SMILES N1(C(C(Cc2cc(C)[nH]n2)NC(=O)OC(C)(C)C)=O)CCC(C)(F)CC1 c1(C(N2CC(O)(CCNC(C3N(C)CCCC3)=O)C2)=O)ccc2c(c1)CCC2 c1(OC)ccnc(C(=O)NCC2CC(C)N(C(c3cc(C(N)=O)c[nH]3)=O)C2)c1C C1(OC)CN(C(=O)CN2CCC(C)CC2)CC1NC(C1CCCN(C(C)C)C1)=O Cc1nn(C)nc1C(=O)NC1COCC1CNC(=O)CC(C)c1ccccc1 C1(O)(C(C(=O)NC(c2cnsc2)C)NC(CCCOCC=C)=O)CCCCC1 C(=O)(N=c1[nH]c(Cl)c(Br)nc1Br)c1sc2c(n1)CN(C(C=CC)=O)CC2 c1(C(=O)NCC=CCNC(C2C(C)(C)CC2)=O)ccc2cc(Cl)ccc2n1 C(=O)(C(C(C)O)N(C)C)NC(c1cn(CCCNC(c2cccs2)=O)nn1)C(C)C c1(C(N(C(C)CNC(=O)CCN2CCC(C(N)=O)CC2)C)=O)ccc(O)nn1 c1(C(C)C)cc(C(=O)NC2CCCC(NC(=O)CN(CC(C)(C)C)C)C2)nn1C Cc1nccnc1C(C)NC(C1CSCN1C(c1c[nH]nc1Cl)=O)=O Cn1cnnc1CCC(=O)N(C1CCN(CCC=CC(=O)O)C1)CCO N1(C(CS(=O)(=O)NC)=O)CC(NC(C2(N(C)C)CCCSC2)=O)CC(C)C1 c1(C(N2CCCCC(Nc3c(C#N)c(Cl)ncn3)C2)=O)cc2cccc(F)c2o1 Cc1cc(-c2cncc(C(=O)Nc3nc(-c4ccccc4)c(Br)s3)n2)cc(C)c1 C1(C(=O)OC)CC(C)N1C(=O)CCC1CC1.C12(CC1C)C(=O)N2 CCC(CN=c1[nH]c(NC(CCO)C(F)F)nc2ccc(Cl)cc12)OC c1(OC)cc(Cl)ccc1CN=C(NC(C)C)NCC12CC(CN1C1CC1)C2 C1(O)(C(=O)NC2CN(C(c3c(OC)c(C)cs3)=O)CC2O)CCC(C)(C)CC1 c1(CC(=O)NCC2(O)CCN(C(C(COC)(C)C)=O)CC2)nnc2n1CCOC2 N1(C(C)CNCc2nnc(C3CC3)n2C)CCn2ncc(C(F)(F)F)c2C1 C(=O)(CC(O)C(C)C)N1CCC(C(C(=O)NCCc2ccn(CC)n2)C)C1 c1(CC(C)C)ncc(C(=O)NC(C)(C)CNC(C2CC2(F)Cl)=O)s1 c1(C(=O)NC23CN(C(c4c(CC)c(C)ccc4)=O)C(C2)C3)cc2ccccn2n1 C1(NC(c2cn(CCC(C)C)nn2)=O)CN(C(=O)C=Cc2ccoc2)CC12CC2 c1(CC)cncc(C(=O)NC2COCC2CNC(=O)C(C)(C)C)c1 c1(C(=O)NCCCC2CCN(C(C(OC)OC)=O)CC2)cn2ncccc2n1 Cc1csc2c(N(C3CCCNC3)C(c3c[nH]c4ccc(Cl)cc34)=O)ncnc12 N1(C(c2nccnc2Cl)=O)CCC(NC(C2(F)CCC2)=O)C(F)C1 N1(C(C(C(CC)C)O)=O)CCC2(CCCC2N2CCC3(CC2)CC(=O)N3)CC1 O=C(CCCSc1ccccc1)NCCCN(C(=O)Cc1cccnc1)C1CC1 CC1(C)CC(NC(C2CC(O)C2)=O)CN(C(c2cc(N)cc(F)c2Br)=O)C1 N1(C(C2=C(C)OCCC2)=O)CC2CCCCC2(NC(=O)C=C(Cl)Cl)C1 c1(OC)ncc(F)c(Nc2ccc(NC(c3cc(F)c(C)s3)=O)cc2)n1 C1(C(=O)NCC2CC3(CC3)CN2C(c2cc(F)cc(F)c2)=O)CCCC1C1CC1 N1(C(C2(CC)CC2(F)F)=O)CCCN(C(=O)C(C)(F)CC)CC1 CCC(C)(C(=O)NCCCCC(C)NC(=O)COCc1nc[nH]n1)C(N)=O c1(NC(C(C2CN(C(=O)C(F)C(F)(F)F)C2)OC)=O)cnc2ccnn2c1 C1(N(C(c2cn(CC(F)(F)F)nn2)=O)CC)CCCN(C(C2CC2C)=O)C1 CS(=O)(=O)c1cncc(C(=O)NC2CCCN(C(C34COCC3C4)=O)C2)c1 N1(C(COC(CC)C)=O)CCC2CCN(C(c3c(O)cc(F)cc3F)=O)CC2C1 N1(CC)CCC(CNC(c2ccc(-c3cnn(C)c3)s2)=O)C1 c1(OCC(=O)OCC)cc([N+](=O)[O-])ccc1NC(c1ccc(Cl)cc1)C N1(C(CCC(C)OCC)=O)CCC(NC(c2occ3c2CCC3)=O)CC1C C1(C(N2CC3C(CNC(c4cc(C)sc4)=O)(C3)C2)=O)CC2(C1)CC(C)C2 c1(CNCc2cn(-c3c(C)ccnc3)nn2)ccc2nnnn2c1 N1(C(CNC(C)=O)=O)CCC(NC(=O)Cc2scnc2-c2ccccc2)C(F)C1 Nc1cc(C(=O)NCC2(NC(=O)CC3(O)CCC3)CC2)cc(F)c1 C1(CC(=O)NCc2cc(C(=O)NCC3(O)CCC3)ccn2)CC(=O)NC1=O N1(C(CNS(NC)(=O)=O)=O)CC(CNC(=O)Cc2nonc2C)N2CCC1C2 c1(OC)ccc(Cl)c(C(N2CC(NC(c3c[nH]c(C(N)=O)c3)=O)C3(CC3)C2)=O)n1 c1(OC)cc(-c2c[nH]nc2NC(c2ccnc(F)c2)=O)cc(F)c1CS(C)(=O)=O CC1(C)C(NC2CCC23CCCC3)CC1O N1(C(C2(CCC)CC(=O)C2)=O)CC2(CC(CC(=O)NCC(C)C3CC3)C2)C1 C(C(CC(=O)NCC1C2CCCC12)NC(=O)CN1CC(=O)NC1=O)OC CC1=NOC(C(N2CCCC2CN(C(=O)CN2CC3CC3C2)C2CC2)=O)C1 C1(C(=O)NCC2(C(C)(C)C)CCN(C(CP(C)(C)=O)=O)C2)CC1C1(C)COC1 N1(C(C(=O)NCCCF)C(C)Cc2c(OC)cccc2)CCNC(=O)C12CCC2 S(=O)(=O)(c1cnc2ccccc2c1)N(C1CCCC(C)C1)C C1(C(=O)NC2(CC#C)CC2)CCN(C(c2[nH]ccc2COC)=O)CC1(C)C N1(C(CC)=O)CCCC(C(N2CCC3C(NC(c4ncn(C(C)C)n4)=O)C23)=O)C1 c1(C(=O)NC2(CNC(C(CC)C)=O)CCCC2)cnn(-c2ccc(F)cc2)c1C CC1CC(NC(C2(C)CCN(C)C2=O)=O)CCN1C(=O)Cc1cc(Cl)cc(Cl)c1 C(=O)(C(CCCCN)CC(F)(F)F)N1CC(NC(Cc2cc(C)on2)=O)C1 CC1(C)CN(C(=O)CC23CCC(CC2)C3)CC(CNC(=O)C=CC=C(Cl)Cl)O1 N1(C(=O)CCn2nc(O)c3ccccc23)CCCC2(CCN(c3nccs3)C2)C1 C1(C(N2CCC(NC(Cc3nc(NC=O)sc3)=O)C2)=O)CC2COCC2C1 c1(C(=O)NCC2CCCN(C(C(C)SCC)=O)C2)c(OC)cc(Cl)cc1F C(CCN=C(NCc1ccc(SC)o1)N1CCC(C(F)(F)F)(CO)C1)OC Cc1ccc(N2CCCC2NC(=O)COC(C)(C)CN2CCNCC2)cc1 N1(C(C(C)C(F)F)=O)CC2CC(C1)C(CO)C2NC(C1C2C3CCC(C3)C12)=O C(=O)(C(C#N)C(C)(C)C)NC(C)(C)CCNC(=O)Cc1cncc(O)c1 N1(C(CC)=O)CC(C)N(C(c2cc(Br)c(Cl)cc2OC)=O)CC1C C(C1=CCN(C(C2CCCC23CCC3)=O)CC1)NC(=O)CCC1CCOC1 c1(C(N(C2CCN(C(=O)CC3CC34CC4)C2)C)=O)ccnn1CC1CCC1 CC1CCN(C(c2csc(CNC(C3(N4CCCC4)CC3)=O)c2)=O)CCO1 C1(C2CCN(C(=O)C(C)(C)CS(C)(=O)=O)CC2)(NC(C(CC)CCOC)=O)CC1 N1(C(c2c(CC)c[nH]c2)=O)CC2CCN(C(=O)C(COC)N(C)C)CC12 C1(C(N(C2(CC)CCN(C(c3coc(CSC)n3)=O)C2)C)=O)CC2COCC2C1 N1(S(=O)(=O)CCCl)CCN(Cc2cc(Cl)cc(Cl)c2F)C2(CC2)C1 N#CC1CN(Cc2cccs2)CC1NC(C1(c2cncc(Br)c2)CC1)=O C1(NC(c2c(Cl)cn(CC)n2)=O)CC(CNC(C2SCCS2)=O)C12CCC2 C#Cc1ccc(C(=O)N(C)CCOCCNC(C2CC2CC)=O)cc1 C(=O)(CC(C)(C)C(=O)NCC1(NC(=O)C(C)O)CCOCC1)OCC c1(CC(C(=O)NCC(N(C(COCCCC)=O)C)C2CC2)O)ccc(Cl)cc1 C1(NC(=O)CC2CCOC2)(CO)CCCN(C(c2ncccc2C(F)(F)F)=O)C1 C1(C(N2CCC(CCNC(CC3C(C)CCO3)=O)C2)=O)CC(=O)NC(=O)C1 C1(NC(C2C(C(C)NC(C(CC)CN(C)C)=O)C2)=O)CC2(CCCCO2)C1 CCC(C)CCCC(=O)NC(C1CCCN1C(c1cccc(C#N)c1C)=O)C Cc1ccc2c(CNC(N3CCC(O)(Cc4ccc(Br)cc4)C3)=O)cn(C)c2c1 C1(C(C)CNC(=O)C(C)(C)c2ccccc2)CCN(Cc2ccccc2Br)CC1 CC1CCCC(C)N(C(c2conc2CNC(=O)C(C)n2cccn2)=O)C1 C1(C(=O)NCC(=C2CN(C(CC3(CSC)CC3)=O)C2)F)CCCCN1S(C)(=O)=O c1(C(N2C(CNC(CC(C)OC)=O)C(C)(C)CC2)=O)cccc2c1C(=O)CC2 c1(C(N2CC(O)(CNC(c3ccc(C(C)=O)cn3)=O)C2)=O)cc(O)nc(O)n1 CC(O)C(=O)N=c1ccn(C2CN(Cc3nc4ccccc4s3)C2)[nH]1 C1(NC(C2N(C(C(NOC)=O)=O)CCOCC2)=O)CCOCC12CCC2 N1(C(C(C(C)CC)N(C(CC=CC)=O)C)=O)C2CCC1CC1(CC1)C2 c1(NC(c2ccc(C3CC3)c(F)c2)c2n(CC(=C)C)nnn2)ccc(F)c(Br)c1 C1(CC(=O)NC(CNC(C2(SCC)CC2)=O)C(C)C)CCCCCO1 C1(NC(CCc2nc(C)sc2)=O)C2COCC1CN(C(c1cnncc1C)=O)C2 C=CC1CN(C(C2C3CC4C(C3)C24)=O)CC1NC(=O)C(C)CC(N)=O CC1(C(N2CC(OCCNC(c3ccnc(-c4ncc[nH]4)c3)=O)C2)=O)CC=CCO1 CC(C)=C=CC(=O)NCCCN(C(=O)CC(C)C)C1CC1 C1(SCC)CCC(C(N2CC(c3cn(C4CCCC4C(=O)O)nn3)C2)=O)CC1 CCC(CC)(CO)C(=O)NC1CC(NC(=O)Cn2cc(Br)nn2)C1 CC(C)(C)C(C(=O)N1CC2CC2(CNC(c2cc(C#N)c[nH]2)=O)C1)C1CCCC1 C1(C(N2C(CC(=O)NCc3c(COC)ocn3)CCC2)=O)CCCN1C=O N1(C(c2[nH]cc(C)c2)=O)CCN(C(=O)CCc2c(C)nc(C)nc2O)C2CCC12 C(=O)(C(C)CCCCCC)N1CC(C(N2CC(C#C)(F)C2)=O)C(C)(C)C1 c1(C(c2n(CCC)nnn2)NCCCN(S(=O)(=O)CC)C)ccnc(Cl)c1Cl C1(C(N(C(CCCC)C)C)=O)CN(C(=O)Cc2c(C)cnn2C)CCN1C c1(OC)c(Cl)cc(C(=O)NCC23CC2CN(C(c2cnnc(O)c2)=O)C3)nc1Cl Cn1cnc(CCC(N2CC(O)(C(F)C(=O)NCc3ncon3)C2)=O)c1 CCCC(CCCNC(C1CCCSC1)=O)NC(c1cc(CSC)c(C)s1)=O N1(C(C)=O)CCCC1(C)C(=O)NCC1(O)CCN(C(=O)CCCC2CC2)C1 C#Cc1c[nH]nc1C(=O)NCC1CC(F)CN1C(c1ccoc1Cl)=O c1(C(=O)NC(CC=C)CNC(c2ncn(CC)n2)=O)ccc(C2CC2)cc1C c1(CC)ccc(C(=O)NC2CCC(C)N(C(c3cc[nH]n3)=O)C2)cc1CC N1(C(C(C)N(C(c2cnnc(C)c2C)=O)C)=O)C2CCC1CC(C)C2 c1(N2C(CNC(C(C(CC)O)C)=O)CCC2)nc2c(F)cc(Cl)cc2s1 C(CC(CC)C(=O)NCC(O)CC(=O)NC(C)C(C)C(=O)OC)=CC C(=O)(CCCC(C)(C)C)N1CC(C(=O)NCCCC(=C)Cl)C(C)C1 n1(CC)cc(C(=O)NC23CC2CN(C(C2CCN2C)=O)C3)c(C)n1 c1(C(=O)N(c2cnc(C3CCNC3)s2)Cc2ccco2)ncc(Cl)cn1 C1(N(C(c2coc(Cl)n2)=O)CC)CCCN(C(=O)Cn2ncc(Cl)c2C)C1 c1(C(=O)NCC2C(C)CCN(C(=O)C(C)(C)CO)C2)ccc(S(N)(=O)=O)nc1 C(=O)(C(C)(C)C1=CCSCC1)N(CC(C)(C)NC(C1CCCC(CNC)C1)=O)C CCCC(CCCNC(C1CCC(O)CC1)=O)NC(=O)CCF CC1(C)CCCOC1CC(=O)NC(CO)CCCNC(=O)C(F)(F)C1CC1 CCC(CC)C(c1nnnn1C(C)CC)NCc1csnn1 CC1OCCOC1C(=O)N(C)CCNC(=O)C(C1(O)CCCC1)F CN1C(C(N)=O)CCC1C(N1CCOC(CCNC(c2cnc[nH]2)=O)C1)=O C1(CNC(CC(C)(C)NC(=O)CCNC(=O)CO)=O)CC2(CCCO2)C1 c1(C(=O)OCCN2CCN(C(c3c(OC)ccs3)=O)CC2)cc(F)c(Cl)c(Cl)c1 C#CCC(CC(=O)N(C(C)C(=O)N(C)C)C)NC(=O)C(C1CC1)OC c1(CC(N2CC(C)N(C(C3CN(C)CCO3)=O)CC2)=O)cncc2ccccc12 CC1CN(C(=O)CC2CC(=O)C2)CCN1C(c1c[nH]nc1-c1ccco1)=O c1(C(=O)NC2C(NC(CCCNC(N)=O)=O)CCCC2)ccc(S(N)(=O)=O)o1 c1(CC)nc(C)oc1C(=O)NCCOCC(=O)NCC(O)CO C1(C(N2CC(O)CC(NC(C(CCSC)(C)C)=O)C2)=O)CCc2c[nH]nc2C1 c1(C(N(C2CCN(CC(O)COC)C2)CCC)=O)ccc(CC(C)C)cc1 c1(O)ccc(CN2CC3C(NC4CCN(Cc5cc[nH]n5)CC4)C3C2)cc1.CC c1(C(=O)NC2C(NC(=O)CSC3CCCO3)C2)cc(C(F)(F)F)ccc1F C12(C(N3CC(CNC(CC4(C)CC4(F)Cl)=O)C3)=O)CC3CC(C1)CC(F)(C3)C2 C(CCCC(=O)NC1CC(C)(C)C1)NC(C(C)(C)F)=O N1(Cc2cc(C(F)(F)F)c(F)cc2)CC2CN(C(=O)Nc3cccc(C)c3)CC12 N1(C(C(CC)CO)=O)CCC(C2CCN(C(=O)C(C3CCOCC3)C)CC2)CC1 c1(NC(C2C(NCc3cn(CC)nc3)C2)=O)cc(F)ccc1C c1(C(=O)NCCC(C)NC(c2n[nH]c(C3CC3)c2Cl)=O)cncc2cccnc12 C(CC(N)=O)(C(=O)N1CCC(C)(C)CC1)NC(c1c(OC)noc1C)=O C(=O)(CCCCO)NC(CNC(CCSC)=O)C C1(N(C2CCOCC2)C(C(N)=O)=O)C2CC(n3cc(-c4ccncc4)nn3)C1C2 c1(OC)ncc(C(=O)OCC(n2cc(-c3cncc(N)c3)nn2)C)cc1C C(=O)(CS(=O)(=O)C(C)C)NC(CNC(CCC(=O)NCC)=O)CC(C)C Cc1ccc(Br)cc1CC(=O)NCC1CCCN1Cc1ccc(Br)cc1Br N1(C(C2(F)CCN(C(CC3(OCC)CC3)=O)C2)=O)CC(C#N)C2(CCC2)C1 C(=O)(C#CC1(C)COC1)N1CC(N2CCN(C(C3C(C)OC(=O)N3)=O)CC2)C1 C1(CNC(=O)C=Cc2ccco2)CC2(CCC2)CN1C(c1ncc(Cl)nc1Cl)=O c1(C(=O)NC(CC(C)NC(C(CCC)=CCC)=O)C)[nH]c2ccc(C)cc2c1C N1(C(CC2(C)CCCC2)=O)CCC2(CCN(C(=O)CC3(C)CCS(=O)(=O)N3)C2)C1 C(=O)(C#CC1CC(F)(F)C1)NC(CNC(C(CCCC)(C)F)=O)(C)C C1(CCC)(NC(=O)CCc2cc(C)[nH]n2)CCCN(C(=O)CS(=O)(=O)CC)C1 c1(C(=O)OC(c2ccccc2)COC(C)=O)cc(F)c(O)c(Cl)c1 C1(C(=O)NCC(CC=C)(C)C)CC(C)(C)CN1C(c1ccnc(O)c1F)=O c1(CCC(=O)N(CC(C)(C)CNC(c2cnn(C)n2)=O)C)ccc(C2CC2)cc1 C1(NC(=O)COc2cncc(Cl)n2)COC2(CCCN(C(C3CC(O)C3)=O)C2)C1 CCCC(C)CC(C)NCc1cccc(N(CC(F)(F)F)CCC)c1 c1(CC(N2CCC(C)C(NC(=O)CNC=O)C2)=O)cccc2ccoc12 CCCCC(CNC(c1ccc(SC)cc1)=O)NC(c1n[nH]cc1C1CCC1)=O C1(CC(=O)NCC(C)(O)C2CC2)C2CN(C(c3csc(Cl)c3)=O)CC12 CC(C)CC(O)C(C)C(=O)N1CCC(N=[N+]=[N-])(C(=O)NC2CC(N3CCCC3)C2)C1 N1(C(C)C)CCCC1C(=O)NCCCCNC(=O)Cc1cc(C(F)(F)F)n[nH]1 c1(C(N2CCOCC(NC(C(CC)(C)C)=O)C2)=O)cc2c(F)cc(F)cc2[nH]1 c1(OCCC(=O)NCC=CCNC(CSCC)=O)ccccc1F N=c1[nH]cncc1C(=O)NCCN(C(=O)CC1CCCC(=O)N1)CC1CC1 c1(OC)cc(Br)ccc1CCC(=O)NC1CN(C(=O)CNC(C)=O)CC1C Cc1c(C(=O)NC(C)(CO)C(=O)NC2CCN(CCF)C2)ccn1C c1(C(=O)NCC2(C)CCCN2C(C2CCSCC2)=O)ncc2ccccc2c1O N1(C(C2C(C)OC(=O)N2)=O)CCC(F)(C(=O)NCC2CCSC2)CC1 C(=O)(CCN=C(NCC(c1cnn(C)c1)O)NCC1CCCC1O)NC(C)C C#Cc1ccc(NC(C2CCC(C3CC3)N2C(c2coc(N(C)C)n2)=O)=O)cc1 c1(COCCC(=O)NCCn2ccc(C)n2)ccccc1Br CC(C)(CC(=O)NCC1CCC1NC(c1cc(F)ccc1F)=O)CC(F)(F)F C(CC(C)C)(C(=O)N1CCC(F)(C(=O)NOC)CC1)NC N1(C(c2c(C)ncs2)=O)CC(NC(=O)C(C)CC(C)(C)C)CC(C)(C)C1 CC(C)(CO)C(=O)NCC1CCCCN1C(c1ccc(C2(F)CC2(F)F)cc1)=O C1(NC(c2cccc(OCCC#C)c2)c2nnnn2C2CC2)CCN(C)C(C)C1 c1(C(=O)N(C2CCOCC2)CCO)c(-c2ccccc2)noc1C1CC1 N1(C(c2n(CCC)ncc2)=O)CCCC(NC(c2cncc(C(C)(C)C)c2)=O)C1 C1(C(N2CCC(NC(c3c(C)cc(F)nc3)=O)(CF)C2)=O)CC(C)CC(C)(C)C1 C12(CNC(C3N(CC)CCCC3)=O)CCC(CC1)CN2C(=O)C(C#N)C(C)C CC1(C)CCC(CN2CCC(c3ccccc3Br)C2)OC1 C#CCCN=C(NCC1CC(C)CO1)N1CCc2cc(OC)c(Cl)cc2C1 C1(C(C)C)CC(C(N2CC3CC2C3NC(=O)Cn2cccnc2=O)=O)CCO1 C1(CNC(C2C(CC)CCC2)=O)CC(O)CN1C(=O)CCCc1ccsc1 C1(C(N(C)CC2CN(C(=O)C=Cc3ccnn3C)CCO2)=O)CC(C)(C)CCO1 CC(C)(CNC(C1(C)CC2CCC1O2)=O)CC(=O)NCCc1ccnc(O)c1 C12(NC(C(CCCC)C)=O)CC(C)(C1)OC21CN(C(=O)CC(C)C)C1 CC1=C(CNC(C2CC(NC(=O)Cc3ccoc3)C(O)C2)=O)COCC1 C1(NC(C(F)=CCC)=O)CCCC(N(C)C(c2cc(Br)cn2C)=O)C1 C1(N(C)C)CCCN(C(C2CC(C)(C)CO2)=O)C1.C12(CCCCC1)CC(=O)NC2 N1(C(c2c(C)ncs2)=O)CCN(C(=O)Cc2cc(CF)on2)C(CS(C)(=O)=O)C1 CC1(C)COC(C(=O)NCC(C2CCC2)NC(=O)CCN2CCOC2=O)C1 CC1(C)CCN(C(C2CCC3(CCC3)CO2)=O)CC1NC(c1coc(Cl)n1)=O c1(C(=O)NC(C2CCCCC2C)C)cc2c(cc1F)NCCC2 S(=O)(=O)(c1ccc(N2CC3CC2C3)cc1Br)NCC1C(C)C1 N1(C(C2(CC)CN(C(Cc3cn(CC)nn3)=O)C2)=O)CC2C(C1)C2(F)F C1(C(=O)NCC(CNC(CC2(OC)CCCCC2)=O)O)CNC(=O)C(C)(C)C1 C(=O)(C(C(C)CC)N(C)C(c1ccncc1O)=O)NC(C#C)C(C)(C)C CCC(C#N)C(=O)NCC1CCCN1C(=O)CCCSC(C)(C)C N1(C(C(=O)NCCn2ccc(C#N)n2)=O)CC2COCC(C2)C1 C1(C(=O)NC(c2c(C)nns2)C)CC(C)(C)CCN1C(=O)CC12CCCC1C2 N1(C(C(C)(C)C2CC2)=O)CCN(C(=O)CC2(CC3CCOCC3)CC2)C(CO)C1 CCC(C)CC(C(=O)NC1CCCCCC1)NC(=O)CC1(N(C)C)CCC1 C1(NC(C2(CSC)CCC2)=O)CCOCC1C(=O)NCCc1ncnn1C N1(C(c2c(C)cc[nH]2)=O)CCCC2(CCCN2C(c2cc(F)cnc2O)=O)C1 N1(C(Cn2c(C)nnn2)=O)CCC2CN(C(c3ccc4c(c3)NCC4)=O)C(C)C12 c1(C(=O)NC2CN(C(C=CCCC)=O)CC(O)C2)cc(F)c(F)cc1OC C1(CN=[N+]=[N-])(N(CC(=O)NC2CC2)C(c2cc(F)ccc2I)=O)CCCCCC1 C(=O)(C1CCc2c[nH]nc21)N1CC2C(CN3C(C)CCCC(C)C3)(CCC2)C1 c1(OCC=C)ccccc1C(=O)NCC1CC2CC2N1C(C1(CN(C)C)CC1)=O c1(C(N2CC=CC(NC(c3c(C)snn3)=O)C2)=O)cc(F)c(C#N)c(F)c1 n1(CC)cnc(C(=O)N(Cc2nccs2)CC2CC2)c1 c1(C(N2CC(C(C(=O)NCc3ccco3)OC)C2)=O)cncc(F)c1C C(=O)(C1CCc2ccccc21)NC1C(C)(C)C(C(N2CCC3(CCC3)C2)=O)C1 C=CC(O)C(C)(C)C(=O)N1CCCC(C)(C(C=O)OCCCSC)C1 c1(OC(CC)C(=O)NCC2CC(NC(=O)CCc3nccs3)C2)ccccc1F CC1CN(C(=O)CC2(O)CC2)CCN1C(c1ccc(-n2cccc2)cc1)=O C12(C(=O)NCCCN(C(c3cc[nH]c3C)=O)CC)CC(c3ccccc3)(C1)C2 C(C(C)(C(=O)NCC(C1CC1)N(C)C(C1CCCN(C)C1)=O)OC)OC c1(OCC)ccccc1-n1nnc(NC(=O)CCSC(F)(F)F)c1C CN1C(=O)CSC1=CC(=O)N1CCC(NC(c2ccnc3cccnc23)=O)C1 C1(CN(C(C(C)OCC=C)=O)C)COCCN1C(c1cc(C2CCCC2)[nH]n1)=O C1(F)(C(N(CC(C)O)CC(F)F)=O)CCN(C(=O)CSC2CC2)CC1 Cc1cc(F)cnc1C(=O)NCC1CC(CNC(c2ccccc2CO)=O)CO1 CC12CN(C(=O)C(N3CCC(Cc4cccc(Cl)n4)C3)=O)CC1(C)CS(=N)(=O)C2 C1(NC(=O)NC(C(C)(C)OC(=O)C(F)(F)F)=O)CCN(CSC2CC2)CC1 C=CC(CCC)CC(=O)N1CCC2(C(=O)NC3C=CCC3)CCCC12 N1(C(C(C)OC)=O)CC2(NC(C3CC3c3csc(Br)c3)=O)CCC1CC2 C1(CN(C(=O)CCSc2ccc(C)cc2)CC)CCCN(C(=O)CS(C)(=O)=O)C1 N1(C(CCC=C(C)C)=O)CCC2(CC1)CC2C(=O)NCCc1cccs1 C1(N(C(=O)CCC2CCCO2)Cc2ccccc2)CCCN(CC2CC2)CC1 C1(CC(N2C(CNC(C3CC3C3CC3)=O)CCC(C)C2)=O)CCCC2(CCC2)O1 c1(C(C)=O)ccc(=NCCNC(c2cc(Br)ccc2N(C)C)=O)[nH]c1 S(=O)(=O)(c1cnc2sccc2c1)N1CC(N(C)Cc2cccc(C)c2)C1 C12(CNC(c3c(CC)n[nH]c3)=O)CCC(CC1)N(C(C1(C)CCC13CCC3)=O)C2 c1(C(=O)NC2CN(C)C2)ncccc1NC(C1CC1CN)=O.C(C(F)(F)F)O C(C(=O)NCC(C)(O)CNC(c1ncnn1CC)=O)(C(C)C)OCC CC(C)CC(C(=O)NCC1C=CCOC1)NC(c1cnc(S)nc1)=O C1(NC(C2(F)CC2)=O)CCCN(C(=O)CCOC2CC2)C1 CC1CC(C(=O)NC2CCCCCC2NC(c2cn(C)nc2C(C)(C)C)=O)=NO1 CN1C(=O)CCC1(C)CNC(C1(CO)CCN(C(C2CCCC2C2CC2)=O)C1)=O c1(CS(C)(=O)=O)cccc(CNC(C2CCCN(c3ccccn3)C2)=O)c1 C(=O)(CCCS(C)(=O)=O)NCCC(C)CCNC(=O)CSc1ccnc(Cl)c1 CCC(CC)CC(F)C(=O)NC1CC(C(C)NC(c2cc(C)oc2CC)=O)C1 c1(N2CC(C(C)NC(c3cccnc3N(C)C)=O)C2)nc(Cl)nc2c1CCOC2 C1(O)(CNC(C2CCN2C(CC(F)(F)F)=O)=O)CCOCC1 C12(C(=O)NCC(CC)NC(C3(SC)CC3)=O)CCN(CC1)CC2 C=CCC(C(=O)N1CC(C(N)=O)(N(C)C)C1)NC(=O)Cc1cn[nH]c1 C(=O)(C1=CCC(C)CC1)NCC(CC)NC(c1nccc2ccsc12)=O N(C1CCCOc2ccc(Br)cc21)C(=O)NC1CN(C)CC1c1ccccc1 C1(C(C(=O)NC2C3CCN(C(c4ccnnc4)=O)C23)O)CCS(=O)(=O)CC1 C1(NC(CCC(N)=O)=O)CC2CC(C1)N(C(=O)CCC(=O)OCCC(N)=O)C2 C1(C(=O)NCCOCCC(=O)NC(C(CCC)O)C)CCC2(CCC2)O1 C1(CC(=O)NCC(CCCC)NC(c2cc(O)ccc2N)=O)CCCC(C)(C)O1 c1(C(C)C)ccc(C(N2CC(O)(CNC(c3ccc(-c4ccco4)s3)=O)C2)=O)o1 CN1CCN(C(c2cn3c(n2)SCC3)=O)C(CNC(C2(C)C=CCC2)=O)C1 c1(C(=O)NCC2(C)C(C)CN(C(=O)C(C)(C)C(C)O)C2)c[nH]c2ccc(F)cc12 c1(OCCC)cc2c(cc1CNC1(C(=O)O)CC(C(=O)O)C1)OC(C)C2 c1(C(C(=O)NC23CC(CNC(C4C(C#C)C4)=O)(C2)C3)O)ccc(C2CC2)cc1 c1(C(N2CCC(NC(CSCCC(C)C)=O)C2C2CC2)=O)ccc2ccsc2c1 C1(C(=O)NCC(CC(C)C)NC(c2cc(O)cnc2Cl)=O)(OC)CCC(C)CC1 C(CN=C(NCc1cn(C)nc1Br)NC1CC1)NC(=O)NC c1(OCC)cc2ccccc2cc1C(=O)NS(=O)(=O)CCC1CC1 c1(C(N2CC3CC(C(=O)NC)(C3)C2)C(=O)NC)ccc([N+](=O)[O-])c(Cl)c1 C(=O)(CCCCCn1cnnn1)NC1(CNC(C2C(C)C2)=O)CCOCC1 c1(C(=O)NCCCCN(C)C(c2cnc(O)n2C)=O)ccc(Cl)c(C(F)(F)F)c1 N1(C(C(C)CC2CC2)=O)CCN(C)CC1CNC(C1CCOC1C(N)=O)=O N1(C(CC2CCC(NC(C3(C)ON=C(C)C3)=O)C2)=O)CCCC(C)(CO)C1 CCC(C#N)(CC)C(=O)N1CCC(CNC(C2CC23CCSCC3)=O)(OC)C1 C1(C(=O)N(c2nc(C(=O)N(C3CCCC3)CCCCC)co2)CC)OC2CCC1C2 C(=O)(C(C)Cc1ccccc1)NCCN(C(=O)Cc1nccn1C)CC c1(C(N2CC(NC(CCC(=O)NC)=O)C(F)C2)=O)cccc(S(=O)(=O)C(C)C)c1 c1(C(N2CC(C)N(C(=O)C(C)CN3CCOCC3)CC2)=O)cccc2occc12 C12(CCC)CC(CC)(CN1C(=O)C(C)NS(=O)(=O)CCC)C2.C(=O)(CCOCC)NC C1(CN(CC(C)NC(=O)CCn2cccn2)C)CCC1C(F)(F)F C(C(F)(C(=O)N1CC2CC1CC2CF)C(C)C)NC(C1C(C(=O)OC)C=C1)=O C(C(CC(=O)NCC1CC1c1ccco1)C1CCC1)NC(C(OC)OC)=O N1(CCN(C)CCSc2nc(C)on2)CCN(C2CCSC2)CC1 C(C(C(C)(C)C)NC(=O)CNC(=O)CC(F)(F)F)NC(Cc1onc(C)n1)=O C1(c2n(C(c3ccc(C(F)F)nc3)C)cnn2)CCCN(C(=O)CCC(C)C)C1 C1(CNC(C(CC=C)CC)=O)CC2CCC1N(C(=O)CC(O)C(C)CC)C2 C1(NC(c2c(CC)cco2)=O)C2CCC1N(C(=O)Cc1cnc[nH]1)C2 C1(OCC(=O)NC(C)(C)CCNC(=O)Cc2nc[nH]n2)CCCCCC1 N1(C(c2c(C)ccnn2)=O)CC(F)(F)CC1CNC(=O)CCC(C)C Cc1[nH]nc(C(N2CC3(NC(=O)C(C)N(C)C(=O)OC(C)(C)C)CC2C3)=O)c1C N1(C(C2(C)CC2)=O)CCC(C2(NC(c3sc(Cl)cc3Br)=O)CC2)C1 C1(CC)CCN(C(=O)C2=C(C)OCC2)C(C(N2CCC=C(F)C2)C2CC2)C1 O=S(Cc1ccccc1)CCNC1CC1Nc1ccccc1 c1(C(=O)NC(C(CO)NC(c2c(F)ccc(OC)c2)=O)C)cc2c(s1)CCCC2 C1(OCC)CCCC1NC(c1c[nH]nc1CCNC(=O)CCc1ccncc1)=O c1(OC)n[nH]c(C(=O)NCCOCCNC(C2CCC(O)CC2)=O)c1Br C1(C(N(C)CC2CCCN2C(=O)CCCC(F)F)=O)CCCc2ccccc2C1 C1(NC(C2CN(C)C(=O)N2)=O)CCC2CN(C(=O)COCC3CCCO3)CC2C1 c1(C(=O)NC(CNC(=O)C=Cc2ccccc2Cl)CO)c[nH]c2cccnc12 C1(C(=O)NCC(N2CCC2CNS(CC)(=O)=O)=O)CCCN1C(C)C NS(=O)(=O)c1ccc(C(N2CC(NC(=O)C(F)(F)c3cncs3)CC(F)C2)=O)o1 c1(CN2CCC(NC(C3CCC(=C)CC3)=O)C(O)C2)cn(C)c2ncccc12 C(=O)(C(C(C)(C)C)C1CCC1)N1CC(N(C(c2cnc(CC(C)C)s2)=O)C)C1 c1(C(=O)NCC2C(OCC)CN(C(c3cc(Cl)no3)=O)C2)c(Cl)ccc(C)c1O N1(C(c2c(CC)nn(C)c2Cl)=O)CCCC(N=c2[nH]nc(C(C)(C)C)s2)CC1 N1(C(CC2CCCN(C)C2)=O)CC=C(CNC(C2(O)CCCCCC2)=O)CC1 c1(CCC)cc(C(=O)NC(C)CNC(c2ncccc2C(F)F)=O)sc1C c1(OCC)ccnn(CCCn2cncn2)c1=O.C(F)(C(=O)NC)=C.C12CC1NC2=O CCC(CCCC(=O)N1CC2CC2(C(=O)OC)C1)NC(C1OCCC1(C)C)=O c1(C(=O)OC)cccc(CNC(C)(C)CCCF)c1Br N1(CC)CCCC(C(=O)NCC2(C(=O)COC)CC2)C1.C123COC(C1)(C2)C3 N1(C(C2CCCC2O)=O)CC2CCCC2(C(=O)NCC2=CCCCC2)C1 C1(C(N2CC3N(C(C(CCCCC)O)=O)C(CC3)C2)=O)CC2(CCOCC2)CO1 c1(COC)cc(=NCCC2CCC(NC(c3csnc3C)=O)C2)[nH]cn1 CC(CC(F)(F)F)C(=O)NCCCOCCNC(=O)C(O)C1CCC1 N1(C(c2cccc(OC)c2C)C(=O)NC2CC(F)(F)C2)CCC2CCC(O)C1C2 C(=O)(CCCC(F)(F)F)NC(C1CC=CCC1)C(=O)NCc1cc(C)oc1 N1(C(c2cc(CCC)[nH]n2)=O)CC2(COC(CNC(=O)C(C(C)C)OC)C2)C1 Cc1cc(Cl)c(C(=O)NC2CC2NC(c2ccnc(CO)c2)=O)cc1N C(CN(C)C)(C(=O)NC1(C(C)O)CC1)NC(C(C)n1ccnn1)=O CC(N=[N+]=[N-])C(=O)N1CCC1c1cn(C2CCCCC2OC(F)(F)F)nn1 n1(C(C)(C)C)cc(C(=O)OCC[SH]=Cc2ccccc2)c(Br)n1 C(=O)(C1CCCn2nccc21)N1CCCC(NC(=O)C2=CC3CCCC23)CC1 C(=O)(CS(=O)(=O)CC(=O)NC1CCCCC1NC(c1cnc[nH]1)=O)OC C=CCC(CC(=O)NCC1(C)CCCCO1)NC(C1CCCCCN1C)=O C1(NC(Cn2ncn(C)c2=O)=O)CC2CC(C1)N(C(C1COC(=O)C1)=O)C2 O=C1CN(CCOC2CCCC2)C(=O)N1C(c1ccco1)c1nncs1 NS(=O)(=O)N1CCC(C(=O)NCCNC(c2coc(C(F)(F)F)n2)=O)CC1 C(=O)(C(C)n1cncn1)NCCCN(C(C1(CC)CC1)=O)C CC1CN(C(=O)C(=O)NCCOc2cccnc2)CCC1C c1(OC)ccc(C(=O)NC2CC(C(=O)Nc3cc(Br)cnc3O)C2)c([N+](=O)[O-])c1 N1(C(Cc2cc(CC)no2)=O)CC(CNC(c2scnc2C2CC2)=O)CC(C)C1 Cc1ccc(C(=O)C(N2CCC(N(C)C(c3nocc3C)=O)CC2)=O)cc1 c1(CCCC(=O)NCC2(CNC(C3(C(N)=O)CC3)=O)CC2)ccc(F)cc1 C1(NC(N)=O)CCN(C(=O)CN(C(=O)CN2CCNC(=O)C2)C2CC2)CC1 CCC(CC(C)C)C(=O)N1CCC(N(C)C(c2ncncc2F)=O)C1 N1(C(c2cn(CCC)nn2)=O)CCN(C(c2cnn(CC(=O)NC)c2)=O)C2CC12 C(=O)(C1=NN2CCCN=C2N1)N1C(CNC(CCCCSC)=O)CCC(C)(C)C1 c1(CN2C(C(=O)Nc3cccnc3C(F)(F)F)CC(=C)C2)ccc(C#N)c(Cl)c1 Cc1cc2cc(NC(C3CCN(C(=O)Cc4ccn(C)n4)CC3O)=O)ccc2[nH]1 C(C(CO)(CO)NC(=O)Cc1nocc1C)N(C(C(COC)NC(C)=O)=O)C C(CCCCCCC(=O)N1CC(CNC(c2ncc[nH]c2=O)=O)C(C)(C)C1)SC N1(C(c2c(C)nn[nH]2)=O)CC2(CCCC2NC(C2CC(=O)N(CC3CC3)C2)=O)C1 C1(CNC(COC)=O)CCC12CN(C(c1cc(F)ccc1C)=O)C2 C1(CNC(C(CC)SC)=O)CN(C(C2(CCF)CCC2)=O)CCC1(C)C c1(SC)ccc(O)c(NC(=O)NCC2CC(NCCS(N)(=O)=O)C2)c1 n1(CC)cc([N+](=O)[O-])c(C(=O)NCC2CN(C(=O)COC(C)C)CC2C)n1 C(=O)(CC(O)CC(C)(C)C)NCC1C(C(N2C(C(N(C)C)=O)C=CC2)=O)CCO1 c1(C(N2CCN(CCCN(C(CCC)=O)C(C)C)CC2)=O)c(C)cc(Br)cc1F c1(C(N2CCC(NC(C(CCC)CC)=O)C(F)C2)=O)ccc(O)c2c1CCCC2 S(=O)(=O)(c1cccnc1N(C)Cc1ccc(C)s1)NC(c1cc(C)on1)C C1(CN(C(C)CC(=O)NC2CC2)C)CCCN(C(C2CC23CCC3)=O)C1 C1(O)(C(=O)NC2CCN(C(=O)OC)CC2)CCN(C(C2CC23CCCC3)=O)CC1 c1(C(=O)NCCCCN(C)C(C2CC2F)=O)c(O)nnc2c1CCCC2 C12(NC(C3C4CCC(C4)C3C(F)F)=O)C3C4C1C1C2C3C41C(F)(F)F C1(C(=O)NCCN(C(CCc2cc(C)no2)=O)C(C)C)CCC2C1C2(F)F C1(NC(C2C(CC)C2)=O)CC2CC1N(C(C1(F)CCC1)=O)C2 c1(C(=O)NCC2(F)CC(NC(C3C(C)CC=CC3)=O)C2)ccc2ncsc2c1 N1(C(c2cncc(C3CC3)c2)C(=O)NCCCOC)CC(C)CCC12CC2 c1(N2CCC(C(C)NC(c3ccoc3)=O)C2)nc2c(cc1C#N)CCC2(C)C c1(C2(C(=O)NCC3N(C(COc4cc(C)on4)=O)CCC3)CC2)cccnc1Cl c1(OC)cccc(CCC(N2CCCC(NC(=O)C(C)(C)C#N)C2C)=O)c1F c1(C(C(N2C(C)(CNC(=O)Cc3cc[nH]c3)CCC2)=O)O)ccc(F)c(Cl)c1 C1(=O)C(C)(CSC)N1.c1(C=O)cnc(=N)[nH]c1.N(C)(CCSC)CC C(CCC(=O)NCC1C(C)(C)C1(C)C)(C(C)C)NC(C1C(C(=C)C)OCC1)=O c1(C(N(C(C)C(=O)NC2CC2)CC)=O)oc(CNC(c2ccc[nH]2)=O)cc1C c1(OCC)cc2c(cc1NC(N1CCN3CC(C)CC3C1)=O)OC(C)C2 C1(NCC(=O)NC(c2ncccn2)CC)CCOC(c2cccc(F)c2)C1 c1(OC)ccc(OC)c(C(O)C(C)NCCC(C)N2CCCC2)c1 N1(C(CN(C)CC)=O)CC(C)(C)OCC1CNC(=O)C(C)(F)C(C)(C)F NC(CCc1c[nH]nc1C(F)(F)F)C(=O)Nc1cnn(Cc2ccccc2)c1 C1(CNC(CCC)=O)CCN(C(=O)COCc2nc[nH]n2)C1(C)C c1(Nc2ncc(C(N(C3CCNC3)CC)=O)cn2)cccc([N+](=O)[O-])c1[N+](=O)[O-] c1(N2C(C3(N(C(=O)C=CC4CCCO4)C)CC3)CCC2)ncnc2c1CCCC2 CC1(C)CC(C(=O)NC2CC3(C2)CC3NC(c2ccc(C3CC3)o2)=O)CNC1=O Cc1[nH]c2c(C(=O)NCCN3CCC(N(C)C)CC3)cccc2c1C N1(C(C(CO)N(C)C)=O)CCC2C(C1)CN2C(c1ccn2nccc2n1)=O N1(C(C2(C(C)NC(C3CC3(C)C)=O)CC2)=O)CC2(C)COCC2(C)C1 CN1C(=O)C2CC1CCN2C(=O)C(N1CCCC1c1ccc(F)nc1)=O C1(CC(=O)NC(C(=O)NCC2CC(OC(C)(C)C)C2)C2CCCC2)COCCO1 Cc1cccc2cc(C(=O)NC3CC3NC(=O)C=Cc3ccc(Cl)s3)cnc12 N1(C(c2c(CC)c[nH]n2)=O)CCOC2CN(C(C3(C)CC=CCC3)=O)CC12 N1(C(C(n2c(C)ccn2)C)=O)CC(NC(c2cnc(C(N)=O)s2)=O)CC1CO c1(C(=O)NC2CCN(C(CCOC(C)C)=O)CC2CO)cc(Cl)c(N)cc1F Cc1sc(N)c(C(=O)NCC2CC(NC(=O)C(C)OCC(F)(F)F)C2)c1C C(C(=O)NCC(CO)NC(c1cnc(C)c(N)c1)=O)(C(C)(C)C)SC N1(C(CC2C(C)(C)C(O)C2)=O)CC2(C=C(C(=O)NOC3CCOCC3)CO2)C1 Cc1nc(NCc2ccsc2Cl)cc(N(C)Cc2ccc(C)s2)n1 C1(C(=O)NCCC(C)N2CCCC2)CC=CCN1C(=O)C=C(C1CC1)C1CC1 C(=O)(C1=CC2(CCOCC2)C1)N1CCC(CNC(CC(C)F)=O)C(F)(F)CC1 Cc1cc(C)nc(-c2cn(CC(=O)NCc3nnnn3C)nn2)n1 c1(COCC(=O)NCCC(=O)NC2N(C(C=C(C)Cl)=O)CC2)ccccc1C C1(CNC(C(C)OCC(F)(F)F)=O)CC(F)(CNC(C2CC(C3CC3)C2)=O)C1 N1(C(c2nccc(OC)c2)=O)CCC(CNC(c2cc(Br)n(C)n2)=O)C12CC2 Cn1ncc(C(=O)NC2(CNC(C3CC4C=CC3C4)=O)CC2)c1N CC1(C)CN(C(C2CCCC2(F)F)=O)CC(CNC(C2(C(N)=O)CC2)=O)O1 c1(OC)cc(C(=O)NCC2C=CCN2C(C2CCCOC2)=O)ccc1C(F)F C(=O)(CCC(=O)C1CCc2ccccc21)NC(c1cc(F)c(F)c(F)c1)CN CCC(CC(=O)N1CC(C2(NC(=O)CCNC(c3cccs3)=O)CC2)C1)C(C)C c1(CNC(=O)NC(C#C)(C)CC)nn(C)c(C)c1Br C(C(C)(C)CNC(=O)C(O)C1CCCC1)NC(C1C(F)(C(=O)OC)C1)=O C1(CNC(C=C(CC)C)=O)CCN(C(C2CC2C2(C)COC2)=O)CC1(F)F Cc1cccc(C(O)C(=O)NC(CO)CCCNC(=O)Cc2ccn(C)n2)c1 C1(C(N(C(C(C)C)C)C)=O)CC(C)CN(CCNC(=O)C(F)(F)F)C1 c1(OC)ccccc1NC(=O)CC1CCCN1c1ncc(C2CC2)cn1 C=C1CCC(C(=O)NC2CC(CCC(N3CCCC(N(C)C)C3)=O)C2)CC1 C1(CNC(CNC(C)=O)=O)CCN(C(c2c(C)nsc2C)=O)CC1CO c1(C(=O)OC)cocc1C(=O)NCCOCCNC(C1CCN1C1CCCC1)=O c1(C(N2CC(F)(CNC(CCOCCC)=O)C2)=O)ccc(C)c2c1NCCC2 C1(NC(C(C)=C(CC)C)=O)CCCC12CN(C(=O)C(c1c(F)cccc1F)C)C2 c1(C(=O)NCCC(=C)CNC(=O)CN(C)CCO)cc(S(N)(=O)=O)cs1 c1(C(=O)NC(CNC(C(C)SCCCC)=O)C(C)(C)C)cnc2cc(C)nn2c1 c1(C(C(=O)NCC2(C)CCCN2C(=O)COC2CCC2)O)ccc(C#N)cc1 c1(CNS(CC(C)C)(=O)=O)ccc(Cl)cc1Cl.c12ccccc1CC(=O)N2 c1(C(=O)NC(C(C)NC(c2nccc(CC)c2)=O)(C)C)nccc2ccn(C)c12 c1(CNC(c2ccccc2-c2ccccc2)CC)ccnc(OC)c1Cl N1(C(c2ncc(Cl)s2)C(=O)NCCSCc2ccncc2)CCC(CF)CC1 c1(C(=O)NCCN2CCN(C(=O)C(F)(F)CF)CC2)cc2cn[nH]c2cn1 c1(C(=O)NOC2CCOC2)n[nH]c(CC2CC(Cl)=NO2)c1Cl N1(C(C(C)CC2CCC2)C(=O)NC2CCCC2)CCc2cc(F)cc(Br)c2C1 c1(CNC(C2CC(F)(F)C2)(C#C)C)ccc(Br)c(Cl)c1 N1(C(c2scc(OC)c2)=O)CC(C(=O)O)OCC12CC2 c1(C(N2CC(NC(C(CSC)C)=O)CC(C)(C)C2)=O)ccc2c(O)ncnc2c1 CC(C)C(CC(=O)N1CCN(C)C(CO)C1)NC(c1cc(F)ccc1F)=O N1(C(C(=O)NCC(C)C)c2cc[nH]n2)CCC(=C(F)F)CC1 Cc1cnc(NC2CC(C#N)C2)c(S(=O)(=O)NC(CO)CCC(C)C)c1 N1(C(c2c(C)nn(CCO)c2)=O)CCC2(CC1)CCN(C(C1CC1C)=O)CC2 N1(C(CC(C)F)=O)CCC(C(=O)Nc2ccccc2CN2CCN(C)CC2)CC1 c1(C(=O)NC(CNC(=O)CC2OCCCO2)C2CC2)cccc(=O)o1 C1(C)(CCC(=O)OC)CCCN1C(=O)C(c1cccc(I)c1)N c1(CNC(c2cnc(-c3ccccc3)s2)=O)cccc(OCC2CCCO2)c1 C(C(CNC(=O)Cc1ccsc1)S(C)(=O)=O)NC(CC1C(C)(C)C(O)C1)=O CONC(=O)C(=O)NC1CC(N(C)C(c2cn(C)cc2C)=O)C1 n1(CC(=O)NCC(CCOC)NC(C2C3CCOCC23)=O)ncccc1=O c1(C(N2CCN(C(CC(=O)OC)=O)C(CC#N)C2)=O)c2c(nn1C)CCC2 c1(C(=O)NCC2C(C)CN(C(=O)CC(=O)NC3CC3)C2)ccc(O)c(C(N)=O)c1 c1(C(N2CC(C)(NC(C(CCC)C)=O)C2)=O)cc2cc(N)ccc2[nH]1 C(CNC(C1C(C)CCN1C(c1cccc(C)n1)=O)=O)(CC(C)C)OC C1(N(CCC(F)(F)F)C(c2c(C)nn[nH]2)=O)CCC2(CC1)CNC2 C(=O)(N=c1ccc(C2CCOCC2)n[nH]1)N(C)CCOc1ccncc1Cl C1(C(=O)NCCCNC(COC(CC)(C)C)=O)CCN(C2CC2)C1 c1(C(CCC)=O)ccc(NC(C2(S(C)(=O)=O)CC2)C)cc1 N1(C(=O)OC(C)(C)C)CCN(C2CCN(C(=O)OCc3cscc3Br)C2)CC1 c1(C2C(C(=O)NCC(C(C)C)NC(C3CN(C(N)=O)C3)=O)C2)c(F)cccc1Cl C1(CNC(C2(F)CCN(C(c3ccc(Cl)cn3)=O)C2)=O)CCC2(CC1)CC2 c1(OCC(CN(CCOC)CCN(C)C)O)cccc(Cl)c1 C(=O)(C1=CC2(CCOC2)C1)NCC(CCCC)NC(C1(CC)CCOC1)=O c1(NC)nc(C(=O)N(C)CC2CCCCN2C(C2CCSC2)=O)ccc1[N+](=O)[O-] c1(OC)cc(C(N2CC(NC(=O)C=C(C)C(C)(C)C)C(O)C2)=O)c(O)c(Cl)c1 c1(C(N2CC(NC(C(C(CC)C)O)=O)C2)=O)c(Br)sc2ccccc12 N1(c2nc(C)nc(N3CC4CCC(C3)O4)c2)C2CCC1CC(CC(F)F)C2 C1(C(N2CCC(C)C(F)(F)C2)=O)COCCC12CN(C(=O)C(C)(C)C#N)C2 c1(C(N2CCS(=O)(=O)CC2)C(=O)NCCCC)sc(=O)n(C)c1Cl C1(C)(C(=O)NCCC(C)C)CCN(Cc2ccccc2C(=O)O)C1 N1(C(c2ccc(C(C)=O)cc2)=O)CCN(C)C(CNC(=O)C(C)c2ncco2)C1 N1(C(CN(C2CCCOC2)CC)=O)CC(C)(C(=O)NOCCCF)C1 N1(C(C(C(C)C)OC)=O)CCC2(C)CN(C(C3CCC(C(C)(C)C)O3)=O)CC12 c1(OC)ccc2oc(C(N3CCC4CCC34CNC(C3(C)CC3)=O)=O)cc2c1 CC1CN(C(=O)CNC(C2CCC(C)(O)CC2)=O)CC(=O)N1 Cc1cn2c(n1)C(C(=O)N(CCCCNC(=O)CC1(O)CCCOC1)C)CCC2 c1(N2CC3CC(NC(c4cc(CCC)[nH]n4)=O)C3C2)cc(C)c(C#N)cn1 N1(C(C(C)=CC)=O)CCN(C(C2CCC(=O)N(C(C)C)C2)=O)C(CC(F)F)C1 c1(C(=O)NC2C3CN(C(C(COC(C)C)(C)C)=O)C2C3)cc2cccnc2[nH]1 c1(C(=O)NC2CN(C(Cc3cnc(C)s3)=O)CC(C)C2)cnc2ncccc2c1 c1(C(=O)NCC2N(C(C(C)(C)CO)=O)CC2)nc2nc(O)c3ccccc3n2n1 c1(C(N2CCN(C(C(c3cccc(F)c3)(C)O)=O)CC2)=O)nc2ccccc2s1 N1(C(c2cn(C)nc2N)=O)CCN(C(=O)CCS(N)(=O)=O)C(CO)C1 Cc1cc(C(=O)NC2CN(C(C3CC4CCCCC34)=O)CC2O)n2nccc2n1 C1(C(=O)NCCCN(C(CCc2cc(C)n(C)n2)=O)C)CCc2c(nnn2C)C1 CCCCS(=O)(=O)CC(=O)NC12CCCC(NC(c3ccns3)=O)(C1)C2 C1(F)(C(N(CCC(=O)NC(C)CCC2CCCO2)C)=O)CCCC1 Cc1nc(C)c(C(=O)NCC2COCCN2C(=O)Nc2ccccc2F)[nH]1 c1(NCC(C)(C)C(=O)N2CCCC2C2CCC(N)CC2)ncc(C(=O)OC)cc1Cl c1(NC2C(C)CN(C(=O)C(=O)N(C)C)C2)ccc(C(F)(F)F)cc1[N+](=O)[O-] CCC(O)C(C)(C)C(=O)NCC1C=CC(NC(=O)CC2CC(C)C2)C1 C12(NC(C(CSC)C)=O)CC3CC(C1)CC(NC(C1CCCCN1C)=O)(C3)C2 C1(C(N(C2COC(C)(C)C2)C)=O)CCN(C(C2CCCC(C#N)C2)=O)CC1(C)C C1(NC(CC)=O)CN(C(c2ccc(-c3sccc3C)s2)=O)C2(CCCOC2)C1 C1(C(C(=O)NC2CCN(C(C3(C)CCOCC3)=O)C2)(C)C)CCS(=O)(=O)CC1 Cc1cc(C(=O)NCC2CCCN2C(c2cnn[nH]2)=O)n(C2CC2)n1 C1(C(=O)NCCCN(C(C2(C=C)CCC2)=O)C)CNC(=O)CC1C N1(C(c2cc(C(=O)OC)no2)=O)CCCC2(CC(NC(=O)C(F)=C(C)C)CO2)C1 CCC(F)(C(=O)OC)C(=O)N1CC2C(N(C)C(c3cc(F)cnc3O)=O)C2C1 Cc1cnc(C(=O)NC(CCNC(C2(CF)CC2)=O)C(C)C)c(O)c1 C(c1ccc(F)cc1)=CC(=O)NCC(C)NC(=O)C=Cc1ccsc1 c1(CC)oc(C)cc1C(=O)NC(CO)C(=O)N(C1CC2CC2C1)C Cc1nc(C(N2CCSCC2CCNC(=O)C(N2CCCCC2)C)=O)c(C)s1 c1(C(N2CCN(C3CN(C(c4nc(Cl)sc4Cl)=O)C3)CC2)=O)ccc(O)nn1 c1(C(N2CCC(c3n(C)ncc3)C2)C(=O)NCC2CCOC2)ccc(Cl)cc1Cl