=O)Nc2ccccc2)(NC(=O)NCC2C(=C)C2)CCOCC1 96592,c1(NC(C2(N(C(CSC(C)C)=O)C)CC2)=O)cnn(C2CCC2)c1 96593,c1(C(C(=O)NCC)N(Cc2nnc(C)o2)CC2CC2)cc(Br)c(OC)cn1 96594,C1(CNC(CC(C)C2CC2)=O)CCCCN(C(C2CCCC(O)C2)=O)C1 96595,N1(C(CCCN(C(C)C)C)=O)CC(C)(C)CC1CNC(c1[nH]nnc1C1CC1)=O 96596,N1(C(c2c(C#C)c[nH]n2)=O)CC(C)CCC1CNC(=O)CCOC(C)=O 96597,N1(N2CCCC(C(=O)NCCNC(=O)C(C)C)C2)CCC(C)CC1.C(=O)OC 96598,c1(C(N2CCC3(NC(Cc4c(C)noc4C)=O)C(C2)C3)=O)ccc2nn[nH]c2n1 96599,c1(CC(=O)NC2CCCCC2NC(C2CC3C=CC2C3)=O)cccnc1Br 96600,C1(OC)CC2CC(C(=O)Nc3cccc(CNC(=O)C=CCF)c3)CC12 96601,c1(C(=O)NC2CN(CC)C2)n[nH]c2cc(-c3ccn(C4CC4)n3)ccc12 96602,c1(-c2ccc(C(=O)NCCC3(OC)CN(C(C=NOC)=O)C3)s2)cccc(F)c1 96603,Cc1ccc2c(Nc3ccc(CCC(N4CCC(F)CC4)=O)[nH]3)ncnc2c1 96604,C(c1cccnc1)=CC(=O)NC(C)CNC(c1cnc(C2(C)OCCO2)s1)=O 96605,C(=O)(C1=CC2CCC1C2)N1CCN(C)C(CNC(C23CCC(CC2)CC3)=O)C1 96606,c1(CCn2c(CC(C)NC)nc(C3CCC(C)CC3)n2)cccc2ccccc12 96607,c1(CNC(C(=O)NCc2cc(C(F)F)cc(F)c2)=O)cccc2c1OC(F)(F)O2 96608,n1(CCC)cc(C(=O)NCC2C=CC(NC(=O)C(C)SCC)C2)c(C)n1 96609,C1(C(=O)NCC2CCCC(NC(c3ccncc3F)=O)C2)(SC)CC(F)(F)C1 96610,CCCC(CCC)CC(=O)NC(C)(CO)C(=O)NCC(O)C1(Cl)CC1 96611,CP(C)(=O)CCC(=O)N1CCCCC(CCC(=O)NC2CC3(CCC3)C2O)C1 96612,CCC(C)(F)C(=O)N(CCNC(=O)COCCOC)CCOC.c1ccncc1 96613,N1(C(CSCC(C)C)=O)CCC(CC(=O)N(C2CCC2)CC2CC2)C1(C)C 96614,c1(CCC(=O)NC2C(CNC(Cc3cc(C)sc3)=O)C2)cnc2ccccc2c1 96615,N1(C(C2(COC)CC2)=O)CCOCC(C(=O)Nc2c(C(N)=O)cccc2C)C1 96616,C(=O)(C1CC(=O)Nc2ncn(C)c21)N1C(C)CN(C(C2CCSCC2)=O)CC1 96617,c1(C(=O)NC2C(C)N(C(c3cnc(C4CC4)nc3O)=O)CC2)cc(Cl)cc(Cl)c1 96618,C1(C(c2cn(C(C(N3CCC(N(C)C)C3)=O)(C)C)nn2)N(C)C)CCNC(=O)C1 96619,c1(COC)ncc(C(N2CCCC2CNC(=O)C(C)S(N)(=O)=O)=O)c(O)n1 96620,c1(CC)ccc(C(N2CCC(C(=O)NCC3CCC(F)(F)C3)C2)=O)cc1 96621,N1(C(CN(C(C)=O)C)=O)CCCCC(CNc2ncc(C)c(C)n2)C1 96622,C(=O)(C1OCCn2ccnc21)NCCCN(C(C(CC)(C)O)=O)C 96623,C(c1ccc(F)c(F)c1)=C(C)C(=O)N(C)CC1CN(C(=O)C=CC(C)C)CCO1 96624,c1(C(N2CC(NC(c3cc(OC)ns3)=O)CC2(C)C)=O)cc2cc(Cl)cnc2[nH]1 96625,CS(=O)(=O)c1cc(C(N2CCN(C(=O)C=CC3CCCO3)C(CCO)C2)=O)cs1 96626,c1(C(=O)NCC2(CNC(C3C(CC)C3)=O)CCCC2)ccc(P(C)(C)=O)nc1 96627,N1(C(CCC(C)=O)=O)CC2CC(C1)N(C(c1cccc(C3CC3)c1)=O)C2 96628,c1(C(N2CC(C)C(NC(c3ccc(CC4CC4)s3)=O)C2)=O)coc2c1CSC2 96629,N1(C(C)C)CCCCC1C(=O)N(C)CCOCCC(=O)NC1(c2cccs2)CC1 96630,C=CC(C)(CCOC)C(=O)NCC(C)C(F)C(=O)N1CC(C)=C(C)C1 96631,c1(C(=O)OCCSCC)ncsc1CC 96632,c1(N2CC=CC(NC(CNC(CC)=O)=O)C2)cc(C)ncc1C#N 96633,C12(C(=O)NCC(CNC(=O)CN3CCCC3=O)F)CC(C1)C(C(F)(F)F)O2 96634,c1(C(N2CCCCC(NC(C(CC=C)(C)C)=O)CC2)=O)cnn2c1CC(C)CC2 96635,C#CCCCC(=O)NC1(CCNC(c2cc(C(F)(F)F)n[nH]2)=O)CC1 96636,CCC(C(=O)NC(c1ccccc1)C(=O)Nc1ccsc1)NC(C)=O 96637,C1(CNC(C2(CC)CCCC2)=O)CCN(C(C23CCC(CC2O)C3)=O)CC1(F)F 96638,c1(OC)cc(CC(=O)N(C)CC2CN(C(C3CC34CC4)=O)CC23CC3)ccc1C 96639,c1(C(=O)NC2C(NC(C(C)O)=O)C2)cc2ncccc2[nH]1 96640,C(=O)(C(CC1CC1)c1ccccc1)N(CC(C)NC(=O)C(C)(C)NS(C)(=O)=O)C 96641,C(=O)(CC1OCc2ccccc21)N(CC(C)NC(CCC(=C)Br)=O)C 96642,C1(C(=O)NCC2(C)CCN(C(C)=O)C2)CC2(CCOCC2)CN1 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96661,CCS(=O)(=O)CC(C)NC(=O)C(N1CCCC(C(F)(F)F)CC1)=O 96662,C1(CC(=O)N(C(C)C)CCN(C(=O)C=Cc2ccco2)C)CC2(CCC2)CCO1 96663,c1(C(N2CCC(COC)(NC(=O)C(C)n3cnnn3)C2)=O)c2c(nn1C)CCC2 96664,c1(C(N(CC(CNC(CC2C(CC)C2)=O)(C)C)CC)=O)cc(=O)cc[nH]1 96665,c1(OC)cccc(CCNC(=O)NCCC(O)COC)n1 96666,Cc1noc(C(=O)NCCC(C)N(C(=O)C(C)Cc2c(C)n[nH]c2C)C)c1C 96667,c1(OCC(=O)NC2(CCCNC(C3(CO)CC3(F)F)=O)CC2)cccnc1 96668,N1(C(CC2(OCC)CCC2)=O)CCOC(CNC(c2nnc(S)n2C)=O)C1 96669,C12(C(N3CC(Cn4cc(C(CC)O)nn4)OCC3)=O)CCCCC(=O)N1CCC2 96670,c1(OC)cc(C(F)F)ccc1CNc1ccc(-c2nncs2)cc1 96671,C1(C(=O)NC(C(=O)NCCSC(F)F)C2CCCC2)CCC(O)C1 96672,C1(CF)(CNC(c2sccc2Cl)c2nnnn2CCN2CCOCC2)CCCO1 96673,C1(C(=O)NCCC(=O)OCCCC)CCCN(C(C2(C)CCOC2)=O)C1 96674,c1(COCCCNC(=O)NC(C)CN(C)CC2CCNCC2O)ccccc1Br 96675,CCCCCC(C)(CC)C(=O)N1CC2(CCC2NC(=O)CSC(F)(F)F)C1 96676,n1(Cc2ccc(OC)cc2)[nH]nnc1=NCC(CSC)SC 96677,N1(C(CC)C(=O)NCC(C)NC(=O)Cn2cnnn2)CCN(C(C)C)CC1 96678,C1(C(N2C(CNC(c3cc(F)ccc3Cl)=O)CCC2)=O)CCn2c(O)nnc2C1 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96748,c1(C(N2C(CNC(CC(=O)NCC)=O)CC(OC)C2)=O)cc2c(=O)[nH]ccn2n1 96749,c1(C(C(=O)NC(CNC(CC(C)F)=O)(C)C)C)nc(F)ccc1Cl 96750,C1(C(=O)NCCCOC=C)C2CCCC2CN1C(=O)CN1CCCCC1=O 96751,N1(CC(=O)N(C(C)CNC(=O)CN(C2CCCC2)C)CC)CCC(C)C1 96752,c1(OC(C2C3CC(N)C(C3)C2)=O)c(Br)cc(Br)c2cccnc12 96753,Cc1cc(C(F)(F)F)nn1CC(=O)NC1CCCCC1NC(c1ccc[nH]1)=O 96754,N1(C(CCCOCC)=O)CC2(CCN(C(=O)C(C)CCO)CC2)C1C(C)C 96755,CC1=C(C(=O)N2CC(NC(c3ccsc3CN)=O)C(C)C2)CCO1 96756,CCC(C(=O)NC1CC(C)(CN(C(=O)C=CC(=O)N(C)C)CC)C1)C1CCC1 96757,N1(C(C=C(CC)C)=O)CCC2(CCCN2C(c2cnc(C(C)(C)C)nc2C)=O)C1 96758,c1(C(=O)NCC(C2CC2)NC(C2CC23CC(O)C3)=O)ccc(Br)cc1Br 96759,N1(C(CC(CCC)C)=O)CC(CNC(=O)CN2CCC(C)(C)C2)OC(C)(C)C1 96760,Cc1ccc(C(N2CC(C(F)C(=O)NOCCN(C)C)(O)C2)=O)c2c1CCCC2 96761,c1(CC(=O)NCCC2(NC(=O)Cc3ccncc3Cl)CC2)ccc(Cl)cn1 96762,CC(C)C(CCN(C(=O)CC1CCSC1)C)NC(=O)CC1CCC(=O)N1 96763,Cc1cc(=NCC2CCSC2(C)C)[nH]cc1S(=O)(=O)N1CCOC(CCO)C1 96764,Cc1c(NC(=O)N(C)CC2CCN(CC(F)F)CC2)cnn1C1CC1 96765,c1(CC(=O)NCCCN(C(C23CCCCC2C3)=O)CC)ccc(S(C)(=O)=O)cc1 96766,CC1CCC(CC(N2CCC(Cc3cn(CCCCN(C)CC)nn3)C2)=O)OC1 96767,Cc1nn(C)c2nc(CSCCNC(C3CCCC4CCCCC34)=O)cc(O)c12 96768,C1(C(N(C2CNC(=O)C23CC3)C)=O)CCN(C(=O)CCC2(C)N=N2)O1 96769,CCC(CCC(=O)NC(CC(=O)NC)c1cccs1)NC(=O)C(C)(C)N(C)C 96770,C(=O)(C(F)(F)C(C)O)N1CC(OC)C(C(=O)N(C(CF)CF)C)C1 96771,N1(C(C2CCC(C)(C)O2)=O)CCC2(CCC(NC(=O)CC3CCCOC3)CC2)C1 96772,CCCCCC(CC)C(=O)NC(C)C(C)(C)NC(c1ccc(CC)[nH]1)=O 96773,c1(CCC(=O)NC(C2N(C(c3cnc(SC)s3)=O)CCC2)C)ccnc(Cl)c1 96774,N1(Cc2nc(CC(C)C)on2)CCC(O)C(C(N2CCN(C3CC3)C(C)C2)=O)C1 96775,N1(C(C(C)=CC)=O)CC(NC(=O)CC2COCCO2)CC2(CCC2)C1 96776,N1(C(c2c(NC)cc(Cl)cc2)=O)CCN(C(=O)CC(=O)NC2CC2)C(C)C1C 96777,c1(NC(c2n(CCCF)nnn2)c2ncoc2C2CC2)cc(F)cc(F)c1 96778,N1(C(CC(C)(C)N(C(C2CCCC(C)C2)=O)C)=O)CCCc2occc2C1 96779,c1(C(C)=O)ccc(NC(=O)C(=O)NCC(Cc2ccc(Cl)cc2)C(=O)O)cc1 96780,Cc1ccc(CCC(=O)NC2C=CCN(C(C3(C(F)F)CC3)=O)C2)cn1 96781,C1(C)(C(N2CCC(C(C(N3CC(C#C)C3)=O)F)C2)=O)COCCO1 96782,C1(NC(C(C)C#N)=O)CCOC12CCN(C(=O)CC1(C)CCS(=O)(=O)N1)CC2 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96818,CC1CCN(C(=O)CCc2ccc(Cl)cc2F)CC1CNC(=O)CN(C)C(N)=O 96819,C1(NC(=O)CSc2ccccc2)CCN(C(c2ccccc2Br)=O)CC1 96820,C(=O)(CS(=O)(=O)CCO)NC1C(C)CN(C(=O)CCc2cccc(Cl)c2)C1 96821,C(CC(C)(C)CC(=O)N1CC(c2cc(O)no2)C1)OC.C12CC=CCC1C(=O)NOC2=O 96822,C(N=c1[nH]c(=N)[nH]c(=NC2CCCCC2N(C)C)[nH]1)c1ccc(CC)cn1 96823,CC(CC(=O)N1CC(O)(CN(C(=O)CC2COC(=O)N2)C)C1)CC(F)(F)F 96824,CC1OCCCC1C(=O)NC1CCOC1C(=O)NC1(C2CC2)CCC1 96825,c1(C(=O)NC2CC(CCNC(C=CC(C)C)=O)C2)cc2c(s1)CCS(=O)(=O)C2 96826,C(COCC(N1CC(C(=O)N(C)C)C1)=O)(C(=O)N1CC(O)(C(F)(F)F)C1)N(C)C 96827,C1(C(=O)NC(c2nncs2)C)CN(C(C2CC2Cl)=O)CC12CCC2 96828,c1(S)nnc2ccccn12.N1(CCCOC)CCCC(C(=O)NCCCNC)C1 96829,c1(C(CC)C)ccc(C(C(=O)NCCC2(C)CC2)N(C2CCCCCC2)C)cc1 96830,N1(C(C(C)(C)OCC)=O)CCC(N(CCO)C(c2sccc2F)=O)CC1 96831,Cc1cc([N+](=O)[O-])c(Cl)cc1NC(c1ccc(NCc2ccn(C)n2)cn1)=O 96832,C1(CC(N2CCC3OCCC3C2)=O)CCc2ccccc2N1 96833,c1(NC(CNC(C(C)=C(CC)C)=O)(C)C(C)C)nc(C)nc2sc3c(c12)CCC3 96834,C1(CC(NOC(C(=O)OC)C)=O)CN(C(c2c[nH]nc2C2CC2)=O)CC1C 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97119,C1(NC(C(N2CCN(C)CC2)C)=O)CC2C(NC(=O)C(C)(C)O)C2C1 97120,N1(C(c2c(C)cncc2)=O)C2CCC(C2)C1CNC(=O)CNC(n1cncn1)=O 97121,C1(C)(CC(=O)N(C)CCNC(c2csc(C3CC3)n2)=O)CCS(=O)(=O)N1 97122,C(CO)(CO)(CO)NC(C1(CCNC(C(C)C2CCCO2)=O)CC1)=O 97123,N1(C(C(C)c2cc[nH]n2)=O)C2CCC1CC(CNC(C1(CF)CCC1)=O)C2 97124,N1(C(C(=O)NCc2ccc(OC)cc2)c2ccon2)CCC(C)C(C)(C)C1 97125,C(=O)(CC(F)(F)C(F)F)NCC1N(C(c2ccc(CC)c(Cl)c2)=O)CCC1CC 97126,c1(CC(=O)OC)ccc(O)c(NC(C2C3CN(C(c4cnn(C)c4)=O)CC23)=O)c1 97127,N1(C(c2ccc(CNC(c3c(C(C)C)cco3)=O)cc2)=O)CCC(O)CC(C)C1 97128,C1(C(=O)NC)CCCCC1NC(=O)CCCCNC(=O)CN(C)CCOC 97129,C1(CNC(c2c(C)n[nH]c2)=O)C(C)CCCN1C(C1CN2CCN1CC2)=O 97130,C12(C(=O)NCC3(CNC(C=CC(CC)C)=O)CCC3)CCCC1(C(N)=O)C2 97131,c1(C(=O)NC(CC=C)CNC(=O)CN(S(C)(=O)=O)C)cccc2oc(C)nc12 97132,CCN=c1[nH]c(C(N2CCN(C)CC2CNC(c2c(C)ccn2C)=O)=O)cs1 97133,c1(C(N2CCCC(NC(C(C)N(C)C)=O)(CO)C2)=O)cc(F)cc2nn(C)cc12 97134,c1(Cn2cc(C3CN(C(C4N(C)CCC4)=O)C3)nn2)ccc(I)c(Cl)c1 97135,N1(C(CC2(OC)CCC2)=O)CCOCC(NC(c2cccc(OCCF)c2)=O)C1 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97153,N1(CC2CN(S(C)(=O)=O)C2)CCc2c([nH]c3cc(Br)ccc23)C1 97154,c1(OC)c(Cl)cc(C(=O)NC2CC(NC(c3c(C)coc3C)=O)CC2O)nc1Cl 97155,N1(C(CC(C)F)=O)CCN(C(=O)CC2CCC(F)(F)CC2)CC12CCC2 97156,C(=O)(C(CC1CC1)NC(=O)COC1CCN(C(=O)CN(C)C2CC2)C1)OC 97157,C1(NC(C2CCC(C)C2)=O)CN(CCCC(C)(C)C)CCC1C 97158,CC1(C(=O)NCC2CCC(F)(CNC(c3ccn(C(F)F)n3)=O)C2)CCC(=O)N1 97159,Cc1cc(C)c(C(N2CC(NC(=O)C(O)CN(C)C)C(C)C2)=O)cn1 97160,c1(C(=O)NC2CCN(C(c3cnc(CCC)s3)=O)C(C)C2)cc(F)c(C)cc1Cl 97161,C=C=C(C)CC(=O)NCCN(CC(C)O)C(=O)CN(C)C1CC1 97162,c1(NC(CCC=C)=O)cnc2c(c1)CN(S(=O)(=O)CC(C)C)CC2 97163,C1(NC(CCc2cc(OC)no2)=O)(CO)CCN(C(C2COCCO2)=O)C1 97164,N1(C(CCC(N)=O)=O)CC2CCCCN2CC1CNC(=O)CC1CCOCC1 97165,N1(C(c2cnc(C)s2)=O)CCC(C)(C(=O)NCCC2CCCC2(C)C)C1 97166,C1(CC)(NC(=O)CNC=O)CCN(C(=O)C(C)Cc2ccc(F)cc2F)CC1 97167,N1(C(CC2ON=C(CC)C2)=O)CC(F)(F)CC1C(=O)NCC(F)C(C)(C)O 97168,CC1(C)CC1(C#N)C(=O)NCC1(CNC(c2nc(Cl)sc2Cl)=O)CC1 97169,CC(C)C(O)CC(=O)NCC1(NC(c2ccc(-c3nccs3)cc2)=O)CCOC1 97170,N1(C(C=CCOC)=O)CCCC(C)(NC(c2cn3ccsc3n2)=O)C1 97171,C1(C(CO)NC(C=C(C)CCNC(=O)CCOCC2CC2)=O)CCOC1 97172,c1(OCC)cccc(N2CCOCC(CNC(c3cnsn3)=O)C2)c1[N+](=O)[O-] 97173,c1(C(N2CCC(CNC(C(C)(C)C3CCCO3)=O)C2)=O)ccc(C2CC2)nc1 97174,C#Cc1ccc(C(=O)N(C2CC(NC(C3(CC(C)C)CCNC3=O)=O)C2)C)cc1 97175,Cc1cccnc1C(=O)NC1CCCC1n1cc(COCC(C)C)nn1 97176,C1(c2sccn2)CCCN(CCc2ncc[nH]2)C1.c12cn(nn1)C2C1CC1 97177,N1(C(C2C(c3c(C)nn(C)c3C)OCC2)=O)C2CCC1CN(C(C13CC(C1)C3)=O)C2 97178,c1(CNC(CN(C(C)=O)C)=O)ncccc1CNC(C1CN(C)C1)=O 97179,C1(NC(C(Cc2ccoc2)NC(c2c(C)n(C)cn2)=O)=O)CCNC(=O)CC1 97180,C1(CCNC(C=CCOCCOC)=O)CN(C(=O)CS(N)(=O)=O)CCCO1 97181,c1(N(C(c2ccnn2CC)C(=O)NC(CC)C)C)ccc(C)c(F)c1 97182,C1(C2CCN(C(C3CC3OCC)=O)CC2)(NC(C=C(CCC)CCC)=O)CC1 97183,CC1(C)CCC(F)(F)CC1C(=O)NC1CCN(C(C2CCSCC2)=O)CC1F 97184,C1(CC(=O)NC2CCCC(NC(=O)C=C3CCCCC3)C2)(OC)CCCCC1 97185,C(=O)(C1=COCCO1)NCC1C(NC(c2n[nH]c(C)c2Cl)=O)CCCC1 97186,N1(C(c2c(CCC)nco2)=O)CCCC2CN(C(c3cccc(C)c3)=O)CCC12 97187,CS(=O)(=O)c1ccc(OCC(=O)NC2(CNC(C34CCCCC3C4)=O)CC2)cc1 97188,c1(Cc2n(C(C)(C)C)cnc2)ccc(NC(CC(N)=O)c2ccccc2)cc1 97189,CON(C(=O)C=CCN(C)C(c1sccc1C#N)=O)C(C)C 97190,C1(c2cn(C3CN(C(C(C)(C)OC(C)=O)=O)C3)nn2)C(C)(C)C1(C)C 97191,N#CC1CCC(C(=O)NCC=CCC(=O)N(C2CCCCCC2)CCO)C1 97192,C1(NC(c2scc(C(C)=O)c2)=O)CC(NC(c2cncc(C(F)F)c2)=O)CC1O 97193,C1(C)(CN(C(=O)CC2C=CCC2)C)CCCC1NC(c1sccc1Cl)=O 97194,Cn1ncc2c(C(=O)NCC3CC3NC(c3cnc4c(c3)NCC4)=O)ccnc12 97195,N1(c2ccn(C)n2)Cc2ccc(Nc3cc(O)nc(C4CC4)n3)cc2C1=O 97196,c1(OC)ccc(C(N2CC(N(C(=O)Cc3ccc(O)nc3)C)C(F)C2)=O)cc1F 97197,c1(CNCNC2CCN(C(C)=O)C2)c(I)ccnc1F 97198,N1(C(C23C(C)(C)C(CC2)C3)=O)CC2CCC(CNC(=O)C3CC3)C2C1 97199,N(C(O)=C(C(=O)C(C(CCC)O)=O)OC)CCCCCNC 97200,c1(OCC)ccccc1C1(C(=O)NCC(O)CNC(=O)C(C)NC(C)=O)CC1 97201,c1(C(N2CCCC(C)(NC(C(C)n3cccn3)=O)C2)=O)ccc2[nH]ccc2c1 97202,N1(C(=O)OC)CCC(NC(=O)NCCC(O)C(F)F)CC1 97203,C1(C2CC2)(CNC(COCCN(C)C(C2CC2Cl)=O)=O)CCC1 97204,c1(CC)cc(NC2CCCCC2C(N)=O)cc(=O)o1 97205,C(c1cn[nH]c1)=C(C)C(=O)N1CC(n2cc(CNC(c3cocn3)=O)nn2)C1 97206,N1(C(C)=O)CCCC1C(=O)NCC1(F)CC(NC(C2CC(C)=NO2)=O)C1 97207,C(=O)(C(C)(C)n1cc(NC(=O)C(N2CCC2(C)c2ccccc2)=O)cn1)OCC 97208,c1(C(=O)NCCC2CCN(C(C(COC)O)=O)C2)ccc(OC)c(SC(C)C)c1 97209,c1(C(=O)NC2C(CNC(c3c(C)c[nH]n3)=O)CCCC2)cc(Cl)ncc1Cl 97210,C1(CC(=O)OC)CC2(CCN(C(c3cc(C)c(Cl)s3)C(=O)NCC3CC3)C2)CO1 97211,C1(C(N(CCOC)C2CC2)=O)CCCN(C(c2cc(OCC)cnn2)=O)C1 97212,Cc1cnsc1C(N1CCCC1C(C)(C)CNC(=O)Cc1cnn(C)c1)=O 97213,c1(C(=O)NC(c2ccc(Oc3cccc(F)c3)nc2)C)ccnc(S(C)(=O)=O)c1 97214,c1(NC(C2CC(CNC(c3ccc(C)s3)=O)C2)=O)ccccc1N=[N+]=[N-] 97215,C(=O)(CC(C1CC1)NC(C1CCCN1C(C1CCCO1)=O)=O)NC 97216,c1(OC)ccc(C(=O)NCCC2CN(C(C3C(C)(C)C3(C)C)=O)CCO2)nc1N 97217,N1(C(c2c(CC)cno2)=O)CCOCC1CC(=O)N(C1CCN(C)C1=O)C 97218,c1(CC(=O)NC2CC(CNC(c3c(CC)ncs3)=O)C2)cc(O)nc(O)n1 97219,C1(OC)CN(C(=O)CC(C)SC)CC1NC(=O)CCC1CCCCCC1 97220,N1(C(COCCC=C)=O)CCN(C(C2CCC(=O)N2C)=O)C(C(C)(C)C)C1 97221,n1(CC)ncnc1CNC(=O)C(C1CC1)N(C(=O)CN(CC(C)(C)C)C)C 97222,N1(C(CC2(C)CC2(Cl)Cl)=O)CC2CCC1C1CN(C(=O)CCc3ccon3)CC21 97223,N1(C(c2cn(-c3cccc(Cl)c3)nn2)=O)CCC(O)C12CCSC2 97224,C(=O)(C1CCCc2cccnc21)NC1(C2CN(C(c3c(C)noc3N)=O)C2)CC1 97225,N1(C(C2(CC=C)CC2)=O)CC(C(=O)NCC2CC(C(C)(C)C)C2)C(F)(F)C1 97226,N1(C(CC(CC)C2CC2)=O)CCC2(CC1)CCN(C(C1CC(=C3CC3)C1)=O)C2 97227,C1(C(N2CCCC(CN(C(=O)CCF)CC)C2)=O)CCC2(CCC2)CO1 97228,c1(C(=O)NC2C(NC(c3cc(OC)ncc3)=O)C2)cc2cc(Cl)ccc2s1 97229,C(=O)(CC1=NN(C)C(=O)C1)NC12CC(CNC(C(CC=C)(C)C)=O)(OC1)C2 97230,S(=O)(=O)(c1ccc(N2CCC(NC3CCN(CC)C3)C2)c(Br)c1)N(CC)CC 97231,N1(C(CCC)=O)CC2CCCC2(CNC(=O)CN2CCn3ccnc3C2)C1 97232,Cc1cccc(C(C(C)C)NC(=O)NCCc2nc(C(C)(C)C)no2)c1 97233,C1(CNC(Cc2cc(C)on2)=O)CCC(C)CN1C(=O)C=Cc1cnn(C)c1 97234,CCC(CC(C)C)C(=O)NCC1CCCC1C(=O)NC1(C(=O)OC)CC1 97235,N1(C(c2cc(C)no2)=O)CCCC(C(=O)NCC23CCCC2C3)C1 97236,C1(CNC(C(CC)OC)=O)CN(C)CCN1C(=O)CCOCC(C)C 97237,c1(OCCC)ccc(C(=O)NC(c2cnc(C)o2)(C)C)cc1OCCC 97238,Cc1ccc(F)c(OCC(=O)NC2CN(C(=O)CCn3ccnc3)CCC2C)c1 97239,Nc1cc(C(N2CCN(C(=O)Cc3cncnc3)C3CC23)=O)c(F)c(F)c1F 97240,C1(C(=O)NCCCNC(=O)Cc2cncnc2O)CCC12CCOCC2 97241,C1(CNC(C=CC)=O)C2CN(C(c3cc(CCCCC)[nH]n3)=O)CC12 97242,N1(C(C2CCN(OC)CC2)=O)CCC2CN(C(=O)C(O)C(F)(F)F)C(C)C12 97243,C1(CC#C)(C(N2CC(O)C(O)C2)=O)CCN(C(c2cc(CC)oc2C)=O)C1 97244,N1(C(C(C)NC(N)=O)=O)CC(NC(=O)C(F)(F)c2nccs2)C(C)C1 97245,C1(OC)(CNC(C2CC(O)C2)=O)CN(C(C2(c3ccccc3)CC2(Cl)Cl)=O)C1 97246,CCC(CC)C(=O)NCCN(C(c1c[nH]nc1Br)=O)C1CC1 97247,c1(N(CC=C)C)nc(N2CCCC(CC=C)C2)c2c(n1)CCCCCC2 97248,c1(CC(N2C(CN(C(C(CC)(C)OC)=O)C)COCC2)=O)cnc2ncccn12 97249,C1(CNC(c2ccc(C)cc2F)=O)CCCCN(C(C2CCC(=O)NC2)=O)CC1 97250,C(C(N)CC(C)(C)C(=O)N1CCC(N(C)Cc2ccccc2)C1)OC 97251,c1(CCC(=O)NCC(CNC(C)=O)=O)ccn(C)c1 97252,c12ccc(c(F)c1)[nH]2.C1(C(=O)NCCC#C)C2CN(C(=O)OC)CC12 97253,c1(C(=O)NC2(CCCC(=O)N(CC(=O)NC3CC3)C)CCC2)ccc(F)cc1F 97254,CCCCC(CC)CC(C(=O)NC)NCC1(C(=O)OCC)CCOCC1 97255,CC(CC(=O)NC1CC(C)(NC(C2CNC(=O)CC23CC3)=O)C1)C(F)(F)F 97256,c1(C(=O)NC(c2nc(C)on2)C=Cc2ccccc2)ccc(N2CCCCC2)cc1O 97257,N1(C(Cc2ccc(C)o2)=O)CC2CN(C(=O)Cc3sc(O)nc3O)CC2C1 97258,C1(N(C(C(CSCC)NC(C2CC(=O)C2)=O)=O)C)CCCC(C)C1C 97259,c1(C(=O)NCC(CCNC(CN(CCC)C)=O)O)c(F)c(F)cc(F)c1F 97260,CC(C)P(=O)(CC(=O)NCCCCN(C)C)C(C)C.C1(=O)CCOCC(C)(C)N1 97261,C1(C(N2C(CN(C(CC(C)N(C)C)=O)C)CCCC2)=O)CNC(=O)CC1(C)C 97262,C1(C(N(CC(C)(C)NC(=O)CNC(c2cccnc2)=O)C)=O)COCCN1C=O 97263,C1(CC)CN(C(c2cc(C(C)C)on2)=O)CCN1C(=O)CCc1ccccc1O 97264,Cc1ccccc1OCCCC(=O)NC1CCCC1NC(C1(O)CC(CF)C1)=O 97265,N1(C(CCCC(=O)NCC)=O)CC(NC(c2noc(C3CC3)c2C)=O)CC12CCC2 97266,N1(C(C(CC)NC(C)=O)=O)CC(C)C(N=c2[nH]n(C(C)C)cc2[N+](=O)[O-])C1 97267,C(C(C)(C)C(=O)N(C)CCN(C)C(N)=O)N(C(=O)C=C1CCCCC1)C 97268,Cc1cccc(CCNC(=O)CC2CCCN(C(C3CC=CC3)=O)C2)c1 97269,c1(C(N2CC(OCCNC(C(CC=C)OC)=O)C2)=O)cc2n(n1)CCCN2 97270,CCCC(CNC(c1cc(Cl)n(C)n1)=O)C(=O)NCC(O)C=O.OCC 97271,Cc1ccc(C(O)Cc2cn(C(C)C(=O)N(C)CCN3CCCC3)nn2)cc1 97272,N1(C(c2nn(C)c(Cl)c2)=O)CC2CCCC(NC(C3(O)CC4CCC3C4)=O)C2C1 97273,C#CCC(C(=O)NC)NC(c1coc(CNC(=O)CSC2CC2)c1)=O 97274,c1(C(=O)NCCC(C)NC(c2ncc(F)cc2N)=O)cc(Cl)cc(Cl)c1 97275,N1(C(CC=CC=C)=O)CC2(CCN(C(c3sccc3Cl)=O)CC2)CC1C 97276,C1(CNC(=O)CCOC2COC2)(NC(c2cc[n+]([O-])cc2)=O)CCOCC1 97277,Cc1cn(C)nc1C(N1CC(n2cc(Cn3cncn3)nn2)C(O)C1)=O 97278,C1(CC)CN(C(=O)CC2CCOCC2)CCN1CC.c12ccn(n1)CCNC2=O 97279,c1(CC)ccc(C(N2CCOCC2CNC(=O)CC(C)COC)=O)nc1 97280,C1(CC(=O)NC(C)C(C)(C)NC(c2cccc(C(F)(F)F)c2)=O)CCC(=O)N1C 97281,N1(C(c2nccc(C)c2)=O)CCN(C(c2cnc3[nH]cncc2-3)=O)C2CCC12 97282,Cc1nccn2ncc(C(=O)NCCC(C)NC(c3cc4c(s3)CCCC4)=O)c12 97283,c1(C(=O)NC(CNC(c2c(C)nc(OC)s2)=O)C)cnc(O)c(C(F)(F)F)c1 97284,c1(C(=O)OC)cnc(N2CCN(C(c3ccnn3C)=O)CC2C)nc1C 97285,c1(C(=O)NCC2CC(CC(=O)NCC(c3ccsc3)C)C2)ccncc1N=[N+]=[N-] 97286,C1(CC(=O)NCCOC2CCN(C(c3c(C)cno3)=O)C2)CCC(C)(C)CC1 97287,c1(C(=O)NC2CCN(C(c3cc(OC)cc(Cl)c3)=O)C2C)cccc2cnnn12 97288,c1(C(N2C(C(=O)O)C3CC3C2)=O)cnn2ccsc12 97289,O=C(C1CCCc2nn[nH]c21)N1CCC2(CCCN(C(=O)CO)C2)C1 97290,N1(C(C(C=C)C)=O)CC2CCCC(N(C)C(c3nnsc3CC)=O)C2C1 97291,N1(C(C(CC)COC)=O)CCCC(F)(CNC(=O)CSCc2cccc(Cl)c2)C1 97292,CC1CN(C(C2CC2(Cl)Cl)=O)CC1CCNC(C1CCCCCC1)=O 97293,c1(OC)ncc(C(=O)NCC(C2CC2)NC(=O)CCNC(C2CCCCC2)=O)s1 97294,c1(C(C)NC(=O)CCCNC(=O)CN2CCC2C)nccn1C(C)(C)C 97295,C1(CC(N2CCC(C)(CCC)C2)=O)CC2(C1)CN(C(C1(C)CNC(=O)N1)=O)C2 97296,C(=O)(CCCCCF)NCC(C)(C)NC(C(C(=O)N(C)C)C1CC1)=O 97297,c1(COCC(=O)NCC(COC)NC(C2CCCN2C2CC2)=O)ccccn1 97298,CC(C(=O)OC(C)(C)C)C(=O)NCC1(C)CN(C(=O)Cc2ccsn2)C1 97299,C(C(C)C(=O)N(CC(O)CO)CC)NC(CCOCC#C)=O 97300,c1(CN(C)Cc2cccc(Cl)c2)ncccc1F.C12CCN(C1)C(=O)C(=O)NC2 97301,c1(C(C(=O)N(C2CCCC2)CC2CC(NC(=O)C=CCF)C2)O)ccc([N+](=O)[O-])cc1 97302,c1(NC(C(CC)n2cnc(-c3nn[nH]n3)n2)=O)ccc(Br)c2c1CCO2 97303,C=C(C)C1CN(C(=O)CCN(C(=O)C(c2ccccc2)C)CCCO)CCO1 97304,c1(OC)cc(OC)nc(N2CC(CO)(NC(=O)C(O)C(C)C)C2)n1 97305,C(CC(C)C)(C(=O)NCC(n1ccnn1)C)ONC(c1c(CC)ncs1)=O 97306,c1(-c2c(F)cncc2)ccc(C=NOCCN2CC=CCO2)cc1 97307,CC1CCCC1(C)C(N1CCOC(C(C)NC(=O)Cn2cc(N)cn2)C1)=O 97308,CC1(C)CCCC(CCN(C(c2ncc(Cl)s2)C(=O)NCCCOC2CC2)C)C1 97309,C1(CNC(CCn2c(C)ncc2)=O)CCN(C(=O)CCc2cncnc2)CC1O 97310,CCCCC(O)C(=O)N1CCN(Cc2cnc(OC)c(Cl)c2)C2CC12 97311,C1(Oc2cnc(C(=O)NCC3(C(=O)OC)CC(CC)C3)s2)CCN(CC)CC1C 97312,CC(Cn1cccn1)C(=O)NCc1n[nH]cc1C(=O)N(C1CCCC1C)C 97313,C1(N(C(c2c(OC)csc2)=O)C)CCCCC1NC(c1cncc(C(F)F)c1)=O 97314,C1(NC(c2ccc(O)cc2)=O)COCCN(C(C2CCN(C3CC3)C2=O)=O)C1 97315,C(CCO)(C(F)F)N(C(C(C1CN(C(c2n(CCC)ncc2)=O)C1)O)=O)C 97316,C#Cc1cc(NC(=O)C(C2CCCO2)NC(=O)Cc2csnn2)cc(F)c1 97317,c1(OC)ncc(C(=O)NC(C)C(CO)NC(c2ccc(F)cc2SC)=O)cc1C 97318,c1(CCC(=O)N(CCNC(C(C)(C)OC(C)=O)=O)C)ccc(Br)nc1 97319,c1(N2CC3(CN(C(=O)C=Cc4ccc(Cl)nc4)C3)C2)ncnc2ccc(Cl)cc12 97320,c1(OC)ccccc1C(=O)NC1CC(CNC(=O)CC2(O)CC2)C1 97321,C1(C(=O)NCCNC(c2ccc(CC)cc2F)=O)CC(=O)N(C)C(=O)N1 97322,Cc1ccc(C(N2CCN(C(C3(c4ccc(F)cc4)CC3)=O)C3CC23)=O)cc1Cl 97323,Cc1cc(C(=O)NCC(C2CC2)NC(c2cnn(CCF)c2)=O)n[nH]1 97324,CCC(C)CC(=O)NC(c1ccc(C2CC2)s1)C(=O)N(C)Cc1cccc(C)c1 97325,C1(C(N2CCN(C(c3ncn(C)c3)=O)CC2)=O)CCc2nnnn2C1 97326,c1(OC)cc(CC(N2CCC(NC(C3CC3C)=O)C2(C)C)=O)ccc1Cl 97327,C(=O)(C(CCc1ccccc1)N1CCOC(CSCC)C1)NCCOC.C(C)(=O)O 97328,N1(C(c2sc(C)cc2Br)C(=O)NC(CC)C)Cc2cc(Br)ccc2CC1C 97329,N1(CCOC)CC(O)CC1=O.C(c1cn(C(C)C)cn1)=CCOC(=O)OC(C)(C)C 97330,c1(C(N2CC(CC)C(NC(=O)COC3CC=CC3)CC2)=O)cc2cccnc2s1 97331,c1(CNc2nnc(CC)n2CC(=O)OC(C)(C)C)cccc(S(F)(F)(F)(F)F)c1 97332,Cc1ncn(C)c1C(=O)NC1(CO)CN(C(=O)CSc2ccc(Cl)cc2)C1 97333,C1(NC(c2ccc(CCCC)cc2)=O)CCN(C(C2(C3CC3)CCC2)=O)CC1O 97334,C12(NC(COc3cccc(SC)c3)=O)CCC(CN(C(C)=O)C1)C2 97335,N1(C(c2cnc(C3CCCO3)s2)C(=O)NCC)CCC(O)CC(C)(C)C1 97336,Cc1nc(NCCC2=CCCC2)cc(N2CCCN(S(C)(=O)=O)CC2)n1 97337,c1(C(=O)NCC(=C2CN(C(CCCSC)=O)C2)F)ncc(Cl)nc1Cl 97338,C=C(C)CC(C(=O)NCCNC(c1cccs1)=O)NC(=O)CC1(O)CCCCC1 97339,C(C(=O)Nc1noc(C2(C)CC2)n1)(C(C)C)OC 97340,C=C=C(C)CC(=O)NCCN(CC(C)O)C(=O)CC1CC(OC)C1 97341,C(Cc1cc[nH]n1)(C(=O)N(CCCN(C)C)CC)NC(C=CCC)=O 97342,Cc1cc(Br)ccc1CC(=O)NC1CC1NC(C1(C)CC(C)(C)C1)=O 97343,CCCC(C)(O)CC(=O)NCCCN(C(=O)C(c1ccc(C(F)(F)F)cc1)O)C 97344,Cc1cc([N+](=O)[O-])cc([N+](=O)[O-])c1NC(C1CCN(C(C2(O)CC2)=O)CC1)C 97345,CC(C)C(C)CC(=O)N1CC(N2CCN(C(=O)CCC3CC3(F)F)CC2)C1 97346,c1(CNC2C(C(=O)Nc3ccc(Cl)cn3)C2)c(Br)cccc1Br 97347,c1(C(N2C(CNC(C(CC)O)=O)CC(F)(F)C2)=O)cc2c(cc1F)NC(=O)CC2 97348,c1(C(C)(C)C(O)NC(=O)CCF)cccc(I)c1 97349,CCC(C)CC(C(=O)NCC1CCCN1C(C)=O)NC(c1cnn(C2CC2)c1)=O 97350,c1(C(=O)Nc2cnccc2[N+](=O)[O-])cc(-c2ccc(CO)o2)cc2c[nH]nc12 97351,CC(C)C(C)CC(=O)N(C1CC(C(=O)NCC(O)(C2CC2)C2CC2)C1)C 97352,c1(C(N2CCCC(CNC(C3C(C=C)C3)=O)C2)=O)cc2nccc(C(F)F)n2n1 97353,Cc1ccc(CN2CC(C)(CC(N3CCOC(C#N)C3)=O)C2)cc1Cl 97354,CC(CN(C)C)CCC(=O)NCCN(C)C(C1CCC(F)(F)C1O)=O 97355,C(CC(C)(C)C)(C(=O)NCC1CCC=CCCC1)NC(C(SC)SC)=O 97356,C1(C2CCN(C(c3cncs3)=O)C2)(NC(CC=C)=O)CC1 97357,C(C)(CC(C)(C)C)(c1nnnn1C1COC1)NC1CCC(CC)CC1 97358,c1(C(=O)NCCN(C)C(c2ccc(Cl)c(Cl)c2)=O)cc2sccc2[nH]1 97359,c1(-c2cccc(OC(C)=O)c2)nc2c(s1)CCN(C(C1C3COCC13)=O)C2 97360,C1(C(=O)NC2(C)CCN(C(=O)OC)C2)(CNC(c2ccco2)=O)CCOCC1 97361,Cc1cc(=NC2CCCn3ccnc32)[nH]c(N2CCC(C)C2)n1 97362,N1(C(c2c(C)cccc2)=O)CCN(C(=O)COCc2nc[nH]n2)CCC1C 97363,C1(C(=O)NC(CNC(c2cc(C(C)=O)sc2)=O)C(C)(C)C)CCCC2(CC2)C1 97364,C#Cc1cccc(C(N2CC=CCC2C(N2CCCC(C(C)(C)C)C2)=O)=O)c1C 97365,Cc1cnn(C)c1CC(=O)NCC(CC(=O)NC(C)(C)CC(C)C)C1CCC1 97366,c1(C(N2C(CC#C)(C(=O)NCC3CC(F)(F)C3)CCC2)=O)cc(C)cc(C#N)c1 97367,c1(C(=O)NC(C)C(C)NC(=O)CCNC(C2CCC2)=O)ccc2ncccc2c1 97368,c1(C(N2CC(NC(C(CCC)C)=O)C(O)C2)=O)sc2ncccc2c1Cl 97369,c1(C(=O)NC(C(C)C)CCN(C)C(c2cccc(O)n2)=O)ccc2c(c1)CCOC2 97370,C1(NC(c2cc(C)nc(O)n2)=O)C2CCCCN(C(c3c[nH]cc(Cl)c3=O)=O)C12 97371,C(=O)(C1=COCCC1)N(C)CC1CCN(C(C(CC2CCC2)OC)=O)C1 97372,C(=O)(C1=COCCC1)N1C(C)CC(NC(C2CNC(=O)O2)=O)C1 97373,C(C)(C(=O)N(C)CC1CN(C(C2(C(C)(F)F)CCC2)=O)C1)NC(CC)=O 97374,C1(CNC(Cn2c(C)ccn2)=O)CCC2CN(C(=O)CCc3nncs3)CC12 97375,c1(-c2onc(-c3cccc(OC)c3)n2)cccc2cc(OC)ccc12 97376,C12(CCNC(c3cccc(CCC)c3)=O)CCC(C1)N(C(=O)C(C)N(C)C)C2 97377,CC(F)(F)CCCC(=O)NC1CC(NC(=O)Cc2cnsc2)C12CCC2 97378,CC1=C(C(=O)NCCN(CCCN(C)C)C(=O)CN2CCNC(=O)C2)CCO1 97379,C1(C(N2C3C(CNC(C(C(C)O)C)=O)CC(CC3)C2)=O)CCc2cnn(C)c2C1 97380,N1(C(C(C)(C)O)=O)CC2CCC1CN2C(C1(C#N)CCC1)=O 97381,C1(C(=O)NC(CCCNC(c2c(Cl)cc(C)s2)=O)C)CCCC2(CCC2)O1 97382,C1(C)(C(=O)NC23CC(NC(CCSC)=O)(C2)C3)C2CCC(C2)C1(C)C 97383,N(C1C(=O)Nc2ccc(F)cc21)C(C1=C(C)OCC1)=O 97384,N1(C(=O)C(F)=CCCF)CCC(C2CCN(C(C3CC3F)=O)CC2)C1 97385,CN1CCC12CN(C(C1C(NC(=O)COCCCN(C)C)C1(C)C)=O)C2 97386,CCC(C(=O)OC)C(=O)NC(CCOCCO)C(=O)NC1CC(CO)C2CC12 97387,c1(C(=O)NCC2CN(C(c3cccc(C(=O)NC)n3)=O)C2)sccc1S(N)(=O)=O 97388,C(=O)(C1CC(C)(C)Oc2ccccc21)N1CCC(NC(c2n(C)cnc2)=O)C1 97389,N1(C(C(=O)NCC(c2cn(C)nc2)(C)O)=O)CCc2c(ncn(C)c2=O)C1 97390,O=C(C1CCCn2cncc21)NCC1CCCCN(C(=O)C2=CCCCO2)C1 97391,Clc1ccc(-c2nc(CN3CC4CC4C3)n(-c3cccnc3)n2)cc1Cl 97392,N1(C(C2(COC(C)C)CC2)=O)CC(N(C(=O)C(C)CN2CCOCC2)C)C(O)C1 97393,Cc1ccc(C(=O)NC23CC2CN(C(c2ncn(C)n2)=O)C3)c2ccccc12 97394,c1(C(=O)NC(c2ccc(F)cc2)CNC(CC(C)CF)=O)cnn2ccccc12 97395,c1(C(N2C(CNC(=O)C(O)CC3CCCC3)CC(O)C2)=O)c[nH]c2ncccc12 97396,Cc1ccc([N+](=O)[O-])cc1C(N1CC(O)CC1C(=O)Nc1cnc(Br)c(Cl)c1)=O 97397,C1(C(=O)NCC2CC(NC(COC(C)(C)C)=O)C2)CCC(n2cccc2)CC1 97398,c1(C(=O)NC(CC)(C)CNC(=O)CC2CCC23CCC3)nsc2ccccc12 97399,Cc1[nH]nc(C(=O)NC2CN(C(=O)C=CCF)CC2C(F)F)c1C 97400,N1(C(C(C(=O)OCC)(C)C)=O)CCc2ccccc2C(NC(=O)CCC2CC2)C1 97401,CON(C(=O)C1=CC2C=CC1C2)C1CCOCC1 97402,CC1(C)CCOC1CC(N1CCCCC1C1CCN(C(=O)C(O)C2CCC2)C1)=O 97403,C1(C(=O)NCCCCCC#C)C2CCC(C2)C1NC(C1CCC2(CC2)C1)=O 97404,N1(C(CC(C=C)C)=O)CCC2CCCC12C(=O)NCCCC(=C)Cl 97405,C(=O)(C1=NOC(C)(C)C1)N1C(C(=O)Oc2ccccc2)CCC1.C1C(O)CN1C 97406,Cc1cc(C(N2CCCN(C(=O)CCCN3CCCC3)CC2C)=O)cc2c1CCC2 97407,CCC(C)(C(=O)NC(C1CCN(C(=O)C(C)=CC2CC2)CC1)C)C(N)=O 97408,Cc1noc(C)c1C(C)C(=O)NCC#CCNC(=O)Cc1ccccc1F 97409,c1(C(=O)NC(CCCC)CNC(=O)CC(C)C2CC2)cc(C)c(C)c(Br)c1 97410,c1(NCC(C)N(C(=O)CC2CCS(=O)(=O)C2)C)cc2nn[nH]c2cc1[N+](=O)[O-] 97411,N1(CC(=O)N(CC)CC2CCC2)CCN(C(=O)C(C2CCC(=O)N2)C)CC1 97412,C1(C(N(C2CCSCC2)C)=O)CCCC(NC(=O)Cc2ccc(Cl)s2)CC1 97413,c1(OC)cc(C(N2CCC(CO)(NC(=O)CN(C)C)C2)=O)cc(F)n1 97414,C1(NC(C2(CC=C)CCCC2)=O)CC2CCC(C1F)N2C(=O)CC1CC1CC 97415,c1(CC)ccc(C(=O)NCC2CC(NC(=O)CCCc3nccs3)C2)c(O)c1 97416,c1(C(C(=O)NCCC(CNC(C(C)(C)OCC)=O)O)CC)c(C)noc1C 97417,C(C)(CO)(CC(C)C)NC(CC1(CNC(C(COCC)C)=O)CC1)=O 97418,Cc1cc(Cl)cc(Br)c1NC(C1CC(C)CN1C(c1cnc(O)cc1O)=O)=O 97419,C(=O)(CS(=O)CCC(F)(F)F)NC12C(CN(C(C(C)NC(C)=O)=O)C1)C2 97420,N1(C(c2ccc(OC(F)(F)F)c(F)c2)=O)CCC2CN(C(C3CC34CC4)=O)CC12 97421,N1(C(C2(C)CC2(Cl)Cl)=O)CCC(C)(NC(=O)CN2CCS(=O)CC2)C1 97422,N1(C(c2occ(C)c2)=O)CC2(NC(c3c(-c4ccsc4)noc3C)=O)CCC1C2 97423,CCC(C)(O)C(=O)NCCCN(C(=O)CC1CCCS1(=O)=O)CCO 97424,C12(C(=O)NCCC(C=C)C)CC(CN1C(=O)CC1C=CCCC1)C2 97425,C(=O)(C1CCCc2nncn21)N1C(CNC(C(C)S(N)(=O)=O)=O)CCC1 97426,n1(CCC)cc(C(=O)NCC2CCCC2NC(=O)C(C)SC(F)(F)F)cn1 97427,c1(-c2c(C(=O)Nc3n(C)nc(O)c3)csc2)c(Cl)cc(F)cc1Br 97428,c1(C(N2CCC(C)C2c2cccc(NC(=O)OC(C)(C)C)c2)=O)cc(O)nc(O)n1 97429,c1(C(=O)NCC2(F)CC(NC(C3ON=C(C)C3)=O)C2)ccccc1CC#N 97430,c1(C(=O)NOCc2ccccc2)ncn(Cc2cc(C(F)F)no2)n1 97431,C1(C(=O)NCC(C)(C2CCC2)NC(C=COCC)=O)CC2(C1)CC(O)C2 97432,CCCCC(CNC(C1OC(C)CC1C)=O)NC(=O)C(C)CSC 97433,CC1=C(C(=O)N2CCC(NC(c3c(F)ccc4nc[nH]c34)=O)C2)C(=O)OC1(C)C 97434,N=c1[nH]c(=NCC2CCOCC23CCCC3)[nH]c(=NCCn2ccnc2)[nH]1 97435,c1(C(=O)NC(CC=C)CNC(=O)CC(C)P(C)(C)=O)ccc2c(O)ncnc2c1 97436,CC(C(=O)NCC1(F)CN(C(c2ccc(Cl)cc2O)=O)C1)C1=CCCC1 97437,c1(C(N2C(C(N3CCCC(C)CC3)=O)CC2)=O)ccc(C#N)cc1Cl 97438,Cc1cc(C(=O)N(CC(C)NC(C2(O)CCCC2)=O)C)ccn1 97439,CCC(CCC(=O)NCCF)NC(C1CCC(=O)NC1)=O 97440,Cc1nc(C(=O)N(CCNC(=O)Cc2cn(C3CC3)cn2)C(C)C)c(C)s1 97441,S(=O)(=O)(c1ccc(C(N2CCCC2C(N2CCCC(F)C2)=O)=O)cc1)NC 97442,CCCCCC(F)C(=O)N(C(C)C(N1CCOC2(CC2)C1)=O)C 97443,N1(C(c2nn(CC)nc2C)=O)CC(C)OC2(CCN(CC3CCOCC3)C2)C1 97444,N1(C(C2(C)CC(=C)C2)=O)CC2CC(C1)CN(C(=O)CCOC1CCC1)C2 97445,C1(CO)C=CCN(CCCOC2CCOCC2)C1 97446,N1(C(C(=O)N(c2ccccc2C)C(CC)C2CC2)=O)CCCC(C)(CC#N)C1 97447,N1(C(C2CCN(C(C(C)CC3CCCC3)=O)C2)=O)CCC2(CCCCC2)C1 97448,c1(OC)ccc(C=CC(=O)NCCNC(=O)CC2CCCC(C)C2)cc1Cl 97449,C(CC(O)C(=O)NOCCCCCC1CC1)NC(CC(C)C(F)F)=O 97450,c1(NC(C(N2CC(N(C)C)C2)=O)=O)cc2c(s1)CCC2C(=O)OC(C)(C)C 97451,C(=O)(C1=CCN(C(=O)C(c2ccccc2)F)C1)NC(C#C)CC 97452,c1(C2OCCN(C(=O)NCCC(CC)CO)C2)cc(OC)c(OC)c(F)c1 97453,C(=O)(CCCCC(F)(F)F)N(C)CC1CCCC(NC(COCCSC)=O)C1 97454,C1(N(C(C(CC)CC(C)C)=O)C)CCCC2CN(C(c3csc(=N)[nH]3)=O)CC12 97455,c1(-c2nc(CCC)nn2Cc2cccc3ccccc23)ccc2nnc(C)n2c1 97456,C(=O)(C(C)C(C)C(C)(C)C)N1CC(CCNC(c2c(OC)cc(F)cc2)=O)C1 97457,CC1(C)CC(CC(=O)NC23CC(CNC(C4C5CCC(F)(F)C45)=O)(C2)C3)C(=O)O1 97458,CC(C)(CNC(C1CCCN(C(c2cccc(=O)o2)=O)CC1)=O)CN=[N+]=[N-] 97459,N1(C(c2cn(C(C)C)c(=O)cc2)=O)CCC2CN(C(C3(O)CCOC3)=O)CC12 97460,N1(C(CSc2ccc(C)cc2)=O)CCC(NC(=O)CN2CC(C)C2)CC1C 97461,c1(CC(=O)N(CCCNC(CC(C)SC)=O)C)cccc(OC(F)F)n1 97462,c1(-c2onc(C3(c4ccc(C)cc4)CCOCC3)n2)ccc2c(c1)NC(=O)NC2 97463,C1(C(N2C(CCNC(C(C(C)C)NC=O)=O)CCCC2)=O)CCCCN(C)C1=O 97464,c1(N(CCCN(C(C=COCC)=O)C)C)cc2c(cn1)C(=O)CCC2 97465,C1(CNC(COCC)=O)CCN(C(C2(c3c(Cl)cccc3Cl)CCC2)=O)CC1C 97466,C1(CN(C(C(C)(C)OCC)=O)C)CCCN(C(=O)CCC(=O)c2ccc(C)s2)C1 97467,Cc1cc(C(=O)NCCN(C(C2CCC(=O)NC2)=O)C(C)C)cc(C)c1O 97468,C1(C(=O)NCC(C)(O)CO)C2CN(C(=O)Cn3nccn3)CC12 97469,C1(C(=O)OC)OC2CCC1(NC(c1c[nH]cc1Cc1ccccc1)=O)C2 97470,N1(C(C(C)OCC=C)=O)CC2(CNC(=O)CN3CCC(C)C3)CC1(COC)C2 97471,c1(N(C(CC(CC)C)=O)C2CNCC2C#N)nc(-n2cccn2)cc(C)n1 97472,C=C(C)CCCC(=O)N1CC(C(=O)NC(C)(C)CCCF)OC(C)C1 97473,C1(C(=O)NCc2cccc(NC(CC(C)SC)=O)c2)C2CC3C(C2=O)C13 97474,CC(C)(CCNC(c1ccc(NC=O)cc1)=O)CN=c1[nH]c2cc(Br)cnc2s1 97475,C1(NC(C(N2CCSCC2)C)=O)CN(C(c2ccc(N)cc2O)=O)CC12CCC2 97476,C1(C(N2C(CN(C(CCC3C(C)C3)=O)C3CC3)CCC2)=O)CCCC1C1CC1 97477,N1(C(c2cc(OCC)n[nH]2)=O)CC2(C1)CN(C(=O)C(=O)NOC)C2 97478,Cn1cnc(CC(O)C(=O)NCC(C)(CO)NC(=O)CCCc2ccsc2)c1 97479,C(CN=c1[nH]c(C#N)c(Cl)s1)C1CC(C(=O)NCC2C(C(F)(F)F)CN(C)C2)C1 97480,c1(C(=O)NCc2cc(C(N(C(CO)C3CC3)C)=O)sc2)cnn(C)c1Cl 97481,C(=O)(CCCC(=O)N1CCOCC1C(=O)NCC1(C)CC(O)C1)OCC 97482,c1(C(N2CCC(NC(C3CCN(C)C3)=O)C2)=O)cc2n(n1)CCCCO2 97483,C(=O)(C(C)(C)CNC(=O)Cc1ccnn1C)NCC(CC)CC 97484,CC(=O)C(C(C)C)NC(=O)NC1CCOC1.C12CCCCN1OC2=O 97485,c1(C(N2CC(C(C)NC(c3cccn3C)=O)C2)=O)ccc(Br)cc1O 97486,c1(C(C)C)nnc(C=CC(=O)NCCC2(CNC(C3CC4(C3)CC4F)=O)CC2)o1 97487,O=C1COc2cc(C(N3CCN(C(c4ccc(F)cc4)=O)CC3)=O)ccc2N1 97488,c1(SCC)cc(=NCCc2ccccc2C(=O)O)[nH]cc1Br 97489,C#CCC(C(=O)NCC(C)CNC(c1ccn(CC(C)C)n1)=O)C1CC1 97490,C1(CNC(C2(OC)CCSC2)=O)CC2(CCN(C(=O)C(CO)C(C)C)C2)CO1 97491,C1(C(=O)NCC2(C#C)CCCC2)CCC2(CC2)N1C(c1ccc(C)n1C)=O 97492,C1(CNC(c2cn(CCOC)c(=O)cc2)=O)CC12CCN(C(=O)C(C)C#N)CC2 97493,C1(C(N(CC(=O)OCC)C)=O)(CNC(=O)CN2CCCC2=O)CC12CCC2 97494,C(=O)(N=c1[nH]oc2c1COCC2)n1cc(C(=O)OC)c(O)nc1=O 97495,c1(C(C(=O)NCCCc2cncc(C(=O)OC)n2)(F)F)cc(Cl)nc(Cl)c1 97496,c1(C(=O)NC(C2CCN(C(c3ccc(Cl)nc3)=O)C2)C)cc2cc[nH]c(=O)c2s1 97497,C(C(CC)(CC)Sc1ccccc1)N(C)C.C12COCC1NC2=O 97498,C(=O)(C(C)(C)C(N)=O)NCC1C(NC(C2N(C(=O)NC)CCC2)=O)CCCC1 97499,N1(C(C(C(=O)OCC)OC)=O)CCC(CC)CC1C(=O)Nc1ccc(Cl)cc1 97500,C1(N(C(CC2CN(C(C)=O)C2)=O)Cc2coc(C)c2)CCN(CC(F)(F)F)C1 97501,C(=O)(CC1=CCN(C)CC1)N1CC(NC(N2CCC(C)CC2)=O)C(C(F)(F)F)C1 97502,C1(C(CC)NC(c2cnc(CC)[nH]2)c2nnnn2C2CC2)CCCCCC1 97503,c1(C(=O)NCC2C(C)CN(C(=O)CS(N)(=O)=O)CC2)cnc2ncc(Cl)cn12 97504,CCC(C)CCC(=O)OCCOC(c1cn(CC)c(C)n1)=O.C1(C)CCC1 97505,N1(C(CCN(C)CC)=O)CCN(C(c2ccncc2C)=O)C2CC12 97506,N1(C(CC=CC(C)(C)C)=O)CCC=C(C(=O)NCc2ncccn2)C1 97507,C1(C)(NC(C2C(CCC)C2)=O)CCN(C(c2ncoc2-c2ccccc2C)=O)C1 97508,c1(OC)cc(C)c2cc(C(=O)NCCc3nnc(C(F)F)o3)[nH]c2c1 97509,C1(C(N2C(CCNC(C(N3CCNC3=O)C)=O)CCCC2)=O)CC2(CC2)CN1C 97510,Cc1ccc(SCC(=O)NCC2C3CN(C(C4CCC(O)CC4)=O)CC23)cc1C 97511,c1(C(=O)NC2CC(CNC(C3CSCCS3)=O)C2)ncn2c1CCCC2 97512,N1(C(c2nc(CC)sc2)=O)CC2(CC2)CC1C(=O)NCC1(O)CCCOC1 97513,C1(C(N2C(CN(C(c3cnc(C(C)C)[nH]3)=O)C)CCCC2)=O)CCCC(=O)N1C 97514,Cc1cnc(F)cc1NC(=O)CN1CCC(C(=O)OC(C)(C)C)CC1 97515,NC(=O)CCC(=O)NCC1CCCCN1C(C1(F)CCOCC1)=O 97516,Cc1ncc(NC(=O)CCn2cc(-c3cc(F)ccc3F)nn2)c(C)n1 97517,C(C(C)(C)C#CC(=O)NC(c1cccnc1)CO)NC(CCc1c(C)noc1)=O 97518,N1(C(C(n2cc(CCN(CCOC)C)nn2)C)=O)CC(C)(C)OC(C)(C)C1 97519,N#Cc1ccc(NC(=O)C(=O)NC(C2CCCCC2)Cc2ccccn2)cc1F 97520,C(=O)(C#CC1CCC1)N1CCC(C(C)(C)NC(c2ccc(OC)nn2)=O)C1 97521,c1(C(N2CCCN(C(c3cccnc3)=O)CCC2)=O)cc(Br)c2occc2c1 97522,C1(NC(Cn2cccc(C)c2=O)=O)CC(N=c2[nH]cnc3cnccc23)C1 97523,C1(NC(c2c(C)c[nH]n2)=O)C(C)(C)CN(C(C2CCNC(=O)C2)=O)CC1(C)C 97524,C1(C)(CNC(c2c(CC)nc(C)[nH]2)=O)COCCN(C(C2CC(C(F)F)C2)=O)C1 97525,CC1(C)CC(c2nnnn2C2COC2)(NCc2scnc2Cl)CC(C)(C)S1 97526,c1(OC)cc(C(F)(F)F)cc(Cl)c1.N12CCCC(C1)CNC(=O)C1CC1C2=O 97527,C12(NC(C(CCC(C)C)O)=O)CCCC(CN(C(=O)CS)C1)C2.C1(O)CC1 97528,c1(C(N(c2ncc(F)cn2)C(C23CC(N)(C2)C3)=O)=O)cc(Cl)cnc1F 97529,c1(NC(CC2CC(C)N(C(C3CCC(O)C3)=O)C2)=O)cnc2c(c1)CCC2 97530,C1(C(N(CCCCNC(C(C2CC(F)(F)C2)OC)=O)C)=O)CCC2CC1CO2 97531,C12(CNC(CCC(=O)OC)=O)CCCC1CCN2C(c1ccsn1)=O 97532,N1(C(=O)NC2(C)CC(C(=O)OCC)C2)CC(c2ccc(OC)cc2)OC(C)C1 97533,c1(C(=O)NCC(C)CNC(c2ccc(F)c(F)c2)=O)cccc2c[nH]nc12 97534,c1(C(=O)NC(c2cn(C)nn2)C(=O)NCc2n(CCC)ncn2)ccc(Cl)cc1 97535,CCCC(C(=O)N1CC(CNC(C2CNC(=O)N2C)=O)C1)C(C)C 97536,c1(CCCC)cc(NCC2CN(C(C3CC4CCC3C4)=O)C2)n2ncnc2n1 97537,c1(C(N2CC(CNC(C(C(C)O)N(C)C)=O)C(O)C2)=O)ccc2c(n1)CCCN2 97538,N1(C(CC2(OC)CCC2)=O)CCC2CCN(C(=O)CC(O)CC(C)(C)C)CC2C1 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97731,N1(C(c2c(CC)[nH]cc2)=O)CC(NC(C2CC2c2cccc(Cl)c2)=O)CC(O)C1 97732,Cc1cc(Cl)ccc1NC(=O)C(C)(C1CCC1)NC(C1CC(CF)C1)=O 97733,N1(C(c2c(C)nc(Br)s2)=O)CCC(C)(NC(C2CC(CF)C2)=O)CC1 97734,c1(NC(C)=O)nc(CC(=O)NCC(C)CNC(=O)Cc2scc(C(N)=O)c2)cs1 97735,N1(C(C=C(CCC)C)=O)CCN(C(c2cncc(-n3cnnn3)c2)=O)C(CF)C1 97736,N1(C(Cc2cn(CC)nn2)=O)C(CNC(=O)COC(C)=O)CC2COCC12 97737,N1(C(C2CCCC(C)(C)C2)=O)CCC2(CCCCC2NC(=O)Cc2cn[nH]c2)C1 97738,Cc1cc(=NC(=O)C(=O)Nc2sccc2Cl)[nH]n1-c1ccc(Cl)cc1 97739,c1(C(=O)NC2(C)CCN(C(C(C)NC(C)=O)=O)C2)cc2cc(Cl)cnc2[nH]1 97740,c1(C(N2C(C(N3CC(C#C)C(O)C3)=O)COCC2)=O)cccc2c[nH]nc12 97741,C(=O)(C1CCc2c[nH]nc21)N(CCC(C(C)(C)C)NC(COCCOCC)=O)C 97742,C(=O)(C(C)C(C)C)NC(C(C)NC(c1n(CC)ncn1)=O)CO 97743,C(CCC(C)(C)C(=O)NCC(O)CC(C)C)NC(C(C)=CC(C)(C)C)=O 97744,CCCCCCCCC(=O)NC(CC)CCCC(=O)NCC12CCC(CC1O)C2 97745,C1(CNC(CC(C=C)C)=O)CC2CCC1N2C(c1ccc(CO)s1)=O 97746,Cc1cccc(Cl)c1C(N1CCC(C)C1CNC(=O)CCOCCN(C)C)=O 97747,C(=O)(C#CC1CCCCC1)N(C)CC1CCCCN1C(C1CC(O)CN1C)=O 97748,CCC(C)C(C(=O)NCCCCn1ccnc1)N(C(=O)CC(F)(F)F)C 97749,C1(C(N(CC(C)NC(=O)CCc2ccc[nH]2)CC)=O)CCCN1C1CC1 97750,n1(CC(=O)NC(CCOC)CNC(c2cc(OC)cnn2)=O)nc(O)ccc1=O 97751,C1(C(=O)NCCNC(C2(C(=O)OC)C(=C)CC2)=O)CCCCN1N=O 