C1(CNC(Cc2cn(CC)nc2)=O)CN(C(=O)CC2COCC2O)CC(C)(C)C1 C1(OC)CN(C(=O)CCCSC)CC1NC(C1(C(C)C)CNC(=O)C1)=O N1(C(CS(CC)(=O)=O)=O)CC2(C1)CN(C(=O)C(C)Cc1ccncc1)CC2CO N1(C(C2CN(C(C)=O)C2)=O)CC2(C(N3CCSC(C)(C)C3)=O)CC1CO2 C1(SC(C)(C)C)CCN(C(=NCC=CBr)NC2CC2)C1 Cc1ncnc(C(=O)NCCC2CCCN(C(=O)CC(C)F)CC2)c1C c1(C(=O)NCc2ncc(C)c(C)c2)nccc2c(Cl)cccc12 c1(C(=O)NC(c2ccncc2)CC)cccnc1CNC(c1coc(C)c1)=O C1(O)(CCNC(CCOCCOC)=O)CCCN(C(c2cnn3c2SCC3)=O)C1 c1(C(N(CC(C)NC(c2c(C)cns2)=O)C)=O)nccnc1N C(c1ccoc1)=CC(=O)NCCN(CCC)C(C1CC1OCC)=O Cc1oc(CNC(=O)CC2C=NN(C)C2=O)nc1C(N1CCC(C(F)F)C1)=O N1(C(CC)=O)CCC2(CCN(C(c3cccc(N(C)C)c3)=O)C2)C1 C1(N(C(C23C(CN(C(C(CC)N(C)C)=O)C2)C3)=O)C)CN2CCC1CC2 c1(N2CCC(CN(C(CC3(COC)CC3)=O)C)CC2)ncnc2cccnc12 Cc1cc(C(=O)NC2CCC(C)(CNC(=O)CC3C=CCCC3)CC2)ccc1Cl Cc1cnc(C(=O)N(C)CCNC(c2csc(-c3ccccc3)n2)=O)cc1Cl C(=O)(CC(C)C(F)F)NCC(=O)NCC(=O)NC1(CC)CCOCC1 c1(C(=O)O)cc(S(=O)(=O)N(C2CCCCCCC2)c2ccccc2)ccn1 CCCC(CC(C)C)C(=O)N1CCC(CNC(=O)C(F)OC)C(C)C1 C1(NC(CC(C)Cc2cccc(F)c2)=O)CCN(C(=O)C(F)(F)CO)CC(O)C1 C(=O)(CCCCC(N)=O)NC(CC)CNC(=O)C=CC(c1ccccc1)=O C12(C(=O)NCC(c3ccccc3)CNC(CCOCC)=O)CC(F)C1C2 CCCCCC(O)C(=O)NC1(COC)CCCN(C(c2nccc(C)c2F)=O)C1 c1(OC(c2nc(Cc3ncccc3F)no2)C)cc(F)ccc1Br c1(C(N(C2C(NC(C(C)S(N)(=O)=O)=O)CCCC2)C)=O)cnc2c(c1)CCCO2 C=CCC(C)(CC)C(=O)NC1C2CN(C(C3(OC)CCS(=O)(=O)C3)=O)CC12 C(CCC(=O)NO)NC(CC1CCN(C(C2N(C(C)C)CCC2)=O)C1)=O N1(C(C(C)c2ccco2)=O)CCCCC1CNC(=O)CNC(=O)C1CC1 N1(C(CNC(CNC(C)=O)=O)=O)CCC(OC(C)C)CC1.C1(=O)C(C)(CO)N1 CC1CCCN(C(=O)Nc2cccc(I)n2)C1CO c1(C(=O)N)conc1C1CC1.CC1C(=O)NC(C)CCN1C.N(C)C Cc1ccc([N+](=O)[O-])c(C(N2CC(NC(C3(O)CC3(C)C)=O)C(O)C2)=O)c1 c1(C(=O)NCC(CNC(CN(C)C2CC2)=O)F)cc2cccc(Br)c2s1 C1(NC(c2ncn(CC)n2)=O)CC2CC(NC(=O)Cn3ncn(C)c3=O)CC12 C(=O)(C(C)C(C)S(C)(=O)=O)N(C(C)C)CCN(C)C(C1(O)CCOCC1)=O c1(C(=O)OCC)sc2nc(CC)nc(NC3CCCc4nc(C)sc43)c2c1C CC1(C)NC(=O)N(CC(=O)NCC2CC3CC(C2)N(c2ccncn2)C3)C1=O C1(C(N2CC(CC(CNC(C(COC)O)=O)(C)C)C2)=O)CC2(CC2)CN1C N1(C(C(CCC=C)NC(=O)COC2(C)CCCC2)=O)CCC2(CCCC2)CC1 C1(N(C(=O)CC2(C)CC2)C)CN(C(c2ccccc2OCC(F)(F)F)=O)CC1F C1(OCC)CN(C(=O)C(c2ccccn2)O)CC1NC(=O)CSC1CCOCC1 c1(OCC)nc(C(=O)NC(C)CNC(c2nc(O)sc2C)=O)cc2ccccc12 C1(C(=O)NC(COCC)C(=O)NCCc2ncc(C)cn2)CC(C)(C)CN1C c1(NC(CC)CSC)[nH]c(=NCC(C)(CC)OC)nc2c1ncn2CC Cn1nc(C(=O)NCC2CN(C(=O)C=C3CCCCC3)C3CC23)cc1C(F)F C1(C)(C(=O)NCC2OCCN(C(C3C(CCC)CCC3)=O)C2)CC(OC)CN1C N1(C(CCOCC#C)=O)CC(C(=O)N(C)CC2CCCC2(C)C)C(C)C1 c1(OC)cc(C(=O)NCCC2CCC(NC(=O)Cc3cccs3)C2)cc(Cl)c1O N1(C(c2c(C)ccnn2)=O)CC(NC(c2c(C3CCC3)cnn2C)=O)CC(C)C1 n1(CC)cnc2[nH]c(=NCC3(C)CCOCC3)[nH]c(=NC(C)C(C)CO)c12 CC1CCCC(CC(N2CCC(OCCNC(C3(c4cccs4)CC3)=O)C2)=O)C1 C12(C(=O)NC3CCC(C)CC3)C3CC1C1C(C(N4CCOC(C)(CO)C4)=O)C3C21 Cc1[nH]cc(C(=O)NCCCC2CCCCN2C(=O)CCC(C)(C)F)c(=O)c1Cl c1(C(=O)NC(CN(C(CC(C(CC)C)O)=O)C)(C)C)cccc2c1COCCN2 CC1CN(C(=O)CN(C)C2CC2)CC(C)N(C(c2cc3c(s2)CC(C)(C)C3)=O)C1 C1(c2nnnn2C)(NCC2(COCC)CCCC2)COCCOC1 N1(C(C(C)CF)=O)CC(NC(c2ccc(-c3cccs3)o2)=O)C(O)C1 C1(C(N(CC=C)CCOC)=O)CCCN(C(=O)COC)C1 N1(C(CCC(C)C)=O)CCC2(CCCN(C(=O)CCCn3cccc3)C2)C1 n1(CC(N2C(CO)CC(NC(C(=O)NCC)=O)C2)=O)ccc(=O)n(C)c1=O.C1CC1 c1(OC)cc(C(=O)NCC(O)CCNC(C2OCC2(C)C)=O)cc(Cl)c1 c1(C(N2CCn3c(C)cnc3C2)=O)ccnc2cc(Cl)ccc12 Cc1cc(C(=O)NCCN(C(=O)CC(C)c2ccccc2)C)nn1C N1(C(N2C(c3nc4ccc(C)cc4[nH]3)CCC2)=O)CC(C2CC(=O)NC2=O)C1 Nc1cc(F)c(F)cc1C(N1C2CCC1CC(NC(C1CC=CCC1)=O)C2)=O N1(C(=O)Cc2ccnc(O)c2)CCC2CCN(C(=O)COC3CC(F)(F)C3)C2C1 c1(CNC(C=CC(C)(C)SC)=O)cnn(C)c1C(N1CC(CO)C1)=O C#Cc1ccc(NC(=O)CCN(CCO)C(c2cccc(OC)c2OC)=O)cn1 c1(COC)ccoc1C(N1CCCC1C1CCN(C(=O)CCC2(O)CCC2)C1)=O C1(OC)CC2CC(C(=O)NCCC3(C)CCN(C(c4scnc4C)=O)CC3)CC12 Cc1ccc(C(=O)N(C)CC2CN(C(=O)C(F)C3CCC3)CC23CC3)c(N)c1 N1(C(C2(CC#C)CCCC2)=O)CCC(NC(=O)C(c2cnn(C)c2)O)CC(O)C1 C(CCC(C(=O)NCC(O)CCC1CC1)NC(c1cc(F)ccc1O)=O)OC C(C1CCCCc2ccccc21)SCc1c(OC)nc(C(C)C)cc1 C#CC1(O)CCCN(C(C2CN(C(c3cc(C(C)=O)on3)=O)CC2OC)=O)C1 N1(C(C(CC=C)CC)=O)CCN(C(c2csc(C(C)C)n2)=O)C2CCC12 c1(-n2cc(C(C)NC(C3CCOC3)=O)nn2)cccc(CC=CCO)c1 C(CN=c1[nH]c2c(c(=NC3CCCC3)[nH]1)COC2)(c1ccc(C)cc1)N1CCCC1 c1(CC(NNC(=O)NCc2ccc(OCC)c(Br)c2)=O)nc2ccc(C)cc2[nH]1 C(=O)(C(O)C(C)(C)C)NCC1(CN(C(=O)C(c2ccccc2)O)C)CC1 C1(CNC(c2ccn(CC(=O)OC(C)(C)C)n2)=O)C2CN(CC=CCO)CC12 C1(NC(c2cc(C)n(C)c2)=O)CCN(C(=O)CCc2cc(Cl)no2)CC1C(C)C N1(C(c2ncn(CC)n2)=O)CC(NC(c2cnncc2O)=O)C(O)C1 Cn1cnc(N2CCC(CCNC(c3cccc(F)n3)=O)C2)c(Br)c1=O c1(C(N2CCCC(NC(C3CCSC3)=O)C2)=O)c(Cl)nc2cc(Cl)ccn12 O=C(C1=CCOC1)NCCCOCCCNC(c1cscn1)=O C1(CNC(c2nc(Cl)cs2)=O)CC12CCN(C(=O)CCc1nc[nH]n1)CC2 c1(OC)c(C(=O)NC(C2(O)CCN(C(=O)C(F)C3CCC3)CC2)C)ccnc1F C1(NC(=O)Cc2ccccc2F)CCCC2CN(C(=O)CCc3nc[nH]n3)CC12 c1(CNC(C(C2CCC2)NC(COCCC)=O)=O)ccc(CC)o1 C(=O)(C1=CCC(NC(c2csc(=N)[nH]2)=O)C1)NCC(CC(=O)NC)C N1(C(C2(CC)CC2)=O)CC2CN(C(C3CCC=CCC3)=O)CC(C1)O2 C1(OC)CN(C(=O)CC2CCOC2)CCC1NC(C1(C)CCC(C)(C)C1)=O N1(C(COc2cccc(C)c2)=O)CCCCC(CNC(=O)CC2CCCC2C)C1 N1(C(C2CC(C)(O)C2)=O)CC2CC(C1)N(C(=O)CCC1CC1CC1CC1)C2 CC1CN2CCN1CC2C(=O)N(CCCNC(C12CCC(CC1)OC2)=O)C1CC1 N1(C(=O)Cc2cc[nH]c2)CC2CCN(C(c3sccc3Cl)=O)CC2C1 c1(OC)c(C(=O)NC2CCC(NC(=O)C=Cc3ccncc3)C2)cc(F)cc1F C1(C(=O)NCC(C)(Cn2cccn2)NC(CNS(C)(=O)=O)=O)CCS(=O)(=O)N1 c1(NC(CC2(OC)CN(C(=O)C(C)(C)C(C)O)C2)=O)ccc(C)cc1C C#Cc1cccc(OCC(=O)NC2CC3CC2N(C(=O)CC2CC4(CC4)C2)C3)c1 C(=O)(CC(O)(C(F)(F)F)c1ncco1)NCC=CCNC(c1c(C)cncc1)=O C(=O)(NNc1cccc2c1OC(F)(F)O2)c1nc(-c2cn(C)nc2)sc1 N1(C(C2CCC(=C)CC2)=O)CC=C(CC(=O)NC2CSC2)CC1 c1(-n2cc(CC3(CO)CCN(C(C(C)=O)=O)C3)nn2)ccc(F)cc1Cl CC(C)CC(C)(C)C(=O)NCCn1cnc(C(N2CCOCCC2C2CC2)=O)c1 c1(C(N)=O)ccc(C(=O)NC2CCCC2NC(C2CC3CC3C2)=O)cc1 N1(C(C(C)Oc2ccc(F)cc2F)=O)CC2=C(C1)CN(C(C1(C#N)CCC1)=O)C2 C(=O)(C1=COc2ccccc2O1)NCCCCC(C)NC(=O)C=CC(=O)NC1CC1 C(=O)(C(C)CC(=O)NCC1(C(=O)NCCC(C)N2CCCC2)CC=CC1)OC O=C1NCCOc2ccc(CNCC3CCCN(Cc4ccccc4)C3)cc21 Cc1ccc(C(=O)NC2CC(O)CN(C(c3ccc(O)cc3)=O)C2)cc1C c1(NC(C(C)(C)C)C2CCCCC2)cc(Cl)cc(Br)c1 C1(NC(CC2(N(C)C)CCC2)=O)CCN(C(=O)CC2CCC=CCC2)CC1 c1(OCC)nc(Cl)ccc1C(N1CCCC(CNC(C23C=CC(CC2)C3)=O)C1)=O c1(CNC(CC2N(C(C3(C(N)=O)CCC3)=O)CC2)=O)ncccc1O N1(C(CCC2C(C)C2)=O)CCC(C2CCCCN2C(n2cc(C#N)cn2)=O)CC1 Cc1csc2cc(C(=O)NC3CC3CNC(=O)C(N)=O)[nH]c12 C(=O)(C(CCC(N)=O)n1cc(CO)nn1)N1CCC(n2c(C(C)N(C)C)cnn2)CC1 c1(NC(C(=O)Nc2cccc(-c3ccncc3)c2)=O)ccc2c(c1)CCNCC2 N1(C(CN(C(CC2ON=C(C)C2)=O)C)=O)CCN(C(=O)C=CCF)CC1 N1(C(COCCC=C)=O)CC2CN(C(c3cnc(NC)c(Cl)c3)=O)CC2(C)C1 C(=O)(CC(C)C(C)(C)NC(c1sc(C)cc1C)=O)NC1CC(C)(CC)C1 C=CC1(O)CC(NC(=O)NC2CCCCC2NC(=O)OC(C)(C)C)C1 Cc1ccc(C(=O)N(C2CCCC(N(C(=O)COCC(F)F)C)C2)C)nn1 c1(C(=O)NCCCN(C(=O)C(C)C2CCC2)CC)cc2ccncc2s1 N1(C(N2CCC(OCC)C(C)C2)=O)CCCc2ccc(C(=O)OC)cc2C1 Cc1ncc(CC(=O)NC2(CNC(c3csc(-c4ncccn4)n3)=O)CC2)o1 C1(CC(=O)OC)CCCN1C(C1C=CC(NC(C2CCC(=O)N2)=O)C1)=O Cc1noc(C2CC2)c1C(=O)NCC1(C)CCCN1C(=O)CC1(C)CCCCC1 c1(C(N2CC(NC(c3c(C)sc(CC(C)C)n3)=O)C2)=O)sccc1S(N)(=O)=O N1(C(COC)=O)CCC(CON(C2C3CCC23)C)CC1 N(C(=NCc1ccc(F)cc1)N1CCC(F)C1)CC1N(CC)CCC1 C1(CC(=O)NC(C(C)C)CCN(C(=O)C=CCO)C)NC(=O)CNC1=O N1(C(C(C)n2cccc2)=O)CC=CC1CNC(c1ccsc1C(F)(F)F)=O c1(C(=O)NCCC2(CNC(C3CC4CCC4C3)=O)CC2)ccnc2ccsc12 CC1CCCn2cc(C(N3CC(O)(CNC(=O)C(c4ccccc4)O)C3)=O)nc21 C1(C(N2CCC(Nc3nc(OC)cc(OC)n3)C2)=O)CCC2(CC1)CNC(=O)C2 CC(C)(CS(C)(=O)=O)C(=O)NC1CN(C(=O)CCCCC2CC2)C2(CCOC2)C1 C1(NC(C2N(CC)CCC2)=O)CCCCN(C(c2cc3ccccc3[nH]2)=O)CC1 CC1CCC(O)(C(=O)NC2COCCN(C(C34CC(C3)C4)=O)C2)CC1 Cc1ccc(-n2nnc(C(=O)NCCC3COCCN3C(=O)C(C)C)c2C)cc1 c1(C(=O)OCCC2C(C)(C)CCO2)ccc2c(=O)[nH]ccc2c1 Cc1noc2cc(C(N3CC4CC(NC(=O)CC(C)(F)F)CC4C3)=O)ccc12 C1(CNC(C(C)(C)N(CC)CC2CC2)=O)CN(C(=O)CCOC(C)C)CC1(F)F c1(C(=O)NC2C(C)N(Cc3c(Cl)cccc3Cl)CCC2)cnc2cnccc2c1 c1(C(=O)NC2C3OCC(NC(C4CCC(C)O4)=O)(C3)C2)cccc(O)c1[N+](=O)[O-] N1(C(c2n(CC#C)ccc2)=O)CC(C)C(C2CN(C(=O)CC3(C)CC3(F)Cl)C2)C1 N1(C(COC(CC)C)=O)CCC(NC(=O)C=Cc2ccc(C)o2)C12CCC2 c1(C(N(C)CC2(NC(C=C(CC)C)=O)CC2)=O)nccc(Cl)c1C N1(CC=CCNC(=O)Nc2ccc(C(C)C)cc2)CC2C3C=CC(CC3)C2C1 c1(CC)nnc2n1CCCC2C(=O)NCC(C)(C)OCCNC(=O)CC1(C)CC1 C(=O)(C1=COCCO1)N1C(CNC(CC2CC(OCC)C2)=O)C=CC1 C(c1ccc(=N)[nH]c1C)=CC(=O)NCC1C(NC(CCSCC)=O)CC1 C(=O)(C1=CNC2=NCCCC2=C1)NCCN(C1CCCCCC1)C(C(CC)C)=O C1(C(=O)NC(C)CC(N)=O)CC2CCC(C1)N2C(C1CC1(C)C(F)F)=O C(=O)(C1=CCCCC1)N1C(CNC(c2csc(O)n2)=O)CCCC1 N1(C(=O)OC(C)(C)C)CCC(C(=O)NCC2CC(=C3CC3)C2)CC1(C)C c1(CC(=O)N(CC(CNC(CC2CC(C)C2)=O)O)C)cccc(C(F)(F)F)n1 C(CN=c1[nH]c(N2CCC(S(=O)(=O)C(C)C)C2)nc2c1CCCC2)SC C1(C(=O)NCCCCC(C)NC(CC(CC)CC)=O)CCCCN(C)C1=O C1(C)(N(CCOC(C)C)C)CCCN(C(=O)CCNc2ccccc2)C1 N1(C(C2OCCN(CC)C2)=O)CCCCC(NC(c2ncoc2C(C)(C)C)=O)C1 CC1(C)C2CCC1(C(=O)NC13CC(NC(c4cc(Cl)ns4)=O)(C1)C3)CC2 CC1=C(F)CN(C(C2CCC(n3cc(-c4csc(C)c4)nn3)C2)=O)CC1 C1(CCC)CN(C(=O)CC(C)(C)OC)CCN1C(c1ccnc(SC)c1)=O C1(C(=O)NCC(=O)OCC)CCN(C(=O)Cn2nnnc2C)C1 Cn1cnc(CCNC(C(CCCO)c2ccccc2)=O)c1 C1(C(N2C(C(C)NC(=O)CCC3CCCN3C)CCC2)=O)CC12CC(C)(C)C2 Cn1cccc1C(=O)C(=O)NC1CC(CNC(c2ccnn2C2CC2(F)F)=O)C1 CON(CCO)C(=O)c1cc(CNC(c2c(O)cccc2F)=O)[nH]n1 C(=O)(CC(C)C(=O)NC(C(=O)Nc1cnn(CCF)c1)C1(C)CC1)OC N1(C(CN2CC(C)(C)C2)=O)CC2(CCC2)CC1CNC(C1CC2CCC(C1)N2C)=O c1(CN(C)C(c2cc(C(N)=O)co2)=O)cccc(C(=O)NC2CCCCCC2)n1 CC(C)(C)CN=C(N(C)C1CC1)N1CCn2c(COc3ccncc3)nnc2C1 c1(C(N2C(C)C(NC(=O)CCC3CCC3)CCC2)=O)ccnc2ccnn12 C(=O)(C(CC)(CC)OC)N(C(CC(=O)NC1CC(CC)OCC1)CC)C CCC(C)(C)CCCC(=O)NCCC(C(N1CCC12CCCSC2)=O)OC C1(OC2CCCN(CCC)C2)CC2(CCN1C(=O)C(CC1CCC1)OC)CC2 O=C(CCC(=O)c1ccc(F)cc1)NCc1ccnc(C(=O)NC2C(CO)C2)c1 Nc1cc(F)c(C(=O)NC(CNC(=O)CCC2CC2)CO)cc1F c1(C2(NC(C(CCC)OC)=O)CC2)cnc2ncccc2c1 C1(N(C(=O)C(c2cccnc2)OC)CC)CCCN(C(C2CC(F)(F)C2)=O)C1 c1(C(N(C2CCN(C(=O)CN3C(=O)CNC3=O)CC2)CC)=O)ncc(F)cc1F C1(CNC(c2n(CCCC)nnn2)(COC)CC)CCC(S(C)(=O)=O)CC1 C(CCOCC)(C(=O)NCc1occc1C)NC(CC1CC(=C)C1)=O C1(NC(CC(C=C)CC)=O)CN(C(c2cc(CC)[nH]n2)=O)CCC12CCC2 C1(CNC(c2cc(C(F)F)no2)=O)CN(C(=O)CCc2cnc(O)[nH]2)CC1O CCC(O)C(C)C(=O)NC1CCC(NC(=O)CCCc2csc(=N)[nH]2)CC1 C=CCC(CNC(c1sccc1F)=O)NC(=O)C(n1ccc(C(F)(F)F)n1)C N1(C(CCSCC)=O)CCC(F)C(NC(C2CC23CCC3)=O)C1 N1(C(CC2(C=C)CN(C(C(C)OCC#C)=O)C2)=O)CCC(C)CC(C)C1 CC1(C)CC(NC(=O)C=C2CCC2)CN(c2ccncc2C#N)C1 c1(C(=O)NCC23CC2CN(C(=O)CCn2ccnn2)C3)cncc2nc(O)[nH]c12 n1(CC)ncc(C(=O)NC2CCOCC2NC(=O)COC2CC2)c1C C(=O)(C1=CC2CCCCCC12)N1CC2CCC(NC(=O)CCCCF)CC2C1 C(=O)(C(C)(O)C(C)C)N(C1CCCN(C(=O)Cn2cc(C3CC3)nn2)C1)CC c1(C(=O)NC(CCN(C(Cc2cn(CC)nc2)=O)C)C)ccncc1C(F)F c1(C(N(CC(C)NC(c2cccc(Cl)c2F)=O)C)=O)cccc(Cl)c1O N1(C(c2c(C)coc2)=O)CCC2C1CCCN2C(c1nnn(C(C)C)c1C)=O N1(C(C(C)(C)C2CC2)=O)CCN(C(C2C=CCC2)=O)C(C2CC2)C1 c1(C(=O)NCCCN(C(C(CCCC#C)C)=O)C)ccc2ncc(Br)n2c1 c1(C(=O)NC2CCCC2CC(N2CCC(C(F)F)CC2)=O)cnc2n1CCC2 Cc1ccc(C(=O)NCC2CN(C(=O)CCC(F)(F)F)CCO2)cc1Cl c1(C2c3n(nnn3)CCCCN2)cccc(NC)c1F.C1(C)(OCC)CCC1.OC N1(C(C2CN(CC(C)C)C2)=O)CCCC(CN(C(=O)CCN(S(C)(=O)=O)C)C)C1 C(=O)(CCC(=O)c1ccc(Cl)s1)NC(CNC(c1nc(COC)sc1)=O)(C)CO CC(c1ccccc1F)=CC(=O)NC(C)(C)C(C)NC(c1c[nH]cc1Br)=O c1(C(N2CC(NC(=O)CN3CSCC3=O)C(F)C2)=O)oc2ccccc2c1Cl C12(NC(Cc3c(CSCC)cccc3)=O)CCCC1N(C(c1cocn1)=O)CC2 c1(C(=O)NCC(CO)NC(CCC(C)CN(C)C)=O)c[nH]c2cccc(C#N)c12 C1(C(=O)NCC(C)(F)F)CC12CCN(C(=O)C=Cc1cc[nH]n1)C2 c1(C(=O)NCC(C)N(C(C(CCC)OC)=O)C)cccc(C2=CCOCC2)c1 Cc1cn2nc(C(=O)NC3(CO)CCN(C(=O)CC4CCOC4)C3)cc2c(=O)[nH]1 C1(C(=O)NCC(CCC)(C)C)CC(C)(C)CCN1C(c1ccc(F)cc1F)=O c1(C(=O)NC2(CNC(c3ccc(O)nc3Cl)=O)CCC2)ccnc2ncnn12 Cn1ncnc1CNC(c1cn(CCNC(C2CCCC2)=O)cn1)=O C1(C)(CNC(CC2(CSC)CC2)=O)CCCN1C(=O)Cc1ccc(C)nc1 CCC(C)(CC)C(=O)NC(C)C(C)C(=O)Nc1cnc(Cl)nc1C c1(CC(=O)NCC2(NC(=O)CCc3cnc[nH]3)CCOC2)ccc(F)c(F)c1 N(C(=NCCc1ccn(CC)n1)N1CCC(c2ccccc2F)C1)C(CC)C c1(C(=O)NCCC2COCCN2C(C2CCCCO2)=O)c[nH]nc1[N+](=O)[O-] c1(OC)cc(F)c(CN(CC(c2ccoc2C)=O)C)c(F)c1 C=CCCC(C)(C)C(=O)N1CC(OCCNC(=O)CSCc2cccs2)C1 CCCCCCn1cc(CN(C2(C)CCC2)CC)nn1 Cc1nc(C(=O)NCC(C)(CO)NC(c2cscc2Cl)=O)nn1-c1ccccc1 c1(OC)ccc(CC(O)C(=O)NC(CO)C(C)NC(=O)Cc2c[nH]nc2O)cc1 C(N=c1[nH]cnc2cc(F)ccc12)C12C(CN(C(c3nccc(C)c3)=O)C1)C2 N1(C(CN(C(C)C)C(c2ccnc(CO)c2)=O)=O)CCCCC1CO N1(C(c2c(C)cccn2)=O)C2CCC1CC(C(N1CC(C)C1(C)C)=O)C2 c1(CC)ccc(CC(=O)NCC2(O)CC(NC(C3COC(=O)C3)=O)C2)cc1 N1(C(c2c(C)nc(C(C)C)o2)=O)CCN(C)CC1CNC(C1CC12CC2)=O C#Cc1ccc(F)cc1OC(C1CCCC1NC(=O)OC(C)(C)C)=O N1(C(C2CN(CC)C2)=O)CCCC(CN2CCN(C(=O)CSS(C)(=O)=O)CC2)C1 c1(CC)cc(C(N2CC3CC2C3NC(=O)CC2(CC(=O)OC)CC2)=O)c(C)o1 N1(C(C(C2CCCC2)NC(CC)=O)=O)CCCCC1CNC(=O)CN(C)C1CC1 c1(CC(=O)NC(C(C)(C)C)CNC(c2cncc(F)n2)=O)ccc(C#N)cc1F C1(NC(=O)CC(O)c2ccccc2)(CNC(=O)C(O)C2CC2)CCCCC1 CC1(C)CC(NC(=O)C=Cc2cn[nH]c2)CN(C(c2cnn(C3CCC3)c2)=O)C1 CCC(CC)(CO)C(=O)N(CC(C)NC(C1(C)CC(C(=O)OC(C)(C)C)C1)=O)C C1(C(N(CC(=C)C)Cc2cscn2)=O)CC12CCN(Cc1ccccn1)CC2 CC(C)CC(CNC(=O)C(CC1CC1)CC1CC1)NC(=O)Cc1ccccc1Cl c1(NC(=O)NC(C)CO)onc2ccccc12 N1(C(c2scc(C(N)=O)c2)=O)CCN(C(C2CC2CF)=O)C(c2ccccn2)C1 c1(CNC(C2C(C3C(C)C3)C2)=O)cccc2c1CCN(c1nnco1)C2 N1(C(C(C)CC2CC2)=O)CC(C(N2CCC(c3cnn[nH]3)C2)=O)CC(C)(C)C1 C1(NC(C(CC)OCC)=O)CC2CN(C(c3ncc(Br)cc3O)=O)CC12 Cn1cc(Cl)cc1C(=O)NCC1CCCCC1NC(c1cnccc1Cl)=O c1(C(=O)NCC2CC(CNC(c3cn[nH]c3)=O)CO2)cnc(O)cc1F C1(C(=O)NC(CC=C)CNC(=O)Cn2ncnn2)CCC2(CCC2)C1 C1(C(N2C(CC)CC(C)C2)=O)CCC2(CC2)N1C(c1cc[nH]c1)=O n1(CCC)nnnc1C(C1CC1C1CC1)NCCNC(=O)C(C)C C12(CC(=O)N(CC(C)NC(=O)C(C)CC3CCCC3)CC)CCC(CC1)OC2 C12(C(=O)NC3C(NC(C4(OC)CCC4)=O)CCCC3)CCCN(CC1)S2(=O)=O C1(C(N(C)CC2CN(C(c3c(O)cc(C)nn3)=O)C2)=O)CCc2nnc(O)n2C1 C(C(F)(F)C(=O)N1CC(NC(c2cc(=O)cc[nH]2)=O)C(CC2CC2)C1)OC CCC(CC)C(F)C(=O)N1CCCC(F)(C(=O)NCC(n2cccn2)C)C1 C1(C2CCC2)(C(N(CCN(C(=O)C=CI)C(C)C)C)=O)CCC1 C1(CCC)CN(CCC2CCOC2)CCO1 C(=O)(CC(C)(O)C(F)(F)F)N1C(C)CC(NC(CC2(C=C)CCC2)=O)C1 N1(C(C(C)OCC=C)=O)CC(=O)NC(=O)C1 N1(C(C=NOC)=O)CCC(C)N(C(=O)CCOc2ccc(Cl)cc2F)CC1 Cc1cc(C(=O)NC2CCC(C)N(C(c3cc(C#N)c[nH]3)=O)C2)cnc1C C1(NC(c2cc(C)nc(C)n2)=O)CCC2CC1CN2C(c1nc(Cl)ccc1N)=O N1(C(c2n(C)nc(C(F)F)c2)=O)CC(NC(c2ccc(F)s2)=O)C2(CC2)C1 C(=O)(N=c1ccc(C(C)(C)C#N)n[nH]1)N1C2(CCC(C)C2)C1=O.C1(OC)CC1 CCCCC(C)(C)NC(C1CC(C)CN1C(=O)C(F)CC1CCOC1)=O C1(C(=O)Nc2ccc(CC(=O)OC)cc2)CC2(CCOCC2)CO1 c1(OCC)ccc(CCC(=O)NC(CNC(C2CCN(C)CC2)=O)C2CC2)cc1 CCN=c1ccc(C(N2CCCCC(NC(=O)C(C)OC3CCCC3)C2)=O)c[nH]1 N(C(=NC(C)c1nncn1C)NCC1CC1(F)F)C(CC)CC Cc1nn(C(C)C)cc1COC(c1ccc(CC(=O)N(C)C)cc1)=O c1(C(=O)NC2(CNC(CCC)=O)CCCC2)cnncc1C C(N=c1[nH]c(=NC2CC2C(C)(C)C)c2cc(F)cc(F)c2[nH]1)c1cncc(C)c1 c1(CN2C(CN(C)C(C3C=CCCC3C(=O)O)=O)CCCC2)ccc(Br)c(O)n1 N1(C(C(=O)NCC2(OC)CCCCCC2)=O)CCC(C)CC(C)C1 n1(-c2scc(CC(=O)NCCN(C3CCO3)CCC)n2)c(C)ccc1C C(=O)(C1CCc2nccn21)NC(C)C(C)C(=O)NCC1CN(C(N)=O)C1 C1(CC(N2C(C(C)O)CC2)=O)CN(C(=O)CCCn2cccc2)CCO1 Cc1nccnc1C(=O)NC(C)CCN(C(=O)Cc1cncs1)C C(C(C)(C)C#CC(=O)NCc1csc(C)n1)NC(C(C)=CCC)=O CC1CN(C(C2(C#N)CC3(CC3)C2)=O)CCC1NC(C1(C2CC2)CCC1)=O CC1(C(=O)NCC#CCNC)CC12CCN(C(c1cc(C3CC3)[nH]n1)=O)CC2 c1(CC)c(NC(N2CCCC2Cn2ccnc2C)=O)cnn1-c1ccccn1 N1(C(CC=CC=C)=O)CC(CC(N2CCC(C)(F)C2)=O)C2(CC2)C1 c1(OC)cc(C(N2CCOC3CC23)=O)c(NC(c2cccc(O)c2F)=O)cn1 C1(C#N)(C(=O)NC(C)CCCl)CC2CCC1CC2 N#Cc1c([N+](=O)[O-])cccc1S(=O)(=O)NC(CCCO)C(=O)O N1(C(=O)NC2CCC(C)C2)CCN2CCCC2C1 C1(C(NOCC=C)=O)CN(C(=O)COCC2CCC2)CC12CC2 CCCC(CC1CCCCC1)C(=O)NCC(C)(C)OCCNC(c1ccsc1)=O c1(SC)cccc(NC(=O)Cc2ccc(C3CCNCC3)cc2)c1 Cc1ccoc1CC(=O)N(C)CC1(CNC(=O)CC2COC(=O)N2)CC1 c1(C(N2C(C)(CNC(C3C(CC)OCC3)=O)CCC2)=O)cc(O)cc(O)c1 C=CC(CC(=O)NCCCNC(c1sc(F)cc1Br)=O)c1ccccc1 C1(NC(C2N(C(COCCCOC)=O)CC=CC2)=O)CC(C)(C)OC1=O Cc1csc(=O)n1CC(=O)NC1COCC1N1CCN(C(=O)CCC2CC2)CC1 c1(OCCC(=O)NC(C)C(C)OC(C)(C)C)cccc(Br)c1 N1(C(CC2N(CC)CCC2)=O)CCC(NC(=O)Cc2ccc(C)s2)C1C C(=O)(C(C)C(C)c1ccccc1Cl)NCCCN(C(c1c(CC)noc1)=O)C c1(C(C)C)nccc(C(=O)NCC2(C)CCCN2C(=O)Cc2ccc(Cl)s2)n1 C1(CNC(C)=O)C=CCN1C(=O)CCCc1ccc(C)o1 N1(C(C(C)O)=O)CCC(CCN(C)C(C2(c3ccsc3)CC2)=O)CC1.C1CC1 c1(-c2cccc(C(C)(C)C(F)(F)F)c2)ccc(S(=O)(=O)N2CCC2C(=O)O)cc1 C(C)(C(=O)NCC(=O)NCC1CC1)N(C(CSCC)=O)C1CC1 CC(C)CCC(F)C(=O)NCCOCCOCCCNC(=O)C(C)C#N C1(CC=C)(NC(C2CCC2CC(=O)NCC2CC(CF)C2)=O)CCOC1 c1(OC)ccc2c(CNCC34CC3CN(C(c3cnc(Cl)c(F)c3)=O)C4)c[nH]c2c1 C1(C2CCN(C(=O)CC(O)CN(C)C)CC2)(NC(C2C(C)CC(C)O2)=O)CC1 C1(CC(=O)NCCC2CC(NC(Cc3cn(C)nn3)=O)C2)CCCCCC1(F)F C1(C)(C(=O)NCC2(NC(c3c(SC)ccs3)=O)CCOC2)CCC(=O)N(C)C1 C(=O)(CCS(=O)(=O)Cc1ccncc1)NCCCNC(CSC(C)(C)C)=O C1(C(C)NC(=O)CCCC(N)=O)COC(C)(C)CN1C(c1cnc(O)c(F)c1)=O CC(C)C(N=[N+]=[N-])C(=O)NC(Cc1cn[nH]c1)C(N1CC2(CCCN2C)C1)=O c1(CNC(c2coc(C(F)F)n2)=O)n[nH]c2c1CN(C(c1cnc[nH]1)=O)CC2 CCCCCC(C)(CC)C(=O)NCCC1(O)CN(C(=O)CC2CC2(Cl)Cl)C1 c1(C(=O)NC(C)CN(C)C(C2CC2C2CC2)=O)cc2ccccc2n1C C1(F)(CNC(C(C2CC2)OCC)=O)CCC(CNC(=O)C=CSC)CC1 c1(C(=O)NCC2(O)CN(C(c3n(CCC)ncc3)=O)C2)nn(C(C)C)cc1Br C1(C(N2CC(NC(=O)CCCCN(C)C)C2)=O)(COC)CCCCO1 c1(C(=O)NCCN(CCC)C(c2ccn(C)c2)=O)ncoc1-c1cnn(C)c1 C(CCNC(c1cc(CC(C)C)on1)=O)(C(=O)NOC(c1ccccc1)C)OC c1(OC)ccc2cc(C(N3CC4CC(NC(=O)C(F)C(C)C)C3C4)=O)n(C)c2c1 N1(C(c2c(C)cc(C)nc2S)=O)CCC2CCN(C(C3CCNC(=O)C3)=O)C2C1 C=CC1OCCC1C(=O)NC(C1(O)CN(C(=O)CC2(C(F)(F)F)CC2)C1)C C1(=O)C(C)N1C.C(CCOCC(=O)N(CCCNC(=O)N(C)C)C)N(C)C N1(C(C=C(C)C)=O)CCCCC1C1CCCN(C(=O)C2=C(Cl)CC2)C1 C1(CNC(C(n2cc(Cl)cn2)C)=O)CCN(C(c2ccc(F)c(F)c2)=O)C1(C)C c1(CN2CCC(O)(C(=O)Nc3cccnc3Cl)C2)ccc(Cl)c(I)c1 C1(C(=O)NCC2CN(C(=O)Cn3cnccc3=O)CC2O)COC2(CCC2)C1 Cc1nn(C2CCCN(C(C3CCC=CO3)C(=O)NC(C)(C)C)C2)c(C)c1Cl C12(C(=O)NCC(CNC(c3ccc(CC)[nH]3)=O)(C)C)CCC(C1)OC2 c1(C(N2C(CNC(CCCC=C)=O)C(C)CCC2)=O)nccc2ncccc12 CC1C(NC(=O)C(=O)NCc2sccc2F)CCCN1C(=O)OC(C)(C)C C#CCC(CC#C)C(=O)N1CC(CNC(=O)CC(C)C(F)(F)F)C(COC)C1 Cc1cccc(N)c1C(=O)NCC#CCNC(=O)C(C(C)C)c1ccccc1 Cc1ccc(NC(C2CCN(C(c3c[nH]ccc3=O)=O)C2C)=O)c(O)n1 N1(C(c2c(CC)noc2)=O)CC2(CC(NC(=O)C(N3CCCC(C)C3)=O)CO2)C1 Cc1[nH]c2ccccc2c1C(=O)NC1CCCC1C(=O)NC(C1CCOC1)C c1(N2CC(CC)C3(C2)CCC3)[nH]c(=NC2CC(OC)C2)nc2c1cnn2C(C)C N1(C(COCCC#C)=O)CCCC1C1CCN(C(=O)CSCCN(C)C)C1 C(=O)(C(F)C(C)(C)O)NCC1C(C)CCN1C(=O)C=Cc1ccccn1 N1(C(C2(C#C)CC(=O)C2)=O)CCC=C(C(=O)N2CCC=C(C)C2)C1 c1(C(CNC(c2cc(C)[nH]n2)=O)NC(=O)C(F)(F)c2cscn2)ccc(F)cc1 C1(CC)(NC(=O)Cc2cccc(C)c2F)CCN(C(=O)Cc2conc2C)CC1 C1(C2(C(=O)NC(C)Cn3cncn3)CC2)CCCN1C(c1cccnn1)=O CCCCCC(=O)N1CCCC(N(C)C(C2CC2(F)F)=O)C1 C1(CNC(Cn2ccc(C)n2)=O)CN(C)CCN1C(c1ccc(C(C)C)cn1)=O c1(C(N(C2CC(N(C(=O)CSC(F)(F)F)C)C2)C)=O)cccn2ccnc12 C1(C(=O)NC(CNC(c2c(CC)n(C)nn2)=O)C2CC2)C2CCCCCC12 N1(C(C(COC)OC)=O)CC(NC(c2ccoc2)=O)CCC(O)C1 C1(C(N2C(CCNC(=O)C(F)C3CC3)COCC2)=O)CC2CCC1CC2 c1(-c2cn(CCN(C(c3cc(C)[nH]c3C)=O)CC)nn2)ccc(-c2ccccn2)cc1 NS(=O)(=O)c1ccc(C(=O)NC2CC3(C2)CN(C(=O)Cc2cncnc2)C3)[nH]1 C1(NC(=O)C(O)C2CC2)CCN(C(c2cscn2)=O)C(c2ccccc2)C1 C1(C(=O)NCCOCC#C)CCC2CCC1N2C(c1cnn(CCO)c1)=O C12(C(N(CCCNC(=O)Cc3cc[nH]n3)CCO)=O)CCC(F)(CC1)CC2 N1(C(c2cn(C)nc2)=O)CCC(NC(c2ccc(C#N)o2)=O)C(CO)C1 Cc1cc(C(N2CC(N3CCN(C(=O)Cn4cnnc4O)CC3)C2)=O)c(O)nn1 CC(C)(CCC(=O)NC1CC1CNC(=O)CN=S(C)(C)=O)c1ccccc1 N1(C(c2c(CC)nc[nH]2)=O)CCC2CN(C(=O)C(O)CC[S+](C)C)CC2C1 C1(C(=O)N(C)CC2(O)CN(C(=O)C(N)=O)C2)(OC)CCCC(C)C1 CN1CCN(c2ncc(C(=O)NCC34CC3CN(C(=O)C=C(Cl)Cl)C4)s2)CC1 c1(NC(CC)(CNC(=O)C(C)CF)CC)ccc(C#N)c(C)n1 c1(C(N2C(C(=O)Nc3cc(OC)cc(F)c3)CC2)=O)c[nH]c2ccc(F)cc12 C1(NC(CC2N(C)CCCC2)=O)CCCCCCC1NC(=O)CCn1cccc1 CS(C)(=O)=NCC(=O)NC1CCN(C(c2ccnn2CCF)=O)CC1CO c1(OC)ccc(C(N2CCN(C(=O)Cn3cnnc3O)C3CC23)=O)cc1Cl C(CCCC(C)NC(=O)C(CC1CC1)CC1CC1)NC(CCCSC)=O C(=O)(C1=C(Cl)CCCC1)N1C(CCNC(c2ccn(C3CC3)n2)=O)CC(F)(F)C1 CC1CC(NC(=O)C(=O)Cc2ccccc2)CCN1C(c1cocn1)=O CCC(CC)C(=O)N(C(CC)CC(=O)NCCC1(COC)CCC1)C c1(C(=O)NCC(CC)NC(c2cnc(C)[nH]2)=O)c(C)oc(C)c1Br C(=O)(CCCNC(=O)CSC1CCCC1)NCC(C)(C)OCC C(CCCNC(=O)CCC1CCCOC1)(c1ccccc1)NC(C=C(C)Cl)=O CCCC(C(=O)N1CC(CCNC(=O)CSC(F)F)C1)S(N)(=O)=O c1(C(=O)NCC2CC3(CN(C(c4ncn(CC)c4)=O)C3)C2)c(C)cc(F)cc1C C1(C(N2C(C(C)C)CCC2)=O)CCN(C(=O)COC2CC=CC2)O1 C1(CC)(NC(=O)C(C)CC(F)F)CCN(C(c2ccncc2)=O)CC1 c1(CC)sc(C(=O)NC(C2CCN(C(=O)C(C3CCOCC3)O)C2)(C)C)cc1C c1(N(CC=C)C)ccc(Br)c(S(=O)(=O)NCCc2c(F)cncc2F)n1 c1(CC(=O)NCCO)ccccn1.C1(C(=O)O)CC1 C1(CNC(C2(OC)CCCCC2)=O)CC2CCC(C1)N2C(=O)C(C)C1CC1 N1(C(Cc2c(OC)c(F)ccc2)=O)CC2CCCC(C1)N2C(=O)C(=O)NC(C)C Cc1cccc2[nH]c(C(N3CCC4CCC(C3)N4C(=O)CNC(N)=O)=O)cc12 C1(C)(C(=O)NC2C(NC(c3n(C)ccc3)=O)COCC2)CCC(O)CC1 C(C(CC)(CC)NC(=O)CCCCN1CCCC1)NC(C(CC)O)=O C12(NC(c3ccn(CC(C)C)n3)=O)CCCC1CN(C(C1(CF)CC1)=O)C2 C(=O)(C(C)(C)CC(C)C)NCC1N(C(c2cnc(CC)[nH]2)=O)CC1 C1(C(N(CC(C)NC(C2CC23CCOC3)=O)C)=O)COCCN1CC(F)F Cc1cc(Br)c(Cl)cc1NC(C1C(Nc2ncccc2C(F)(F)F)C1)=O C1(C)(CNC(CCC(C)O)=O)CCCN(C(=O)CC2CCC(C)C(C)C2)C1 C1(CNC(CCCN(C)C)=O)CC2CCCCC2N1C(=O)Cn1cnc(C#N)n1 N1(C(CC(C)OC)=O)CC(NC(c2[nH]nc(C(F)(F)F)c2C(C)C)=O)C(C)C1 c1(C(=O)NC2CC3CN(C(C4CN(C(C)=O)C4)=O)C2C3)c(C)[nH]c2ccccc12 Cc1ccc(C(=O)NC(C2CCN(C(=O)CC3COCCO3)CC2)C(C)C)c(C)c1 c1(OC)ccc(CNC(C2CN(C(C3CCCCO3)=O)CC23CC3)=O)c(OC)c1 C(=O)(C#CC1CCCCO1)NCCCN(C(c1c(Br)ccc(C)n1)=O)C(C)C Cc1cc(CO)oc1C(=O)NC1CN(C(c2nc(Cl)cs2)=O)CC1C c1(C(C)C(=O)NCC2(F)CN(C(=O)CCN3CCCC3)C2)nc(F)ccc1Cl N1(C(c2ccc(C)c(O)c2)=O)CCc2cc(C(=O)NCC(C)CCl)ccc2C1 N1(C(CCC)=O)C2CCC1CC(CNC(c1ccc(OC(F)F)cc1)=O)C2 c1(C(=O)NCC2CC(NC(C(C)N(CC(F)(F)F)C)=O)C2)ccc(N)cc1Cl C(=O)(C(CNC(c1ccn2nccc2c1)=O)CC(C)C)NCCN(C(=O)OC)C C1(CNC(C2CCC(=O)NC2)=O)CC2(CCN(C(c3cc(Cl)cnn3)=O)C2)CO1 CN1CC(C)(C)CC1C(N1CC(c2c(F)cccc2Cl)C1)=O Cc1cc(C(N2CC(NC(=O)C=C3CCOCC3)CCC2C)=O)nc(C)c1 C(=O)(C1=NOCC1)N(CC(CC)NC(=O)Cc1cccc(OC(F)F)n1)CC N1(C(C(C)n2cncn2)=O)CCC2CCN(C(C3CCC3)=O)C2C1 CN1N=CC(CC(=O)NCC2CN(C(C3CCS(=O)(=O)C3)=O)C2)C1=O CCC(C#N)C(=O)NC1(C)CC(NC(c2cc(CCCO)on2)=O)C1 c1(CNC(CC(C)c2ccccc2)=O)ccc(CNC(c2cnsc2)=O)c(F)c1 c1(NC(CNCC2CC(OC)(CN)C2)=O)ccc(C)c(Br)c1 C1(CC(=O)NC2(COC)CN(C(=O)C(CO)N(C)C)C2)CC2(CC2)CO1 C(=O)(C1=CCc2ccccc21)NCC1C(NC(c2cc(C3C(C)C3)on2)=O)CCC1 c1(CC(N2CCOCC(NC(C3(O)CCCC3)=O)C2)=O)c[nH]c2ccccc12 Cc1nn(C2CC2)cc1C(=O)NC1CC(NC(C2(C(=O)OCC(C)C)CC2)=O)C1 c1(C(=O)NCC(CNC(C2N(C(C)=O)CC(O)C2)=O)C)cncc(Cl)c1C N1(C(C(COC)(C)O)=O)CCN(C)C(CNC(c2ccc(C(C)(F)F)cn2)=O)C1 c1(OC)cc(C(N2CCC(O)C(C(=O)Nc3cccc(CO)n3)C2)=O)cnc1Cl C#CC1(C(N2CCC(O)(CC)C2)=O)CN(C(=O)CCCC2CCCO2)C1 N1(C(C(C)N(CC)CC)=O)CCC2CCCC12C(=O)NCC1CCC(C)(CC)O1 C(=O)(CCCCCCC(=O)NC(CO)C(C)NC(=O)C(=O)NCC(F)F)OC N1(C(C)=O)CC2(CC2)CC1C(=O)NC1CC(O)CN1S(C)(=O)=O C(=O)(CC1=CCCC1)N(CCn1cc(-c2ccc(C)nc2)nn1)CC CN1CC2CC1CN(C(C1N(C(=O)COC(C)(C)C)CCC1(C)C)=O)C2 C1(NC(C2CCCC(C)CC2)=O)CC2CCC1N(C(=O)C=Cc1cccnc1)C2 C1(CNC(c2c(CNC(CCC#C)=O)ocn2)=O)CCC(=O)NC1C C1(C(N(C)C)=O)CC2(CCN(C(=O)NCc3c(I)ccnc3O)CC2)CO1 c1(C(C)C)ncc(Br)c(=NC(CNC(C2CCC(=O)N(C(C)C)C2)=O)CO)[nH]1 C1(C)(CNC(c2cc(C(C)C)[nH]n2)=O)COCCN(C(=O)C(C)c2ccsc2)C1 c1(C(=O)NC(C)C(=O)N(C2CN(C(=O)C(O)CF)C2)CCO)ccc(F)cc1F c1(N(S(C)(=O)=O)C)nc(N2CCN(CC3(CO)CCCO3)CC2)c2c(n1)CCS2 N1(C(c2ccc(OC)cc2)=O)CC(C(N2CC(C(C)C)C2)=O)CCC1(C)C C(C1CCOCC1)=CC(=O)NC(CNC(C1CC2C=CC1O2)=O)C1CC1 N1(C(C(CSC)O)=O)CC(NC(=O)CCc2csc(C)n2)C(C2CC2)C1 CCC(C)(C(=O)NCCOCCCNC(=O)Cc1ccoc1)OC N#Cc1cnn2cc(CN3CCN(C4CCCS(=O)(=O)C4)CC3)cnc12 C(=O)(CCCCC(C)C)N1CCCC(O)(CN(C(CC(C=C)C)=O)C)C1 C(C(O)C(C)(C)C)NC(c1scc(CNC(C2C(C(=O)OC)C2)=O)c1)=O c1(C(N2CCC3CCN(C(CCC)=O)CC32)=O)cc([N+](=O)[O-])cc(S(C)(=O)=O)c1 CCC(C)(C)C(O)C(=O)NCCC(=O)NCCSCCC(=O)CO C#Cc1ccnc(C(=O)N(C(C)C(=O)NCC2=NOC(C)C2)C)c1 c1(C(=O)NC2CC(F)(CNC(C(CC)N(C)C)=O)C2)[nH]c(C)nc1C c1(C(=O)NCCCC(CCC)NC(C2CCN(C)C2=O)=O)cn2cccnc2n1 Cc1noc(C)c1CC(=O)NC1CCCCN1C(=O)C=CC(=O)NC1CCCCC1 C1(C2CCC2)(C(=O)NC2C(CNC(=O)C(c3cccc(Cl)c3)O)C2)CC1(F)F C1(N(C(c2cc(C)cc(F)c2N)=O)C)CCCC2CN(C(=O)C3=CCSC3)CC12 C#CCC(CC(=O)NC(c1nnnn1C)C)NC(C1(C)CCOCC1)=O C1(C2CCSCC2)(NC(c2n(CCC)nnn2)(C)CSC)CC1 C(=O)(C(CC(C)C)OC)NC(C(C(C)C)NC(COCC=C)=O)C c1(C(=O)OC)cc(N(C2CCN(C(c3nc(=O)n(C)[nH]3)=O)CC2)CCO)nc(C)n1 N1(C(CC(C)=C(C)C)=O)CCCCC1CC(=O)NCCCCC1CC1 C1(NC(=O)CCCn2cncn2)CCN(C(c2cn(CCCF)nn2)=O)CC1F C1(O)(CC(=O)NCCCC2N(C(C(C)C)=O)CCCC2)COC(C)(C)C1 C12(C)CCC(C1)N(C)C2.C(=O)(CCOCC(=O)NC1CCC1)OC c1(C(N2CCC(CC(C)CO)CC2)=O)ccc(S(=O)(=O)C2CCC2)cc1 c1(OC)c(Br)ccc(F)c1C(c1nnnn1C(C)C)NC1C=CCC1 C(C(CC(=O)OCC1Cc2ccccc2N1C)C(F)(F)F)N(C)C C(=O)(C(C)CC(F)(F)F)NC1C(SC)CN(C(C2C=CCS2)=O)C1 c1(C(N(C2CCN(C(C34CCC3C4)=O)C2)C)=O)cccc(C#N)c1 c1(C(N2CC(CC=C)(NC(c3nc(C)sc3C)=O)C2)=O)cc(C#N)ccc1O C(=O)(CCC(O)C(C)(C)C)NCC(C)N(C(c1cc(SC)ncc1)=O)C N(C(=NCCCF)NCCc1ccc(F)cc1Br)C1N(C)S(=O)(=O)CC1 C1(F)(CNC(c2c(C)cnn2C)=O)CC2CCC(C1)N2C(C1CCC(C)(C)C1)=O CC1CN(C(c2cccc(C#N)c2)=O)CCC1N(C(=O)C1=CCOCC1)C N1(C(CC(=O)NCC)=O)CC(NC(=O)COC2CCOC2)C(c2cnn(C)c2)C1 c1(OCC)cc(Cl)ccc1C(=O)NC1CN(C(C2CCCC2(F)F)=O)C1 c1(C(N2C(C)CCC(NC(C3CC34CCOC4)=O)C2)=O)cccc2c1OCCN2 c1(OC)ccc(C(N2CCCC(C(N3CC4CCC(C3)O4)=O)C2)=O)cc1F C1(NC(C(CC#C)NC(=O)CCCCC#N)=O)CC2(C1)CC(C#N)C2 N1(C(COCC)=O)CCN(C(c2sc(F)cc2C)=O)CC1COC CCCCC(C(=O)N1CC(C(N2CC(C)(OC)C2)=O)CC12CCC2)C(C)C C(CC1CC1)(CC(=O)N1CCOCC1CCO)NC(c1ccn(COC)n1)=O N1(C(c2c(C(C)C)occ2)=O)CCC(CO)(CNC(=O)CC(C)F)C1 CCC(CCC(=O)N(C(C)CN(C)C(c1ccc(C(=O)OC)s1)=O)C)OC C(=O)(C1=CC2CCCC12)NCC1(O)CCN(C(C(C(C)(C)C)NC(N)=O)=O)CC1 C1(CC(=O)NC2(CCC)CC2)CCCN(C(C2CC(F)C(=O)N2)=O)C1 C12(CNC(C3CC(C#N)C3)=O)CCC(NC(=O)Cc3cccc(Cl)c3)(CC1)CO2 CC1=C(C(=O)Nc2ccc(-c3ccc(OC(C)(C)C)cc3F)nc2C)CCO1 N#CC1CN(Cc2ccccc2)CC1C(=O)N(c1cc(Cl)ncc1F)c1ncncc1F N1(C(c2ccc(C#C)o2)=O)CC2CCCC2(CNC(=O)CC2(C)CC(F)(F)C2)C1 c1(N(C(CN(C(Cc2c(CC)cccc2)=O)CC)C)CC)ncc2ncnc-2[nH]1 CC1CN(C(c2cnnn2C)=O)CC1NC(C1(C)C=CCC1)=O N1(C(C2N(C(c3c(CC)nn(C)c3)=O)CC(C)C2)=O)CC2CC2C2CC12 C1(NC(C2CCSCC2)=O)CCCC(CC(=O)NCC(CN(C)C)O)C1 C1(C(=O)NCC2CC(F)(CNC(Cc3n[nH]c(=N)s3)=O)C2)CCCN1C=O C#CC1CN(C(=O)C(CC2CCC2)NC(C2CC(CF)C2)=O)CCO1 N1(C(c2c(C)cnnc2)=O)CC2CCCC(C1)N2C(C12CCC(C)(CC1)CC2)=O c1(OC)cncc(C(=O)NCC2(F)CCC(CNC(C3(CCF)CCC3)=O)C2)c1 c1(C(=O)NCCC2(O)CCN(C(=O)CCC3CC3(F)F)C2)cc(Cl)cnc1O c1(C(N2CCC(N(C(=O)C3=NOCC3)CCC)CC2)=O)cn2c(n1)CCC(C)C2 C1(NC(NC(C#C)C(C)C)=NC)CCOC2(CCC2)C1 C(C(C(=O)NC1(CO)CC(F)C1)C(C)(C)C)NC(CCCC#C)=O CC(C)CC(C)(CNC(C1CC(C)(C)O1)=O)NC(=O)CCC(C)(F)F C#CC1(C=C)COCCN1C(c1cc2ccncc2o1)C(=O)NCC Cc1cnn(C)c1CC(N1CC(N(C(=O)CN2CC(C)C2)C)C(O)C1)=O C(=O)(C1c2c[nH]nc2CN1C(=O)CSC(F)F)NCc1cc(OC)ncn1 N1(C(c2ccc(CN=[N+]=[N-])o2)=O)CCC(NC(=O)CCSC2CCCC2)C(O)C1 c1(CC)cc(F)ccc1C(=O)NC1(CCNC(C2(CC)CCCC2)=O)CCC1 C1(C(=O)NCC2(CNC(c3c(C)cc(Br)o3)=O)CCC2)CCC2CCC(=O)N12 O=C1NCC2(CCN(c3nccc(N4CCC(CC5CCOC5)C4)n3)CC2)N1 