97752,c1(C(=O)NCC(C2N(C(C(COCC)C)=O)CCC2)(C)C)c(OC)cccc1Cl 97753,c1(NC(C(=O)Nc2cn(CC)nc2)=O)ccc(C(=O)N(CC(C)C)C)cc1 97754,CCCCCC(=O)NC(Cc1ccco1)C(=O)NCc1cc(C(N)=O)no1 97755,c1(OC)cc(N)c(Cl)cc1C(=O)N(C1CCN(C(C2(C)C=CCCC2)=O)CC1)C 97756,C=C1CON(C(=O)C23CC2CCN3C(=O)Cc2cccnc2O)C1 97757,C(N=c1nc2sccc2c(NC2CCCCCCCC2)[nH]1)C1(C)CC1(Cl)Cl.C1CCN1 97758,N1(C(C2(CC(=O)OC)CC2)=O)CCC(C(C)C(=O)Nc2ccccc2)C1 97759,CCS(=O)(=O)CCCCCN1CCC(N(C)C(=O)Nc2ccccc2)C1 97760,CON(CCC(=O)N(C)C)C(=O)NC(CO)CC(C)(C)C 97761,Cn1cc(C(=O)NCC(C2CC2)NC(c2cccc(=O)o2)=O)c(-c2ccoc2)n1 97762,C1(NC(C=C(C)C2CC2)=O)CC(CNC(c2cc(CO)c(C)o2)=O)C1(C)C 97763,N1(C(CC=C=C)=O)CC2CC(NC(=O)CS(=O)(=O)CCC)C(C2)C1 97764,CCCC(C(O)C(=O)NCc1cc[nH]n1)NC(c1cc(C)nnc1C)=O 97765,CCC(C)(C(=O)NCC1(C)CC(F)(F)CN1C(c1ccc(F)cc1)=O)C(N)=O 97766,C12(C(=O)NC3CC4(C(NC(c5ccc(SC)cc5)=O)C4)C3)CCC(C)(CC1)OC2 97767,N1(C(C(C2CCCCC2)C)=O)CCCC(C2CN(C(=O)C(F)(F)C(C)O)C2)C1 97768,O=C(NN1CCOCC1)N1CC2CCCCC12c1ccc(NC(=O)OC(C)(C)C)cc1 97769,c1(COC(c2ccc(-c3ccc(OC)nc3)nc2)=O)ccc(OC)cc1F 97770,C(=O)(CC(CC)C(F)F)N(CC(=O)NCc1cccnc1)CCC 97771,N1(C(c2oc(CC)c(C)c2)=O)CC2(CC)CC1(CNC(c1sccc1F)=O)C2 97772,C1(CC(=O)N(CC(COCC)O)C)CN(C(c2nnsc2C)=O)C(C)(C)C1 97773,c1(SCC(=O)NC2C3CC2CN(C(C2CCC2CF)=O)C3)cc(Cl)ccc1Cl 97774,C1(NC(C2N(CCC)CCC2)=O)CCCN(C(C2(CC)COC2)=O)C1 97775,c1(C(n2nc(-c3cccnc3)nc2N(C(=O)CO)CCF)C)cccc(Cl)c1 97776,Cc1cc(=NCCCCC2(C)OCCO2)[nH]cc1S(=O)(=O)N(C)C(C1CCC1)C 97777,CCS(=O)(=O)CC(=O)NCC12CCC(CN1C(=O)CC1CC(F)(F)C1)C2 97778,C1(C(=O)Nc2ncc(C)s2)COCCC1C1CCNCC1 97779,C(=O)(CC(C)(C)C#N)NCC1CN(C(c2ccc(C(C)C)cc2)=O)CC1C 97780,Cc1ncc(-c2cn(CC3CCCC(NC(=O)C(C)(F)F)C3)nn2)n1C 97781,N1(C(C2(CC=C)CN(C(=O)CC(C)CC(=O)OC)C2)=O)CC(C)(C)CCC1C 97782,C1(C2CCC2)(C(=O)NC(C)CCCNC(C2CCC=CO2)=O)CCC1 97783,CC(C)CC(C(=O)N1CCCC1CNC(N)=O)NC(=O)CN1CCC(C)C1 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97802,Cc1cc(C(=O)NC2(CNC(c3ccccc3Br)=O)CCOC2)cc(O)c1 97803,c1(C(=O)NCC(c2ccc(OC)cc2)NC(CN(C)CC)=O)cn(C)c(O)n1 97804,C1(C(=O)NC(CCNC(c2n(CC)ncc2Cl)=O)C)Cc2nnsc2S1 97805,C1(NC(C2(OC)CC2)=O)CCCCN(C(=O)CC2(O)CCCOC2)C1 97806,N1(CCc2ccc(OC)cc2Br)CCC(C2CC(OC)(OC)C2)C1 97807,n1(CC(=O)NCC(CNC(C(CC)c2cccnc2)=O)F)c([N+](=O)[O-])cnc1C 97808,c1(OC)cccc(CC(N2CC3CC2C3C(=O)NCc2cccc(F)n2)=O)c1 97809,C1(c2nc(C)[nH]n2)COCCN1C(c1ccc(Br)cn1)C(=O)NCC(C)C 97810,Cc1ccc(F)c2oc(C(=O)NC3CCC(N4CCN(C(=O)CO)CC4)C3)cc12 97811,c1(C(=O)NC)ccc(C(=O)NC2CCC2NC(c2cc(O)ccc2Cl)=O)cc1F 97812,C1(C(CC)C)CCN(C(=O)C(CCC2CCC2)NC(=O)CCCCOCC)CC1 97813,n1(CC(=O)NCCCOCCNC(=O)Cc2cc[nH]n2)cc(CO)nn1 97814,C1(NC(Cc2c(C)nc(C)s2)=O)CCC(C)N(C(c2cncs2)=O)C1 97815,CCCC(C)(O)C(=O)NCCCCCCNC(=O)CNC(c1ccc(C)cc1)=O 97816,N1(Cc2cn(CCNC(=O)CCc3nc[nH]n3)nn2)CCC(F)(F)CC1 97817,O=C(C1=CSCCO1)NCC1(CNC(c2ccc([N+](=O)[O-])o2)=O)CC1 97818,N1(C(C=CCC2(N(C)C(C3CCC3C)=O)CCC2)=O)CCCCC1CF 97819,CCC(C(=O)N(CCCNC(=O)CC1CC(F)C1)C)NC(N)=O 97820,N1(C(c2cnn(-c3ccccn3)c2)=O)CC2CCCC(C1)C2(F)F 97821,C1(CC)C(=O)NCCN1C(=O)C(F)C(C)CNC(=O)COc1cnn(C)c1 97822,c1(CN(C2CC2)Cc2nc(C3C(C)N(C)CC3)on2)c[nH]c2cccnc2c1=O 97823,C(=O)(C1=NOC2COCC12)NCC1CCC(C(=O)NC(C)C(C)(C)C)O1 97824,N1(C(CC=CCCCCC)=O)CCC(C)(C(=O)N(C2CC3(CCC3)C2)C)C1 97825,c1(C(=O)NCc2c(C(N3C(COC)CCC3)=O)c[nH]n2)cncc(C)c1 97826,N1(C(C(C)C(F)F)=O)CC(NC(=O)CC2CC(C)(C)C(=O)N2)CC12CCCCC2 97827,N1(C(C2CCN(C)C2=O)=O)CC(C2CCN(C(c3ncn4c3CCC4)=O)CC2)C1 97828,Cc1cccc(C2(C(=O)NC(C3CCN(C(C4(O)CCSC4)=O)C3)C)CC2)c1 97829,C1(CN(C2CSCC(=O)N2)C(C2N(C(C(N)=O)=O)CC(O)C2)=O)CN2CCN1CC2 97830,CN1CCC2C(CCCN2C(c2cn(C)nn2)C(=O)NC2COC2)C1 97831,Cc1noc(C2CN(C(=O)CC(C)N(C(=O)C(C)OCCN(C)C)C)C2)n1 97832,Cc1cc[nH]c(=N)c1C(=O)NCC1(C)CCN(C(c2c(C)nc(C)n2O)=O)CC1 97833,C1(NC(C2CC(CCC)(CC)C2)=O)CC2CC(NC(=O)C(F)(F)C3CC3)CC2C1 97834,C1(C(N(C2CCN(C(c3n[nH]c(O)n3)=O)C2)CCO)=O)CCC2CC2C1 97835,C(=O)(CCC(=O)NC(C)C)NC(C(c1ccccc1)NC(c1cnc(C)s1)=O)C 97836,C1(CC(=O)OCCCC(=O)NC(c2nccn2C)C)NC(=O)OC1C 97837,N1(C(c2c(CC(C=O)(C)C)cnnn2)=O)CCN(C)C(COC)C1.CCO 97838,c1(OC)cccc(C(F)F)c1C(N1CCC(NC(=O)C(C)(C)CF)C(CO)C1)=O 97839,n1(CC)nccc1C(=O)NCC1CC1CNC(=O)CNC(c1cnn(C)c1)=O 97840,c1(C(C(=O)NCC=C)N(C)Cc2cnn(C3CC3)c2)cccc(O)n1 97841,C=C=CC(C)C(=O)NCC(C)(C)OCC(=O)Nc1ccc(O)nc1 97842,CN1CCC2(CCN(C(C3C4CCC(C4)N3C(=O)CCC(F)(F)F)=O)CC2)CC1 97843,CC(C)C(O)C(F)(F)C(=O)NCC1CC(F)CN1C(C1CC2CCC1CC2)=O 97844,C1(C(N(CC(=O)NC2CCN(CC3CC3)C2)C)=O)CC2(CCO1)CC2 97845,n1(CC)nc(C(=O)NC(C2CCN(C3CCN(C4CCC4)C3=O)C2)C)c(C)n1 97846,c1(CC)cnc(C(N2CC(NC(c3ccc(NC(C)C)cc3)=O)CC2C)=O)cn1 97847,c1(SC)ccccc1C(=O)NC1CC(F)(CNC(=O)C(C2CC2)SC)C1 97848,CC(C)C(C(C)C)NC(=O)NCC1CCC(C)C1 97849,C1(COC)CCN(C(=O)C(CC2CCC2)NC(c2ccns2)=O)C1 97850,c1(C(N2CCC(N(C(c3cnn(C)n3)=O)CCO)C2)=O)cnn(C)c1Br 97851,C1(C)(C(=O)NC(c2cccnc2O)C)C=CCN1C(c1cc(C2CC2)[nH]n1)=O 97852,C(=O)(CCC(N)=O)N(C1CCN(C(=O)C(CCSC)N(C)C)C1)CC 97853,c1(C(=O)NC(C2CCN(C(=O)CSc3ccccc3)C2)C)ccc2scnc2c1 97854,c1(C(=O)OC)ccc2cnn(CC(N3C4CSCC3CC(=O)C4)=O)c(=O)c2c1 97855,CC1CC=CCC1C(=O)NC(c1cnn(C)c1)C(=O)NC1CCC(F)CC1 97856,N1(C(CS(CCC)(=O)=O)=O)CCCC12CCN(C(c1ccccc1[N+](=O)[O-])=O)C2 97857,N#CC1(C(N2CCCCC2C(=O)NC2CC(NC(N)=O)C2)=O)CC2CC2C1 97858,c1(NC(=O)C(N2CCC(c3nccs3)C2)c2cccs2)ccc(F)cc1 97859,N1(C(C=C)=O)CCC2(CCC2)C(NC(C2CCc3cncn3C2)=O)C1 97860,Cc1noc(CCNCC(=O)Nc2ccc(CN3CCOCC3)cc2)c1C 97861,c1(Cc2cn(CC(CC)O)nn2)ccc(Cl)cc1.C1(C)C(=O)N1C1CC1 97862,N1(C(C(C)CCN(C)C)=O)CCc2nc[nH]c2C12CCN(C(=O)C#CC1CC1)C2 97863,C=CCC(Cc1ccccc1)N=c1nc2c(ncn2C)c(NC2C=CCCC2)[nH]1 97864,C1(CNC(C2C3C4CCC(C4)C23)=O)CCCC2CN(C(=O)CC3(O)CCC3)CC12 97865,N1(C(C2(CC#C)CCOC2)=O)CC(C)N(C(=O)CC2CC(C)(C)C2)C(C)C1 97866,c1(C(=O)NCCn2cc(CCCC(O)c3cccs3)nn2)ccc2nccn2c1 97867,N1(C(C=Cc2ccc(C)o2)=O)CCOCC(CNC(c2c(C)cnn2C)=O)C1 97868,N1(C(C2(CC=C)CC=CC2)=O)CCN(CC(=O)NC(c2nn(C)cc2O)C)CC1 97869,CC(C)(C(=O)NCC(C1CCCC1)NC(=O)Cc1cnc[nH]1)Oc1ccccc1 97870,C12(C(=O)NC3C(CNC(C(C)OCCCC)=O)C3)CC3CC1C2C3O 97871,C1(C2CCOCC2)(C(N2CC(CNC(=O)CCc3ccccn3)C2)=O)CC1(F)F 97872,S(=O)(=O)(c1cc(C(N)=O)co1)N1C(C)CCCC1 97873,c1(CC(=O)Nc2c(OCC(C)C)cccc2)csc2nc(-c3ccccc3)cn12 97874,C1(C(N2CC(NC(N)=O)C2)=O)CCCC(NC(c2cccnc2)=O)CC1 97875,C1(NC(c2nc(Cl)sc2Cl)=O)CCCCN(C(C2CN3CCC2CC3)=O)CC1 97876,N1(C(c2nc(COC)sc2)=O)CC2CC1C2CNC(c1n[nH]cc1F)=O 97877,Cc1ccc(F)c(CNC(C2(C)CCCN2C(=O)CCN2CCCC2=O)=O)c1 97878,c1(NC(C2(C)CCN(C(C=C(C)c3ccco3)=O)C2)=O)c(O)cccc1O 97879,c1(NC(=O)C(=O)NCC2CN(C(C3CC4CCC34)=O)C2)cccc(C(F)(F)F)c1 97880,c1(OC)c(C(=O)NCC(C)(C)CNC(=O)CCCc2ncc(C)o2)cccc1N 97881,n1(CC)cnc2c(NC3CC(NC(=O)COCC4CC4)C3)ncnc12 97882,C1(NC(c2ccc(C)cc2)=O)CN(C(=O)C(C2CCCCC2)N(C)C)CC1(C)C 97883,C1(CC(=O)NC(C2CCN(C(=O)CC3CCCC3C)C2)C)CN2CCN1CC2 97884,c1(CC(=O)NC(CC)(C)CNC(c2n[nH]cc2Br)=O)ccc(F)c(F)c1 97885,c1(C(=O)NCCCN(C(C(C)OCC2CCCO2)=O)C2CC2)ccc(=O)n(C)n1 97886,C1(C(N2CC3CCC(CC)(C2)C3)=O)Cc2c[nH]nc2CN1C(=O)OC(C)(C)C 97887,Cc1cc(C2CCCN2C(=O)NC(c2cccc(Cl)c2)CF)c(C)o1 97888,c1(C(=O)NCCC(CC)(CC)NC(=O)C(F)=C2CCC2)nn2cccnc2c1Cl 97889,N1(C2CCC(NC(C3(C(N)=O)CC3)=O)C2)CCN(C(=O)C=Cc2cnc[nH]2)CC1 97890,C#CC1(NC(=O)C(CC(C)CC)NC(c2coc(C)n2)=O)CCCCCC1 97891,N1(C(CNC(C(CC)C)=O)=O)CC2C(NC(=O)CCCCN3CCCC3=O)C2C1 97892,c1(CC)c(C(=O)NCC2CC(C)N(C(c3cnn(C)n3)=O)C2)cccc1C 97893,C1(NC(c2c(C)nn(C3CC3)c2)=O)C2CC3CN(C(=O)C(C)(F)F)C1C3C2 97894,c1(C(=O)NC2(CN(C(=O)Cc3cn[nH]c3)C)CC2)cc2cccc(Br)c2o1 97895,c1(COC(C)(C)C)cc(C(=O)NC2CCC2NC(c2csnn2)=O)no1 97896,C(=O)(C(C#N)CC1CC1)NCC(C)(C)NC(C1CC(CCC)C1)=O 97897,c1(CC(=O)NC2C(NC(Cc3cc(C)ns3)=O)COC2)cccc(C(C)C)c1 97898,C1(NC(c2c(OC)cc(C)cc2)=O)C(C)CCN(C(=O)C(C)C2CCOC2)C1C 97899,C1(CC)CCNCC1.c1(Cn2ncnc2C(C2CCCCN2)C)nn(C)cc1C 97900,c1(C(=O)NCC2CC(NC(C=CCC)=O)C2(C)C)ccc2c(n1)OCCO2 97901,C1(C(N(CC(CC)NC(c2cscc2C2CC2)=O)CC)=O)CCC(C)(C)C1 97902,Cc1cccc(F)c1CNC(C1CCCN(C(C2CC2C)=O)C1)=O 97903,CCC(C)(CO)C(=O)NCc1cccc(CNC(C2CC3(C2)CC3(F)F)=O)c1 97904,c1(C(N2C(Cn3cc(COC)nn3)CCC2)=O)ccc(S(F)(F)(F)(F)F)cc1 97905,CC1CC2(CCN(C(c3ccc(Br)cc3Cl)C(=O)NCc3ccco3)CC2)CO1 97906,N1(C(C(C)CF)=O)CC2CC(NC(=O)CSCc3ccccc3Cl)C1C2 97907,N1(C(C(=C(C)C2CC2)F)=O)CCCN(C(=O)CC2(C)CCS(=O)(=O)N2)C(CO)C1 97908,C1(NCC(C)(O)C2(C)CC2)CC(=O)N(O)C1.C12CCN1C(=O)C2 97909,CC(c1ccccc1)=CC(=O)NCC1(O)CCN(C(c2nnsc2SC)=O)C1 97910,c1(COC)csc(C(=O)NCC2(CO)CN(C(=O)C(F)=C(C)C)C2)c1 97911,C(=O)(CCC(=O)CCC(=O)c1ccsc1)NCCC.c12c(cccc1C#N)C(=O)N2 97912,C12(CNC(=O)CCn3ccnn3)CCC1CN(C(c1coc(Br)n1)=O)C2 97913,C1(NC(c2cccc(C)c2Cl)CO)CCCCC(O)CNCC1 97914,CC1CN(C(=O)C(C)NC(=O)OC(C)(C)C)CCN(C(C2CCCN2C)=O)C1 97915,S(=O)(=O)(c1ccc(NCC2(C)CC2(F)F)c(Cl)c1)N1CCCC2(CC(OC)C2)C1 97916,C1(N(C(c2cc(CC)sn2)=O)C)CCC(NC(C2CCCC2C)=O)CC1 97917,c1(C(N2C(C(=O)NC3CC(C(=O)OC)C3)CC2)=O)cnc(C2CC2)nc1 97918,C12(NC(C(c3ccc(C)cc3)C)=O)CCC1CN(C(=O)CN(C)C(C)C)C2 97919,CC(=O)CCCC(=O)NCC(=O)NCCCN(c1noc2c1CCC2)C 97920,c1(C(=O)NCCN(C(=O)C(C)(CC)CO)CCC)ccc(Cl)nc1OCC 97921,N1(C(C2N(C)CCCC2)=O)CCC2(CC(NC(c3cc4n(c3)CCOC4)=O)C2)C1 97922,c1(OC)cc(N(C)CC2CCN(C(=O)CC3COC(=O)C3)C2)nc(OC)n1 97923,c1(C(N(C)CCNC(c2ccc(=N)[nH]n2)=O)=O)ccc2oc(O)nc2n1 97924,C1(C(N2CC(CC)(CC)C2)=O)(CF)CCN(C(=O)CC2CC2COC)C1 97925,C1(CC=C)(NC(=O)CCCNC(C)=O)CC2CCC(C1)N2C(c1cnn(C)n1)=O 97926,CC(C)C(F)(F)CC(=O)N1CCN(C(C2CC(CC(F)(F)F)C2)=O)C(C)C1 97927,N1(C(=O)CCc2nc[nH]n2)CCN2C(=O)NCCC2C1 97928,C(=O)(CCN=C(NCc1cccc(C)c1C)NCC12CCC(C)(CO1)C2)NC 97929,CC1CN2CCN1CC2C(=O)NCCC(C)N(C)C(c1ccccc1N(C)C)=O 97930,C(=O)(CCC(CC)OC)NC(CCCNC(C1(COCC)CCC1)=O)C 97931,c1(CC)ccc(OCC(N2CCCC2CCNC(=O)Cc2nnc(C)s2)=O)cc1 97932,N1(C(c2csc3ccccc23)C(=O)NC(CC)C)CC2CCC(C1)C2(F)F 97933,Cc1ccc(SCC(=O)NCC(C)NC(c2cc(C)nn2C2CCC2)=O)cc1 97934,c1(C(C)C)ncncc1C(N1CCN(CC(C)NC(=O)CC2(C#N)CC2)CC1)=O 97935,C1(CN(C(c2cn(CCC(C)C)nn2)=O)C)C2CN(C(=O)C(CO)N(C)C)CC12 97936,C1(NC(CC(C)C)=O)CC(NC(c2ccc(O)c(C(C)C)c2)=O)C12CCOCC2 97937,C1(NC(=O)CCN2CCOC2=O)CN(C(C2CC3(C2)CC32CC2)=O)CC12CC2 97938,c1(C(=O)NC2CN(C(c3c(C)cc(N)cc3)=O)CC2F)cccc2c[nH]nc12 97939,C1(NC(CCN(C(C)=O)C)=O)CCN(C(=O)CSc2nncn2C)CC1C 97940,c1(CC(N2CC(CNC(=O)C(O)C3CC3)OCCC2)=O)ccc([N+](=O)[O-])cc1 97941,CC(C)C(C(=O)NCCOC1CC1)C(C)NC(C1CC(F)(CF)C1)=O 97942,C=CCC(C)(C)CCNC(C1CCOCCN1C(=O)Cc1ccco1)=O 97943,N1(C(C2CC(=C)C2)=O)CCOC2(CCS(=O)(=NC(=O)C3(C)CCCC3C)CC2)C1 97944,C1(C(N(C(C)C(=O)NCCCC(C)CO)C2CC2)=O)CCC(=O)N(C)C1 97945,C(C)(C)(CCC(=O)N1CSCC1C(=O)NCc1snnc1C)OC 97946,CC(C)C(F)(CNC(C1(Cl)CC1(F)F)=O)C(=O)N(C)CC1CCCCCC1 97947,N1(C(CC(C(C)C)C)=O)CCC(CNC(=O)CCCCN2CCCC2)C(F)(F)CC1 97948,C1(NC(NCC2(CO)C(C)(C)C2)=NCCCOCCO)CCc2ccccc2C1 97949,CC(=O)CCC(=O)N1CC(NC(C2(c3ccccc3Br)CC2)=O)CC1C 97950,c1(C(c2nnnn2C)NCc2n(CC)ccn2)cncc(-c2cccc(F)c2)c1 97951,C1(C(=O)NCC2N(C(C(C)(C)C(N)=O)=O)CCC2)CN2CCCC2CO1 97952,C1(C(=O)NCCn2c(CC)nnc2)C(C)CCN1C(c1cncc(F)c1)=O 97953,N1(C(C(CC)NC(N)=O)=O)CCC(OCCCNC(=O)C=CC(C)CC)CC1 97954,C(=O)(C1CCCn2nccc21)N1CC(CNC(c2ccc(=O)n(CCO)c2)=O)C1 97955,N1(C(c2cc(C)c(C)nn2)=O)CC(NC(c2cnn(C)c2)=O)CC12CCCOC2 97956,C1(NC(C(CNC(c2nnc(O)nc2O)=O)O)=O)CNC(=O)C12CC2 97957,N1(C(c2c(CC)ncs2)=O)CCC(C(N2CC(NC(N)=O)C2)=O)CC1C 97958,CC(CCNC(C1CCCCC1)=O)CCNC(=O)CCN(c1ccc(Cl)cc1)C 97959,c1(COC)cc(N2CCCC(C3CCCCN3C(C3CC3C(C)O)=O)C2)ncn1 97960,N1(C(C)=O)C2CCC1CC(C(N1CCCC(C(N)=O)(N(C)C)C1)=O)C2 97961,Cc1noc2ncc(C(N3CC(CNC(c4cc(F)cc(Br)c4)=O)C3)=O)cc12 97962,C12(C(=O)NCCC3CN(C(COCC=C)=O)CC3C)CCC(N(C)C)(CC1)CC2 97963,C1(NC(c2cccc(COC)n2)=O)CN(C(C2CC2C)=O)CC(C)(C)C1 97964,C1(C(=O)NCc2c(OC)nsc2)C(C)OCCN1C(=O)CC1CCN(C)C1=O 97965,N1(C(c2c(C)cc(CO)o2)=O)CC2(CNC(=O)C(C3CCOCC3)O)CCC1C2 97966,c1(CC)nc(N(C)C)co1.C1(C(=O)N(S)C)C(C)CN1C(=O)OC(C)(C)C 97967,N1(C(C2(CCC=C)CC2)=O)CCC2(CC1)OCCC2NC(=O)CC(F)F 97968,N1(C(C23CCCC2C3)=O)Cc2cc(Cl)ccc2CC1CO 97969,C1(CNC(C=CCC)=O)(CO)CCCN(C(=O)C(C)OCCCCCC)C1 97970,c1(C(=O)NC2(CF)CCN(C(C(C)(C)c3cc[nH]n3)=O)C2)cc2c(s1)CCC2 97971,O=C1OC(CNC(c2cccs2)C2CC2)CCC12CC2 97972,c1(N2CC(NC(C)=O)C2)cccc(CCC(=O)NC2C3COCC23)c1 97973,C1(NC(C(C)n2cncn2)=O)(CO)CCN(C(=O)CC2(CN(C)C)CCC2)C1 97974,C(=O)(CCC(F)(F)Cn1cc(CC(O)C2CC2)nn1)N(C)Cc1cc(Cl)sc1Cl 97975,C12(CNC(c3scc(C)c3)=O)CCCC1N(C(=O)CNS(C)(=O)=O)CCC2 97976,C1(CC(=O)NCCC(=O)NCC#C)CCCN(C(=O)C(C)SC(C)C)CC1 97977,C=CC1(C(N2CCC(O)(C(N)=O)C2)=O)CCN(C(c2ccc(Cl)o2)=O)C1 97978,c1(C(=O)NCCCNC(=O)C=CCN2CCCC2)c(Cl)csc1Cl 97979,CC1(C)CC(CNC(=O)Cn2cccn2)N(C(C2CCC(C)(C)O2)=O)C1 97980,C1(C(N2CCC(NC(C(C)=C3CCC3)=O)C2C)=O)CCOC2(CCC2)C1 97981,C(CCN(C)C)(C(=O)NC1COCCC1O)NC(C1C(C)=CCS1)=O 97982,CCCC(CCCNC(=O)C=Cc1cocn1)NC(=O)CC1(C)CCC1 97983,c1(C=O)cc(=N)[nH][nH]1.C(C(C)(C)O)N1C(=O)CC2(CC2)C1.CO 97984,C(=O)(C(C)C(F)(F)C(F)F)NCC(CNC(c1ccc(C(C)C)nc1)=O)(C)O 97985,c1(C(=O)NC2CN(C(c3c(CCC)nco3)=O)C2)ccc(O)c2c1CCCC2 97986,c1(NCCC(CC)O)ccc(S(=O)(=O)N2CCOC(C(C)(C)OCC)C2)cc1Br 97987,N1(C(c2cc(CNC(C(c3cncnc3)C)=O)no2)=O)CC2CCC(CC2)C1 97988,N1(C(C(C)C)=O)CCCC(C2(NC(C3CC(OC(F)F)C3)=O)CC2)C1 97989,C1(NC(C(N2CCC(C)CC2)=O)=O)CC2CCC1N(C(=O)C(C)C(C)O)C2 97990,CCC(C)(C)C(C)CC(=O)N1CC(NC(c2cc(C(C)(C)C)c[nH]2)=O)C(F)C1 97991,C(=O)(CCCN(C)N=O)N1C(C(C)NC(C2CC3C(C2)C3(F)F)=O)CCC1 97992,CC(C)(CN=c1ccnc(C2CC2)[nH]1)NC(=O)CCCCc1cnn[nH]1 97993,c1(OC(C2C(C)(C(=O)Nc3ccc(C(=O)OC)cc3)C2)=O)ccc(Cl)c(Cl)c1 97994,O(S(=O)(=O)c1cc(Br)ccc1Br)c1ccc(CC)cc1Nc1ccc(OC)cc1 97995,N1(C(c2c(OC)csc2)=O)CC2CCCCC2(CNC(=O)C(C)(F)F)C1 97996,N1(C(C(C2CC2)OC)=O)CCCC1C1CCN(C(C2CC(C(F)(F)F)C2)=O)C1 97997,Cc1c(Br)noc1C(N1CCC(O)(CN(C(=O)C2=C(Cl)CC2)C)C1)=O 97998,S(=O)(=O)(c1c[nH]ccc1=NCC1CCS(=O)(=O)N1C)NC(C)Cn1ccnc1 97999,C1(C(=O)NC(C)CF)C2CCC(C2)N1C(c1ncccc1Cl)=O 98000,c1(C(N2CCC(N(C(C3CC3C)=O)CC)C2)=O)ccc2oncc2c1 98001,C1(C(=O)Nc2cnc(I)cn2)CN(C(c2cccc(CO)c2)=O)CCC1O 98002,C1(C(=O)NCC(F)(F)F)CCCN1C(=O)NCc1ccccn1 98003,c1(C(NNC(C2COCCN(C(C)=O)C2)=O)=O)ccc(Cl)c(Cl)c1F 98004,c1(C(=O)NCC(C)CN(C)C(C2CC(F)(CF)C2)=O)c(C#N)ncn1C 98005,C1(NC(c2cc([N+](=O)[O-])c[nH]2)=O)CC2CCC1N(C(=O)Cc1ccno1)C2 98006,c1(C(N(CCC(C)NC(c2ccc(C3CC3)o2)=O)C)=O)ncccc1Br 98007,C(CNC(=O)CC1CCCOC1)(CC(=O)NOCC(=O)OC(C)(C)C)OC 98008,c1(OCC(=O)NC2CC(NC(C3C=CCC3)=O)C(O)C2)cccc(Br)c1 98009,C1(CC(N2CCC(CCNC(=O)CN3CCCNC3=O)C2)=O)CC2C=CC1CC2 98010,N1(C(CCOCC#C)=O)CCCC(CCNC(c2cc(CC)[nH]n2)=O)C1 98011,Cc1nc(NCc2n[nH]c3c2CCC3)cc(=NCCc2nccn2C2CC2)[nH]1 98012,C=CC1(CC(N2CC(CO)(CF)C2)=O)CN(C(C2CCC(C)C2)=O)C1 98013,C1(CN(C(=O)Cn2cccn2)C)CCCN1C(C1(CF)CC1)=O 98014,CC1(C)CC(CO)CN(C(C2CC=CCN2C(c2ccc3cncn3c2)=O)=O)C1 98015,C#CCCCC(=O)N1CCCC1C(C)NC(C1CC=C(C)CC1)=O 98016,c1(C(N2C(C(N3C(COC)CCCC3)=O)CC2C)=O)cc2cccnc2[nH]1 98017,c1(CNC(C(CC=C)C)=O)ccc(CNC(C2CC(C)N(C)C2)=O)c(F)c1 98018,Cc1cc(C(=O)NC2CC3(C2)CC(C(=O)Nc2cc(I)ccc2C)C3)cc(O)n1 98019,CC1CC=C(C(=O)N2CC(C)(C)CC2CNC(c2sccc2C(C)(C)C)=O)CC1 98020,C1(CNC(C(c2c(OC)cccc2)C)=O)CCC2(CN(Cc3cnn(C)c3)C2)O1 98021,N(C(=NCCC1CCCCO1)NCC1CCC1)CC1(F)CC1 98022,C1(CNC(CC2(C)CC2(F)Cl)=O)CC2(CO1)CN(C(=O)COCCCN=[N+]=[N-])C2 98023,C1(CNC(c2cc(C)ns2)=O)CCC2(CCN(C(C3(C)CC(F)C3)=O)CC2)O1 98024,N1(CC(=O)NC(CC)CN(C(C2(OC)CCC2)=O)CC)CCC(C)C1 98025,N1(C(C(CCCOC)C)=O)CC(C)CN(C(c2ncn3ccccc23)=O)C(C)C1 98026,C1(CNC(C2C(C)(C)C2)=O)CCCCCN1C(=O)C=Cc1cc(Cl)sc1Cl 98027,C1(CC)CC(O)CN1C(c1occc1CNC(=O)Cn1cnnc1)=O 98028,C1(C2CC2)(C(N(CC=C)C)=O)CN(C(=O)CC2CCC(C)C2)C1 98029,CC1CC2(CO1)CN(C(c1coc3c1CN(C(=O)COCC1CC1)C3)=O)C2 98030,c1(C(N2CCC(NC(CC3C=NN(C)C3=O)=O)(CO)CC2)=O)cc2ccncc2s1 98031,c1(C(N2C(CC)CCOCC2)C(=O)NCCCF)c(C)nn2cccnc12 98032,c1(NC(=O)NC2CCc3c[nH]nc3C2)nc2ccccc2cc1[N+](=O)[O-] 98033,C=CCCC(C)(C)C(=O)N1CC2CC2(CNC(c2ccnc3[nH]nnc23)=O)C1 98034,c1(CC(=O)OC(c2ccc(OC)cc2)CC)c(F)cccc1F 98035,c1(C(=O)NCC2C(CNC(c3ccc(SC)cc3)=O)C2)cc(C2CC2)nc(Cl)c1 98036,C1(CC=C)CCCCC1(c1nnnn1CCCF)NC1COCCOC1 98037,C(=O)(CC(C)C(C)(C)C)NC(C1CCCC1)CNC(c1nc(CC)sc1N)=O 98038,c1(OC)cc(C(=O)NCCC2(O)CN(C(c3cc(Cl)ccc3O)=O)C2)cc(Cl)n1 98039,C1(CC(=O)OC)C(C(=O)NCC(c2ccccc2)(C)F)C1(C)C 98040,CC1CC(C(=O)N(C2CCCCCC2)CCNC(c2cncc(F)c2)=O)C(=O)O1 98041,N(C1CC(C)n2ncnc21)C(C1CCCN(C(CCOC(CC)C)C)C1)=O 98042,C1(NC(Cc2nc(C(C)C)on2)=O)CC(F)CN(Cc2ncccc2C(F)F)C1 98043,c1(-c2ccc(C(C)=O)cc2)cnc2ccc(C(=O)NC3CCCN(C(C)=O)C3)cn12 98044,N1(C(C(C(C)C)OCC)=O)CC(NC(=O)C=CS(C)(=O)=O)CCC1C 98045,CC(CN(C)C)CC(=O)NC1(CNC(c2cnc(Cc3cccs3)s2)=O)CCC1 98046,N1(C(CCC#CC)=O)CCC(NC(=O)C(C)NS(=O)(=O)CCCC)C(F)(F)CC1 98047,N1(C(c2cnc(C(C)C)[nH]2)=O)C2CCC1CC(CNC(C1CC13CC3)=O)C2 98048,C(C(C)(CO)NC(=O)CCC1(C)CN(C(C2CCN(C(C)C)C2)=O)C1)OC 98049,c1(CC)ncncc1C(N1CCN(C(CNC(C2CC(O)C2)=O)C(F)F)CC1)=O 98050,c1ccc(Cl)cc1.C(=O)(CCCOC(=O)C(c1c(C=O)cno1)OC)OC 98051,C(CCCC(=O)NC(C)(C)CN=[N+]=[N-])N(C(=O)C=Cc1ccccc1)C 98052,C(C(=O)Nn1cnn(C)c1=S)N1CC2(N(C(CCCC#CC)=O)CC2)C1 98053,N1(C(C(CC(C)C)(C)C)=O)CCC2(CCC2NC(c2ccsc2Cl)=O)CC1 98054,CC1CN(C(C2(O)CC3CCC2C3)=O)CCC1CNC(=O)CC1CCCCC1O 98055,C1(C(=O)NCCCN(C(C2N(CCC)C(=O)CC2)=O)C)CC2(CCCCC2)CO1 98056,C1(CN(C(CNC(C)=O)CC)C(c2c(CC)noc2)=O)NC(=O)NC1=O 98057,c1(CC)nnc(N2CCC(OCCNC(=O)Cn3cnnn3)C2)o1 98058,N1(C(C(CCC2CCC2)NC(C(C(CC)C)N(C)C)=O)=O)CCOC(C)(C)CC1 98059,C(C)(CO)(C(=O)NC1CCN(CCNC(=O)CC2CCCCC2C)CC1)OC 98060,C1(O)(C(N2CC(NC(c3cnc(SC)s3)=O)C2)=O)CCCCCC1 98061,CC1(C#N)CC2(CC(c3nnnn3CC(F)F)(NC3(CF)COC3)C2)C1 98062,C1(NC(CCCC(=O)NCC)=O)CCN(C(c2ncc(F)cn2)=O)C12CCC2 98063,CCOC(C)(C)c1ccc(NCCSCC(=O)NC(N)=O)cc1 98064,N1(C(C(C)Cn2cccn2)=O)CCOC2(CCN(C(=O)C(=O)NC3CC3)C2)C1 98065,C=CCCC(C)(C)C(=O)NC1CCCC1NC(=O)C(CC)NC(N)=O 98066,c1(C(=O)OCCSc2n(C)cnc2)cc(NC(=O)OC(C)(C)C)ncn1 98067,N1(C(C(CNC(C(c2ccccc2)OC)=O)C(C)C)=O)CCC12CCC(O)CC2 98068,C1(N(C(=O)CCC2CC2CC2CC2)C)CCCN(C(C2(C(N)=O)CCC2)=O)CC1 98069,C(=O)(CCC(C)(C)N(C)C)N1C(C(=O)NC(c2nc(C)[nH]n2)(C)C)CC1C 98070,C(=O)(C1CCc2c[nH]nc21)N1CC(CC(=O)NCc2cnns2)(OC(C)(C)C)C1 98071,CC(c1ccccc1F)=CC(=O)N(CCN(C(=O)CCC(C)N(C)C)CC(C)O)CC 98072,N1(C(c2cccc(CC=C)c2)=O)CC2(C(=O)N(CC(C)C(F)(F)F)C)CC1CO2 98073,Cc1cc(C(N2C(C(=O)NCC3(CO)CC4CC4C3)CCC23CC3)=O)nc(C)c1 98074,CC1=C(C(=O)NC2CC(CNC(=O)Cn3ccc4ccccc34)C2)CCS1(=O)=O 98075,c1(NCC(CN(C(CNC(C)=O)=O)C)C)c(C#N)cnc2c(C)cc(F)cc12 98076,C1(CNC(C2(CC(=O)OC)CC2)=O)CCCN(C(=O)Cc2nocc2C(C)C)C1 98077,C1(NC(c2cc(CNC(CC3N(C)CC=CC3)=O)on2)=O)CCc2nncn2C1 98078,Cc1csc2cc(C(=O)NC3CC3NC(c3cc(F)cc(F)c3)=O)[nH]c12 98079,Cc1cc(Cl)c(C(N2CCN(C(=O)CC3OCCCC3(C)C)CC2C)=O)cc1N 98080,c1(C(=O)NCC(=O)NCC(C)CN(C)C(c2ccc(F)nc2)=O)ccc(N)cc1 98081,N(C1CCCc2n[nH]cc21)C(C(CC)(C)CNC(c1c[nH]nc1OC)=O)=O 98082,c1(C(=O)NC2CCC(NC(c3n(CC=C)ccc3)=O)CC2)ccc(SC)cc1Cl 98083,N1(C(C(C)=C(C)C)=O)CCN(C)CC1CNC(=O)C(O)C(F)(F)F 98084,c1(C2(C(=O)NCC3CCN(S(C)(=O)=O)C3)CCCC2)cc(F)ccc1F 98085,C12(C(N3CC(C(=O)N(C)Cc4cc[nH]n4)(CC)C3)=O)CCCC1C2(F)F 98086,c1(C(=O)NC2CCCN(C(c3n(CC)c(O)nc3)=O)C2)cc(F)cc(F)c1 98087,N1(C(CCCC#N)=O)CCCCCC1CNC(=O)CCCn1ccnn1 98088,C(c1ccc(Cl)cc1)(C(F)(F)F)=CC(N1CCN(C(C(C)O)=O)C2(C1)CCC2)=O 98089,C1(=CC(=O)NCC=CCNC(CN(C)C(N)=O)=O)CCC(C(C)(C)C)CC1 98090,CCC(C)C(O)C(C)C(=O)N1CCOCC1CC(=O)NCCSC 98091,N1(C(c2ncn(C)n2)C(=O)NCCCC)CCN(C2CCOCC2)CC1 98092,C1(C(=O)NC2CCCCC2O)(CNC(c2c(CC)ocn2)=O)CC(C)(C)C1 98093,c1(C(=O)NCCC(C)NC(=O)CC2COC(=O)C2)cncc(C(F)F)c1 98094,C1(C(N2CCC(CCNC(C3CN(C(N)=O)C3)=O)C2)=O)Cc2cccnc2C1 98095,c1(N(CC(CNC(C(CC)CCOC)=O)C)C)nc(O)c2c(ncn2C)n1 98096,Cc1csc2c(C(=O)NC3CCC(CCNC(c4cnc(O)o4)=O)C3)ncnc12 98097,CC1CN(C(C2COC(=O)N2C)=O)CC(C)CN1C(=O)CN(c1ccccc1)C 98098,c1(C(N(CCC(C)NC(Cn2c(C)ncc2)=O)C)=O)cc(F)cc([N+](=O)[O-])c1 98099,Cc1ccc(N)cc1C(N1CC(CCNC(C2(O)COC2)=O)C1)=O 98100,Cc1ccc(C(=O)NC2CCC(C(=O)Nc3ncc(CCO)s3)OC2)cc1F 98101,C1(NC(C(=Cc2cccs2)C)=O)CCCN(C(=O)C(n2ccc(C)n2)C)C1C 98102,Cc1nccnc1CNC(=O)CCCN(C(=O)C(C)CC#N)C 98103,c1(C(=O)NC2CC3CN(C(C4CN(CC)C(=O)C4)=O)C2C3)cccc2[nH]ncc12 98104,C(CCC(C)CC(C(=O)Nc1ccc(F)cc1)N1CCCC1C(N)=O)=C(C)C 98105,CC(Cc1cccc(F)c1)CC(=O)N1CCN(CCNC(C2CCCS2)=O)CC1 98106,CCC(C(=O)NCC(C1CCC1)NC(=O)CCCNC(N)=O)N(C)C 98107,C1(C(=O)NC2C(CC)N(C(=O)CN3CCC(F)CC3)CC2)CC2CC(=O)C1C2 98108,CCC(CC)(C(=O)N(CC(C)N(C(=O)C(C)C(C)C)C)C)c1ccccc1 98109,C1(NC(C2C3CCC(C3)N2C(c2cscn2)=O)=O)CCCC1C1CCCC1 98110,C(C(=O)N1CCCC(CNC(C2(C(F)(F)F)CC2)=O)C1)(C(C)O)NC(C)=O 98111,C1(C(N(C)CC2C(NC(CC(=O)NCC)=O)CCC2)=O)CC2(CCC2O)C1 98112,C1(NC(c2c(C)ccnc2)=O)C2CCCN(C(c3ccncc3)=O)C12 98113,Cc1cc(NC(C2CN(C(=O)CCc3cc(F)cc(F)c3)CCN2)=O)cc(F)n1 98114,c1(CC)ccnc(C(N2CC(N(C)C(c3cc(Cl)c(Cl)s3)=O)C2)=O)c1 98115,C12(NC(=O)C=Cc3cnc[nH]3)CCN(C(C3(O)CCSCC3)=O)CCC1C2 98116,C1(NC(C(c2ccccc2Cl)C)=O)CC(F)(F)CC1NC(c1cc(C#N)c[nH]1)=O 98117,N1(C(CCC2CCN(C(C3(C)CC(F)(F)C3)=O)C2)=O)Cc2n[nH]cc2C1CO 98118,C=CCC(C(=O)NC1CC2(CCN(C(=O)CN3CC=CC3)C2)C1)C(C)(C)C 98119,N1(C(c2c(Cl)cc(C)s2)=O)CCC(NC(C2SC3C=CC2CC3)=O)C(CO)CC1 98120,C1(C(F)F)(OC)CC(C(=O)NCCC2CN(C(=O)CC3CC3C)C2)C1 98121,c1(C(=O)NC2(C)CN(C(C3CCCCC3C3CC3)=O)C2)cccc2[nH]ccc12 98122,N1(C(C(=O)NC(C)C)C(C)C2CCCCC2)CC(C)NC(=O)C12CC2 98123,N1(C(c2ccc(CC#N)cc2)=O)CC=C(C(=O)Nc2ccccc2C2CC2)C1 98124,c1(C(C(=O)NCC(C)(C)OCC(=O)NC(C)CC2(O)CCC2)=O)cccn1C 98125,C1(NC(C2CCCNCC2)=O)CCCC(Nc2ccncn2)C1 98126,N1(C(c2c(CC)ccc(F)c2)=O)CC2CCC(C1)N2C(c1cc(Cl)c(Cl)s1)=O 98127,Cc1nn(CC(=O)NC2CN(C(c3nc(O)sc3C)=O)CC2CO)c(=O)o1 98128,c1(C(N2CC=CC(NC(c3c[nH]nc3[N+](=O)[O-])=O)C2)=O)c(O)cc(O)cc1O 98129,C1(NC(C(C)N2CCC2)=O)CC(C)CN(C(c2cccc(Br)c2F)=O)C1 98130,C(=O)(C(C)CS(C)(=O)=O)NCCCN(c1ccccc1)CCCC 98131,n1(C(C)C)cnc2cc(NCC3CCC4(CCOCC4)O3)ccc12 98132,N1(C(CCc2cn(C)nn2)=O)CCC2CCCC12C(=O)NOCc1cn[nH]c1 98133,c1(C(=O)NC2CCC(CNC(C3N(CC)CC3)=O)C2)c(C)ccc(Br)c1F 98134,c1(CC(=O)NC2C(NC(CC=CC)=O)C2)ccc(Cl)c(C)c1 98135,Cc1cccc(C(CNC(=O)Cc2nnc(O)s2)NC(C2CCSC2)=O)c1 98136,c1(CNC(C(N2C(C)(C)CC(CO)C2)=O)=O)cccc2c1OC(F)(F)O2 98137,C1(CC=C)(C(=O)NC2CCC(CNC(C3(O)COC3)=O)C2)CCOCC1 98138,C=CC1CCCN(N2CCCC2c2c(F)cccc2F)C1 98139,N1(C(C2CC(O)(CC#C)C2)=O)CCOCC1CNC(c1c[nH]nc1F)=O 98140,CN1CC=CCC1CC(=O)NC1CCCCC1NC(c1ccsc1C(F)(F)F)=O 98141,c1(C(N2CCC(C)CC2C(=O)NOCCC2CC2)=O)c[nH]c2ccccc12 98142,c1(C(=O)NC2CC(NCc3cc(C)[nH]c3C)C2)c(F)c(F)c(O)c(F)c1F 98143,c1(NC(=O)CCc2ccc(C(=O)NC3CC3(F)F)[nH]2)ncc(F)cc1O 98144,NC1COCCC1NC(=O)NCCSC1CC1 98145,C1(OC)CCn2cc(C(=O)N(C(C)CNC(=O)Cn3cnc(C#N)n3)C)nc2C1 98146,C=C(C)C(CC(=O)N1CCCC1CN(C(=O)CC1(O)CCC1)C)OCC 98147,c1(CC)nc[nH]c1C(=O)NC(C)CCN(C(=O)CNS(N)(=O)=O)C 98148,C12(C(=O)NCC3OCCN(C(c4ncn(C(C)(C)C)n4)=O)C3)CC(C1)S(=O)(=O)C2 98149,C1(C)(OC(=O)CCC2CC2(C)C)CN(C(=O)CC(C2CC2)CN(C)C)C1 98150,C(=O)(CS(=O)(=O)CCC(F)(F)F)N1CC(N(C(COCc2onc(C)n2)=O)C)C1 98151,N1(C(C(C=C)O)=O)CC2CCC(C1)N2C(=O)Cc1cc(COC)on1 98152,C(=O)(CC(C)(C)CNC(=O)C=CC1CCCCC1)N(CC)Cc1ccn(C)n1 98153,CC(CNC(c1ccc(F)c2c1CCC2)=O)N=c1[nH]ccn2nnnc12 98154,N1(C(c2c(C(C)(C)C)ccs2)=O)CC2CCCC2(Nc2nc3cccnc3s2)C1 98155,c1(C(N(CC(CNC(CC2CC(C(=O)OC)C2)=O)C)C)=O)c(C)n[nH]c1C 98156,CC1(C)C(NC(=O)CCCCCNC(=O)CCC(=O)NC2CC2)CC1(F)F 98157,C1(NC(c2cncc(C)n2)=O)CCSC12CN(C(c1cc(C(F)F)ccn1)=O)C2 98158,C12(CNC(CCC=C)=O)CC(NC(=O)C(COC)NC(C)=O)(CO1)C2 98159,C1(C(=O)NCCC(CCC)C2CC2)CN(C(=O)C(C)(C)C(C)O)CC1(F)F 98160,C(C(C)(C)CN=c1cccc(S(=O)(=O)NC(C2CCC2)C)[nH]1)OC 98161,N1(C(CC(CC)C(C)C)=O)CCCC2(CCN(CCO)C2)C1 98162,C(=O)(C(C)(C)C)NCCC(=O)NCCN(C(CSCC=C)=O)C1CC1C 98163,c1(C(=O)NCCCNC(c2nc(CCC)oc2)=O)cncc(C(C)=O)c1 98164,c1(C(N2C(CN(C)C(c3cc(Cl)no3)=O)CCC2)=O)cnc(Cl)cc1N 98165,c1(C(=O)NC(CSCC)C(N2CCC(NC(N)=O)CC2)=O)cnc(F)cc1C 98166,C(C(C)CN=c1[nH]c(=NCCS(=O)(=O)CCO)[nH]c2cccnc12)OCC 98167,Cc1ccc(C(N2CC3(CNC(c4cnns4)=O)CC2CO3)=O)c(O)c1 98168,S(=O)(=O)(c1ccc(NCCCC(=O)NC2CC2)c(Cl)c1)NC(CCCCC)C 98169,CN1CCN(C(C2CCCN2C(=O)CC2CCCCC2)=O)CC1C1CC1 98170,c1(CNC(c2c(Oc3cccnc3)cccc2F)C)ccnc(C#N)n1 98171,C1(O)(C(N2CCC(N(C(=O)C(C)O)CCOC)CC2)=O)CCC(C)CC1 98172,N1(C(CC2(OC)CCC2)=O)CCOC2CCN(C(C3CC3(F)F)=O)CC12 98173,Cc1ccc(C(N2CC(CNC(=O)C(C)NC(C)(C)C)C2)=O)c2cccnc12 98174,c1(C(N2CCN(C(C3C(C)(C)COC3)=O)CC2CCO)=O)cnn2cccnc12 98175,N1(C(C=C(C)C)=O)CC2(C=C(C(=O)N3CC(C(F)(F)F)C3)CO2)C1 98176,C1(CNC(c2ccnc(S)c2)=O)CC12CCN(C(=O)CS(=O)(=O)C1CC1)CC2 98177,C(=O)(CC(C)C(C)(C)NC(=O)CCc1cc(C)[nH]n1)N(CCOCCO)CC 98178,Cc1cc(NC(C2CC(C)CN2Cc2ccc(I)c(F)c2)=O)ccc1O 98179,C1(CCNC(CC=C=C)=O)CCCN(C(=O)CC2(C#N)CCOCC2)CC1 98180,C(=O)(CC(C)(C)C(C)(F)F)NC1C(NC(CCC(C)C#N)=O)CCCC1 98181,C1(CNC(C2(N(C)C(C3(C4CC4)CC3)=O)CCC2)=O)CCCC1(C)C 98182,C1(C(NOCCC(C)O)=O)CN(C(=O)OC(C)(C)C)CC12CCC2 98183,C1(C(=O)NCC2C3CN(C(c4cnn(CC)c4Cl)=O)CC32)COCCN1C=O 98184,C#Cc1ccc(OCC(=O)NCC2(CNC(=O)C(C)CC)CCC2)cc1 98185,C1(CNC(N(CC(=O)NC(C)(C)C)C)=O)(CNC(=O)C2CC2)CCN(C)CC1 98186,C(C1CCCCC1)=CC(=O)NCc1cc(C(=O)NCc2c[nH]nc2C2CC2)no1 98187,CC(C)(F)C(=O)N1CCC(C(=O)NOCCOC=O)C1 98188,CC(CN=c1[nH]c(=NCC23CC(C2)C(C(F)(F)F)O3)[nH]c2cccnc12)C(F)(F)F 98189,c1(C(=O)NC(CCCNC(C=CCCC(C)C)=O)C)cc2scnc2[nH]1 98190,C1(NC(c2c(C)cc(SC)s2)=O)CC2CC1N(C(=O)Cc1cc(C)on1)C2 98191,c1(C(C(=O)NCC)N(C(C#N)C2(SC)CC2)C)ccc2nc(C)oc2c1 98192,c1(C(=O)NCCN(C(C(C=C)(C)C)=O)CC)cc(=O)n2nccc2[nH]1 98193,C1(C(N(C)CCOCCNC(c2cc(C(F)(F)F)n(C)n2)=O)=O)CCC12CCCO2 98194,N1(C(C=C(CC)C)=O)CC(C)(CNC(C2CCCCS2)=O)CC1(C)C 98195,C1(NC(CC(C)OC)=O)CCCC(NC(=O)Cc2ccc(Br)nc2)C1.C1CC1 98196,C(C(CCO)N=c1[nH]c2c(c(=NCCCn3ccnc3)[nH]1)CCCCC2)N(C)C 98197,c1(C(N(CC(N2CCC(N(CC)CC)C2)=O)C)=O)ccc(Cl)nc1OC 98198,C=C(C)CC(C(=O)NC1CC(CCNC(C2Cc3nccn3C2)=O)C1)OC 98199,C1(CNC(C2(C#C)CC2)=O)CN(C(c2cc[nH]c2CCC)=O)CC12CCC2 98200,c1(C(N2CC(N(C(=O)Cn3cnccc3=O)C)C2)=O)c2c(nn1C)CCOC2 98201,Cn1cc(S(N)(=O)=O)c(C(=O)NCC2CC(O)CN2C(C2CCCC2)=O)n1 98202,c1(C(=O)NC(CC)CNC(=O)C2=C(C)OCC2)cc2c(Cl)c(F)ccc2[nH]1 98203,c1(C(=O)NCC2CC2NC(C2CC(C(F)(F)F)C2)=O)ccc(F)c2c1OCC2 98204,C1(C(N(C2CCN(C(=O)C(C)(O)C3CCC3)CC2)CC)=O)CCC12CCC2 98205,C(=O)(CS(=O)(=O)C1CCCC1)NC1C(NC(C(C(CC)CC)OC)=O)C1 98206,C1(NC(CC(C)(C)SC)=O)CC(O)CN(C(c2cccc(O)c2Cl)=O)C1 98207,C1(NC(c2c(C)cccc2O)=O)CC2CCC1N(C(C1CSC1)=O)C2 98208,c1(C(=O)NC2CCOC2C(N2CC(CO)C2)=O)cncc(O)c1 98209,Cc1nc2cc(CNC(C3CN(c4ncc(C)c(C)n4)CCC3O)=O)cnc2[nH]1 98210,c1(C(=O)NCCN(C(=O)C(F)(F)C2CC2)CCOC)c[nH]cc(C)c1=O 98211,C=C=CC(C)C(=O)NC1(C(N2C(C(=O)OC)CC2C)=O)CC1(C)C 98212,c1(C(=O)NCCc2c(CNC(CC(C)F)=O)nco2)cnc(Cl)cc1N 98213,c1(C(=O)NCCC2(CNC(CC(C)c3ccco3)=O)CC2)nccc2ccsc12 98214,Cc1cc(=O)c(NC(=O)C(C(C)NC(c2csc(Cl)c2)=O)C(C)C)c(C)[nH]1 98215,C1(CC=C)(C(=O)NCc2nc(C(N3CCCC3C(=O)NCC)=O)co2)CCOC1 98216,c1(CC)noc2ncc(C(=O)NCC(F)CNC(c3cscn3)=O)cc12 98217,c1(C(C(=O)N(CC(CN(C)C(c2cnc(O)o2)=O)O)C)(C)C)ccc(O)cc1 98218,c1(NC(C(Cc2cc[nH]n2)NC(C(C)=C2CCCC2)=O)=O)ccc2c[nH]nc2c1 98219,N1(C(C(C2CN(C(CCOc3cc(C)[nH]n3)=O)C2)O)=O)CC2C(C1)C2(F)F 98220,c1(CN2C(C(N3C(C(=O)OC)COCC3)=O)CC(F)C2)cc2cc(Br)ccc2[nH]1 98221,Cc1cc(O)ccc1C(N1CCC(NC(=O)C(=O)Nc2c(F)cccc2F)C1)=O 98222,C(=O)(CCCCCCNC(=O)Cn1ccccc1=O)NC(C)C(C)(C)O 98223,N1(C(C=CC)=O)CC(NC(c2ncsc2CC)=O)C(SC2CCCCC2)C1 98224,N1(C(C(C)OCOC)=O)CCC(O)(CCNC(C2(COC)COC2)=O)C1 98225,C1(OC)CC(C(N2CCCCC2CNC(=O)CC2CCCSC2)=O)CC1OC 98226,c1(N(C2CCN(C(=O)CSCCNc3ccccc3)C2)C)ccccc1 98227,c1(C(C)C)ccc(Cl)cc1C(=O)N(C(C)CNC(=O)Cc1cnoc1)C 98228,N1(C(C)C)CCCC1C(=O)N(CCC1CCC1)CCNC(=O)CCc1cnc(O)[nH]1 98229,C(=O)(C1=CCCCO1)NCC1C(C)CCN1C(=O)C(C)(C)OCC(F)(F)F 98230,N1(C(C2N(C=O)CCC2)=O)CCN(C(=O)Cc2c[nH]nc2O)CC(O)C1 98231,C1(C(=O)NC(c2ccccc2)CNC(CCSC)=O)CC(=O)C12CCCC2 98232,c1(C(n2cc(-c3scc(C)n3)nn2)C(N)=O)cccc(F)c1 98233,O(NC(=O)CC(CNC(=O)CC1CC1)OC)CC#C 98234,c1(CC(=O)N(CCN(C(C)C)C(c2ncccn2)=O)C)cn(C)nc1Cl 98235,O=C(CS(=O)(=O)N1CCOCC1)NCC1CC(O)CN1C(=O)C=CC1CCCO1 98236,C(=O)(CCC(C)(C)F)N1CC(C2N(C(c3cc(C)n(C)c3)=O)CCC2)(O)C1 98237,N1(C(c2n(CC)ncn2)=O)CC(NC(c2ccccn2)=O)C(CC(C)(C)C)C1 98238,Cc1cc(=NCC23CCCCC2CN(C(=O)C2=NOCC2)C3)[nH]cn1 98239,C=CCC(CNC(C1CCN1C)=O)NC(=O)C(C)NC(=O)C1CC1 98240,N1(CCOC)CC(C(=O)NCC2CCC2NC(c2cc(C)ns2)=O)CC1=O 98241,c1(C(=O)NCCN(C(Cc2cc(C)[nH]n2)=O)CC2CC2)cc(C)c(N)cc1F 98242,N1(C(CSCCCC)=O)CCC2(CC1)CCN(C(=O)CCC1CCCCN1C)C2 98243,CC1(C)CC(CC(N2CCCCC2CCCNC(=O)CCn2ccnc2)=O)CO1 98244,n1(CC(N2CCC(CN(C(C3C(C)OCC3)=O)C)C2)=O)nc2ccccn2c1=O 98245,C(=O)(C(C(C)CC)N(C)C(c1ccccc1Br)C)NCC(=C)C 98246,N1(C(C2CC3OC2C2CC32)=O)CCC2CN(C(c3ccnc(C(F)F)c3)=O)C2C1 98247,C(CCCC(=O)NCCn1cccn1)N(C)C(c1[nH]nnc1C1CC1)=O 98248,C1(C#N)(C(=O)NC2CCN(C(c3c(Cl)nc(OC)s3)=O)C2)CC12CCC2 98249,N1(C(CC(CC)(C)C)=O)CCC2(CC1)CC2CNC(=O)CCn1nc(C)nc1C 98250,C1(NC(C2N(CCCC)CCOC2)=O)CCN(C(C2CC2CCOC)=O)C(C)C1 98251,C1(C(C)C)C2CCN(C(=O)C(C3CCN(C(c4nc(=N)cc[nH]4)=O)CC3)C)CC12 98252,c1(C(N2CC(OC)C(NC(=O)C3=CC(O)CCC3)C2)=O)ccc2[nH]c(=N)[nH]c2c1 98253,c1(C(=O)NCC2C3CN(C(C(c4cccnc4)C)=O)CC32)c(O)cccc1F 98254,c1(NC(C(CC)O)=O)ccc(C(C)NC(=O)COc2ccsn2)cc1 98255,C1(CNC(c2c(C(C)C)nns2)=O)C2CN(C(C3CCCN3S(C)(=O)=O)=O)CC12 98256,C(=O)(C(CC)C(C)O)NC1(CC=C)CCN(C(=O)CCc2ccc(O)nn2)C1 98257,CCCC(C(=O)N1CC(C)(CCC(=O)NC(c2nccnc2C)C)C1)NC(C)=O 98258,C1(NC(C(CC)C)=O)CCCCCC1C(=O)NCc1ccc(Cl)cc1 98259,N1(C(=O)CCF)CCC2CN(C(=O)CCCOc3ccccc3Cl)CC2C1 98260,C1(C(N2CC3CC3(C(=O)NC3CCC3)C2)=O)CCC(C(F)(F)F)CC1 98261,C(=O)(C1CCCc2nc[nH]c21)N1CCC(NC(C(CC)(F)F)=O)CC1 98262,C1(C)(C(=O)NCCCN(C(C2C(C)(C)OC(=O)N2)=O)CCO)CCCCNC1=O 98263,N1(C(Cc2c(C)ocn2)=O)CC(NC(C2CC3CC3C2)=O)CC(C)C1 98264,C(=O)(C(F)(F)C(F)(F)F)NC(CCCC)CNC(c1ccccc1Br)=O 98265,c1(-n2c(-c3ccc(-c4[nH]cc(C#N)c4)cc3)ncc2)ccc(F)cc1F 98266,C1(CNC(C=CC=CC)=O)CCN(C(c2ncc(C)cc2F)=O)C1(C)C 98267,N1(C(CSCCC)=O)CCN(C(=O)CCC2COC(C)(C)O2)C(C2CCC2)C1 98268,c1(C(=O)NC2CCN(C(C(C(C)C)CN(C)C)=O)C2)cc(F)cc2cnccc12 98269,c1(-c2cn(C(C3(C)CCOC3)C3CCOCC3)nn2)ccnc(F)c1 98270,c1(NCC2(C)CN(C(=O)NC3CC3)C2)ncc(CO)cc1Cl 98271,c1(C(N(CC(=O)N(CCC#C)C)C)=O)ocnc1C(C)C 98272,c1(CN(C(=O)CC2CCN(CC3CCOC3)C2)CC=C)c(F)cccc1F 98273,C1(C(=O)NCC(CC=C)C(=O)OC)CCC2(CC1)CCC2O 98274,c1(C(N2C(CNC(c3cncc(C)c3)=O)CC(C)(C)C2)=O)cncc2nc[nH]c12 98275,N1(C(C2(OCC)CCC2)=O)CC2CCN(C(c3nnc(C)s3)=O)C2C1 98276,c1(C(N(CCCNC(=O)CCCc2cnn[nH]2)C)=O)ccc2oc(O)nc2n1 98277,N1(C(c2ccc(CC)nc2)=O)CCCN(C(c2ccsc2SC)=O)CC1C(C)C 98278,C1(CCC2CC2)CN(C(c2cn(CCC(C)C)nn2)=O)CCN1C(=O)C(=O)OC 98279,c1(C(N2CC(CN(C)C(c3ccc(F)s3)=O)OCC2)=O)cccc(F)c1N 98280,Cc1nc(C(=O)NCc2csc(C(=O)N(C)Cc3ccncn3)c2)cn1C 98281,CC1(NC(c2cn(Cc3ccccc3)nn2)=O)CN(C(c2cscc2F)=O)C1 98282,C1(NC(c2n[nH]c(C)c2Cl)=O)CCN(C(=O)C(C)CCO)CC1C 98283,C1(CNC(COC2(C)CN(C(c3c[nH]c(C#N)c3)=O)C2)=O)CCCC(F)C1 98284,CCCN=C(NCCCN(CCC)CC)NCC1CCCCC1 98285,c1(OC)cc(CCC(=O)NC2CCCN(C(C3CCOC3C)=O)C2)ccc1Cl 98286,Cc1ccnc(C(=O)N(CCCOCCN(C(=O)CC2(C)CC2(Cl)Cl)C)C)c1 98287,c1(C(N(C2CN(C(CC(=C)C)=O)CC2F)C)=O)cnc(O)c(Cl)c1 98288,c1(C(=O)NCC(C(C)C)NC(C(CC)N(C)C)=O)cc2ccccc2n1C 98289,CCC(CC)C(F)C(=O)NC1(C(=O)NC2C(C)CCC2C)CCN(C)C1 98290,C=CC(C)CC(=O)NCC(CNC(=O)CCC1CC(NC(=O)OC(C)(C)C)C1)CO 98291,c1(C(=O)Nc2ccc(COC(C3(OC)CCC3)=O)cc2)cccc(C)c1C#N 98292,C1(NC(C2(C#N)CCC2)=O)CCN(C(c2cnc(O)s2)=O)CC1c1ccccc1 98293,c1(NCCN(C)C(c2cccc(F)c2F)=O)nc(Cl)nc2nc(Cl)n(C)c12 98294,N1(Cc2c(Br)ccc(C)c2)CC2CC(NC(=O)Cc3c(C)noc3C)CC2C1 98295,C1(C(=O)NCc2nnn(CC)n2)C(C2CC2)CCN1C(C1CN2CCC1C2)=O 98296,C1(C(=O)NCC(CC)N(C(=O)CCC2CCC(C)O2)C)CC(F)(CF)C1 98297,C1(NC(c2c(C(C)(C)OC)cccc2)=O)CC(O)CN(C(=O)C(C)=CC2CC2)C1 98298,Cc1c(Br)ccc(F)c1C(=O)N(C)CCNC(=O)CC1CNC(=O)C1 98299,Cc1[nH]c(C#N)cc1C(=O)NCc1cccc(C(N2CC(C)(C)C2)=O)n1 98300,C1(NC(CC(CCC)(C)O)=O)CN(C(C2CCCCN2N=O)=O)CC2(CCC2)C1 98301,C1(NC(CC2OCCN(C(C(C)OCC(C)C)=O)C2)=O)CC2CC1CC21CC1 98302,C12(NC(=O)COC3COC3)CCCN(C(=O)CCCCF)CC1C2 98303,Cc1cc(=NC2CC3CN(C(=O)CC4(C)CCCC4)CC23)[nH]c(Cl)n1 98304,C(c1cnc(O)nc1O)=CC(=O)NC(C)(CNC(c1ccccc1Cl)=O)C1CC1 98305,c1(N2Cc3c(C)cccc3CC2)nc(=NCC(C)CCO)[nH]c2ccccc12 98306,C1(C(N(CCOC)CC)=O)(CNC(=O)C(C)n2cccc2)CCCC1 98307,c1(CCCC(=O)NCC(CNC(CNC(CNC(C)=O)=O)=O)O)ccc(O)cc1 98308,C1(C(=O)NCc2ccc(CNC(c3cn(C4CC4)nn3)=O)cc2)(CC)CC=CCC1 98309,C(=O)(C(C)(C)CS(N)(=O)=O)Nc1ccc(F)cc1C(F)F.CC1(C)C2CC1NC2=O 98310,Cc1cc(C)n(CC(N2CCC(C)(CNC(=O)C(C)C(C)(C)C)C2)=O)c(=O)n1 98311,N1(C(C(CC=C)CN)=O)CCc2sccc2C1CC 98312,c1(OCC(N2CC(C3N(C(C(C)(C)C)=O)CCC3)(O)C2)=O)cncc(F)c1 98313,C1(C(N(CCC)C)=O)CCN1C(=O)CSc1nc[nH]n1 98314,C1(C)(NC(C2N(C(CS(CC)(=O)=O)=O)CCOCC2)=O)CCCCC1(C)C 98315,c1(OC)cc(C(N2CCCCC2CNC(C2CCS(=O)(=O)N2C)=O)=O)cc(C)n1 98316,n1(CC)cc(Cl)c(C(N2CCC(N(C(=O)CC3CCS(=O)(=O)C3)CCO)C2)=O)n1 98317,C1(C)(CC(=O)NCCOC2CCN(C(C3(C(C)C)CC3)=O)C2)CCS(=O)(=O)N1 98318,N=c1[nH]c2c(s1)CN(c1nnnn1CCCCCC(=O)OCCO)CC2 98319,CCCC(C(=O)N1CC2CC1(CNC(c1nccnc1N)=O)C2)S(N)(=O)=O 