CC1(F)CCN(C(C2(C)CN(C(=O)CCn3cccc3)CC2C)=O)CC1 Cn1ccc(C(N2C3CCC2C(CNC(C2CC2c2cccs2)=O)C3)=O)cc1=O Cc1ccn(C(C)C(=O)NCCNC(C2CN(C(C3SCCS3)=O)C2)=O)n1 C1(CC(=O)N(CC(C)O)CCNC(c2c(C)n[nH]c2)=O)CC(C)(C)CO1 C1(O)(N(C)C)CCN(C(=O)C(C2CCCCC2)NC(C2(C(N)=O)CC2)=O)C1 Cc1n[nH]cc1C(c1nnnn1C1(C)CC1)NCC(Cc1ccoc1)CO C(=O)(CCC(=O)c1ccc(F)cc1)NC1C(CNC(C(C)(F)F)=O)CCC1 C1(C(N(C)CC2N(C(CCSCC(C)C)=O)CCOC2)=O)Cc2cccnc2C1 C1(Cn2cc(CCCSC)nn2)N(C(C23CSCC2C3)=O)CC1(C)C c1(NC(=O)NCC2(CCCC)CCCC2)c(Cl)cc(Cl)c(Cl)c1F c1(NCC2C(C)CN(C(C3CNC(=O)CC3C)=O)C2)c(C#N)c(=O)n(C)c(=O)n1C N1(C(CCNC(=O)OC)=O)CCN(C)C(CNC(c2cc(C3CC3)[nH]n2)=O)C1 n1(CC)cc(CC(=O)NC2CC(CNC(=O)C(C)C(C)(F)F)C2)c2ccccc12 c1(C(=O)OCC)ncc(Br)cc1NCC1(c2cccs2)CC1C C1(C)(NC(C2(CC#C)CCCO2)=O)CCN(C(=O)C#CC2CC2)CC1 N1(C(c2c(S(C)=O)cccc2)=O)CCC(C2CCCN(c3nnns3)C2)CC1 CC1(C)C2CCC1(C(N1CCN(C(c3cc4scnc4[nH]3)=O)CC(O)C1)=O)CC2 c1(OC)c[nH]c(C(=O)NCCCCCCNC(=O)Cc2cncn2C)cc1=O Cc1cccc(C(=O)NCCC(C)CCNC(=O)C(F)n2ccnc2)c1C C1(c2ccccc2F)(C(=O)NC(C(C)NC(=O)C(C)C)CO)CCCCC1 C1(CCNC(c2cccnc2)=O)CC(N=c2nn[nH]n2-c2ccccc2)C1 C1(NC(C(CC)NC(N)=O)=O)CCN(C(=O)C(Cl)=CCl)CCC1(F)F C1(O)(CCNC(C2CC(OC)C2)=O)CCCN(C(=O)CCCc2nncn2C)C1 c1(C(C(=O)NCC(C)NC(C2C3CCC23)=O)C)ccc2c(c1)OCCO2 CN1CC(C)(C(=O)NCCn2cc(-c3cnn(C4CCC4)c3)nn2)CCC1=O N1(S(=O)(=O)CC2(C(F)(F)F)CCC2)CCOC2(CCCCC2)C1 C1(NC(C(CCN(C)C)O)=O)CC2CC1N(C(C1(CCO)CC1)=O)C2 c1(C(=O)NCCOC2CN(C(c3ncc(F)cn3)=O)C2)ccc(Br)c(O)n1 C1(C(F)(F)F)(C(N2CCN(C(C(C)OCCC#C)=O)CC2)=O)CC2CCC1CC2 CC(C)P(=O)(CC(=O)NCC1(O)CCN(C(C2CC=CCC2)=O)C1)C(C)C CCCC(C)CN=c1ccc(S(=O)(=O)NCCC(O)CN(C)C)c[nH]1 c1(C(N(CC(C)N(C(=O)CCC=CBr)C)C)=O)cc(N)cc([N+](=O)[O-])c1 CCC(CC)(CCNC(C1CCC(C)(O)CC1)=O)NC(=O)C(COC)CC c1(C(=O)NC2C(NC(c3c[nH]c(C)c(Br)c3=O)=O)CC2)cccn2c(O)nnc12 C1(CC)CN(C(=O)C(C)NC(c2cc(CO)c(C)o2)=O)CCN1C C1(NC(=O)NC(Cn2ncc(C)c2)C)C(C)CCC1C N1(C(C2(OC)CCN(C(=O)Cc3ccnn3C)C2)=O)CC2COCC2(C)C1 C(=O)(C(CCCC)C(C)C)NCC(C(=O)N(C(C=C)C1CC1)C)CC1CC1 N1(C(c2cn(CC=C)nn2)=O)CCOC2(CCN(C(C3(CC)CC3)=O)C2)C1 C(=O)(C(C)(C)CF)N(C(CC)C(=O)NC1CCCC1CN(C)C)C c1(C(N2CCC(NC(CCCC)=O)CC2C)=O)ccc(Cl)c(F)c1F CCC(CN=c1ccc(S(=O)(=O)NCC2CCOCC2)c[nH]1)C1CCOCC1 Cc1cccc2[nH]c(=NC3CC(CNC(=O)C4=CCCC(C)(C)C4)C3)sc12 N1(C(=O)NCCn2nnc(C)n2)CCC(OC)C1(C)C C1(C(N2C(C)CC(CNC(=O)Cc3ccccn3)C2)=O)CC2C=CC1C21CC1 CC1CSCCCN1C(C1CC(C)N1C(=O)CC1OCCO1)=O C1(C(=O)NCCOC2CN(C(c3cn(C4CCOC4)nn3)=O)C2)CCCCS1 N1(C(c2c(CCC)nns2)=O)CCC(F)(F)C(CNC(c2sc(F)cc2C)=O)C1 C1(C(=O)NCC=CC)CCN(C(=O)Cc2cccnc2)C1C N1(C(=O)Nc2cc(C)[nH]c2C)CCCc2cccc(OC(F)F)c21 N1(C(CCn2cc(C(=O)OC)nn2)=O)CCOC(C)C1CO.C12CC(C1)NC2=O CC(C)CC(C)CC(=O)N1CCC(F)C(NC(=O)C(C)(C)n2cnnn2)C1 c1(C(N2CC(CC)C(C(=O)N(C(C)C(N)=O)C)C2)=O)cccc(C)c1O N1(CC)N=C(C(=O)NCC2CCN2C(c2cc(C3CCC3)[nH]n2)=O)CCC1=O N1(C(C2(C(=O)OCC)CC2)=O)CC(COC)CC(C)C1 C1(C(=O)NCC2N(C(c3cc(C(C)C)n(C)n3)=O)CC=C2)CN(C)C(=O)CCO1 CC1C(NC(C2CCCS2(=O)=O)=O)C(C)CCN1C(=O)CC1CN2CCN1CC2 CCCC(CCO)NC(=O)Nc1ccnc(N2CCC(C)C2)c1 c1(C(N2CC(OCCNC(CC3(C)CCCO3)=O)C2)=O)ccccc1NCCO c1(C(=O)NCC2CC(NC(CCOC)=O)C2(C)C)ccc2nnn(C)c2n1 C1(CC(C)C)(C(=O)NC2CCC(CNC(C3(C#N)CC3)=O)C2)CCNC1=O c1(C(N(C(C)CNC(=O)CSc2nncs2)CC)=O)cn(C)cc1C(F)(F)F c1(C(=O)NC2CC(CNC(C(C)NC(=O)NC)=O)C2)cnc(C(C)C)nc1O N1(C(CC2(C=C)CN(C(C3(C(N)=O)CC3)=O)C2)=O)CC(C)OCCC1C N1(C(c2nc(C)sc2)=O)CC2CC(C1)C2C(=O)CC1CCCC1C c1(C2(C)CC2)ccc(C(=O)NCC2CC(F)(F)CN2C(c2cnsn2)=O)cc1F C1(C)(c2cn(C(C)C(=O)Nc3cccc(OC(F)(F)F)c3)nn2)CC2CC2C1 C(=O)(C(C(C)NC(c1ncccc1Cl)=O)C(C)C)Nc1c(OC)cc(F)cc1 C12(CNC(c3ncn(C)c3)=O)CC1CN(C(=O)CCCC1CCOCC1)C2 C1(CNc2n(CCF)nc(-c3ccccc3)c2)CN2CCC1CC2 C(=O)(CCCC(C)(C)C)NCC(CNC(C=C1CCC(C)C1)=O)C c1(CC)oncc1C(=O)NC1CCC(CNC(=O)C(N2CCOC2=O)C2CC2)C1 C=C(C)c1cccc(NC(=O)C(CCC)NC(=O)CC2CC(F)(F)C2)c1 c1(CC)nc(N2CC3CC2(CNC(=O)CC(C)(O)COC)C3)c(F)c(Cl)n1 CC1(C)CCC1C(=O)NCC1(CNC(c2ccn(C3CCCC3)n2)=O)CC1 N1(C(C(CC)SC)=O)C(C)C2CC1C2NC(=O)CNC(C1CCCC1)=O C1(NC(C2(CC#C)CCCCC2)=O)CC2CCC(C1)N2C(=O)C1=C(C)CCCC1 c1(C(=O)NC2C(C)N(C(=O)CC3CCSCC3)CCC2)cnc(O)n(C)c1=O c1(CC)cccc(C(N2CCOC(C(=O)N(CC(C)O)CC)C2)=O)n1 N1(C(c2sccc2Cl)C(=O)NC(C)C)CCC(C(F)(F)F)(C(F)(F)F)C1 C1(OC(=O)NC(C)(C)C)CN(C(=O)CCF)CC1NCC.C12SCCN1C2=O c1(CC)scnc1C(=O)Nc1nnc(N(C(=O)C2CC2)C2CC2)s1 C1(C(=O)NCCCN(C(CC=C)=O)C)CC2(C1)CC(F)C2 C1(NC(=O)CCc2ccccc2)CCSC12CN(C(=O)C(C1CCOCC1)O)C2 C1(C(C(=O)Nc2c(C)csc2)C)CCN(C(c2ccc(C#N)s2)=O)CC1 C(=O)(CCN(OC)C(=O)C(C)c1cccs1)NC1(C=C)CCCC1 CCCCC#CC(C)(C)NC(C1CC(O)CN1C(C1CCC(=O)N(C)C1)=O)=O Cc1cc(=NC(C)c2ncnn2C(C)C)[nH]c(=NCc2nccc(O)n2)[nH]1 C(CC(O)C(=O)NCC(CC1CCCC1)C(=O)NCC(c1ccccc1)C)SC C1(c2onc(CN(C)C)n2)CN(CC2(C)CSCCO2)CCO1 N1(C(c2cc(C)[nH]c2C)=O)CCCC(CO)(NC(C2CCSC(C)C2)=O)C1 c1(CC)occc1C(=O)NC1(C(=O)N(CCF)CCOC)CC1(C)C c1(C(N2C(C)(CNC(c3ccoc3C3CC3)=O)CCC2)=O)ccc(F)c(C#N)c1 c1(C(C(N2CC(C)(NC(C(C(C)C)N(C)C)=O)C2)=O)N(C)C)c(F)cccc1F C(=O)(C(O)CCCNC(=O)CC1CSC1)NC(C1CCOC1)C#C N1(C(CCc2cc(C)on2)=O)CCCC(C2CN(C(=O)C(C)c3cc[nH]n3)C2)C1 c1(OCC(=O)NCC(CC)NC(c2cncc(F)c2)=O)cncc(Br)c1 C1(NC(C(C)(N(C(c2cc(OC)n[nH]2)=O)C)C2CC2)=O)CCN(C)C(=O)C1 C1(C(N2CCC(NC(CN(C(C)C)C)=O)C2)=O)CC(c2ccccc2)=NO1 C1(C(=O)NCC(C#C)CC)C(C)CCN1C(=O)C=Cc1cocn1 N1(C(CN(c2nn[nH]c2C(C)(C)C)C(C)=O)=O)c2ccc(Cl)cc2NC1(C)C c1(C(=O)NC2(C(=O)Nc3ccc(Cl)nc3)CC2)ccnc(O)c1 Cc1cncc(C(=O)NC2CCCC(NC(=O)CCc3ccccc3Cl)C2)c1 N1(C(C)C)CC(C(N2CCCC2C(C)(C)NC(C2CC2(F)F)=O)=O)CC1=O c12ccccc1CCS2.C1(CC(=O)OC)CCCC(C)C1 c1(C(=O)NC2(C)CN(C)C(=O)CC2)cc2n(c1)CCCNC2=O c1(CC(=O)NCC(CNC(C2(CC=C)CCC2)=O)C)ccc(F)c(Br)c1 CC1CC=C(C(=O)NC2CCCCC2NC(=O)COc2ccc(Cl)nc2)CC1 N1(C(c2ccc(N(C)C)cn2)=O)CCCCCC(Nc2ccccc2[N+](=O)[O-])C1 c1(C(=O)NC(c2cn(-c3ccc(OC)cn3)nn2)(C)C)ccc(Br)c(F)c1F O=C(C1=CCCCO1)NCc1cc(C(=O)NCc2noc(C3CC3)n2)cs1 N1(CC(=O)NC2(C)CCN(C(CC=CC=C)=O)C2)CCSC2CCCCC12 CCCC(C)(CCC)C(=O)NC1C2CC3C1C3C2C(=O)NCC(C)(COC)CC C(c1ccc2c(c1)COCC2)=CC(=O)NCC1CC(NC(COCCC=C)=O)C1 N1(C(C2N(C(c3cc(C)c(C)nn3)=O)CC(O)C2)=O)CC2(CCC1CO)CC2 C(=O)(C1=CCCCCC1)NC(CN(C(C(C(=C)C)(C)C)=O)C)C N1(C(CC2OCCC(C)(C)C2)=O)Cc2ccccc2C(NC(=O)CC2(C)CC2)C1 c1(CC(=O)NCC(CC)NC(=O)CC(C)(C)COC(C)=O)ccc2[nH]ccc2c1 N1(C(c2c(C=C)cnn2C)=O)CC=C(C(C)(C)C(=O)NCC)C1 c1(OC)cc(CNC(Cn2cncn2)C(=O)O)cc(C#N)c1 CC(C)CC(O)C(=O)N1CCOCC1CNC(=O)CCN1CCCCCC1 c1(C(=O)NCCC2CC(OC)CN2C(C2CCOC2)=O)c(F)cc(Cl)cc1F C1(CNC(C(CC=C)C)=O)CC2(CCOCC2)CN1C(=O)C(F)=C1CCCC1 c1(C(N2CCC(C(C)NC(=O)Cn3cc(Cl)cn3)C2)=O)ccc2nc(O)oc2c1 C1(CC(=O)NCC2(O)CCC2)COCCN1C(c1scnc1C(F)F)=O C1(NC(c2cnc(CC)s2)=O)CC2(C1)CC2NC(c1cn[nH]c1)=O S(=O)(=O)(c1ccc(NC2CCCC3CC23)cc1Br)N1C(C(N)=O)CC(F)C1 c1(CC)ccc(C(N2CCCC(c3cn(C)nn3)C2)C(=O)NCC2CC2)cc1 N1(C(=O)CC2CCCCO2)CCOCC1NC(CC1CC(NS(C)(=O)=O)C1)=O Cc1cc(Cl)c(Cl)cc1C(N1CC(NC(c2c(C)cccc2C)=O)C(F)C1)=O Cc1ccc(S(=O)(=O)C2(C(=O)NC3CCNS3(=O)=O)CCCC2)cc1 C1(COC)CN(C(C2CC2c2cnc[nH]2)=O)CCN1C(C1(F)CCCC1)=O c1(C(=O)NCCN(C(=O)CC2OCCC2C)CCC)c[nH]nc1C1CC1 C1(NC(C2CCCN(c3nccs3)C2)=O)CCC2(CCNCC2)C1 c1(CC)noc(C(=O)NCCCCCCNC(c2ccc(C(C)=O)nn2)=O)c1C Cc1cc(C)c(C(=O)NC(C2CC2C(=O)NC(C)Cc2nn[nH]n2)C)s1 CCCCCC(CC)C(=O)NCC(=O)NCC(=O)NC12CC1COC2(C)C C(=O)(C#CC1(C)CC1)NC1(CN(C)C(C2(C)CC2c2ccccc2)=O)CC1 CCC(CN(C)C)CC(=O)N(CCC(=O)NCc1nc(CO)n[nH]1)CC C(CCCCC(=O)N(C(C)CCNC(c1cn(C2CCC2O)nn1)=O)C)=CC CC(C)CC(C(=O)NCC1(O)CCCN(C(=O)Cc2ccco2)C1)C(N)=O C(=O)(C(C)CS(C)(=O)=O)N(C)CC1CCCN(C(c2cncc(C(C)C)c2)=O)C1 N1(C(c2cc(C(C)=O)c(O)cc2)=O)CCC(C2(NC(=O)CC3CC3(Cl)Cl)CC2)C1 N1(C(CCOCCOCC)=O)CCC2(CCN(C(c3ccc(C#N)[nH]3)=O)C2)C1 N1(c2nnc(CC)o2)C(CNC(=O)C=Cc2cocn2)CC2COCC12 c1(C(CNC(=O)CCc2cnn[nH]2)=O)ccccc1Cl c1(C(N2CCC(CC=C)(NC(c3cc(C)sc3C)=O)C2)=O)cccc(F)c1F c1(CC)noc(C)c1C(=O)NCC1(F)CC(CNC(C2CC2F)=O)C1 N1(C(C(CCN(C)C)NC(=O)CC2CCC(=O)N2C)=O)CCc2ncncc2C1 Cc1nc2ccccc2n1CC(=O)NC1CN(C(C2CCSC2)=O)CC1O CC1(C)CC(N=c2ccn3nccc3[nH]2)CN(c2ccncc2)C1 C(C)(C(=O)N1CC(c2ncccn2)C1)(C1CCC1)NC(COCCN(C)C)=O c1(COC(C2OCCN(C(CC(C)C)=O)C2)=O)cc(F)cc2c1CCC2 c1(C(=O)NC(C)C(C)NC(=O)C=Cc2ccccc2)ncc(Cl)cc1Cl c1(OC)ncnc(OC)c1C(N1CC(CN(C)C(C2CCCCC2(F)F)=O)C1)=O CP(C)(=O)CC(=O)NCCNC(=O)NCC1CCCN(C(c2ccoc2)=O)C1 CC1(C(=O)NCCC2CCN(C(=O)C=CCO)C2)CC(c2ccccc2Cl)=NO1 c1(C(N(CCN(C(c2cc(C)on2)=O)C(C)C)C)=O)cc(F)cc(Cl)c1N c1(CC)cc(C(=O)NCC2CC2C(=O)NC2CC(CC)(CC)C2)on1 C=Cc1ccc(CC(=O)NCCC2CC(NC(=O)CN3CC4CC4C3)C2(C)C)cc1 c1(C(N(CC(CN(C(C2C(OC)CC2)=O)C)O)C)=O)cccc(C)c1[N+](=O)[O-] c1(NC(C2CC3CC3N2C(=O)C(c2ccccc2Cl)O)=O)ccc(F)cc1O c1(COC(C(C)OC)=O)cc(=O)n2c(n1)CCCC2 c1(C(N2CCCC(Cn3cc(C4(O)CC4)nn3)C2)=O)cnc2cccnn12 CC(C)(C)CCCCNC1(c2nnnn2C2CC2)CCCCCC1 n1(CC(=O)N(C2CC2)CC2CCC(NC(=O)CC3CCCCC3)C2)nnc(=O)[nH]1 c1(C(=O)NCCCCCCN(C(=O)CC2CCC(=O)N2)C)ccc([N+](=O)[O-])s1 CC1CC(NC(c2occ3c2CCC3)=O)CN(C(=O)Cc2cnns2)C1 CC1(C(N2CC(c3ccc(Br)cc3)C2)=O)COC(=O)N1 C1(CC(=O)NCCNC(C2C=CCCC2)=O)COCCO1 C1(C2CC2)(CNC(Cn2c(C(F)F)cc(C)n2)=O)CCN(C(=O)C(Cl)=CCl)C1 C1(CC=C)CCCCN1C(c1c[nH]nc1CNC(=O)CC1CC=CCC1)=O C1(C(N2C(COC)(CNC(c3cocn3)=O)CCC2)=O)CC2C(C1)C2(F)F C1(COC)CCC(NC(=O)CC2CCCN2C(=O)CC2CC(SC)C2)CC1 c1(C(=O)NS(C)(=O)=O)cccc(NCCc2ccc(Cl)cc2)c1 C1(NC(c2c(C)nc[nH]2)=O)CCCCC1C(=O)NCC1(O)CCOC1 O=C(NNc1cc(F)cc(F)c1)N1CC(F)CC1c1nn[nH]n1 C1(CNC(=O)CC2CCCOC2)CC2CCCCC2N1CC=CCl c1(CN=c2scc(-c3c(OC)cccc3)[nH]2)cccn2c(O)nnc12 C1(NC(c2cccc(CC)n2)=O)(CC)CCCN(C(C2CCC2)=O)C1 N1(C(c2n(CC)nnc2)=O)CCC2CCN(C(=O)C=Cc3nccs3)C2C1 C1(C2CN(C(=O)C(C)(C)C3CCCC3)C2)(NC(C(n2c(C)ncc2)C)=O)CC1 CCCCC(=O)NC1CC(C(F)C(=O)N2CC(C3CCCCO3)C2)C1 C1(NC(CCc2ncc(C)[nH]2)=O)CCN(C(=O)COCC2CCOC2)CC1CO C1(C(N(C(C)CCCO)C)=O)COCCC1NC(=O)CC1CCCC(C)O1 C12(CNC(C3CCC4(CC4)C3)=O)CC1CN(C(=O)C=CCO)C2 c1(C(c2nnc(-c3ccccc3)s2)SCCN(C)C)ccc(Cl)cc1 c1(C(=O)NCCN(C(C2CCC(C(C)C)NC2=O)=O)C)cn2cc(Cl)cnc2n1 C(=O)(C1CCc2c[nH]nc21)NC(CCC=C)C(=O)NCc1ncc[nH]1 C1(CNC(=O)C(N2CCC(C3CC3)C2)=O)CCC2(CCCCCC2)O1 N1(C(c2c(C)[nH]nc2Cl)=O)CCCC(C)C1CNC(C1CC(=O)NC(=O)C1)=O Cc1cc2c(cc1C)C(C(=O)NCCCCC(C)NC(C1CCCSS1)=O)CO2 C1(C(=O)OC)CCC1(C)C(=O)N(CCCNC(=O)C(C)CC)CC1CC1 c1(C(=O)O)cccc2c(CNC(C3(F)CCC(F)(F)CC3)=O)ccnc12 C(=O)(C(C)CN(C(=O)C=C(C)C)C)N(C1CCCOC1)CC N1(C(C(C)(C)CC2CCCCC2)=O)CCN(c2ncc([N+](=O)[O-])cn2)CC(O)C1 CCCN(C1CC1)N(C)Cc1cn2cccc(Br)c2n1 CC(C)C(F)(CNC(=O)CC1OCCCO1)C(=O)NC(c1cccnc1)CO N1(CCC)CC2CCN(C(=O)C(C)CCC(C)(C)C)CCC2C1 c1(C(N2CCC(CC)CC2C(N2CCC=C(Cl)C2)=O)=O)cccc2ccccc12 c1(-c2cc(C(N(C3CN(C(C(CSCC)O)=O)C3)C)=O)no2)ccc(OC)cc1 N1(C(C=C=C(C)C)=O)CCCC(C)C1CNC(c1cn(C)ccc1=O)=O N1(C(c2cccc(C(C)C)n2)=O)CCCC12CCN(C(c1cncs1)=O)CC2 N1(C(C(C(C)(C)C)NC(C)=O)=O)CC2CC(C1)N(C(=O)CCC1OCCO1)C2 Cc1cc(N2CCN(C(C)C(=O)N3CCCC3)CC2)cnc1O N1(C(C2CC(OCC)C2)=O)CCCOC(CNC(=O)C(c2ccccc2)C)C1 N1(C(C(C)CC(F)F)=O)CC2COCCC2(NC(c2ccc(Cl)cc2Cl)=O)C1 C(c1ccsc1)=CC(=O)NCC(CC)NC(C1(N2CCNC2=O)CC1)=O C1(OC)COCCC1CC(=O)NC1CC(CNC(c2ccoc2C2CC2)=O)C1 c1(C(N2CCN(C(C(=O)NC(C)C)=O)C(C)C2C)=O)nnc(O)c2ccccc12 c1(NC(C2CC(F)CN2C(c2c(F)ccnc2Cl)=O)=O)ncc([N+](=O)[O-])cc1Br C(CN=c1ccnc(NC2CC(COCC(F)(F)F)C2)[nH]1)C1CC(C)C1 C1(NC(c2scc(C)c2C)=O)CCC2(CCN(C(=O)CSc3ccncc3)C2)C1 C1(CNC(C2N(S(C)(=O)=O)CCCC2)=O)CCCC12CCN(C(=O)COCCF)CC2 c1(NC(c2n(C(CC)C)nnn2)c2scnc2Cl)cccc(OCCCC#N)c1 CC1(C)CC(F)(F)CN1C(=O)Cn1cc(CN2CC(O)CCC2=O)nn1 c1(C(=O)NCC(CC)NC(C2OCCO2)=O)ccnc(C(C)(F)F)c1 c1(CC)cccc(F)c1C(N1CCC(C)C1CNC(=O)C(C)(C)c1cccs1)=O N1(C(C(C#C)(C)C)=O)CCCC(C(=O)NCC2(CO)CC3CC3C2)CC1 N1(C(C(CN(C)C)(C)C)=O)CC2(NC(=O)C(C3CCCCCC3)O)CCC1CC2 C(=O)(C(C)(C)CS(C)(=O)=O)NCC(C(C)C)NC(c1cc(F)c(CO)c(F)c1)=O N1(C(COCCCCC)=O)CCC2CCN(C(=O)C3CC3)CC12 c1(C(N2C(CNC(c3c(SC)ccs3)=O)CC(C)(C)C2)=O)cc2ccncc2[nH]1 Cc1cc(Br)cnc1C(=O)NCC1CCN(C(C2CC(N3CCCC3)C2)=O)C1 C(C)(C(=O)NC1CCCCN(C(=O)CCc2cncn2C)C1)(C(C)C)OC CC(C)(C)C1=NOC(C(=O)NCCNC(c2cc(CC3CCCCC3)on2)=O)C1 Cc1cccnc1C=CC(N1CCC(NC(=O)CCc2cn(C)cn2)CC1C)=O N1(C(c2ccc(C)c(F)c2)C2CC2)CCn2ncc(SC(F)F)c2C1 N1(C(c2cc(Cl)cc(Cl)n2)C(=O)NC(CC)(C)C)CCC(C2CCCC2(C)C)C1 CC(C)C(C(=O)OCC)NC1(C)CS(=O)(=O)C1.S(=O)(=O)(C1CC1)NC N1(C(CCNC(=O)NC2CC2)=O)CCOCC(C(=O)NCC2CCC(F)(F)C2)C1 C(CCCCC(=O)NCC1CCN(C(=O)C=Cc2ccccc2)C12CC2)SC C(=O)(C1=CC2(CCOC2)C1)N1C(C)CC(NC(=O)CC2CC(=O)C2)CC1 C1(C)(CC)C=C(C(=O)NC(C(=O)N(C)CC)C2CCC2)C1 CC1(C#CC(=O)NCC23CC2CN(C(=O)C(c2cc(Cl)cc(Cl)c2)=O)C3)CC1 C1(NC(C(C2CN(C(C(C3CCCC3)OC)=O)C2)OC)=O)CCCCC1 C1(CC(=O)NCC2(F)CN(C(=O)COCCc3ccccc3)C2)CC=CCC1 C(=O)(CC(CC)C(C)C)NCC(CCCC)NC(c1ccsc1Br)=O N1(C(COC2(C)CCC2)=O)CC2(CC(C(=O)N(CC3CC3)CC3CC3)CO2)C1 N1(C(C)=O)CCCC(C)C1CNC(=O)CCc1ncc[nH]1 c1(OC)ccc(CCC(=O)NC(C)CN(C(=O)CC2CCCCO2)C)cc1OC C1(C(=O)NC2C=CC(CC(=O)NCCOCCC)C2)CC2OC1C1CC21 N1(C(c2c(CC)nccn2)=O)CC2CC1CN2C(=O)Cc1cccc(C(N)=O)c1 C1(C)(C(N2CCCC(CN(C(C(C(=O)NC)(C)C)=O)C)C2)=O)CCC(C)C1(C)C N1(C(C2C(C=C)CC2)=O)CCN(C(c2ccc(CNC(N)=O)cc2)=O)C2(CC2)C1 Cc1ccc(S(=O)(=O)NCC2CC(OC(C)(C)C)C2)c(C#N)c1 C1(C(=O)NC2CCN(C(c3nc(NC(C)=O)sc3)=O)CC2)CCS(=O)(=O)C(C)C1 N1(C(C2(C(=O)OC)CC2)=O)CCCC(NC(=O)Cn2ncn(C)c2=O)C1 Cc1ccc(OCc2nc(CC3CC=CCC3)n(-c3ccccc3)n2)cc1 Cc1cccnc1-n1cc(-c2ncccc2C)nn1 C1(NC(C(=O)NC(C)C)=O)CCN(C(=O)C(c2ccccc2F)N(C)C)CC1 N1(C(CC(C)(C)O)=O)CCC2(CCC2)C(NC(C2CCC(=O)NC2)=O)C1 N1(C(C2C3CN(C(=O)Cc4ccc(F)cn4)CC32)=O)CC2CCC(C1)O2 c1(C(N(CC(CN(C(C(CC)F)=O)C)O)C)=O)cc(OC)ccc1[N+](=O)[O-] c1(C(=O)NCC(CNC(C2(CSC)CC2)=O)C)cccc(C2OCCO2)c1 c1(C(=O)NCC(CCOC)NC(C=COCC)=O)cc(OC)c2c(c1)CC(C)O2 c1(OCC)cccnc1C(=O)NCC1C2CN(C(=O)CC3CCC(F)(F)C3)CC12 C1(C(C(=O)NCC(CC)CO)(C)C)CCCN(C(c2cscc2C)=O)C1 N1(CC(N2CCC(CNC(c3c[nH]cc(C)c3=O)=O)C2)=O)CCc2sccc2C1 C1(C(=O)NCC(COC)(C)CO)CCOCCN1C(=O)Cn1ncnn1 c1(CC(N2C(CN(C(=O)CC3(N(C)C)CC3)CC)CCC2)=O)ccccc1O C(c1ccncc1)=CC(=O)NC12CC(CNC(C(C)OCC(F)(F)F)=O)(C1)C2 CCCC(C)(O)CC(=O)NC(CC(=O)NCCc1cnc(C)cn1)C1CC1 c1(C(=O)NCCC2N(C(C(CC=C)C)=O)CCC2)c[nH]c2cccc(F)c12 C1(C)(CNC(c2c(C)nn(C)c2)=O)CCC(NC(C2CC2c2cnc[nH]2)=O)CC1 C1(NC(C2CCC(=O)NC2)=O)CCS(=O)(=O)C12CN(C(=O)CCC[N+](=O)[O-])C2 c1(N2CCC(C(F)(F)F)C2)nc(N2CCC3(C=CCO3)CC2)nc2c1CSC2 c1(C(C)NC(c2c(CC)cncc2)c2nnnn2C2CC2)ccc(Br)c(C)c1 C12(CNC(CC=C=C)=O)COCCN1C(=O)CN(C(c1cccc(Cl)c1F)=O)C2 N1(C(C2(C)CC=CCC2)=O)CCCC(C(=O)N(C2CC2)C2CC2)CC1 C(=O)(CC(C)(C)F)NCC1C(NC(c2cc(OC)ns2)=O)CCC1 C1(NC(c2csc(Br)c2)=O)CCN(Cc2cc(Br)c[nH]2)CC1F C(=O)(C1CCCc2nc(C)[nH]c21)N1CCN(C(c2nccc(C)c2)=O)CC12CC2 O=C(CCC1=CCCCC1)NCC(C1CC1)NC(c1ccsc1)=O C1(C(=O)NC(C2CN(C(c3cnc(SC)s3)=O)C2)C)COC2COCC12 c1(C(N2CCN(CCNC(CCC#N)=O)CC2)=O)cc(F)cc2nc[nH]c12 c1(CC(=O)N(CC(CN(C(Cc2nnc(C)o2)=O)C)O)C)ccc(C)c(C)c1 C1(C(N2CCCN(C(c3ccc(C)nc3C)=O)CC2)=O)CC2CSCC(C1)C2 c1(C2(C(=O)OC)CC2)ccc(-c2ccnc(NCc3ccc(F)cn3)c2)cc1 N1(C(C2C(C)OC(C)C2C)=O)CC2(C)CN(C(=O)C3=CCCO3)CC2(C)C1 N1(C(CSSC)=O)CCC(N=c2[nH]c(-c3ccccc3)nc3c2CCC3)C(C)C1 c1(OC)ccc(CCC(N2CC(CNC(C3CCC3)=O)C(C(F)(F)F)C2)=O)cc1 C(C(C)C(=O)NC1COCC1NC(c1csc(Cc2ccccc2)n1)=O)OC c1(OC)ccc(C(=O)NCC2CN(C(=O)C=CSC)CC2C(F)(F)F)c(C)c1 C12(CNC(=O)COCC3CCCC3)CC1CN(C(c1ccc[nH]1)=O)C2 N1(C(CC)=O)CC(NC(c2csc(Br)c2)=O)CC12CCCCCC2 N1(C(c2c(CC)oc(C)c2)=O)CCN(C(=O)C(C)(COC)COC)CC1C N1(C(c2nc(C)c(C)[nH]2)C)CCC(O)(Cc2cn(C3COCC3O)nn2)CC1 CC1CCCN(C(=O)C=Cc2cnn(C)c2)C1CNC(=O)CCCC#N C(=O)(C(O)CCC(C)C)NC(C(=O)NC(CC=C)CO)CN=[N+]=[N-] C(C(C)(C(=O)NCC1C(C)CCN1C(c1ccn(CCO)c1C)=O)OC)OC c1(N2CCC(C=C)CC2)[nH]c(=NCc2c[nH]nc2C2CCCCC2)nc2scnc12 n1(CC(=O)NCC(C)(Cn2cccn2)OC)ccc2c(C)cccc12 c1(NC(N(CC(O)C2CC2)C)=O)ccc(N2CCOCC2)nc1C C(=O)(CCCCCCCC1CC1)NCc1cn(CCN(CCCN(C)C)C)nn1 C1(C2CCN(C(=O)Cn3ccnn3)C2)(NC(C(C)C(C)(F)F)=O)CC1 C1(C(N(CCCCN(C(c2c(C)[nH]c(C#N)c2)=O)C)C)=O)CCCC1S(C)(=O)=O c1(CC)nn(C)c(CC)c1C(=O)N(C)CC1CCCN1C(=O)CSC(C)C C1(C(C)C)COCCN(C(C2CCC2NC(C2(C)CC3CCC2O3)=O)=O)C1 C1(C(=O)NCc2c(COC)noc2)CN(C(=O)CC(C)(F)F)CC12CC2 C(CCN=c1cc[nH]cc1S(=O)(=O)NCC1CCOC(C)(C)C1)OCC c1(N2CC(NC(CCC(C)SC)=O)(CO)C2)ccnc2ncnn12 CCCCCCCC(=O)NC(C1CN(C(=O)CC2CC(F)(F)C2(F)F)C1)C CCC(CC(=O)NC1(C)CCN(C(=O)CCn2ccnc2C)C1)C(C)(C)C N1(Cc2ccc(C)o2)CC2CCN(S(=O)(=O)c3ccc(O)cc3)CC2C1 c1(CC)ccc(O)c(C(=O)NCC(CC(C)C)NC(c2cccc(C)c2F)=O)c1 Cc1ccc(OCC(N2CCN(C(=O)CC3(C)CC3)C3CC23)=O)c(Br)c1 C1(CC)C(N)CCCN1Cc1ccc(N2CCCC2)o1 CC1CN(C(c2cc(F)c[nH]2)=O)CCCN1C(c1c[nH]c(=N)o1)=O Cc1n[nH]c(C)c1CCC(=O)NCC1CCCN1C(C1CC1c1cccnc1)=O c1(NCCNC(=O)OCC(C)(C)C)ccc(OC(F)(F)F)cc1.ON c1(C(N2CC3C(NC(C4CCC(CC)CC4)=O)(C3)C2)=O)nccc(Cl)c1O C(=O)(CS(=O)(=O)C(C)(C)C)NC(C)CC(C)NC(C1(c2ccccc2)CCC1)=O C1(CC(N2C(C)CC(CNC(C3(C)C(C)CCC3)=O)C2)=O)CN2CCC1CC2 Cc1c(C(N2CC3CC(NC(c4ccccc4Cl)=O)C2C3)=O)cnc2ncnn12 CCC1CN(C)CCNC(=O)C1.C(C)(CCC(C)(C)C)OC(C)(C)C CCCC(C(F)(F)F)NC(=O)CC1CCCN(C(=O)COC2(C)CCC2)C1 Cc1n[nH]c(C)c1C(C)CC(=O)NCC(F)CNC(=O)CNC(c1ccco1)=O Cc1ccc(C(=O)N(C2CN(C(=O)CCCC(C)(F)F)C2)C)c(N)c1C C12(NC(C(CCC#C)O)=O)CC3CC(C1)CC(CNC(c1ccnn1C)=O)(C3)C2 Cc1ccc(CC(N2CCN(C)CC2CNC(=O)COCC(F)F)=O)c(F)c1F C(=O)(C(C)C(C)(F)F)NCCC(C)NC(c1ccc(-c2cnc[nH]2)cc1)=O N1(C(c2cncc(F)c2C(F)F)=O)CC2CCC(C1)N(C(=O)C=CC(F)(F)F)C2 C#CCCCCCCC(=O)NC1(C(N2CCOC(C)CC2)=O)CCOCC1 C1(C(=O)NCCCN2C(C)CCCC2)CN(C(c2cncc(O)c2)=O)C(C)(C)C1 C1(C2CC2)(C(=O)NCCc2cc(C(N(C3CCN(C)CC3)C)=O)no2)CC(=O)C1 CC1(C)CC(CCNC(=O)CC2(NC(=O)CCc3cccn3C)CC2)CO1 c1(C(N2CC(COC)N(C(=O)CCCCCF)CC2)=O)ncnc2c(C)csc12 CC12CC(NC(C3CC4CCC(C3F)N4C(=O)CNC=O)=O)(C1)C1(CCC1)O2 c1(C(=O)NCC2(C)CCCN(C(C(C)OCCCC)=O)C2)cn2c(n1)CCCC2 N1(C(C(COC)(C)O)=O)CC2CC(NC(c3ccc(OC)nc3Cl)=O)CC2C1 N1(C(C2(C)CCCN(C(C(CCSC)(C)C)=O)C2)=O)CCOC2(CCC2)CC1 c1(C(C)C(=O)NCCOCCN(C)C(C2CC2(F)F)=O)ccc(Br)s1 c1(C(N2C(C)CC(CNC(c3ncc(C)nc3)=O)C2)=O)cc(N)cc(N)c1 C=CCC(CNC(=O)CCNc1ccccc1)NC(=O)C=C(Cl)Cl c1(CNC(C(C)OC(C)=O)=O)ccc(C(N2CCC2(C)C(C)C)=O)s1 c1(OCC(=O)NC(CC(=O)OC)C)cnc(SC)nc1O N1(C(C2=NOC(CNC(C(COCC)N=[N+]=[N-])=O)C2)=O)CCn2cc(C)nc2C1 C1(C)(CC)C=C(C(=O)NC2COCC2NC(c2ccc(F)cc2)=O)C1 C1(C(=O)NCC(CC=C)NC(=O)C=C2CCCC2)CCN(c2nncs2)CC1 C(CCC(C)C(=O)NC1CCCC(NC(=O)CCCNS(C)(=O)=O)C1)OC CCC(CNC(=O)CCCn1cc(-c2ccc(C)cc2C)nn1)CC(F)F C1(C(N2CC(NC(C=CCOC)=O)C(C(F)F)C2)=O)CS(=O)(=O)CC(=O)N1 S(=O)(=O)(c1ccc(NCCSC(C)C)nc1)NC1CC(OC)C1(C)C Cc1cc(C(=O)NCC2CC3CC3N2C(=O)COCCCF)n(C)n1 C1(C(=O)NCCC#CCO)(CNC(c2cc(CCO)on2)=O)CC2(CC2)C1 Cc1cc(C(=O)NC2CS(=O)(=O)CC2NC(c2sccc2C(F)F)=O)cc(O)n1 C1(C(=O)NCC(C)(CNC(=O)C2=C(C)CC2)OC)CC(C)(C)C(C)(C)C1 Cc1csc(CCNC(=O)C(CNC(c2c[nH][nH]c2=N)=O)N(C)C)n1 c1(N(C(N2CCCC2)=O)CC2CC(C)OCC2)csc(N=S(C)(C)=O)n1 c1(C(C2(NC(=O)NC3(C(C)C)C(CC)C3)CC2)OC)ccc(C#N)cc1 CP(C)(=O)c1cnn(CC(=O)NCCOc2cc(Br)ccc2C(N)=O)c1 C(C(C)N=c1cccc(S(=O)(=O)NCC(c2ccccc2)(C)C)[nH]1)N(C(C)C)C N1(C(C(C)SC)=O)CC2(CC(C(=O)NOCC(F)(F)F)CO2)C1 N1(C(c2c(OC)cc(C)cc2)=O)CC2CCCC(CNC(=O)C(C)OC)(C2)C1 N1(CCC(=O)N(c2ccc(C)c(C(=O)O)c2)CCSC)CCC2(CC1)OCCO2 C1(NC(C2(C)CS(=O)(=O)C2)=O)CCC2(CCCN(C(c3cc(Cl)c[nH]3)=O)C2)C1 C#Cc1cncc(NC(=O)C(CCF)NC(=O)Cc2cn(C)cn2)c1 c1(C(N2CC(C(C)NC(=O)Cn3cnnn3)C2)=O)cccn2c(O)nnc12 CC(C)C(F)C(=O)NC1CC(NC(c2ccc(SCCCO)cc2)=O)CC1O c1(C(=O)NC(C(C)OC)C(=O)NCC2(CC3CC3)CC2)ncc(C)cc1C C1(NC(c2ocnc2C(F)F)=O)CCN(C(C2CCCC23CC3)=O)CCC1CO C(=O)(CC(O)CC(C)(C)C)N(CC(=O)NC(c1cc(C)on1)C)CCOC C1(CN(C)C(=O)NC2(C(F)(F)F)CC(O)C2)CCC2CC2C1 C1(CNC(c2scc(OC)c2)=O)CCCCN(C(=O)Cc2cc(C)cc(F)c2)C1 c1(CNC(C2(F)CN(C(CC(CC)SC)=O)C2)=O)ccc(C(C)C)cc1F c1(C(N2C(CNC(c3c(C)ccs3)=O)CC(F)C2)=O)cc2c(Cl)cncc2s1 C1(NC(CC(CCC)O)=O)CN(C(c2ccsn2)=O)CC(F)(F)C1 C(=O)(C1Cc2ccccc21)N(C(=O)C#CC1CC1)C(CN(CC)CC)C C(=O)(CCC(F)(F)F)NCCC1(C)CCN(C(c2c(C(C)C)ncnc2)=O)C1 C1(C(=O)NCC(=C)Br)COC2(C1)CN(C(=O)C(C)=C(C)CC)C2 N1(C(Cc2ccc(C)o2)=O)CCC(C)N(C(c2n[nH]c3c2COC3)=O)CC1 c1(C(=O)NCC2(NC(C(C3CCC3)OC)=O)CCC2)ccc(Cl)cc1 Cc1nc2ncc(C(=O)NC3CC3CNC(=O)C(C)Cc3ccccn3)cc2o1 c1(C(N2CCC(NC(C3C=C(C)CS3)=O)CC(F)C2)=O)ccc2[nH]nc(Cl)c2c1 N(C(=NCCC1COC(C)(C)OC1)NC(CC)CC)CC1C(C(=C)C)CNC1 C12(C(=O)NCCCNC(C(CCO)N(C)C)=O)CCC(C(F)F)(CC1)CC2 c1(NC(N2CCC2C2CCOC2)=O)ccc(F)c(F)c1 C1(C(C(=O)NC(C)CC2(NC(c3occc3C3CC3)=O)CCC2)C)CCOCC1 c1(OC)ncc(NC(C2CC23CCN(CSC)C3)=O)cc1CO.c12ccc(o1)C2 S(=O)(=O)(c1c[nH]ccc1=NCCCCc1ccccc1)NCC1(C)CCCO1 C1(C2(C(=O)NCCOCC)CC2)CCCN1C(=O)CC1CCC(C(F)(F)F)O1 c1(NC(CCOCCNC(CC)=O)=O)sc(C)nc1C C1(C(=O)OC2C(=O)NC3CC2C3)(OC)CCOCC1.C(C)(C)(C)OC(=O)NCCF CN=c1[nH]nc(CC(=O)NC2CC2NC(c2ccc(SC)cc2)=O)s1 C1(O)(CCn2cc(CCS(N)(=O)=O)nn2)CCCN(C(=O)C2=NOCC2)CC1 C(=O)(C#CC1CCCCO1)NCC1OCCC(NC(c2c(Cl)cnc(C)n2)=O)C1 N1(C(=O)CC2COCCO2)CCC2OCCN(C(c3cccnn3)=O)C2C1 N1(C(CCC2(C#N)CCC2)=O)CC2CCC2(C(=O)NC2CC(CO)C2)C1 c1(C(=O)NC2(C3CN(C(C4C(C(C)C)C4)=O)C3)CC2)ncccc1N=[N+]=[N-] C1(C(=O)NC(C=C)CO)CN(C(=O)CCCNC(C)=O)CC1C=CC CC1CCN(C(C2CCCN(C(c3cc(=O)cc[nH]3)=O)CC2)=O)CC1(F)F c1(C(N2CCC(C)(CNC(c3cc(F)c[nH]3)=O)C2)=O)ccc(O)c2c1CCCC2 c1(C(N(C2CCCN(C(CC)=O)C2)C)=O)cccn2c(O)nnc12 C1(C(=O)NCC2(OC)CN(C(C3CC(C)(C)CN3C)=O)C2)CCS(=O)(=O)C(C)C1 C1(CC(N2CCCC2(C)C2CCOCC2)=O)(NC(=O)OC(C)(C)C)CC(F)(F)C1 Cc1nc(N2CCOCC2)sc1CC(=O)NC1(CC(F)F)CC1 c1(C(N2CCC(NC(c3cc(Cl)cnn3)=O)C(O)C2)=O)ccn2ccccc12 c1(C(N(C2CCN(C(c3cc(CCC)n(C)n3)=O)C2)C)=O)[nH]cc2c1CCCC2 c1(CC)cc2c(NCC3CCCC3NC(C3(O)CC(C)(C)C3)=O)nc(C)nc2s1 Cc1ccc(F)cc1C(=O)NC(c1nocc1C(=O)NC1CCCCCCC1)C CCCCCCCCCn1cc(CN2CCCC(F)(F)CC2)nn1 N1(C(c2ccn(CCOC)n2)=O)CCC(NC(c2cc(F)n[nH]2)=O)C1C1CC1 S(=O)(=O)(c1cc(C(=O)NC2CC(CCNC(C3(C)CCC3)=O)C2)c(C)o1)NC C1(NC(C(Cc2ccc(OC)c(O)c2)N)=O)CCOC2(CCS(=O)(=O)CC2)C1 Cc1nc(C#N)cc(=NC(C)CC(C)NC(C2(C)CCCCC2)=O)[nH]1 C1(NC(C2CCCN(C(CC3CCC(C)NC3=O)=O)C2)=O)CC2C=CC1C21CC1 n1(CC(=O)N(CC(CNC(C(CC)(F)F)=O)C)C)ncc(C)cc1=O c1(C(N2C(C(C)NC(c3nccc(C#C)c3)=O)CCC2)=O)ccn2cccc2c1 CCCCC(C)C(=O)NCC(CNC(c1ccc(Br)cc1Cl)=O)CO C12(C(=O)NCC(CNC(C(C(C)C)n3cccc3)=O)C)CC(C)(C1)OC21CCC1 CC1(C)COCC1CNC(=O)NC1CC1c1ccc(C(F)(F)F)cc1 c1(N(C(=O)CSC2CCSC2)CCN(C)Cc2cnn(C)c2)cc(O)ccc1F C1(C(N(C)CCC2CC2)=O)CC(CCNC(=O)COC2CCC2)C1 Cc1cc(F)ccc1S(=O)(=O)N(CC1OCCCO1)CC1(C)COC1 c1(C(=O)NCC(C)NC(C=C(C)c2ccsc2)=O)cc2c(ccn2C)[nH]1 N1(C(CSCC=C)=O)CC2CC2(CNC(C2CC(C(F)F)C2)=O)C1 N1(C(CC#C)=O)CC2CCC2(CCNC(c2ccsc2Cl)=O)C1 C(=O)(C(CO)C(F)(F)F)N1CC(CC)(NC(c2cncnc2C2CC2)=O)C1 C1(CC(=O)NCC2(CNC(CCc3ccn(C)n3)=O)CCC2)CCOC(C)(C)C1 C1(OCC(=O)NC2(COC)CCC2)CCN(C(c2conc2C2CC2)=O)C1 c1(C(C(=O)NCC2CN(C(C=NOC)=O)C2)O)cccc(Cl)c1 CCCCC(C)(F)C(=O)N1CC(CCNC(C2CC23CCCC3)=O)(OC)C1 Nc1cc2c(cc1C(=O)NCCCCCNC(=O)CCc1cncnc1)OCO2 N1(C(C2(CC)CCN(C(C3CCN(C)CC3)=O)C2)=O)CCOC2COCC12 C(=O)(C(C)(C)C(=O)N1CCC(CC(=O)NCC2CC3(CC3)C2)C1)OCC c1(C(N(C2CCS(=O)CC2)CC)=O)cccc(-c2ccccc2CN(C)C)c1 N1(C(=O)NC(c2scc(C(=O)OC)n2)C)CCOC(c2cccc(O)c2)C1 N1(C(C(C)(C)OC(C)C)=O)CCCC(CCC(=O)NCC(C)CC2CCC2)C1 C1(NC(CCNC(CCP(C)(C)=O)=O)=O)CCn2ncnc2C1 C(CNC(=O)CC1CC(CF)C1)(C(C)(C)C)NC(c1ccn(CC(C)C)n1)=O Cc1nc(CC(=O)N(CCC(C)NC(C2CCCO2)=O)C)c(Cl)s1 c12ccnc(c1)C(=O)N(C)C2.C1(C(C)(F)F)(C(=O)NC2(CO)CC2)CCC1 c1(C(=O)NC(CC)CNC(=O)C(c2c(C)n[nH]c2C)C)cc2ccnc(Cl)c2[nH]1 c1(CC(=O)NC(C)CC2CN(C(=O)CC3CCC4CC34)C2)c[nH]c2ncccc12 C1(C(=O)NCCC2(O)CCN(C(c3cccnc3O)=O)C2)CN2CCCN1CC2 S(=O)(=O)(c1c(OC)noc1CC)NCC1(F)CC(C(=O)OCC)C1 CC1CCN(C(=O)Cn2nncc2N=[N+]=[N-])CC1N(C)C(c1cccc(Br)c1)=O CCCCCCC(=O)NC(CCC1CCC1)C(N1CC(S(C)(=N)=O)C1)=O N1(C(C2C(OCC)CC2)=O)CC2(CCN(C(c3cnc(O)n(C)c3=O)=O)C2)C1 c1(C(C(C)NC(C(=O)Nc2ccc(OC)cc2OC)=O)O)ccc2c(c1)OCO2 C(C(C(=O)OC)n1cc(CNC(=O)NC)nn1)OCC.c1(C(=O)NCC)scnc1C C1(CNC(C(C)SCC)=O)CC2(CO1)CN(C(c1c(Cl)nn(C)c1C)=O)C2 C(=O)(CC1=CCCC1)NC1CCC(NC(C(CC)(O)c2cccc(Cl)c2)=O)CC1 C(=O)(C#CC1(C)COC1)N1CCCC(C)(C(N2CC(C(CC)C)C2)=O)C1 C1(C(N2CC(C(c3ccccc3)C)C2)=O)Cc2cc(F)ccc2O1 c1(C(N(c2nc(OC)c(C)cn2)C2CNCC2F)=O)cc(F)cc(F)c1OC N1(C(CCNS(C)(=O)=O)=O)CC(CO)(NC(c2cncnc2)=O)C1 c1(C(=O)NC(C2(C(=O)NC3CC(N4CCC4)C3)CC2)C)cccnc1 C(c1sc(Cl)nc1Cl)=CC(=O)NCC1C2CN(C(CNC(=O)NC)=O)CC21 c1(C(N(CCCCN(C(=O)C(F)CC2CC2)C)C)=O)cnc(O)cc1C(F)(F)F c1(C(=O)N(C2CC2)Cc2ccccc2)cc(O)ccc1C(F)F C(=O)(C1=Cc2ccccc2C1)NC1CC(C(=O)NC2CN(c3ccncc3)C2)C1 C(CCCC(=O)NCC12CC(CO1)C2)NC(C1(C)COC1)=O Cc1c([N+](=O)[O-])c(C(=O)NCCc2cnc(C3CC3)nc2)nn1C C1(CNC(C(OC)OC)=O)COCCN1C(=O)Cn1cc(-c2ccccc2)cn1 C12(NC(C3C(C)C3C)=O)CCC1CN(C(=O)CCc1cc(Br)ccc1F)C2 CC1CN(C(=O)CC2CN(Cc3cccc(-n4cncn4)c3)CCO2)CC(=O)N1 C(=O)(C(CC=C(Cl)Cl)c1ccccc1)N1CC(C(CC)CC)C1 C(C)(CC(=O)N1CCC(CN(C)C(c2c[nH]nc2C(F)(F)F)=O)C1)OC C1(C(N2C(C3(NC(Cc4c(C)occ4)=O)CC3)CCC2)=O)CCC12CCC2 N1(CC(C)C)CCC(C(=O)NCC(C)CN(C(=O)Cc2nccn2C)C)C1 C12(CNC(Cc3cc(COC)on3)=O)CC1CN(C(=O)CCNC(C)=O)C2 c1(NC(C2N(c3cc(SC)ncn3)C3C(C2)C3)=O)cc(F)c(O)cc1Cl n1(CC(=C)C)nnnc1C(CCOC)(C(c1noc(C2CC2)n1)OC)OC CCCC(CNC(=O)C(CC)CCOC)C(=O)N1CCC(NC(N)=O)CC1 C(=O)(CCn1cccn1)NC(C1C(C(N(C(C)(C)C)CCN)=O)C1)=O c1(CN(C)Cc2nc(C)c(Br)s2)cccnc1[N+](=O)[O-] C1(NC(Cc2c(CC)cc(F)cc2)=O)CN(C(=O)CC2CC2)C2(CCC2)C1 N1(C(C(C2(C)CC2)NC(=O)COCC(F)F)=O)CC2CC2(CO)C1 Cc1nn(C)cc1CN1CC(NC(=O)C(c2cccc(Cl)c2)(C)C)C(F)C1 c1(CC)ncncc1C(=O)NCC12CC1CN(C(=O)C(=Cc1cccnc1)C)C2 C(=O)(CCCC(N)=O)NC1(C)CCN(C(Cc2c(C)cco2)=O)C1 C(=O)(C(C(=O)NC1CCN(C(=O)C(C)(CC)CC)CC1)OC)OCC C#CC12CCC(NC3CCN(C(=O)OC(C)(C)C)C4CCC34)(CC1)CC2 CCCC(CC)CC(=O)NCCC(F)Cn1cc(-c2ccc(C)cn2)nn1 c1(C(=O)NC2CC(CNC(CC(=C)C)=O)C2(C)C)ccc2cc(O)ccc2n1 N1(C(c2c(CC)ocn2)=O)CCC(F)C(NC(C2(C)CCN(C)CC2)=O)C1 C1(NC(CC=CC=C)=O)(CC)CCCN(C(C2CCC3CC2CO3)=O)C1 N1(C(C2CC23CC3)=O)CCCC2CN(Cc3nnc(-c4ccccc4F)s3)CC12 C=CC1CN(C(=O)CN2CCCCC2=O)CC1NC(=O)CCc1cn(C)cn1 N1(C(c2c(C)nc(C)o2)=O)CCCC(C)(CNC(=O)C(c2ccccc2)F)C1 C1(N(C(=O)CN2CC3CC3C2)C)CN(C(c2cc(C(F)F)nn2C)=O)CC1F CC(C(=O)NC(C)(CNC(c1cc(C(C)C)cnc1O)=O)CO)C(F)(F)C(F)F c1(OCC=C)ccccc1C(=O)NCC(F)CNC(C1C(C)(C)C1(C)C)=O CCC(C)C(C(=O)N1CC(CC(=O)OC)C1)N(C)C(c1cnsc1C)=O c12ncccc1[nH]c(=O)[nH]2.O=C(CC(C1CC1)C1CC1)NCCC1CCC2CC12 c1(COC)cnc(OC)c(C(=O)NC2COCC2NC(C2C=CCCC2)=O)c1 c1(C(N2CCN(C(c3ccc(OCF)nc3)=O)C3CC23)=O)ccc(O)c(O)c1 CC(C)(C(=O)NC1CC(CCNC(c2ccc(Br)cn2)=O)C1)C(F)(F)F C12(NC(CNC(C3C(C)C3)=O)=O)CC(C(=O)NC3(CCO)CCC3)(C1)C2 N1(C(CONC(c2c(C)ocn2)=O)=O)CC=CC1(C)CO c1(C(N(C2CCN(C(c3cc(C(N)=O)[nH]n3)=O)CC2)CC)=O)cc(Cl)c(Cl)[nH]1 CC(c1cccc(Br)c1)=CC(=O)NC1CN(C(C2CC2F)=O)CC1(C)C C1(NC(c2c(SC)ccs2)=O)CCC2CC1CN2C(=O)CC1(O)CCCOC1 C=CCC(CC=C)C(=O)NC1CCN(C(C2CCOCC2)=O)C12CCC2 C(N=c1nc2ncn(C)c2c(NCc2cccnc2Cl)[nH]1)c1cccc(C)c1F C1(COC)(CNC(C2CC23CC(O)C3)=O)CCCN1C(=O)C(C)(C)F c1(OC)ccc(C2CSCCN2C(=O)CCCN2CCOC2=O)cc1 C(=O)(CC(C)C(=O)N1CCN(Cc2cn(-c3ccc(F)cc3Cl)nn2)CC1)NC c1(C(N2CC(CC(C)NC(c3cc(Cl)c[nH]3)=O)C2)=O)ccc2[nH]nc(O)c2c1 