98320,C1(CCNC(C(C)NC(=O)Cn2cnnn2)=O)CCCCN1C(=O)CNC=O 98321,C1(C)C(C)C(=O)N1.C12(NC(C3(COC)CCC3)=O)CC(C)(C1)C2 98322,CCCCC(C(=O)NCC(C)(C)CNC(c1cn(C)[nH]c1=N)=O)C(C)C 98323,C(=O)(C1=NOC(C)(C)C1)NC(C(C)C)CC(=O)NC(c1nccc(O)n1)C 98324,c1(SC)cc(C(=O)NCC2CC(NC(C3CC=CCO3)=O)C2)nn1C 98325,c1(C(=O)NCC2CC(NC(c3cc[nH]n3)=O)C23CCC3)c[nH]c2cnccc12 98326,N1(C(C(c2ccnn2C)NC(c2c(C)csn2)=O)=O)CC2CC1CS2=O 98327,C(C(C(C)C(C)C)NC(=O)CSC)NC(CCc1cncc(OC)c1)=O 98328,C1(c2n(CCOC)nnn2)(NCC2COC2)CC2CC1CC21CC1 98329,n1(CCC(N2CC(O)(C3CCCN3C(=O)C3=CCC3)C2)=O)cnc2ccccc12 98330,c1(N2CC(C)(CCO)OCC2)ccncc1S(=O)(=O)NCC(C)(C)c1cccs1 98331,c1(C(NOCC(=O)NC(CC#C)C)=O)ccc(O)nn1 98332,N1(C(c2cc(OC)cc(=O)o2)C(=O)NCC(=C)C)CC2COCC(CO)(C1)C2O 98333,CC(O)(Cn1ccccc1=O)C(=O)NC1CC(F)(CNC(=O)Cn2cnnc2)C1 98334,Cc1ccc2c(=NCc3nc(=N)[nH][nH]3)[nH]c(=NCCC(C)(C)C)[nH]c2c1 98335,c1(NCC(COC)(C)CO)[nH]c(=NCCc2ncccc2C)nc2scnc12 98336,N1(C(C(=O)NC(C)C)=O)CCC(C)(CCNC(C2C=CCCC2)=O)CC1 98337,c1(C(N2CC3C(C(=O)NCCOCC)(C3)C2)=O)ccc2c(c1)C(=O)CC2 98338,N1(C(C(COC)NC(C)=O)=O)CCN(C(=O)C(O)CC(N)=O)C(C)C1 98339,N1(C(C(CC)OC)=O)CC2(C1)CN(C(=O)C(CC(C)C)OCC)CC2CO 98340,C1(C(=O)N2CC2)(OCC)CCCCC1.C12CCCC(C1)NC2=O.O(C)CC 98341,CC(C)C(C)C(=O)NC1(NCc2ccc(OC(F)F)cc2)CCC1 98342,C(C(=O)NCCN(C(=O)C(c1cscn1)N(C)C)C)(OCC)OCC 98343,c1(C(=O)NC2CN(C(=O)C(F)CC3CCCCC3)CC2O)ncc(Cl)cc1O 98344,N1(C(CCN(C(CCC)C)C)=O)CCN(C(C2CC3(C2)CC(O)C3)=O)C2(CC2)C1 98345,Cc1cc(C(N)=O)sc1Cc1ccccc1.C1(=O)C(=O)NCCCN1 98346,C1(C(N(C2(CC(=O)NCCC3(C)CCOC3)CC2)C)=O)CCCC(=O)N1 98347,C1(CC)CCCN(CC(=O)NC2CN(C(=O)CC3(C#N)CC3)CC2O)C1 98348,n1(CC)ncc(C(=O)NC2CC(NC(=O)CCC3CCCCN3C)C(O)C2)c1C 98349,C1(N(CCCO)C(C2(C(C)NC(=O)COCCF)CC2)=O)C2CCCC12 98350,N1(C(c2cn(CCOC)nc2)=O)CCC(CCN(C(=O)C(C)SC(C)C)C)CC1 98351,C(CNC(C1C2(CC2)C12CC2)=O)(C(C)(C)C)NC(CC1C(CC)C1)=O 98352,C#Cc1ccc(F)c(C(=O)NC2CCN(C(=O)C(C)(CO)OC)CC2)c1 98353,c1(C(N2CC(CCCNC(C(CC)OC)=O)OCC2)=O)cc(F)ccc1C1CC1 98354,CCC(CNC(c1ccc2cc[nH]c2n1)=O)(CC)C(=O)NCC1CCOC1CC 98355,CC1CN(C(C2CN(S(=O)(=O)C(F)F)C2)=O)CCN1C(C1COC(=O)N1C)=O 98356,C1(NC(c2c(OC)csc2)=O)CCN(Cc2c(C)noc2C)CC1(C)C 98357,CCC(CC(=O)N(CC(O)CNC(c1ccn(CC)c(=O)c1)=O)C)C(F)F 98358,c1(C(C(=O)NCC2N(C(C=CC=CC)=O)CC=C2)C)ccc(SCC)cc1 98359,c1(C(c2nnnn2CCOCC2CC2)NCCC=C=C)cc2nc(Cl)ccc2s1 98360,c1(CNC(=NC)NCCC(C)CCC(=O)NC)nnn(C)c1N 98361,C1(C(N2CC(CCCCNC(C(C)=C(C)C)=O)C2)=O)C2Cc3cc(Cl)ccc3C12 98362,N1(C(CCC2CCCN(C(CCN(CCC)C)=O)C2)=O)CCOC(CC)(CC)C1 98363,C1(C(=O)Nc2ccc(OCC(=O)OC)cc2)CCCCC1(OC)OC 98364,N1(C(Cn2c(C)nc(C)n2)=O)CCC(C(=O)NCCc2nncn2C)CC1(C)C 98365,N1(C(C2(C)ON=C(C)C2)=O)CC2CN(C(c3cc4cnccc4o3)=O)CC2(C)C1 98366,C1(NC(CC=C)=O)CCN(C(c2occc2C)=O)C1C(C)(C)C 98367,C1(C(=O)NC2C(NC(c3c(C)nc(C)s3)=O)COCC2)CCC(=O)N(C(C)C)C1 98368,c1(OCC=C(C)C)cccc(C(=O)NC2CCC(NC(c3cncs3)=O)CC2)c1 98369,CC(CC(=O)N1OCC(F)(F)C(=O)NCC(C)C1)C(C)(C)C 98370,CC(CC(=O)N1CC(NC(c2cccc(Cl)c2)=O)C1)C(=O)c1ccccc1 98371,c1(NC(CC(CCC)NC(c2cn3ccccc3n2)=O)=O)cnc(C)c(C#N)c1 98372,CCCCCCCCCCCC(=O)NCC1CCCN(C(C2CCSC2)=O)C1 98373,c1(C(=O)NC2CC(CCC(=O)NCCC(C)(C)OC)C2)c(C)nsc1N 98374,c1(C(N(CCNC(C(CC)N(C)C)=O)CCOC)=O)nc(C)ncc1Br 98375,C1(NC(c2cnc[nH]2)=O)CN(C(=O)CC2CC3(CC3)C2)C2(CCCCCC2)C1 98376,C1(NC(C(C)OCCC=C)=O)CCCC12CCN(C(c1cc(Cl)sc1Cl)=O)CC2 98377,c1(C(=O)NC2CCCC(NC(C=CSC)=O)CC2)ccn2c(O)nnc2c1 98378,N1(C(C(C2(O)CCC2)NC(=O)CCN2CCOCC2)=O)CC(F)(C2CC2)C1 98379,N1(C(C(=O)NCC)=O)CCOCC1CN(C(=O)C(C)(C)c1cncs1)C 98380,C1(c2nnc(N(C(COC)C)C)n2Cc2ccc(C)c(C)c2)CC2(CCOC2)C1 98381,N1(C(C2(COC)CC2)=O)CCC2(CCC(NC(C3CC(C4CCCC4)C3)=O)C2)C1 98382,c1(C(=O)NCC(CC=C)NC(=O)C(F)n2ccnc2)cnc(C(F)(F)F)nc1 98383,C(=O)(N=c1nc(C2(C)CC2)[nH]s1)N(C)Cc1c(C)n[nH]c1 98384,Cc1cc(N2CCCC(C)C2CNC(=O)C(C)(C)CC(C)(C)C)ncc1[N+](=O)[O-] 98385,c1(OC)c(NC(C2CC3CC3N2Cc2c(F)ccc(C)c2Br)=O)ccc(F)c1F 98386,N1(C(c2c(CC)n(CC)nc2)=O)CC2(C=C(C(=O)NCC(O)CC(C)C)CO2)C1 98387,N1C(CC(=O)NCC2(C(=O)NCCc3cc[nH]n3)CCC2)CCOCC1=O 98388,C1(C)(NC(c2n(C)nnn2)c2ncoc2C(C)(C)C)CN2CCC1CC2 98389,c1(N(c2n(C)nnc2)C(C2CNC2)=O)ccn2ncc(Br)c2n1 98390,C1(CNC(c2ccc(OC)s2)=O)CC(C)(C)CCC1NC(=O)C(C)(C)CC(F)F 98391,C(=O)(C1=CCCCC1P(C)(C)=O)NC1C(CNC(C(C)(C)c2ccccc2)=O)C1 98392,c1(C(N2C(CN(C(C(COCC)C)=O)C)COCC2)=O)cncc2c1CCC2 98393,N1(C(c2c(C)cco2)=O)CCC(C(=O)NOCCN(C)C)C12CC2 98394,C1(NC(=O)COCC2CCCO2)CCCC(NC(=O)Cc2nccc(O)n2)C1 98395,N1(C(CC(CC2CN(C(=O)OC(C)(C)C)C2)O)=O)CCC2CCCC12c1ccco1 98396,N1(C(CN(C(c2ccc(N(C)C)nc2)=O)CC)=O)C2CCC1CC2 98397,CCC(CC)CC(=O)N1CC=CC(C(=O)NCC=CC(=O)OCC)C1 98398,N1(C(c2n(C)nc(C(F)F)c2)=O)CCC(NC(C2CC2(C)C)=O)C12CCC2 98399,N1(C(CCCC(=C)C)=O)CCCC(C2CCN(C(C3CN4CCN3CC4)=O)C2)C1 98400,c1(C(=O)NCCCn2cc(C3CCCC3O)nn2)cnn2cccc(Cl)c12 98401,c1(N(C(C)=O)CC)ccc(C(=O)NCC2(c3ccccc3Cl)CCOCC2)cc1 98402,c1(C(=O)NCC2C(NC(C(CC)O)=O)CCCC2)c(C)sc(C)c1C#N 98403,CC1CCCN(C(c2cnc(Cl)s2)=O)C1CNC(C1C2COCC12)=O 98404,C(C(C)CC(F)(F)F)NC(C(c1ccnn1C)NC(C(C)SC)=O)=O.C1CO1 98405,c1(CCC(=O)NC2(C)CC(NC(C(C)=CC)=O)C2)ccc(F)cc1Cl 98406,Cc1cc(Br)cc(C(N2CCC(O)(C(=O)NC3CCOCC3)CC2)C(=O)NC)n1 98407,c1(CC(N2C3C(NC(COCCOC)=O)C(C3)C2)=O)ccc([N+](=O)[O-])cc1Cl 98408,c1(NCC)cccnc1C(=O)NCC1CCC1NC(C1(n2cccn2)CC1)=O 98409,O(N1CCC(CC(=O)N(C(C)CN(C(=O)CC(C)COC)C)C)CC1)CC 98410,C1(NC(c2ncn(C(C)C)c2)=O)CCOCC1NC(=O)CC(=O)NC1CC1 98411,C1(C(C)NC(=O)C(C)n2cccn2)CCN(C(c2ccnnc2Cl)=O)CC1 98412,c1(C(C)C)ccc(F)cc1C(N1CCC(NC(=O)C(O)C2CC2)C(O)C1)=O 98413,C#Cc1cccc(CC(=O)NCC2(NC(c3ncccn3)=O)CCCCC2C)c1 98414,C1(C(N(C2CCN(C(C(CC)C)=O)C2)C)=O)CCn2c(cnc2C)C1 98415,O=C1CCCc2ccc(C(N3CCCCC34CC(NC(=O)C(O)CF)C4)=O)cc21 98416,c1(NC(C2C(NCc3cccc(C)n3)CCC2)=O)cc(F)c(F)cc1[N+](=O)[O-] 98417,N1(C(c2cnc(C(C)C)s2)C(=O)NC)CCN(C(=O)OC(C)(C)C)CC1C 98418,c1(C(N(C2CCN(C(c3cc(C)on3)=O)C2)CCO)=O)cc(N)cnc1C 98419,O=C1NC(=O)C2(CCN(C(=O)C(=O)NC(c3ccc4ccccc4c3)CF)C2)N1 98420,O=C(C1=CCCC1)NC1CN(c2cc(-n3cncn3)ncn2)CC1F 98421,C(c1c(F)cccc1F)=CC(N1CC(OCCNC(C(C(C)OC)O)=O)C1)=O 98422,N1(C(c2ccn(C(C)C)n2)=O)CC(NC(=O)CCC2CCCO2)CC(O)C1 98423,Cc1cc(C(N2CCCC(CNC(=O)CCF)C2)=O)cc(I)c1 98424,c1(SC)nccnc1-c1nc(C2C=CCC2)n(C(c2cnn(C)c2)C)n1 98425,N1(C(C(CC)Oc2ccccc2)=O)CCC2CN(C(c3ccn(C)c3)=O)C2C1 98426,C1(C(N(CCCCCNC(C(COC)N(C)C)=O)C)=O)OCCOC1(C)C 98427,c1(C(=O)NC2CC3(C(NC(c4c(N)cc(Cl)nc4)=O)C3)C2)n[nH]c2c1CCSC2 98428,C1(C(=O)NCc2cccc(CNC(CCCC#C)=O)c2)CCn2c(C)cnc2C1 98429,c1(C(=O)NCC(CC=C)NC(C2CCC(CO)CC2)=O)cc(C#N)ccc1F 98430,C(CCCCCC(=O)N1CCC(O)C(F)(F)C1)NC(C1CC2CCC1CC2)=O 98431,CCCCC(C)CCC(=O)NCC1(NC(c2ccc(O)cn2)=O)CCOCC1 98432,n1(CC)c(N(CC)CC)nnc1N1CCC(CN)CC1.N1(CCOC)CCN(C)CC1 98433,C(N=C(NC1CC1)NC1CC(C)(C)CCc2ccccc21)c1c(C)ncs1 98434,C1(CNC(COCC(C)(C)C)=O)CC(CNC(c2cc(C3CC3)cs2)=O)CO1 98435,n1(CC(N2CCC(CN(C(c3c(OC)scc3)=O)C)C2)=O)nc(C)c(Cl)c1C 98436,C(=O)(CCC(C)(C)[N+](=O)[O-])NCC1C(C(=O)NC(CC=C)C2CC2)CCO1 98437,CC1(C)CN(C(=O)COc2ccccc2F)CC1NC(=O)CCCC#N 98438,CC(C)(C)CC(C)(C)C(=O)NC1CN(C(=O)C(O)CC2CCCCC2)C1 98439,Cc1ccc(NC(C)CN(C)C(c2sccc2C(F)F)=O)c([N+](=O)[O-])c1 98440,Cc1cccc(C(C)C(=O)N(CCNC(=O)C#CC2CC2)CC2CCCCC2)c1 98441,CCC(C)CCC(=O)N(C1CCCCC1NC(C1(n2cnnn2)CC1)=O)C 98442,C1(C(=O)NC(CCSC)Cc2cccnc2)CCCCC(C)(C)C1 98443,c1(C(=O)NC(CC)CNC(=O)C(C(C)C)OC)c(Cl)nc2ccccn12 98444,c1(C(=O)N(C2CC2)CC2CCCN2C(c2csnn2)=O)coc2c1CS(=O)(=O)C2 98445,C1(C(N2C3C(NC(C(C)OCCOC)=O)C(C3)C2)=O)CCCC2(CCOC2)O1 98446,N(C(=NCCN1CCOCC1(C)C)NCCOC)C(c1cccc(C)c1)C#C 98447,C(=O)(C#CC1CCCC1)NCC(CC=C)C(=O)NC(CCOC)C(N)=O 98448,N1(C(c2cc(SC)oc2C)=O)CCC2(CCC2NC(c2occc2C)=O)CC1 98449,C=CCC(C)C(=O)N(C1(C(=O)N(C)CCn2ccnc2)CC1)C 98450,Cc1nn(CCO)c(C)c1C(=O)NCCCNC(=O)Cc1ccccc1Cl 98451,C1(COC)(NC(=O)Cc2nnc(C)s2)CCCN(C(c2ccc(OC)cn2)=O)C1 98452,c1(OCCC(=O)NC2C(NC(C(CCC)C)=O)COCC2)c(C)cccc1C 98453,C(=O)(C(O)CC(C)C)NC(c1nc(C(=O)NCc2nc(C)cc(C)n2)co1)C 98454,C12(NC(c3nc(CCOCC)oc3)=O)CCN(C(=O)CNC=O)CCC1C2 98455,c1(OC)nccc(Br)c1NC(=O)NCC1(C(N)=O)CCOC1 98456,C1(NC(C2CC(C)(CC)C2)=O)CN(C(C2C3CCC(=O)C23)=O)CCC12CCC2 98457,C(c1ccc(S(C)(=O)=O)o1)=CC(=O)NC(CNC(CCCC(C)C)=O)C1CCC1 98458,N1(C(C(C)C2CCCO2)=O)CC2CC(C1)N(C(c1cc(N)cc(O)c1)=O)C2 98459,C(C)(C)(C(C)CC(=O)NCC1CC12CC2(F)F)NC(CC1(NC(C)=O)CC1)=O 98460,N1(C(=O)COCC2CCCCO2)CCN(C(=O)C(O)C2CCCC2)CC2(CC2)C1 98461,C(C1=CCN(C(=O)CC(F)(F)F)CC1)NC(Cn1c(C(C)C)nnn1)=O 98462,C(=O)(CCCC(F)(F)C(F)(F)F)NCC1(NC(c2nc(C#C)sc2)=O)CC1 98463,C1(C(C)(C)C)CCC(NC(=NCc2cnccn2)NCC(F)F)CC1 98464,N1(CCC)CCCCC1CN=C(NC(CC)CC)NC1CCS(=O)(=O)C1 98465,C1(NC(c2cnc(C(C)C)s2)=O)CC2CCC1N2C(=O)CC1CC(=O)NC(=O)C1 98466,c1(C(=O)NC2CCCN(C(c3cccc(SC)c3)=O)C2C)cc2cccnn2c1 98467,C1(SC)CN(C(C2(O)CC(F)(F)C2)=O)CC1NC(C1(C)CC1(F)F)=O 98468,C1(NCc2cccc(-c3nnc(C)o3)c2)CCC(C)(C)CC1C(=O)O 98469,Cc1oc(C)c(CN2CCC(NCCN3CCCCC3)CC2)c1C 98470,C(c1ccc(F)cc1)=CC(N1CC(NC(c2nccc(N(C)C)c2)=O)C2C1C2)=O 98471,Cc1cccc(C)c1NC(=O)C(c1ccccc1Cl)N1CCC(C)(O)C1 98472,c1(C(=O)NC(CN(C(c2cccc[n+]2[O-])=O)CC)C)cc(C(F)F)ncn1 98473,c1(NC(C(CN(C)CC)C)=O)cccc(NC(=O)CCNC(=O)OC(C)(C)C)c1 98474,CCCC(C)(O)C(=O)NC1CC(CC(N2CCC2CC2CC2)=O)C1 98475,N1(C(c2ccc(C(C)=O)o2)=O)CCOCC1CC(=O)NCC1(C)CCCC1O 98476,N1(C(C(C2CCCO2)NC(CCCCOC)=O)=O)CCC2(C1)CN(C)C2 98477,CC(F)(F)CCCC(=O)N1CCC(CO)C(NC(=O)COc2cccc(Cl)c2)C1 98478,C1(C(=O)NCC2(CCC)CCC2)CCC(n2cc(-c3csc(C)c3)nn2)C1 98479,c1(C(=O)NC2COCCN(C(C3CC4(CCC4)CO3)=O)C2)ccc2ccnn2c1 98480,N1(C(CC(CC(C)(C)C)O)=O)CCCC(C2CN(C(=O)CCn3cncn3)C2)C1 98481,c1(C(N(C2CCN(CC)C2)C)=O)cnc(CNC(=O)C(n2ccnc2C)C)nc1 98482,CC(C)C(CCNC(c1cnn(CC2CC2)c1)=O)NC(=O)Cc1cn(C)nn1 98483,c1(OC)cc(OC)cc(NCCSc2n[nH]c(Br)n2)c1 98484,c1(NC(C2CC23CC(NC(C2CCC2)=O)C3)=O)ccccc1CCO 98485,N1(CC)CC(C(=O)NCC(c2ccccc2)NC(c2ncn(CC)n2)=O)NC1=O 98486,CN1CCN(C(C2(C)CC2(C)C)=O)CC1C(=O)NCc1ccc(F)cc1 98487,N1(C(C2C(C=C)OCC2)=O)CCCN(C(c2nc(C)n(C)c2C)=O)C(C)C1 98488,c1(C(N2CC(N(C(=O)C3=COCCO3)C)C(C)(C)C2)=O)ccnc2ccncc12 98489,c1(C(=O)OC)ccc(CC(=O)NC2CN(C(c3ccnn3C)=O)C3CC23)cn1 98490,CS(=O)(=O)CCC(=O)NCC(CC1CC1)C(=O)NCCC1NC(=O)NC1=O 98491,C1(OC)CCn2cc(C(=O)N(C)CCN(C(=O)C(C)C#N)C)nc2C1 98492,N1(C(C)=O)C(C)CN(C(c2cn(C)nc2Br)C(=O)NC2CCCCC2)CC1C 98493,O=C(C1CC(O)c2ccccc21)OCc1c(F)cc(O)c(Br)c1F 98494,CC(C)CC(O)C(=O)N(C(CNC(=O)CCC(=O)c1ccc(Cl)cc1)C1CC1)C 98495,N1(C(CNC(CC2(OC)CCC2)=O)=O)CCCC(C)C1Cc1cc(C)cc(F)c1 98496,N1(C(CS(CC)=O)=O)CCC2(CCCCN(C(C3(c4ccccc4)CC3)=O)C2)C1 98497,C(=O)(C(C)CS(C)=O)N1C(CNC(c2c(NC(C)=O)c[nH]c2C)=O)CC(F)C1 98498,c1(OC)ccc(CCC(=O)NCC(C)N(C)C(c2cccs2)=O)cn1 98499,C(CC(=O)NC(C)CNC(=O)C=C(C)C(C)C)OCCC 98500,Cc1nc(C(=O)N(C)CCOCCCNC(=O)CC2(C)CCCO2)co1 98501,C1(CC)(CC)CC(NC(=O)Cn2nccc2C)CN1C(=O)CSC1CC1 98502,C(=O)(C(O)CC(C)(C)C)NCCCCNC(C(c1c(C)n[nH]c1C)C)=O 98503,Cn1ncc2c(C(N3CCC3CNC(c3ccc4c(n3)CCO4)=O)=O)cccc12 98504,CC12CC(NC(c3csc(O)n3)=O)(C1)C1(CN(C(=O)CC3=NNC(=O)C3)C1)O2 98505,Cc1cc(CCC(c2nnnn2CCC2CC2)NCc2cc(C(N)=O)no2)no1 98506,C(C)(CNC(=O)C(=O)NCC(C)OC(F)F)(CO)OC 98507,C1(C(C)C)CCCC(C(N(CC(F)F)CCO)=O)C1 98508,c1(C(=O)OC(C(=O)Nc2c(C)ccc(N(C)C)c2)C)ccc(S(=O)(=O)N(C)C)cc1 98509,C(CC(C(=O)N1CC(SC)C1)NC(=O)CC1CC=CCC1)OCC 98510,c1(CNC(Cn2ncc(C)c2)=O)cccc(-n2cc(C3CCNC(=O)C3)nn2)c1 98511,c1(C(=O)NC2CC(NC(C(C)N(C)C)=O)C2)ccn2ncc(Br)c2n1 98512,N1(C(CC(=C)C)=O)CCC2(NC(=O)C(=Cc3cccnc3)C)CCCC12 98513,N1(C(CCc2ccc(C)o2)=O)CCC(O)CC1C(=O)NOC(C)(C)C 98514,N1(C(c2c(OCC)nccc2)=O)CC2CCCC(NC(c3ccsn3)=O)(C2)C1 98515,N1(C(C(CC(=C)Cl)NC(=O)C=C(C)C2CC2)=O)CCc2nc[nH]c2C1 98516,c1(-c2cc(C(=O)NCCC(C)N(C)C(C3CC4CC4C3)=O)no2)cccc(Cl)c1 98517,c1(OCC)cncc(C(=O)NCC(C2CCC2)NC(=O)CC2CCN(C)C2=O)c1 98518,c1(CCC(=O)NCC(CC)NC(c2cn(CC(=O)OC)nn2)=O)ncccc1C 98519,CC1CCc2ncc(C(N3CCC3C3CC(F)(F)C3)=O)n2C1 98520,c1(CC)cc(N2CC3C(CNC(c4n[nH]cc4Cl)=O)C3C2)nc(CC)n1 98521,CCC(O)CC(=O)N1CC=CC1(C)C(=O)N(C)CCn1cnnc1 98522,N1(C(CN2CCC(OC)CC2)=O)CC2CN(C(=O)CSC)CCC2(CO)C1 98523,N1(C(c2c[nH]c(=NC)s2)=O)CCC(NC(=O)CN2CCCNS2(=O)=O)C(F)C1 98524,Cc1ccn(CCC(=O)NCC2CC(O)(CNC(=O)Cc3csc(C)n3)C2)n1 98525,C1(CNC(C(C)NS(C)(=O)=O)=O)CC2(CCC2)CN1C(c1cc(=O)cc(Cl)[nH]1)=O 98526,CCCCS(=O)(=O)NC(C)C(=O)NC1(CCNC(c2nnn(CC)c2C)=O)CC1 98527,N1(C(CC=CC=C)=O)CCN(C(c2ccc(Cl)c(CC)c2)=O)C2(CC2)C1 98528,C1(C(N2C(CC(=O)N(c3ccc(F)cn3)CC)CCCC2)=O)CC(C)(C)CN1C 98529,C1(C(=O)NC2(CO)CN(C(=O)CCCCc3cnn[nH]3)C2)CCC2(CCOC2)O1 98530,N1(C(c2cnc(CC)s2)=O)CC(C)CCC1CNC(=O)CNS(N)(=O)=O 98531,C1(CNC(=O)C(F)Cc2ccccc2)CN(C(C2(F)CC2)=O)CCCO1 98532,C(CN=c1[nH]cc(C(=O)NCC(c2ccc(OC(C)C)cc2)(F)F)s1)OC 98533,N1(C(c2c(SC)snn2)=O)CCCCC1CCCNC(C1CCS1(=O)=O)=O 98534,c1(C(=O)NCC2(C)CCCN2C(c2cccc[n+]2[O-])=O)ccc2scnc2c1 98535,C1(CNC(COCC=C)=O)COC(C(F)(F)F)CN1C(=O)CC1CCC(C)CC1 98536,CCC(C)C(C(=O)N(CC(O)CN(C(=O)C(c1cccc(O)c1)C)C)C)OC 98537,N1(C(CN(C2CCCCC2)CC)=O)CC2CC(C(=O)NCc3nnsc3C)CC2C1 98538,c1(C(N2CCC(O)(C(N3CCOC(CO)C3)=O)C2)=O)c(F)cncc1F 98539,C#CCC(CC#C)C(=O)NCC(C1CCN(C(C2(C)CCN(C)C2=O)=O)CC1)F 98540,CC1CN(CC(=O)CCc2c(F)cccc2F)CC2(CCCOC2)O1 98541,CCC(O)CC(=O)N1CC(CC(C)NC(c2cc(-c3cccs3)on2)=O)C1 98542,C1(C(=O)NCCN(C(=O)CCCc2cnn[nH]2)CC(C)O)CCC2(CCC2)OC1 98543,C1(C(=O)NCC(C(C)C)NC(CC(C(F)(F)F)OC)=O)COc2ccccc2O1 98544,N1(C(c2ccc(OCC#C)cc2)=O)CCN(C(=O)COCC#N)C2CC12 98545,CN1CCOCC1C(N1CC(CO)(NC(c2ccc(C(C)(C)C)nc2)=O)C1)=O 98546,CC1CC(C(=O)NCC(C)(O)C2CC2)N(C(C2CC(CF)C2)=O)C1 98547,C(CC(F)F)(C(=O)NCC1(C)CCCO1)N(C)C(C1CC(C2CC2)=NO1)=O 98548,C1(c2cn(CC3CC(F)(F)C3)nn2)(NC(=O)CC2CCCO2)CCCOC1 98549,C(=O)(CCCC(C)(C)NC(=O)C=Cc1cccnc1)N1CCC(CC)C1 98550,C1(NC(=O)CN2CCCNC2=O)CN(C(c2conc2C(F)(F)F)=O)CCC1O 98551,N1(C(C=C2CCC(C)C2)=O)CCOC(C(C)NC(C2CCCN(C(N)=O)C2)=O)C1 98552,C(=O)(C(CNC(c1csc(F)c1)=O)CC1CC1)NCC1C(CCC)C1 98553,C1(C(=O)OC(C)C(=O)N(C)C)CN2CC1CNC2=O.C(=O)(C(C)(C)C)OC(C)(C)C 98554,c1(CNCC2CCCN(c3cc(C(C)O)ncn3)C2)cc(Br)ccc1OC(F)F 98555,C1(NC(Cc2cn(CC)nn2)=O)CCC(C)N(C(=O)CC2(C)OCCO2)C1 98556,N1(C(C(C=C)(C)C)=O)C(CNC(=O)CCOC)CC2COCC12 98557,N1(C(C2CC(CS(N)(=O)=O)C2)=O)C2CC1CN(C(=O)Cc1ccoc1)C2 98558,O=C(CCCC(F)(F)F)OC1CCCCC1F 98559,C(CCN=c1[nH]c(N2CCN3CCOCC3C2)nc2c1SCC2)NC(C)(C)C 98560,CCCC(C)(CC)C(=O)NCc1ncccc1CNC(=O)Cc1ccsc1C 98561,c1(-c2c(OCC(=O)OC)ccc(Br)c2)ccc2c(c1)C(C)C(C)O2 98562,C1(C(N(C2CCN(C(c3cc(CCCO)on3)=O)C2)C)=O)CCCS(=O)(=O)N1 98563,C1(C(=O)NC(CC)C(=O)N(C)C)CC(NC(C2(C)CC(C)=NO2)=O)C(O)C1 98564,c1(C(N2CC(CNC(CN(C(C)C)C)=O)C(C)CC2)=O)cn2cc(Cl)cnc2n1 98565,c1(CNC(c2cc(CNC(C(CC)(C)O)=O)no2)=O)cc(C)cc(F)c1 98566,Cc1cc(C(N2C3CCC2CC(NC(C2(C)CC=CCO2)=O)C3)=O)cn(C)c1=O 98567,N1(C(C)=O)CCOC2(CCN(C(=O)C3CC3)C2)C1.c1cc(C)nc2c1c(C)nn2C 98568,C1(C2(N(C(=O)C=CC3CCCN3C(=O)CCCC(C)=O)CC)CC2)(OC(C)=O)CCC1 98569,c1(CNC2CCN(C(Cc3ccc(OC)cc3)=O)C2)c[nH]c2cccnc12 98570,CCCCCC(C)CC(=O)NCCN(C(=O)C(F)CC1CCCC1)C 98571,N1(C(c2cccc(C(C)C)n2)=O)CC(CNC(=O)COC2CC2)N2CCC1C2 98572,C(CC(F)F)(C(=O)NCc1cc(O)cc(F)c1)N(C)C(c1ccnc(CO)c1)=O 98573,C1(CNC(Cc2nnc(C)s2)=O)CCC(CNC(=O)C(C)C(C)O)CC1 98574,n1(CC(=O)NC2C3N(C(c4c(C)cn(C)c4)=O)C(CC3)C2)cc2ccccc2n1 98575,N1(C(C=C(C)C(=O)O)=O)CCC2CN(C(c3cn4cccc(C)c4n3)=O)C(C)C12 98576,C1(CNC(C2N(C(N)=O)CC(O)C2)=O)CC2(CC2)CN1C(=O)CCC1CC1 98577,C1(CC)CN(C(=O)NC2CCN(c3cccc(Cl)c3)C2=O)CCO1 98578,c1(NC(=O)OCC(C)NC(c2ccccc2)C)ccc2ncccc2n1 98579,N1(C(C(C)(C)CF)=O)CCN(C(c2cc(F)c(CO)c(F)c2)=O)CC(O)C1 98580,c1(C(=O)NC(C2(O)CN(C(Cn3ncc(C)c3)=O)C2)C)nc(C2CC2)ncc1Cl 98581,N1(C(C(C=CCCC)O)=O)CCN(C(=O)CNC(=O)OCc2ccccc2)CC1 98582,Cc1cc(C(N2CCCC2CCCNC(C2CC23CCSCC3)=O)=O)nc(C)c1 98583,CC(C)CC(C(=O)NC(CCF)C(=O)NCCCOC1CCC1)C(N)=O 98584,c1(C(=O)NCC(C)NC(c2ccc(C(F)C(F)(F)F)cc2)=O)ccnc(Cl)c1N 98585,c1(C(=O)NCC#CC(=O)NCC2CN(C(C)=O)C2)c[nH]c(=S)cn1 98586,c1(C(=O)NCC2(NC(CC3N(C)C(=O)CC3)=O)CCC2)cncc2c1CCCC2 98587,C(=O)(NNC(=O)c1ccc(I)cc1)C1C(C)OCC1 98588,Cc1c(Cl)ccc(Cl)c1NC(=O)CC1CCCN1C(=O)Cc1ccc(Br)cc1Br 98589,C(=O)(CC(C)CC(C)(C)C)N1CCC(CNC(c2ccc(C=C)cc2)=O)(CO)C1 98590,c1(COC)csc(C(=O)N(CCNC(C2CCCC2O)=O)C2CC2)c1 98591,N1(C(C#CC)=O)C2CCC1CN(C(c1ccc(Cl)nc1F)=O)C2 98592,C12(C(N3CC(O)CC(NC(c4ccncn4)=O)C3)=O)CCCC(CCC1)C2O 98593,C(C)(CCC(F)(F)F)(C(F)(F)F)NC(c1ccc(OCC)cc1)C 98594,C(=O)(CCC(C)(C)[N+](=O)[O-])NCC1OCCN(C(C(C2CCC(=O)N2)C)=O)C1 98595,CC1CCC(NC(c2cc(C(F)(F)F)cs2)=O)CN1C(=O)CC1CCCC(=O)N1 98596,C1(C(N2C(CNC(=O)Cc3cnns3)CC2)=O)CC12CCCCCC2 98597,c1(C(=O)NCC(CNC(CCC=CCC=C)=O)(C)O)c(C)c[nH]c1CC(N)=O 98598,C1(C#N)(C(=O)NCCn2cc(CNC(CN3CC(C)C3)=O)nn2)CC12CCC2 98599,C(=O)(CCS(C)(=O)=O)NCC(C)(CO)NC(=O)CSCCCc1ccccc1 98600,N1(C(C(CN(C)C)N(C)C)=O)CC(O)(C2(CNC(C3(C)COCCO3)=O)CC2)C1 98601,C1(CCNC(=NCCC)NC2CCNC(=O)C2)CCC2(CC1)OCCO2 98602,c1(C2C(C(=O)NC3(C)CC(NC(C4(Cl)C(C)(C)C4)=O)C3)C2)ccncc1F 98603,c1(C(N(CC(C)N(C(=O)C(c2ccc(C(F)F)cc2)C)C)C)=O)cc(Cl)cn1C 98604,C1(CNC(Cc2c(C)nc[nH]2)=O)CN(C(=O)CC2CCC(C)C(C)C2)CCCO1 98605,Cc1nc2ccccc2n1Cc1nc(-c2cc[nH]n2)nn1C1CC(OC(C)C)C1 98606,CC(C)CC(CNC(c1cnn[nH]1)=O)C(=O)N(C)CCc1ncon1 98607,N1(C(COCCOC)=O)CC(CO)C(C)C1.c12cc(n(C)c1)CCn1cc-2nn1 98608,c1(CC(=O)Nc2ccsc2NC(c2cc(O)no2)=O)cccc(F)c1[N+](=O)[O-] 98609,C1(CNC(C2(CC=C)CCCC2)=O)CC2CCCCC2N1C(=O)C(CCC)OC 98610,C1(CNC(C2(NC(C(CC3CCC3)OC)=O)CCSC2)=O)CCCCC1(C)C 98611,c1(C(=O)NCCCCN(C(Cc2cc(C)sc2C)=O)C)cc(O)nc(O)n1 98612,c1(C(N(CC(CNC(CCC)=O)(C)C)CC)=O)cc(C)nc(N(C)C)n1 98613,C1(NC(C=C(C)C(C)(C)C)=O)CCC(NC(=O)CC(O)c2ccccc2)CC1 98614,Cc1c(C(=O)NCC2(CNC(C3CC4C(C3)C4(C)C)=O)CCCC2)cccc1N 98615,Cc1cc(C(=O)NC2CC2CNC(c2ncc(Cl)s2)=O)cc(C)c1Cl 98616,C1(NC(=O)CC2COCCO2)CCOC12CCN(c1ncc(O)cn1)CC2 98617,C(=O)(C1=CC(C)(C)C1)N1CCC(CC(C)NC(=O)CCC2CCCCO2)CC1 98618,c1(OC)c(NC(C2CC(F)CN(C(=O)CCC3CC3)C2)=O)cccc1Cl 98619,CC1(C)Cc2c(cnn2-c2ccccc2)CN(C(c2cc(I)cs2)=O)C1 98620,C1(CCNC(CCCNC(N)=O)=O)CCN(C(=O)Cc2ccsn2)CC1 98621,O=S1(=O)CC(N2CCN(Cc3ccccc3)CC2)C(CNc2cc[nH]n2)C1 98622,CCCCS(=O)(=O)CC(=O)N1CC2C(CN(C(=O)Cc3cn(C)cn3)C)C2C1 98623,n1(CCC(=O)NC2CN(C(C3CC3C(F)F)=O)CC23CC3)ncc2c1CCCC2 98624,N1(C(C=CC)=O)CCC(C(C)NC(C2(CCS(N)(=O)=O)CCC2)=O)CC1 98625,C1(NC(c2ccc(C)o2)=O)CC2CCC1CC2NC(C12CCCC1C2)=O 98626,N1(C(C2C(NC(CNC(C3C(C)C3)=O)=O)CCO2)=O)CCC(C(=O)N(C)C)CC1 98627,C1(CC)CN(C(=O)Cc2ccnc(Br)c2)CCN1C(c1nc(O)c(C)s1)=O 98628,C1(C)(C(=O)NC2C3CN(C(C(c4ccccc4)N(C)C)=O)CC32)C(C)(C)C1(C)C 98629,N1(C(C2(F)C(C)OCC2)=O)CC2CN(C(=O)COc3cccc(F)c3)CC(C1)O2 98630,N1(C(C2C(C=C)C2)=O)CC2CCC1C(NC(=O)COc1cccc(F)c1)C2 98631,C(=O)(C(CC)(CC)C(C)C)NC(c1ccnn1C)C(N1CCC(=CCC)C1)=O 98632,c1(C(N2CCC(CC)(NC(=O)CCCCF)CC2)=O)cccc2c1C(=O)NC2=O 98633,c1(N2CCCC(C)CC2)nc(=NCCCc2ccccc2Br)[nH]c2ccccc12 98634,C(c1cccnc1)=C(C(=O)NC1C(NC(c2[nH]cc(C(=O)OC)c2)=O)CCC1)F 98635,N1(C(C2(CCCC)CCC2)=O)CCC(C=CC(=O)Nc2csnc2OC)CC1 98636,C1(C(N2C(C(N(CC(C)(C)N(C)C)C)=O)COCC2)=O)CC2(C1)CC2(F)F 98637,c1(C(=O)NC(C)CN(C(=O)CSc2nc[nH]n2)C)ccc(F)c(Cl)c1N 98638,N1(C(C2(C)CC(F)(F)C2)=O)CCC(O)C(NC(C2CC23CCC3)=O)C1 98639,c1(NC(N2CCOC(C3CC3)CC2)=O)ccnc2c1CCC2 98640,c1(CCC(N2CC(C(C)NC(=O)CC(O)C3CC3)C2)=O)cccnc1Br 98641,c1(C(=O)NC2CC(CNC(C(Cc3ccccc3)OC)=O)C2)cccc(C)c1F 98642,C12(CNC(C3N(CC)CC3)=O)COCCN1C(=O)CN(C(c1cnc(S)[nH]1)=O)C2 98643,c1(CC)ocnc1C(=O)NC(C)C(CO)NC(c1cc(F)n[nH]1)=O 98644,C12(NC(C(CC)CC)=O)CC3CCC(C1C2)N3C(=O)Cc1cn(C)nn1 98645,c1(N2CCN(c3ccc(CC)cc3C)CC2)ncnc2cc(C#N)ccc12 98646,N1(C(Cc2c(C)ncnc2C)=O)CCC2CN(C(=O)CC3NC(=O)NC3=O)C2C1 98647,c1(N2CCCC(C#N)CC2)nc2c(c(=NC3CCc4nn[nH]c4C3)[nH]1)COC2 98648,C(=O)(C(C)(C)C(C)O)NCC1(C(C)NC(c2nc(CC)sc2)=O)CC1 98649,c1(CC)cc(CNC2CCC2C)on1 98650,c1(C(N2CCCC(NC(C34CCC(C3)C4)=O)C2)=O)ccc(Cl)cc1NCC1CC1 98651,N1(CC)CCOC(C(N2CCC(CNC(C3(COC)CC3)=O)C2)=O)C1 98652,Cc1cc(C(=O)N(CCCN(C(=O)CC2CC2C)C)C)c(C)n1-c1nccs1 98653,C1(CC(=O)N(CCCNC(=O)CC2(O)CCC2)C)CCOC(C)(C)C1 98654,C1(CNC(C(CC=CC)C)=O)(NC(c2cc(C)cc(O)n2)=O)CCC(C)(C)CC1 98655,c1(C(c2nnnn2CSc2ccccc2)NC(CCC)C)cc(Cl)n(C)n1 98656,c1(C(N(CC(CC)NC(=O)CCCn2cncn2)C)=O)cnn2cccc(Cl)c12 98657,C1(CCNC(c2c(Cl)cn(CC)n2)=O)CCN(C(C2CC=CC(O)C2)=O)C(C)C1 98658,C1(C(N(C)Cc2ncc(C)o2)=O)CC12CC(NC(=O)CC1CCOC1C)C2 98659,c1(C(=O)OCC)cc(C(N2CCCC2CNC(c2c[nH]nc2CC)=O)=O)nn1C 98660,n1(CCC)ncc(C(=O)NC(CNC(C2CCCN2CC(C)C)=O)C2CC2)c1C 98661,CC(CCN(C)C)C(=O)NC1CC(C)N(C(=O)CCC(=O)N(C)C)C1 98662,C1(CN(C(c2n(CC)nnc2)=O)C)COCCN1C(c1nncs1)=O 98663,C#CCC(C)(C(=O)NC1CC2CC3C(C2)C13)NC(=O)CC1CCCC(C)C1 98664,C(=O)(CC(CC)NC(=O)C(O)C1CC1)NCC(=O)OCC=C 98665,C1(NC(C2C(C(C)(C)C)C2)=O)CC2CC1N(C(C1CN3CCC1CC3)=O)C2 98666,c1(CCC)nc(C(=O)NC(C2CCN(C(=O)CSC3CC3)C2)(C)C)co1 98667,N1(C(COCCCOC)=O)CCCC(C2CCN(C(=O)COCCF)CC2)C1 98668,C=CCCCC(=O)NCC1CCCC(CNC(=O)CCc2cnc(C3CC3)o2)C1 98669,C1(C)(NC(Cc2nnc(C)s2)=O)CCCN(C(C2CC(C)(C)CCO2)=O)C1 98670,C=CC1(NC(=O)C(F)CC2CN(C(c3cccc(CO)c3)=O)C2)CCOCC1 98671,c1(NCc2ccc(OC)cc2F)cc(S(=O)(=O)N(CCCO)CC)ccc1C#N 98672,CC#CCC(C)NC(=O)CN(CCC)C(c1cccnc1)=O 98673,C1(CNC(c2nc(CC)sc2)=O)CCC(C)N(C(C2(c3cccnc3)CC2)=O)C1 98674,C(=O)(C(CN=[N+]=[N-])NC(c1n[nH]c2c1CCC2)=O)N(C)CC1CCCN(C)C1 98675,N1(Cc2cn(CCCNC(C(CC=C)NC(C)=O)=O)nn2)CC(O)CCC1=O 98676,CN=c1ncc(-c2cnc(NCc3ncc(C)cc3F)nc2)c[nH]1 98677,CCC1=C(C(=O)N(C)CC2CCCN(C(c3cnncc3NC)=O)C2)CCCO1 98678,N1(CCC(=O)NC23CC(C2)N(C(c2cnoc2C2CCC2)=O)C3)C(=O)CCC1=O 98679,c1(C(=O)NCCN(C(=O)CC2C(=O)NN=C2C)CC)ccc(P(C)(C)=O)s1 98680,C1(C(N2CC(C)N(C(=O)C=Cc3ccccc3)CC2)=O)CC2(C1)NC(=O)NC2=O 98681,c1(C(=O)NC2CCC(NC(C3C(C)=C3)=O)C2)c(C)c(C)nn(C)c1=O 98682,c1(CCNC(c2cnn(C)c2OC)c2n(CCOCC)nnn2)ccccc1C 98683,c1(C(C(=O)NC)N(C)CC2(C)CCCO2)cn(C)c(=O)n(C)c1=O 98684,C(=O)(C#CC1CCOC1)N(CCOCCNC(c1cnc(C(C)C)s1)=O)C1CC1 98685,N1(C(C2(C)N(C)CCC2)=O)CCCC(CO)(CNC(=O)CCc2cnccn2)C1 98686,c1(CCCCC)cc(C(=O)NC2(CO)CN(C(c3cc(C(N)=O)co3)=O)C2)n[nH]1 98687,c1(C(C(=O)NC(C(C)NC(C(C)Cn2ccnc2)=O)CO)(C)C)ccccc1Cl 98688,C1(CNC(C2(CF)CCC2)=O)CCCC1C(=O)NCc1cscn1 98689,c1(COC)ncc(C(=O)NC(C)(CNC(C2CNC(=O)N2)=O)C2CCC2)s1 98690,CC(N=c1nc(N2CCC(CCC(C)O)CC2)c2c([nH]1)CSC2)c1cscn1 98691,N1(C(c2cc(Cl)ccn2)=O)CC2(CCCN2C(=O)N(CCCl)CCO)C1 98692,c1(NC(C(=O)NCCC2CCCS(=O)(=O)C2)=O)cccc2c1OCCCO2 98693,N1(C(C2CN(C)C(=O)C2)=O)CC2(CCCC(CNC(=O)C(F)=CCCF)O2)C1 98694,c1(NC(=O)NCc2cc(Br)nn2C2CCCCO2)cc(-c2ccccc2)ccn1 98695,c1(NC2CN(C(CC(C)c3ccccc3)=O)CC2C)cccc(F)c1C#N 98696,C(=O)(CS(=O)(=O)C1CCCC1)NCC1CN(C(C(CSC)OC)=O)C2(C1)CCC2 98697,N1(C(CNC(c2ccc(Cl)cc2)=O)=O)CC2CC2(NC(C2C3CCCCC23)=O)C1 98698,C#CCC(C)(C(=O)NC1CC1(C)CCC)NC(=O)CCOC1CCCC1 98699,C1(C(N2CCCCCC2)C(=O)NC(C)Cc2ccccc2)C2CCOCC12 98700,C(c1c(C)cccc1C)=CC(=O)NC(CCC)CNC(C1(n2cnnn2)CC1)=O 98701,c1(C(=O)NC(CC=C)CNC(C2CCCCCN2C)=O)cc2cc(C)ccc2o1 98702,C1(C)(CCNC(C2N(CC)CCC2)=O)CCN(C(=O)CCc2cccn2C)C1 98703,c1(COC(c2ccc(CN3CCCC3=O)cc2)=O)cccc2sccc12 98704,C(CC(F)F)(C(=O)N(C12CCC(CC1)CC2)C)n1cc(-c2cccc(C)n2)nn1 98705,Cc1nc2cc(C(N3CC(NC(=O)CC(C)P(C)(C)=O)C(O)C3)=O)cc(O)c2[nH]1 98706,C1(C(=O)NCCN(C(C2(COC)CCCCO2)=O)C)CC(=O)N(OC)C1 98707,c1(CC(=O)NC2CC(C)(NC(CCC3N(C)CCC3)=O)C2)cc(F)ccc1O 98708,c1(NC(C(c2cc(CC)on2)N(C(C)CCC#N)C)=O)cccc(OC)c1 98709,c1(CNCC2(F)CCCN(C(C3CC3F)=O)C2)sc(Br)c2c1OCCO2 98710,c1(C(N2C(CC(=O)Nc3c(O)ncnc3O)COCC2)=O)ccn2nccc2c1 98711,C(C(C(=O)NCC(C1CCCC1)NC(c1ccn(C)n1)=O)N(C)C)N(C)C 98712,c1(C(N(C)CCN2CCN(C(C3CC3C(F)F)=O)CC2)=O)cnc2[nH]ccnc1-2 98713,c1(NC(c2cccc(Br)c2)=O)ccc2[nH]cc(-c3ccc(C(=O)O)c(F)c3)c2c1 98714,c1(C(N(CCCOCCN(C(C(C)SC)=O)C)C)=O)c(C)oc2ccccc12 98715,CC(CC(=O)N1CCOC(CC(=O)NCC(F)Cl)C1)C(C)(C)C 98716,CC1(C)CC(C(=O)NC(C)(CO)C2CC2)CN(C(C2(C3CCCC3)CC2)=O)C1 98717,Cn1nc(C2CC2)c(Br)c1C(N1C(C(=O)O)CSC1c1ccncc1)=O 98718,Cc1nc(C(C)(C)C)nc(O)c1C(N1CCCC(C)(NC(C2CC2CF)=O)C1)=O 98719,C(=O)(C(C(C)(C)C)N1CCCC1=O)NC1CCN(C(c2ccc(OC)cn2)=O)C1 98720,N1(C(COCCCC(C)C)=O)CC(CNC(C2CCC(N(C)C)CC2)=O)C(C)C1 98721,N1(C(C(C)(C)C2CCCCC2)=O)CCC(O)(CCNC(=O)CSC(F)F)C1 98722,Cc1ccc(C(N2CC(NC(c3ncoc3C(C)C)=O)CC(C)C2)=O)c(N)c1C 98723,N1(C(C(N2CC(C)C2)C)=O)C(C)CN(C(=O)CC2CCC(C)(C)O2)CC1C 98724,C(=O)(C#CC1CCOCC1)NC1C(NC(c2c(C)noc2C)=O)CCCC1 98725,C1(N(C(=O)CSCCOC(C)C)CCC)CCN(C(=O)C(COC)N(C)C)C1 98726,C#Cc1cccc(C(=O)NC(CNC(c2ccc[nH]2)=O)CCOC)c1F 98727,C=CCCN=C(NCc1ccc(O)cc1Cl)N1CCCC(CC)C1 98728,C(=O)(C(C)(C)CC(C)(C)C)N1CCCC(O)(CN(C(C(C)C(C)(C)C)=O)C)C1 98729,c1(CN2CCC3(C(C(=O)Nc4ncc(C#N)cn4)C3)C2)ccc([N+](=O)[O-])c(Br)c1 98730,c1(C(=O)NCC2N(C(c3cc(CC)c(Cl)cc3)=O)CC2)ccc(N)c(C)c1C 98731,c1(CN2C(C(N(CCCCC=C)C)=O)CC(O)C2)cccc(C(C)(C)C)c1O 98732,c1(C(N2CC(NC(CC(CC)C)=O)C(C#N)C2)=O)cccc2c(Br)n[nH]c12 98733,N1(C(c2ccc(OC)cc2)=O)CCN(C(=O)Nc2cc(Br)ccc2OC)CC1C 98734,c1(C(N(C)CC2(O)CCN(C(Cc3nc(CC)sc3)=O)C2)=O)cccc(N)c1C 98735,N1(C2CCN(C(C(C)C)=O)CCC2C)CCC2(CC1)OCCc1ccsc12 98736,c1(C(=O)NCC(CNC(=O)C(C)(O)C2CCC2)OC)cc(F)c(Cl)cc1Cl 98737,c1(C(N2CCC(NC(C(CCCC)CC)=O)C2)=O)ccc2c(=O)n(C)c(C)cc2n1 98738,c1(OCC)ccc(CN(c2cc(NCC3CC(O)CN3C)ncn2)C)c(F)c1 98739,C1(C(N(C)CC2CCN(C(CCC=CCC=C)=O)CC2)=O)Cc2ccccc2C1 98740,N1(C(C=C(C)C(C)(C)C)=O)CC(O)CC1CNC(=O)C(O)C1CC1 98741,c1(C(=O)NCC(C(=O)NC(CCC)C(=O)N(C)C)O)cc(C)c(C)nn1 98742,N1(C(c2cccc(SC)c2)=O)CC2(C1)OC1(C)CC2(NC(C2CCC(C)O2)=O)C1 98743,Cc1cnn(C)c1CNC(C1C(C)CCN1C(=O)CC(C)(C)C)=O 98744,C1(C(N(C2CCOC2)C)=O)(CF)CCN(C(c2ccn(C(F)F)n2)=O)C1 98745,N1(C(CCOCCNC(c2cc(C)nnc2)=O)=O)Cc2ccc(O)cc2C1 98746,CCCC(C)CCCC(=O)N(CC(O)CNC(=O)Cc1csc(CC)n1)C 98747,C1(CC)CN(C(=O)C(O)COCC)CC1NC(c1cc(-c2ccccc2)no1)=O 98748,C(C)(C(=O)NCCC1CN(C(C2(N(C)C)CC2)=O)CCCO1)(C(C)C)OC 98749,C1(C(=O)NCCN(C(c2nc(OCC)oc2)=O)C2CC2)CCCC12CC2 98750,C1(CNC(C(C)NC(c2ccc(C)cc2Br)=O)=O)CC(C)c2ccccc2N1 98751,N#Cc1cnc(N2CCC(F)(F)C(CNC(c3cccc(Cl)c3Cl)=O)C2)c(Cl)c1 98752,N1(C(c2sc(C)c(Br)c2)=O)CCC2CN(C(c3c(F)cccc3Br)=O)CC12 98753,C1(C(=O)NCC(C)OCC=C)(OC)CCN(C(C2COCC(C)O2)=O)C1 98754,Cc1cn2ccnc(C(=O)NC3CCCC3CNC(c3cncs3)=O)c2n1 98755,CC(=O)CCCCC(=O)NCC(CNC(=O)C(c1ccnn1C)C)CO 98756,CONC(=O)C(=O)NCCC1CCC(NC(C2C3CCCCC23)=O)C1 98757,C1(C(N(CCC(C)NC(=O)Cn2cnc(C(N)=O)n2)C)=O)C(C)(C)C1(F)F 98758,c1(C(C)=O)cc(C(N2CCCC(NC(=O)Cc3cc(C)no3)CC2)=O)ccc1O 98759,C(=O)(CN1C(=O)Cc2ccccc21)NC1CCCC(NC(c2c(OC)n[nH]c2)=O)CC1 98760,C1(NC(c2c(OC)cccc2)=O)COC2(CCN(C(c3coc(CO)c3)=O)C2)C1 98761,c1(CN2CC(OC)C(NC(=O)CSC(C)=O)CC2)c[nH]c2cc(Br)ccc12 98762,c1(CC(N2CCC(NC(Cc3c(C)cccn3)=O)C2)=O)ccc2oc(O)nc2c1 98763,C1(C(N(C(C)C(=O)N(C)CCc2cc[nH]n2)CCC)=O)CCC(CC)O1 98764,N1(C(C(C)CO)=O)CCC2(CCCC2NC(=O)C=CC2CCOCC2)CC1 98765,C1(C(=O)NCc2c(C)nccc2)CCC(O)CN1C(c1cc(C#N)oc1C)=O 98766,c1(NC(=O)NC)cccc(C(=O)NCC(C)(C)NC(C2CCC(O)C2)=O)c1 98767,C1(CC#C)(C(=O)N(C2CCCCC2O)C)CCN(C(C2CCOC2C(C)C)=O)C1 98768,C12(NC(=O)CCC3CCCO3)CC3CCC(C1C2)N3C(=O)CC1(C(F)(F)F)CC1 98769,N1(C(C2(OCC)CCSCC2)=O)CCCC(NC(C2(C)CCCOC2)=O)CC1 98770,c1(C(=O)NCCOCCN(C(c2cc(C(C)=O)[nH]n2)=O)C)noc2c1CCCC2 98771,c1(C(=O)OC)cccc2c1N(CCC(C(Cl)Cl)NC(=O)OC(C)(C)C)CCC2 98772,c1(C(=O)NC2CC(CNC(C(CC)OCC)=O)C2)ccc(OC)cc1F 98773,C(=O)(CC(C)CC(C)(C)C)NC(CCNC(c1c(C)ncs1)=O)C(C)C 98774,c1(C(=O)NCCN(C(=O)C(F)CC2CCC2)C2CC2)cc(OCCF)cc(F)c1 98775,n1(CC(N2CCn3nc(Br)nc3C2)=O)ncc2c(c1=O)CCCC2 98776,C1(C(N2CCC(=C)C2)=O)CC2CC1CC2NC(c1cc(C)nnc1C)=O 98777,C1(C2CCN(C(C3CCCOCC3)=O)CC2)(NC(C(C(C)C)NC(C)=O)=O)CC1 98778,C(=O)(C(C)C(=O)NC1(CO)CN(C(C2(C(C)C)CCC2)=O)C1)OC 98779,C(=O)(C1c2c[nH]nc2CN1C(=O)CC(=O)N(C)C)N(CCC)C(C)C 98780,C1(CNC(CC2CCCN(C)C2)=O)CN(C(=O)Cc2cccnc2)C(C)(C)C1 98781,c1(C(N(CCC)CCNC(C2(F)CCC2)=O)=O)cc(C)c2c(c1)CCC2 98782,C1(CC)CN(C(c2cnns2)=O)CC1NC(c1ccc(CS(N)(=O)=O)cc1)=O 98783,CC1Cn2nccc2CN1C(=O)CC12CCC1CN(C(c1ccn(CCF)n1)=O)C2 98784,C#Cc1cnn(C)c1C(N1CCC(CCN(C(=O)COC(C)C)C)CC1)=O 98785,c1(SC)cccc(C(N2CCC(NC(c3cncc(C)n3)=O)C2)=O)c1O 98786,N1(C(c2ccc(SC)o2)=O)CCC2(COC(CNC(C3(C)CCSCC3)=O)C2)C1 98787,c1(C(=O)NC(C)CNC(C2(c3ccc(Cl)cc3)CCC2)=O)c[nH]cc(Br)c1=N 98788,c1(C(N(CCNC(C2CCC(COC)O2)=O)CC)=O)c(Cl)ccc(OC)c1N 98789,c1(C(N2CC(F)CC(NC(c3n(C)c(CO)cc3)=O)C2)=O)c(Cl)ccc(Br)c1F 98790,C1(CNC(c2ccc(I)c(O)c2)=O)CCNCC1(F)F 98791,C1(NC(c2cncc(C)n2)=O)CCN(C(=O)CC2CCC(=O)N2)CC1C 98792,C(=O)(C1=C(C)CCOC1)N1C2(C(=O)NC(c3nn[nH]n3)CC)CC2CC1 98793,c1(C(=O)NCC(CNC(C2CC(C)(CC)C2)=O)F)cc(C)ccc1[N+](=O)[O-] 98794,CC(C)C(F)(F)CC(=O)NC1CCC(C)N(C(c2cc(N)c(Cl)cn2)=O)C1 98795,C1(CC(=O)NCCC(CNC(=O)CC2OCCC2C)OC)CCCN(C)C1 98796,c1(N(C)C)cc(NC(=O)C(c2ccc(Cl)s2)NC(=O)OC(C)(C)C)cc(Br)c1 98797,c1(CC(=O)NCCC(C)N(C(CC(C)C)=O)C)coc2ccc(F)cc12 98798,C1(NC(c2n(CCSC)nnn2)C2CC(F)(F)C2)C(C)CCC1C 98799,c1(CC)cccc(C(=O)NC2CCC2CNC(C2(C)C=CCC2)=O)c1N 98800,c1ccc(C)cc1.C#CCCCN(CC(=O)NCC(=O)NCCC(=O)OC)C 98801,C1(C(=O)NCC(CCNC(C2(C)CC(F)(F)C2)=O)O)COC2(CCC2)CO1 98802,c1(CC)cc(C(=O)NCCCNC(=O)C(c2ccc(C)cc2)C)cn(C)c1=O 98803,c1(C(N2CC(C)N(C)C(C)C2)=O)ccc(S(=O)(=O)NCC2CCOCC2)cc1 98804,N1(C(C(C)CN(C)C(c2cnoc2C2CC2)=O)=O)CC2CCN(C)C2C1 98805,C(S(=O)(=O)C(C)C(=O)N1CCN(C)C(CF)C1)c1c(-c2cccc(OC)c2)n[nH]c1 98806,Cc1c(C(N2CC3C(N(C(=O)C(F)CC4CC4)C)C3C2)=O)oc2c(Cl)cccc12 98807,c1(C(N(C(C)CNC(=O)Cc2conc2C)CC)=O)cc(F)ccc1N 98808,c1(C(C)=O)cc(=NCC2CN(C(C3CC(C)CO3)=O)CCO2)[nH]cn1 98809,N1(C(C2CC=C(C)CC2)=O)CCCC(C2CC2NC(=O)C(C)(C)C(F)F)C1 98810,N1(C(CCCOCCOCC#C)=O)CC2CC(NC(c3ccc[nH]3)=O)C1C2 98811,c1(NC(C(C(C)NC(C2C(C(C)C)CCO2)=O)(C)C)=O)cccc([N+](=O)[O-])c1 98812,C12(C(C)C)CCC(NC(=O)C(Cn3cccn3)NC(=O)CN3CC=CC3)C1C2 98813,c1(C(N2C(CC)C(NC(=O)CCCC(F)(F)F)CC2)=O)ccc2nn[nH]c2c1O 98814,C(C)(C)(CC(F)C(=O)NC(C1CCOC1)CO)NC(CC1CCN(C)C1=O)=O 98815,c1(C(N(CCCNC(=O)C(C2CC2)C2CC2)CC)=O)c(C)nn(C2CC2)c1Cl 98816,CN=c1[nH]cc(C(N2CCCC(NC(=O)CCCSc3ccc(F)cc3)C2)=O)s1 98817,C1(C(N(CC(COC)O)C)=O)COCCN(C(c2ccnn2C(F)F)=O)C1 98818,Cc1cc(C(N2CC(N(C)C(c3cnoc3C)=O)C3(CC3)C2)=O)nc(N(C)C)n1 98819,C1(S(C)(=O)=O)(C(=O)NC2CC(C)(NC(CC3C(C)C3(F)F)=O)C2)CC1 98820,N1(C(Cc2c(C)ocn2)=O)CCC(C)(C)C1C(=O)NCCN1CCOCC1 98821,c1(CC)cn2c(n1)CC(C(=O)NCC(CC)NC(c1ccc(=O)n(C)n1)=O)CC2 98822,c1(N(C)C)ccnc(C(=O)NCCC2CCCN2C(=O)C=Cc2ccco2)c1 98823,C1(NC(=O)CC2CC=CC2)CCC(O)CN(C(C2(c3ccc(Cl)cc3F)CC2)=O)C1 98824,c1(OC)ccc(C=CC(=O)NC(C)(C)CNC(C2CCCC(O)C2)=O)cc1F 98825,c1(C(N2CCC(N(C(=O)CN(C)C3CC3)CC)C2)=O)cccc2nsnc12 98826,Cc1cc(-c2cnccc2C(=O)Nc2cnn(CCO)c2)ccc1OC(F)(F)F 98827,N1(C(C)CC(F)(F)F)CC(C)(C)CCC1CNC(=O)CCc1cccc(F)c1F 98828,C1(NC(CCN(C)CC)=O)CCN(C(C2(n3cnnn3)CCCCC2)=O)CC1OC 98829,Cc1sc(C(=O)Nc2ccc(-n3cccc3)cc2)c(C)c1Br 98830,c1(NC(=O)NC2CCCN(CCC(=O)OC)C2)ccc(F)cc1C 98831,C(C(C(=O)N1CCC(CN(C)C)C1)n1cc(-c2csnn2)nn1)OCC 98832,CC(C(=O)NCc1cccc(COC2CCOCC2)c1)C(C)(C)C 98833,C(=O)(CCCCN(C)C)NC(CN(CC(=O)N(c1ccccc1)CC)C)C 98834,C1(C)(C(C)(C)C)CC(C(=O)NCC(O)CNC(C2CSCCS2)=O)C1 98835,C1(NC(=O)C(O)C2CCCC2)CCC2CN(C(c3cc4c(s3)CCC4)=O)CC2C1 98836,C1(CCC#C)CCCN(C(=O)CCC(C)NC(=O)C(C)C(C)C)C1 98837,Cc1c(C(=O)NCCCCNC(c2csc(C)c2C)=O)cc(F)cc1Br 98838,N1(C(CCCOCC=C)=O)CC(NC(c2nc(O)c(C)s2)=O)C(n2ccnn2)C1 98839,C1(COC)CCCC1NC(=O)CC1(C)CCN1C(C)=O 98840,CCC(CC(=O)NC1CCC12CN(C(c1cc[nH]n1)=O)C2)C(C)C 98841,c1(-c2onc(CN(C(=O)OC(C)(C)C)CC)n2)cc(CO)cc(C)c1 98842,C1(CNC(c2c(C(C)C)csc2)=O)CCCCN(C(=O)COc2ccsn2)C1 98843,C(C(C)CC(C)C)NC(c1ccncc1)CC 98844,N1(C(C2CCN(C(c3nc(C)c(C)s3)=O)C2)=O)CCC(C)C2(CCC2)C1 98845,C1(C)(CNC(c2[nH]cc(C)c2)=O)CN(C(=O)CCNc2ccccn2)CCO1 98846,C1(NC(c2c(C)n(C)nc2)=O)CC12CCN(C(C1CC3CC3C1)=O)CC2 98847,n1(CC)nc(C)c(C(=O)NCC2(NC(=O)C(C)S(C)(=O)=O)CCCCC2)c1C 98848,C1(C)(C(=O)Nc2c(CC)noc2)CCCN1C(=O)CCCn1ccnn1 98849,c1(OC)cc(C(=O)NCC=CCNC(C2(CO)CCCC2O)=O)cnc1C 98850,C1(CNC(c2cc(OC)no2)=O)N(C(=O)Cc2cc(C)cc(F)c2)CCC1(C)C 98851,N1(C(C(C=C)O)=O)CC(F)CC1CC(=O)NCc1cncc(F)c1 98852,c1(OC)ncccc1C(=O)NCC(C)(C1CC1)NC(c1ccoc1Cl)=O 98853,CCCCCC(O)CC(=O)NCCN(C(=O)CC(C)C)Cc1ccccc1 98854,c1(CC(=O)NC2CN(C(c3c(C#C)c[nH]n3)=O)CC2C)coc2cc(F)ccc12 98855,C12(CO)COCC(Nc3ncc(Br)cc3C(F)(F)F)(C1)C2 98856,C(=O)(C(C(C)C)n1cncn1)NC(CCCNC(CC1(C(=O)OC)CCCC1)=O)C 98857,c1(CNC(C(CC)n2ccnc2)=O)cnn2c1CN(c1nnc(C3CC3)o1)CC2 98858,Cc1ccc(NC(=O)C(=O)N(CC(C)CNC(=O)CNS(N)(=O)=O)C)cc1 98859,C1(NC(CCC#CC)=O)CN(C(C2CS(=O)C2)=O)CC1(C)C 98860,N1(C(C)C)CCCC(CN2CCCC2c2cc(Br)cs2)C1 98861,S(=O)(=O)(c1c(C)noc1C)NCC(=O)NCC1C(NC(CCCCCC=C)=O)C1 98862,c1(C(N2C(CNC(C=CSC)=O)CC3(CC3)C2)=O)cc2c(Cl)cccc2s1 98863,c1(C(=O)NCC2C(NC(CCC#CC)=O)COC2)ccc(Cl)c2c1OCCO2 98864,N1(C(CCCC#CC)=O)CC2(C1)C(NC(=O)C#CC1CCOC1)CCS2(=O)=O 98865,N1(C(CCC=C(C)C)=O)CC(N=[N+]=[N-])CC1C(=O)NCCN1CC=CCC1 98866,C(=O)(CCC1=NNC(=O)CC1)NC1CN(C(CN(CCC)C)=O)C2(C1)CCOC2 98867,CC(C)(C)C(O)C(=O)NC1CN(C(C23CC2CNC3=O)=O)CC12CC2 98868,N1(C(C(=O)NC(C(=O)NCC(=C)C)C2CC2)C)CCOCC1 98869,C1(C(=O)NCC(C)CNC(C2(CO)CCOCC2)=O)(COC)CCCOC1 