C1(NC(CC=C)=O)CN(C(c2nnn(Cc3ccncc3)c2C)=O)CC(C)(C)C1 CC1CN(C(c2sccc2Cl)=O)CCC1NC(=O)Cc1cnn(C(F)F)c1 N1(C(C=C(CCC)CCC)=O)CCN(C(C2(C)SCCCS2)=O)CC12CC2 C1(C)(C(N(CCC(N)=O)C)=O)C=CCN1C(=O)COCC1CC1 CCCCC(C)CCC(=O)NCC1C=CC(NC(c2ccoc2Br)=O)C1 c1(OC(=O)NCCC2C(CCN(C)C)COC2)cccc(F)c1 c1(OC)nccc2c(C(=O)N(C)CCNC(c3cc(C#N)c(C)cn3)=O)c[nH]c12 N1(C(Cc2c(C)ocn2)=O)CCC2(CC1)CN(C(=O)C1=CCCCO1)CC(C)O2 c1(C(N2CC(C)SCC2)C(=O)NCc2nnn(C)n2)ccc2c(c1)OCCO2 N1(C(CC(C)SC)=O)CCC(C(=O)NC2C(=O)N2)C1.C(C)(C)OC1CC1 Cn1nnc2c(C(=O)NC3CCN(Cc4ccccc4Cl)CC3(C)C)ccnc12 c1(CC)ccc(C(N2CCCC(NC(=O)CCC(C)CN(C)C)C2C)=O)c(O)c1 N1(C(CC2(CNC(CN(CCC)C)=O)CC2)=O)CC(CO)CC1CO c1(C(=O)NC2CC(CCNC(CC3CC(=C)C3)=O)C2)conc1C(C)C c1(C(=O)NC2CC3CN(C(C(C)(C)CC#N)=O)C2C3)ccc2ncnn2c1 CC1(CCC(=O)NCC(=O)NCC(=O)NC2CC2)CN(C(=O)CC(N)=O)C1 C1(C(=O)NC(c2ccccc2)CNC(C(C)NC(CC)(C)C)=O)CC(C2CC2)C1 C#Cc1cc(C(=O)NC2CCC(C)N(C(=O)C=Cc3cnc(C)s3)C2)ccc1Cl CCC(CC(=O)N1CCN(C(c2cc(C)nc(O)n2)=O)C(CF)C1)C(F)F C1(C(N(CCNC(C(c2cncnc2)C)=O)C2CC2)=O)CCCC(C#N)C1 CC(C)CC(CNC(=O)C(N1CCCCC1=O)C)NC(=O)C(c1ccccc1)=O CC(C(=O)Oc1ccc([N+](=O)[O-])cc1)C(=O)NNc1nc(Cl)ncc1Br c1(C(=O)NCC(CCCC)NC(c2ccncc2)=O)[nH]cc2c1CCC2 C(=O)(C(C)(CCC)CCCCCC)NC1CC(NC(C2C(C=C)OCC2)=O)C1 N1(C(Cc2c(C)nsc2)=O)CC2CCCN(C(C3CC4C=CCC(C3)C4)=O)C2C1 c1(OC)cccc2c1C(C(=O)NCC1CSCCS1)CC2 C1(CNC(C2CC(C(C)C)OC2)=O)CC12CCCCC2 C(c1cnn(C)c1)=C(C(=O)NC1CCC(CNC(c2c(CCC)[nH]cc2)=O)C1)C c1(CCC(=O)NCCCOCCC(=O)N(CC(C)C#N)CC)nc(C)cs1 C(CC1=CCN(C(c2c[nH]nc2C(C)(C)C)=O)CC1)NC(C1(C)ON=C(C)C1)=O C1(NC(Cn2cc(CNC(C=C(C)C(F)F)=O)nn2)=O)CC2(C1)CC(C)C2 N1(C(C2CCN(C(C)=O)C2)=O)CCOC(CNC(=O)C(F)(F)c2cnccn2)C1 C1(C(N2CC3C(CNC(c4cc(C)[nH]c4C)=O)C3C2)=O)CCCCC1(C)C C1(CC)CN(C(c2ccccn2)=O)CCC1NC(c1ccc(OC)s1)=O C1(OCC)CC2(C1)CC2C(=O)OC(C)C.C(C1C(=O)S1)NC(C)=O.OCC NS(=O)(=O)c1c[nH]c(C(=O)NC2CC(C(=O)O)C2)c1 c1(NCC(N2CC(O)(CCNC(CC3(C=C)CCC3)=O)C2)=O)ccccc1C c1(OC)ccc(C(=O)NC2CCCC(NC(=O)CC3CCC3)C2)c(C)c1 C(C(C)(C)CC(=O)NC(C)CC(=O)NCC1CCC2(CC2)CO1)OC C(=O)(C1CCc2c[nH]nc21)NC(CCNC(C(=Cc1ccccc1)CC)=O)C C1(NC(CN(S(CC)(=O)=O)C)=O)CCC(C)(CNC(C2(C(F)(F)F)CC2)=O)C1 N1(C(C(C)OC)=O)CCC2(C(=O)Nc3cccc(F)c3C(C)C)CCCC12 CC1CC(NC(C23CC(C(F)(F)F)(CO2)C3)=O)CN1C(=O)C=CC1CCCCC1 C(c1cccnc1)=C(C)C(=O)N(CCN(C)C(C1(C)CC1F)=O)C(C)C N1(C(Cc2n(C)nnc2)=O)CC2CCC2(CCNC(=O)CC2(CO)CC2)C1 CC(C(=O)N(CCCN(C)C(C1CC(N2CC(O)C2)C1)=O)C)C1CCC1 c1(C(=O)NCC2(F)CN(C(CCCCNC(N)=O)=O)C2)cc2cc[nH]c2cn1 c1(NC(C)=O)cccc(C(=O)NC(C2CCCCN2C(=O)C(C)C)C)c1 N1(C(C=Cc2c(C#N)cccc2)=O)CCC2C(CCN2C(C2CC2C(F)F)=O)C1 C(COCC)(C(=O)NC1(CC)CCCO1)NC(CSCC#C)=O c1(C(CC(=O)NC2CC(C)(NC(CC(C)SC)=O)C2)C)c[nH]c2ccccc12 c1(C(N2CCOCC(NC(C=C(C)Cl)=O)C2)=O)cc2c(ccn2C)[nH]1 C(CCC(O)C(=O)NCC(C)(C)CC(F)F)NC(C(C)c1cccs1)=O c1(C(N2CCN(C(CN3C(=O)COCC3)=O)C3C2C3)=O)c(F)cc(F)cc1Cl Nc1cc(F)c(C(=O)N(CCNC(c2cn3ccncc3n2)=O)C2CC2)cc1Cl N1(C(c2cc(C)sc2)=O)CCCC(C)C1CNC(C1(O)CCCC1)=O c1(C(N(CC(CC)NC(C(C(CC)C)O)=O)C)=O)c(F)cc(C)cc1Br c1(CC)cc(C(N2CCC(COC)(NC(=O)CC(C)(C)N(C)C)C2)=O)cc(O)n1 C1(CC=C)CCCCN1C(C1C(C)CN1C(=O)C=CCC)=O C1(C(N2CC(C)CC(NC(C(CCC)NC(C)=O)=O)C2)=O)CC2C=CC1C21CC1 c1(OC(COC(C(CC#C)C)=O)C)ccccc1C#N Cc1c(F)ccc(C(N2CC(C3(NC(=O)CCC4CCOC4)CC3)C2)=O)c1C C1(NC(c2ccn(CC)c2C)=O)(CC)CCN(C(=O)C(C)S(C)(=O)=O)CC1 CCC(CC(=O)N1CCN(C(c2cc(C)ncn2)=O)C(CS(C)(=O)=O)C1)C(C)C C(=O)(CCCCCCSC)N(CC(CC)NC(c1cccc(C2CC2)c1)=O)C CCC(O)CC(=O)NC1CCC1NC(c1ccc(-c2ccc(C)cc2)cc1)=O CCC(CNC(=O)CC(C(C)C)NC(=O)CC(C)CCO)(CC)CO C1(NC(C2CN(C(=O)NC)C2)=O)CC(NC(C2CC(C(C)C)C2)=O)C12CCC2 N1(C(c2c(C)nc(C)o2)=O)CC2CCN(C(=O)C(F)(F)c3ccncc3)CC2C1 C=CCC(CC(=O)NCc1nc(C)c(C)s1)NC(c1cc(CC)no1)=O N1(C(C(CC(C)C)C)=O)CCCC(C2(NC(c3ncc(Cl)cc3F)=O)CC2)C1 c1(CC)c(C(=O)NC23CC2CCC(C(N)=O)C3)cnn1C(C)(C)C c1(C(N(CCC)N)=O)nc(O)c2cc(C)cc(C)c2n1 C(C(C)(CC(C)C)NC(c1nsnc1O)=O)NC(Cc1c(C)cnn1C)=O CC1CCCn2ncc(C(N3CC(F)(CNC(=O)CCc4ncc[nH]4)C3)=O)c21 C1(F)(C(N(CC(C)NC(=O)C(c2ccc(Cl)cc2)(C)O)C)=O)C(C)(C)C1(C)C C(CCC)(C(=O)NC1CC(NC(=O)C(c2ccccc2F)C)C(O)C1)=CCC N1(C(C(CC)C(C)O)=O)CCCC(C2CCN(C(C3COCCO3)=O)CC2)C1 c1(C(=O)NC2CCN(C(CSCCCC)=O)C(C)C2)cccc2cccnc12 Cc1nc(CN(C(C)(C)C)C(C2CCCC2(C)C)=O)nn1-c1nc[nH]n1 C1(C(=O)NC23CC(C2)C3)(CC)CCCN(C(=O)CC2CCCOC2)C1 C(CN=c1cc(C)nc(N(C)CCC2CCCO2)[nH]1)c1n(CC)cnn1 C1(C(=O)NC2COCC2NC(C2CC=CCO2)=O)(NC(N)=O)CCCCC1 c1(C(=O)NC(CC)(C)CNC(c2cscc2C)=O)cc2c(cc1C)OCO2 C(C)(C)(CCC(=O)N1CC(=O)NCC1C(=O)NCCOCCC1CC1)OC C(=O)(CC(F)(F)C(F)F)N(CCCNC(=O)CCC(F)(F)F)CC c1(OC)cccc(C(=O)N(CC(C)C(=O)N(C)C(c2nc(C)no2)C)C)c1 C(=O)(C1=CC2(CCN(C(=O)CCc3csnn3)C2)C1)N(CC(O)C(C)(C)C)C c1(C(=O)NC(c2ccc(OCC)c(OC)c2)C)c(C)ccc(Cl)c1O C1(CCNC(=O)CCOC2(O)COC2)CCCN(C(C2CC2c2cccs2)=O)C1 c1(CC(=O)NC2C(NC(CC3ON=C(CC)C3)=O)C2)ccnc2ccccc12 CCC(CC(=O)N1CCC(C(=O)NCC(C)C(C)O)(C(C)C)C1)CC(C)C c1(NC(C(c2nc(CCCC)sc2)N(CC(C)SC)C)=O)cccc(Cl)c1 N1(C(C2CC(C#C)(O)C2)=O)CCC(NC(=O)C(CSC)OC)C(O)C1 Cc1sc(Cl)nc1C(=O)NC(CNC(C1(Cl)CC12CCC2)=O)C(C)(C)C c1(CC)ccc(O)c(C(=O)N(C)CC2CCCN(C(=O)C(=O)NCC(F)F)C2)c1 c1(OC)cc(-c2cncc(NC(=O)C(c3ccccc3)C)c2)ccc1O c1(C(=O)NC2(CC(=O)Nc3ccc(Cl)nc3Cl)CCC2)ccc(F)c(Br)c1 C1(NC(c2c(C)oc(Cl)n2)=O)CCN(C(=O)CCC(C)(C)C)C(C2CC2)C1 C(=O)(CCC(F)(F)C(F)(F)F)NCC1N(C(=O)C(O)CC2CC2)CCN(C)C1 N1(C(C2C(NC(Cc3c(C)nccc3)=O)C=CCC2)=O)C2C=CCC1CCC2 C1(CNC(C(CC)N(C)C)=O)CCCN(C(=O)C(CO)N(C)C)C1 C=CCCC(C(=O)NC1CCOC1)NC(=O)CC1(C)CC1 N1(C(CSC(C)C)=O)CC(C)CN(C(c2ccc(F)cc2Cl)=O)C(C)C1 C1(C(N2CC(F)(CNC(c3cc(CCCO)on3)=O)C2)=O)CN2CCC1CC2 C(=O)(CCCCC(C)C)N1C(CO)CC(NC(c2ccc(C)cc2Cl)=O)C1 C1(NC(c2n(CC)ncc2Cl)=O)CC2CCC(C1F)N2C(=O)C(CC)(CC)CO CC(C)CC(C)(C)OC(=O)NC(C)CC1CCCCO1 Cc1ccncc1-n1cc(C2CCN(C(C3CCC(C(N)=O)CC3)=O)C2)nn1 C1(NC(C(C2CCN(C(=O)C3=CCCOC3)CC2)C)=O)CC2(CCCO2)C1 c1(C(=O)NCC2CC(F)(CNC(C3(C)C=CCC3)=O)C2)cccc2nc(O)oc12 C1(OC)CC(C(=O)N(C)C(c2cnn(C)c2)C)N(C(=O)C(CO)NC(N)=O)C1 C1(O)(CCNC(CSCC#C)=O)CCCN(C(c2nocc2C(C)C)=O)C1 c1(C(=O)NC2(C(=O)N(C)C)CC2)ccccc1CNC(C(C)OCC(F)(F)F)=O C1(C(=O)NC(C2N(C(C=CCOCCOC)=O)CCC2)C)(CCF)CCOCC1 Cc1cc(C)c(C(N2CCC3CC23C(=O)NCc2ncnn2C(C)C)=O)cn1 c1(C(N2C(COC)(CNC(=O)CNS(N)(=O)=O)CCC2)=O)ccc(F)c(O)c1 C12(C(=O)NC(CNC(=O)C(F)CC3CCCC3)C3CC3)CCC(CC1F)C2 C1(F)(CC)CN(C(=O)C#CCNC(=O)COC2CCCCC2)C1 c1(C(N2CCCN(C(C=C(COC)C)=O)C(CO)C2)=O)ccc2nc(O)[nH]c2c1 c1(CC(=O)NCC#CCNC(=O)CC2CC3COCC23)c(F)c(F)cc(F)c1F N1(C(C(N(C(C(C)Oc2ccccc2)=O)C)C2CC2)=O)CC2(CCCO2)C1 N1(C(CC2(C)CCC(=O)C2)=O)CCCC(O)(c2cn(-c3ccnnc3)nn2)CC1 Cc1cc(C(N2CCCC2C(=O)Nc2cccc(F)c2O)=O)ccc1F c1(N(C)Cc2ccccc2F)ccn2ncc(S(=O)(=O)NCC3CC3)c2n1 c1(C(c2nnnn2CC2CCCO2)Nc2n(CCC)ccn2)ccncc1Cl C(CC(C(=O)N1CC([N+](=O)[O-])C1)NC(=O)CC1(N(C)C)CC1)SC n1(CC)nc(C)c(C(N2CCOC(C)C2c2nn[nH]n2)=O)c1C(F)(F)F C1(C#N)(C(N(CC(C)CNC(c2cnc(C3CCC3)o2)=O)C)=O)CCOCC1 N(C(=NCCc1nc(-c2ccccc2)no1)NCC1CC1)C1C(C)CCCC1 C1(NC(c2ccc3nccn3c2)=O)CN(C(=O)Cc2cn[nH]c2)CC(F)(F)C1 C1(=O)CCCCCn2cc(nn2)-c2cccnc2N1.CC1CC1CC(=O)O N1(C(C(C2CCC2)OCC)=O)CCCCC1CCCNC(=O)CCc1cnc[nH]1 C1(C(C)NC(=O)C2=CCC2)CN(C(c2cc(C3CC3)cs2)=O)CCO1 c1(C(N2C(C(=O)Nc3scc(C(C)(C)C)n3)COCC2)=O)cc(I)ccc1Cl C(=O)(C(F)CC(C)(C)NC(c1cn(C)c(C)n1)=O)NC(CC=C)CC C(CC(C(=O)Nc1cccc(Cl)c1)NC(c1n[nH]c(C)c1Cl)=O)=CC c1(CN2C(C)(C(=O)Nc3ncc(Br)nc3I)CC2)c(F)cc([N+](=O)[O-])cc1F c1(C(=O)NCC2CN(C(C3(CC)CCC3)=O)C2)ccc2nc(O)oc2c1 c1(N2C(C)CNC2)c(Oc2cccc(Cl)c2)ccc2ccccc12 c1(C(N2CC(N(C)C(C3CCC34CCC4)=O)C2)=O)ccc(C(F)F)c(F)c1 c1(CC)c(C(N2CCCC2C(C)(C)C(=O)NCC(C)O)=O)nnn1C CCCC(C(=O)N1CCOCC1)OC(C1(C(=O)OC)CCC1)=O C1(CNC(C2C(C)CCN2C(=O)CC2CC3(CCC3)C2)=O)CC(C2CC2)=NO1 Cc1cccc(C(=O)Nc2ccsc2C(N2CCOCC2C(C)C)=O)c1C Cc1ccc(Br)cc1C(N1CCCC(C(=O)NCc2cscn2)C1)=O C(=O)C#CC(C)(C)O.C(C)(CN=[N+]=[N-])CC(=O)N.CC1=CC(=O)NC1 c1(C(=O)NC2(CC=C)CCN(C(C3CCN3CC)=O)C2)coc2c1CCCC2 N1(C(Cn2ccc(C)n2)=O)CCC2(CC1)CCN(c1ncnn3ccc(Br)c13)C2 c1(C(C(=O)NC2CN(C(c3occ(C)c3)=O)CC2F)(F)F)ccc(F)c(F)c1 CCC(CC)C(C)C(=O)NCC(C1CCCC1)NC(c1cc2c([nH]1)CCC2)=O N1(C(c2cccc(CCC)c2)=O)CCN(C(=O)C(F)CC2CCCC2)CC(O)C1 C(=O)(C(COCCC)N(C)C)N(C1CCN(C(c2cnc(C)s2)=O)C1)CCC c1(CC(=O)NCC=CCNC(C(COC)(C)O)=O)cc(Br)ccc1OC N1(C(=O)OC(C)(C)C)CCC(F)(CNC(C2CC(C(F)F)C2)=O)C1 N1(C(=O)OC(C)(C)C)CCn2c(CNC(C3(C)CCCNS3(=O)=O)=O)nnc2C1 c1(NCCc2c(SC)cccc2)ccc(S(=O)(=O)N(C)CCOCC2CC2)cc1Br CC1CN(C(=O)CCOC2CC2)CC1CNC(c1csc(C(N)=O)n1)=O n1(CC(=O)OCC)c(N2CCC(C)C2)nnc1-c1cc(Br)c[nH]1 N1(C(C(c2cn(C)nc2)(C)C)=O)CCC2(CC1)CC(NC(C1(N=[N+]=[N-])CC1)=O)C2 C(=O)(CCC(C)(C)[N+](=O)[O-])N(C1CCN(C(c2c(OC)c(Cl)ccc2)=O)C1)C c1(C(N2C(C)C(NC(C3CC(F)C(=O)N3)=O)CC2)=O)cncc2c(O)nccc12 CN1C(=O)CC(CNCC2CCC2C(=O)O)C1c1ccc(Cl)c(Cl)c1 CC1(C)CN(C(C2CCC(CC(=O)O)C2)=O)C(C)(C)C1O N1(C(c2ccc(OC(C)C)cc2)=O)CC2(CCC2NC(=O)C=C2CCCCC2)C1 c1(C(=O)NC2(CNC(CCC(C)SC)=O)CC2)ccc(C(F)(F)F)c(F)c1 C#CCCCC(C)C(=O)NC(CCC1CCC1)C(=O)NCC(C#N)CC c1(C(=O)NCC2N(C(C=C(CCN(C)C)Cl)=O)CC2)c(Br)ncn1C CC(CC(=O)NC1CN2CCC1CC2)C(C)(C)NC(C1CN2CCN1CC2)=O Cc1cc(C(N2CC(CNC(C3(C(F)F)CCOCC3)=O)C3CC23)=O)c(C)n1C Cn1ccc2cc(NC(C3COC4CN(C(C5CCCCO5)=O)CC34)=O)ccc12 c1(C(N2C(CCNC(CC(n3c(CC)ncc3)C)=O)CCC2)=O)nn(C)cc1N N1(C(C2(CC)CNC(=O)C2)=O)CC2(CC(C(N3CC(=O)NC(C)C3)=O)CO2)C1 Cc1ccc2c(c1)C(C(=O)N1CC(OCCNC(c3ccc(F)o3)=O)C1)C2 C1(NC(c2ccc(SC)s2)=O)CN(C(c2cc3ccoc3s2)=O)CC(F)(F)C1 c1(OC)cc(C(=O)NCCc2cn(CC3CC(F)(F)C3)nn2)cnc1OC C1(NC(C2(SCC)CC2)=O)CN(C(=O)C2=NNC(=O)C2)CCC1O C1(CC)C(C(=O)NC2(CO)CC(O)C2)CCCN1C(=O)C(C)COC c1(OCC)ccc(C(=O)NCC2CCC(C)CN2C(=O)C2=COCCO2)cc1N C1(NC(CSCCC(C)C)=O)CCN(C(=O)Cc2ccoc2)CC1C C(=O)(C(C)(O)C(F)(F)F)N1CCC(OC)(CNC(C23CCCC2C3)=O)CC1 CC(C)CCCCC(=O)N(C)CC1CN(C(C2CCC3CCC2O3)=O)CCO1 C1(C)(C(N(CC(C)NC(c2csc(C3CCCC3)n2)=O)C)=O)CC2(CCC2)C1 N1(C(c2cncc(SC)c2)=O)CCC2(CCC2NC(=O)Cn2nnc(C)n2)CC1 c1(Nc2scc(-c3cc(O)c(O)c(O)c3)n2)ncnc2[nH]ccc12 C#Cc1cc(F)c(C(=O)N(C)CCOCCN(C(=O)C(N)=O)C)c(F)c1 C(=O)(C(C(C)C)N(C(=O)CC1(C)CCCC1)CC)OCC.C1C(C)N1 N1(C(C23CC(COC)(OC2)C3)=O)CCCN(C(c2cnns2)=O)C(C)C1 C(=O)(C(CC(C)C)NC(C)=O)N(CC(C)NC(c1c(COC)ncs1)=O)C c1(C(N2CCC(CNC(c3c(COC)ncs3)=O)C2)=O)cc([N+](=O)[O-])ccc1C c1(C(=O)NCC(CNC(C2(C)CC=C(C)CC2)=O)(C)C)coc2c1C(O)CCC2 C12(C(=O)NC(CC)CNC(C3CCCN3C(=O)NC)=O)CCCC1CCC2 C1(CN(CCCc2cccc(C)c2)C)C(C)CCCN1C(c1cnc(O)n1C)=O N1(C(C(C2CC2)NC(C(C)=C2CC2)=O)=O)CCC2(C1)CN(C)C2 C1(C2CCC2)(C(N2CC(O)(CNC(C(c3ccccc3)OC)=O)C2)=O)CC1(F)F c1(OC)ccc(Cl)c(CC(=O)NCC(C2CC2)NC(C2CC2F)=O)c1 Cc1cccc(C(=O)NCCCOCCNC(=O)C=CCNC(=O)C2CC2)c1 C(=O)(C1=NOC(C)C1C)N1C(CC)C(NC(c2ccnn2C(C)C)=O)CC1 c1(NCCC(Cc2cccs2)NC(c2ccc(C)[nH]2)=O)cnc(Cl)c(Br)c1C C1(C2(C)CC2)(C(=O)NCC2C(C(=O)NCCC(C)CO)CC2)CC1 C#CC(C)(C)C(=O)NCCC(C)NC(c1c(Cl)noc1C)=O c1(CC(C)C)cc(=NCCC2(NC(c3cnoc3)=O)CCCC2)[nH]cn1 C#CCC(O)C(=O)NC1CC1CNC(c1cnn(-c2ccc(Cl)cc2)n1)=O CCC1=C(C(=O)NC2CCC(C(=O)NCC3CC(C)=NO3)C2)CCCO1 c1(-c2cn(CC(=O)NCc3c[nH]nc3C3CC3)nn2)c(C(=O)OC)cnn1C C#Cc1cc(NC(=O)C(CC2CCC2)NC(C2CCCC(C#N)C2)=O)cc(F)c1 Nc1cccn(CC(=O)NCC2(NC(C3SCCS3)=O)CCCCC2)c1=O C1(CNC(C(C)OCCOCC)=O)CCC(C(N2CCC(F)(CF)C2)=O)CC1 N1(C(C2(C)CC(=C)C2)=O)CCC=C(C(=O)N2CCCC(N(C)C)CC2)C1 c1(C(=O)NC(CNC(C(CC)(C)OC)=O)C)ccc(C(F)(F)F)c(F)c1 C1(C(N(C(CNC(=O)CCCCO)C2CC2)C)=O)CC(=O)NC1(C)C N1(C(Cc2cc(C)on2)=O)CCC(NC(=O)CC2CC3CCC2O3)C2(CCC2)C1 C1(C(N2CCC3(C(CNC(C=CC(C)C)=O)C3)CC2)=O)Cc2n[nH]cc2C(=O)N1 C1(C[Si](C)(C)C)CCC(N=c2nc(-c3cc(Cl)cc(Cl)c3)[nH]o2)C1 CC1CN(C(=O)C(C)S(N)(=O)=O)CCCN1C(c1cccc(C(F)(F)F)c1Cl)=O CCCC(C)CC(=O)NCC(C1CCCCC1)NC(C12CC(C1)C(C)O2)=O N1(C(C(C2CC2)OCC)=O)CC2(CCC2NC(c2ccc(OC)s2)=O)C1 c1(NCC)cncc(C(N2CC=CC2CNC(c2ncn(C(C)(C)C)n2)=O)=O)c1 S(=O)(=O)(c1cccc2c1OCCCO2)NC(c1ccc(=NC)[nH]c1)=O C(C)(C(F)(F)C(F)(F)F)=CC(=O)N.C(C(CNC(C1CC1C(=O)C1CC1)=O)CO)OC Cn1cc(C(=O)NC(CNC(C2(S(C)(=O)=O)CCC2)=O)CO)n(C)c1=O c1(C(=O)NCC(CC)NC(c2cnc[nH]2)=O)cc(S(N)(=O)=O)co1 c1(C(=O)NC2CCS(=O)(=O)C2)n[nH]c2cccc(-c3cncc(CO)c3)c12 N1(C(c2cncc(CC)c2)=O)CCN(C(C23CCCC(C2)OC3)=O)C(CCO)C1 CC1=NOC2(C1)CC(C(N1CCC(NC(=O)C=Cc3ccoc3)C1(C)C)=O)C2 c1(C(=O)NCC(CC)NC(=O)C(F)(F)C2(O)CCC2)ccc(COC)s1 C1(NC(CCOC)=O)CCCC1NC(=O)COCC1CCC1 Cc1cc(C)c(CC(=O)NCC(C2CCCN2C(=O)COC(F)(F)F)(C)C)c(O)n1 c1(C(=O)NC2C(NC(CCc3cc(C)on3)=O)COC2)cnc2[nH]ncc2c1 CCC(COC)C(=O)NC1CCCC1CC(=O)NCC1CC(C(C)C)C1 CC(C)(CO)CC(O)CNC(c1ccccc1OC(F)(F)F)CO Cc1cc(C(=O)N(C2CCCN(C(=O)C(N3CCNC3=O)C)C2)CCF)n(C)n1 Cc1ncc(C(=O)NC2CC(C(N3CCC(CC(N)=O)C3)=O)C2)cn1 N1(C(c2c(CCC)n[nH]c2)=O)CCN(C(=O)C(COC)OC)CC(C)(C)C1 CC(C)C(C(=O)NCC(C)CNC(c1ccon1)=O)NS(N)(=O)=O N1(C(c2ccc(CC)cc2)=O)CC(C)N(C(=O)CCCCC(C)C)CC1C N1(C(C(C(C)C)c2ccccc2)=O)CCN(C(=O)CCCCC#N)CC(CO)C1 c1(CNC(C2(C)CCN2Cc2cnc(Br)s2)=O)cc(F)ccc1Br CC1(CNC(=O)CCN2CCOCC2)CCN(C(c2cnc(C3CC3)s2)=O)C1 c1(CNC(C)=O)cccc(C(=O)NC)c1.C1(CC(=O)NCC(CO)SC)CC=CCC1 C1(NC(c2sccc2-n2ccnn2)=O)CN(C(=O)Cn2ccnn2)CC1C(F)F N1(C(c2ccc(C(C)=O)o2)=O)CC(NC(=O)C(C#N)CC2CC2)CC1C C(N=c1nc(N2CCSCC2)c2sccc2[nH]1)c1ccc(SC2CCCO2)cc1 C(CC(=O)NCC1(C)CCN(C(c2ccc(SC)cc2)=O)C1)(C(C)C)OCC C1(C(C)C)CN(C(=O)CC(C)c2cnn(C)c2)CCN1C(=O)C1=COCCO1 N1(C(CCc2cc(C)on2)=O)CCC(C)(CNC(=O)Cc2ccc(Br)cn2)C1 n1(CCC)ncc(C(=O)NCC2CN(C(c3cc(F)cs3)=O)C2)c1C C(=O)(C1=NN(C)C(=O)CC1)N1C(CC)C(NC(c2cncn(C)c2=O)=O)CCC1 c1(C(N(CCOCCO)CC)=O)cn(CCNC(c2cnns2)=O)cn1 c1(CCC)ccc(NC(N2CCCC(C(C)Sc3ccccc3)C2)=O)c(C#N)c1 N1(C(c2c(N)cnc(Cl)c2)=O)CC2CCCN(C(c3cnn[nH]3)=O)C2C1 C1(C(=O)NOC2CCN(C)C2C)N(C(C2C=C(C)CS2)=O)CCC1(C)C C1(C(N2C(CNC(C3CCCN3CC(F)(F)F)=O)CC2)=O)CCS(=O)CC1 N1(C(C(C)NC(C2(c3ccc(C#N)c(Cl)c3)CCCC2)=O)=O)CCN2CCCC2C1 CC(Cc1ccccc1)C(=O)NCCC(C)(C)NC(c1cc(C(N)=O)no1)=O c1(C(=O)NC(C2CCN(C(c3c(C)ccc(O)c3)=O)C2)C)c[nH]c2cccnc12 CC(F)(F)C(C)(C)CNC(=O)C(=O)N(CCO)CC1CCC(=O)N1c1ccccc1 CCCC(CCC)=CC(=O)N(CCNC(=O)Cn1nccn1)C1CC1 CC1(C)CCCN(S(=O)(=O)N2CCC(CF)CC2)CC1 CC1CCC(CNC(c2nccnc2C(F)(F)F)=O)N(C(=O)Cc2ccco2)C1 C1(C(=O)NCCCN(CCO)C(c2scnc2C)=O)(OC)CCOC1 O=C(C#CC1CCCO1)NCC1CN(C(=O)C=CBr)CC12CCC2 CON(CCC(=O)NC(c1ccoc1)C)C(=O)C1=C(C)OCC1 C(=O)(C(CC1CCOCC1)NC(=O)CC1(CO)CC1)N(CC)CC1CCCC1 C(=O)(CC(C(F)(F)F)NC(c1csc(O)n1)=O)NCC(COC)OC N1(C(=O)Cc2ccccc2F)CCCC2C1CCN2c1ncnc2sccc12 C1(CC)CN(C(C2CC(F)(F)CS2)=O)CCN1C(=O)CC12CCC(CC1)C2 C1(NC(CSCCCC)=O)CCC12CN(C(c1ccco1)=O)C2 c1(NC(C2CC(C)(C(=O)OC(C)(C)C)C2)=O)ccc2c(c1)C(O)CC2 c1(COC(=O)CC2CC=CC2)cccc2c(Br)cccc12 N1(C(C(CN=[N+]=[N-])NC(=O)CCOCC2CC2)=O)C2CCCC1CC(O)C2 c1(C(N(CC(F)(F)F)CC(C)C)=O)cnc2ccccc2c1Br Cc1cc2sc(NC(=O)NCC(=Cc3ccc(F)cc3)C)nc2cc1F N1(C(c2c(C(C)C)nns2)=O)CC2CCC1CN2C(c1cnc2ncccn12)=O C1(C(=O)NCCC)CCN(C(=O)C(CC(C)(C)C)OC)C12CCC2 N1(C(c2cc(CNC(CCC(=O)NCCC)=O)no2)=O)CCC(CO)C(C)C1 N1(C(CC2ON=C(C)C2)=O)CCC12CN(C(C1CCN(C)CC1)=O)C2 C#CC1(NC(C2CCCCC2NC(=O)C(C)(C=C)CC)=O)CCCOC1 C(=O)(C(CCF)NC(C1C=CCN(C(c2oc(C)cc2C)=O)C1)=O)OC C(=O)(CC(C)C(C)C(C)C)N1CCC(CNC(c2c(OC)scc2)=O)C(C)C1 c1(C(=O)NCC(C)N(C(C(C2CCC2)OC)=O)C)c(C)cncc1F C1(NC(CN(C2C=CCCC2)C)=O)CC(F)(CNC(=O)CNc2ccncc2)C1 c1(OC)ccc(C)c(C(=O)N(C(CNC(c2cc(O)no2)=O)C2CC2)C)c1 C(=O)(C1=CNC2=NCCCN12)N1CC(CN(C(=O)C=CC(F)(F)F)C)OCC1 c1(C(=O)NC2C3(CC(C(=O)OC)C3)CC2)cc(Br)c2c(c1)[nH]c(=N)n2C c1(SCC)cccc(C(=O)N(C2CN(C(c3cccnc3C)=O)C2)C)c1 C1(O)(CN(C(CSCC(C)C)=O)C2CC2)CCN(C(=O)CC2CCCOC2)C1 C1(OC)CC(NC(=O)CCc2cc(C)on2)CN(C(C2CC(C)(O)C2)=O)C1 N1(C(C=C(C)C2CC2)=O)CCOC2(CCC(N=c3nc(C(C)C)[nH]s3)CC2)C1 C(C(C(C)(C)C)NC(=O)CC(C)O)NC(C1N(CC)CCC1)=O C1(NC(C2(N(C)C(C3CCC(=O)O3)=O)CC2(C)C)=O)CC12CCCC2 Cc1ccc2cc(C(=O)NC(C)(C)CN(C(=O)C=Cc3cn(C)nn3)C)[nH]c2c1 n1(CCC(=O)NC2(CNC(C(CC)(C)OC)=O)CCCC2)ccc(O)nc1=O c1(C(=O)NCC(CC(C)C)NC(C=C(COC)C)=O)ccc2c(c1)CCCS2 c1(C2C(C(N3CC(C)(NC(c4n(CC)ncc4)=O)C3)=O)C2)ccc(Cl)nc1 C1(c2n(C)nnn2)(NC(CC2CC2)C2CC2)CC2(CCCOC2)C1 CCCCC(CC)C(=O)NCc1occc1C(=O)NCC(CC)n1cccn1 c1(CC(N2CC3C(CNC(c4c(C)ncnc4)=O)C3C2)=O)cccc2c1OCO2 N1(C(c2ccc(CC)o2)=O)CCN(C(=O)C2=C(Cl)CCOC2)CC(O)C1 C(=O)(C1CCCn2c(Br)cnc21)NC(C)CNC(=O)Cc1cc(F)ccc1O N#CC1CN(c2ncc(I)cn2)CCN1c1ncncc1F C=C1c2ccccc2C(=O)N1C(C)C(N1CCC(C)S(=O)(=O)CC1)=O N1(C(C=CCN(C)C)=O)CCN(C2CCN(C(c3csnn3)=O)C2)CC1 CCCCCCC(C)C(=O)NCCCC1CN(C(=O)CSCCC(C)C)CCO1 C(=O)(C(F)C(C)(F)F)NCC1(COC)CCCN1C(c1cccc(C(C)C)n1)=O O=C(CC(C1=CCCC1)N(c1ccccc1F)C(c1ccnnc1)=O)N.C1(C)CC1 c1(Sc2ccc(NC(N3C4CCC3CC4)=O)cc2)ccc(Br)cc1 C1(NC(C(CC=CC)NC(c2ccn(C(F)F)n2)=O)=O)CCC(=O)NC1C C1(OC)CC2(C1)CC(C(=O)NC1CN(c3ncc(Cl)c(O)n3)CCC1C)C2 c1(C(=O)NCc2ncccc2C(N2CCCC(O)C2)=O)cnc2c(Cl)cccn12 C1(NC(=O)Nc2ccc(OCC)cc2)CCN(C(=O)CC(C)(C)O)CC1F C1(CC=C)(NC(c2ccc(OC)cc2)=O)CCCN(C(=O)C(COC)N(C)C)C1 CC1(C(=O)NC2COCCC2NC(C2(C(N)=O)CC2)=O)CC(F)(F)C1 c1(C(=O)NCC2COCCO2)cccc(N2CC=CC2)c1 N1(C(C(c2c(C)noc2C)C)=O)CCC(NC(c2ccn(C)n2)=O)C(C)(C)C1 N1(C(c2nc(C(C)C)sc2)=O)CC(CNC(=O)COCC(F)F)CC1C C1(OC)CC(C)CN(C(c2ccc(OC3CCC3)cc2)C(=O)NCCCF)C1 C1(CN(C)C(C2(CO)CC2)=O)CCCCN1C(=O)CCc1cccnc1Cl C1(C(C)C)CN(C(c2ncn(C)n2)=O)CCN1C(c1cc(Br)n(C)n1)=O n1(CC)nc(C(=O)NCC2CC(C)N(C(=O)Cc3ncoc3C)C2)cc1C Cc1ccc2cc(C(=O)NCCCn3cc(-c4coc(C)n4)nn3)sc2c1 c1(SC)cn(C)nc1C(=O)NC1C=CC(CNC(C2CC=CCO2)=O)C1 C(CC)(C(=O)NC1CC(CSC2CCCN2C(=O)C=CC(=O)NC2CC2)C1)=CC C1(CC=C)(C(=O)NC(c2nc(C)no2)C)CCCN1C(=O)Cc1ccn(C)c1 C1(C(N(CCNC(=O)CSc2cccc(Cl)c2)CC)=O)CCCCC12CCC2 N1(C(C2(C(N)=O)CCC2)=O)C2CCC1CC(O)(CNC(C1(C(F)F)CC1)=O)C2 c1(C(=O)NC2(COC)CN(C(CSCCCC)=O)C2)ccc(C)nc1N CC1=NOC(C(=O)NC(CNC(=O)CNC(c2cccc(F)c2)=O)C2CC2)C1C N1(C(CCc2ncc(C)[nH]2)=O)CC2(CCOCC2)C1c1cn(-c2nccs2)nn1 c1(C(N(CC2CC(O)C2)C)=O)cnccn1.O=C(CNC1CC1)N c1(C(=O)OC)cc(Nc2ncc3c(n2)CCC3)c2ccncc2n1 N1(C(c2scc(C)c2)=O)CC2CCCC(NC(c3cnoc3)=O)C2C1 N1(C(CCC)=O)CCC2(CCC(NC(C3CCC(O)CN3C)=O)CC2)C1 C1(NC(CNC(CC)=O)=O)CCN(C(c2cc(Cl)n[nH]2)=O)CC1O CC1(C2(C(=O)NCCc3cc(C(=O)O)no3)CC2)CC1 C1(C(N(CCC(C)NC(=O)C(C)(C)C2CCCO2)C)=O)CCC(N(C)C)CC1 n1(CCC(=O)NCC(CN(C(Cc2cc(C)n(C)n2)=O)C)O)ccc(O)nc1=O c1(CN(C2C(C)(C(F)F)C2)Cc2ncccn2)cccc2ccoc12 c1(C(N2C(CNC(C3C(C)(C)C3)=O)C(O)C(O)C2)=O)cc(=O)c2ccccc2[nH]1 C1(NC(c2cc(C(C)C)on2)=O)CC(O)CN(C(C2OCCCC2(C)C)=O)C1 c1(C(N(C(C(=O)NC)CO)C2CC2)=O)nc(C(=O)OC)co1 C1(NC(C(COC(C)(C)C)N(C)C)=O)CCC2(CC1)CC(NC(C1CC1F)=O)C2 C=CCC(C)(C)CC(=O)NC1COCC1NC(C1CCCN(C(=O)N(C)C)C1)=O Cc1nn(C)c(C)c1C(=O)NCc1cc(C(=O)O)ccc1C(F)(F)F N1(CC(=O)N(C)C)CCCC(N(C(=O)CC2(C(F)F)CC2)C)C1 N1(C(CS(CC)(=O)=O)=O)CC(C)N(C(c2ccc(C)c(Cl)c2)=O)CC1C C(C(=O)N1CC(C)(O)CO1)N(C(=O)CC1=CCCC1)C(C)C C1(N(C(=O)C(C)c2ccsc2)CC(=O)NC(CCC)c2ccco2)CC(C#N)C1 C(=O)(CCCS(=O)(=O)N1CCCC1)NCCN(C(CC(CCC)C)=O)CC N1(C(C(CC#C)NC(c2cccc(CO)c2)=O)=O)CCCC(C)(C#N)C1 Cc1ncnc2c1CC(C(=O)NCCC(C(C)C)NC(c1cc(O)cs1)=O)CC2 N1(C(C2C(C)C2C)=O)CCCC(C2CCCN(C(C3(C)CCCCCC3)=O)C2)C1 C1(C(N2CC(CNC(c3cc(C)ns3)=O)C(C)(C)C2)=O)Cc2c(C)cccc2N1 S(=O)(=O)(c1cccc2cnccc12)N(C(C(F)(F)F)C1CC1)CC1(C)CCC1 C(CCCC(=O)N(CC(C)(C)CNC(C1CCC1c1nc[nH]n1)=O)C)(OC)OC c1(C(N2CCCC(NC(CC3CCC(C)C3)=O)CC2)=O)c2c(nn1C)CCCC2 c1(OC)cnc(Cl)nc1N1CC2C(NC(=O)CNC(=O)C3CC3)C2C1 CCCC(C)(O)CNC(=O)CC(c1cccc(C(F)(F)F)c1)C N1(C(CN2CCC(C)(C)C2)=O)CC2ON=C(CNC(=O)CCNC(=O)CO)C2C1 CCCCC(O)C(=O)NC1(C)CC(C(=O)NC2(C)CCOCC2)C1 n1(CC(=O)N(C(C)CCNC(c2nc(C3CC3)cs2)=O)C)nc(O)ccc1=O C(CCS(C)(=O)=O)(n1cc(C2CC3C=CC2C3)nn1)OCCOC Cc1nc(C)c(C(=O)N(C2CCN(C(=O)CCc3nc[nH]n3)CC2)C)c(C)n1 N12CC(C(F)C1)NCc1cc([nH]c1)C2=O.c1(C=O)c(C)ncn1C.CO c1(C(=O)OC)ccc(C)nc1N1CCCC(C(N2CCNC(=O)C2C)=O)CC1 c1(C(N2CC(C)N(C(c3ccc(N)cn3)=O)CC2)=O)ccc(Cl)c(S(C)(=O)=O)c1 C(=O)(C1COc2ccc(Cl)cc21)N1C(Cn2cc(CC(=O)O)nn2)CC(O)C1 c1(C(=O)NCCN(C(Cc2cc(C)[nH]n2)=O)C(C)C)nccc2occc12 C12(C(N3CCC(O)(CNC(CN(C(C(C)C)=O)C)=O)C3)=O)CC=CCN1CCC2 CC(C(=O)NCC1=CCCN(C(C2(F)CCOC2)=O)C1)S(N)(=O)=O C(C(=O)NNC(=O)COc1ccc(C(=O)N(C)C)cc1)C1C(C)CCO1 C1(CC(=O)N(CCCNC(CCCNC(=O)OCC)=O)CC)CCC(C)CO1 Cc1cc(C(=O)NC2CC(C)N(C(c3cn(-c4ccn(C)n4)cn3)=O)C2)ccn1 N1(C(CCCCCC)=O)CC2=C(C1)CN(C(C1CC(F)(CO)C1)=O)C2 c1(C(N2CC(COC)N(C(C3CC3(C)C)=O)CC2)=O)ccccc1P(C)(C)=O C(=O)(C(C)(F)C(=O)N(CC(C)NC(=O)CN1CCCC1)C)OCC N1(C(=O)NCC(C)Cn2ccnc2)CCCC1CN1CCOCC1 C12(C(N3CC(C)C(CC(=O)NCC4CNC(=O)C4)C3)=O)CCCC1OCC2 C#CCCCC(C)(c1nnnn1C1CCC1)NCC1CC(C)(C)OC1=O Cc1ccccc1SC(C)C(=O)NC1CN(C(=O)C=CCn2cncn2)CC1O C(=O)(C(F)(F)CCn1cc(Cn2ccnc2)nn1)N(C1C(C)C1C)CCO CC1CC(C(=O)NCCC2CN(C(=O)CCc3ncc(C(C)(C)C)o3)C2)CN1C N1(C(c2cn(CC)nn2)=O)CCC2CN(C(=O)C(F)(F)C(O)C3CC3)CC2CC1 C1(C(N2CC(c3cn(-c4nccs4)nn3)C2)=O)CCCCC1C1CC1 Cc1ccc2cc(C(N3CCC(NC(C4CCC(C)CC4)=O)C(C)C3)=O)cn2c1 C1(C(=O)NC(C(C)C)C2CCCC2)CN(C(=O)C=CC(=O)OCCO)CC1C(C)C c1(OC)cccc(NC(=O)NCCSCc2cc(-c3cncc(Br)c3)no2)c1 c1(C(N(C2CCCCC2NC(C23CC(F)(C2)C3)=O)C)=O)cccn(C2CC2)c1=O C1(C(N2CC3(CCN(C(C4(C5CC5)CC4)=O)C3)C2)=O)COc2cc(F)ccc2O1 c1(CCOC(CCNC(C)=O)=O)cc(C)c(F)cc1Cl C1(C(=O)NCc2c(C(=O)NC3COC(C(F)F)C3)c[nH]n2)CC12CCCC2 c1(C(C)NC(c2c(C)nns2)=O)cccc(N2CCOC2=O)c1 c1(Cc2cn(CCNC(C(CN(CC)CC)F)=O)nn2)cccc(S(C)(=O)=O)c1 c1(C(=O)NCC2CC3CC3N2C(=O)CC2CC=CC2)[nH]nc2ncnc(O)c12 C(=O)(C1CCc2scnc21)N(Cc1ccc(C)cc1)CSC1(O)CCCS(=O)(=O)C1 c1(CC(N2CCCCC(NC(C3(Cl)C(C(C)=O)C3)=O)C2)=O)cnc2cccnn12 C1(CCC(=O)NCC2CN(C(c3c[nH]nc3-c3ccncc3)=O)C2)CCOCC1 c1(OCC(=O)N(C(C)CNC(c2ccc(C(C)O)cc2)=O)C)cc(F)cc(F)c1 C(=O)(C(C(C)O)NC(C1CCOC1C)=O)N(CCC#C)CCOC C1(F)(CNC(c2ccc(C)s2)=O)CCN(C(c2cccc(OC(C)C)c2)=O)CC1 c1(C(N(CCOC)CCNC(C23CC(C)C2C3)=O)=O)cccc(C(C)C)n1 c1(C(N2C(CC(=O)NCC(CCOC)O)CCC2)=O)ccn2nccc2c1 N1(C(=O)CN2CCSCC2)Cc2n[nH]cc2C1C(=O)NCC1(O)CCCCCC1 C12(C(=O)NCC(C(C)C)NC(C3(C)CC(C)C3)=O)CC(C)(CCO1)C2 Cc1cc(N)cnc1C(=O)NC12CC(C1)N(C(C1CCS(=O)(=O)C1)=O)C2 C#CCCCCCCCNC(=O)C(C1CCC1)NC(=O)CC(O)CC(C)C C(=O)(CC1=CCCC1)NC(C1N(C(C(SC)SC)=O)CCC1)C c1(C(N(C)CC2N(C(C3(CC(C)C)CCCC3)=O)CCC2)=O)cccnc1O c1(OC)ccc(C(N2CCC(OCc3ccnnc3O)CC2)=O)c(OC)c1Cl c1(C(=O)NC2C(NC(c3ccnnc3O)=O)CC2)nccn2ccnc12 N1(C(C2=CC(C)(CC)C2)=O)CCC2CCN(C(c3sc(C)nc3C)=O)CC12 c1(OC)ccc(OC)c(C(=O)NC(CCNC(C2CC(F)(CO)C2)=O)C(C)C)c1N c1(NC(C2(F)CN(Cc3n(C)ncc3)C2)=O)ncc(C#N)cc1I CCCCCCC(C)(C)C(=O)N1CC(O)(CCNC(=O)C=CC=C(Cl)Cl)C1 c1(C(=O)NC2(CNC(c3cc(CC)sc3)=O)CCCC2)oc(C)nc1C c1(C(=O)NC2(CNC(COC)=O)CCC2)cc2c([nH]1)CCOC2 C=CCC(CC)C(=O)NC1(c2cn(CCSCCO)nn2)CCOC1 N1(C(=O)NCc2c(CC)c(F)ccc2)C(C)CS(=O)(=O)CC1C CC1CCC(C(=O)N2CC(n3cc(CN(C4CC4)CC4CC4)nn3)CO2)CC1C n1(CC)nc(C)cc1C(=O)NCC1(C(N)=O)CN(C(=O)CC2CN(C)CC2O)C1 c1(N2CC(N3CCN(C(C4CCN(C)C4)=O)CC3)C2)ncnc2n[nH]cc12 C1(CC(=O)NCCCOCCNC(CCCN(C2CC2)CC)=O)CCCC12CC2 C1(NC(=O)COc2ccsn2)COCC1NC(C1(O)CC(c2ccccc2)C1)=O C1(C(C)NC(=O)Cc2ccnn2C)CCN(C(C2CC2C2CCCO2)=O)CC1 N1(C(C2C(CC)CCC2)=O)CCCOC(CNC(c2nnsc2C)=O)C1 CC12CCC(C)(O1)C(C(=O)NCCN(C(=O)CCCn1cncn1)C1CC1)C2 C1(C(N2CCC(CNC(CC=C)=O)C(C)C2)=O)C2CCC1(C)C2(C)C N1(C(=O)Cc2ccccc2CO)CC2OCC(NC(C3CC(C(F)F)C3)=O)C2C1 C(=O)(CCCOC)N(CC(CC)NC(c1cc(C2CC2)ns1)=O)CC N1(C(c2nc(C)n(C)c2)=O)CCC(NC(=O)C2=C(Cl)CCOC2)CC(C)(C)C1 C=C(C)C(O)CC(=O)NC(C1CCCC1)CNC(c1cc(-c2csc(C)n2)c[nH]1)=O N1(C(CC(=O)OC(C)(C)C)=O)CC2CC1C2NC(C12CCCCC1C2)=O C(=O)(C1=CCC(F)(F)CC1)NCCN1CCC(NC(C(C(C)SC)O)=O)CC1 C1(CNC2CN(C(=O)OC(C)(C)C)C3(C2)CCC3)CCc2nncn2CC1 c1(OC2CCN(Cc3ccc(OC)cc3)C2=O)ccc2c(c1)C(C)(C)C(=O)N2 c1(CCC(=O)NCCC2(C)CCN(C(CCCC#C)=O)C2)nnc(O)nc1O Cc1ccc(Cl)c(O)c1C(=O)N(C)CC1CCCC(NC(=O)C2=CC(C)(C)C2)C1 c1(C(N2CCC3CC(C2)CN(C(C2(CF)CC2)=O)C3)=O)ccc2cnccc2n1 CC1(C)CCC(F)(F)CC1C(=O)NCC=CCNC(=O)C1=CCCC1 C1(C#N)(C(N2CC(CNC(CCC=CC(C)C)=O)C(O)C2)=O)CC2(CC2)C1 CC1(C)CN(C(=O)C(C)(C)C2CCC2)CC(CNC(=O)CCOCCN(C)C)O1 N1(C(c2ccc(N(C)C)nn2)=O)CCN(C(=O)COC2CCC2)C2CC12 N1(C(C2CC(=C)C2)=O)CCC(NC(=O)C=C(C)C(F)F)C(CC)C1 Cn1cc(C(=O)NC(CNC(=O)C=C2CCSCC2)CO)c(C2CCC2)n1 C1(C(N2CC(C3OCCN(C(C#CC(=O)N(C)C)=O)C3)C2)=O)CCn2cnnc2C1 c1(C(=O)NCC(CNC(CC(CCC)(C)O)=O)(C)C)cc(=O)c2ccncc2o1 C(C(F)(C(=O)N1CCCC(C)(C#N)C1)C(C)C)NC(C1CC(OCC)C1)=O N1(C(CCc2n(C)c(S)nn2)=O)CC2CCN(C(C3(F)CCCOC3)=O)CC2C1 Cc1cc(=NC(CNC(=O)Cc2ccc(O)nc2)CO)[nH]c(C)c1C#N c1(C(=O)NC2(CCC)CC2)ccoc1CNC(=O)C(C)(C)OC CCC(C)C(=O)NCC1(NC(=O)CN2CCSCC2)CC(OC)C1 N1(C(CC(C)c2ccsc2)=O)CCCC(CO)(CNC(C2CN(S(N)(=O)=O)C2)=O)C1 C(=O)(C(F)(F)CCc1ccccc1)NCC(CNC(C1(C)CCC(=O)C1)=O)OC C1(C(N2CC(OC)C(NC(C3CC4CCC3O4)=O)C2)=O)CC2(C1)CS(=O)(=O)C2 N1(C(C2(CC=C)CC2)=O)CCC2CCN(C(c3cccc([N+](=O)[O-])c3C)=O)C2C1 C1(C(=O)NCC(C)(C2CC2)NC(c2c(C(C)C)occ2)=O)CCN(C)C1C N1(C(C2CCN(C(N)=O)CC2)=O)C2CCC1CN(C(C1C3CCCC13)=O)C2 C1(C(=O)NC(C)CC(C)O)(SC)CN(C(=O)COCCSC)C1 c1(C(=O)NCC(C2CC2)NC(CCSC)=O)cc(C#N)c(F)cc1F CCC(C(=O)NCCOC1CCN(C(=O)Cn2ncnn2)C1)N(C)C C1(C(NOCC(C)C)=O)C2CCC1N(C(c1ccccc1C1CCCO1)=O)C2 C1(NC(C2C(NC(C(C(C)C)=O)=O)CCC2)=O)CCCC2(CC1)CC2 CN1C2CCC1CC(=CC(=O)NC13CCC1CN(C(c1cccc(F)c1)=O)C3)C2 c1(CC)ccc(CN2CCC(OCC(=O)NCc3nc(CC)on3)C2=O)cc1 CC1CC(C(N2CCC2(C)CCO)=O)CCN1C(c1csc(F)c1)=O C1(CNC(c2occ(C(N)=O)c2)=O)CCCCN(c2ccc(C#N)nc2)C1 N1(C(C2C(c3n(CC)ccn3)C2)=O)CCC2(CC1)CCN(C(C1CC(C)(O)C1)=O)C2 C1(C(N(C2CCOC2)C)=O)C2CN(C(C3(C(F)(F)F)CCC3)=O)CC12 N1(C(C(C)SC(F)(F)F)=O)CCC(CNC(=O)CC2CCCC(C)C2)C12CCC2 C1(N(CC=C(C)C)C(=O)NC2(c3ccccc3)CC2(C)C)C(C)CCC1C c1(N2CCCC(CCNC(c3cnc(COC)s3)=O)C2)ncc([N+](=O)[O-])cc1C C1(C(=O)NCc2n(CC)cnn2)CCN(C(c2snnc2C)=O)C1C C(=O)(CCCN=[N+]=[N-])N1C(CC(=O)NC(C=C)C2CCC2)CC1 CC(C)CCC(=O)NCCCC(C)NC(c1ccc(C2CCCCC2)s1)=O CC(O)C(C)C(=O)NC1C2CC1N(C(=O)CCCc1nc(-c3cn[nH]c3)no1)C2 C1(CC#C)(C(N2CC(N=[N+]=[N-])C2)=O)CCN(C(=O)CC2CCCO2)C1 N1(C(CC)C(=O)NC(C)(C)CN(C)C(C2(O)CCC2)=O)CCN(CCO)CC1 C12(NC(c3cnc(C(C)C)[nH]3)=O)CCCC1CN(C(C13CCC(CC1=O)C3)=O)C2 C(=O)(C#CC(C)(C)CNC(c1nc(O)sc1C)=O)N(CCSC)CC C1(CC(=O)NC(C)C(=O)N(C23CC(C2)C3)C)CCOC1=O CC(C)C(O)CC(=O)N1CC(NC(c2ncc[nH]c2=O)=O)CC(O)C1 C(=O)(C1CSc2ccccc21)N1CCC(NC(C2CC(=O)N2)=O)C(CO)CC1 N1(C(C(C(C)C)C#N)=O)CCC(C2CC2)C1C(=O)Nc1ccc2nncn2c1 CC1CC2CN(C(=O)C(O)CC(F)(F)F)CC2N1C(=O)CN1CCC(=O)CC1 c1(C(=O)NC2C(NC(c3c(OC)cc(O)nc3)=O)CC2)cc2cccn2cn1 C1(NC(Cc2n(C)nnc2)=O)CC2CC1CN(C(C13CCC(CC1)OC3)=O)C2 N1(C(CCC(C)OC)=O)CCC2(CC1)CN(C(C1CCCC(F)(F)C1)=O)C2 c1(C(=O)NCC(CC)NC(C2(C(=O)OCC)CCC2)=O)csc(C(F)(F)F)n1 c1(C(=O)NC2CCCC2NC(C2(n3cc(Cl)cn3)CC2)=O)cc(O)ccc1F c1(OC)cc(CN2CC(NC(C3(C#N)CC3)=O)C2)cc(CN(C)C)c1O N1(C(c2nn(CC)c(O)c2)=O)CC2(CC2)CC1CC(=O)NCCCS(C)=O C1(NC(C2C(OC)CN(C(COCCCC#C)=O)C2)=O)COCCN(C)C1 C1(N(C(CCOC(C)C)=O)C)CN(C(=O)CC2CCCN2C(C)C)CC12CC2 CC(C)C(C)CC(=O)NC1(CCNC(C2(F)CCCOC2)=O)CC1 N(C1CCOc2cc(F)cc(F)c21)C(C(=O)NCCC(C)C)=O c1(OC)ncc(Cl)cc1C(N1CCC(NC(c2cc(Cl)n(C)n2)=O)C(O)C1)=O c1(OC)cc(OC)nc(Nc2cc(Cl)ccc2C)n1.C12CCN1C2=O N1(C(C(CC=CCC)C)=O)CCC(CNC(c2nnsc2SC)=O)C12CC2 N1(C(CC(CNC(COCC(=O)NC)=O)O)=O)CC(=O)NCC1C(N)=O c1(NC(C2N(c3ncc(C)c(C)n3)CCCC2)=O)cc(Br)c([N+](=O)[O-])cn1 C1(CC)CC(c2nnnn2C2CC(F)(F)C2)(NC2CSC2)CCO1 C1(NC(C)=O)CC2(C1)CN(C(c1cccc(CO)c1F)=O)C2 N1(C(=O)CCSc2ccc(F)cc2)CCC2CN(C(=O)C3=CCCC3)C2C1 c1(C(C(=O)N(C2CN(C(C(CC)SC)=O)C2)C)O)ccc(Br)cc1 CC(C)C1=NOC(C(N2CCCC2CCCNC(=O)C=CC=C(Cl)Cl)=O)C1 N1(C(C(C=CCCC)O)=O)CC(NC(c2cnc(C)n2C)=O)CC2(CCC2)C1 N1(c2n(CC(=C)C)c(-c3cnn4cc[nH]c34)nn2)CCCC(C2CCC2)C1 C1(C(N2C(C)CN(C)CC2)=O)CCN(C(=O)C(C)N=[N+]=[N-])CC1(C)C C(=O)(C1=CC2CC=CCC12)NCCC1CC(NC(c2cc(C)c(Cl)c(N)c2)=O)C1 C1(N(C(C2(C(=O)OC)CC2)=O)CCN2CCCC2=O)CC2CC1CN2 C1(NC(c2[nH]c3ncn(C)c3c2)=O)CCN(C(c2cc(Cl)no2)=O)CC12CCC2 C1(NC(C(CC)F)=O)CN(C(=O)CSCc2ccc(Cl)cc2)CC1C c1(C(=O)NCC(C2CCCC2)NC(C(C)(C)N(C)C)=O)cccc2c1CCN2 Cn1cc(-c2cccs2)cc(NC(CC(=O)OC(C)(C)C)=O)c1=O C=CCCCCC(=O)N1CCOC(CNC(C2CC(Oc3ccccc3)C2)=O)C1 CC(C)(CC(F)(F)F)C(=O)N1CCC(OCCNC(=O)CN2C(=O)CCC2=O)C1 CC(CC(=O)NC1COCCC1NC(=O)C1=CCCSC1)C(F)(F)F c1(C(=O)NC2CCC(C(=O)NCc3occ(C)n3)CC2)ccn2nccc2c1 C(=O)(CC(C)(C)C(F)(F)F)NCCCN(C(=O)C(c1cccc(F)c1)(C)O)CC CC1=C(C(=O)NCC2CC3CN(C(=O)C(C)C(=O)OC(C)(C)C)CC23)CCC1 c1(CNC(C(F)=CCC)=O)cc2n(n1)CCN(C(c1nc(C)no1)=O)C2 C1(C)(NC(c2nccc(OC)n2)=O)CCCN(C(C2(O)CCOC2)=O)C1 Cn1c(CO)nc2cc(C(N3CCC4CC4(NC(=O)CC4CC4)CC3)=O)ccc12 c1(C2C(C(N(CCCNC(C(CC)(C)O)=O)C)=O)C2)c(Cl)cccc1Cl C(CC(C)C)(C(=O)NCC(CC(F)(F)F)NC(c1coc(C(=O)OC)n1)=O)OC C1(O)(CNC(C2(CCOC)CCC2)=O)CCCN(C(=O)CCn2ccc(C)n2)C1 c1(C(=O)NC2C(CCC)CN(C(=O)C(C)(C)OC(C)C)C2)cc2ccncc2[nH]1 Cc1nn(C)c2nc(O)cc(C(=O)NC(C)CC(C)NC(=O)CC3CC=CC3)c12 N1(C(C(C)C2CCCC2)=O)CC2(C(=O)NCCCC(C)(F)F)CC1CO2 N1(C(CC)=O)CCN(C(c2ccc(CC)nc2)=O)CC(O)C1 C(C(C)(COC)CC)NC(C(C=CC)O)=O.C1C(=O)N1CC(C)C C1(N(C(=O)C(C2CCOCC2)O)C)CCCCN(C(=O)CN2CC3C=CC2C3)C1 C(C1CCc2cc(F)ccc21)N(C(c1ccc(C(F)(F)F)cc1)C)C1CC1 C1(NC(COCCN(C)C)=O)CN(C(=O)C(CO)N(C)C)CCO1 N1(C(C2C(C)CC2)=O)CC(CNC(c2cn(C(C)(C)C)cn2)=O)CC1(C)C N1(C(C(C=C=C)C)=O)CCN(C(c2cc(Br)ccn2)=O)C(c2cn[nH]c2)C1 FC(F)(F)C(C(F)(F)F)Sc1nc(C2CCC2)nn1-c1cncc(Br)c1 N1(C(C2CC(OC)C2)=O)CC=CC1(C)C(=O)NCCCC1CCCCO1 C(c1ccncc1)=C(C(=O)NC(CN(C(c1nnc(C(F)(F)F)s1)=O)CC)C)C C1(CCNC(COCCC#C)=O)CCN(C(c2ccnn2C(F)F)=O)C(C)C1 N1(C(C2C(C)C2)=O)CCC(CNC(=O)C(C)Cc2ccccc2F)C1(C)C N1(C(CC(CNC(c2c(COC(C)=O)occ2)=O)OC)=O)CC2CC1CS2=O C12(CNC(Cc3cccc(OCC)c3)=O)CCCC1CCN2C(=O)CN(C)C N1(C(C23N(C(=O)Cc4ccco4)CCC2C3)=O)CCC([N+](=O)[O-])CC1 N1(C(c2c(N)nccn2)=O)CCCC(NC(c2nn[nH]c2Cl)=O)C(F)C1 C1(NC(CC2N(C(C)=O)CCC2)=O)CCN(CCNC(=O)Cc2cnns2)CC1 C#Cc1ccnc(C(N2CCC(C(C)C(=O)NCc3cc(=O)cc[nH]3)C2)=O)c1 c1(-c2cn(CCCNC(=O)COCCN[SH]=O)nn2)ccc(F)cn1 N1(C(=O)Cn2ncnn2)CCC2CN(C(C3(n4cncn4)CC3)=O)CC2C1 CCC(C)(F)C(=O)N1CCC(NC(=O)C(O)Cc2[nH]cnc2C)CC1 CCC(CC)(C(=O)NC1CC(C)N(C(=O)Cc2cnsc2)C1)OC N1(C(=O)C=CCNC(C2CCN2Cc2ccccc2)=O)CCC12CCCOC2 Cc1ncc(N)cc1C(=O)N(C)CCNC(c1cnoc1-c1ccccc1Cl)=O N1(CC(C)C)CC2(CN(C(=O)CC(C)C3CC3)CCO2)C1 C1(NC(c2c(C)nc[nH]2)=O)CCN(C(c2cnn(C3CC3)c2Cl)=O)CC1(C)C C1(C(CNC(=O)CC2OCCO2)NC(CN(C)CCO)=O)CCCCC1 C1(C(=O)NC(CCC)c2nn[nH]n2)CCn2c(C(F)(F)F)nnc2C1 C#Cc1ccnc(C(N2CC(NC(=O)CCc3ccc(F)cc3)CC2C)=O)c1 c1(N(CC(C)(C)O)C(N(CCCCO)C)=O)cnc(C(F)(F)F)cc1 N1(C(c2c(C(F)(F)F)nn(C)c2C)=O)CCOC(C)(CNC(=O)C(C)(C)C(F)F)C1 C1(NC(C(COC)O)=O)CCOCC1NC(C1(C(F)(F)F)CCCC1)=O CN=c1c(C(=O)NC(C)C(C)NC(=O)Cn2cncc2C)c[nH]c2ccccc12 C1(C(=O)NCC(CCC)OCC)C(C)OCCN1C(=O)C(C)N(C)C N1(C(C(C)OCCOC)=O)CCC2C(NC(=O)CCc3cnc[nH]3)CC12 c1(C(CNC(=O)C(C)(C)C2CCCCO2)N(C)C)ccc(CCC(=O)OC)cc1 c1(N2C(CNC(c3c(CC)noc3)=O)CC3(CC3)C2)nc(O)c2ccccc2n1 C(c1ccc(O)cc1)=CC(=O)NC1CC(C(N2CCC(N(C)C)C2)=O)C1 C1(C(=O)NC(C)CC(C)NC(=O)CC2CCC2)(OC)CCOCC1 c1(CC(=O)NCCC(CC)(C)NC(=O)C=CC(C)(C)SC)cccc(C)c1C N1(C(C(CC)OC)=O)CC2(CCCCN(C(C3(OC)CCCC3)=O)C2)C1 N1(C(c2cncc(C)c2)=O)CCC2(CCN(c3cc(C)ncn3)C2)C1 CC(C)C(C(=O)NC1CCN(C(C2(C)CCCCC2)=O)C1)c1cccnc1 C1(NC(c2n(CC)ncc2)=O)C2CCC1CC(NC(c1cc(C)ccc1N)=O)C2 C1(C(=O)NC2C(NC(CCC(=O)NCC)=O)C2)CCc2nc(C(C)C)[nH]c2C1 c1(OC)cc(OC)c(C(=O)N(CC(C)O)CCNC(=O)CNC(C)=O)cc1Br N1(C(COCCC=C)=O)CCC(C2CC2)C1CNC(c1ccc[n+]([O-])c1)=O C(=O)(C1=NNC(=O)C1)NCCN1CCN(C(c2cc(C(=O)OC)ncc2)=O)CC1 C#CCCCC(=O)N(C1CCN(C(=O)C=C2CCCO2)CC1)CCOC Cc1n[nH]c(C)c1C(C)C(=O)NC1CN(C(=O)Cc2ccccc2)CC1CO c1(C(N2CC(F)(C(=O)Nc3cnoc3)C2)=O)cccc(F)c1 c1(C(c2nnnn2CCO)Nc2c(Cl)cc(C)c(Br)n2)cccc2cnccc12 C1(NC(c2n(C)nc(CC)c2Cl)=O)CC2CCC1N(C(=O)CC(C)C(C)C)C2 S(=O)(=O)(c1cc(Br)c(Br)s1)N(C1C(C)CCNCC1)CC=Cc1ccccc1 c1(C(N(CCCCNC(C(C)NC(CC)=O)=O)C)=O)cccc([N+](=O)[O-])c1 N1(C(C2N(CCC)CCC2)=O)CCCN(C(=O)CS(=O)(=O)NC)C(C)C1 CCCCC(CC(=O)NC1CC(CCC(N)=O)C1)NC(C12CCCN1CCC2)=O C(=O)(CCCCCNC(=O)Cc1n[nH]c(C)n1)N1C(CC)(CC)CC1 CC1C(C)N(C(=O)CC23COC(C)(C2)C3)CCN1C(c1nc2ncccn2n1)=O C(=O)(CS(=O)(=O)Cc1cccs1)N1CCN(CCNC(=O)Cc2cnns2)CC1 C1(CNC(C2(CC)CCN(C(=O)C(c3cnn(C)c3)C)C2)=O)CC2CCC(C1)C2 N1(C(c2ccc(-c3ccco3)[nH]2)=O)CCCCC2(CCN(C(=O)C(Cl)=CCl)C2)C1 C(=O)(C(F)CCC(C)C)NCC1ON=C(C(=O)NCC2OCCN(CC)C2)C1 c1(NC)cccc(C(N2CC=CC(NC(=O)C=C3CCC(C)CC3)C2)=O)n1 c1(N2CCC(C)C(NC(c3c(C)onc3)=O)C2C)ncc2ncn(C)c2n1 c1(C(N2CC(NC(C(N3CCOCC3)C)=O)C2)=O)ccc(C2CCC2(C)C)cc1 Cc1ncccc1NC(C1CN(C(C2CCNC(=O)C2)=O)CCO1)=O C1(NC(CC=CC(C)(C)C)=O)CCCC(C(=O)NC2(CC(C)(C)C)CC2)C1 c1(C(=O)NCC2C(NC(=O)CCCC3CCC3)CC2)cc(O)nc2cnccc12 c1(CCOC(C2C(CCC)CCC2)=O)cncc(C)n1.N12CC(C1)OCC2=O C1(C2CCOCC2)(C(=O)NC(CNC(c2c(Cl)ccc(C)c2)=O)CO)CC1(F)F C1(C(=O)NCCSCCC=C)CCC(O)CN1C(c1ccn(C)c1CC)=O N(C1CCCc2ccc(Br)cc21)C(C(C)(C)C(C)C)c1n(CC(=C)C)nnn1 N1(C(CCC(=C)Br)=O)CCC(CO)(NC(=O)CC2CCCNC(=O)C2)CC1 c1(C(N2C(CNC(c3cn(CC)nc3)=O)CC(O)C2)=O)cc(F)cc([N+](=O)[O-])c1 c1(CNC(=NCC=C)NC(CC)C(F)F)ccc2c(n1)CCCC2 CCC(C)C(O)C(=O)N1CCN(C(c2ccc(C(C)(C)C)cc2)=O)C(CCO)C1 c1(CC(=O)NC(C(C)NC(=O)C(C)C(F)(F)F)(C)C)noc2ccccc12 C1(C(N(CCNC(C(C)NC(C)=O)=O)C)=O)C(C)(C)CCCC1(C)C CC1CN(C(=O)C(CN(C)C)NC(=O)C(C)n2ccnn2)C(C)C1C N1(C(C2(SC)CC2)=O)CCC2CN(C(=O)CC3CNC(=O)O3)CCC2C1 C1(NC(CC(C)F)=O)CCC(O)CN(C(=O)CP(C)(C)=O)C1 C(CC(=O)NC1CCC(NC(=O)CCC#N)C1)(C(F)(F)F)N(C)C1CC1 N1(C(CC(CC)(C)C)=O)CC2(CCNC(c3ncsc3NC)=O)CCC1CC2 C1(C(=O)NC2CCN(C(c3ccn(CC)n3)=O)C2C2CC2)CS(=O)(=O)CC12CC2 C1(NC(c2cnco2)=O)CC(C(=O)NCC2(CO)CC23CCC3)=CC1O C1(CC(N2CC(CNC(C3C(C)C3)=O)N(C)CC2)=O)CC(C)CC(C)(C)C1 c1(N2CCC(N(C(C(C)OCCCCCC)=O)CCC)C2)cc(C)ncc1C#N N1(C(Cc2nccc(OC)n2)=O)CC(C)CN(C(=O)C=CC(=O)N(C)C)C(C)C1 c1(C(=O)NCC(C)CNC(=O)CCC2CCN(C)CC2)cc(C#N)c(N)cc1O N=c1[nH]c(=NCc2ccc3c(c2)OC(F)(F)O3)[nH]c(=NC2C=CCCCC2)[nH]1 Cc1cc(N)c(C(N2CCCCC2CCNC(C2(C)CCCO2)=O)=O)cc1C c1(C(=O)NC2CCN(C(c3c(C)sc(O)n3)=O)C2(C)C)ccc(F)c(F)c1Br CC1(C)CN(C(C2CC3(C2)CC(F)C3)=O)CC(CNC(c2cnccn2)=O)O1 C1(CC(N2CCCC(OCCCN(c3c(C)nns3)C)C2)=O)CCCCC1(C)C C1(C(C)NC(c2cocn2)=O)CN(C(c2cnc(Cl)cn2)=O)CCO1 C1(C)(CNC(C(CCOC)(C)C)=O)COCCN(C(C2(C)C=CCCC2)=O)C1 N1(C(c2n[nH]c(C)c2O)=O)CCOCC(NC(=O)C=CCN2CCCC2)C1 N1(C(c2c(Cl)cc(C)s2)=O)CCC(C2(NC(c3ccc4n[nH]cc4n3)=O)CC2)C1 c1(CSCCC)ccc(C(N2CC(C(C)NC(c3cnc(S)[nH]3)=O)C2)=O)o1 C1(C(=O)NC2(C)CN(C(c3nn(C)c(F)c3)=O)C2)CC2OC(C)(C)OC2C1 C(=O)(C1=CN(C)S(=O)(=O)N=C1C)N1CCC(CNC(C(C)OCC#C)=O)C1(C)C C1(CNC(CCn2cc(CN(C)S(N)(=O)=O)nn2)=O)CCCC12NC(=O)NC2=O C=CC(CC)CC(=O)NCCC1(O)CCN(C(c2cnc(OC)c(C)c2)=O)C1 N1(CC)C(C)CN(C(=O)C(c2cc(C)cc(C)c2)NC(C)=O)CC1C C1(C2CCN(C(=O)CNC(=O)NC3CC3)C2)(NC(=O)CC2COC(=O)C2)CC1 C1(SCC)CCC(C(=O)NCC2CCCC2NC(c2cccc[n+]2[O-])=O)CC1 C=CCC(C)(C(=O)N1CC(C)(C)CC1CNC(c1ccncn1)=O)N(C)C C1(=CC(=O)NCC2COCC2NC(=O)C=C(Cl)Cl)CN2CCC1CC2 c1(C(N2CC(O)(CCNC(=O)C3=COCC3)C2)=O)ccc2scnc2c1 C(CC(C)C)(C(=O)NCC1(COC)CCC1)ONC(C(C)NC(CC)=O)=O c1(C(N(CC(C)CC(C)C)CCC)C)cccc(C)c1 C(=O)(CCCCCc1cccs1)NCC1C(NC(c2c(C)occ2)=O)CC1 C1(C(=O)NC2CN(C(C3CCC(C(N)=O)CC3)=O)C2)CCC2(CCC2)O1 N1(C(C2CC(N(C)C)C2)=O)CCC2(CCC(NC(C3CSCC(=O)N3)=O)C2)CC1 C(=O)(CCCS(N)(=O)=O)NC1CCN(C(c2ccc(C)nc2)=O)CC1C N1(C(c2nnc(C)s2)C)CCC(C)(NC(=O)CC2CC=CC2)C1 Cc1cc(NC(=O)C(C)(C)C2CCN(C(=O)C(C)O)C2)cnc1O N1(C(=O)Nc2nccc(-c3ccc(Cl)cc3)n2)CCCC2(CCCNC2=O)C1 Cc1ccc2[nH]c(C(=O)Nc3cccc(Cn4cccn4)c3)c(Cl)c2c1 Cc1cc(=O)oc2ccc(OCC(=O)NCC(O)CCNC(=O)CN(C)C)cc12 c1(C2(CC)CCC2)csc(NC(=O)C=CC(c2cnn(C)c2)=O)n1 Cc1cc(=NCc2nc3ccccn3c2Cl)[nH]c(N2CCC3(CC2)CSC3)n1 C1(C(N(CCCNC(CCC=CC(C)C)=O)C2CC2)=O)CC1C1CCCC1 c1(C(=O)NC2C(NC(=O)CC(O)c3ccccc3)COC2)ccccc1NC=O c1(C(=O)NCCC(O)C(=O)N2CC(N3CC(F)C3)C2)ccn2nccc2c1 N1(C(C(C2CCCC2)NC(C)=O)=O)CCCC1C(=O)NC1CCN(CC2CC2)C1 c1(OC)c(C(N2CCCCC2c2cn[nH]c2)C(=O)NCCCSC)cccc1F N1(C(C=CCOC)=O)CC(CO)C2(CCN(C(=O)C(C)(C)CC3CC3)CC2)C1 N1(C(c2c(C)con2)=O)CCC(NC(=O)C=Cc2cnn(C)c2)C1C1CC1 Cc1c(C(=O)NCC2N(C(c3ccc[nH]3)=O)CCC2(C)C)c[nH]c1C#N c1(C(N(CCCCNC(CCOC(C)C)=O)C)=O)cncc(-n2ccnn2)c1 C1(C(=O)NC(C)(C)CNC(=O)C(c2cccc(Cl)c2)(C)C)CC1C1CCCC1 C1(N(C(CC(OCC)OCC)=O)C)CCCN(C(=O)C(C)(C)C)CC1 c1(C(N2CC(O)(CCNC(C3CC(OCC)C3)=O)C2)=O)cnn(C(C)(C)C)c1C C1(OC)CN(C(c2ccns2)=O)CCC1NC(=O)CN1CC2CC2C1 S(=O)(=O)(c1cc(F)c(F)c(F)c1)N1CC(C(=O)Nc2cccc(C#N)c2)OCC1 n1(CC(=O)NC(CNC(c2cscc2-c2ccccc2)=O)CO)nnc(=O)[nH]1 C1(C(=O)NCC2CCCN2C(c2cc[nH]n2)=O)(CSC)CCOCC1 c1(C(C(=O)NC(C)CC)N(CCOCC=C)C)cccc(C2CCCC2)c1 c1(OC)cc(N2CC(O)(CNC(C3CCC(NC)CC3)=O)C2)nc(C(F)(F)F)n1 C1(C(N2C(CC(C)C)CC2)=O)N(C(C2CCC(=O)CC2)=O)CC12CCCC2 C1(C(=O)NC(c2ccc(F)cc2)CNC(CCCOC(C)=O)=O)CCCC1(C)C N1(C(C(COCC)NC(c2cncnc2C)=O)=O)CC(N(C)C)C2(CCC2)C1 CCCCC(CCC)NC(=O)CC(C)(C)NC(C1CC(F)C(=O)N1)=O C12(CNC(C(C=C)O)=O)CCCCC1N(c1ncc([N+](=O)[O-])cc1Cl)CC2 N1(C(=O)C=CCN2CCOCC2)CCC2CC(C1)CN(C(=O)C(O)C1CCCC1)C2 c1(C(=O)NC(C)C)c(C(=O)NCCN(C(C2CC2F)=O)CCOC)cnn1C C(C(C)CC(=O)N(C1CC(C(=O)Nc2cnc(SC)nc2)C1)C)OC N1(CCCCCC)CCC(N(c2ccc(F)cc2)C(c2nc(C)c(C)o2)=O)C1(C)C CC1(C)CC(CNC(=O)CC2CCCC23CC3)CN1C(=O)Cn1cnc(=N)[nH]1 c1(CCC)nc(C(=O)N(C)CCNC(C2CC(C)CO2)=O)co1 Cc1cc(C(N2CCCC(O)(CN(C(=O)CN3CC=CC3)C)C2)=O)c(C)cn1 c1(C(=O)NCC2N(C(CCN(CCCCC)C)=O)CCC2)ncc(C)cc1OC c1(C(=O)NCC2N(C(CC3(C)CCCO3)=O)CCC2)ccc(Br)cc1F C1(NC(C(c2cnn(C)c2)C)=O)CCCCCC1NC(c1cnc(O)n1C)=O C1(CNC(C(C=CC)O)=O)CN(C(=O)Cn2cc(C#N)cn2)CCC1C Cc1c(CC(=O)NC2CC(CC(=O)NC34CCC(CC3)C4)C2(C)C)ncn1C C12(NC(c3ccc(SC(F)(F)F)cc3)=O)CC1CN(C(=O)Cn1cc(Cl)cn1)C2 Cc1cnc(NC(CC2CC2)CO)c(S(=O)(=O)NCc2ccnc(Cl)c2C)c1 c1(C(=O)NC2CCCN(C(=O)C(F)OC(F)(F)F)C2)ccc2ccccc2c1F C1(C)(CC(N2CCC(OCC(N3C(CC)(CC)CC3)=O)C2)=O)CCOCC1 Cc1nc2sccn2c1C(=O)N(C)CCC(=O)COCCN.c1(O)cnn(C)c1 c1(C(N2CCC(C(C(C)C)NC(=O)COCC3CC3)CC2)=O)cc(=N)[nH]c(Cl)n1 c1(CC)cc(=NC(=O)C(CCC2CC2)NC(=O)CC2COCCO2)[nH]n1C C1(C(=O)NCc2cc(-c3cccc(C)c3)no2)CCC(C)(C(F)(F)F)CC1 N1(C(C2C(C)OCCC2)=O)CCC(NC(c2ccc(CO)c(F)c2)=O)CC1C N1(C(C(=O)NCCOC)C2CC(C(=O)OC)C2)CCCC1C(C)(C)CO C1(NC(C(C)N2CCC2)=O)CCCCCC1n1cc(CC(C)(C)O)nn1 c1(OC)c[nH]c(C(=O)N(CCC(C)NC(=O)CC2CC=CC2)C)cc1=O C1(c2cn(CC3(O)CCN(C(CC)=O)C3)nn2)CC2(C1)OCCO2 C(=O)(C1=NOCC1)N1CCC(CN(C(C(c2ccc(F)cc2)OC)=O)C2CC2)C1 c1(C(N2C(C(=O)NCC3(C)CCC3)COCC2)=O)cc([N+](=O)[O-])c(O)cc1O C1(NC(Cc2c(OC)cccc2)=O)CCN(C(=O)C(C(C)C)C2CCC2)CC1F c1(OC)ccc(C(=O)NC(C)CN(C(=O)CSCC(N)=O)Cc2nncs2)cc1 Cc1onc(C(N2CCC23CN(C(C2CCC(=O)N2C)=O)C3)=O)c1[N+](=O)[O-] C1(CCN(C(CCCOCC=C)=O)CC)CN(C(c2ccc(C(N)=O)[nH]2)=O)CCO1 c1(OC)cc(F)ccc1C(=O)NC1(CNC(=O)C(C)CC2CCC2)CC1 N1(C(C(C)N(C(Cc2nc(C)oc2)=O)C)=O)CC(C)(C)OCC1C N1(c2ncc(OC)cn2)CCN(C(c2cc(Br)cnc2Cl)=O)CC12CC2 N1(C(COCCOCC)=O)C2CCC1CC(O)(CNC(c1cc(C)ns1)=O)C2 c1(CC)cn2c(n1)CCC(C(=O)NCC1CC(F)(F)CN1C(C1CC1C)=O)C2 N1(C(C2CC2F)=O)CC2CCC(C1)N2C(c1ccc(Br)nc1Br)=O c1(C(N2C(CCC)(C(=O)NC)CCC2)=O)cc2c(F)c(F)cc(F)c2[nH]1 c1(C(=O)NCC2OCC(CNC(=O)Cc3cc[nH]n3)C2)ccc2ncnn2c1 c1(C(N2C(CN(C(=O)CC3CC4CC4C3)C)CCC2)=O)cnc(N)cn1 c1(CC(N2CCC(N(C(C(C(C)C)C)=O)C)CC2)=O)cc(Cl)cc2ccccc12 C1(CC)CCN(C(=O)CCOCC(C)(C)C)C1C(=O)NCc1cnn(CC)c1C c1(N(CC(CN(C)C(C2CCC(F)(F)C2)=O)O)C)ccccc1[N+](=O)[O-] c1(NC(=O)COc2ccccc2)cccc(OCCCNC(C2C(C)C2C)=O)c1 C1(C(=O)NC(C(NOCc2ccc(C)cc2)=O)C)CCC(C)(O)CC1 N1(CCC)CCCN(C(C2COCCC2NC(=O)C(F)(F)CC)=O)CC1 c1(N2CCS(=O)(=O)NC2)nc(NCCC(O)C2CCC2)c2cccc(Cl)c2n1 C1(C(=O)NC(C=C)(C)CC)CCN(C(=O)Cc2cccs2)C1(C)C C1(NC(c2ccns2)=O)CN(C(C2CCCOC2)=O)CC2(CC2)C1 C1(C(=O)NC2CN(C(c3c(OC)n[nH]c3)=O)C(C)(C)C2)CC(C)(C)OC1(C)C c1(SC)cccc(C(=O)NC2CCOCC2NC(=O)C(C)(C)C(N)=O)c1[N+](=O)[O-] c1(OC(C)C)ccc(NC(c2c(Br)ncn2C)=O)cc1Br C1(CC(=O)NC2C(C)COCC2)N(C(=O)CCC=CC(C)C)CCC1(C)C N1(c2n(C)c(CC(c3ccccc3)(C)O)nn2)CCc2c(cnn(C)c2=O)C1 CC1(C)CN(C(c2c(F)cc(Cl)cc2Cl)=O)CCC1NC(=O)Cc1ccon1 N#Cc1cc(C(=O)C(=O)NCCn2cc(C(C3CC3)C3CC3)nn2)ccc1F C(CN=c1[nH]c(Cl)ncc1Cl)C1(C(=O)OC)CC1 CC1(C)CC(NC(=O)C2=CSCCO2)CCN(C(C2CCn3cnnc3C2)=O)C1 c1(SCC)ccccc1C(=O)NCC1CN(C(C2CC2(C)C(C)C)=O)CCO1 c1(C(C)(F)F)ccccc1C(N1CCN(C(=O)CC2CCC3CC23)CC1)=O N1(C(CCC(C)C)=O)C2CC1CN(C(=O)CNC(=O)COc1ccccc1)C2 N1(C(C(CCC)OC)=O)CCN(C(=O)COc2ccon2)CC(O)C1 N1(C(C(C(C)C)C2CCC2)=O)CCC(C)N(C(C2CN(C3CCC3)C2)=O)CC1 CCCCC(C)C(=O)NCCCN(C(=O)CC(C)(C)OC)CCO c1(N(CCCCOC)C)nc(NCC(C2CCCCCC2)SC)c2ncsc2n1 N1(C(C(CC)n2cncn2)=O)CCOCC1CNC(c1oc(C)nc1CC)=O C(=O)(C(C)SC(F)(F)F)NC(CNC(=O)C1CC1)C1CCC1 N1(C(CC2(C)CCOCC2)=O)CCC2(CC1)CC2CNC(=O)C(F)(F)C(F)(F)F c1(C(=O)NCC2(CNC(CCN(C)CC)=O)CCCC2)cccc(C(C)C)c1N O=C1Cc2cc(NC(C3(C)CC3)=O)ccc2N1.c1(C(=O)N)ccccc1Cl S(=O)(=O)(c1ccc(NC2CC3(C2)CC32CCC2)cc1Cl)N(C)Cc1cscc1Br CC1(NC(c2ccccc2)=O)CCN(C(=O)CC2(O)COC(C)(C)C2)CC1 N1(C(c2c(F)cc(OC)cc2Cl)=O)CCc2[nH]nc(CNC(=O)C(C)(C)F)c2C1 C1(CNC(C=CCOC)=O)CC2(CCOCC2)CN1C(c1cc(O)nc(C)n1)=O C(=O)(C(CC(C)C)ONC(C1CC(=O)NC1(C)C)=O)NC(CCC)CO c1(CC)nnc(C)cc1C(=O)NC(c1ccccc1)CNC(C1CC(C)(O)C1)=O c1(CC)ccc(O)c(C(=O)NCC2CN(C(C3CCCC3(F)F)=O)CC23CC3)c1 C1(CNC(CC(CC)(C)C)=O)CN(C(=O)C(O)CCC(C)C)CCC12CCC2 CCC(N)CCC(=O)NCc1ccc(Oc2ccccc2Cl)cc1 Cc1cc(C)c(C(=O)NCC(C)CNC(c2cn(C(C)(C)C)nc2C)=O)[nH]1 C(=O)(C(C)CC(F)(F)F)N1CCC(C#C)(C(=O)Nc2ccccc2OC)C1 C1(O)(CNC(CCC(C)SC)=O)CCN(C(c2cn(C)c(C)n2)=O)CC1 C1(CN(C(=O)CC2OCCC2(C)C)C)CN(C(=O)COCC2CC2)CCO1 C(=O)(C1NCc2n[nH]cc21)NC(CC(=O)OC)c1ccccc1 C12(NC(C3CCCC3)=O)CCCC1N(C(=O)C1=C(Cl)CCOC1)CCC2 C1(C(=O)NC(CCC)C(=O)NC(COC)CCOC)CCCCC1(C)C CN1CCCC(C(C)(C)C(N2CCC(F)(CNC(C3CC(CF)C3)=O)C2)=O)C1 c1(NC(C(CC)Cc2ccccc2C)=O)ccc(C)nc1CNC(C1CC1F)=O N1(C(c2ncc(OC)cn2)C(=O)Nc2ccccc2)CCC(C)(O)CC1 Cc1nc2sccn2c1C(N1CCC(CNC(=O)C(O)C(C)(C)C)C12CCC2)=O C1(NC(c2cc[nH]c2)=O)CCCC2CN(C(C3(n4cnnn4)CC3)=O)CC12 C1(NC(c2nc(-c3cccnc3)cs2)=O)CCNCC1CO N1(C(CC(CNC(C2CC(OC)(OC)C2)=O)OC)=O)CC2CC(O)CC1C2 c1(CNc2c(C)nc(-c3cc(OC)cc(OC)c3)s2)ccc2oc(C)nc2c1 CC(CC(=O)NC1CCC(N(C(=O)CCC2(C)N=N2)C)CC1)C(F)(F)F N1(C(CC=C(C)C)=O)CCC2(CO)CN(C(=O)CSc3ccc(O)cc3)CC2C1 c1(CN(C(=NC)NCC(=O)NC2CCCC(C)(C)C2)C)ccc(F)c(F)c1 c1(C(N2CCCC(C)C2CCNC(C2(O)CCC2)=O)=O)noc2cc(F)ccc12 C1(C#N)(C(=O)NCC(CNC(CC(C)OC)=O)OC)CC(=O)C1 C1(NC(Cc2cc(C)sc2)=O)CN(C(C2(CO)CC(C)(C)C2)=O)CC2(CC2)C1 C(=O)(C1=CC2CCCC12)NCC1(CNC(c2[nH]c(=NC)sc2)=O)CC1 Cc1ccc(C(=O)NC2(CO)CN(C(c3cc(C(F)F)nn3C)=O)C2)nc1C CCCC(C(O)C(=O)NCC(C)(C)CO)NC(C1(C)CCOCC1)=O N1(C(C(C2CN(C(c3c(C(C)C)nco3)=O)C2)O)=O)CCC(C(F)F)CC1 C(C(C)(C)CC(=O)O)NC(c1cnn(C(C)C)c1Br)=O C12(NC(c3ccnnc3O)=O)CCCC1N(C(=O)C=CSc1nc[nH]n1)CCC2 C(=O)(C1=CS(=O)CCC1)NCC(CN(C(c1c(NC(CC)=O)cccc1)=O)C)C N1(c2cccc(C(C)=O)c2)CCC(N=c2[nH]c3c([nH]c2=O)CC(F)(F)CC3)CC1 N1(C(C2N(CC)CC2)=O)CCC2(CCCC2NC(C2CCCC3CC23)=O)CC1 C1(CNC(CSCC=C)=O)N(C(C2CCC(=O)N2CCC)=O)CCC1(C)C C1(C(N(C2CCN(C(C=CCC)=O)CC2)CC(C)C)=O)Cc2nccn2C1 CC(CNC(C1CN(CC(F)(F)F)C1)=O)CN(C(=O)CCc1cn[nH]c1)C CN1C(=O)C(=O)N(CC(=O)NCc2ccnc(N3CCNCC3)n2)C1=O C1(c2ccccc2)(CNC(=O)NC(c2cc(F)cc(Br)c2)C)NC(=O)NC1=O N1(S(CC=C)(=O)=O)C(CNc2ccnc(C3CC3)n2)CCC1C c1(OC)ccnc(C(N2CC(CCNC(c3conc3C3CC3)=O)C2)=O)c1C C(CCCCCNC(=O)CCc1cnn(C)c1)NC(C1C(CC)CCC1)=O c1(OCC(=O)NC2C(NC(C(C)O)=O)CCCCC2)cccc2cccnc12 C1(CNC(CC(C)OC)=O)CC2(CO1)CN(C(=O)CC1(C(F)(F)F)CC1)C2 Nc1nc2c(cc1C(N1CC3CCC(C1)N3C(C1CCCCO1)=O)=O)CCCC2 N1(C(c2[nH]cc(OC)c(=O)c2)=O)CCC2CCCN(C(C3C4CCCC34)=O)C2C1 N1(C(COCCCCC)=O)CCC(N(CCC)C(C2(C)CCOC2C)=O)CC1 c1(CC(=O)NC2CC(OC)C2)c[nH]c2cc(F)ccc12.N12CCC(CC1C)C2=O Cc1ccc(O)c(C(=O)NC(c2ccnn2C)C(=O)NC(CO)C(C)C)c1 C1(CN(C)C(C2CCCN2C(=O)Cc2cncs2)=O)CCCC2CC12 C(C(C)(C)CC1CN(C(c2nocc2Cl)=O)C1)NC(C(=O)NCCOC)=O N1(C(c2ncc(CC)s2)C(=O)NC2CCC2)CCOCC(C2CCC2)C1 C(C(C)(C)CNC(=O)CC1CC1(Cl)Cl)N(C(=O)Cn1ccc(C(F)F)n1)C NS(=O)(=O)CCCCCC(=O)N1CC(NC(c2cnco2)=O)CC(O)C1 c1(NC(CNC(c2cnc(C(C)O)s2)=O)C2CC2)nc2c(cc1C#N)COCC2 N1(C(c2cc(OC)n(C)n2)=O)CC(C2(NC(=O)Cc3nn(C)cc3Cl)CC2)C1 c1(CC)c(C(=O)N(C)CC2CCCC2NC(C2CSCCS2)=O)ccn1C CC1CCC(CC(=O)NC2(CF)CCN(C(=O)COCCN(C)C)C2)CC1 N1(C(CC2(C)CCCO2)=O)CCC(C2(NC(=O)C(F)=CCCF)CC2)CC1 c1(OC)cc(OC)c(C(=O)NCC(C)N(C(=O)C(C2CC2)OC)C)c(OC)c1 N#CC1(O)CC(C(N2CCC(CNC(=O)C(O)CCn3cncn3)C2)=O)C1 C1(NC2CC(OCC(=O)NC(CN(CC(C)C)C)C)C2)CC2(CC2)C1 CCCCC(CNC(C1CC1C#N)=O)NC(c1ccoc1CC(N)=O)=O Cc1c(C(=O)N(CC(C)(C)NC(=O)CC(C)C(F)F)C)cc(C(C)C)n1C c1(NCCC(C)(C)OC)cc(=NCc2ccc(S(C)=O)cc2)[nH]cn1 N1(C(C2(C(=O)OC(C)=O)CC2)=O)CC(OCCOCC(F)F)C1 Cc1onc(Br)c1C(=O)N(CCC(C)NC(C1CC1F)=O)C N1(C(c2c(CC)nns2)=O)CCCN(C(c2ccc(C)cc2)=O)C(CO)C1 N1(S(CCOC)(=O)=O)CC2CCC1CN2C(=O)CCN1CCCCC1 C(C(=O)NCCCCc1ncc[nH]1)(C1CCCO1)NC(C1CC(CF)C1)=O N#Cc1ccc(C(N2CC3CC2C3NC(=O)CN2CCCNC2=O)=O)c(O)n1 C(=O)(C#CC1CCCCO1)NCC1C(NC(c2ncc(C)cc2F)=O)CCC1 C(=O)(C(O)C(F)F)N(CCN(C(c1cccc(Br)c1)=O)CC)CC CC(C)(O)C#CC(=O)NC(CNC(=O)C(C)(C)CC1CCOC1)CO N1(C(c2c(C)ncnc2)=O)CCCC(C2(NC(=O)CNC(=O)C(C)(C)C)CC2)C1 C1(NC(c2n(CC)nnc2)=O)(CC)CCN(C(=O)Cc2ccc(C)cc2)CC1 C1(NC(CC2(N(C)C)CC2)=O)CC=C(C(=O)NCC(C2CCCC2)O)C1 CC(C)C(C(=O)NOCC(F)(F)F)NC(=O)CCCCC1CC1 N1(C(CC(C(C)C)O)=O)CCC2(CC1)CN(C(c1cccc(N)c1)=O)CCO2 CC1(C)CN(C(=O)C2=NOCC2)CCC1C(N1CC(O)(CO)C1)=O C1(C(N(CCOCCNC(=O)C(CN(C)C)NC(C)=O)CC)=O)CCCNS1(=O)=O N#Cc1cc(Br)ccc1C(=O)NC1CCN(C(C23CC(CO2)C3)=O)C1 C(=O)(CC(C)(C)CC(=O)N1CCC2C1CCCN2C(=O)Cn1nnnc1C)OC N1(C(c2cnc(CC)[nH]2)=O)CCC2CCN(C(=O)Cn3ccc([N+](=O)[O-])n3)C2C1 n1(CCN(CCOCC=C)C)ncc(C#N)c1N C(N=c1[nH]c2c(c(=NC(C)C3CCOCC3)[nH]1)COCC2)C1(C(C(C)C)O)CC1 c1(C(C)(C)OC)nc(C)c(C(=O)N(C)CCNC(c2ccncc2C)=O)s1 N1(C(C(C)Cn2cccn2)=O)C2CCC1CN(C(=O)COCCCF)C2 C#CC(C)(C)C(=O)NCC(C)N(C(=O)C(C1CCOCC1)F)CC C1(N(C(=O)Cc2cnns2)C)CCN(C(=O)C(c2ccccc2)O)CC1 CC(C)(C)C(C(=O)N1CCC(F)(CO)C1)NC(c1ccncc1O)=O C(=O)(C(C)(F)C(C)(C)F)N1CCN(C(CCCCC)=O)C(CCOC)C1 C1(C(N2CCC(C)(NC(=O)C(=O)N=S(C)(C)=O)C2)=O)CCCN(S(N)(=O)=O)C1 c1(C(=O)NCCN(CCC)C(c2cccnc2OC(F)F)=O)ccn(C)c(=O)c1 O=C1NCc2c(C(=O)NC3CCN(C(c4cc(O)ncn4)=O)C3)cccc21 CC1CN(C(=O)CSC(C)(C)C)CC1n1cc(C2C(Cc3cccs3)C2)nn1 n1(C(C)C(=O)NCC2CCS(=O)(=O)C(C)(C)C2)c(=O)oc2ccccc12 C1(NC(C(CC)SC)=O)CN(C(=O)CCNC(=O)OC(C)(C)C)CCS1 C1(C(=O)NC(C)CCN(C)C(c2cncc(N)c2)=O)CCS(=O)(=O)C1(C)C c1(C(C(=O)NC(=O)C=CCC(C2CSC2)C)O)cncn1C C(C)(CCCCNC(=O)Cc1cn(C)nc1C)NC(COCC#C)=O CC1C(NC(=O)C(C)(C)CC(F)F)C2CCN1CC2 N1(C(C(CSC)C)=O)CC(CNC(c2cnc(C(F)(F)F)c(F)c2)=O)C(C)(C)C1 C1(CNC(=O)C2=CCCCCC2)CN(c2ccncc2C#N)CCC12CCOC2 O=C(CNC(=O)C(F)(F)F)N1Cc2ccccc2C(=O)N1 CC(C)C(C#N)C(=O)NC1C=CC(C(=O)NCCc2cc[nH]n2)C1 C(=O)(C(C)C(C)C(C)(C)C)N(CCOC)CCNC(c1cccnc1C1CC1)=O CCC(C)C(C)C(=O)N1CC(n2cc(CN(c3cccc(C)c3C)C)nn2)C1 C1(N)CC2CC(C1)N(C(=O)C=CC=C(Cl)Cl)C2.CCCCCC=CCC=O c1(CC2CCN(c3nc(Cl)ncc3F)C2)ccc(F)c(F)c1.C(CCO)N1C(=O)N1 CCC(CCC(C)C)N1CCCC(C(=O)NCC2CCC(=O)N2C2CC2)C1 Cc1ccc(CCC(=O)NC23CC2CN(C(=O)Cc2cccnc2O)C3)cc1 O=C(C1CCCc2nnnn21)NC1CCOCC1NC(C1(C2CC2)CC1)=O C(=O)(C(C(C)(C)C)OC(C1(c2cc(OC)cc(F)c2)CCCC1)=O)OC C(CC(C)C(=O)N1CSCC1C(N1CCC(C(F)F)C1)=O)=CCC CN1C(=O)CCCC1C(=O)NC1CCCCN(C(=O)C(C)(C)c2ccno2)C1 c1(CNC(c2cnsc2)=O)ccc2c(c1)CCCC2NC(c1cccnc1O)=O c1(C(=O)NC(C(C)NC(CCS(=O)(=O)NC)=O)C)ccc(C#N)c(Cl)c1 C1(C)(C(=O)NCCC(C)N(C(c2cnc(OC)nc2)=O)C)CCCNC1=O C(C(C(C)C)NC(=O)C(F)(F)c1nccs1)NC(CSCCCC)=O C1(CCC)COCCN1C(=O)C(=O)NC1(CO)CC1(C)C C1(NC(c2c(C)cco2)=O)CCCCC1NC(=O)C(C)Sc1nnnn1C1CC1 c1(CC(=O)NCc2cccc(NC(=O)C(Cl)=CCl)c2)ncc(F)cc1F CC1(C)CC(CO)CN(CC(=O)Nc2cnc(Cl)c(F)c2)C1 C1(CNC(c2c[nH]nc2Cl)=O)CC2(CC2)CN1C(C1CC2CC2C1)=O CCC(CNC(c1ccsn1)=O)(CC)NC(=O)CC1CCN(CC(F)F)CC1 C1(F)(C(=O)NCC(NOC)=O)CCN(C(=O)C(C)(C)CSC)C1 CCC(CC(=O)N1CCC1Cn1cc(C2CC23CC3)nn1)C(F)F N1(C(C=CSC)=O)CCC(NC(c2cscc2SCc2ccccc2)=O)C12CC2 C1(C(N(CC(=O)NOCCCOC(C)C)CC)=O)CCOC(C)C1 C=CCC(C(=O)N1CCCCCCC1C(=O)NCCC1CCN(C)C1=O)C(C)C C(=O)(CS(=O)(=O)CCC(F)(F)F)NC1C(NC(c2cc(C(C)C)[nH]n2)=O)COC1 Cc1cc(=NCC(C)N(C(=O)C(C)c2ccco2)C)[nH]c(C(C)(C)C)n1 C(C)(C)(C(=O)NCCC(C1CCC1)NC(c1cn(CC(=O)N(C)C)nn1)=O)OC c1(C(C(=O)NCCOCC)N(CC(C)(C)C2CCOC2)C)sc(Br)cc1Cl Nc1c(C(=O)NCC2(CNC(C34CCCCC3C4)=O)CCC2)sc2nccnc12 C1(OC)CC2N(C1)C2.C(=O)(C(C(C)C)c1ccc(Cl)cc1)Nc1ncc(Br)cn1 c1(C(=O)NCCCCCCCn2cc(CC=C)nn2)ccc(S(C)(=O)=O)c(C)c1 c1(C(=O)NC(CC(C)C)CNC(c2cccc(O)c2)=O)coc2c1C(=O)NCC2 N1(C(CCC)=O)CC(O)C(O)C1CNC(=O)CC1CCN(C)C1=O C1(C(N(C)CC2CCN(C)C2)=O)C2CC1N(C(=O)CC1CCCN1C)C2 C(C(=O)N(C1CCN(C(C2(c3ncco3)CCC2)=O)C1)CCO)(C(C)C)OC N1(C(c2nc(COC)[nH]n2)=O)CCOCC(CNC(C2CC(C)CO2)=O)C1 CCC(CO)C(=O)NCCCCC(C)NC(c1scnc1C1CCCC1)=O C1(NC(c2ccc(Cn3ccnn3)o2)=O)CN(C(C2(Cl)CC2)=O)CC2(CCC2)C1 C1(CCOC)CN(C(c2sc(=N)[nH]c2C)=O)CCN1C(c1ccns1)=O C(CCF)(C(=O)NCc1cc(OC)ns1)NC(c1c(CC)c[nH]n1)=O N1(C(C(c2ccccc2)NC(CC)=O)=O)CCC12CCC2 N1(C(C2C(=C)C2)=O)CCCC(C2(NC(C3CC(O)C3)=O)CC2)C1 N1(C(c2nocc2C)C(=O)NCCCCCC)CCc2c(Cl)cccc21 N1(C(C2(C)C(C(=O)OC)C2)=O)CCC2(CC1)CC(NC(=O)CCCC(C)C)C2 C(=O)(CCCCC(F)F)N1CCC(N(C(=O)COCC2CCCCO2)CCC)C1 CCC(CC(F)(F)F)C(=O)N(C(C)CNC(=O)C(F)C(C)(C)O)C N1(C(C(CC)CCc2ccccc2)=O)CC2CCC1CN2C(=O)C1=CC(C)(C)C1 N1(C(c2cc(SC)oc2)=O)CCOC2CN(C(=O)Cn3cncn3)CC12 C1(C(=O)NCC2C(OCC)CC2)CC2(CCN1C(=O)CC1C=CCC1)CC2 C(=O)(CC(C=C)CC)N1CCC(N(CC#C)C(C2CCCC2C)=O)CC1 c1(-c2n(CC=C)nc(-c3ccnn3C)n2)cc(OC)c(O)cc1C O=C(C1=CC2(CCN(C(=O)C3CC3)C2)C1)N1CCC(CSC)C1 CN1CCc2cc(C(=O)NCC3CC(CNC(=O)C4=CCCC4)CO3)ccc21 C1(CNC(C2(CC)CCC2)=O)CC(O)(CNC(=O)CC=CC(C)(C)C)C1 C(=O)(CC(CNC(c1ccc(F)c(F)c1C)=O)C(C)C)OC C(=O)(C#CC1CCOC1)NCC(c1ccc(C)cc1)NC(C1CC(O)C1)=O C1(C(=O)NC2CN(C3CN(C(c4csc(Cl)c4)=O)C3)C(=O)C2)CC12CC(F)(F)C2 N1(C(CSCCC)=O)CCC(O)(C2CCN(C(=O)C=Cc3cscn3)CC2)CC1 C12(CCNC(=O)C=CC3CCCO3)CCC(C1)N(C(c1ccc([N+](=O)[O-])s1)=O)C2 c1(CC(N2CC3(C2)CN(C(=O)Cc2sc(O)nc2O)C3)=O)ncc(Cl)cc1Cl C1(CC)CC(C(=O)NCC2CCN2C(c2c(N)cnn2C)=O)CCO1 c1(C(N2CCCC(C)(CNC(C(C)C3CC3)=O)C2)=O)cc(C#N)ccc1N c1(CC(=O)N(CC(CNC(CSCCCC)=O)O)C)noc2ccc(OC)cc12 c1(SC)ccc(O)c(C(=O)N(CCNC(C2CCSC(C)C2)=O)C2CC2)c1 C(c1c(Cl)cccc1Cl)=CC(=O)NC1C(F)CCN(C(CCOCCOC)=O)C1 c1(C(=O)NC2CCN(S(=O)(=O)Cc3cccs3)C2)cc(C(F)(F)F)ccn1 C(C)(C)(CN1C(=O)CCc2cc(Br)ccc21)n1cc(COC(C)=O)nn1 C(=O)(C(C)C(CC)CC)NCC(N1CCN(C(CCCC(=C)C)=O)CC1)=O c1(C2(NC(c3cc(=N)[nH]o3)=O)CC2)ccc(Br)cn1 N1(C(=O)C2CC2)CCCC(CNC2(C)C(C(NOC(C)(C)C)=O)CC2)C1 N1(C(CCN(C)CC)=O)C2CCC1C(CNC(=O)Cc1cccc(C(N)=O)c1)C2 c1(CCC)ccc(CC(=O)NC2CC(CNC(C3CC3C)=O)C2)cc1 N1(C(c2c(CC)nc(C)s2)=O)CCP(=O)(OCC)CC1 C(=O)(C1c2c[nH]nc2CN1C(c1cnc(=N)[nH]c1)=O)NCC(C(=O)NC)(C)C N1(C(C=CC2N(C(C(COC)COC)=O)CCC2)=O)CC(OC)CC(C)(C)C1 C1(NC(=O)Cn2cncn2)CCSC12CN(C(C13CCC(F)C1CC3)=O)C2 C(CN=c1[nH]c(C2CCCC2)nc(=N)[nH]1)(C(C)(C)C)NC(C(C)O)=O c1(C(=O)NCCC(C)(C)NC(c2occ(C)c2)=O)cc2n(n1)CC(F)C2 n1(CC(=O)OC)cc(C)nn1.C(=O)(C(CC)OC)N(CCN(C(C)=O)C1CC1)CC c1(C(N(CC(C)NC(=O)CC(=O)c2cnn(C)c2)C)=O)ccc(O)cn1 N1(C(c2cc(SC)oc2)=O)CCSCC1CCNC(=O)CC1CCCO1 CN1CC(C(N2CC3CC2C3C(=O)NC2(C3CCC3)CC2)=O)CCC1=O C1(OC)(OC)COC(NC(N2CCC(C(O)C(F)F)CC2)=O)C1 C1(C2CCN(C(=O)CC3C=CCCC3)C2)CCCCN1C(=O)C(F)CC1CC1 Cc1cc(C(C)C(=O)NCC2CN(C)CCN2C(C2CCCCS2)=O)cc(F)c1 C1(NC(CCOCCCOC)=O)CCCCC1C(=O)NCCCCC1CC1C c1(C(N(C2CC(NC(C3CCCOCC3)=O)C2)C)=O)cc2cccnc2[nH]1 Cc1cc(Cl)cc(C(=O)N(C2CC(NC(=O)CN3CCSCC3)C2)C)c1O CC(=O)CCCC(=O)NC1CC(F)CN(C(=O)CCN2CCN(C)CC2)C1 N12CCC(O)(CC1)C(=O)N1CCC(CC1)C2=O.N1(CC)CCCC(C(F)(F)F)C1 CCC(CC)C(C)C(=O)N(CCCNC(=O)COC(C)(C)C)C1CC1 N1(C(c2ccc(CC)cn2)=O)CC2CC(NC(c3ccn(CCOC)n3)=O)C1C2 N1(C(C(C)=C(CC)C)=O)C(C(N2CC(C(=O)OCC)C2)=O)CC1C C1(CNC(COc2ccc(C)cc2)=O)CCC(C)CN1C(=O)Cc1cnns1 N1(C(C(C)=C(C)C)=O)CC(NC(c2nn[nH]c2Cl)=O)CC2(CCOCC2)C1 c1(C(=O)NCC(C2CCOC2)NC(c2nc(C(C)=O)sc2)=O)nnn2c1CCC2 CCC(N=c1ccnc(N(C)CC2COCCO2)[nH]1)c1ccc(F)cc1F c1(COC)nccc(NCC2COCC(C)O2)n1.C1=NC(=O)C1 N1(C(C(C)S(C)(=O)=O)=O)CC2CCN(C(=O)C(C)(Cl)Cl)CC(C2)C1 C1(CC(=O)NCc2cnn(C3CC3)c2)CCN(C(=O)CC2C=CCC2)C1 N1(C(CCSCC)=O)CCC(C)(C)C(C(=O)NC(c2ccco2)CO)C1 N1(C(=O)Nc2cc(Cl)ccc2Cl)CCN(Cc2cc(Cl)ccn2)CC12CC2 C1(C2CC2)(C(=O)NCCN2C(C)COCC2)CN(C(c2cncc(O)c2)=O)C1 C1(CNC(C(=Cc2ccncc2)C)=O)CCN(C(=O)C(C)OC(C)(C)C)C(C)C1 CCCCCC(O)C(=O)N1CC2C(CC(=O)NC3CCCC4(C3)N=N4)C2C1 CC(CCNC(=O)C(C)n1ccnn1)NC(=O)Cc1cnoc1 C1(C)(C(=O)OC)CN(CC2CCC(=O)N2C)CCO1 c1(C(=O)NCC(CNC(C(C)n2cccn2)=O)O)cc2c(o1)CCCNC2=O c1(NC(c2c(NC(c3ccc(F)c(F)c3)=O)c[nH]n2)=O)ccc(Br)cc1Cl n1(CC(=O)NCC2CC(NC(c3cnn(-c4nccs4)c3)=O)C2)cc(CO)nn1 c1(C(=O)NCCN(C(C(CC)F)=O)CCOCCO)oc(C)nc1C Cc1cc(N)ccc1C(=O)NCC(C)(C)CN(C)C(C1CCN1C)=O c1(C(N2CC(OC)(CNC(=O)C(O)Cn3cncn3)C2)=O)cncc(N)n1 C12(NC(c3cc(C)cc(C)c3)=O)CCCC1N(C(=O)CC1CCCCO1)CCC2 C(=O)(C(C)C(O)CC)NCCC(C)(C)NC(C1(CCC=C)CC1)=O C(=O)(C(C)CC(C)(C)C)NCCC(C)(C)NC(CSc1ccc(C)cc1)=O N1(C(c2cn3ccsc3n2)C(=O)NC)CCc2c(C(=O)OC)n[nH]c2C1 CC(N=c1ccnc(N2CCC3(CCCO3)CC2)[nH]1)c1cccc(F)c1F Cc1nc(C2CCCN(C(C3CCC3CC(=O)O)=O)C2)oc1C(=O)OC(C)(C)C CC(CC(=O)OCC1CSCN1C(=O)C(C)(C)C)NC(=O)Cc1ccccc1 C1(CNC(c2c(CCC)nns2)=O)CCCN(C(C2CC(C#N)(OC)C2)=O)C1 N1(C(c2ccn(C)n2)=O)CCC(C2CCCN2C(C2CCC(=O)N2)=O)CC1 C1(C(c2nnnn2C2CC2)(C)NCc2cc(Cl)ccc2F)Cc2ccccc2C1 CC1CC(NC(C2(F)CC2)=O)CCN1C(c1cccc(Cl)n1)=O C1(CC(C)C)(C(=O)NC2CCCC2CNC(=O)Cc2ccco2)CCCC1 N1(C(C23CC(CO2)C3)=O)CC2CN(c3nnc(O)s3)CC2C1 N1(C(C)C)CCN(C(=O)NCC(C2CCOCC2)F)CC1C C1(CNC(C2CC(OC)C2)=O)CCCCC1NC(c1cn(C)nc1C1CCC1)=O N1(C(C(=O)NC2CC2)=O)CC2(CCCCN(C(c3cc4ncccc4s3)=O)C2)C1 C(=O)(C(=O)N=c1nc(-n2cccn2)[nH]o1)N(c1cc(Br)ccc1C)CCC C1(CN(c2nc(C(C)(C)C)ns2)C)CCCCN1C(C1CCNC(=O)C1)=O C1(NC(Cc2c(C)nc[nH]2)=O)CN(C(=O)Cc2ncccc2C2CC2)CC1(C)C Cc1cc(-n2cc(C3CCCCN3C(=O)CN3CCOC3=O)nn2)cc(C)c1Br S(=O)(=O)(c1cccc2nsnc12)Nc1cccnc1.N12CCC(C1)CN(C)CC2 c1(C(=O)NC2(c3cn(CCC(=O)NC)nn3)CCC2)cc(P(C)(C)=O)cs1 c1(CC(=O)NCC(CNC(C2CCN(CCC)CC2)=O)O)nsc2ccccc12 N1(C(C(CCN(C)C)O)=O)CCC2(CC1)CC2CNC(C1(CF)CCOCC1)=O c1(CN=C(NC(C)C)NCC2CCCN2C)cc(Cl)ccc1N1CCC(O)CC1 