98870,N1(C(Cc2ccc(C)s2)=O)CCC2CN(C(C34CCC(=O)N3CCS4)=O)CC2C1 98871,C(=O)(CCCCSC)NC(C1CN(C(c2ccc(COC)o2)=O)C1)C 98872,c1(CN2C(c3ccc(CC)o3)CCOCC2)cccc(S(F)(F)(F)(F)F)c1 98873,CCCC(CCC)=CC(=O)N(C(CNC(=O)C(C)(C)n1cnnn1)CC)C 98874,CC(=O)C(C)CC(C)C(=O)NC1CCC(CNC(C2(F)CCCCC2)=O)CC1 98875,C1(NC(C(CCSC)NC(N)=O)=O)C2CCC1N(C(c1ccsc1Cl)=O)C2 98876,c1(CC(=O)NCc2occ(NC(=O)OC(C)(C)C)c2)cccc(Cl)c1I 98877,N1(C(CC(C)(C)F)=O)CCN(C(=O)C=Cc2nccs2)CC1C1CCC1 98878,C1(NC(C2C(=C)C2)=O)CCC12CCCN(C(C1COCCN1C=O)=O)C2 98879,c1(CC(C(N2CC(c3cn(CC(COC)O)nn3)(F)C2)=O)OC)ccc(C)cc1 98880,C1(NC(N(CCC)C)=O)CC(=O)N(OCc2ccccc2)C1 98881,N1(C(C(C)NC(C)(C)C)=O)CC2CC(NC(c3coc(C(F)F)c3)=O)C1C2 98882,c1(N2CCC(SC(F)(F)F)C2)[nH]c(=NCc2cn(C3CC3)nn2)nc2sccc12 98883,C1(CC(N)=O)CN(CC(c2ccc(-c3ccccc3)cc2)O)CCO1 98884,C1(C)(C(N2CCC(CNC(C(F)(F)C3(OC)CCC3)=O)C2)=O)CNC(=O)C1 98885,C1(NC(c2cn(CC3CCCO3)nn2)=O)COCCC1NC(C1(CO)CCC1)=O 98886,C(=O)(C(C)(C)CC#N)NCC1(C(C)(C)O)CN(C(CSCCC)=O)C1 98887,c1(C(C(=O)NCCOC)N(C2CCCC2)CCOC)cc(OC)c(Cl)cc1F 98888,C1(F)(CNC(c2n(CC)nnc2)=O)COCCN(C(=O)CS(=O)(=O)NC)C1 98889,C=C(C)CCNC(=O)COCCNC(C1CC1(C)C)=O 98890,C(=O)(CC(C)c1cccnc1)NCC1(NC(C(C)C)=O)CCC1 98891,c1(NC(C2CC3OC2C2CC32)=O)nc(=O)c(Br)c[nH]1 98892,C1(CNC(c2cc(C)n(C)n2)=O)(CO)CCCN(C(C2CCN(C)C(C)C2)=O)C1 98893,N1(CCNC(C2OCCN(CC)C2)=O)CCCN(C(=O)CC2(N(C)C)CCC2)CC1 98894,C1(NC(CCC=C)=O)COC2(CCN(C(=O)Cc3cn4c(C)csc4n3)C2)C1 98895,N1(C(C2(OC)CCSCC2)=O)CC2CC1CN2S(C)(=O)=O 98896,C(=O)(C1=CC2C=CC(C1)C2)N1CCC(NC(C2(CC)CC2)=O)C(C)C1 98897,c1(Cn2ncc(C)c2)ccc(C(=O)NC2CC2CNC(=O)CC23CC(C2)C3)cc1 98898,N1(C(CCc2c(C)n(C)nc2)=O)CCCC(C)(NC(c2ccn(C)n2)=O)C1 98899,c1(CC)cnn2ccc(C(N3CCC(C)N(C(=O)C(CO)C(C)C)CC3)=O)nc12 98900,c1(CC(=O)NC2CN(C(=O)C3=CCCS3)CCC2CO)cccc2ccccc12 98901,N1(C(C)=O)CCCC(C(N2CC(NC(=O)Cn3cc(C(C)O)nn3)C(F)C2)=O)C1 98902,C1(C(N2C(C)CC2)=O)CCCC(NC(=O)COCC2CC2)C1 98903,C1(C2(O)CCC2)(C(=O)NCC2CCC(NC(C(n3ccc(C)n3)(C)C)=O)C2)CC1 98904,CC1=NS(=O)(=O)N(C)C=C1C(=O)N1CCOC2CN(C(=O)CCS(C)=O)CC12 98905,N1(C(c2c(CCC)nco2)=O)CC2CC(NC(c3occc3CN(C)C)=O)C2C1 98906,CCCC(C(=O)NC(CCC)CCCNC(=O)CCCOC(C)=O)OC.OCC 98907,C(=O)(C(O)CC(F)(F)F)N1CCC(N(C(=O)COCCCN(C)C)CC#C)CC1 98908,c1(OCc2n(C)ccn2)ccc(CNc2cccc(-n3ccnc3)c2)cc1 98909,Cc1nn(C)c(=O)c(C(N2C3CCC2CC(NC(c2cnccn2)=O)C3)=O)c1C 98910,c1(C(N2CCC(CC)C2CNC(=O)Cc2ccn(C)n2)=O)cn2c(n1)CCC2 98911,N1(C(CC#C)=O)CCC2(CCCN(Cc3cc([N+](=O)[O-])ccc3O)C2)CC1 98912,S(=O)(=O)(c1ccccc1C(=O)NCC1(NC(=O)COC(F)(F)F)CCC1)N(C)C 98913,C(CCCCC(=O)N1CC(C(N2CCOC(CC)C2)=O)(COC)C1)OCC 98914,C=CCCCCCC(=O)NCC=CCNC(C1CNC(=O)N1C)=O 98915,CC1CCCC(C)N1CC(=O)N(C1CN(C(c2cccc(=O)n2C)=O)C1)C 98916,C1(C(N2CC(NC(c3c(C)cc(F)cn3)=O)CC2(C)C)=O)CC2(CCC2)CCO1 98917,C1(C(=O)NC2(C)CN(C(c3cn(CC(N)=O)nn3)=O)C2)CCC2C1C2(F)F 98918,c1(CNC(=O)C(=O)N(c2ccc(CO)cc2)CCN2CCCC2)ccccc1Br 98919,C1(C(=O)NCCCN(C(=O)C(C)Oc2ccc(C)cc2)CC)CC(=O)N(OC)C1 98920,C=CC(C)(C)CC(=O)NCC1(C(=O)NC(C(C)(C)O)C2CC2)CCCC1 98921,C=CC(CCC)CC(=O)NC1CN(C(=O)Cn2nc(C)c(C)c2C)CC(F)(F)C1 98922,C(=O)(C(O)C1=CCCCC1)NCCC1CCN(C(c2n(C)nc(C)c2Cl)=O)C1 98923,C(CC1c2ccccc2CCN1C(c1ncc(C)cc1C)=O)NC(C(C)=CC)=O 98924,C1(C(=O)NC(CC(C)NC(C2N(CC)CCCC2)=O)C)CCC2CC(C)CN2C1 98925,N1(C(C=CC(C)(C)SC)=O)CC(CNC(c2ccnc(C)c2C)=O)N2CCC1C2 98926,c1(CC)cc(C(=O)NCCC2CCN(C(=O)CCC3(C)CC3)C2)c(C)o1 98927,N1(C(CSC(C)C)=O)CCCC2(CNC(=O)Cc3ccns3)CCCC12 98928,n1(CCC)nc(CO)nc1-c1ccn(-c2ccc(C(F)(F)F)cc2)n1 98929,c1(C(=O)NCC2N(C(CCCC)=O)CC(C)(C)C2)cc(Br)cc([N+](=O)[O-])c1C 98930,c1(OC)ccc(C(C)C(N2CCCC2CNC(=O)CC2(C(F)F)CC2)=O)cc1F 98931,c1(C(N2CC3CC(NC(C4(COC)CC4)=O)C3C2)=O)ccc2ncnn2c1 98932,c1(C(N(C(CCNC(CCCOC)=O)C)C)=O)sc(Cc2ccccc2)nc1C 98933,c1(C(N2CC(C(C(=O)NCCC(=O)NO)OC)C2)=O)ccccc1F 98934,C(=O)(C(CC(C)C)OC)NCC(CCCC)NC(C1CC(CF)C1)=O 98935,C(=O)(C(C)(C)CCCF)NCC1(C)CCC(NC(CN(CC)CC)=O)C1 98936,C(=O)(C1CC(=O)Nc2ncccc21)N(CCCNC(=O)C1CCc2nccn21)C 98937,C(CC(C(C)C)NC(c1cncc(O)c1)=O)NC(C1(c2c(C)cno2)CC1)=O 98938,C(=O)(CCC(C)(C)F)NCCCC(C)NC(=O)C1=NOC(C(C)(C)C)C1 98939,C1(NC(c2ccn(C3CC3(F)F)n2)=O)CN(C(=O)COC2CC2)CC12CCC2 98940,C1(C#N)(C(=O)NCC(=O)NCC2(CO)C(C=C)C2)CC(=O)C1 98941,c1(-c2cn(C(CNC(c3c(CC)con3)=O)C)nn2)c(F)c(F)c(N)c(F)c1F 98942,c1(C(=O)OCC23CC(C(=O)OC)(OC2)C3)ccnc(Br)c1N 98943,C1(CC(=O)OC)(NC(c2cc(COc3ccccc3)on2)=O)CCCS(=O)(=O)C1 98944,c1(C(N2CCC(NC(c3cnn[nH]3)=O)C2)=O)nnn(C2CC2)c1-c1ccccc1 98945,CC1CC(=O)NCC1C(=O)NC1(C2CCCN2C(c2cc(O)cs2)=O)CC1 98946,c1(N(C(C(C)C2CC2)C(=O)NC(C)(C)C(F)F)C)ccc2c(c1)CCC2 98947,N1(C(C2(C=C)CCC2)=O)CCC2CC2(C(=O)Nc2cncnc2O)CC1 98948,C1(C(=O)OCC)CNC(=O)CC12CCN(Cc1ccc(OC)c(OC)c1O)CC2 98949,c1(C(C(=O)NCCN(C(CC(C)OC)=O)C2CC2)(C)C)ccc(Cl)nc1 98950,C1(NC(C2CC23CC3)=O)C2CC(O)C1N(C(c1ccccc1-c1cc[nH]n1)=O)C2 98951,c1(C(=O)NC(C(C)C)CNC(=O)CC2CCC(C(F)(F)F)O2)cnc(N)c(O)c1 98952,C1(CNC(CN(C(C(C=C)OC)=O)CCOC)=O)CCCC12CCC2 98953,C(=O)(C(CCCC)NC(c1ncc(F)cn1)=O)NC(C=C)C 98954,N1(C(Cn2ncc(CC)c2)=O)CC2COCC2(C(=O)NC(c2ccncc2)C)C1 98955,C1(CN(C(CC(C)c2ccccc2)=O)C)CCCN(C(C2(F)CC2)=O)C1 98956,C12(C(N3C(CNC(C=C4CCN(C)CC4)=O)CCCC3)=O)CCC(C1)C2(C)C 98957,C1(CC(=O)NC2CC(NC(c3ccc(C(=O)OC)o3)=O)C2)C(=O)NN=C1C 98958,c1(C(N(CC(C)N(C(c2ccc(C)nc2)=O)C)C)=O)n[nH]c2c1CCOC2 98959,Cc1cnccc1C=CC(=O)NC1CCCC(NC(c2c(C)nn(C)c2Cl)=O)C1 98960,Cc1oc(Br)cc1C(=O)NC1CC2(C1)CC2NC(=O)CN1CCCNC1=O 98961,N1(C(c2ccc(CC)cn2)=O)CC(CNC(=O)CCCc2cccs2)CC1(C)C 98962,CC1C(N(C(=O)CCC2CCCN2)C(=O)CN(C2CCCC2)CCO)CCCN1C 98963,C(c1c(Cl)nc2sccn12)=CC(=O)NC1C2CCN(C(=O)C(O)CC(F)(F)F)C12 98964,C(C)(CN=c1[nH]c(Cl)ncc1C(F)(F)F)N(C(c1c(CC)nc(C)[nH]1)=O)C 98965,c1(C(=O)NCC2N(C(C(C)CF)=O)CCN(C)C2)cccc2c1COCC2 98966,C1(CNC(c2ccsc2F)=O)CCC(NC(c2[nH]nnc2C2CC2)=O)C1 98967,C(CNC(=O)CSc1nnnn1C)(CC(F)(F)F)NC(C(C)CSC(F)(F)F)=O 98968,c1(C(C)NC(c2n(CCSC)nnn2)c2cscc2C)ccncc1Cl 98969,CC1CCN(C(C2(CO)COC2)=O)CC1NC(=O)CC(F)(F)Br 98970,c1(OC)ccc(C)c(C(=O)N(C2CCN(C(=O)CCC(C)SC)C2)C)c1 98971,c1(CC)ccc(F)cc1C(=O)NCCCC1CCCCN1C(c1[nH]ccc1C)=O 98972,C1(CCC(=O)NC(C2CCCC2)CSC(C)C(=O)NCC)(N(C)C)CCCCC1 98973,c1(C(N2CCC(C(C)(C)NC(CC3N(CC)CCC3)=O)C2)=O)ccc(CO)cn1 98974,c1(C(C)C)ccc(C=CC(=O)NC2COCCN(C(=O)CCC3CC3)C2)cc1 98975,c1(CC(=O)N(C)CC2N(C(C(C)SC)=O)CCOC2)coc2ccc(F)cc12 98976,CN1CC(O)CC1C(=O)NC1CC(C(N2CC(n3cnnn3)C2)=O)C1 98977,C1(N(C(C=CC=CCC)=O)C)CCN(C(c2cc(Cl)ncc2OC)=O)CC1C 98978,CC1(C)CC(CC(=O)NC2(C3CCCN3C(C3CC=CCO3)=O)CC2)CCO1 98979,C1(NC(C2(SC)CN(C(C(CCC)CC)=O)C2)=O)CC(C)(C)OC1(C)C 98980,CC(C)(O)C(C(=O)NC1CCCC1O)NC(c1cnn(C2CC2)c1)=O 98981,C(C(C)CC(=O)NCC1(C(N)=O)CN(C(=O)C=CCn2cncn2)C1)OC 98982,N1(C(CC=CC=C)=O)CC(C2CC2)(C(=O)Nc2ccc(F)c(CO)c2)C1 98983,C=C(C)CC(C(=O)N1CC(NC(=O)OC)C1)NC(c1cn(CC)cn1)=O 98984,N1(C(C(C)OCC(C)C)=O)CC(NC(c2coc(Cl)n2)=O)CC12CCCCC2 98985,C1(OC)(CNC(C2CC3CC3C2)=O)CCN(C(=O)CCc2ccc(O)cc2)CC1 98986,C(=O)(CCCNC(=O)CC1CC(NC(C2CCCN2C(N)=O)=O)C1)NC 98987,c1(CN(C)C)ccc(C(=O)NC23CC(NC(=O)CCOc4cccnc4)(C2)C3)o1 98988,N1(C(C2CCC3CC23)=O)CCOC2(CCCN(C(c3ocnc3C(F)F)=O)C2)C1 98989,c1(C(=O)NC2C3CN(C(CCC(C)SC)=O)C2C3)ncc(Cl)cc1F 98990,C12(C(=O)NCC(N(C)C(C3C4CCC(=O)C34)=O)C3CC3)CCCCC1C2(F)F 98991,Cc1n[nH]c(C)c1CNC(=O)CC1CCN(c2ccnc(C(C)(C)C)n2)C1 98992,C(=O)(CC(O)CC(C)(C)C)N1C(C(=O)Nc2c(CC)c(F)ccc2)C=CC1 98993,c1(C(=O)NCCN(C(C)C)C(C2CCCCO2)=O)c(Cl)c([N+](=O)[O-])nn1C 98994,C12(C(=O)OCC)CCC(C(N3CCCCC(CNC(C)=O)CC3)=O)(CC1)CC2 98995,N1(C(c2nn(CC)c(C)c2)=O)CCC(N(C)C(c2cc(OC)nn2C)=O)C(C)C1 98996,N1(C(Cc2cccc(SC)c2)=O)CCN(C(C)C)CC1C.C12(CC1)C(=O)N2 98997,C1(NC(c2ccc(C)nc2)=O)CS(=O)(=O)CC1Nc1cnc(C#N)cn1 98998,N1(C(C=COCC)=O)CCC2(CCCC2NC(=O)CCc2cccc(C#N)c2)C1 98999,Cc1ccc2c(C(=O)NCC3(F)CC(CNC(c4cnco4)=O)C3)cnn2c1C 99000,c1(C(N(CCCNC(=O)CC(C)C)CC)=O)ccc2oc(N(C)C)nc2c1 99001,c1(C(=O)NCC(CNC(C2CCC(=O)N2)=O)CO)c[nH]c(=O)c2ccncc12 99002,c1(NC(N2CCC(N(C)CC)C2)=O)ccnc(S(C)(=O)=O)c1 99003,C1(NC(COCCCN(C)C)=O)CN(C(c2cc(F)cs2)=O)CC1F 99004,c1(OC(C)C(N2CCCC2CCNC(C2(c3ncco3)CC2)=O)=O)ccccc1 99005,c1(C(=O)NC)ccc(C(=O)N(CC(O)CNC(=O)C(F)n2ccnc2)C)cc1F 99006,c1(C(=O)NC2CN(C(c3nn(CC)c(C)c3)=O)CC2F)cc(Br)ccc1O 99007,c1(CC)cnc(C(=O)NCC2CC2NC(c2cccnc2C)=O)cn1 99008,c1(CNC(CC=C(C)C)=O)ccc(F)cc1Cl.n12cc(nn1)C(=O)NCCC2.OCN 99009,N1(NC(C2(CC)CCC(C)CC2)=O)CCC(N=c2ccc3nccn3[nH]2)C(F)(F)C1 99010,c1(C(=O)NC(c2cn(C(C)C)nn2)(C)C)cccc2scnc12 99011,N1(C(C2(CC#C)CCOC2)=O)CCCC(NC(c2c[nH]c(=N)s2)=O)CC1 99012,N1(C(Cc2c(C)ccnc2)=O)CC(F)(F)CC1CNC(C1CCCOC1)=O 99013,c1(C(=O)NCC2(F)CCN(C(C(=CC3CCCC3)C)=O)C2)cccn2cncc12 99014,c1(C(=O)N(C2(CCNC(=O)C(c3ccccc3)F)CC2)CCO)cnc2sccn12 99015,C1(F)(C(=O)Nc2nccnc2Br)CCN(C(c2occc2Br)=O)CC1 99016,N1(C(C(F)OC)=O)CC(O)(CCNC(c2ccncn2)=O)C1 99017,C1(C(=O)NCCCN(C)C(C2C(Cl)(Cl)C23CC3)=O)CCc2ccccc2C1 99018,N1(C(=O)Nc2c(CC)ccc(C(F)(F)F)c2)Cc2ccccc2SCC1C 99019,c1(NCCC(C)F)nc2ccccc2nc1NCCCN1CCCOCC1 99020,N1(C(c2c(C)n(C)cc2)=O)CCN(C(C2(C)CC(F)C2)=O)C2(CCC2)C1 99021,C(=O)(CC1CCc2ccc(O)cc21)NC(C)(C)CNC(C1OCCC1(C)C)=O 99022,N1(CC(=O)N(c2scc(-c3ccc(CCCC)cc3)n2)CC)CC2CC(F)(C2)C1 99023,c1(N2CCC(O)(CCNC(CC)=O)CC2)nc(C(=O)NC)nc(C)c1Br 99024,C1(CC)CN(C(c2csc(Cl)c2Cl)C(=O)NCc2ccc(F)cc2)CCN(C)C1 99025,C1(C(N2CC(CNC(c3n(C)c(=O)ccc3)=O)OCC2)=O)CCc2nn[nH]c2C1 99026,C(=O)(CCC(C)(F)F)NCCN(C(C1(OC)CCC1)=O)CCOCCO 99027,N1(C(c2cncc(N)c2)=O)CCCC(C2(NC(=O)Cc3ccsc3)CC2)C1 99028,C1(CN2CCC(NC(C3CCC3)=O)CC2)CCC12CCNCC2 99029,c1(C(=O)NCC2(OC)CN(C(C(CC)O)=O)C2)nc2n(c1C(C)C)CCCC2 99030,N1(C(C(C(C)NC(=O)CC2(N(C)C)CCC2)(C)C)=O)CCC12CC(C)(CO)C2 99031,C(CCCCC(=O)NCC1CCN1C(c1ncccc1O)=O)=CC 99032,Cc1ccc(F)c(C(=O)NC2CCC(N(C)C(c3cccnc3)=O)CC2)n1 99033,N1(C(C(C)n2cccn2)=O)CC(NC(c2n[nH]cc2Br)=O)CC2(CC2)C1 99034,c1(C(N2CC3C(CNC(CCCC#N)=O)C3C2)=O)cc2ccccn2n1 99035,S(=O)(=O)(c1cc(C)ccc1C)N1CCC(NC(C(C)(C)OC)=O)C(F)C1 99036,N1(C(c2cnc3cn(C)nc3c2)=O)CCS(=O)(=O)Cc2ccccc21 99037,C=CCS(=O)(=O)C(N1CC(CNC(=O)OC(C)(C)C)C1)=O.C12CCN(C1)C(=O)C2 99038,C(=O)(C(C(C)(C)C)C1CCC1)NC(Cc1c(C)ccs1)=O 99039,c1(C(=O)NC(c2ccc(OC(F)(F)Cl)cc2)C)c(Br)cnn1C 99040,N1(C(C2N(C)CCC2)=O)Cc2ccccc2C1CNC(C1CCCO1)=O 99041,c1(C(=O)NC2(CN(C)C(C3CC34CC(N(C)C)C4)=O)CC2)cc(C#N)cn1C 99042,CC1C(NC(=O)C(C)(O)C2CC2)CC2CCC1N2C(c1cc(Br)c[nH]1)=O 99043,Cc1ccc(OCC(N2CCC(CCNC(=O)CSCC(C)C)C2)=O)cc1 99044,CCC(C)(CO)C(=O)N1CCCC(n2cc(-c3ccnc(OC)c3F)nn2)C1 99045,Cc1[nH]nc(C(N2CCCC2CN(C)C(C2C3CCN2CC3)=O)=O)c1[N+](=O)[O-] 99046,CN1CCCC1CC(=O)NC1CC(NC(C2(C(=O)NC(C)(C)C)CCCC2)=O)C1 99047,C(=O)(CCCC(C)(C)CC)N1CCC(C(F)F)(CNC(C2CCN(CC)C2)=O)C1 99048,N1(C(C(CCCCC)C)=O)CC2(C=C(C(=O)Nc3cccc(C)n3)CO2)C1 99049,C(=O)(C(O)CCC(C)C)NCCN(C(=O)CN1CC2CCC1C2)CCC 99050,CCC(CC(=O)NC1(CCNC(=O)CCSC)CCC1)c1ccccc1 99051,c1(OC)ccc(OC)c(C(N2CCCCC2C2(NC(=O)C=CBr)CC2)=O)n1 99052,CC1CCCN(C(c2ncccc2C2CC2)=O)C1CCNC(c1cnc(Cl)s1)=O 99053,C=CC(C(=O)NCC(CC)NC(=O)C(C)(F)c1ccon1)OC 99054,C(=O)(CC(C)C(=O)NCC1(CNC(=O)Cc2ccsn2)CCOCC1)OC 99055,c1(CNC(C)=O)ccc2c(c1)CN(C(c1cc3c(cc1O)OCO3)=O)C2 99056,c1(C(=O)NC(CC(N)=O)C(N2CCC3C(C2)C3(F)F)=O)ccn2cncc2c1 99057,C1(C(=O)NC2(C(C)NC(=O)CCc3cncnc3)CC2)CC12CCOCC2 99058,Cc1ccccc1-n1ccc(C(=O)NC(C)CCNC(=O)CSC2CC2)n1 99059,c1(C(=O)NCC(CNC(C2C(C(N)=O)C2)=O)F)ccsc1Cl 99060,C1(N(C)C)CCc2nc(NC(c3cc(Cl)cc(C#C)c3NC(C)=O)=O)ncc2C1 99061,N1(C(c2cc(OC)cc(F)c2)C(=O)Nc2nnn(C)n2)CCn2c(cnc2CO)C1 99062,c1(C(=O)NC(CNC(C(n2ccc(C)n2)(C)C)=O)(C)C)cnc2n1CCCC2C 99063,N1(C(c2cncc(C=C)c2)=O)CC2CCC1CN2C(c1cccc(C)n1)=O 99064,N1(C(C2C(NC(C(CCCC)O)=O)C2(C)C)=O)CC2CCCC(C2)C1 99065,c1(CC(N2CC(NC(CCN(CCC)C)=O)C2)=O)cc(C(F)(F)F)cc(F)c1 99066,C1(CC)CN(C(=O)C=C(C)c2cccs2)CCC1NC(=O)Cc1ccnn1C 99067,N1(C(c2n(C)ncn2)=O)CCCC2(NC(c3cccc4cnnn34)=O)CCCC12 99068,c1(CCCC(=O)NC(C(C)NC(C(CCOC)C)=O)CO)c(F)cccc1F 99069,CCCC(C)(O)CC(=O)NCCOCCOCCCNCC1CCN(OC)CC1 99070,N1(C(C2CCN(C(Cc3cn(C)nc3)=O)C23CCC3)=O)CCC2(CCOC2=O)C1 99071,c1(C(=O)NC(c2nc[nH]n2)C)conc1CNC(=O)CCc1cncn1C 99072,[N-]=[N+]=NC1CC(C(=O)NCC2CC=CCC2)N(C(c2cnn3ccccc23)=O)C1 99073,C(c1ccc(C)cc1C)=CC(=O)NCC1CC(NC(C2CN(CC)C(=O)C2)=O)C1 99074,c1(NC(=O)NC(c2cccs2)C)c(Br)nnn1C 99075,C(CC(C(=O)N(C)Cc1ccc(C)nc1)OC)NC(C1CC(CC)C1)=O 99076,c1(OCC)cncc(C(=O)NCC(F)CNC(c2c[nH]cc2Br)=O)c1 99077,Cc1cc(C(N)=O)cc(C(=O)NCC2CC2NC(c2ccc(O)c(Cl)c2)=O)c1 99078,N1(C(c2n(C)nnc2)=O)CCCC(C(=O)NC2(C(C)(F)F)CC2)C1 99079,N#Cc1ccc(CN2CCC(NC(c3sc(Cl)cc3Cl)=O)C2)nc1 99080,C1(NC(C(CC)F)=O)CC2CCC1N2C(=O)COCC1CCCC1 99081,c1(C(=O)NC2(CO)CCCN(C(C=CC(C)(C)SC)=O)C2)cccc2[nH]ncc12 99082,C1(NC(CCCOCCC)=O)CN(C(=O)COC2CC=CC2)C2(CCOCC2)C1 99083,c1(C(N2CCC(O)(CN(C(=O)C(C)(C)NS(C)(=O)=O)C)C2)=O)noc2c1CCCC2 99084,n1(CC)nc(C(=O)NCc2cn(CC(=O)N(C3CCC(C)(C)C3)C)nn2)cc1C 99085,CC1(N2CCC2)CCN(C(C(=O)Nc2cccc(C3CC3)n2)C2CCOC2)C1 99086,CCCC(C)C1C(=O)NC2(C)CCCN1C2.C(=O)(C(C)(C)C)NCC(F)F 99087,C(=O)(CCC(C)CCN(C(=O)CCc1ccc[nH]1)CC)OCC 99088,CCCC(CNC(C1CC1CC(C)C)=O)C(=O)NCCC(C)(C)CO 99089,C12CCCCCN1C(=O)N2.c1(CC)c(-c2cn(C(C)C(=O)OC)nn2)cnn1C 99090,N1(C(C(COC)O)=O)CC2(CCCC(CNC(=O)CCNC(=O)C(C)(C)C)O2)C1 99091,C1(OC)CCC(C(=O)NCCCCNC(C2CC(n3cccn3)C2)=O)C1 99092,c1(CC(N2CC(NC(C(C)N3CCC3)=O)(CO)C2)=O)ccnc(Br)c1 99093,C1(C(=O)NC2CCC(O)C2)CCCC2CN(C(C3(F)CCCC=C3F)=O)CC12 99094,N1(C(C(C2(O)CN(C=O)C2)F)=O)CC(F)C(F)C1.c12cn(nn1)C2.C1CC1 99095,N1(C(CC2C(=O)NCCC2)=O)CCC(CNC2CCC3(CCC3)C2)C(O)C1 99096,C1(S(C)(=O)=O)(C(N(C2CCCC(NC(c3ncccc3F)=O)C2)C)=O)CCC1 99097,C1(C(=O)NC2CC(CC(=O)OC)C2)CC1C1CN(C(C2CC3(CCCO3)C2)=O)C1 99098,Cc1ccc(CN2CCC(C(=O)NOC3CC4CCC3C4)CC2)c(Br)c1 99099,C(=O)(CC(C)(C)N(C)C(c1ccn(CO)c1C)=O)NCC(C(=O)OC)OC 99100,c1(OCC)cnncc1C(N1CCC(C2CCCCN2C(c2ccsn2)=O)C1)=O 99101,N1(C(=O)Cc2cnn(C(F)F)c2)CCC(CNC(C2(Br)CCCC2)=O)CC1 99102,c1(OC)cc(O)ncc1C(N1CCCCC(NC(=O)C(C)=CCO)C1)=O 99103,N1(C(C=CCC)=O)CC(OC)CC1CNC(=O)C(Cc1ccsc1)NC=O 99104,c1(C(N2CC(C(=O)OC)CC(OC)(OC)C2)=O)cnc2ccccc2c1OC 99105,N1(C(CCC)=O)CCCC(C(=O)OCC2COCCC2C(N2CCCC2)=O)C1 99106,Cc1nnc2n1CC(C(=O)NC1CC(NC(=O)CN=S(C)(C)=O)C1)CC2 99107,Cc1csc2c(CNC(=O)NCc3ccc(C#N)cn3)cccc12 99108,CN1CCOC(C(=O)NCC(C(=O)NCCC2CCN(C)C2)N(C)C)C1 99109,C(C(=O)N1CC(C(C)NC(=O)CC2(C)CC2)C1)(C(C)C)OCC 99110,CCCCC(O)CC(=O)N1CC(CC(F)C(=O)NCCC(O)CC)C1 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99214,C1(CC=C)(NC(=O)CC2C=CS(=O)(=O)C2)CCN(C(=O)CCN2CCC(O)CC2)C1 99215,C12(C(N3CCC(C)(C(N)=O)C3)=O)CCC(CC1NC(=O)CC1CC(=O)C1)C2 99216,C1(C)(C(=O)NCC(C)NC(Cc2ccc(C)cc2F)=O)CCc2ccccc2C1 99217,C(=O)(CCCC(C)(C)NC(c1cc2cc[nH]c2cn1)=O)NC(CC(C)C)CO 99218,C1(C(N2CCN(C(CC(=C=C)C)=O)CC2C)=O)CC(C(C)(C)C)=NO1 99219,c1(C(=O)NCC(C)(C2CCC2)NC(C2COC2)=O)coc2cc(F)ccc12 99220,c1(CC(C(=O)NCCOCCNC(C2CC3C=CC2C3)=O)O)cc(Cl)cc(Cl)c1 99221,c1(CCC(=O)NCC(C2CC2)NC(C(c2cccnc2)N(C)C)=O)ncccn1 99222,n1(CC(=O)NCCCCCN(C(CCCC=C)=O)C)c(C)cc(C)nc1=O 99223,C(=O)(C1=NN(c2ccc(C)cc2)C(=O)CC1)N(C1CCC(NC(CC)=O)C1)C 99224,c1(NC)cccc(OC)c1C(=O)Nc1ccc(CNc2cnc(Br)c(C)c2)s1 99225,Cc1ncc(C(=O)NCCCCC(=O)NC2CC3C=CC2C3)c(=N)[nH]1 99226,c1(CC(=O)NC2CCCN(C(C3C(CC)C3)=O)C2)ccc(C)c(O)c1 99227,N1(C(C2CN(C)C(=O)C2)=O)CCC(CNC(c2ccc(CCF)cc2)=O)C12CC2 99228,CCC(C(=O)NCC1CC(F)(F)CN1C(C1CCCC(=O)N1)=O)C(C)C 99229,N1(C(C2(CF)CCN(C(c3c(CCC)nco3)=O)C2)=O)CCCC(O)(CO)C1 99230,N(C(=NCC(C)(O)c1cccc(Cl)c1)NC1CCCC1)Cc1ccn(CC)n1 99231,Cc1noc2nc(C(=O)NCCOC3CCN(C(C4CCSC4)=O)C3)ccc12 99232,Cc1ccc2c(=NCC3CC=CC3)[nH]c(=NCC(CO)C3CCOC3)[nH]c2c1 99233,c1(NC(CC(C)NC(CSC)=O)C)cc(OC(F)F)ccc1[N+](=O)[O-] 99234,C=CC1(C(N2CC(NC(=O)CP(C)(C)=O)C(O)C2)=O)CCCCC1 99235,N1(C(CNC(C=CC)=O)=O)CCN(C(C2(OC)CC(C)(C)C2)=O)CC1 99236,C=CCC1C(=O)N1.C1(CC(=O)OC)CC(NC(=O)C(C2CC2)OCC)C1 99237,C1(NC(C(C)Oc2ccc(F)nc2)=O)CCN(C(C2CC(F)(CF)C2)=O)CC1O 99238,C1(C)(C(=O)NCC(C)=CC(=O)NCCn2cncn2)CCC(=O)N1 99239,c1(C(=O)NCCN(C(C)C)C(C2CC3CC3C2)=O)cc(C2CCCCC2)[nH]n1 99240,CCC(CC(=O)N1CCN(C(c2cccc(C)n2)=O)CC1C1CCCC1)C(F)F 99241,Cc1nnc(CNC(c2nnnn2C2CCC2)Cc2ccccc2)n1C1CC1 99242,N1(C(C2(OC)CCSC2)=O)C(CNC(c2ccc(F)cc2Cl)=O)CC2COCC12 99243,C(CNC(C1CNC(=O)N1C)=O)(CC(C)C)NC(C(C)SCC)=O 99244,C(=O)(C1=NOC(CNC(c2c[nH]c(=N)o2)=O)C1)NCC=CC 99245,C1(F)(C(=O)NC2CCC3(C(C)C)C2C3)CCCN(C(=O)CC(C)n2cccn2)C1 99246,CN1CC2CCCC(C1)N2C(=O)C(CC(N)=O)NC(C1CCCN1C1CC1)=O 