N(C(=NCCOC)NC(c1ccnc(C)n1)C)CC(C)OC c1(C(=O)NCC2CCCCN2C(=O)CCCCCF)ccn2cncc2c1 CCC(Cc1ccccc1)CC(=O)N(C(C)CNC(=O)C(F)(F)C1CC1)CC N1(C(COCC(C)C)=O)CCCCC(N(C)C(C2CN(C(C)C)C2)=O)C1 C1(NC(c2cnc(C3CCCC3)s2)=O)CCCCN(CCCC2CCOC2)C1 N1(C(C(CSC)OC)=O)CC(C2CCCCN(C(c3ccc(Cl)c(F)c3)=O)C2)C1 CN1CCCC1(C)C(=O)NCC(c1ccccc1OCc1ccccc1)N(C)C N1(C(CN(CCC#C)C)=O)CCC(CCC(=O)N2CC(CC3CCC3)C2)CC1 c1(C(=O)NCC2N(C(C(CC)Oc3ccccc3)=O)CC2)cnc(N)cn1 c1(C(N(C)CC2(CNC(c3c(C)cccn3)=O)CC2)=O)ccc2nncn2c1 Cc1nc(C)c(CC(=O)NC2C=CCN(C(=O)CC3(O)CCOC3)C2)s1 CC1(C)CN(C(C2(O)CCCCCC2)=O)CC(C)(C)S1(=O)=O S(=O)(=O)(c1ccc(F)c(Cl)c1)N1CC(F)CC(C(=O)Nc2c(NC)cncc2)C1 C1(CNC(C(C=C)O)=O)CC2CCC(C1)N2C(=O)C(c1cccc(Cl)c1)C c1(CN2CCC(=O)N(Cc3ccccc3)CC2)cc2cc3c(cc2[nH]1)OCCO3 C(=O)(CC1C(=O)Nc2c(F)cccc21)NC(CN(C(c1csc(C)n1)=O)CC)C c1(C(N2CCC(C(=O)NC3(C)CC3)CC2)C(=O)N(C)C)ccc(Br)cc1[N+](=O)[O-] C1(CN(C(C2(C)CC(C)=NO2)=O)CC)CC2CCC(C1)N2C(C)=O C12(CNC(CCCCCCC)=O)CCCCC1N(C(c1cc(C#N)no1)=O)CC2 Cc1csc2c(CC(N3CCCC3C(=O)N(C)C3CC3)=O)cccc12 N1(C(CCN(C)CC)=O)CCC2CN(C(c3cc(C#N)ccc3F)=O)C(C)C12 c1(C(C)C)ccc(OCCC(=O)NCCC(C)NC(C2CCC23CCC3)=O)cc1 C(=O)(CCCCCF)N(C)CC1C2CN(C(C(C)OCC#C)=O)CC21 Cc1ccnn1CC(N1CC(CNC(=O)C(F)C2CCC2)C1)=O C1(CNC(=O)Cc2ccon2)COCC1NC(C1(c2ccccc2)CCC1)=O Cc1cc(C(=O)NC2CCN(C(=O)CCn3cccn3)C(C)C2)ncc1Br C1(F)(NC(CN2CC(C)(OC)C2)=O)CCC(NC(C2CN(C(=O)CCS(C)=O)C2)=O)C1 C1(C(=O)NC2CC(CCNC(CSCCOC)=O)C2)CCOC(C(C)C)C1 CC1CN(C(=O)CCOCC(F)F)CCN(C(c2cc(C(C)(C)C)on2)=O)C1 N1(C(c2c(OC)nccc2)=O)CCC(NC(c2csc(C)n2)=O)C(F)C1 N1(C(CCCCC)=O)CCCOC(CNC(c2n[nH]cc2Br)=O)C1 N1(c2nc(C)nc3c2cc[nH]3)CCC2(CN(C(C3CCCC3O)=O)CC(C)O2)C1 C(CN=c1nc2sccc2c(NCC2CCC(=O)N2)[nH]1)C1CC(C)C1 C(=O)(C1Cc2ccc(F)cc21)NC1CC2(CCCN(C(C(CC)(C)CC)=O)C2)C1 C1(NC(C(CC)N(C)C)=O)CN(C(c2c(Cl)ccc(O)c2Cl)=O)CC2(CCC2)C1 c1(CC(=O)NC2(C3CCCN3C(c3cnc(Br)s3)=O)CC2)nc2ncccn2n1 c1(C(N2C(CNC(c3c(C)n(C)cc3)=O)CC2)=O)cc2n(c1)CCCC2 c1(C(=O)NCC(CC)(C)NC(c2n[nH]cc2[N+](=O)[O-])=O)ccc(C)c(Cl)c1F N1(C(c2ccn(Cc3cn(C(C)C(=O)O)nn3)c(=O)c2)=O)CC(=O)NC(=O)C1C c1(OC)ccc([N+](=O)[O-])c(C(N2CC3C(NC(=O)CCC#N)C3C2)=O)c1 CC1(C(=O)NC(CNC(C2CCCN2N=O)=O)C2CCC2)CS(=O)(=O)C1 C1(C(C(=O)N(C2CC2)CC)C)CCCN(C(C2CCC2)=O)C1 c1(C(N2CC=CC(NC(C(C)SC)=O)C2)=O)c[nH]c2ncc(Br)cc12 CC1CCC(CNC(=O)C(C)(C)C(F)F)CN1C(c1coc(C#N)c1)=O C1(NC(CC2(C)CC2(F)F)=O)CCN(C(c2ccncc2N)=O)C1C1CC1 C(=O)(C(C)CCC(C)(C)C)N1CC(N(C(C2C(COC)(COC)C2)=O)C)C1 CC1CC(CNC(=O)CC2CCC3(CC2)CC3)CCN1C(=O)CC1(C)CCCO1 C1(NC(C(=O)NCCOC)=O)(CO)CN(C(=O)CCCOC2CCOCC2)C1 Cc1cccc(C)c1C(=O)NC1CC2(C1)CC2NC(=O)CC1(C2CC2)CC1 C1(N(C(C2(COC)CCCC2)=O)CC)CCCN(C(c2cc(F)cc(F)c2)=O)CC1 c1(OC)ccc(C(=O)NC(C)COCC(F)(F)F)c(Br)c1F c1(N(CC(=O)NCC)C)cc(C)nc(NC2CCCOC2c2nccn2C)n1 C1(NC(C2C(C(=O)OC)C=C2)=O)CC2(CCC2)C1OC C1(CC(=O)N(CCNC(c2c(SC)n(C)nc2)=O)C2CC2)CCC(F)(F)CC1 CC1(C)OCc2c1n[nH]c2C(=O)NC1CC(NC(c2cnc(S)nc2)=O)C1 N1(C(C2CCCN(C)C2)=O)CCC(C(=O)NC(c2ncc(F)cn2)C)C1(C)C C1(NC(C=CC(CC)C)=O)CCCCC1CC(=O)NC1CCCC1 C#Cc1ccnc(C(=O)NCCN(C(=O)CCc2nncs2)CC(C)O)c1 N1(C(c2c(C)nc(C(C)C)s2)=O)CCOCC(NC(=O)C(C)(O)C(C)C)C1 C1(F)(CNC(=O)Cc2cnns2)CCC(CNC(=O)CN2C(=O)CCC2=O)C1 c1(C(=O)NCc2c(CNC(CC3C(C)OCC3)=O)nco2)c(F)ccc(F)c1Cl C1(CNC(CC(CC)C2CC2)=O)CCC2(CN(C(c3cc(CC(C)C)c[nH]3)=O)C2)O1 CC1(C)CC=C(C(=O)NCC23CCC2CN(C(c2ocnc2C2CC2)=O)C3)CC1 C(CCCCNC(C12CCC1CC2)=O)NC(=O)CCF CC(C)(O)CC(=O)NC(C)(C(N1CC2CCC1C2)=O)C1CCC1 C1(F)(C(N2CCC(C(C)C)(CO)C2)=O)CCCN(C(=O)CNc2ccccn2)C1 N1(C(C(c2cccc(C)c2)C)=O)CC2(CNC(c3c[nH]nc3C)=O)CC(F)(C1)C2 c1(OC)cc(C)cnc1C(N1CCCC(CNC(=O)C(O)CSC)CC1)=O C1(C(C)(C)C)CC(CNC(=O)CCc2ccsc2)CN(C(c2ccon2)=O)C1 N1(C(C2CCCCN2Cc2cccnc2)=O)CCC(C2CCOC2)CC1 C(=O)(C1=NN(c2ccccc2)C(C(=O)NCc2coc(C)n2)C1)OC C(=O)(C(C)(F)C(C)(C)F)N1CC(N(C(=O)CCC(c2c(F)cccc2F)=O)C)C1 C(=O)(C(C)CCCC(C)C)NC(C(=O)Nc1c(OC)ccc(C)c1)(C)CO Cc1ccc(CNC(=O)COC2CN(C(c3ncccc3N)=O)C2)c(F)c1 C1(CCOC)CN(C(c2cnsn2)=O)CCN1C(=O)CC1(C)CCC1 CCCC(C)(CC)C(=O)N1CC(C)C(C)(CNC(=O)CCCc2ccccc2)C1 N1(C(C=CC(=O)N(C)C)=O)CC(F)(F)CC1CO.c12cc(no1)C(=O)NC2 c1(C(=O)OCC)ccc(C(N2CC(NC(c3cccc(C)n3)=O)C(C)C2)=O)cc1 CN1CC=CCC1CC(=O)NCCN(C(C1(CO)CC1(F)F)=O)C1CC1 c1(C(N2CCC(CNC(C(COC)OC)=O)CC2C)=O)ccc2ccccc2c1 C=CCC(CC=C)n1cc(CONC(=O)Cc2cccc(C)c2)nn1 CCCC(C)(O)CC(=O)NC1C=CCC(C(=O)NC2CCN(C(C)=O)C2)C1 C(=O)(C1=COCCO1)NCCCN(C(=O)CCc1c(F)cccc1F)C C1(C(N(CCC)CCNC(C2(C)CCC(=O)N2)=O)=O)CCCCCC(=O)C1 C1(NC(CC2CCN(C(c3c(C)nn[nH]3)=O)CC2)=O)CC2CCC(C1)N2C Cc1nnc(CCNC(=O)C(CC2CCCC2)NC(=O)Cc2cnsc2)n1C c1(CC(C)C)ccc(C(=O)NCCCN(CCO)C(C2CC(OC(F)F)C2)=O)s1 N1(C(=O)CC2CCC2)CCN(C(C2CC(F)C2)=O)C(c2ccccc2)C1 C(CC(C)C(=O)NC(C1CCN(C(=O)CCc2cccnc2F)C1)(C)C)OC c1(C(N2CC3(CC(NC(C4CCC5(CCC5)C4)=O)C3)C2)=O)cnc2n1CCOC2 Cc1cc(O)c(C(N2CC(N(C(=O)CN3C(=O)CCC3=O)C)C2)=O)nn1 C(=O)(N=c1ncn(C(C)(C)C)[nH]1)N(C(c1ccccc1)C)CCOC c12ccc(cc1)C(C)NC2.n1(CC=C)cc(C(=O)NC(=O)CN(C)CC)cn1 C1(NC(C2CCCOCC2)=O)CN(C(C2SCCS2)=O)CC12CC2 C1(COC)(CNC(=O)CNCCCc2ccc(C(=O)OC)cc2)CCC(=O)N1 C=CCC(C(=O)NCCN(C)C(c1[nH]c(=N)sc1CC)=O)C(C)C c1(C(=O)NCC2N(C(C=C3CCN(C)CC3)=O)CC=C2)csc2nccn12 c1(CCC)nc(C)c(C(N2CCCC2C2(NC(c3cnn(C)n3)=O)CC2)=O)o1 c1(C(N2CCCC(N(C(=O)CC3CCCC3(F)F)C)C2)=O)ccc(N)c(Br)n1 C1(CNC(CC2C(C)(C)C2(C)C)=O)CN(C(=O)CC2CCCOC2)CCCO1 C(C(=O)N1CC(F)(CNC(C2CC2C(F)(F)F)=O)C1)(C(C)C)c1cc(C)no1 C(C(=O)Nc1ccnc(N2CCCCC2)n1)(C(C)C)n1ncc(C)c1 c1(C(=O)NC(C(C)NC(c2c(C)con2)=O)CO)cnn(-c2ccccn2)c1C C1(NC(C2N(C)C(=O)CCC2)=O)CCC2CCN(C(C3(n4ccnn4)CC3)=O)C12 C1(C(N2CC(OC)(CO)C2)=O)CCCN(C(=O)C(n2cc(C)cn2)C)C1 N1(Cc2cccc(N(C)CC)c2)CCC2(CCCOC2)C1 CC1(C)CC(C(N2CCC(C3CCC3)C2)C(=O)C)CC(C)(C)C1.CCCN c1(C(N2C3CN(C(CC(C)=C(C)C)=O)C(C3)C2)=O)cc2ccc(N(C)C)cc2[nH]1 c1(NC(CC)=O)ccc(Nc2ccncc2F)cc1.C12CCN(C1)C(=O)C2 N1(C(C2=CC(C)CC2)=O)CCCC2(C1)OCCCO2 C(=O)(C(F)CC(C)(C)C)NCc1cc(C(N2CCCC(C=C)C2)=O)sc1 Cc1cc2ncnn2cc1NC(c1cnc(CN)nc1C)=O c1(C(=O)NCCN(CCOC)C(C2CCCCC2OC)=O)c(C)cnn1C N1(C(c2c(NC)cnc(Cl)c2)=O)CCC(NC(=O)C(CO)N(C)C)C12CCC2 c1(OC)nccc(C(=O)NC2CCC2NC(c2sccc2C(C)C)=O)c1F N#Cc1c(F)cc(C(=O)NCC2(NC(c3cnc(O)o3)=O)CC2)cc1F C1(C(=O)NCC(CCO)OC)CCCN(C(C23CSCC2C3)=O)CC1 c1(C(=O)NCC2C(CC(=O)N(C(CC)CSC)C)C2)ccc(Cl)cn1 C(C1(C)CCOCC1)=CC(=O)N(C)CCN(c1ncc(Br)c(O)n1)C c1(C(=O)NC2C=CCN(C(CC(CN(C)C)O)=O)C2)c2ccccc2nn1C CN(C)NC(=O)CCC(=O)NC1CCC1CNC(=O)CC1CCC(O)C1 CCCCC(CNC(c1cccc(COC)n1)=O)NC(C1(C(F)F)C=CCC1)=O C(=O)(C1CCCc2ccccc21)NCCCNC(CN1CCC(C)(C)C1)=O C1(CC=C)(NC(=O)C=CC(C)CC)CCN(C(=O)CCS(N)(=O)=O)CC1 c1(CCC(N)=O)nc(CSCc2ncccn2)n(-c2ccc(Cl)cc2)n1 C1(NC(CN(C)CC)=O)CCN(C(=O)CN2CCOCC2=O)C(C2CC2)C1 c1(N(C)CC2CCCN2C(=O)C#CC2(C(F)(F)F)CC2)ncc(C#N)cc1F N1(C(c2nc(C)[nH]c2Br)=O)CCN(C(C2CC(O)C2)=O)C(C)C1C C1(C(=O)NCC2N(C(c3c(C)cncc3)=O)CC(O)C2)CCCCC1(F)F Cc1cc(C(N2CCCC(CN(C)C(C3CCCSS3)=O)C2)=O)cc(C)c1 Cc1c(C(N2CC3(CCC3NC(c3sccc3F)=O)C2)=O)cncc1Br N1(C(c2cnc(CCC)s2)=O)CCC(NC(c2cnoc2CC(C)C)=O)C(O)C1 Cc1cc(C(=O)NCC(Cc2ccccc2)NC(=O)C=CCO)cn1C(C)C C1(C)(CC(=O)NCC(C)N(C(C2CC(C#C)(O)C2)=O)C)CCS(=O)(=O)N1 Cc1cc(O)ccc1CC(N1CC2CC2(NC(=O)CCN(C(=O)CO)C2CC2)C1)=O C1(C(=O)NC2(CO)CC2)CC2(CC2)CN1C(=O)CC1CCCOC1 N1(C(Cc2ncc(C)[nH]2)=O)CC(CNC(c2ccc(Cl)cn2)=O)C(C)(C)C1 CCCCCCCCCCCC(=O)N1CC2CC1CN(C(=O)CC=C(Cl)Cl)C2 N1(C(C(C)CN(C)C)=O)CCCCCC(NC(=O)COCC2CCCC2)C1 C1(C(=O)OC)CCCN(C(=O)C(N2CCC3(CC2)CC3)=O)CC1 c1(C(N2CCC(NC(=O)COCCc3cccs3)C2)=O)ncccc1C(F)F c1(C(C)NC(N(CCC)C(C)C)=O)ccc(-n2ccnc2)cc1 CCC1=C(C(=O)NCC2CCN2C(=O)CC(C)OC)CCCO1 C(=O)(CC(O)C(C)(C)C)NCC1(C)CCCN(C(c2n(C)ncc2)=O)C1 N1(C(C2C(OCC)C2)=O)CCC(OCCCNC(=O)Cn2nccn2)CC1 C1(CNC(=O)CO)CN(C(c2ccncc2-n2cccn2)=O)CC1(F)F C1(NC(C2(C)CCCN2C(=O)OC(C)(C)C)C)CC2OC(C)(C)OC2C1 N#Cc1ccc(C(=O)NCCNC(c2ccnnc2Sc2ccccc2)=O)o1 N1(C(c2c(CC)nn(C)c2)=O)CCC2(C1)CN(c1cc(C)nc(C(F)(F)F)n1)C2 C1(C2CCN(C(=O)CNC=O)CC2)(C(=O)NCC(CCC)O)CCOCC1 C12(NC(=O)CCC(F)(F)F)CCCC1(F)CN(C(=O)CCC1CC1(F)F)C2 c1(C(=O)NC2CCCC(CNC(C(C)=C(C)C)=O)C2)c(F)ccc(F)c1O c1(C(N(C(CC)C(=O)NOC2CC2)C)=O)cc(C)c(C)cc1C C(=O)(C1Cc2ccccc21)N1C(C(=O)NCC(C(CC)C)CO)CCC12CC2 Cc1ccc(CN2CC(C(=O)NC3CN(C(c4ccnnc4)=O)C3)CC2=O)cc1 C1(CNC(C2CC(OC)C2)=O)CN(C(c2cc3ccsc3s2)=O)CC(C)(C)O1 c1(C(N2CC(C)CC(CNC(C(C)C3CCC3)=O)C2)=O)c[nH]c2nccc-2c1 C(=O)(CS(=O)(=O)C1CC1)N1CC2C(CCNC(c3ncc(NC)nc3)=O)(CC2)C1 N1(C(c2c(OC(F)F)cccc2Cl)=O)CCC2CN(C(c3cnc[nH]3)=O)C2C1 CCC(CCC(=O)Nc1cnc(C)c(Cl)c1)NC(C1CC(C)(C)CO1)=O C1(C(=O)NC(c2cccc(Cl)c2F)C)CCC(=O)CC1C c1(C(N2CC(CSC)OCC2)C(=O)NCC2CC2)ccc2ccc(F)c(F)c2n1 N1(CC2NC(=O)OC2)CCCC(CNC(C2CC(c3ccccc3)C2)=O)C1 Cc1cnn2ccc(C(N3CCCC4(NC(=O)CCC(F)F)CCCC34)=O)nc12 c1(C(=O)NCC(CNC(C2C(C)OCCC2)=O)C(F)(F)F)[nH]nc2ncccc12 c1(N(CC#CC)C)nc(=NCC2CCC(F)C2)nc(N2CCOCC2)[nH]1 CC1COCC1(c1nnnn1C1CCCC1)NC(c1nnnn1C1CC1)C C(=O)(C(C)C(O)CC(C)C)N1C(CNC(c2c(C)c(F)cnc2)=O)CC2(CC2)C1 C(C(N=[N+]=[N-])C(=O)N(C)CC1CN(C(c2cc(C)cnc2C)=O)C1)OCC c1(C(N2CCC(C(C)NC(C3(C#N)CCC3)=O)CC2)=O)cc(C(F)(F)F)ccc1O c1(-c2nn(CCOC)c(CCCS(=O)(=O)N(C)C)n2)cc(F)c(N)c(F)c1 CC1CCC(C(F)(F)F)CN1C(c1ccc(CCN)cc1F)=O C1(C(=O)NC2CCC(NC(C3CC3c3cccs3)=O)C2)(CO)CC(F)(F)C1 C1(CNC(c2c(C)ccnc2)=O)CN(C(=O)Cc2ccoc2)CCC12CCC2 C(CCOCCO)(C(=O)NC(c1ccn(C)n1)C)NC(C(CSC)O)=O c1(C(N(CC(CC)NC(=O)CC2C=CS(=O)(=O)C2)C)=O)nc2nc(C)ccn2n1 c1(CC)ccc(C(N2C(CNC(c3n[nH]c(C)c3Cl)=O)CC3CC23)=O)cn1 Cc1cccnc1C(=O)NC1C2CN(C(c3ccncc3Br)=O)CC12 N1(C(C2CN(Cc3cc(C(=O)OC)[nH]c3)CC(F)C2)=O)CC(F)(F)CC1C#N C#Cc1cc(C(=O)NCC(C(C)C)NC(=O)C(C)(O)COC)ccc1C C1(C(=O)NCc2scc(CNC(c3n(C)cnc3)=O)n2)CCC2(C1)CC2(F)F N1(CC2(O)CN(C(C3(SC)CC3)=O)C2)C(C)CCC1C.C12(CCC1)C(=O)NC2 C12(NC(C(=O)NCCOCCOC)=O)CCCN(C(=O)CCC(C)(C)C)CC1C2 c1(NCC(CSC)OC)ccc(S(=O)(=O)NCc2cncs2)c(Cl)c1 Cn1c(CN(C2CCS(=O)(=O)C2)CC2CCCO2)nc2ccccc2c1=O c1(C(=O)NC2C(O)CCN(C(CCOCC#C)=O)C2)ccc(OC)c(OC)c1C C(CCCC(C)NC(=O)Cn1ccsc1=N)NC(C=C(C)Cl)=O c1(C(N(CC(C)NC(=O)CCOC2CC2)CC)=O)csc(Cl)c1Cl C1(C(=O)NCC(C)N(C(c2c(SCC=C)cccc2)=O)C)CC2(CCCC2)CO1 c1(OC(C)C)ccc(Cl)c(C(N2CCCC(O)(CNC(c3ccco3)=O)C2)=O)n1 C1(C2CC2)(CNC(c2cc(OC)c(C)nc2)=O)CCN(C(c2c[nH]nc2C)=O)C1 N=c1ccc(C(=O)NC2C=CC(CNC(c3cn(CC(F)F)cn3)=O)C2)n[nH]1 c1(NC(C2CS(=O)(=O)CC2N2CCOCC2)=O)nc2cccc([N+](=O)[O-])c2s1 c1(C(C)NC(C(=O)NCCCC)CC)ccc(OC)cc1 c1(C(=O)NC(CNC(C(C=C)(C)C)=O)(C)CO)cc(C)cc2c1NCCC2 Cc1cccc(N)c1C(=O)NC1CC(O)CN(C(=O)CC2CSCCS2)C1 C1(C(=O)NCC2C(C(F)(F)F)CCN(C(CSC)=O)C2)CCc2nn[nH]c2C1 Cc1cc(C)c(NC(=O)CCC2CC(NC(=O)C=CC(=O)NC3CC3)C2)s1 c1(NC(C2N(Cc3c(C)n(C)nc3)CC2)=O)ccc(Cl)c(F)c1Cl N1(C(c2cc(C)no2)=O)CC2CC(C1)CN(C(c1ccnc(Cl)c1N)=O)C2 c1(C(=O)NC2CCN(C(=O)Nc3c(Cl)cccc3Cl)CC2)ccc2c[nH]nc2c1 CC(C(=O)NCCCOCCO)C(C)NC(c1nccnc1O)=O c1(CC(=O)NCC2CN(C(C=CCOC)=O)C3C2C3)c(C)nn(C)c1Cl C1(C(N2CCC(NC(CCC(=C)Br)=O)C2)=O)CCC(C)(O)CC1 c1(CN2C(C(=O)NC3(C(=O)OCC)CCC3)CC(O)C2)cc(I)ccc1F c1(CCC(=O)NCCCN(CCCNC(C2CC23CC3)=O)C)ccnn1C C(=O)(C(C)CC(C)(C)C)N1CCC(=C)CC1C(=O)NCCc1nc(C)oc1C Cn1ccc(=O)c(C(N2CC=CCC2C(=O)NC2CC(O)C(F)C2)=O)c1 CCCCCC(C(=O)NCC1CCN(C(=O)C=CSc2nc[nH]n2)C1(C)C)C(C)C c1(CN(C)C(C2(CO)CN(C(=O)CCNC(=O)N(C)C)C2)=O)ccon1 Cn1cc(C=CC(=O)NCCC2CCCN(C(=O)COC3CCCC3)C2)cn1 N1(C(COc2cc(C)on2)=O)CCC(C)CC1CNC(=O)C(C)NC(N)=O C1(NC(C=C(C)Cl)=O)CC2CC1CN(C(c1ccc(S(N)(=O)=O)s1)=O)C2 C1(NC(CCCC#CC)=O)CCOC12CCN(C(=O)CC1NC(=O)NC1=O)CC2 C1(C(=O)NCC(=O)NCC2CC(F)(F)CO2)(OCC)CCOCC1 C1(NC(CCc2c(C)cccc2)=O)CC2CC1N(C(C1(F)CC1C)=O)C2 N1(C(c2ccc(C#N)cc2)=O)CCN(C(C2CCSCC2)=O)CC(CO)C1 CCC(C)C(C)C(=O)N1CCC1CNC(c1ccc(-c2ccco2)s1)=O Cn1cccc(C(=O)NC2(C3CCCN3C(=O)C(F)CC3CC3)CC2)c1=O N1(c2cc(SC)nc(C)n2)CCC2CN(C(c3cnc(N(C)C)o3)=O)CC12 N1(C(C(CC2CCOCC2)NC(c2c(C)scc2)=O)=O)CC(CO)C1(C)C CSC1=C(C(=O)NCCC2(O)CCCN(C(=O)Cc3cnnn3C)C2)CCCC1 c1(C(=O)OCC(=O)N(c2cscn2)CCC(C)N(C(C)=O)C)n[nH]c2c1CC1CC21 c1(C(N2C(CC(N3CCC(C)CC3)=O)COCC2)=O)c2c(nn1C)CCC2 c1(CC(=O)NCC2CN(C(c3cc(O)no3)=O)CCCO2)n[nH]c2c1CCCC2 C1(NC(C(C)C)=O)COC2(CCN(C(=O)C(C)n3ccnc3)C2)C1 c1(C(=O)NC2(C)CC(C(N3C(C(=O)OC)C=CC3)=O)C2)ccc(C#N)c(C)n1 N1(C(c2c(SC)cccn2)=O)CCCCC(C2CN(C(=O)C(C)=C(C)C)C2)C1 N1(C(c2c(C)nn(C3CC3)c2)=O)CC2CCC(C1)N2C(C1CCCC1C)=O CC1CC(NC(=O)Cc2ccc(F)c(F)c2)CN(C(c2cc([N+](=O)[O-])n[nH]2)=O)C1 CCC(CCCC(=O)N(C1CCCC1(C)O)C)NC(=O)C(C1CCCCC1)O N1(C(C(CCN(C(=O)OC(C)(C)C)CCO)(C)C)=O)CC2(CCCO2)C1C1CC1 C1(NC(c2ccc(Cl)cn2)=O)CCN(C(c2csc(Cl)n2)=O)C12CC2 CC1OCCC1CN(C(=O)C=CCC1(NC(=O)Cc2ccoc2)CCC1)C c1(C(N2C3CN(C(c4cnc(O)[nH]4)=O)C(C3)C2)=O)c(Cl)cc(Cl)cc1Cl c1(C(=O)NC(CNC(C=C(C)Cl)=O)CO)cc2cc(C)ccc2[nH]1 C(=O)(CC(C)C(=O)NC(Cc1ccccc1Br)C(N1CCC(F)(F)C1)=O)OC C1(O)(CCNC(C(C)N2CCC2)=O)CCCN(C(c2cc(=O)c(O)c[nH]2)=O)C1 C(=O)(CC(C(F)(F)F)n1cccn1)N(CC(C)(C)CNC(=O)Cc1ccsn1)C N1(C(CCOCC)=O)CC(NC(=O)C2=C(Cl)CC2)C2CC12 CC1(F)CN(C(=O)CN2CCOCC2)CCN(C(=O)CC2(CO)CCCC2)C1 C1(C2(NC(C3CCN(C(=O)c4occc4C)O3)=O)CC2)(OC)CCC1 N1(C(c2c(C)ccs2)=O)CCC(C)(C)C1CC(N1CCC(C)(CO)C1)=O N1(C(CC(CC)NC(CCCC#C)=O)=O)C2CCC1COC2 CC1=CCC(C(=O)NCCC2(C(N3CCSCC3CN(C)C)=O)CC2)CC1 c1(OC)ccccc1CC(C)(C)C(=O)NCC(CNC(C1CC1(F)F)=O)CO c1(C(=O)NCC2CC(NC(C=Cc3n(CC)ncc3)=O)C2)c(Cl)c(C)nn1C Cn1ncc(C(=O)NC(CC2CCC2)C(=O)NC2(c3nc[nH]n3)CC2)n1 C(=O)(CCS(=O)(=O)CC(C)C)N1CC(NC(c2ncnc(C)c2C)=O)C2C1C2 C(=O)(C(C(C)(C)C)C1CCC1)N(C)CC1(NC(c2ccc(OC)cn2)=O)CC1 N1(C(c2c(CC)scc2)=O)CCN(C(=O)C(CO)N(C)C)CCC1C C1(C2C(C)CCC2)NC(=S)N(c2ccc(F)cc2F)C2=C1C(=O)N(C)C2C C(CNC(C1CCO1)=O)(C(=O)N1CC(O)(c2cc[nH]n2)C1)N(C)C C1(C(N(C(COC)COC)C)=O)C=CCCN1C(=O)CC1CCC(C)(C)C1 C1(C)(C(=O)NC(C)C(=O)NCCC(Cl)Cl)C=CCCC1 CC1CC(C)C1CNCc1cn(CCNC(=O)OC(C)(C)C)cn1 N1(C(C2CC(CCC)OCC2)=O)CC=C(CCNC(c2cn(C)cc2C)=O)CC1 C1(NC(CCOCCOC)=O)CN(C(C2CC(C)(C)O2)=O)Cc2ccnn2C1 C1(CN(C(C2(COC)CCC2)=O)C)CCN(Cc2ccccc2)C1 C1(CNC(C2=NOC(C)C2)=O)C(C2CC2)CCN1c1nnc(C(N)=O)s1 C=C1Cn2c(C(N3CC4CCC4(NC(C4CC4(C)CC)=O)C3)=O)nnc2S1 c1(CCC(=O)NC2CC(NC(COC(CC)C)=O)C2)ccc(F)cc1Br C1(NC(c2cc(C)n(C(F)(F)F)n2)=O)CC(C)CN(C(c2ccc(O)nc2)=O)C1 Cc1cc(C(N2CCCC(CF)C2)C(=O)NCc2cccs2)cc(C)c1F c1(OCC=C)ccccc1CC(N1CCC(N(C(=O)C(C)CCC)CC)CC1)=O c1(C(=O)NCC(CC)O)cccnc1CNC(=O)CCOCC1CCC1 c1(C(C(=O)OCC=CC)C)cccc(NC(Cc2ccccc2)CO)c1 CC(C)C(C#N)C(=O)N1CCOCCC1C(=O)NC(C)C(C)(C)C N1(C(c2c(OC(F)F)cc(C)s2)=O)CCN(C(C2CC(C)C2)=O)CC(O)C1 c1(C(=O)NC2C(C)(C)N(C(=O)Cc3ccsn3)CC2)noc2c1COCC2 CC(C)CCCC(=O)NCC1CN(C(=O)C2=CCCCO2)CC1O C(=O)(C1CCC(=O)c2cccn21)N1CCN(C(C(C(C)C)NC=O)=O)CC1C C(CN=C(NCC1CCC1)N1CCOC(C2CCCO2)C1)c1ncc(C)cn1 Cc1nocc1CNC(=O)C(C1(O)CCC1)NC(=O)C(C1CC1)SC Cc1c(C(N2CC=CC2CNC(=O)C(C)C(C)C)=O)cc([N+](=O)[O-])cc1Br C=C(CNC(=O)CC(C)C(C)(C)NC(=O)Cc1cnc(C)s1)c1ccccc1 N1(C(c2cnc(C)s2)=O)CCC(C(CO)NCC2(c3ccncc3)CC2)CC1 C12(C(=O)NCC3(CC(=O)NC(c4nc(C)on4)C)CC3)CCC(CC1F)C2 C1(NC(C(CCCC)C)=O)CCC2(CC1)CN(C(=O)CSc1ccc(OC)cc1)C2 C1(NC(c2cnc(CCCC)s2)=O)CCN(C(c2oncc2CC)=O)CC1(C)C C1(C(N(C)CCN2CCCCC2)=O)N(C(=O)CCCC#N)CC12CCCC2 c1(C(N(c2ncccn2)CC(C)C)=O)nnn(C)c1N C1(CC(=O)NCCCN(C(C2CCCCO2)=O)C(C)C)(OC)CCOCC1 N1(C(c2cnccc2)c2nc[nH]n2)CCCN(CC2CCCOC2)CC1 C(=O)(C1=CS(=O)(=O)CCC1)NC(C)C(C)NC(c1cn2c(n1)CCCC2)=O CCC(C)(COC)C(=O)NCC(CO)NC(=O)C(C1CCCCC1)N(C)C(C)C C(=O)(C(C)C(C)C)NCC1C(NC(c2nc(C(C)C)oc2)=O)COC1 c1(C(N2CCC(CCC(=O)NC(C(N)=O)C3CC3)C2)=O)cnc(O)c(Cl)c1 CC1CN(C(C2CN(C(c3c[nH]nc3C(F)F)=O)CC2(C)C)=O)CC1(C)CO N1(c2cc(C)nc(CO)n2)CCC2(COC(CNC(=O)C=C3CCCCC3)C2)C1 C1(C(N(CC=C)CC)=O)CC(O)CN1C(C1CCNC1=O)=O Cc1cnc2n1CCC(C(=O)NC1(Cc3ccccc3)CCOCC1)C2 Cc1ccc(O)c(C(=O)NCCCCCCNC(c2cc(C)[nH]n2)=O)c1 c1(COC)nn(C)cc1C(=O)NCC1C=CCN1C(=O)C(O)COC N1(C(c2on(C)c(=O)c2)=O)CC2(CCN(C(C3(CC4CCC4)CC3)=O)C2)C1 c1(C(N(CC(C)(C)NC(C23CCCC2C3)=O)C)=O)n[nH]c2c1CCC2 Cc1cc(C(=O)NCCC(C)(C)CNC(=O)CC2CCCCO2)[nH]c1C.C(C)(C)C CCC(C)(C)C(=O)C(=O)N1C(OC)CCC1c1ccccc1 C(C(O)C(=O)NCC(C1CC1)NC(=O)CSC)=CCCC N1(C(C2(C)CC(F)C2)=O)CCN(c2ccc(C(F)(F)F)cn2)C(CCO)C1 c1(NC(c2c(C)noc2C)=O)c(Cl)ncn(C)c1=O C(=O)(CCC(C)(F)F)N1CCC(N(C(c2cccc(SCC#C)c2)=O)CCC)C1 c1(C(=O)NCC=C)ccc(C(=O)NC(C)(CNC(C2C=CCC2)=O)C(C)C)cc1 c1(-c2cc(NCc3c(C)cccn3)ncc2)cccc(O)c1C C1(NC(C(C=C)(C)CC)=O)CC2(CCN(C(=O)CNC(c3cscn3)=O)CC2)C1 CCCC1C(=O)NC2(CCC2)C(=O)NCCCN1CC(C)C.C(=O)(N(C)C)OC C1(C(=O)NCC23CC(C(=O)NCCCOCC)(C2)C3)CCC(C2CC2)C1 c1(CN(CCCNC(=O)CSC(F)F)C(C2CCCC2)=O)cccnc1 N1(C(Cc2cc(COC)on2)=O)CCC(C)(NC(=O)Cn2ncnc2N)C1 C1(CNC(C=CC(=O)OC(C)(C)C)=O)CN(C(=O)C(O)CC(N)=O)C2(CCC2)C1 c1(C(CNC(=O)C(=O)N(C)C)NC(CCn2c(C)ncc2)=O)cccc(C(F)F)c1 N1(C(c2n(CCC)ncc2)=O)CC(NC(=O)Cc2nonc2C)C(CO)C1 C1(NC(CCCOC)=O)CN(C(c2cnn(C(C)C(C)C)c2C)=O)CCC1F c1(OCC)ccc(Cl)c(C(N2CCCC(C)C2CNC(=O)C(Cl)=CCl)=O)n1 C(=O)(C(C)(C(F)F)NC(=O)OC(C)(C)C)NC(C)CC(C)NC(=O)C(C)CN(C)C c1(C(N2C(C)(C)C(CNC(=O)Cn3ccnn3)CC2)=O)ccc(N)c(F)c1F Cc1[nH]c2ncccc2c1C(=O)NCCCC1CN(C(=O)CS(N)(=O)=O)CCO1 c1(N2CCCCC(C)C2)nc2c(c(=NCCS(=O)c3ccccc3)[nH]1)SCC2 N1(C(COCC=C)=O)CCCC(O)(CNC(c2cc[nH]c2C2CC2)=O)C1 C#CCCCC(C)C(=O)NC1C=CC(CC(=O)N(CCC(C)(C)O)C)C1 C12(CNC(CN(C3CCC3)C)=O)CC(CO1)N(C(=O)CCc1n[nH]c(=N)s1)C2 c1(C(=O)OCC)nc(C(=O)NCCCNC(C2(C(C)C)CNC(=O)C2)=O)c(C)s1 CCC(CC)C(=O)NC(Cc1cn(C(C)(C)CC(N)=O)nn1)C(=O)NCCOC N1(CC)CCc2cc(NC(=O)C(=O)N=c3[nH]nc(Cc4ccccc4)s3)ccc21 N1(C(CC2CCC(=O)O2)=O)CCCC(NC(=O)CSCc2cccnc2)C1 c1(C(=O)NCCC(C)N(C(=O)CSc2n[nH]c(O)n2)C)cc2cccc(F)c2s1 C1(NC(c2c(OCC)non2)=O)CCOCC1NC(C1CCC1(OC)OC)=O c1(OCC)cncc(C(=O)N(C(CNC(c2ccnn2CC)=O)C2CC2)C)c1 C1(C(=O)NC2(COC)CCCCC2)COCCN(C(C2(C)CC2C)=O)C1 N1(C(C2C(C(C)=O)C2(C)C)=O)CCC(C)(C)C(C(=O)N(C2CCCC2(C)O)C)C1 N1(C(c2cc(C)n(C)n2)=O)CCC(C)(C)C1C(=O)N(C)C(c1cccs1)C N1(C(CSCC(N)=O)=O)CCCC2(CCN(C(C3CC4CC4C3)=O)CC2)C1 CC1(NC(=O)CCC2CC=CCC2)CCCN(C(C2CC2c2ccccc2)=O)C1 c1(C(=O)NC(CNC(c2cc(CC)[nH]n2)=O)(C)CO)cccc(OCCOC)c1 C1(NC(C(CN(C(c2c(C)oc(CO)c2)=O)C)C)=O)(CO)CCC(C)(C)C1 n1(CC(=O)OCC)cc(C(=O)NCC(O)CN(C(=O)C(C)n2cncn2)C)nn1 N1(C(CCOCC(C)C)=O)CCCC(n2cc(C3(S(N)(=O)=O)CC3)nn2)C1 N1(C(C2(CC)CC2(F)F)=O)CC2CCC1C(CCN=c1cc(C(N)=O)nc[nH]1)C2 C(=O)(C1=NOC2(CCNCC2)C1)N(CCN(CCC1CCC(C)O1)C)C C(CCCC(=O)NCC1(C)CCCS1)N(C(CC(C)F)=O)C Cc1c(CNc2nnccc2F)cccc1N1CCOC1=O C(CC(F)F)(C(=O)Nc1cc(N(C)C)cc(F)c1)N(C(c1n(C=C)nnc1)=O)C c1(NC(C2(C)CN(C(=O)C(C)Oc3ccccn3)C2)=O)nnc2ccc(Cl)nn12 C#CCC(O)C(=O)NC1CCN(C(c2coc(C(=O)OC)n2)=O)C1C CC1(C(N2CCC(CNC(c3cc(F)ccc3Cl)=O)C2)=O)CCC(F)(F)C1 CC1CCC(CNC(=O)C2=CCCOC2)CN1C(=O)Cc1cncnc1 C1(NC(C2C(CNC(c3ccc(C)nc3)=O)CCC2)=O)CC=C(C(C)C)CC1 C12(NC(C3N(CCC)CCC3)=O)COC(C1)C(NC(=O)CCC(=O)OC)C2 C(=O)(C(C(C)(C)C)NC(=O)CC(F)(F)CC)N1CCC(O)(CC)C1 N1(C(C(CCC)N(C)C)=O)CC2(CCN(c3cc(O)nc(=O)n3C)CC2)CC1C CC(C)(CC(=O)NC1CC(NC(=O)C(C)(F)F)C1)C(F)F Cc1ccc2scc(CN3CCN(C(=O)CC(C)C4CCCCC4)CC3)c2c1 C1(CNCC(c2cc(OC)ncc2)(C)C)Cc2cc(C)cc(Br)c2O1 c1(C(N2C(C3(NC(C4CCOCC4)=O)CC3)CCC2)=O)cc2ccccc2[nH]1 c1(CNC(C(=O)OCC)C(O)c2ccc(Cl)cc2)cc(C)c(Cl)c(C)c1 N1(C(C(C2CCOCC2)C)=O)CCN(C(c2cnc(S)nc2)=O)CC1CO O=S(=O)(c1cccnc1NC12CCCC1C2)NCCn1ncc2ccccc12 c1(C(=O)NC(C(=O)OC)(C)C(F)F)ccnc2[nH]c(C(F)F)nc12 S(=O)(=O)(c1cccc(=NCC2CCSC2(C)C)[nH]1)NCC(c1ncc(C)s1)C c1(C(N2CC3CC(NC(c4ccc(SC)s4)=O)C3C2)=O)c(C)ccc(F)c1O Cc1cccc(C(=O)NC2CCC(C(=O)N(C3CCCC3O)C)C2)c1O N1(C(c2c(C#C)c[nH]n2)=O)CCC(C(=O)N(CC(C)O)CC(C)O)C(O)C1 C(=O)(C1CCCc2nn[nH]c21)NCCc1nc(C(C)C)sc1 c1(CC)ccc(CCCC(=O)NCC(O)CNC(c2coc(OC)n2)=O)cc1 c1(C(=O)NCCC(=C)CNC(c2ccnc(O)c2)=O)cc(S(C)(=O)=O)ccc1O C(=O)(CC(C)(O)OC(C)C)N(CCOCCN(C(C(C)CF)=O)C)C C1(NC(C=CCC)=O)CCN(C(C2(C(=O)NC3CC3)CC2)=O)CC1F CC1OCCC1C(=O)NCC1CCCC1NC(=O)CCc1nccs1 C1(C(=O)NCC2C(NC(CCOCC(C)C)=O)C2)COCCN1C1CCCC1 C(C(C(=O)NC1CCN(C)CC1C)C(C)C)NC(C1(CCOC)CCC1)=O c1(CC(=O)NC2CC(CCNC(c3cc(OC)no3)=O)C2)cc(F)ccc1F C(C)(CC1CCC1)(C(=O)NCCCCNC(C1(O)CCOC1)=O)OC c1(C(=O)NCC2(OC)CN(C(C3(C)CCCN3C)=O)C2)ccc(F)c(C(F)F)n1 c1(C(N(CC(CO)(CO)NC(CNC(=O)OCC=C)=O)C)=O)ccc(F)c(F)c1 CC(C)C(O)CC(=O)NC1CCCN(C(c2coc(C(F)F)c2)=O)CC1 c1(C(=O)NC2CC(NC(C3(C)CCC(C)C3)=O)C2)n[nH]c2cccnc12 c1(N(C)C)cccc(CC(=O)N(C2CCCCC2NC(=O)Cc2cnc[nH]2)C)c1 CCC(C(=O)NCC(CO)NC(c1cc(F)cs1)=O)Nc1nc(C)cs1 n1(CC(=O)NC2CN(C(C3(C(N)=O)CCC3)=O)CCC2O)cnc2c1CCCC2 c1(C(N2CC(NC(C(C)SCCCC)=O)(CO)C2)=O)c(C)cccc1F C=Cc1ccc(C(N2CC(N(C)C(C3CC(OC(F)F)C3)=O)C2)=O)cc1 CN1CCC(C)(C(=O)NC2(C)CCCN(C(c3nscc3N)=O)C2)C1=O N1(C(C(C)CC2CC2)=O)CC(C(=O)NC(C)(C)CC2CC2)C(F)C1 CC(CC(=O)NCC(C)NC(c1cnn(-c2ccccc2F)c1)=O)C(F)F C1(NC(c2c(COC)cc[nH]2)=O)(CO)CCN(C(=O)Cn2nc(C)cc2C)C1 C(=O)(CCC(C)CN(C)C)NC1(CNC(Cc2ccc(OC)cn2)=O)CCOC1 C(=O)(CCCC(C)CC)NC(CC#C)CC(=O)NCCCN1CCOC1=O N1(C(CCC#C)=O)CCC2(CC2C(=O)NOCC2CCCC2)C1 N1(C(c2nc(C)[nH]n2)=O)CCOCC12COCCN(C(=O)C=CCO)C2 Cc1ccc(C(N2CCC(C)C2CNC(=O)Cc2cc(Cl)ccc2F)=O)cc1Cl C(=O)(C(C)N=c1cc[nH]cc1)NC1CCN(C(C(C)CO)=O)C1C C1(COC)(NC(=O)Cc2ccsc2)CCN(C(c2cn(C3CC3)cn2)=O)C1 C#Cc1cccc(C(=O)NCC(C2(O)CN(C(=O)C=CC3CC3)C2)(C)C)c1C c1(C(=O)Nc2cc(C(=O)NCCNC(C3C(C)=C3C)=O)on2)[nH]c(=N)ccc1C CC1(CNC(c2ccccc2C(N)=O)=O)CCCN1C(=O)COC1CC(F)(F)C1 c1(OC)nc(Cl)ncc1OC(=O)NC(=O)N(C)C CC1(C)CCN(C(C2CCC3(CC3)C2)=O)C1C(=O)NCC1=CCCCCC1 CC(C)(C(=O)NCC(O)CNC(=O)CCF)C1CC1 c1(CNC(CC2(C)CCN2C(=O)COc2ccsc2)=O)n[nH]c2c1CCC2 C1(C(N(CC(C)C(=O)NCC(c2ccncc2)O)C)=O)CCCCNC1=O N1(C(C(c2n(C)cnn2)(C)C)=O)CCN(C(C2(CF)CC2(F)F)=O)CC12CCC2 Cc1nc(C(=O)NCC2(F)CC(NC(C3COC(=O)N3C)=O)C2)c(C(F)(F)F)[nH]1 CC(C(C)(C)NC(c1cnn(-c2ccccn2)c1)=O)NC(=O)C(=O)N(C)C C1(C2CCCCC2)(NC(=O)CC2CC(C(=O)N3CC4CC4C3)=NO2)CC1 N1(C(C2(C)C(C)C2)=O)CC2COCC(C1)N2C(c1cc2cnccc2[nH]1)=O N1(C(C(C)Cc2cccc(F)c2)=O)CCN(C(=O)Cn2c(C)csc2=O)CC1C C1(C(=O)NCCCNC(=O)OC)CCC2CCC1N2C(c1c[nH]c(C)c1)=O C#Cc1ccc(C(N2CCC(NC(c3cc(F)ccc3F)=O)C(O)C2)=O)cc1C c1(CN2CCC(C(=O)Nc3c(OC)ncc(Cl)c3)C(O)C2)ccccc1[N+](=O)[O-] C1(C(N(CC#C)C)=O)CCC2CCC1N2C(c1ncn(C)c1C)=O O=C1NC2C3(CCC13)OCC1OC1=CC=CC(Cl)=C(Cl)C2CCOCC N1(Cc2c(OCC)cco2)CCC2(CC1)CC2C(=O)Nc1c[nH]nc1Cl C12COCC1C(=O)N2.N1(C(CCNC(=O)OC)=O)CCCC1C(C)(C)O Cc1cc(-c2cn(C3CCN(C(c4c(C)ccn4C)=O)CC3)nn2)ccc1F c1(C(N(C)CCN(C)C(C2CCc3nccn3C2)=O)=O)cc(F)cc2nc[nH]c12 C1(CC)CN(C(c2nnn(CC)c2C)=O)CCC1NC(=O)C(C)NS(C)(=O)=O Cc1cccnc1-n1ccnc1-c1c[nH]c(-c2ncsc2C)c1.c1nccnc1N C(=O)(C(C)(C)CC(C)(C)C)NCC12OCC(NC(C3N(CC)CC3)=O)C(C1)C2 C1(C(=O)NCC(C(C(=O)OC)F)C)CCN(C(C)=O)C(C)(C)C1 C=CCC(C(=O)NCC1CCC(C(=O)NC(c2cn[nH]c2)C)C1)C(C)C n1(CC)cnc2[nH]c(=NCc3cnc(O)[nH]3)[nH]c(=NC3CCOC3C(C)C)c12 c1(CN2C(C)(C(C)NC(C3CC(F)C3)=O)CC2)cccc(C(F)(F)F)c1F CC(C(=O)OC(C)(C)C)C(=O)N1CC2C(CNC(=O)CCC(=O)N(C)C)C2C1 C=CC1OCCC1C(=O)NCCn1cc(C(=O)Nc2ccc(C(C)C)cc2)cn1 N1(C(=O)NCCc2ccc(Cl)cc2C(F)(F)F)CCCC1C1CCCO1 c1(C(C)=O)cc(NCCCNC(C2CCC(=O)N2)=O)ncn1 c1(CC(=O)NC(CCCNC(CC=C)=O)C)coc2cc(Cl)ccc12 c1(NC(COC)COC)ccnn1C1CN(C(c2c[nH]nc2OC)=O)C1 c1(C(=O)OCCc2ccccn2)ccc(NC(c2ccon2)=O)cc1 c1(OC)cc(O)c(CNc2ccc(C(=O)Nc3ccc(Cl)c(F)c3)cn2)cc1Cl c1(C(N(CCCNC(CC=CC)=O)CC2CCCC2)=O)cnc(O)c2cncn12 Cc1cccc(CC(=O)NC2CC2NC(=O)COc2cnc(Cl)cn2)c1 C(=O)(C(CC)CCCC)NC1C(OC)CN(C(c2c(OCC)ccc(C)c2)=O)C1 N1(C(C23CCC(OC)C2C3)=O)CC(NC(c2cnc(C)cc2C)=O)CC(C)C1 N1(C(Cc2n(C)c(S)nn2)=O)CC2CCC(C1)C(NC(=O)C(F)C(F)(F)F)C2 c1(C(=O)NC(CNC(C(C=C=C)C)=O)CCC)cc(N)c(C)cc1C CC1CN(C(C2CCC3(C2)CC3(F)F)=O)CC2(CCN(C(C3CC3F)=O)C2)O1 N1(C(c2cc(OC)n[nH]2)=O)C(C)C2CC1C2NC(=O)CC1CCCCO1 C=C(C)C(CC(=O)NC12CCC1CN(C(=O)CCCC)C2)OCCN(C)C C1(=CC(N2CC3C(CNC(=O)CN4C(=O)CCC4=O)(C3)C2)=O)CN2CCC1CC2 C(=O)(C(O)CCCNC(=O)C(C)CC(C)C)N1CC(OCC)C1 c1(CC)cc(C(=O)OCC2CC2c2ccc(Br)cn2)c(Br)s1 N1(C(C(C)(C)F)=O)CC2CCC1C(NC(C1(n3ccnc3)CCCC1)=O)C2 C1(OCC)CN(C(C2C=CCCC2)=O)CCC1NC(C1CC=CCC1)=O Cc1ncn2ccc(C(N3CCC(CNC(=O)C(C)O)C34CC4)=O)cc12 N1(C(CC(=O)OCC)=O)CCCCC1CN(C(=O)C(C)(C)COC)C c1(C(N2CC=CC(NC(CCCC#C)=O)C2)=O)ccn2c(C)cnc2c1 C1(C(=O)OCC)OCCNCC1N(c1nccs1)C(=O)CN1CCCCC1=O C1(OC(C)C)CCCN(C(=O)CCCCN(C)C(c2c[nH]nc2C(C)C)=O)C1 N1(C(c2ccc(C#C)o2)=O)CCN(C)C(CNC(=O)C=CC=C(Cl)Cl)C1 C1(C(N(CC(CN(C)C(c2n[nH]cc2[N+](=O)[O-])=O)O)C)=O)CCCCC(F)(F)C1 C1(C(=O)NCC2(F)COC2)COCCN(C(c2ccnnc2O)=O)C1 N1(C(C(C(C)C)O)=O)CCC(C2CC2)C1CNC(c1cccc2nsnc12)=O CCCC(CNC(c1cccc(O)c1F)=O)C(=O)N1CC(C)CC1CC C(C(C(=O)NCc1cnc(F)c(C)c1)C(C)(C)C)NC(C(CCCC)C)=O C(CCCCC(=O)NCC(C)C1CCC1)NC(Cc1c(C)noc1C)=O C1(C(=O)NC2(C)CN(C(c3cccc(CS(C)=O)c3)=O)C2)C2CC3C(C2=O)C13 C(c1ccccc1C)=CC(=O)NC1CCC(N(C(C2CC(CC)(CC)C2)=O)C)C1 C12(C(=O)NCC(CC(C)C)NC(=O)C#CC3CCOC3)CCCN(CCC1)C2 C(=O)(C1=NOC(C)C1C)NC(C1C(C(N2C(C(=O)NC)C=CC2)=O)C1)C C(=O)(C(=O)C(C)(C)C)N1CC2C(C(N(C)CC3CC3(F)F)=O)(C2)C1 C#Cc1ccccc1NC(=O)CC1(CNC(=O)C(CC2CC2)OCC)CC1 N1(C(CC2(OC)CCOCC2)=O)CCC(O)(C(C)NC(C2CCCC2O)=O)CC1 N1(C(CC2(OC)CC2)=O)CCC(C(F)(F)F)C(NC(=O)CCCn2cccn2)C1 c1(C(=O)NC2CN(C(c3ccnnc3)=O)CC3(CC3)C2)cnc2ncccc2c1 O=C(C(C1=NOCC1)N1CCCC1C1CC1(F)F)NCc1ccc(Cl)cc1 C(=O)(N1CCC(C(N2CC(CO)C2)=O)O1)c1nc(C(C)(C)C)oc1 C(=O)(C(CNC(c1nc(C)oc1C)=O)CC(C)C)NC(c1nc[nH]n1)CC c1(C(N2CC3C(N(C(=O)C4=CCCC4)C)C3C2)=O)ccc2ncncc2c1 CC(C)C(C)(CNC(C1(CS(C)(=O)=O)COC1)=O)NC(C1CCOC1)=O c1(C(C)NC(C2OCCC2CNC(=O)C(CO)N(C)C)=O)cccnc1O c1(C(N2C(CC(=O)N(C)CC3COCCO3)CC2)=O)ccnnc1O CCCCCCCCC(=O)NC1CCC(C)N(C(c2cc3c(ncn3C)[nH]2)=O)C1 CCC(C)C(O)C(C)C(=O)NC(CC(F)F)C(N1CCC2(CCCC2)C1)=O C1(C(N2CCC(CN(C(=O)C(C)(C)n3ccnn3)C)C2)=O)CCCC(C)(C)CC1 C=CCCCCNC(=O)C(C)(C1CCC1)NC(=O)C(C)NC(N)=O N1(C(=O)C=CCF)CCC2(CCCN2C(C2SCCCS2)=O)C1 c1(C(=O)NC(C(=O)NC(c2nnc(O)n2C)C)C2CCOC2)ccnnc1O c1(C2(NC3C(c4n(CC)ccn4)OCC3)CCC2)ccccc1Br C12(CNC(C3(CC)CC3(F)F)=O)CC1CN(C(C1(CO)CCCCC1)=O)C2 C1(NC(C(C)N(C)C)=O)CCC(F)(CNC(c2cncc(N3CCCC3)n2)=O)C1 c1(NC(c2ncn(C)c2)=O)sc2c(c1C(=O)Nc1ccc(Cl)cn1)CCC2 C1(NC(C(C)(O)Cc2ccccc2)=O)CN(c2ncc(OC(F)F)cn2)CCC1(F)F c1(C(N(CC(CNC(c2nccc(C)n2)=O)C)C)=O)cc(N)c(C)cc1C N(C1CCCn2ccnc21)C(CCC(CC)NC(=O)Cc1cnns1)=O n1(CCOC)cc(C(=O)NCCC2CCCN2C(C2CC(CF)C2)=O)nn1 N1(C(C2(N(C)C)CC2)=O)CCC(F)(F)C(CNC(c2nc(Cl)sc2Cl)=O)C1 N1(C(c2c(C)c[nH]n2)=O)CC(C)CCC1CNC(c1ccc(F)c(CO)c1)=O N1(C(C2C(C=C)C2)=O)CC2CCC1CN2C(C1(C#N)CCOC1)=O n1(CC(=O)NC2(CCNC(CC3(C)CC3F)=O)CCC2)cc(C#N)cn1 C(=O)(C(C)(C)C(C)(F)F)NCC(CC(C)C)NC(=O)C=Cc1ccc([N+](=O)[O-])s1 Nc1cc(C(=O)NCCC2CCN(C(C3(C(F)F)CCCO3)=O)C2)cc(O)c1Cl CC1(C)CC(NC(C2(F)CCC2)=O)CCN(c2ncnc(Cl)c2F)C1 C(c1c(C)noc1C)=CC(N1CCC(N(C(=O)C(C)C2CCC2)CC)C1)=O Cc1cc(C(C(=O)NCc2ccco2)N(C)C(C2(O)CCOCC2)C)cc(F)c1 c1(C(=O)NCCC2C(C)CN(C(c3ccon3)=O)C2)cc2scnc2[nH]1 C#CCC(C(=O)NC(C)CN(C)C(c1ccnc(N(C)C)c1)=O)C1CC1 C1(NC(c2nc(CC)oc2C)=O)CC2CC1CN(C(c1cc([N+](=O)[O-])c[nH]1)=O)C2 CN=S1(=O)CCN(C(=O)C(c2ccc3c(c2)OCO3)=O)CC1 N1(C(C(N2CCN(C)CC2)C)=O)CC2CCN(C(c3cccc(=O)o3)=O)CC2C1 CCCCC(C)CCC(=O)N(C(C)CNC(=O)CC=C(C)C)Cc1ccccc1 N1(CC2CC(C)OCC2)C(=O)CN(CCc2ccccc2C2CC2)C1=O C1(NC(C2CC3(CC(C=C)C3)C2)=O)CC2CN(C(C3(C)CCOCC3)=O)CC2C1 c1(C(=O)NCc2nc(CC(=O)OCC)on2)cnn(CC)c1C1CCCC1 c1(OC)ccc(SCCCC(=O)NC(C)(C)C#N)cc1 C1(C(=O)OCC)(CC)CCCN1C(C12CC(CCO1)C2)=O CCCC(CNC(=O)Cc1ccsc1C)C(=O)NCCCOCC(C)C C(=O)(C(CC(F)F)C1CCC1)NC1C(CNC(c2cc(C)ns2)=O)CCC1 c1(C(=O)NCC(CC)NC(=O)C(C)NC(C)(C)CC)cccc2c1C(=O)CC2 N1(C(C(CC)C)=O)CCCOC(CNC(c2cnc(CO)nc2C)=O)C1 C1(C(=O)NCC(c2ccc(-c3ccccc3)cc2)O)C2CC(C(O)C2O)S1(=O)=O N1(C(C(CN(C)C)O)=O)CC(NC(=O)COCP(C)(C)=O)CC1CO C1(C(=O)NC2(CNc3cccs3)CCC2)OCCCC1c1ccccc1 c1(OC)cc(CN)cc(N)c1O.N1(CCC(=O)N2CC(C)C2)CCN(C(C)C)CC1 C1(NC(C(CC#C)O)=O)CN(C(c2cn(CC3(C)COC3)nn2)=O)CC(C)(C)C1 C1(NC(=O)CCNC(C2CNC(=O)C2)=O)CC2C=CCC(C1)C2 C1(OC(C)=O)CCCN(C(C23CC2CN(c2ncncc2Br)C3)=O)C1 Cc1ccncc1CC(N1CC(OCCNC(=O)CC2CC=CCC2)C1)=O C(CN=c1ccn2ncc(I)c2[nH]1)c1ccc(C)c(O)c1 c1(C(=O)NCCCC(C)(C)NC(CCOCCN(C)C)=O)ccc(O)c(=O)cc1 c1(NC(c2csc(CNC(c3cccnc3F)=O)n2)=O)ncccc1[N+](=O)[O-] Cc1cc(O)c(Cl)cc1C(=O)NC1CCC(NC(=O)CSCCC(C)C)C1 Cc1ccnc(NC(C)(CCCO)c2nnnn2CC2CCCO2)n1 C1(CCCNC(c2cn(CCO)nn2)=O)CCCCN1C(=O)C=CC1CC1 c1(C(N2CCC(CNC(CN(C(COC)=O)C)=O)C2)=O)c(C)oc2ccccc12 Cc1[nH]nc2c1CCC(C(=O)N(C1CN(C(C3CCN(C4CC4)C3=O)=O)C1)C)C2 C1(N(CCNC(N(CC)Cc2ccc(Br)cc2)=S)C)CC(C)N(CC)C(C)C1 C1(CC)CN(C(C2CC2C)=O)CCN1C(c1cc(C2CCCC2)nn1C)=O C1(NC(C(c2cn(C)nc2)=O)=O)CCCC(NC(=O)COC2CC=CC2)CC1 C1(O)(CNC(C2C(C(=O)OC)C2)=O)CCCN(C(=O)CC2(OC)CCC2)C1 CC1CC(NC(=O)CC(C)n2cccn2)CN(C(C2(CF)CC2)=O)C1 CC1CN(C(c2ccns2)=O)CC(CCNC(c2cc(C3CC3)ncn2)=O)O1 C1(CC(=O)N(C)Cc2ccns2)CCN(C(=O)CCC2CC2)C1 N1(C2CN(C(N3C(=O)CCC3=O)=O)CC2=O)CCN(C(=O)CCC2CC2)C(=O)C1 Cc1cc(CCC(=O)NCC(C)CNC(C2CCC2(C)C)=O)on1 C1(NC(C(c2ccc(Cl)cc2F)C)=O)CC2CCC1N2C(C1CCOC1)=O C1(CN(C(C(C)Cn2ccnc2)=O)C)CN(C(c2c[nH]nc2C(F)F)=O)CCO1 c1(C(N2CC(CC(=O)NC(CC)CO)C2)=O)cc(C(F)(F)F)cc(F)c1 c1(C(=O)NCC2(F)CC(NC(C3(C#C)CCC3)=O)C2)c(C)c(C)c(C)c(C)c1C C(=O)(C(CC(C)(C)C)NC(=O)C=Cc1cncs1)NCC1(CCOC)CC1 c1(C(=O)NC2CCCS2)nnc(C)cc1NC(C1CCC(CNC(C)=O)CC1)=O C(CC(O)CNC(=O)C(C1CCCCC1)O)NC(=O)COCCF c1(C(=O)NCCC2CCCN(CC(N)=O)C2)ncccc1Cl C1(CCNC(C2C(C=C)C2)=O)CN(C(=O)COCc2ccnn2C)CCS1(=O)=O N1(C(c2cnn(C)c2Cl)=O)CC(NC(c2nncs2)=O)CC1(C)C N1(C(C(COC(C)=O)C)=O)CCOC(CCC(=O)NC2(CCO)CCCC2)C1 c1(C(C(=O)NCCCCCC)N(C2CCCOC2)CC)cccc(Cl)c1Cl N1(C(CC2N(C(c3c(C)ocn3)=O)CCC2)=O)CCCC(OC2CCC2)C1 c1(C(=O)NC(CC2CCN(C(C3(C#C)CC3)=O)CC2)C)cccc(F)c1C(F)F n1(CC(=O)OC)cnc2c(cnn2C)c1=O.C1(=O)C(N)(c2ccccc2)CN1 N1(C(COCCC)=O)CCN(C(=O)Cc2cccc(Br)c2C)CC1CO N1(C(CC2C(C)CCN(C(Cc3ccn(CC)n3)=O)C2)=O)CC2(COC(=O)C2)C1 C(C(C)(O)CC(=O)NC1CCCC(C(=O)NC2CCC3(CC2)N=N3)C1)OC C(=O)(C#CC1CCC1)N1CC(CCNC(C2(C)CC(C(F)(F)F)C2)=O)C1 Cc1ccoc1C(N1CCCC1CNC(=O)CCNC(=O)CC1CCCCC1)=O N1(C(CC(C)(C)C#N)=O)CCC2(CC2)CC1C(=O)NCc1cccc(O)c1F c1(-c2cn(C3CCN(C(C(CC)COC)=O)CC3)nn2)cc(F)c(Cl)cc1Cl C1(C(=O)NCC(C)(C2CCC2)NC(c2nn(CC)c(C)c2)=O)COC(C)(C)CO1 CC1COCCN(C(=O)C(C)(C)C)C1.S1(=O)(=O)CCN1C C(=O)(CCC(=O)c1ccc(Br)cc1)NC(CNC(=O)C(F)=CCCF)CO C(C(=O)NCC(N1CCCC1)=O)(C1=CCSC1(C)C)N(C)CC1CC(F)(F)C1 n1(CC)ncc(I)c1C(=O)NC.c12cccc(c1)NC(=O)NCC2 C1(C(=O)NCC2CCN(C(c3c(C)nc[nH]3)=O)C2(C)C)CCCCCC1(F)F C(=O)(C(C)C(O)C(C)C)NC1CCC(NC(c2cc(CC)oc2C)=O)CC1 C(=O)(CCN=c1ccc(C)c[nH]1)N1C(CCNC(CCCCC)=O)CC(OC)C1 c1(C(=O)NCC(C)CN(C(=O)C(O)C2CCC2)C)cccc(C(C)(C)C)n1 c1(CSC)ccccc1CC(=O)NCC(C1CCCC1)NC(=O)C(C)N1CCCC1 C1(CNC(C2(SC)CCC2)=O)CC2(CC2)CN1C(C1CCCC(CF)C1)=O c1(CN2CC3C(C(=O)Nc4c(CO)ccc(OC)c4)(C3)C2)c(Br)cc(Br)cc1Br C1(C(=O)NCC2(CO)CCCC2)CC2CC2N1C(=O)Cc1cnns1 c1(C(=O)NC)cncc(N2CCCC2)n1.CCC(C)(C)NC(=O)C(O)C1CC1C CCC(COC)C(=O)NCCCN(C)C(c1cnn(CCC#N)c1C)=O c1(C(N2C(C)(C(=O)NCCCS(C)(=O)=O)CCC2)=O)cnn2cccc(F)c12 CN1CC2CN(C(c3ccnc(F)c3)C(=O)NC3CCOCC3)CCN2C1=O N1(C(CCNC(=O)CO)=O)CCOCC(C(=O)Nc2cnn(C3CC3(F)F)c2)C1 C1(C)(CC)CCCN1C(=O)CCc1ccccc1C c1(-c2c(C)ccc(CO)c2)cc(C(N2CC(NS(C)(=O)=O)C2)=O)c2cc[nH]c2c1 c1(C(=O)NCCCNC(c2ccc(C)nc2C2CC2)=O)ccc2c(c1)NC(=O)C2 N=c1ccc(C(N2CC3C(NC(c4cnn(CC5CCCC5)c4)=O)C3C2)=O)n[nH]1 C1(CNC(C2N(C(CCC(=O)NC)=O)CC2)=O)CC(C)OC(C)C1 C1(C(C)C)CN(C(=O)CC2CC2)CCC1NC(C1(N(C)C)CCCSC1)=O C1(NC(c2c(OC)c[nH]c2C)=O)CC2CCC(C1)N2C(=O)CSc1ccccn1 C1(C)(C(=O)NC2C(C)N(C(=O)CCc3cnoc3)CC2)CCCC1(F)F CCN=c1[nH]c(C(N2CCOC(CCNC(=O)COC3CC(F)(F)C3)C2)=O)cs1 N1(C(C(C2CCOC2)OC)=O)CC23CCCC2(C1)CN(C(=O)CCP(C)(C)=O)C3 c1(CN2CC(NC(C(CCC)N3CCNCC3)=O)C(C)C2)ccnc(F)c1Cl c1(CNC(C(C#C)(C)C)=O)cc(C#N)ccc1Cl C(CC(=O)NC(C)CNC(c1cccc([N+](=O)[O-])c1C)=O)(C1=CCCC1)OCC C1(C(=O)NC2C(CNC(=O)C=Cc3cncc(F)c3)CC2)CCn2nncc2C1 CC(CCCC(=O)Nc1ccc(O)cc1)NC(=O)C(C)(Cl)Cl c1(C(N2CCC(OCC(=O)N(C3(CC)CCC3)C)C2)=O)cccc(F)c1C c1(CC(C)C(N2C(C(=O)NCc3cccc(Cl)n3)CC3CC23)=O)ccc(O)cc1 c1(C(N2CCC(SC)CC2C(F)(F)F)=O)c(F)ccc(Cl)c1Br N1(C(C23N(C(CC(=O)NCC)=O)CCC2CCC3)=O)CCC2C(=O)NCC2C1 C1(CC(=O)N(C(C)C)CCF)CCN(C(=O)CC2CC3(CC3)CO2)CC1 c1(C(N(CC(CC)NC(c2csc(C)n2)=O)C)=O)nc(C(C)C)oc1C C1(NC(c2c(CCC)n(CC)nn2)=O)C(CNC(=O)C=CCF)CCC12CCC2 c1(C=O)nc(=N)cc[nH]1.n1(CCCN(C)NC2CC2)cc(Cn2ccnc2)nn1 C1(c2noc(C3CC3C(C)NC(C(C)(C)C)=O)n2)CC2(CC2)C1 c1(NCCCC(=O)NCC(C)N(C(=O)Cc2cc[nH]c2)C)ccc([N+](=O)[O-])cc1 Cc1nccc(F)c1C(=O)OC(C)C(=O)Nc1ccccc1F N1(C(CCC(=C)Cl)=O)CCN(C(c2cn3c(n2)SCC3)=O)CC1C Cc1oc(C#N)cc1C(=O)NC1CC(CNC(=O)CC2CC(F)(F)C2)C(O)C1 CC1SCCCC1C(=O)NCC1CC(C(=O)NOCC2(C)CCC2)C1 c1(C(N2CC3C(CNC(=O)Cc4ccsc4)C3C2)=O)c(Cl)ccc(Cl)c1O C1(CC(=O)NCC)CCOC1=O.CC(O)CN(C(=O)C=CC1CC1)C(C)C N1(C(CSc2cccc(C)c2)=O)CCN(C(=O)Cc2sc(C)nc2C)C2CC12 c1(C(N(C2CCCC(=O)O2)c2nc(C3CC3)cs2)=O)ccc2ccccc2c1 N1(C(CN2CCC(C)CC2)=O)CC(C)(C)OC2(C1)CN(C(C1OCC1(C)C)=O)C2 c1(C(=O)NC(CNC(C2CC2c2ccsc2)=O)C2CCC2)csc(Cl)c1 C1(C(=O)NCc2cc(C)[nH]n2)CC(C)CN(C(c2occ3c2CCC3)=O)C1 CN1CC2CN(C(=O)CC3(NC(=O)CC4CCCCC4)CC3)CC2C1 N1(C(Cn2nc(C)c(Br)c2C)=O)CCn2c(C(N)=O)nnc2C1 N1(C(C2(OC)CCSC2)=O)C2CCCC1CC(NC(=O)CSc1n[nH]c(O)n1)C2 S(=O)(=O)(c1ccc(NCC23CCCC2C3(F)F)c(F)c1)N(CCC)CC N1(C(C(CC2CCC2)OC)=O)CC2CC1(C(=O)NCC(C)C(F)F)C2 N(C1COc2ccc(F)cc21)C1CCC(C)CC1n1cncn1 N1(C(C(CC2CC2)NC(C2CC(O)(CC#C)C2)=O)=O)CC(CN(C)C)C2(CC2)C1 C(=O)(NN1CCCCC1=O)c1c(OC(C)C(=O)NC2CCCS2(=O)=O)cccc1 C1(C)(CNC(C(COC)C)=O)CCCN1C(c1cnn(C2CCCC2)c1)=O c1(NCC(CCC)O)ncccc1S(=O)(=O)N(C)C.c12cccnc1NC2 N1(C(c2c[nH]c(=N)o2)=O)CCC2C(C1)CN2C(C1CCS1(=O)=O)=O c1(COC(COCCOCC#C)=O)cc(C)c(Br)c(Cl)n1 C=C(C)CCCC(=O)N1CC(NC(C2CCCN2N=O)=O)CCC1C N1(CC2C=CCN(Cc3ccccc3)C2)CC2CC(O)C2C1 c1(C(=O)Nc2c(CNC(C3(COC)CC3)=O)cccn2)cnn2c1OCC2 c1(-n2cc(CNC)nn2)ccc2[nH]c(C(=O)NCC(Cl)=CCl)c(C)c2c1 CC(CN(C)C)CCC(=O)NCC1CC2CCC1N2C(c1ccc(Cl)nc1O)=O c1(C(=O)N=c2cc[nH]cc2O)cnc2cccc(Br)c2c1 C1(OC)CC2CC1CN(C(=O)C(CNC(=O)CCCCN(C)C)CC(C)C)C2 c1(C(=O)NC2CN(C(c3c(C)cn(C)c3)=O)C(C)CC2)cn(C)c2ncccc12 C(CC(=O)NCCn1cc(C)cn1)(C1CC1)NC(CC1(OCC)CCC1)=O C1(C(=O)NC2C(C)CN(C(C3CCOCC3)=O)C2)CCn2ccnc2C1 Cc1ccc2cc(C(=O)NC(C3(O)CN(C(c4cc(=O)cc[nH]4)=O)C3)C)[nH]c2c1 C(=O)(CC(=O)NC1CC1)N(CC(CC)NC(=O)CC(C)C1CCCCC1)CC C(=O)(C(F)C1=CCCCC1)NCC1CCN(C(CN2C(=O)CN(C)C2=O)=O)C1 C1(C(N2C(C=C)CC2)=O)CC(O)CN1C(c1c[nH]c(C#N)c1)=O c1(C(=O)NCC2C(NC(COCCC=C)=O)COC2)cc(N)ccc1F C1(C(=O)NC2C(SC)CN(C(c3coc(SC)c3)=O)C2)COc2ccccc2C1 c1(C(=O)NCC2(O)CCN(C(c3cnc(Cl)[nH]3)=O)C2)nc[nH]c2nccc1-2 C(=O)(C1CCc2ccccc21)N(C(C(=O)NC(CSC)(C)C)C)C C(c1nc2ccccc2o1)=CC(=O)NCC(CO)NC(=O)COCC1CC1 N1(C(Cc2c(C)ocn2)=O)CCCN(C(=O)C(CO)C(C)(C)C)C(CO)C1 N1(C(C(CC)NC(N)=O)=O)CC(C)(C)CC1CC(=O)NC1CC(CN(C)C)C1 C1(C(C)(C)NC(CSCC#C)=O)CCN(C(C2CCCCO2)=O)CC1 C1(C(N2CC(N(CC=C)C)C2)=O)CN(C(=O)CC(C)COC)CC1F C1(CNC(C2C(CC)C2)=O)CCCN(C(C2CC2c2cccnc2)=O)C1 N=c1[nH]c2c(s1)CCCC2C(=O)NCc1ncc(Cl)cn1 c1(COCC(=O)NC(CN(C(Cc2nc(CC)sc2)=O)C)C)ccc(OC)nc1 c1(C(=O)NC(CCN(C(C=CC=CC)=O)C)C)cnoc1-c1ccco1 N1(C(COCCOCCOC)=O)CCN(C(C2CC23CC(O)C3)=O)CC1CO c1(C(=O)NCC(=C)CCNC(C2CC2C(C)(C)C)=O)ccc(-c2cc[nH]n2)cc1 N1(C(C2(NC(C(COC)C)=O)CCN(C)C2)=O)CC(C)C(F)(F)C1 C1(NC(=O)Nc2c(F)cc(C)c(F)c2)CCOC2(CCSCC2)C1 N1(C(CC(=O)NCC)=O)CCC2(CC1)COCC(CNC(C1CCOC1)=O)O2 c1(CC)ccc([N+](=O)[O-])cc1NC(N1CC2NCCOC2C1)=O c1(C(C)C(=O)NCC2(NC(c3ccc(F)cc3)=O)CCOC2)nc(F)ccc1Cl O(CP(C)(C)=O)CC(=O)NC(C1CCCCC1)CNC(C1C(CCC)C1)=O c1(C(N(CCNC(c2scc(C(C)=O)c2)=O)C)=O)n[nH]c2c1CCCC2 c1(CC(C(N)=O)NC(C2C(NC(c3c(C)scc3)=O)CCC2)=O)ccc(O)cc1 C(=O)(C1=C(Cl)CCC1)NC(C(C)NC(=O)CN1CCC(C(N)=O)CC1)CO N1(C(CCc2onc(C(C)C)n2)=O)CCC(NC(c2scnc2Cl)=O)C(F)C1 c1(SCC(=O)NCCN(CC(=O)NCC2(C(C)C)CC2)CC)nc(C)cc(C)n1 C(=O)(CS(=O)(=O)C(C)C)N1C2C(NC(CCCC=C)=O)C(CC2)C1 C1(C(=O)NCC(=CC(N2C(CCC)COCC2)=O)C)CC(C)(C)CN1C c1(C(=O)NCC(CNC(CC(C=C)CC)=O)O)cc(Cl)c(C)cc1Br C1(N(C(c2cn(CCCC)nn2)=O)C)CCCN(C(C2(SC)CC2)=O)CC1 c1(OC)cc(C(N2CC3CC3(C(=O)Nc3cn(C)nn3)C2)=O)c([N+](=O)[O-])cc1O C12(C(=O)NC3CN(C(c4c(C)sc(C(F)(F)F)n4)=O)CC3C)CC1COC2(C)C c1(C(=O)NC(C(NOCC#C)=O)C2CCOCC2)nn(C)cc1C#C C(=O)(C(C)(C)C(C)NC(=O)CC1CCCC(=O)N1)NCC(N(OCC)C)=O N1(C(C2OCCN(CC)C2)=O)CCN(C(c2snnc2C)=O)CC(CO)C1 N1(C(=O)NC)CCOC(C(=O)N(C)CCN(C)C(c2cn(C)nc2C)=O)C1 N1(C(CC2(C=C)CCC2)=O)CCC(C)(NC(=O)C(c2ccccn2)C)C1 c1(C2(C(N3CC(N(C(C=C4CCC(C)C4)=O)C)C3)=O)CC2)ccc(F)cc1Br C(=O)(C1=CC2CCC(C1)N2C(CC(=O)OC(C)(C)C)=O)N1C(C)C(C)S(=O)CC1 c1(C(=O)NC(C)CCNC(c2ccn3nccc3n2)=O)cc(O)c2ccoc2c1 N1(C(C2N(C)C(=O)OC2)=O)CCS(=O)(=O)C(CCNC(c2ccc(O)nc2)=O)C1 CC(C)C(F)(CNC(C1C=CCS1)=O)C(=O)NCC1(c2ccon2)CC1 C1(C(N2CCC(C(C)(C)NC(C(=O)NCC)=O)CC2)=O)CS(=O)(=O)CC(=O)N1 C(CC(C)C(=O)NCC1CC1NC(c1cnc(C2CC2)o1)=O)=CCC Cc1ccc(C(CNC(C2(C)CC2(Cl)Cl)=O)NC(c2cccnc2)=O)cc1 C1(NC(c2c(C)non2)=O)CCCCCC1C(N1CCS(=O)CC1C)=O c1(CCC)cc(C(N2CCC(CN(C(=O)C3=CCCC3)C)C2)=O)sc1C c1(C(=O)NCC2C(NC(C=C(CCC)C)=O)CC2)cc2c(C)ccc(Cl)c2[nH]1 c1(C(=O)NC2CC(n3cc(C4(O)CCOCC4)nn3)C2)cc(Cl)cc2[nH]ncc12 N1(C(c2cccc(CC)c2F)C(=O)NCC2CCOC2)CCCC(C)(C)CC1 c1(CC(=O)C(=O)NC2(CC(=O)Nc3csc(Br)c3)CCC2)ccc(O)cc1 C(=O)(CC(C)(C)C#N)NC1CC(N(C)C(c2n[nH]cc2Cl)=O)C1 C(=O)(C1=CC2(CN(C(c3csc(Cl)c3)=O)C2)OC1)N1CC(C)(C(F)(F)F)C1 C=CCC(CNC(=O)CCCC(OC)OCC)C(=O)N1CC(CC23CC(C2)C3)C1 O=C(CCN=c1[nH]c(=NCCCF)[nH]c2c1CCCCC2)Oc1ccccc1 N1(C(CC=CCC)=O)CCC(NC(c2coc(S(C)(=O)=O)c2)=O)C12CCC2 Cc1nc(F)ccc1CNC(=O)CC1CCCC1NC(C1CC(O)C1)=O C1(CNC(C(c2ccc(Cl)cc2)OC)=O)CCC(C)(C)CN1C(c1ccoc1)=O c1(-c2ccc(C)cc2)nc(C)cc(=NC2CN(C(=O)C(F)C(C)(C)O)C2)[nH]1 N1(C(c2c(SCC)nccn2)=O)CCC2C1CCCN2C(=O)CCC(C)(F)F N1(C(c2c(C)nn(C)c2C2CC2)=O)CC(NC(c2cccn2C)=O)C(C2CC2)C1 CC(C)(F)CCC(=O)NC12CC(C(N3CC(CF)OC(CF)C3)=O)(C1)C2 N(C1CCOc2ccc(Br)cc21)S(=O)(=O)c1cccc(N2CCC3(CCC3)C2)n1 n1(C(C)(C)C)nccc1C(N1CCC(OCCNC(=O)Cc2csnn2)C1)=O C1(CNC(CCc2cccc(OC)c2)=O)C(C)CCCN1C(c1coc(Br)c1)=O C1(NC(CC(C)F)=O)CN(C(c2ccc(-c3ccco3)o2)=O)C2(CCCC2)C1 C1(NC(c2cccc(N)c2O)=O)CCCCCN(C(=O)CCCC2CC2)C1 N1(C(C2CCN(C)CC2)=O)CC(C(N2CCC(CO)C(C)(C)C2)=O)CC12CCC2 c1(C2c3n(nnn3)CCN3CCCC(C3)CCN2)cccc2c1OCC2.CCSC Cc1cc(C(=O)N(C2CCC(NC(c3ccnnc3C)=O)CC2)C)nc(C)c1 C(=O)(CC(F)(F)C(F)F)NCCC(C)N(C)C(C1C(F)(F)C12CC2)=O C1(CC(=O)N(C(CC(C)C)C)C(=O)CN)CC2(C1)CN(C(=O)CN1CCCC1)C2 N1(C(C(C)C#N)=O)CCC(NC(C2CCC(c3ccccc3)C2)=O)C(C)(C)C1 C(=O)(C1=CCC2(COC2)OC1)NCCOCCNC(Cc1nc(C)[nH]n1)=O N1(CCCCCNC(C2CC3C=CC2C3)=O)CCN(C(=O)COCC(F)F)CC1 N1(C(c2cc(C)c(Cl)cc2)=O)CC2OCCN(C(=O)CC3CCCN(C)C3)C2C1 C1(CC#C)(NC(C2CCCCC2CNC(=O)CSCCC(C)C)=O)CCOCC1 CC(CN(C)C)CCC(=O)NCCCN(C(C1(F)CCN(C)CC1)=O)C1CC1 C(=O)(CCC(C)NC(C)=O)NC(CCN(C(Cc1ccc(C(C)=O)s1)=O)C)C c1(C(N2CCN(C(C3C(F)(F)C34CC4)=O)CC2)=O)nnn(C2CC2)c1C(F)F c1(N(C)CCN2CCCCCC2)[nH]c(=NCCc2cn[nH]c2)nc2c1cnn2C Cc1csc2ncc(C(=O)N(CCNC(=O)C(F)C3CCOC3)CC3CC3)n12 c1(OC)cc(CC(=O)NC(C)(C)C(C)NC(=O)CCc2ccsc2)c(F)cc1O CP(C)(=O)C1CCC(C(=O)OCc2cc(-c3ccco3)on2)C1 C(CCC(c1ccccc1)NC(=O)Cc1cnco1)NC(CSCC=C)=O C(C(=O)NC)(C1CCSC1)N(CC(C)C)CC=C C=CCC(C)(CC=C)NC(=O)CCC1(NC(c2ccc(Cl)o2)=O)CCCC1 C1(C(C)C(=O)NCF)CCCN(C(=O)C(C)(C)N(C)C)C1 C(=O)(CCCC(=O)NCC)NCCCC1OCCN(C(C(COCC)C)=O)C1 Cc1cc(C(=O)NC(CNC(=O)C(C)O)C2CCC2)c2cccc(C)c2n1 C1(NC(c2cc(Cl)c(F)c(Cl)c2)=O)CCc2nc(NC(=O)C(O)CCl)sc2C1 CC1(C)CN(C(=O)CCC2CC2(Cl)Cl)CC1NC(=O)C1=NNC(=O)C1 c1(CC(=O)Nc2cncc(CC)c2)cc(Br)ccc1C N1(CC(N2CC(O)(CNC(c3ccc(Br)o3)=O)C2)=O)Cc2ccccc2C1=O CCCCS(=O)(=O)NCC(N1CCOC(C(C)NC(=O)C(F)(F)CO)C1)=O C1(CNC(c2n(CC)ncn2)=O)CCC(C)N(C(c2cnc(C)s2)=O)C1 C1(N(C(CC=CC)=O)C)CCCCN(C(C2CC=C(C)CC2)=O)C1 C1(CC)C(NC(=O)C=Cc2ncc[nH]2)CCN1C(C1CCS(=O)CC1)=O Cc1nc(=NCC2CC3CCC2N(C(C2CCS(=O)(=O)C2)=O)C3)[nH]cc1Br N1(C(C(CCC)C#N)=O)CCC2(CC1)CC2CNC(=O)Cn1cc(C)cn1 N1(C(CC2CC(C)(C)C2)=O)CC(F)(F)CC1CCNC(C1CC1CF)=O N1(Cc2c(C)cccn2)CC2(C1)CN(c1ncc(Br)cn1)C2 C1(C(N2C(C(N(CCCCCC)C)=O)C(O)CC2)=O)CCC2(CC1)CC2 Cc1ccc(C(N)=O)cc1C(N1CCC(NC(c2cccc(Cl)c2)=O)C(O)C1)=O C1(N(C(=O)C(C)=CC(C)(C)C)CC)CCCN(C(c2ccc(N)c(N)n2)=O)CC1 C1(CNC(C2C(NC(c3nc(C)oc3)=O)CC=CC2)=O)CCC(C)(C)CC1 C1(C2CN(C(C34CCCN3CCC4)=O)C2)(NC(C(CC)N2CCCC2=O)=O)CC1 C1(CC(=O)O)(C(N2CCN(c3ccncc3)CC2)=O)CC2(CCOCC2)C1 Cc1ccc2nc(C(N3CC(CN(C)C(c4ccnn4C(F)F)=O)C3)=O)cn2c1 N1(C(C2(C#N)CC(C)C2)=O)CCC(NC(C2(C)CCCC2)=O)C(C)(C)C1 C1(CNC(CC2CCN(C(C34CC(CCC)(C3)C4)=O)C2)=O)CC(=O)N(CC)C1 C1(NC(=O)OC(C)(C)C)CN(C(=O)NCCc2cc(Cl)cc(Cl)c2)CC1C1CC1 C(=O)(CC(C(C)CC)NC(C1CN(C(C)=O)C1)=O)Nc1ccc(CC)cc1 c12ccc(cc1)CC(O)CN2Cc1cscn1.C1(C(=O)OC)CCSCC1 c1(C(N2CCC(CNC(C(C(C)C)N(C)C)=O)CC2)=O)cnn2c(=O)cc[nH]c12 C(N=c1[nH]nc(C(N)=O)s1)C1C(NC(C2(C)CNC(=O)C2)=O)CCCC1 N1(C(=O)C2=CCCCC2)CCC(C2CCCN(C(C3COCCO3)=O)C2)CC1 Cc1ncnc2c1CC(C(=O)NC1(CCNC(=O)C(CO)N(C)C)CC1)CC2 C1(C(N2CC(CC=C)(C(N3CCC=C(C)C3)=O)C2)=O)CCCCC(=O)N1 c1(C(N2CC(NC(C3(C4CCCO4)CC3)=O)C(C(F)F)C2)=O)cc(F)cc(F)c1 N1(C(c2nncn2C)C(=O)NCC=C)CCC(N(C)C)(CC)CC1 C1(O)(CNC(CCCc2scc(C)n2)=O)CCN(C(=O)CSC(F)(F)F)CC1 c1(OC)ccc(CC(=O)NC2CCOC(CN)C2)c(Cl)c1OC S(=O)(=O)(C1CCOC1)Nc1cc(C(=O)OC)nn1-c1ncccc1Cl C1(COC)(CNC(=O)CP(C)(C)=O)CCN(C(C2(C)CCCN(C)C2)=O)CC1 c1(OC)ccc2cc(C(N3CC(CNC(=O)C(C)O)CC(C)(C)C3)=O)n(C)c2c1 C=CCCC(C(=O)OC)NC(c1cc(OC)c(-c2cc(F)cc(F)c2)cn1)=O c1(SC(C(=O)N(C2CCN(C(CCNC(C)=O)=O)C2)C)C)ccc(C#N)cc1 N1(C(c2cc(C)[nH]c2)=O)CC2(CC2)CC1C(=O)NCCc1ccon1 CC1CC(=O)NC(C(=O)NC2(CNC(c3ccc(OC(F)(F)F)c(Cl)c3)=O)CC2)C1 Cc1ccc2nc(C(N3CC(N(C)C(C4CCC5CCC(=O)N45)=O)C3)=O)cn2c1 CC1CCC2(CCC2)CN1C(=O)NC1CC1(c1ccc(Br)cc1)C c1(OC)ncc(C(=O)NCC2CCCCCN2C(=O)CCNC(=O)CO)cc1C C1(CNC(C2(S(N)(=O)=O)CC2)C)CC2(C1)CC(F)C2 Cc1cnn(C(C)C(=O)NC2CCC(CNC(C3CC(F)C3)=O)C2)c1 CCC(C)C(CC(=O)NCCC(C(C)C)OC)NC(=O)C(O)CC(N)=O n1(CC(N2C3CN(C(C(CC(C)C)F)=O)C(C3)C2)=O)ccc2ccc(F)cc12 C1(CNC(c2c(C)snc2)=O)CN(C(c2ccccc2)=O)CCN1C.C1(N)CC1 c1(NCC(C)Cn2ccnc2)ncccc1S(=O)(=O)N1CCCC1C1CC1 N1(C(c2c(N)nccn2)=O)CCOC2CN(C(=O)COc3ccon3)CC12 c1(NC(c2csc(CO)n2)=O)cccc(F)c1F.C12CC(C1)C(=O)NOCCC2 Cc1nc(CC(C)C)c(C(=O)NC(C)C(CO)NC(=O)CSC(F)(F)F)s1 N1(C(C(CC)OC)=O)CC2CCN(C(c3ccccc3C)=O)CC12 n1(CC)ccnc1C(=O)NCCCCCN(C(=O)CC1CC1(Cl)Cl)C c1(C(=O)NCc2ccn(CC)n2)c[nH]c2cc(C3=CCCCC3)cnc12 C1(C(N(CCN(C(=O)CC(C)N2CCCC2=O)C(C)C)C)=O)CCCC(C)(C)O1 C(CC1=CCN(C(c2csnc2Cl)=O)CC1)NC(c1c(OC)ccs1)=O C(=O)(CC(=O)NCC(CNC(=O)CC1CCCOC1)CO)OCC c1(OC)cccc(C(C)=CC(N2CCN(C(c3ccc(C)s3)=O)C(C)C2C)=O)c1 CN1CCC12CN(C(C13CC1CN(C(C1CCCCC1(C)C)=O)C3)=O)C2 N1(C(=O)NC2CCCCC2Oc2ccccc2)CCNC(c2ccc(Br)cc2)C1 N1(C(C2CCC(C)(C)OC2)=O)CCCC12CCCN(C(=O)C=CC=C(Cl)Cl)C2 c1(CCC(=O)NCCC2CN(C(C(C=C)(F)F)=O)CC2C)ccc(Cl)c(OC)c1 N1(C(C(C)OCC)=O)CCC(NC(c2cnc(F)c(Cl)c2)=O)C(CC)C1 c1(C(=O)NCCC(C)NC(C2CCOC2C(F)(F)F)=O)ncc(C(F)F)s1 N1(C(C2(C(C)(C)C)CC2)=O)C(CNC(=O)CC2(O)COC(C)(C)C2)CC2COCC12 CC1CN(C(=O)Cc2cc(Br)ccc2O)CCN1C(C1CCC1)=O C(CCF)(C(=O)N1CCN(C(=O)Cc2coc(-c3ccccc3)n2)CC1)N(C)C c1(OC)ccnc(C(=O)NC(C)C(CO)NC(=O)C(C)P(C)(C)=O)c1OC N1(C(c2c(CC)onc2C)=O)CCN(C(=O)C(C)CF)C(c2ccccn2)C1 N1(C(Cc2nc(=N)[nH][nH]2)=O)CCC(CO)C(NC(=O)Cn2cnc(C(N)=O)n2)C1 N1(C(C2N(C(C(C)NC(=O)OC)=O)CCC2)=O)CCOCC2(CC2)C1 C1(NC(C2CCCOC2)=O)CN(C(c2cc(O)nc(O)n2)=O)CCC1F C(C(CNC(C1C2COCC12)=O)C(F)(F)F)NC(=O)CCSc1ccccn1 c1(C(=O)NC(C)CN(C)C(C2CCC(=O)N2)=O)cncc([N+](=O)[O-])c1 c1(C(=O)NC(CN(C(=O)CC2CC(C)=NO2)CC)C)ccc(COC)s1 c1(C(=O)NCC(C)(CO)NC(CC2(COC)CC2)=O)cccc2nc(C)nn12 c1(C(N(CCNC(c2cccc(CC)n2)=O)C)=O)ccc2c(c1)COCO2 Cc1ccc(Br)c(F)c1C(=O)NC1CCC(C)(CN)CC1 c1(C(=O)NC2CC(NC(c3c(COC)ncs3)=O)C2)cnn(CC(F)(F)F)c1C Cc1ccc(C)c(C(=O)NC2(CCNC(=O)C3=CCSC3)CCC2)c1 c1(CCC(=O)NCCN(CCCN(C)C)C(C2N(CC)CC2)=O)cnc(C)o1 C(C(=O)N(C)OCC)NC(CNC(C(C1CCCC1)OCC)=O)=O N1(C(C=NOC)=O)CC2CC(NC(C3(C4CCOCC4)CC3)=O)CC2C1 C=CC(C(=O)N(C1CCN(C(c2csnc2C)=O)C1)CCO)c1ccccc1 C1(C(=O)OC)C(C(=O)NCCCN(CCCNC(=O)CN(C)C)C)C1C(C)C N1(C(CCOCC#C)=O)C(C(=O)NCC2CCCSC2)CC2CCCC12 c1(C(=O)NC2C(NC(CNC(C(CC)C)=O)=O)CC2)c(C)cncc1C c1(C(N(CC(C)N(C(=O)C(N2CCOCC2)C)C)C)=O)csc(S)n1 C1(C)(C(=O)NCC(C(C)C)NC(C=C(C)Cl)=O)CC(C)(C)C1 Cc1ccc(C(=O)NC2CC(C(N3CC(OCC(N)=O)C3)=O)C23CCC3)nc1O CC(C)C1=CCC(C(=O)NCCC2CC(NC(C3(C)CCCOC3)=O)C2)CC1 c1(CC)oc(C)cc1C(=O)NCC(C(=O)NCc1nn(C)cc1C)N(C)C Cc1cn2ccc(C(=O)NC3COC4(CNC(=O)CSC(C)C)CC3C4)cc2n1 c1(C(=O)NC(C)CCN(C)C(c2c[nH]nc2C(C)(F)F)=O)ccc(Cl)cc1O C(=O)(CCCC(=O)N(C)C)NCC1(CN(C(CC(c2scc(C)c2)O)=O)C)CC1 C(CCCN=[N+]=[N-])NC(C(C1CC1)NC(C(C)n1cccc1)=O)=O O=[N+]([O-])c1ccccc1-c1ccc(C2(NCc3cc(Br)c(O)c(Br)c3)CC2)cc1 C#CCC(C)(C(=O)NCC(=O)Nc1ccccn1)NC(=O)CC1CCOC1(C)C c1(C(=O)NC(CC=C)CNC(C2CN(C(C)=O)C2)=O)ccc2cc(Cl)ccc2c1 C(=O)(C(C(C)C)CN)NC1COCC1Cc1cnn(C(=O)NC)c1 c12ccc(Br)cc1C(=O)N2.c1(C(N(C(C)C)CC)=O)c(I)n[nH]c1C N1(C(C(c2cccc(Cl)c2)C)=O)CCC(NC(c2n[nH]cc2Br)=O)C1C c1(CC(=O)NCC(O)CCNC(c2ccc(C(F)F)nc2)=O)cncnc1O N1(C(C2(OC(C)=O)CC2)=O)CCC(F)(C(=O)NC2(C3CCCO3)CC2)C1 c1(OC)nccc(-c2ccnc(C(=O)Nc3nc(C4CC4)cc(C)n3)c2)c1OC c1(C(=O)NCCCCCNC(C(C)Cn2cccn2)=O)cnc2c(ccn2C)c1 c1(C(=O)NCC(CC(C)C)NC(C2(C)CC=CCC2)=O)c(F)ccnc1Cl C(=O)(C#CC(C)(C)CNC(c1ccncc1Cl)=O)N1CC(O)(C(=O)OC)C1 N1(C(CCN(C)CC)=O)C2CCC1CC(CCNC(=O)C(C)(C)NC(C)=O)C2 CC(c1cccc(Cl)c1)=CC(=O)NC1CCCC1CNC(=O)C(C)C1(O)CCC1 C1(C(=O)OC)OC(C(=O)N(CCCNC(=O)CCSC2CCCCC2)C)CC1C c1(OC)cccc(C2CC(O)CN2C(=O)C(C)n2ccnc2)c1 N1(C(CN(C)CC)=O)CCC(C2CCCN(C(c3cn4c(n3)CCCC4)=O)C2)C1 N1(C(c2c(C)n[nH]c2)=O)CCC(NC(C2CC3(CC3)CO2)=O)C1C C1(CN(C(=O)CSCCC#N)C)CCCN1C(=O)CCc1ccncc1 c1(NC(C2SCCN(Cc3c(C)cc(Br)cc3C)C2)=O)ccc(Cl)c(C#N)c1Cl C(CC1CCC1)(C(=O)N(CC(=O)NCC1(OC(C)C)CCC1)C)OC Cc1cc(C(=O)NCC2CN(C(c3cc(F)cnc3O)=O)CC2(F)F)cc(F)c1 S(=O)(=O)(c1cnn(C)c1)NCC(=O)NC(CC)CNC(C1CC2CCCCC12)=O N1(C(C2(CC=C)CCC2)=O)CCC(C)C(CNC(c2cc(F)cnc2Cl)=O)C1 C#CC1(C(=O)NC(C=C)COC)CCN(C(c2ccc(C(F)F)o2)=O)C1 C(C(C(=O)N(C)Cc1ccc[nH]1)n1cc(CC(C)O)nn1)OCC C=C(C)CCC(=O)NCC(C)(C1CC1)NC(=O)COCCNC(=O)OC(C)(C)C C1(C(N2C(CNC(=O)Cc3csc(S)n3)CC(OC)C2)=O)CCc2ccnn2C1 N1(C(c2c(OCC)cccn2)=O)CCN(C(c2ccc(C#N)[nH]2)=O)C2CC12 c1(C(=O)NCCOC(C)(C)CNC(C2CC2(C)C(F)F)=O)cnn2c1OCCC2 c1(CC(=O)NCC(CC)NC(=O)CC2CC3CC3C2)cnn2ccccc12 C1(NC(CCCc2onc(C)n2)=O)CC2CN(C(c3nc(Cl)oc3C)=O)CC12 C=C(CNC(=O)CSCC1CCCO1)CCNC(=O)Cc1ccccc1 C(C1=Cc2ccccc2OC1)=CC(N1CC(NC(C2CCC(F)(F)CO2)=O)C1)=O C1(NCC2CN(C(COC3C(CC)CCCC3)=O)C(C)C2)CCC(=O)NC1=O C1(CN=C(NCC2(OC)CCC2)NCC(F)F)CCOC2(CCOC2)C1 c1(C(N2CCC3(C(=O)NCC4(F)CCC4)CC3C2)=O)ccnc(Cl)c1F N1(C(C(N)CCSC(F)(F)F)=O)CCCC(c2ccncc2)CC1 N1(CCC)CCC(C(=O)NC2CN(C(=O)CN(C)C(C)C)C3CC23)CC1 c1(CC)oc2ccccc2c1C(N1CCOC2(C1)CN(C(=O)C(C)(F)CC)C2)=O N1(C(C2C(C)C2)=O)CCCCC(C2CN(C(=O)Nc3cc(F)c(F)cc3F)C2)C1 CCCC(C(=O)OC)C(=O)N(CC(O)CN(C(=O)COCC)C)C N1(C(c2nn(C)c(F)c2)=O)CCC2(CCN(C(C3CCCCS3(=O)=O)=O)C2)C1 CCC(C)C(O)CC(=O)NCCC(C)(C)NC(c1cn2ccsc2n1)=O c1(C(C)NC(c2cncc(NC(C3CCOCC3)=O)c2)=O)ccc(Br)c(F)c1 Cc1ocnc1CNC(=O)C(c1ccnn1C)NC(=O)COC1CC=CC1 c1(CC(=O)NCC(CC)NC(c2nocc2Cl)=O)csc(C2CCOCC2)n1 C1(N(C(=O)C=C(C)C)CC)CCCN(C(c2ccc(C(=O)OC)s2)=O)C1 Cc1cc(F)cnc1C(=O)NCC(C1CCCN1C(c1cnc(C)n1C)=O)(C)C C#CCC(C)(C(=O)NC(CO)CC(C)CC)NC(c1nonc1C)=O CC1CN(C(=O)C=CCF)CCN1C(C1CCCN1CC(F)(F)F)=O CC1(C)CCCC(C(=O)NC2(C)CCCC2NC(C2CC3C(C2)C3(C)C)=O)C1 C(C)(CCNC(C1(OC)CC1)=O)N(C(C=C(CC)C)=O)C N1(C(C(C)S(N)(=O)=O)=O)CCC2C1CCCN2C(c1nccc2n[nH]cc12)=O C1(CNC(c2cc(OCC)ns2)=O)N(C(C2CC(C)=NO2)=O)CCCC1(C)C C(=O)(C1CCc2c[nH]nc21)N1CC2CN(C(c3c(C(C)(C)C)c[nH]c3)=O)CC2C1 CC1CC2CN(C(=O)C(C)O)CC2N1C(=O)Cn1cnnn1 O=C1CSCN1CC(N1CCC(Cn2cc(CO)nn2)C1)=O.N12CC=CC1C2 Cc1cc(Cl)ncc1S(=O)(=O)N1Cc2ccc(-c3cnc4ccccc4n3)cc2C1 CCC(C)(C(=O)O)N(C)C(c1ccc(NCCc2ccco2)cc1)=O CCCCS(=O)(=O)CC(=O)NC1CN(C(C2CC(N=[N+]=[N-])C2)=O)CC2(CCC2)C1 CC1(C)CN(C(=O)Cc2ccccc2O)CC1NC(=O)C(O)Cc1ccccc1 CC(C(=O)NC1CCN(C(=O)Cc2nc(C3CC3)nn2C)C1C1CC1)C(C)(C)C Cc1ccc(C(N2CC(CC(=O)NC3CC(C)OC3=O)C3(CC3)C2)=O)c(O)c1 Cc1nc(C(N2CC3CC2CC3N2CCCC(CF)C2)=O)ccc1Br N1(C(C(CSC)C)=O)CC(NC(=O)C(C2CCCCC2)O)C(CC(C)(C)C)C1 c1(C(N2Cc3cccnc3C2)C(=O)NC(CC)(C)C)nc(Br)c2ccccn12 c1(C(N(C(CCNC(c2cc(CC)[nH]n2)=O)C)C)=O)ccc(C(C)=O)cc1 C(CC(=O)N(CC(F)(F)F)CCOC)OCC=CC(=O)NCCCOCCOC.C(C)=C N1(C(c2cccc(OC(C)C)c2)=O)CCC(C)N(C(c2c[nH]ccc2=O)=O)CC1 c1(NC)cnncc1C(=O)N(CC(C)N(C(=O)CC1CCC1C(=O)O)C)C c1(C(=O)NC2CCC(C)N(C(=O)COc3cn[nH]c3)C2)cncc2ncn(C)c12 c1(C(=O)NC(C2CCCN2C(=O)C(F)C2CCC2)(C)C)c[nH]nc1-c1ccoc1 c1(C(=O)NC2CN(C(CCOC)=O)CC(O)C2)nn(C)c(=O)c2ccccc12 C(=O)(C(C=C)CC)NC(COCC)C(=O)N1CC(CC)C1 C1(C(=O)NCCC(C)(C)NC(=O)CN(C)C)(OC)CCSC1 c1(C(=O)NCC(C)NC(C2CC(C)(C)CC(C)(C)C2)=O)cnc2nccnc2c1 C1(CC(=O)NCCC(C)(C)NC(c2cc(OC)n[nH]2)=O)CCCCN1C c1(C(=O)NCC2C(CNC(c3c(COC)noc3)=O)C2)[nH]cc2c1CCCC2 N1(C(c2cncc(OCC)c2)=O)CCCC2(CCC(NC(=O)CC(F)(F)Cl)C2)C1 CCC(CC(=O)NCC(O)(COC)CO)SC.C12C(C1(F)F)CNC2=O C1(C(=O)NCC(C)CNC(=O)CCc2cn[nH]c2)C2CCN(C)CC12 c1(OCC(N2C(CNC(C(C)OC)=O)C3CC3C2)=O)cccc(F)c1F c1(C(N)=O)ccccc1-n1ccc(-c2cnc(C3CC3)nc2)n1 N1(C(c2cnc(C(C)C)s2)=O)CCC=C(CNC(=O)CC(C)(C)CN(C)C)C1 c1(C(N(C(C2CCCCC2)C)C)=O)cccc(CNC(=O)C(F)C2CCOC2)n1 C1(C(=O)NC(C)CNC(=O)CCc2cnco2)CCC(=O)N1 CC1(C)CC(NC(C2(C)CCC(=O)N2)=O)CN1C(C12CC(F)(C1)C2)=O C1(CNC(=O)OC)CC(C)CC(C)(C)C1.C12CN(CCO1)C2=O N1(C(c2c(CC)c[nH]c2)=O)CC(C)(C)C(NC(=O)C(C)CC2CCC2)C(C)(C)C1 C(=O)(C(CNC(C1CCC1)=O)CC1CCCC1)NC(C1CC1(C)C)CC N1(C(C2CC(SC)C2)=O)CCCC(C)(C)C1CNC(c1cncn1C1CC1)=O C1(CNC(c2c(CCC)nns2)=O)CCC(C)N(C(c2ccc(O)nn2)=O)C1 CN=S(=O)(c1ccc(NC(=O)NCC2CCC3C4C=CC(C4)C23)cc1)N(C)C Cc1cccc(F)c1C(=O)NC1CN(C(=O)Cc2ccc(F)cc2)CC1CO c1(C(=O)NCC(CNC(C2CC(F)(F)C2)=O)C(F)(F)F)cccc2c1COC2 c1(C(N2CC(NC(=O)C(C)(C)N(C)C)CC(C)C2)=O)n[nH]c2c1CC1CC21 O=S(=O)(c1cnc(N2CC3CC3C2)c(Cl)c1)N1CC23CCC2(COC3)C1 CC1CCN(C(C2(C)CCN(C(c3ccc(CO)cc3F)=O)C2)=O)CC1(F)F Cc1ccc(C(N2CCC(C)(NC(c3cc4sc(C)cc4[nH]3)=O)C2)=O)c(F)c1F c1(C(=O)NC2CC(NC(c3c(-c4n(C)ncc4)n[nH]c3)=O)C2)cncc(N)n1 C1(NC(c2c(C#N)ccs2)=O)CCN(C(=O)COC(F)F)CCC1(F)F C(=O)(CCCCCCNC(C1CC(=O)CC(=O)N1)=O)NC(C(CC)C)C(=O)NC n1(C(COC)C)nc(-c2cccc(SC(C)(C)C)n2)nc1-c1cnc(Cl)n1C c1(C(N2CC3CC(O)CC2C3)=O)cc(Br)c2nccnc2c1 N1(CC(=O)N(CCNC(C(C(C)SC)O)=O)C(C)C)C(=O)CCCC1=O N1(C(C2C(C(C)C)CCO2)=O)CCCCC1CCC(=O)NC1(C)CC1(C)C CCC(C)C(C(=O)N1CCCC1CNC(C1OCCC1C)=O)N(C)C N1(C(c2cc3n(n2)CCC3)C(=O)NCCOC)Cc2ccc(OC)cc2CC1C c1(C(N(CCC(C)NC(C(CC)OC)=O)C)=O)cc2cc(F)cc(F)c2[nH]1 N1(C(c2cccc(C)n2)=O)C2CCC1CC(NC(C13CCC1C3)=O)C2 c1(C(N2C(CN(C)C(c3nnsc3N)=O)CCC2)=O)ccc(O)nn1 C1(NC(c2cccnn2)=O)CCCC12CN(C(c1cc3nc[nH]c3cn1)=O)C2 C1(C(C)C)CCCC(NC(c2ccc(CNC(=O)CC(C)(F)F)s2)=O)C1 C1(C(N(CC(=O)N(CCCCC(=O)OC)C)CC2CC2)=O)CCC(N=[N+]=[N-])C1 C(c1nc2ccccc2[nH]1)=CC(N1C(CNC(C(C(C)C)(C)O)=O)CC(O)C1)=O C(=O)(CCC(C)(C)[N+](=O)[O-])NC(CNC(CC(C)O)=O)CC(F)(F)F Cc1cn2c(C(=O)NC3CN(C(=O)C(C)CC(N)=O)C4CC34)cnc2s1 c1(C(N(CCC(C(C)(C)C)NC(CCC=C)=O)C)=O)ccnc2cc[nH]c12 C1(C(NOCCOCC)=O)CN(C(=O)C(C)(C)CF)CC(C)O1 c1(C(=O)NC2C(NC(CCCC)=O)CCC2)ccc(C(C)C)cn1 c1(N(C(c2sc3cc(C)sc3c2)=O)C2CC2)cccc2ccc(CN=[N+]=[N-])cc12 CC1CN(C(=O)CCc2nncs2)CC1(C)CNC(=O)C(c1cccn1C)=O C1(NC(=O)COC2CCOC2)(CO)CN(C(C2CC2c2ccncc2)=O)C1 C1(C(=O)NCC23C(CN(C(C4(C#C)CCCC4)=O)C2)C3)CC2(CCOCC2)CO1 N1(C(=O)NC2CCC(Oc3ccccc3)CC2)CCC2(C1)OCc1ccccc12 O=S(=O)(c1cc(Cl)c(I)s1)N1CC(O)CC1c1cc(F)c(F)c(F)c1 C(CC(CC)C(=O)N(CCCCNC(=O)CC(C(F)F)n1ccnc1)C)=CC C1(C(=O)NC(C)CCO)CCCN(C(c2cc(Cl)c(Cl)s2)=O)C1 Cc1cc(C(=O)NCC(C(C)(C)C)NC(C2CCC23CCC3)=O)cnc1O C1(C(N2C(C(=O)NC3CC(C)(CC)C3)C3CC3C2)=O)CC2OC1C1CC21 c1(C(N(CCCNC(c2cnn(C3CC3)c2)=O)CCO)=O)ccc2c(c1)CCO2 N1(C(c2ncn(C)n2)=O)CC2(CC(CNC(c3cnn(C4CCC4)c3)=O)C2)C1 C(=O)(C1=CC(O)CCC1)N(CC(C)N(C(=O)C#CC(C)(C)C)C)C C(CCC(=O)NCCn1cc(-c2c[nH]nc2C(=O)OC)nn1)N(C(C)=O)C1CC1 CCCC(O)CC(=O)NCCCCNC(c1scnc1C(F)F)=O N1(Cc2cnc(CCOC)s2)CCCC(c2cccc(C(=O)OC)c2)C1 N1(C(C2CC(C)CN2C(=O)C=Cc2ccccc2)=O)CCC(O)C(C)(CO)C1 Cn1cc(C=CC(=O)NCCOCCC(=O)NOCCCF)nn1 c1(C(N(C2CCC(CNC(c3cc(C)sn3)=O)CC2)C)=O)cc2cn[nH]c2cn1 C(=O)(C(CC(C)C)NC(c1sc(C)cc1C)=O)N(CCC#C)CC N1(C(C2N(C)CC2)=O)CCCC2(CCCN2C(C2CCc3c[nH]nc3C2)=O)C1 c1(C(N2CCC(OCCCNC(C(C)(C)F)=O)C2)=O)ccc(C2CC2)cc1 CC(C(=O)NCC1(O)CN(C(c2ccc(F)cc2F)=O)C1)S(C)(=O)=O c1(C(=O)NCC2OCCC(NC(C3(CC)CCC3)=O)C2)cc2c(Cl)nccc2o1 C1(CC=C)(C(=O)NCCP(C)(C)=O)CCN(C(=O)C(C)O)C1 C1(NCc2c(OC)nc(Cl)cc2)CC2(C1)CC1(CCCC1)C2 CC1(C)CCN(C(c2cccc(F)c2F)=O)C1CNC(C1(C)CCCS1(=O)=O)=O c1(C(N2CC(NC(c3cocn3)=O)C(O)C2)=O)cnc2ccccn2c1=O c1(CC)ccccc1C(CNC(c1ncncc1Cl)=O)NC(c1cc(F)n[nH]1)=O C(C1=CCN(C(=O)CCCSC)CC1)NC(CCc1onc(C(C)OC)n1)=O O=C1CC2CCC1C(C(=O)Nc1nc(-c3c[nH]c4ccccc34)cs1)C2 C(=O)(CCCCC(=O)NCC(C1CC1)NC(=O)CSCc1cccs1)NC c1(NC(C2CN(C(=O)Cc3ccc(Cl)c(Cl)c3)C2)=O)cccc(C#N)c1[N+](=O)[O-] CON1CCC(C(=O)NCC2C=CCN2C(c2cc(-c3ccco3)[nH]n2)=O)CC1 N1(C(c2ccc(C)nc2O)=O)CCC2C(CCCN2C(=O)Cc2[nH]cnc2C)C1 C(=O)(CS(=O)(=O)C1CC1)NC(C)CN(C)C(C1CCCCN1S(C)(=O)=O)=O C1(NC(=O)Cc2ccccc2)CCN(C(C2CCCC23CC3)=O)CC1 N1(C(c2ccccn2)=O)CCN(C2CN(Cc3scnc3Cl)C2)CC1 Cc1cnc(N2CCOC(C(C)NC(c3cc(Cl)n(C)n3)=O)C2)nc1 c1(OC)ccc(C(=O)NCCC(C)CCNC(c2cc(SC)oc2C)=O)c(F)c1 C(C(C)(C)CNC(c1ccoc1)=O)N(C(=O)CC(C)c1cnn(C)c1)CC Cc1nc(Cl)ccc1CC(=O)NCC1CCCCC1NC(c1ccccn1)=O C1(SCC(=O)NCCC(Cn2cc(C(C)(C)S(C)(=O)=O)nn2)F)CCC(=O)NC1 C1(CC)CN(C(C2CC(=O)N(c3cc(OC)ccc3Cl)C2)=O)CC(=O)N1 C(=O)(CCC(CC)CC)NC(CC)C(=O)NC1CC12CC(O)C2 N1(C(CCC=C(C)C)=O)CCC(O)(C2(NC(C3C(Cl)(Cl)C34CC4)=O)CC2)CC1 C1(CN(C(C2CC(SC)C2)=O)C)CCCN1C(=O)C(C)=C1CCCC1 N1(C(C(N2C(CC)CNCC2)=O)=O)CC2(CCC2)CCC1CC(=O)NCC(F)F C(=O)(C(F)C(F)(F)C(F)(F)F)NCc1cccc(CNC(CCCCOC)=O)c1 c1(C(=O)NC23CN(C(C(COC)(C)OC)=O)C(CC2)C3)cc(F)c2[nH]nnc2c1 C(=O)(CCCCCF)NC(C1CCCN(C(C(COC)COC)=O)C1)C