99247,c1(C(N2CCC(O)C2)C(=O)NCc2ccco2)cn(C2CCOCC2)nn1 99248,C1(NC(c2cc(C#N)no2)=O)CC2CCCC(C1)N2C(C1OC2CCC1CC2)=O 99249,O=C(C(O)C(F)F)NCC1CC(NC(=O)Cc2ccccc2CO)C1 99250,N1(C(C(c2cccnc2)C)=O)CCC2(CC1)CCN(C(c1ccc[nH]1)=O)CC2 99251,C1(CNC(CC(C)(C)F)=O)CC2(CCOCC2)CN1C(=O)C(N)=O 99252,CCC(C)(CO)C(=O)NCC1CC(F)(CNC(c2cnc(S)n2C)=O)C1 99253,C1(CCNC(C2(CN(C)C)CC2)=O)CCN(C(=O)CC2CC3(CC3)C2)CC1 99254,C(=O)(C1=C(F)CN(C(c2cc(F)c[nH]2)=O)CC1)NC1CCCC(C)(C)C1 99255,C(=O)(C(C(F)(F)F)NC(c1cc(-c2cccc(F)c2)no1)=O)OCC 99256,N1(C(C(=O)NCc2cncc(OC)c2)=O)CCC(C)C(NC(N(CC)CC)=O)C1 99257,C1(COC)CN(C(C2(CCn3cncn3)CC2)=O)CCC1NC(=O)CC1CC1C 99258,N1(C(CSCC=C)=O)CCc2nc(-c3ccc(F)c([N+](=O)[O-])c3)sc2C1 99259,CC1(C)CC(NC(=O)Cc2nc[nH]n2)CN(C(=O)C(F)(F)C(C)(C)O)C1 99260,C1(CC)CCN(C(=O)CC2CC2C(=O)N)C1CCc1occc1CC.N(C)(C)N 99261,c1(C(N2C(C)CCC(NC(=O)C(N)=O)C2)=O)ccc(C2=CCCC2)cc1 99262,c1(CC)ccc(F)cc1NC1CCN(C(c2ccc(OCC)nc2)=O)C1 99263,c1(OC)ccc(Cl)c(C(=O)NC2CC3CCC2N3C(=O)C(F)(F)C(O)C2CC2)c1 99264,N1(C(C(CCC)F)=O)CCC(C)N(C(=O)C(n2cc(C)cn2)C)CC1 99265,c1(C(N2CCCC(C(N3CCC(O)C3)=O)C2)=O)ccc(-c2cccnc2)nc1O 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99283,C(=O)(C(N)CC(F)F)NCC(=O)Nc1[nH]nc(-c2nccc(C)c2)n1 99284,C(=O)(CC(C)NC(C1CC(CCNC(=O)CC(=O)OC)C1)=O)OCC 99285,O=C(C1=CCN(C(c2cnns2)=O)C1)NCCOCC(F)F 99286,C(=O)(CC(F)(F)C(C)C)N(CCC)CCNC(=O)C(C)CS(C)=O 99287,C12(C(=O)NC3CC(C)CN(C(c4ccnc(O)c4)=O)C3)CCOC1CC(=O)NC2 99288,CC1(NC(C2CC23CCSCC3)=O)CCN(C(C23CC(CCO2)C3)=O)CC1 99289,N1(C(c2cc(CC)no2)=O)CCC2CC12C(N1CCC(CC(=O)OC)C1)=O 99290,c1(C(N2CC(NC(=O)CC3CC4(CCC4)C3)CC(C)C2)=O)cccc([N+](=O)[O-])c1 99291,N1(C(C2CC(C)OCC2)=O)CC2CC(NC(C3(N(C)C)CCC3)=O)CC1C2 99292,Cc1oc(-c2cccs2)nc1C(=O)NCCOC1CCN(C(=O)CC(C)CF)C1 99293,c1(C(=O)NCCNC(=O)OC)ccoc1CNC(C1C(C)C1C)=O 99294,C=C(C)CC(C)C(=O)NC1(COC)CCN(C(c2nnn(C)c2C)=O)CC1 99295,Cn1cnc2c1CC(NCCCc1nc(O)c3ccccc3n1)CC2 99296,C1(C(N(CC(CC)NC(CC(=C)Br)=O)C)=O)CN(C(C)C)CCO1 99297,C1(C(=O)NCC(CN(C(C(C)CSc2ccccc2)=O)C)(C)C)CCC(C)(C)O1 99298,c1(NCc2[nH]nc(OC)n2)[nH]c(=NC(C)c2nnc(C)o2)nc2c1cnn2C 99299,Cc1ccnn1CCC(=O)NCCOC1CCN(C(=O)CO)C1 99300,N1(C(c2c(C)nc(O)[nH]2)=O)CC(C)CCC1CNC(c1cnco1)=O 99301,CCC(C)(C)CCCC(=O)NCC(C)(C)CN(C(=O)C(C)(F)C(F)(F)F)C 99302,C(c1ccc(F)cc1)=C(C)C(=O)NC1CCN(C(=O)C(C)(C)C2CCOCC2)C1 99303,C(=O)(C(C)(O)C(C)C)NC1CC(CNC(CN(C2CC2)CC)=O)OCC1 99304,C1(CNC(C(C)O)=O)CC2COCC2N1C(=O)C(F)(F)c1cnn(C)c1 99305,C1(NC(CSC(C)C)=O)CCC(C)N(C(c2cc(C3CC3)[nH]n2)=O)C1 99306,CCCCCCn1cc(C2CCN(C(=O)Cc3nocc3C)C2)nn1 99307,C1(CC(=O)NCC(CNC(CCC(=C)Br)=O)OC)CCCCC12CC2 99308,C1(C(=O)NC(C2(C(=O)NC(C3CCOC3)C#C)CC2)C)CCCCCC1 99309,c1(SC)nc(Cl)c(C)c(=NC2CCN(C(=O)CN3CCCNC3=O)C2)[nH]1 99310,Cc1cc(Br)cc2cc(CC(C(=O)O)NC(c3ccc(CN(C)C)o3)=O)oc12 99311,CC(CCc1ccccc1)CC(=O)NCC(C)CN(C)C(c1cnoc1)=O 99312,c1(OC)cc(C)c(C(=O)NC2CC(NC(=O)CC(C3CC3)C3CC3)C2)cn1 99313,c1(SC(C(N2CCCN(CC)C2)=O)C2CCCC2)cc(O)ncc1Br 99314,c1(C(=O)NC2CC(C)N(C(=O)CN(C)S(N)(=O)=O)C2)ccc(O)c(Cl)n1 99315,N1(C(C(=O)NCCSC)c2cnsc2)CCC2NC(=O)CCC2C1 99316,N1(C(C2C(CC)NC2)=O)CC(N(C)C)CC1c1ncc(C(F)(F)F)[nH]1 99317,C1(C(=O)NCC(CCOC)NC(c2c[nH]c(C(F)(F)F)c2)=O)C(C)(C)C1(F)F 99318,c1(NC(=O)NCC2CC(F)(CNC(=O)CN3CCCCC3)C2)c(F)cccc1F 99319,c1(C(C(=O)NCCOC)N(CC(=O)NC(C)C)C2CC2)cc(C(C)(F)F)ccn1 99320,C1(C(=O)Nc2ccc(C(=O)NCC(=O)N(C)C)nc2)CC(N=c2cncc[nH]2)C1 99321,C1(NCc2c(Cl)ccnc2I)CC2(CCN(c3ncc4c(n3)CCC4)CC2)C1 99322,N1(C(CCC2C(=O)NC(=O)N2)=O)CC2(CC(NC(c3cc(F)c[nH]3)=O)CO2)C1 99323,Cc1ccc(C)n1CC(=O)N(CCNC(=O)CC1(C)OCCO1)Cc1ccccc1 99324,C(=O)(CCNC(C=CCOCC1CC(CNC(=O)O)C1)=O)CC.C1(F)(OC)CC1.N 99325,C(=O)(CC(O)CNC(C1CCC1C(=O)OC)=O)N1C(C(C)O)C=CC1 99326,N1(C(CCCN(C(=O)C(F)C2CCCC2)C)=O)CCC(NC(=O)COC(F)F)CC1 99327,c1(C(N2CCC(CNC(COC3C(C)CCCC3)=O)CC2)=O)ccn(C)c(=O)c1 99328,C(=O)(C(CC(C)SC)NC)N1C(C(=O)Nc2c(C(=O)NCC)cccc2)CCC1 99329,C1(CNC(C2C(=C)C2)=O)(CNC(c2nc(Cl)cs2)=O)CC12CCC2 99330,CN=c1cc(C(N2CCOC(C(=O)NC3CCC(C4CC4)C3)C2)=O)cc[nH]1 99331,C1(C(=O)NOC(c2ccccn2)C)(CC#C)CCN(C(=O)CC2CC=CCC2)C1 99332,C(=O)(C1=NOC(C)(C)C1)N(C(C)C(=O)NCC1CCC(CCO)C1)C 99333,c1(C(N2CC(C(C)(C)O)(CNC(CCC(C)(F)F)=O)C2)=O)cc(F)cc2cc[nH]c12 99334,C(=O)(C(O)CC(F)(F)F)N1C(C)(CC)CC(NC(c2cccn2C)=O)C1 99335,C1(C(=O)NCCC(C(=O)N(CCOC)CCO)O)CCCC(C#N)C1 99336,Cc1c(C(=O)NC2CC23CCN(C(C2CSCCS2)=O)C3)cncc1Cl 99337,Cc1sc(=O)n(CCC(=O)NCC(O)CCNC(C2(C3CC3)CC2)=O)c1C 99338,c1(OC)c(C(=O)NCC2CC(NC(=O)Cc3nonc3C)C2)nc(O)nc1O 99339,CON(CCC(=O)NC(C)(C)CCN(C)C)C(=O)C12CCC(C1)OC2C 99340,CC(C)(C#N)CC(=O)N1CC(NC(c2cccc(Cl)c2)=O)CCC1C(F)(F)F 99341,C1(NC(C2(SCC)CC2)=O)CC2(C1)CC2NC(=O)Cc1csc(C2CCCC2)n1 99342,C1(CCNC(COCCCOC)=O)CN(C(=O)CCOC2CCCOC2)CC1C 99343,C(CC1CC1)(CC(=O)NC(CO)CCF)NC(c1cn(CC=C)nc1)=O 99344,N1(C(C(CN(CC)CC)F)=O)CCC(C)(CCNC(=O)Cc2cn[nH]c2)C1 99345,C1(NC(CC(c2c(C)cccc2)C)=O)COCCN(C(=O)CN2CSCC2=O)C1 99346,C(C)(CC(C)NC(C1(C(C)(F)F)CCC1)=O)NC(CCOCC#C)=O 99347,C1(CC(=O)NCc2cc(Cl)n[nH]2)CCCN(C(C23CCCC2CCC3)=O)CC1 99348,C(=O)(C1CCc2c[nH]nc21)N(CC(N1CC(C2(C)CC2)C1)=O)CC1CC1 99349,N1(C(CSCC(=O)OC)=O)CCCC(NC(=O)CN2CC(OCC(F)F)C2=O)C1 99350,c1(C(N(C)CC2(O)CCN(C(C3(C(N)=O)CCC3)=O)C2)=O)cnn2c1OCC(F)C2 99351,c1(NC(=O)NCC(C2CCCOC2)OC)ccc2c(c1)CCCN2 99352,C1(O)(CCNC(c2c(C)ncs2)=O)CCCN(C(C2CCN2C2CCCC2)=O)C1 99353,N1(C(=O)NC(c2ccc(C)cc2)CC)CCN(c2ccc(Cl)cn2)CC1 99354,CCC(C)CCC(=O)N1CC(O)(CNC(C2CCC(F)CC2)=O)C1 99355,N1(CC)CCCC(C(N2CC(N(C(=O)Cc3nc(C(C)(C)C)n[nH]3)C)C2)=O)C1 99356,C1(NC(CCCC)=O)CN(C(=O)C(=O)Nc2ccc(C)c(C)c2)CC2(CC2)C1 99357,Cc1cc(C(N2CCCC2CCCNC(=O)C(=Cc2cscn2)F)=O)ccn1 99358,Cc1cnc(CNC(c2sccc2CNC(=O)CC2CCCN2C(C)C)=O)nc1 99359,C(CCC(N)=O)(C(=O)NCCCN(C)C1CC1)n1cc(CSC)nn1 99360,c1(N(CCCOCC)C)ncc(S(=O)(=O)N2CCC(c3ccco3)C2)cc1Cl 99361,N1(C(C(C(C)C)=O)=O)CC2CN(C(=O)Cc3ccc(F)cc3Cl)CC2C1 99362,c1(OC)ccc(C(O)CC(=O)NC(C2CCC(=O)N2)c2nn[nH]n2)cc1OC 99363,CC1(C)CC(C)(C(=O)NC(CCOCCO)C(=O)NCCc2ccccc2O)C1 99364,n1(CC(N2CC3C(N(C(CN(CC)CC)=O)C)C3C2)=O)nc(C)ccc1=O 99365,c1(C(=O)NC2CN(C(CC(=C=C)C)=O)C3C2C3)ccc(O)cc1C 99366,C1(NC(=O)CC2CC3CC3C2)CN(C(=O)CC2CCCC2)CC2(CCC2)C1 99367,CC1(CNC(=O)C(F)(F)c2ccncc2)CCCN1C(c1ccc[n+]([O-])c1)=O 99368,N1(C(C(=O)NC(C(C)C)C)=O)CCCC(C(=O)CCN2CCCC2)C1 99369,C1(NC(c2nc(CCC)oc2)=O)CN(C(=O)C(C)N2CC(C)C2)CCC1CO 99370,c1(C(=O)NC(C(C(C)C)NC(c2c(C)nncc2)=O)C)cc2ccc(F)cc2o1 99371,C(=O)(C(C)(CC)CO)N(CCC)CCNC(c1onc(Br)c1C)=O 99372,N1(C(CN(C(=O)CC2CCCOCC2)CC)=O)CCC(C)(C#N)C1 99373,c1(C(N(CCC(=O)NC(COC)COC)C)=O)sc(C)cc1C 99374,C1(CNC(C2N(C)CCC2)=O)CN(C(=O)CCC2CC2(F)F)CC(C)(C)O1 99375,Cc1cn(-c2ccc(F)cc2)nc1C(=O)N(CCS(C)=O)C(C)(C)C 99376,CC1CN(C(=O)C=CC2CCOC2)CCCN1C(C12CCCCC(F)(C1)C2)=O 99377,N1(c2n(CCC=C)c(C(c3cccc(OC)c3)C)nn2)CC2CC(O)CC2C1 99378,C1(C2CCCN(C(=O)C(O)CCSC)C2)(NC(c2ccc(OC)cc2Cl)=O)CC1 99379,c1(C(N2C(CCCNC(CC=C)=O)CCC2)=O)ccc(-c2cn[nH]c2)cc1 99380,Cc1scc(CNC(=O)C=CC(C)(C)NC(C2OC3CCC2C3)=O)c1C 99381,CC(N=c1nc2sccc2c(NCc2csc(Br)n2)[nH]1)c1cnccn1 99382,CC(CC(=O)N1CCCC(O)(CN=c2[nH]nc(CO)s2)C1)C(F)(F)F 99383,c1(SC)cc(=NC(=O)C2N(C(=O)Cn3ccnc3)CCCC2(C)C)[nH]n1C 99384,Cc1c(C(N2CCC(C(=O)NCC(C)(O)CO)(CO)C2)=O)ncn1C 99385,C1(C(C)(C)C)CCN(C(=O)CCN(C(=O)CC2CCOC2)CCO)C1 99386,c1(CNC(C=CC(C)(C)NC(=O)C(C2CCOCC2)O)=O)c[nH]ccc1=O 99387,C1(NC(C(C)CC2CCC2)=O)COCCN(C(=O)Cc2cnccn2)C1 99388,c1(C(=O)NC(C(C)C)CCN(C(=O)C(=O)N(C)C)C)cc2n(c1)CCOC2 99389,Cc1c(-n2cc(C3(C)CCCN3C(C3CCOC3C)=O)nn2)cccc1Br 99390,C(=O)(CCCC(=O)N1CCN(C(=O)CCOC2CCOCC2)C(C(F)F)C1)OC 99391,Cc1cnc(NC2C=CCC2)c(S(=O)(=O)NCCCCOC(C)(C)C)c1 99392,C1(NC(c2ccc(C(N)=O)o2)=O)CN(CCN2CCCS2(=O)=O)CC2(CC2)C1 99393,Cn1c(C(=O)NCC2(C(N3CC(N4CCOC4=O)C3)=O)CCCO2)cnc1Cl 99394,N1(C(C2C(C=C)CC2)=O)CCOCC1CCNC(c1nc(Br)sc1C)=O 99395,C1(NC(C2N(CC)CC2)=O)C=CC(C(=O)N(CCC(O)CO)C)C1 99396,C(CN=c1cc[nH]cc1S(=O)(=O)N1CCC(C(C)C)C1)c1c(C)cccc1 99397,Cc1ccc(F)c(C(N2CC=CC(NC(=O)CC(C)C3CC3)C2)=O)n1 99398,c1(-n2cc(CCCNC(c3csc(-c4ccccc4)n3)=O)nn2)cccc(F)n1 99399,Cc1[nH]nc2ccc(C(=O)NC3CC3NC(=O)CCCS(C)(=O)=O)cc12 99400,N#CC1CCN(CC(=O)NC2CC(n3cc(C4CCCC(O)C4)nn3)C2)CC1 99401,c1(CC)cscc1C(=O)NCC1CC1NCC.c1(C=O)ccncc1 99402,N1(C(CCCCC)=O)CC2(C1)CN(C(c1ccc(C3CCCO3)nn1)=O)C2 99403,Cc1ccc2[nH]nc(C(=O)NCCC(C)(C)NC(=O)CN3CCCCCC3)c2c1 99404,C(=O)(C(F)C1=CCCCC1)NC(CNC(Cc1c(C)nc(O)nc1O)=O)C(C)C 99405,Cc1cccn2cc(C(N3CCC3CNC(=O)C(C)Sc3ccccn3)=O)nc12 99406,c1(OCC(N2CC(N(C(c3cc(OCC)n[nH]3)=O)C)C2)=O)cc(C)cc(C)c1 99407,C(=O)(C(C)(C)CS(N)(=O)=O)NCC(CC)NC(=O)Cc1cc2ccccc2s1 99408,n1(C(C)C)ncc(C(=O)NCC(C(C)(C)C)NC(C2(Cl)CC2(F)F)=O)c1C1CC1 99409,c1(C(N2CCC(F)(CNC(c3c(CC)c(C)sc3)=O)C2)=O)ccc2c(c1)CCO2 99410,N1(C(CC2(CSC)CC2)=O)CCC(NC(=O)COC2CCCCCC2)CC1C 99411,N1(C(C2(CC)CCCC2O)=O)CC=C(C(=O)Nc2ccn(C3CC3)n2)CC1 99412,C1(C(=O)NCCN)CCC(CC(=O)C(=O)NC)C1.c1(CCC(=O)N)cncn1C 99413,C(=O)(C(C(C)CCC=C(C)C)N1CCC(C(N)=O)CC1)NCCC(=O)OCC 99414,c1(NC)cc(C(N2CC(C)(NC(=O)C(CC3CC3)NC(C)=O)C2)=O)cc(Cl)n1 99415,C#Cc1cccc(C(=O)NCc2ccc(C(N3CC=CC3C(=O)OC)=O)nc2)c1 99416,c1(C(N2C(C(CNC(CC(COC)C)=O)(C)C)CCC2)=O)cc2occc2[nH]1 99417,CCS(=O)(=O)CC(=O)NCC1CCCCN1C(C1CCCN(C(N)=O)C1)=O 99418,C1(NC(c2c(CC)[nH]nc2Cl)=O)COCCN(C(=O)COC2COC2)C1 99419,c1(C(=O)NC(C2CCN(C(=O)C(C)Cc3ccco3)C2)C)ccnc(Br)c1F 99420,c1(C(=O)NCCCCCNC(Cn2nc(C)n(C)c2=O)=O)ccc2cc[nH]c2c1 99421,Cc1c(C(=O)N(C)CCN2CCN(C(c3ccc(O)cn3)=O)CC2)cnn1C 99422,c1(C(N(CC(CNC(C2CC(CC(=O)OC)C2)=O)O)C)=O)c[nH]nc1C(F)(F)F 99423,C1(NC(CCOC(C)C)=O)CCCC(NC(=O)CCN2CCCCC2)C1 99424,c1(CC)ccc([N+](=O)[O-])cc1C(=O)N(CC(C)(C)NC(c1ccncc1F)=O)C 99425,C1(C(=O)NC(CNC(CCc2onc(C(C)C)n2)=O)(C)CO)CCN(C)C1C 99426,C1(NC(C=C(CC)CC)=O)CCCCCC1C(=O)NC1CCCC1(F)F 99427,c1(CCC)cc(C(=O)NCCC(C)N(C(=O)C(C)Cc2ccncc2)C)n[nH]1 99428,C#CC1(C(N2CCCC(CNC(C3COCCO3)=O)C2)=O)CCCC1 99429,CCC1=C(C(=O)N(C)CC2CCCN2C(=O)CC2COCC(C)(C)O2)SCCO1 99430,C1(CC(=O)N(C)CC2N(C(CCCc3ccc(C)s3)=O)CCC2)COC2CC1C2 99431,Cc1cc(C(N2CC(NC(c3nc(O)c(C)s3)=O)C3CC23)=O)n2nc(C)cc2n1 99432,N#CCC(=O)NNC(=O)CN(c1ccc(Cl)cc1)CC1CCCOC1 99433,c1(C(=O)NCC2CC(NC(CC3N(CC)CCC3)=O)C2)ccc(CC2CC2)cc1 99434,C1(NC(C(C(=C)Cl)(C)C)=O)CCC2CCN(C(=O)CCNC(=O)OCC)C1C2 99435,C1(C)(CNC(C2C(c3c(C)ccnc3)C2)=O)CCC(NC(c2cc[nH]n2)=O)CC1 99436,c1(C(=O)NC(CC)(C)CNC(=O)C(C)NC(c2cccs2)=O)sc(CO)nc1C 99437,C1(C(=O)NC(C2(OC)CCC2)C)CC12CCN(C(c1cccc(F)c1O)=O)C2 99438,N1(C(C=CSC)=O)CCC(F)(CNC(c2cn(C3CC3)nn2)=O)CC1 99439,Nc1cccc(C(=O)NCCOC2CCN(C(=O)C(O)CN3CC=CC3)CC2)n1 99440,C(=O)(C1Cc2ccccc21)N1CCC(C(N(CC(C)CO)C)=O)CC1(C)C 99441,c1(C(CCC#N)=O)ccc(-c2c[nH]nc2C(=O)N(CC)CC2CCCCC2O)cc1 99442,c1(C(=O)NC(C)CCCNC(C2COCCO2)=O)cnc2cc(Br)ccc2c1 99443,CC(C)(C)CC(=O)N1CCCC1CNC(C12CC(c3ccccc3)(C1)C2)=O 99444,N1(C(c2ccc(C(=O)OC)cc2)=O)CC(N(C)C(c2conc2C)=O)C2(CC2)C1 99445,N1(C(Cc2cccc(COC)c2)=O)CCN(C(c2nc(O)sc2C)=O)C2CC12 99446,N1(C(CC(C)CC2CCCN2C(=O)OC(C)(C)C)=O)CCCCC1C1CC1 99447,c1(SC)cc(F)ccc1C(=O)NCCC1CN(C(=O)CN2CCCC2C)C1 99448,Cc1cccc(C2=CCN(C(=O)NCC3C(CO)C3(C)C)CC2)c1 99449,C(CN=c1nc(O)c(Cl)c[nH]1)c1onc(-c2c(C)cccc2)n1 99450,N1(C(C2N(C)CC(O)CC2)=O)CCC(C(N2CC3(CO)CC3(CO)C2)=O)CC1(C)C 99451,CC1COc2c(C(=O)NC3CC4CCC3N4C(=O)CC3CCOCC3)cccc21 99452,c1(C(N2CCCN(C(CC(C)C3CCCO3)=O)CC2)=O)ncccc1N=[N+]=[N-] 99453,C(CC(=O)N1CCCC(CNC(=O)CN(C(=O)C(C)C)C)CC1)(C(C)C)OCC 99454,C(=O)(C1=C(Cl)CCOC1)NCC12CN(C(c3c(OC)cccn3)=O)C(C1)CO2 99455,C1(CNC(C=CCC)=O)CCCC(CNC(=O)C(F)(F)c2cscn2)C1 99456,c1(C(=O)NCC(CNC(C2(CCC)CC2)=O)C)cc(OC)c(OC)cc1O 99457,N(C(=NCCc1ccc(Cl)nc1)NCC1CCCCO1)Cc1c(CC)nn(C)c1 99458,c1(C(N2CCN(C(C3C(C)CCCC3)=O)CC2)=O)cc(P(C)(C)=O)ccn1 99459,CCC(CC(F)F)C(=O)N1CCCC1C(=O)NC1(c2ccc(F)cc2)CC1 99460,CS(=O)(=O)CC(F)(F)CCNC(c1nnn(Cc2ccccc2)c1Cl)=O 99461,N1(C(C2CC(C#C)(O)C2)=O)CCC(C)(C)C1CNC(=O)COc1ccccc1C 99462,c1(C(N2CCC(NC(C3CCCS3)=O)C2)=O)cc(F)c2cc[nH]c2c1 99463,N1(C(c2c(C)cnnc2)=O)CC(NC(c2cc(C3CCC3)nn2C)=O)CCC1C 99464,c1(COC)nn(C)cc1C(=O)N(CCNC(c1cc[nH]c1C1CC1)=O)C(C)C 99465,N1(CC(=O)NCCCN2CCN(C(C(CC)(C)O)=O)CC2)C(=O)NC(C)(C)C1=O 99466,C(=O)(C1=CC2(CCOC2)C1)N(CC(C)(C)CNC(=O)CCCn1ccnc1)C 99467,CC(C)(CCCCNC(c1cc(Cl)ccc1F)=O)NC(c1coc(C2CC2)n1)=O 99468,CC(C)CC(C)C(=O)NCC1CC2CCC1N2C(C1CC=CCC1)=O 99469,S(=O)(=O)(c1ccc(Br)cc1NCC1CCCCCCC1)N1C2CC(=C)CC1CC2 99470,c1(C(=O)NCCC2(CNC(C(CCOC)C)=O)CC2)cc(C)c(F)cc1F 99471,N1(C(C(CCC#C)O)=O)CCCN(C(c2cccc(Cl)c2C)=O)C(C(C)C)C1 99472,CC(C)(O)C(F)CNC(C1(C2CCCN2C(=O)CC2CCCO2)CC1)=O 99473,CC1CC(C(=O)NCCCOCCOCCNC(C2(F)CCCC2)=O)CC(C)C1 99474,CC1C(NC(c2cnccc2Cl)=O)C(C)CCN1C(c1cc(N(C)C)ccn1)=O 99475,c1(OCC)ccc2c(c1)C(NC(=O)N(CCCc1nc(C)cs1)CCO)CCO2 99476,N1(CC(=O)NCC(=O)N(C)CCN(C)C(c2ccccn2)=O)CCCCS1(=O)=O 99477,c1(C(=O)NCC2CCCN2C(c2cnn(C3CCOC3)n2)=O)cnn2c1CCC2 99478,c1(CNCC2(C)CCN(S(=O)(=O)CC3CC(N)C3)CC2)ccc(Cl)c([N+](=O)[O-])c1 99479,C1(NC(c2cc(C)oc2)=O)CCCCN(C(C2CC(OC(C)(C)C)C2)=O)C1 99480,CCC(C)(O)C(=O)N(CCCNC(C1C(C(F)F)C1(C)C)=O)CCO 99481,CC(C)(F)CC(=O)NC1CC(CNC(=O)Cc2c[nH]nc2O)C1 99482,N1(C(c2c(OC)cc(Cl)c(Cl)c2)=O)CCCC2(CCC2O)C1 99483,c1(-n2c(C(c3n(CC)ccn3)NCCn3cncn3)nnn2)ccc(Cl)cc1F 99484,Cc1ncc(Br)c(N2CCOC(C(=O)NC(c3ccc(F)cc3)CO)C2)n1 99485,c1(C(=O)OCC(=O)N(CC)CC)ccc(Oc2cc(F)cc(Br)c2)c(F)c1 99486,Cc1csc(Cl)c1C(=O)NCC1COCCN1C(C1CC(C)(C#N)C1)=O 99487,N1(C(c2cc(CNC(CC(CC)O)=O)[nH]n2)=O)CCOC(C)CC1 99488,c1(COC)cncc(C(=O)N(C(C)CN(C(=O)CCc2cccs2)C)C)c1 99489,c1(CC)cc(C(=O)N(C(C)CNC(c2cc(C)c(CO)cn2)=O)C)ccc1O 99490,CC1SCCCC1C(N1CCC2CC12C(=O)NCCNC(=O)CO)=O 99491,Cc1cn2ccc(C(N3CCC(Cc4cn(CCO)nn4)C3)=O)cc2n1 99492,N1(C(C2ON=C(C)C2)=O)CCN(C(c2ccnc(CO)c2)=O)C(CCO)C1 99493,Cc1nc(Cl)ncc1NC(=O)C(c1ccccc1)NC(=O)CC1CCC(C)(C)C1 99494,N1(C(C(C)S(N)(=O)=O)=O)CC(NC(=O)C(F)(F)C2CC2)CC12CCCCCC2 99495,C(c1ccccn1)=C(C)C(=O)NC1CCC(C)(CNC(c2ccncc2)=O)C1 99496,c1(C(c2nnnn2CCOC)NCCC(CC)CO)sc2ccccc2c1Cl 99497,CC1CCN(C(c2ncsc2C2CC2)=O)CC1NC(=O)CSc1cn[nH]c1 99498,C(=O)(C(C(=O)NCCNC(=O)CC1CC=CCC1)OC)OCC 99499,C=C(C)CC(C(=O)NCC1CCC1C#N)NC(C1(C)COCCO1)=O 99500,N1(C(C)=O)CC(C(=O)NCCN(C)C2CC2)(C(C)C)C1.C12CC1C(=O)N2 99501,C1(CNC(c2cnn(C)c2Cl)=O)CCN(C(=O)C(C)(O)C2CCC2)CCC1(F)F 99502,c1(C(=O)NCC2C(C(N3CCC(CCCC)C3)=O)CCC2)cnc(O)cc1C 99503,C1(NC(C=CCN(C(=O)CCOC2CCCC2)C)=O)CCC(F)(F)C1 99504,C1(CNC(C(COC)N(C)C)=O)CCCC2(CN(C(=O)C(CC(C)C)OC)C2)O1 99505,S(=O)(=O)(c1c[nH]ccc1=NC(C(C)(C)C)C(C)(C)C)NC1CN(C)C(C)(C)C1 99506,C(=O)(C1c2c[nH]nc2CN1C(C1CCC1C)=O)N1CCCC(C)(OC)C1 99507,N1(C(C(CC)F)=O)CCC2(CCC(NC(=O)C=CC(C)C)C2)C1 99508,N1(C(C(C)CF)=O)Cc2ccccc2CC1CNC(=O)C(c1ccccn1)O 99509,N1(C(C(CCOC)NC(=O)C=Cc2ccsc2)=O)CCC2(CCC(O)C2)C1 99510,c1(C(=O)NC(CN(C(=O)C(C)NC(C2CCC2)=O)CC)C)cc(C2CC2)[nH]n1 99511,C1(C(=O)NCC2(F)CC(NC(c3cnc(Cl)s3)=O)C2)CC2C=CCC(C1)C2 99512,O=C1NC(=O)C(CNC(C2CC23CC(NC(c2[nH]nnc2C2CC2)=O)C3)=O)N1 99513,C1(NC(c2cccnc2OCC(F)(F)F)=O)CCN(C(=O)C(C)(C)CO)CC1C 99514,CCC1=NOC(C(=O)N(C2(C(=O)NC3CCNC(=O)C3)CCC2)C2CC2)C1 99515,C(CC(C(C)(C)C)NC(C1CC1OC(C)(C)C)=O)N(C(C=C(C)C(F)F)=O)C 99516,N1(C(CC(C)(C)SC)=O)C2CCC1CC(N(C)C(C1CC3CCC(C1)C3)=O)C2 99517,C(=O)(CC(COC)NC(C12CCC(OC)C1C2)=O)N(CCCCC=C)C 99518,C1(N(C(CC2(CCOC)CC2)=O)C)CCN(C(c2cncnc2)=O)CC1.C1CC1 99519,C(=O)(CCC(C(C)O)NCc1ccc(N(C)C)cc1F)OC 99520,N1(C(C2CC(C#N)C2)=O)CC23CCCC2(C1)CN(C(=O)C1=C(Cl)CC1)C3 99521,CC1CN(C(C2CC(C)(F)C2)=O)CCCN1C(c1cnc(C(F)(F)F)nc1)=O 99522,Cc1ccc(S(=O)(=O)Nc2cccc3nncn23)cc1NC(c1ccc(C)s1)=O 99523,N1(C(CN(C(C(C)C)=O)C)=O)CCC(CNC(=O)C(C(C)C)N(C)C)C12CC2 99524,C(=O)(CCCC(C)(C)C)N1CC(CC)N(C(=O)C(C)NC=O)CC1 99525,C1(CNC(c2cccn2Cc2cccs2)=O)CCCN1C(=O)CCC1CC1(F)F 99526,c1(C(=O)NC(CC)CNC(c2nc(=N)cc[nH]2)=O)ccc(NC)c(F)c1 99527,Cc1nc(Cl)nc(N2CC=C(CNC(c3cc(Cl)cs3)=O)CC2)c1[N+](=O)[O-] 99528,Cc1c(C(=O)NCC2CC2NC(=O)Cn2cnc(=N)[nH]2)[nH]c2c1CCCC2 99529,c1(C(N2CC(CC(C)NC(CN3CC(C)C3)=O)C2)=O)nc(C(C)C)ncc1Br 99530,C(C)(CC(C)(C)C)(c1nnnn1C(C)(C)C)NCc1nccc(C)c1 99531,c1(C(=O)NCC2C(NC(=O)CC(F)F)CCC2)ccc(-c2nc(=O)o[nH]2)cc1 99532,c1(C(C)=O)c(NC(=O)CC2(O)CCOC2)c(C#N)c2n1CCCC2 99533,CC(C)C(C)(Cc1ccccc1)C(=O)NCCc1ccccc1O 99534,c1(CC)cnc(C(=O)NC(c2cccc(C)c2)CNC(=O)C(=O)C(C)C)nc1 99535,n1(C(CC)C)nc(C(=O)NC2(C3CCCN3C(=O)Cc3ccoc3)CC2)cc1C 99536,Cc1cc(Cc2nc(CCC(C)(C)C)nn2CC(C)O)ccc1Br