c1(C(=O)NCC(CC)N(C)C(c2cccc(N)n2)=O)ccccc1NC(N)=O c1(C(N(CCCNC(=O)CCNC(N)=O)CC)=O)ccc2nc(O)[nH]c2n1 c1(OC)cccc(C(F)(F)C(=O)NC(CNC(=O)C=CC(=O)N(C)C)C2CC2)c1 N1(CCCC(=O)N(c2ccc([N+](=O)[O-])cc2)C)CCC(=O)N(CC(C)(C)C)C1=O Cc1cc(CC(N2CC(=C(F)CNC(=O)C(n3nccc3C)C)C2)=O)ccc1O c1(C(=O)NC(C(C)NC(CCCCC)=O)C)c[nH]c2cc(C(=O)OC)ccc12 N1(C(c2cc(CNC(c3cnc(C)s3)=O)no2)=O)CC(F)CC1CO c1(C(=O)NCC2N(C(C(C3CCOCC3)C)=O)CC2)cc(CC2CC2)sn1 N1(CC(=O)N(CCC(=O)OCCN(CCOC(C)=O)C)C)CCC(C)(C)C1 C1(NC(C(C)n2ccnc2)=O)CC2C(NC(=O)CCCn3cncn3)C2C1 c1(-c2cn(CCN(C(=O)CCC(=O)N(C)C)CC)nn2)cccc(S(C)(=O)=O)c1 C(=O)(C(=O)N=S(C)(C)=O)N1CCC(C(C)NC(=O)CC2COC(C)(C)C2)CC1 N1(C(c2c(CC)cc[nH]2)=O)CC(C(=O)N(C2CNC(=O)C23CC3)C)CC(C)(C)C1 c1(CC(C(=O)NCC(C(C)(C)C)NC(CCC(=C)Cl)=O)C)ccc(C#N)cc1 CC1(C)CN(C(C2CC3CCC(C2)O3)=O)C(CNC(c2cnns2)=O)CO1 c1(C(CC(=O)OCC)NC(c2ccc(NS(C)(=O)=O)cn2)=O)ccc(Cl)c(F)c1 Cc1nc2ccc(Br)cc2cc1NC(=O)NNc1cncnc1 c1(C(CC)NC(=O)NC(c2ccccc2)CC)ccc(C)cn1 N1(C(C2(CCOC)CCCC2)=O)CCN(C)C(CNC(C2CC2(C)C(C)C)=O)C1 c1(-c2cccc(NC(Cc3cc(C)no3)=O)n2)cc(N2CCCCC2)ccc1F c1(C(=O)NCCC(C)N(C)C(c2ccc(C3CC3)o2)=O)snnc1C1CCC1 C(C(C(=O)NC1(C(F)(F)F)CC(NC(=O)OC(C)(C)C)C1)N(C)C)SC N1(C(CCNC(N)=O)=O)CC(CNC(=O)C=CC2CCCC2)C2CC12 c1(OC)c(Cl)ccc(C(N2CC(NC(=O)CC3(C)CC3)CCC2C)=O)c1F C1(CNC(C2(C)CC2(F)F)=O)CN(C(C2C3CC4C(C3=O)C24)=O)CCC12CCC2 c1(S)ccccc1.C12(CC(NCC(=O)OC)C1)C(=O)NC2.c1(O)cnn(C)c1 C12(C(=O)NCC(=O)NCC(C)C)CC1CCN2C(=O)CC=C(Cl)Cl N1(C(C2ON=C(CC)C2)=O)CCC(C2CCN(C(=O)C(C)(C3CC3)OC)C2)CC1 C1(C(=O)NCC(C)NC(=O)OC)CSC(C)(C)C1 C1(CNC(=O)CCOCC2CC2)CC12CCN(C(c1ccsc1Br)=O)CC2 c1(C(N2CC(OC)C(NC(=O)CCc3nc[nH]n3)C2)=O)cc(F)c(C#N)c(F)c1 N1(C(CSCC)=O)CCCC(C)(C)C1C(=O)NC1CN(C(N)=O)C1 CC(CN=c1c(C#N)c[nH]c2c(F)ccc(F)c12)N(C)C(c1ccnc(O)c1)=O c1(C(=O)NCC2N(C(C(COC)COC)=O)CC2)ccnc(S(N)(=O)=O)c1 N1(C(C2(OC)CCC(C)C2)=O)CCCC(CCNC(=O)C(F)=CC2CC2)CC1 C1(NC(CC2(C)CCN2C(=O)CCc2nc[nH]n2)=O)COC2(CCC2)C1 c1(NC(CN2CC(CC#C)(C(=O)O)OCC2)=O)nc2cc(F)cc(F)c2[nH]1 C1(CC(=O)NC2CC(n3cc(C(CC)(C)O)nn3)C2)(CO)CCCCC1 C(C)(C)(CC(=O)NC1(CCOC)CCN(C(=O)C(Cc2cnc[nH]2)OC)C1)OC N1(C(c2ccc(I)cc2Cl)C(=O)Nc2c(C)cccc2C)CCCC2CCCC12 CC1=C(C)CC(C)(C(=O)NC(C)CCNC(c2cc(C#N)[nH]c2C)=O)CC1 c1(-c2c(NC(C)=O)cccc2)cccc2[nH]c(C(=O)NCC(O)C(F)(F)F)cc12 C1(C)(C(=O)NCCCCCC)CCN(c2ccnc(N(C)C)n2)C1 CCC(CC)CCC(=O)N1CCCC(C(C)NC(=O)CSC(F)(F)F)C1 c1(OC)cc(O)ncc1C(=O)NC1CCC(Nc2cc(C(C)(C)C)ncn2)C1 N1(C(c2ccc(OC)cn2)=O)CCN(C(c2cnc[nH]2)=O)C2COCC12 C(=O)(CCCc1ccccn1)NC(C1CCCN1C(C1CC1c1ccco1)=O)C CCC(C)C(C)N(C(CC1CCCCO1)C(=O)NCCCF)C C1(C(=O)NC(C2N(C(c3c(C)nc(O)cc3)=O)CCC2)C)CN2CCCN1CC2 CC(C)CCC(O)C(=O)N(C(C)(C)CC(N1CCCNC(=O)C1)=O)C C1(NC(=O)CC2CCC(=O)N2)CCN(C(=O)CC2(N3CCCC3)CC2)CC1O N1(C(CC(C=C)C)=O)CC2CCC1C(CNC(C1(O)CCOC1)=O)C2 N1(C(COC2(C)CCC2)=O)CC(C)(C(=O)NCC2(C)CC(O)C2)CC1(C)C CCS(=O)CC(=O)NC(c1ccccc1CO)CNC(=O)C(C)OC(C)(C)C CC(C)CCC(O)C(=O)N(C)CC1CCN(C(=O)Cn2cnc(C#N)n2)C1 N12CCC(F)(F)C(C1)CNC(=O)C2.c1(C(=O)NC(COCC)C)cnc(S)n1C n1(CCOC)c(C)cc(C(=O)Nc2ccnn2Cc2cccc(OC)n2)c1C FC1(F)CC1C1CCCN(c2nc(N3CCCCCC3)c3ncsc3n2)C1 C1(CNC(c2cccnc2Cl)=O)CCN(c2ccncn2)CC1(F)F C1(n2cc(CC(=O)OCC)nn2)CCCCC1=O C1(CC)(NC(c2ccc(=O)oc2)=O)CCCN(C(c2cc(CSC)c(C)s2)=O)C1 N1(C(N2C(CC)CCC2)=O)CCN(C(=O)Cc2ccn(CC)n2)CC1 C1(CC(C)(C)C)CC12CCN(CC1CCCN1)CC2 c1(C(N(C2CN(C(C3(C#N)CCOCC3)=O)C2)C)=O)c(Br)nc2n1CCC2 N1(C(C(C(C)(C)F)(C)F)=O)CCC2(CCC2NC(c2cc3scnc3[nH]2)=O)CC1 C1(CNC(c2cccc(C(=O)NC)n2)=O)CN(C(=O)C(F)CC2CC2)CCCO1 c1(NC(C2(OC)CCSC2)=O)ccc(NC(=O)C(C)CC(C)C)cc1C C1(CC)CN(C(C2CC3(CCC3)C2)=O)CCN1C(c1ccc(CO)cc1)=O C12(C(=O)NCCC3(OC)CN(C(C4CCCN4C)=O)C3)CC1COC2(C)C C1(NC(c2n(CC)ncc2)=O)CCC2(CC1)CC2NC(C1C2C3CCC(C3)C12)=O C1(N(C(N2C(C)(COC)CC2)=O)C)CCS(=O)(=O)C1 c1(NC)ccc([N+](=O)[O-])cc1C(=O)NC(C)C(CO)NC(C1CC2CC2C1)=O c1(C(C(=O)NCC#CCNC(C2C(C)C2)=O)=O)cc(S(N)(=O)=O)cn1C C1(NC(C2C(C)(CC)C2)=O)CCSC12CN(C(=O)C=Cc1cccc(CO)c1)C2 c1(C(N2CC(C)C(C(=O)NCC3CCC(C)CC3)C2)=O)cncc(C#N)c1 Cc1ccc(C(C)NC(=O)CC2CCCN2C(=O)CCC=CC(C)C)cc1 Cn1cnc2ccc(CN3CCOCC3CC(F)F)cc12 C1(C(N2CCN(C(C=CC)=O)CC2)=O)Cc2nn[nH]c2C(C)C1 Cc1cccc2c(C(N3CCCC(F)(CNC(=O)C(Cl)=CCl)C3)=O)n[nH]c12 CCC(C)C(C(=O)NCC(C)COC)NC(C1CCCC1C(C)C)=O c1(C(N(CCNC(=O)CSc2nncn2C)CC)=O)cnc2cccnn12 C1(NC(=O)CN2CCSCC2)CCCCC1N=c1[nH]c2cc(Br)cnc2s1 C1(C(=O)NCC2C(C)CN(C(c3cnc(Cl)s3)=O)CC2)CCc2nnc(O)n2C1 N1(C(CN2C(=O)CCC2)=O)CC2CCN(Cc3ccc(Cl)s3)C2C1 CCC(CC)(CCOC)C(=O)NCc1ncoc1CNC(C1CC2(CC2)CO1)=O N(C(=NCCc1c(F)cccc1F)NCC(c1ccc(F)cc1)(F)F)C1C(C)C1 C1(C(N2CC(CNC(C3C(C)(Br)C3)=O)C2)=O)Cc2cc(F)ccc2C(=O)O1 c1(COC)cc(C(=O)NC2CCCC2NC(=O)C=Cc2cccs2)n(C)c1 C1(OCC)C(Nc2cc(Cl)ccn2)COC1(C)C c1(C(=O)NC2CCC(NC(C(C)CF)=O)C2)noc2c1COCC2 C1(n2cccn2)(NC(C(CN(C)C)O)=O)CCN(C(C2(NC(N)=O)CC2)=O)CC1 N1(C(C2(CCC)CC2)=O)CCOC(C)(CNC(=O)CCS(C)=O)C1 c1(-c2nccc(NCc3nc(C)sc3)c2)ccc2c(c1)C(C)C(C)O2 n1(C(C)C)cc([N+](=O)[O-])c(=NCC2CCCN(C(C3CC=CCC3)=O)C2)[nH]1 n1(CC(=O)N(C(C)CNC(=O)C(C)(C)C(F)F)CC)ccc2ccccc2c1=O N1(C(C(C)(C)Nc2ccccc2)=O)CCC(CO)(NC(c2occc2Br)=O)CC1 C1(NC(C2C(C)OC(C)C2)=O)(CO)CCCN(C(c2cn(CCO)nn2)=O)C1 N1(C(COc2c(OC)cccc2)=O)CC(NC(c2ccncc2O)=O)C(C)(C)C1 N1(C(Cc2ccc(C)cc2)=O)CC(C(=O)NC(C(N)=O)C2CC2)OC(C)C1 c1(C(=O)NC(CNC(CN(C)C)=O)CC(F)(F)F)sc2cccc(F)c2c1Cl c1(C(=O)OC)cccc2oc(=NCCCCNC(=O)C(C(C)C)NC=O)[nH]c12 N1(C(CC(=O)OCC)=O)CCC2(CCC(C(=O)NCc3ccnc(Cl)c3)C2)CC1 C12(CNC(C(C=C)(C)C)=O)CC(COC)(CN1C(=O)Cn1cc(C3CC3)cn1)C2 C1(CNC(C(C)OCCCC)=O)CC(O)CN1C(c1nc(C)nn1C)=O C(CC(C)CC(C)(C)C)NC(c1ccccc1COC)c1n(CCC)nnn1 C1(CNC(C2(CC)CC2)=O)CC12CCN(C(c1cc(C(C)C)ccc1C)=O)CC2 CCC(C)(COC)C(=O)N1CCCCC(C(=O)NCC(C2CCC2)OC)C1 N1(C(c2cnn(-c3cccc(Cl)c3)c2)C(=O)NCCC)CC(C)CCC12CC2 c1(NC(=O)OCC)cc(NC(=O)NCC2CC(CNC(C)(C)C)C2)c(F)cc1C C12(C(N3CCC(C(C)(C)CNC(CC4(C)CC4)=O)CC3)=O)CCC(F)(CC1)CC2 CC1(CNC(c2ncc(C(F)F)s2)=O)CCN(C(=O)CCCCO)C1 C1(C(=O)NCC2(F)CC(CNC(CC3C(C)OCC3)=O)C2)CC2(C1)CC(O)C2 C=C(Cl)C(C)(C)C(=O)NCC1CCCCN(C(C2CCN(S(C)(=O)=O)C2)=O)C1 c1(C(C(=O)NCC2CN(C(C(CC)N3CCCC3=O)=O)C2)C)nc(F)ccc1Cl C1(C(N2CCCC(N(C)C(c3cnn[nH]3)=O)CC2)=O)CC(=O)C12CCCC2 c1(OCCC)cccnc1C(=O)NCC1CC(F)CN1C(c1ccc(CC)o1)=O C1(C)(C(=O)NC(C(=O)NC)CO)CCCN1C(=O)CC(C1CC1)C1CC1 N1(C(c2c(C)occ2)=O)CCC2CCN(C(C3CCC(N=[N+]=[N-])CC3)=O)CC2C1 N1(C(C(N2CCCC(C(C)N)C2)=O)=O)CCc2cc(Br)cc(F)c2C1 N1(C(c2nc(C(C)=O)sc2)=O)CCC(C(C)C)C1CN(C(c1ccco1)=O)C1CC1 Cc1c(CCC(=O)NC(C)CCNC(=O)CCN(C)CCO)cnn1C N1(C(C=C(c2ccn(C)n2)F)=O)CC(C)(C)CCC1CNC(C1(C)CCCO1)=O c1(CC)c(C(=O)NC(CNC(C2CN(C(C)=O)C2)=O)CC)sc2ccccc12 CCC(C)CCC(=O)NCc1ccc(CN(C)C(C2(F)CC=CCC2)=O)cc1 CC1CN(C(=O)C(Cl)Cl)CC1(C)C(=O)N(C)CC1(CO)CC1 CC1(C(=O)NCCC(O)CNC(C2(Br)CC2)=O)CC(F)(F)C1 C(C(C)C(C)C(=O)N(C)CC1CCN(C(C2CC(OC)C2)=O)CC1)OC N(C1CC2(CN(C(c3ccc(F)s3)=O)C2)n2ccnc21)C(c1ccc(C)nn1)=O c1(C(=O)NCC2=CCN(C(c3c[nH]c(=NC)o3)=O)CC2)cccc2sccc12 N1(C(CC(CC)C)=O)CCN(C(c2c[nH]nc2C)=O)C(CC(C)(C)C)C1 c1(OC)cccc(C(=O)NC2CCCC2(C)NC(=O)CC2CC2)n1 C1(NC(c2cnc(OC)nc2)=O)CC2CC(NC(C3COC3)=O)CC2C1 C1(CNC(C(CC)N(C)C)=O)CCCCC1NC(=O)COc1ccccn1 C1(NC(CCc2nc(C)c(C)[nH]2)=O)CC2CCC(C1)N2c1cc(C2CC2)ncn1 N1(C(C2CN(C)C(=O)N2)=O)CCC(O)C(N(C)C(C2(C)CCN(C)C2=O)=O)C1 c1(CCC(=O)NC(C2(CNC(c3c(C)scc3)=O)CC2)C)ccc(Cl)cc1Cl N1(C(c2c(CC)csc2)=O)CC2(C(=O)NCC(c3nccs3)C)CCC1CC2 N1(C(C=CC(=O)OC(C)(C)C)=O)CC2(CCC(CNC(=O)CC3CC3)O2)C1 Cc1ncc(NC(=O)C(CO)NC(c2csc(=N)[nH]2)=O)c(C)c1C N1(CC)CCOC(C(=O)NC(Cc2cnn(C)c2)C(=O)NCC)C1.C1(=O)CCN1 N1(C(c2cc(OC)c(O)cc2)=O)CCCC2(CCC2NC(C2CC2C(C)C)=O)C1 C(=O)(C(CC(=O)N1CC2(CCC(CNC(C3CC3(F)F)=O)O2)C1)C(C)=O)OCC N1(C(CCN(CCC)C)=O)CCC(C)C(CNC(c2ncsc2NCC)=O)C1 C(=O)(C#CC1CCC1)N1CC(OCC(=O)N(C)CC2CCC(=O)N2)C1 C(=O)(C(Cc1ccsc1O)NC(=O)CCc1cncnc1)OC CCCCC(CNC(c1cc(C(N)=O)no1)=O)NC(c1snc(Cl)c1Cl)=O CC(Cc1ccccn1)C(=O)N(CCCNC(=O)CSc1nnnn1C)C C(=O)(C(C)(F)C(C)(C)F)NCC(C)CN(C)C(c1ccc(C#N)cn1)=O c1(C(N2CC(C(C)OC)C2)=O)cnn(CCNC(=O)C(C)C2CCCO2)c1 c1(NC(=O)NC2(CSc3ccccc3)CCOC2)cccnc1C1CC1 CN1CC(NC(=O)Nc2cn(C3CNC3)cn2)CC12CCOCC2 C(=O)(CC(C)(O)COC)NCC(C1CC1)NC(c1nnn(CC)c1C)=O C#Cc1ccc(C(=O)NCCC(C)(C)NC(c2nc(O)sc2C)=O)c(F)c1 Cc1c(C(N2CCCC(CNC(=O)C(O)CC(C)C)CC2)=O)ccnc1Cl CCC(CC(=O)N1CC(CNC(c2ccc(-c3cccs3)cn2)=O)C(O)C1)OC c1(NCc2c(NC)cncc2)nc2c(c(=NCC34CCCC3C4(F)F)[nH]1)COC2 CC1CC(C)N(C(=O)CSc2ccccc2)CCN1C(c1cc(O)nc(Cl)c1)=O C1(CC=C)(NC(c2cnc(C3CC3)nc2)=O)CCN(C(=O)C(C)n2cncn2)C1 c1(C(=O)NC2CCN(C(COC)=O)C2)cnc2c(c1)CCC(=O)N2 N1(C(=O)OC)CSCC1C(=O)NCC1(F)CC(C(C)(C)C)C1 N1(C(CC(CC)OC)=O)CCC(C2CC2)(CNC(C2CCCN2C(C)=O)=O)C1 C1(C(=O)NC2CC(C(C)O)C2)CCC(O)CN1C(c1cccc(F)c1)=O c1(OCC)cc2ccccc2cc1NC(=O)NCC1CCC(=O)N1C1CC1 N1(C(C(CCCC)F)=O)CCC2(CC1)CC2NC(c1cccc(C)c1)=O c1(NC(C(C2CCN(C(c3ccncn3)=O)CC2)C)=O)nc(Cl)ccc1I N1(C(C(C=C=C)C)=O)CCCCCC(NC(c2cc(C)cc(C)c2C)=O)C1 Cc1cn2cc(C(=O)NC3CCN(C(C4CC(=O)NC(=O)N4)=O)C3)sc2n1 CC1(C)CC(CNC(=O)C=Cc2cnc[nH]2)CN1C(c1cccc(N)c1)=O c1(OC)cc(C(=O)NC2CN(C(=O)CCc3cnn[nH]3)CC2OC)ccc1Cl C12(SCC)CCC(C(=O)OC)(CC1)CO2.c12ccc(N)c(c1)CNC(=O)CC2 N1(C(C(C)C2CCCC2)=O)CC(C2(NC(=O)CCN3CCC3)CC2)C1 n1(CCC(N2CC(C)C(NC(c3cc4sccc4[nH]3)=O)C2)=O)ccc(O)nc1=O Cc1nccn2c(-c3nc(C(C)O)nn3-c3ccc(Br)nc3)cnc12 N1(C(C2N(C(C(CC)n3cncn3)=O)C3(CC2)CC3)=O)CC(O)C(O)C12CCC2 C1(C)(C(=O)NCC(C)(F)CNC(C2CC3CC3C2)=O)CCC2CC2C1 Cc1cc(C)n(CCC(=O)NCC2CCC(NC(=O)COCC3CCCC3)C2)n1 c1(N(c2nc3ccccc3cc2Cl)C)ncnc2c1ncn2C1COCC1O C1(CCNC(C(CC)OC2CCCC2)=O)CCCN(C(=O)Cn2cnnn2)C1 c1(C(=O)NCC2C3CN(C(C4CC(=C)C4)=O)CC32)cc(F)c(C)cc1F N1(C(c2c(C)nn(C)n2)=O)CC(O)(C2(CNC(c3cc([N+](=O)[O-])c[nH]3)=O)CC2)C1 c1(OC)ccc2c(c1Br)CN(CC1COCCC1(F)F)CC2 C(=O)(CC(=O)N1C(C(=O)NC(c2ccncc2)(C)C)CC1C)NCC c1(Cc2ccc(CN(CC)CC)s2)ccccc1NC(N1CC(CN)CC1=O)=O n1(CC)cccc1C(=O)NC1C=CC(C(=O)NC(c2cc(C)on2)C)C1 N1(C(CNS(N)(=O)=O)=O)CCC2(CCN(C(c3n[nH]cc3OC(F)F)=O)CC2)C1 c1(CNC(C2CC=CC2)=O)c[nH]nc1C1CCN(C(C2(C3CC3)CCCO2)=O)C1 c1(NC(CCC2(C)N(C(c3cn(CCOC)nc3)=O)CCC2)=O)cnc(Cl)nc1C c1(C(=O)NCC2OCC(CNC(c3c(OC)ccs3)=O)C2)cccc2nc(C)sc12 C1(OC)CCCC(NC(=O)C(=O)NCCCCCCC2CC2)C1 C=Cn1nccc1C(N1CC(C)(NC(=O)CCOCC=C)C1)=O C1(NC(c2c(C)noc2)=O)CC(F)CN(C(=O)C(C)Oc2ccc(Cl)cc2Cl)C1 CC(CC(=O)NC1CCC(C(=O)NCCCF)C1)C1CCCC1 N1(ONC(=O)C=CCO)CCSCC1c1cccs1.CCF C1(CC(=O)NC(CC)(C)CNC(c2cscc2F)=O)CC=CCN1C CC1CCC(NC(=O)CNC(=O)C(F)(F)F)CN1C(c1ccnc(CO)c1)=O C1(C(=O)NCc2n(CC)cnc2)CCCCC1NC(c1csc(F)c1)=O C1(CNC(c2c(COC)noc2)=O)CC2CC(C1)N(C(=O)CN1CCCCC1)C2 c1(C(=O)NCCN(CCCN(C)C)C(C2SCCCS2)=O)cnn2c1N(C)CC2 C(=O)(C(C)N(C(C1CN(c2ncco2)C1)=O)C1CC1)NCC.OCC N1(C(C2COC(=O)O2)=O)CCC2(CC1)CC(NC(C1(C(F)F)CCC1)=O)CCO2 C1(CC(=O)NCC2(F)CN(C(C(OC)OC)=O)C2)NC(=O)NC1=O C=CCCC(CC(C)C)C(=O)NCC1(NC(=O)CC(C)CC(C)C)CCC1 n1(CC(=O)NC(c2oc(C)nc2C)=O)cc(Cc2ccc(C)o2)c2ccccc12 N1(C(C2C(COC)C2)=O)CC2CC1CN(C(c1cc3occc3n1C)=O)C2 C1(NC(CC2(C(=C)F)CCC2)=O)CC2(CCN(C(c3cccc(N)n3)=O)C2)C1 C(=O)(C#CC12CC3CC(CC(C3)C1)C2)NC(C)CNC12CCC(C#N)(CC1)CC2 C1(NC(CC=CC)=O)CN(C(c2cc(C(C)C)n(C)n2)=O)C2CC12 CC1(C)NC(=O)CC1C(=O)NC(C)(C(=O)NCc1ccc(Cl)nc1)C1CC1 c1(NCc2c(OCC)cccc2)nc(C)ncc1C(C)C CCCC(CC)CC(=O)N1CCCC(CNC(c2ncc(C(N)=O)cc2Cl)=O)C1 Cc1cn2nc(N3CC=C(CNC(=O)CCc4nnc(C)n4C)CC3)sc2n1 C1(NC(c2c(OC)ccs2)=O)CN(C(c2cc(O)nc(Cl)c2)=O)C2(CCOC2)C1 CCCC(CC)CCC(=O)NC1CCN(C(=O)CCSCC(N)=O)C1C CN1CC(NC(=O)CCCCCNC(=O)CC(=O)NC2CC2)CC1(C)C C1(C(=O)NCC(C)O)CC2(CCN(C(=O)Nc3ccc(C(=O)O)cc3)C2)C1 c1(C(=O)NCC(CC)(CC)NC(=O)Cc2cncs2)nccc2n[nH]cc12 C(c1cn(C)cn1)=CC(=O)N(C)CCNC(C1(O)CCSC1)=O N1(C(C(C(C)C)C(C)C)=O)CCC(C2(NC(=O)CCc3ccoc3)CCC2)CC1 C=C(Cl)CC(C(=O)NC)NC(=O)C(C(C)(C)C)NC(=O)CCC(C)(C)F NS(=O)(=O)c1cc(C(N2CC(C3(NC(=O)Cc4ccco4)CC3)C2)=O)c(Cl)o1 N1(C(C(C)CC2CCCO2)=O)CCS(=O)(=O)C(CO)C1 CC(C(=O)NC1CC2(C1)CC(NC(C1OCCN(C)C1=O)=O)C2)C(C)(C)C c1(C(N(CC(C)(C)NC(Cc2ccc(C)c(Cl)c2)=O)C)=O)cc(Cl)cc(F)c1F Cc1cc(C(N2CCCC(C(N3CCC=CC3CN(C)C)=O)C2)=O)nnc1C C(CC(=O)N(CC(O)CN(C)C(c1sc(COC)nc1C)=O)C)(C(C)C)OCC C1(NC(c2ccc(N(C(C)=O)C)cc2)=O)CN(C(=O)C#CC2CC2)CCC1CO N1(C(c2ccc(OC)cc2F)=O)CCC2(CC1)CN(C(=O)CC1CCSCC1)C2 C1(NC(c2cc(CCC)[nH]n2)=O)CC(O)CN(C(C2(CC)COC2)=O)C1 c1(CNC(c2c(COC)noc2)c2nnnn2C2CC2)csc(Cl)c1Cl C(=O)(CCCCCCC(=O)NCCc1ccccc1[N+](=O)[O-])OC CCC(C)C(O)C(=O)NCC1(C)CCN(C(c2ccc(=O)n(CCO)c2)=O)C1 c1(NC(C2N(C(c3cn(CCC)nc3)=O)CCC2C)=O)ccc(O)c(=O)cc1 N(C1CCCc2ncccc21)C(=O)N(CCS(=O)CC(F)(F)F)CCO C1(O)(CNC(C(C)OCCOCC)=O)CCCN(C(=O)Cc2cnsc2)CC1 c1(CCNC(CSCC(CCCC)CCC)=O)ccc2c(c1)OC1(CCCC1)O2 C1(C(N2CCC(N(C(=O)CO)C)C2)=O)CCc2c(ncn2C)C1 S(=O)(=O)(c1ccc(C)cc1)N1CCCC(C(=O)Nc2c(CC)noc2C)C1 C1(N2CCCC(C)(O)CC2)CC2(CCN(C(=O)C=CC(=O)NC3CC3)CC2)C1 N(C1CC(C)(C)Oc2cc(F)ccc21)CC(=O)N(CC(=O)OC)C Cc1cc(C(=O)N(C)CCNC(C2CC2(C)Br)=O)cnc1C(F)F c1(C(=O)OC)ccc(SCCCC(=O)Nc2nnc(C(C)C)s2)cc1 CS(=O)(=O)C1CN(CC=Cc2ccncc2)CC1n1cc(C2(CCO)CC2)nn1 C(=O)(CCCC(C)(F)F)N(C)CC1(O)CN(C(C2CC(C)OC(C)C2)=O)C1 N1(C(C(CC=C)CC)=O)CCOCC(C)(CNC(=O)CCc2cc(Cl)cs2)C1 N1(C(c2c(C)nc(C3CC3)nc2)=O)CC2CCCC1C2CNC(C1CCCO1)=O c1(C(=O)NCC2CCN(C(c3ccco3)=O)CC2)cccc2c1CCO2 CCCC(C)(C)CC(=O)N1CC2CC2(C(=O)NC2(CC3CC3)CCC2)C1 c1(CC(=O)NC(C)(CNC(C2(O)CC2)=O)C2CC2)ccc(Br)s1 C(CCC(C)C(=O)NC1CCC(CNC(c2occc2C(C)C)=O)CC1)OC Cc1cc(C)c(CC(=O)NC2CCN(C(c3cn(C)c(O)n3)=O)CC2)s1 Cc1cncc(NC(C2CCN(C(c3ccc(OCCF)cn3)=O)C2)C)n1 C(C)(CN=c1[nH]c(C)cc(=NCc2nc(C)ccc2Cl)[nH]1)OC N1(C(CC2(COC)CC2)=O)CCC2(CCCCN(C(C3CC3C3CC3)=O)C2)C1 C1(COC)CN(C(C2CCS2(=O)=O)=O)CCN1C(=O)CC1(C)CC1 N1(C(c2csc(-c3ccccc3)n2)=O)CCN(Cc2ccc(O)c(F)c2)C2CC12 c1(C(N(CC(=O)NC(Cc2scc(C)n2)C)C2CCC2)=O)ccc(O)cn1 C1(CN(C(C(C)OC)=O)C)CC(F)CN1C(=O)C(C)Cc1cnco1 c1(C(N(C(C)CNC(=O)CN2CCCOC2=O)C)=O)ncc(P(C)(C)=O)cn1 c1(C(N(C2CCN(C(c3cccn3C)=O)CC2)CCC)=O)cc(OC)ncc1F N1(C(C2OCC(C)(C)C2)=O)CC2(CNC(c3ccc[n+]([O-])c3)=O)CCC1CC2 C1(N(C2(c3cn(C4CCC4)nn3)CCN(C)C2)C2CN(C)C2)CCN(CCO)CC1 N1(C(CCCOCCC)=O)CCOC(C(C)NC(=O)Cc2ccc(OC)cn2)C1 C(C)(C)(CCCC(=O)NCC1CCCC(OC)C1)NC(C(C)=CCC)=O c1(C(N2CC(CNc3nc(C)nc(Cl)c3)OCCC2)=O)cc2c([nH]1)CCCC2 CC1(C)CCOC1CCC(N1CCC(NC(=O)Cn2ccnn2)C1)=O N1(C(CC(CNC(C=CC=CC)=O)(C)C)=O)CC2(CC(CO)CO2)C1 c1(C(=O)NCC(=C)CCNC(=O)C=CC(=O)NCC2CCCC2)ccc(F)cc1 c1(C(=O)NCC2(F)CCN(C(COC(C)C)=O)CC2)cccc(C#CC2CC2)c1 Cc1cn2c(C(N3CC=CC3CNC(=O)COCC(C)C)=O)cnc2s1 C1(NC(C=CC(CC)C)=O)CN(C(c2ncccc2O)=O)CC2(CC2)C1 N1(C(CC(=C)Br)=O)CC(CNC(C2(CCCC)CCCC2)=O)C(O)C1 C1(C(C)C)CCOCCN1C(C1CC2CCC1CC2)C(=O)NC1COC1 c1(C(C)C)ncc2c(n1)CCN(N1CCN(CCNC(C3CCCO3)=O)CC1)C2 Cc1cc(F)ccc1NC(=O)CC1CC(O)CN1C(=O)C(c1ccn(C)c1)C CCCC(C(=O)NCC1CC1CO)NC(=O)C(Cl)Cl C1(NC(C2CCC(C)N(C(=O)OCc3ccccc3)C2)=O)CCC2(CC1)CC2(F)F S(=O)(=O)(c1cn(C)c(=O)n(C)c1=O)N(Cc1ccc(SC)o1)CCO C1(C(=O)NC(C(C)(C)C)CO)C(C2CC2)CCN1C(=O)Cc1ncccc1F C(c1c(Cl)nc2sccn12)=CC(=O)N(C1CN(C(=O)CC2(O)CCOC2)C1)C C(CC(O)CNC(=O)C(C)OC(C)=O)NC(C=C(COC)C)=O C(=O)(C(C)(C)CC(F)F)NC1CC(CCNC(C(C(C)C)c2cnc(C)s2)=O)C1 C1(CNC(C(C=C)OC)=O)CCN(C(c2ccccc2)=O)C1(C)C c1(C(N(CCCNC(C=C2CCC(C)CC2)=O)C(C)C)=O)ccccc1C#N C1(SCC)CCCN(C(=O)CC2CCN(C(=O)Cc3sccc3C)C2)C1 Cc1nn(C)c(C(=O)NCC2(NC(=O)C(C)(C)n3cnnn3)CC2)c1[N+](=O)[O-] C1(C(=O)NCC2CC(C)C2)CC2CN(C(=O)C(F)(F)C3CC3)CC2C1 C1(CC(C)NC(=O)C(O)C(F)F)CCN(C(c2ccc(F)s2)=O)CC1 N1(C(C(CC)COC)=O)CC2(CC2)CC1CNC(=O)Cc1ccccc1C(N)=O N1(C(C(C)=O)=O)CC2(C1)C(NC(c1nc(C)c(C)nc1O)=O)CCS2(=O)=O C(C)(C(=O)OC(C)(C)C)(C(=O)N1C(C)CN(C(=O)C=CC(C)C)CC1C)OC C1(NC(c2cc(COC)c(F)cc2)=O)CC2CN(c3ncc(OC)cn3)CC2C1 Cc1cc(CC(=O)NCc2ccc(C(=O)NCC3(CC(C)C)CCC3)o2)no1 C1(NC(CCC2(CCC#C)N=N2)=O)CC2CCCC(C1)N2C(C1(Cl)CC1(F)F)=O N1(C(CCC(CC)NC(c2nnsc2C)=O)=O)CCC(O)C(F)(F)C1 c1(C(=O)NC2CN(C(C=CC=CCC)=O)CC(O)C2)cc2nccnc2cc1F N(C1CCCc2c1cnn2C(C)(C)C)CC(=O)NC(C)CCO CC1CN(C(C2CCC=CCC2)=O)CC1CC(=O)NC1CCC1(C)C C#Cc1cccc(CNC2CCN(CC(N3CCCCCC3)=O)CC2)c1 C(C(C(=O)NCCc1nncn1C)NC(=O)CC1CC=CCC1)N(C)C C(CC(C(C)C)N(C)C)NC(C(c1ccnn1C)N(C(C=CC(=O)OC)=O)C)=O C=CC(F)(F)C(=O)NC1CC(C)N(C(c2cccnc2NC)=O)C1 c1(C(=O)NCC2CC3(CN(C(CC(CC)OC)=O)C3)C2)n[nH]c2ccc(Cl)cc12 c1(C(N2C(C)C3CC2C3NC(=O)CCCNC(N)=O)=O)c(F)ccc(N)c1F CC1(C)C2CCC(C2)C1C(=O)NCCC1CCCN1C(=O)COC1CCCC1 CN1CC(NC(=O)CC2(NC(=O)CC3CC4CCC3O4)CCC2)CC12CCC2 C1(C(N2CC(F)(CNC(C(COC)C)=O)C2)=O)CNC(=O)N1C c1(CNC(C(C=CC)O)=O)ccc2c(c1)CN(C(c1ccc(F)c(F)c1C)=O)C2 CCCC(C)(O)CC(=O)NC(CC(=O)N(C1(c2cc[nH]n2)CC1)C)C(C)OC C(=O)(C(COC)CC(C)C)NCCC1(C(N2CCC(O)(CC)C2)=O)CCC1 N1(C(c2cccc(Br)c2)C(=O)N(C(CC)(C)C)CCC#N)CC2CCC(C1)C2(F)F c1(OCC)cc(C(N2C(CO)CC2C)=O)[nH]n1.C(Cc1cn[nH]c1)(C(=O)NC)N C(CC1=CCN(C)CC1)NC(C(CCCNC(c1c(C)noc1C)=O)O)=O N1(C(Cc2cc(C)on2)=O)CCC2(NC(=O)OC(C)(C)C)CCCCC12 N1(C(c2cc(CCC)ncc2)=O)CCCC(C)(C(N2CCOC(CO)C2)=O)C1 CCC(CC(F)F)C(=O)N1CC(F)(CNC(c2ccc(=O)n(C)c2)=O)C1 N1(C(C(N2CCCC(O)C2)C)=O)CCCC1(C)CNC(c1ccoc1Cl)=O C1(C(=O)NCc2n(CC)ccn2)CCC2CCC1N2C(=O)CC1CNC(=O)O1 c1(-c2nc(CCC)nn2CCCN2CCOCC2)ccnc(Cl)c1Cl C1(C(=O)NC)C=CCN1C(c1conc1CNC(C1CC1OC(C)(C)C)=O)=O C1(=CC(=O)NCC2N(C(C)=O)CCOC2)CCOc2ccccc21 c1(CN(C)CC2CNC(C)(C)C2)cccc(OCC(F)(F)F)n1 C1(C(=O)NCCC2CCSC2)CCCN(C(C2(Cl)CC2(F)F)=O)CC1 c1(C(=O)NCCN(C(c2c(C)[nH][nH]c2=N)=O)C)cc2cccc(F)c2o1 CC1(C)OCc2cc(C(=O)OCc3cnn(-c4ccccc4)c3N)ccc21 c1(C2(C(=O)NCC3CCC(NC(c4c(C)nc[nH]4)=O)C3)CCC2)ccccc1Cl c1(C(N2C(CC)C(NC(=O)CC3CCCCC3)CC2)=O)ccc2c[nH]nc2c1 O=C(C1CCSc2ccccc21)NC1C2CC1N(C(C1CC3CC3C1)=O)C2 C(=O)(C(C)(COC)CC)NCCCN(C(c1c(CC)occ1)=O)C C(=O)(CC(C)CC(C)C)NCCCC1N(C(CCc2c(C)n[nH]c2C)=O)CCC1 N1(C(C2OCC(C)C2)=O)C2CCC1CC(n1cc(C3(N(C)C)COC3)nn1)C2 c1(CC)cnn2ccc(C(=O)NCCC(C)NC(c3cc(C)[nH]n3)=O)nc12 C12(C(=O)NCC3N(C(c4n(CC)nnc4)=O)CCOC3)CC1COC21CCC1 c1(C(N2C(C)CCC2C(N2CCC(C(=O)N(C)C)C2)=O)=O)ccnc2ncccc12 C1(CC)C(NC(c2ccn(-c3cccc(F)c3)n2)=O)CCN1C(=O)CC(O)CC Cc1ncccc1-c1cn(CC2CCCC2NC(C2CS(=O)C2)=O)nn1 c1(CC(=O)N(C2CCCN(C(=O)Cc3cccs3)C2)CC)cc(F)c(F)cc1F C1(CNC(CC=CC)=O)OCC2CCC1C2.C12C(C1(C)C)NC2=O CCC(C(=O)NCC1CC(F)(CNC(=O)Cn2nnc(=N)[nH]2)C1)C(F)(F)F c1(C(=O)NC(C2CCCCN2C(C2CN(C3CCC3)C2)=O)C)c[nH]nc1[N+](=O)[O-] c1(OC)cccc(C(C(=O)NCc2ccc(F)cc2)N(C2(C)CC(C)(C)C2)C)c1 c1(CC(=O)NC(C)CN(C)C(C2(C#N)CCC2)=O)nn(C)c2ccccc12 C12(CNC(C(CC)CC)=O)CC(NC(c3cscn3)=O)C(CO1)C2 c1(CN2CCC(C)(C(=O)NCC(F)F)C2)cc(F)c(Cl)c(Cl)c1 C1(NC(c2n(C)ncc2)=O)CCN(C(=O)CC2CCCC(=O)N2)C1(C)C C1(NC(C2N(CC)CC2)=O)CC(F)(CNC(=O)C(c2ccccn2)OC)C1 C=CCC(CC(=O)NCc1cncc(OC)c1)NC(C1(C)CNC(=O)N1)=O c1(C(=O)NC23CCC(C(=O)Nc4nnc(Br)s4)(CC2)C3)cc(F)cnc1Cl c1(CC(=O)NC(CNC(CCC(=C)Br)=O)C(C)(C)C)ccc(O)c(Cl)c1 C1(C(=O)NCc2n(C)ncn2)CC2(CC2)CN1C(=O)C(F)F C12(C(CNC(=O)Cc3nc[nH]n3)NC(=O)C=Cc3cccnc3)CCC(CC1)C2 c1(C(N2CC(C)C(NC(c3cnc(N)c(Cl)c3)=O)C2)=O)cccc2c1CNC2=O N1(C(c2c(C)con2)=O)CCC2(CCCC2NC(C2(F)CCCCC2)=O)C1 O=S(=O)(c1ccnn1C1CC1(F)F)Nc1cnn(-c2ccccc2)c1 CC(O)C(C)C(=O)NCC1CCN(C(=O)CSC(=N)N)C1 C(=O)(C1=Cc2ccccc2C1)N(CCCNC(=O)C(O)C1CCCC1)C C1(c2n(C)nnn2)(NCC2(CO)CC2)CC2CCC1CC21OCCO1 c1(-n2cc(-c3cn(C)nc3)nn2)cncc(C(=O)Nc2cccc(Br)n2)c1 C1(C(N(CCNC(C2(C)CC=CC2)=O)CC)=O)CC(O)CN1C(=O)OC(C)(C)C C(N=c1[nH]c(=NCCCN2CCC2)[nH]c2c1CSC2)c1nc(C(C)C)sc1 N1(C(C2C(C)=C2)=O)CC(NC(C2(C)CC=C(C)CC2)=O)CC12CCOCC2 C1(NC(Cc2cc(C)sc2)=O)CC2(CCN(C(=O)C3CC3)C2)C1 c1(C(=O)NC(C)CC(C)NC(c2ncoc2C(C)(C)C)=O)cnc(Cl)c(F)c1N CCC(C)CC(=O)C(=O)N1CC2CC(C1)N(C(=O)C=CCF)C2 CCCCCCCCCC(C)CC(=O)N1CC2CCC(C1)N2C(C1SCCS1)=O C1(=CCNC(C(COC)O)=O)CCN(C(C2CCCCS2)=O)CC1 C(C1c2ccsc2CCN1C(C1CCCCC1)=O)NC(CC1(C)CCC1)=O C1(C(=O)NC2CN(C(c3cnc(N(C)C)n3C)=O)C2)CC2CCCCN2C1 N1(C(CNC=O)=O)CC2CCC2(CC(=O)NC2(c3nn[nH]n3)CC2)C1 Cc1ccc2c(c1)CCC(C(=O)NCC1CCN1C(c1cnsc1C)=O)O2 N1(C(CC2(COC)CC2)=O)CC2(C)CC1(C(=O)NCc1ccc(C#N)s1)C2 c1(C(=O)NC2CCCCCN(C(CC(=O)N(C)C)=O)C2)cc(F)cc([N+](=O)[O-])c1 Cc1c(C(=O)N(C)CC2CCCN(C(=O)C(F)=CC3CC3)C2)ccc(F)c1F C1(C(C)(C)O)CCCN1N1C2CCC1CC(Oc1ccccc1)C2 C1(NC(c2cc(C)c(C(F)F)nc2)=O)CCCN(C(c2sccc2F)=O)CC1F c1(CCC(=O)N(CCC)CCNC(=O)Cc2cnco2)cc(C)cs1 CC1CCN(C(=O)C(C)(C)CN(C)C)CCN1C(C1CCCCC(C)(C)C1)=O Cc1nn(C)c(C)c1C(=O)C(=O)NCCNC(=O)CN1C(=O)CCC1=O N1(C(CSCC=C)=O)CC2(C1)CN(C(=O)C(=O)NCC(F)F)CC(C)(C)O2 CC1CN(C(=O)CCCN2CCOCC2)CC1CNC(c1cccnc1)=O N1(C(c2cccc(CCC)c2)=O)CCC(C)C(NC(=O)CN(C)C(C)=O)C1 N1(C(C2CC=CCN2C(c2cc(CO)on2)=O)=O)CCC(CO)C(O)C1 C(=O)(CC(O)(C(F)(F)F)c1ccccc1)Nc1ccc(OCC#N)nc1 Cc1ccc(F)c(CC(N2CCCC2CN(C)C(C2(O)CC3CCC2C3)=O)=O)c1 C(=O)(C1CCc2nccn21)NC(CCCNC(COCc1cc(C)on1)=O)C Cc1cc(NC(=O)C(O)C2CN(C(=O)CC3CCC(C)CC3)C2)cc(C#N)c1 C12(C(=O)NC(C(C)NC(C(CC)(C)OC)=O)CO)CC3CC(C1)CC(C)(C3)C2 c1(N2CCC(OCCOC)C2)nc(C)cc(=NC(C)CN2CCOCC2)[nH]1 N1(CC)CC(C(=O)N(CC(C)(C)CNC(c2csc(C)c2OC)=O)C)CC1=O C1(NC(=O)CCOC2CCC2)CC2(CCN(C(=O)CC3CCCCCO3)CC2)C1 N1(C(C(=O)NCC#C)C)CC2CCC1CN2C(c1c(Cl)c(C)nn1C)=O CC(C)CC(C)C(=O)N(C1CCN(C(c2coc(C3CCCC3)n2)=O)C1)C c1(CN2CCC(C(C)NC(=O)Cc3occc3C(=O)O)C2)cc2ccccc2o1 c1(C(N2CCC2Cc2c(-c3cn(CCC)nn3)n(C)nc2)=O)c(C)cccc1Cl c1(N(C)C(=O)OC(C)(C)C)ccc2c(c1)CN(C(c1nc(Br)c(Br)cc1Br)=O)C2 c1(C(C(=O)N(C(CC)CNC(=O)OC)C)F)c(F)cccc1F C1(NC(c2c(CNC(=O)CN3CCOC3=O)ocn2)=O)CC2(CCC2)C1O C1(CC(=O)NCC(C)(C)C(N)=O)CCCN(C(=O)CCc2cn[nH]c2)CC1 c1(C(=O)NC(CC(C)NC(C2CN(C(=O)NC)C2)=O)C)cc(C)nc(Cl)c1N c1(C(=O)NCCNC(=O)Cc2ccc(F)cc2C(F)(F)F)cnc2n1CCCC2 CC(C)C(CO)C(=O)NCC1CCC(NC(=O)CC2CCC(C)(C)CC2)CC1 CN1CCCc2ccc(NC(=O)Nc3cc(S(=O)(=O)CF)ccc3F)cc2C1 Cc1ncc(C(=O)NCC2CCCC2NC(=O)Cn2cccnc2=O)n1C N1(C(c2occ(C)c2)=O)CCCC(OCCNC(=O)C(N)=O)C1 CC(C(=O)NC1(CNC(C2C(C)(C)C2(F)F)=O)CC1)S(=O)(=O)c1ccc(F)cc1 c1(CNC(CN(C2CC2)CC)=O)ccccc1CNC(C1C=C(C)CS1)=O N1(C(C2CCC(=C)CC2)=O)CCC2C(CCCN2C(C2CCC(O)CN2C)=O)C1 Cc1ccc(CCNC(C2CCC(C)N2C(=O)C2=NOCC2)=O)cn1 CC1(C)CCCCC1C(N1CCC(C(O)CNC(C2CCC3(CC3)C2)=O)CC1)=O c1(C(=O)NC2C(OC)CN(C(C(CC)F)=O)C2)cc2n(n1)CCNC2=O O=C1NC2(CO1)CC(C(=O)NCC1CCN1C(=O)C1=COCCC1)C2 C1(C2CCCCN2C(C2(F)CC2)=O)(CNC(C23CC(F)(C2)C3)=O)CCOCC1 C1(C)(C(=O)NCC2C(NC(CCOCC(C)C)=O)C2)CC2(C1)CC(F)(F)C2 C1(C(N2C(C)(C)C(NC(=O)Cn3ccccc3=O)CC2)=O)Cc2nccnc2C1 C1(C)(C(=O)NC2CC(CCNC(c3c(C)cn(C)n3)=O)C2)CCOC12CC2(F)F Cc1onc(C(=O)N(C)CCNC(C2CC2CF)=O)c1Br N1(C(C2(CC)CCCC2O)=O)CC2(C1)CN(C(c1[nH]c(C)cc1C)=O)CCO2 C(=O)(CC(C(F)(F)F)NC(=O)C(CC)CCC)NC(C=C)C(F)(F)F C1(CNC(C(CC)C2CCOCC2)=O)CN(C(=O)CNC(=O)C2CC2)CCO1 c1(C(NC(NC(C=C)C)=NCCN2CC2)C)cc2cc(Br)ccc2[nH]1 N1(C(CN(C(C)C)C)=O)CCC(NC(C2CC2(C)C(F)F)=O)C1C(C)(C)C C1(COC)(NC(C(C)C(C)C)c2nnnn2Cc2ccco2)CCCCC1 C(CC(C)(C)C(=O)N1CCC(N(C)C)C1)NC(C(C)OCCC=C)=O CCCC(C)(C)C(=O)N1CCN(C(=O)CCCSC)C(c2cccc(F)c2)C1 C1(CC(=O)NCC#CCC)CC(NC(c2nc(C)oc2C)=O)C1(C)C C1(NC(c2cn(CC(=O)OCC)nn2)=O)C2CCCN(C(C3CCOCC3)=O)C12 N1(C(CCOCC)=O)CC2CC(C(=O)NCC3CC3(C)CC)CC2C1 N1(C(c2ccn(C(C)C)n2)C(=O)NCC2CCCO2)CC(C)CC1C c1(CNC(N(C(C)CC(N)=O)C)=O)ccccc1OC1CCC1 C(C(C)(CC)C(=O)Nc1cnc(C)c(Cl)c1)NC(C1C(CC)CCO1)=O N1(C(C(CC=C)C)=O)CCOC2(C1)CN(Cc1ccc(OC)c(C(F)(F)F)c1)C2 C1(CC)CCCCC1CNC(=O)CSc1ccccc1.c12ncc(s1)c(=O)[nH]2 c1(C(=O)NC(C(=O)NCC(CC)SC)C2CCCO2)ncncc1OC N1(C(C(COCC)C)=O)CCC(NC(=O)CCC2CCC2)CC(O)C1 c1(CC)ccc(C(C)CC(=O)N2CCC(CNC(=O)C=CCF)C2)cc1 CC(C)C(C(=O)N1CCC(C(=O)N(C2(CO)CC2)C)C1C)C1CCC1 c1(C(=O)NCCCC2N(C(c3cc(C)no3)=O)CCC2)c[nH]c2cccnc12 c1(OCCC(=O)NC(C)C(C)NC(=O)C=Cc2cn[nH]c2)cc(Cl)cc(Cl)c1 c1(CNC(C2CN(Cc3c(Br)cccc3Br)CCO2)=O)ccc2ccccc2n1 C1(C(=O)NCC2CCCC(CNC(C3(C(N)=O)CC3)=O)C2)CC2(C1)CC21CC1 c1(CCC(=O)NCC(c2c(C)nn(C)c2)N2CCCC2)ccc(F)c(F)c1 C1(C(=O)NCCN(CCC)C(C2([NH+]([O-])NC)CCCC2)=O)CCn2cc(C)nc2C1 C1(NC(c2ccc(Cl)c(F)c2)C(=O)O)COC2(CCCNC2)C1 C1(COC)(CNC(C2CCOC(C)(C)C2)=O)CCN(C(=O)Cc2ccco2)CC1 c1(C(N2CCN(C(CC3CC(C(=O)OC)C3)=O)C3C2C3)=O)cccc2nccn12 c1(CNC(CC(C(=C)C)O)=O)nc2ccccc2[nH]1.c12cccc(c1)CNC2=O c1(OC)c(C(c2ccccc2)NC(=O)N(C2COC2)C(C)C)cccc1Cl C(=O)(C1CCOc2ccc(Cl)cc21)N1C(CNC(c2cnn(C)c2N)=O)CC1 N1(C(C2C(C(=O)OC)CC2)=O)CCC(C(C)(C)NC(=O)Cc2ccn(C)n2)C1 C=CC(F)(F)C(=O)N1CCOC(CCNC(c2cn(C(F)F)cn2)=O)C1 N1(C(CN(C)CC)=O)CCCN(C(=O)CSc2cn[nH]c2)C(C)C1 Cc1conc1CC(=O)NCC1CC(CNC(=O)CNC(=O)C(F)(F)F)CO1 C1(NC(c2cc(OC)nn2C)=O)CC2CN(C(c3c[nH]nc3OC)=O)CC2C1 CC1(C)C(CNC(=O)CCC2CC(NC(=O)CN3CCC(F)CC3)C2)C1(F)F C1(O)(C(=O)NCC2(NC(c3cn(CCCC)nn3)=O)CC2)CCC(CC)C1 C1(NC(c2c(CNC(C3N(CC)CCC3)=O)nnn2C)=O)CC(F)(F)C1(C)C C1(NC(c2c(C)[nH]cc2)=O)CCCCCC1NC(c1cc(O)cc(Br)c1)=O C1(C)(NC(C2C(C(C)NC(=O)C(C)c3cc[nH]n3)C2)=O)CCC(O)CC1 C1(NC(c2ccc(F)nc2)=O)C2CCC1CN(C(C1CCCC(CF)C1)=O)C2 C1(CC(=O)NC2(CC)CC2)CCN(C(=O)CNC(=O)NC)C1 CCC(C)(C)CC(=O)NCC1COCCN(C(c2cc(C(F)F)ccc2Cl)=O)C1 Cc1cc(CC(=O)NCCOCC(=O)N(CC(C)O)CCO)cs1 N1(C(=O)CC(F)(F)F)CCC2C(C1)CN2C(c1cnn(CC(F)F)n1)=O C(=O)(C1CCc2cccc(F)c21)N(C(C)CNC(c1cc(Br)n(C)c1)=O)C c1(OC)cc(C(N2CCC(NC(=O)Cc3cnsc3)C2)=O)ccc1C#N C1(N(C(c2n(CCC)ncc2)=O)C)CN(C(=O)C(C)NS(C)(=O)=O)CC12CC2 O=C(C1Cc2ccc(Cl)cc21)NCC12CC1CN(C(=O)CCC(F)F)C2 c1(OC)cccc2ccc(C(=O)NCC3(F)CC(NC(C)=O)C3)nc12 C1(CCNC(=O)CCC23CC(C2)C3)CCCCN1C(=O)CN1CCCCCC1 N1(C(C(C)C(F)(F)Cl)=O)CC2CCCC(N(C)C(c3cnc(O)c(F)c3)=O)C2C1 C#CCC(C(=O)N1CCCCC1CF)NC(c1oc(C)nc1CC)=O C1(CNCC(C)O)CCCN1C(=O)CCCC1CC1 C1(NC(C=CC(C)C)=O)CN(C(=O)C(=O)NCC(F)F)C(C)(C)C1 c1(SC)nc(C)c(CCC(N2CCC(C(=O)N(c3ccccc3)C)C2)=O)c(O)n1 c1(OCC(C)C)cccc(C(=O)N(C(C)CN(C(=O)C=C(Cl)Cl)C)C)c1 C(C(C)C)(C(O)C(=O)NCCC1(NC(C2CC2(C)C(F)F)=O)CCC1)OC C12(NC(C=C(C)C)=O)CCC(CC1)N(C(=O)CSc1n[nH]c(=N)s1)C2 C1(NC(c2nc(C)oc2)=O)CN(C(=O)CNC(c2ccc(O)cc2)=O)CC2(CC2)C1 C1(C(N(C(c2c(C)ccc(C)c2)C)C)=O)CC2(CCCC2)CO1 CCC(C)CCCCC(=O)N(CCCCCC(=O)NC1(C)CC(F)C1)C N1(C(C2CN(C(=O)NC)C2)=O)CC(C(=O)N(C2(C)CC2)C)C(C2CC2)C1 C#CCC(C)(C(=O)N=c1cc(C)n(C)[nH]1)NC(=O)CC(O)CC(C)C c1(CN(C)C)ccoc1C(=O)NCC1CCN(C(C2CCC(C(N)=O)C2)=O)C1 C(=O)(CCCCCC(C)O)N(C1CCN(C(c2c(CC)c(C)sc2)=O)C1)CCO N1(C(c2cncc(N)n2)=O)CCN(C(C2CC(F)(CO)C2)=O)C2CCC12 C1(NC(C2CN(CC)C(=O)C2)=O)CC2CN(c3nc(C(C)(C)C)ns3)CC2C1 CC1C(NC(c2cccc(F)n2)=O)CCN1C(=O)Cc1ccccc1Cl CCC(C)(CC)C(=O)NCC1(F)CCC(CNC(c2ccc(C)cc2SC)=O)C1 CC1CC(CNC(c2cnc(N)c(Cl)c2)=O)CCN1C(=O)Cc1cncc(F)c1 C1(C(=O)N(CCCCCO)C)(CC)CCCN(C(=O)C2=C(C)CCC2)C1 C1(NC(CCSCC(N)=O)=O)CCOCC1NC(=O)C(O)C(F)F Cc1cc(CN=c2cc(NCCCC#N)nc[nH]2)nc(Cl)c1Br c1(C(=O)NC2(CC(=O)NCCn3c(CC)nnc3)CCC2)ccc(C#N)[nH]1 C(=O)(N1OC2CCC1CC2)C12N(C(CC)=O)CC(C1)C2 c1(-n2cc(CN(C(C)(C)CO)CC)nn2)c(C(C)C)cccc1C c1(C(=O)NCCCCNC(c2cn(CCC=C)nn2)=O)[nH]c2c(c1C)CCCC2 N1(C(C(CC)NC(C)=O)=O)CC2CCC(NC(c3ccc(C)nc3SC)=O)C2C1 C1(C)(CNC(CC2C(CNC(C3(OCC)CCOC3)=O)C2)=O)NC(=O)NC1=O N#Cc1ccc(CSCC(=O)NC2CC2NC(C2(C3CCC3)CCC2)=O)cc1 C(C)(CNC(c1ccc(O)c(N)n1)=O)(CC(C)C)NC(c1c(C)n[nH]c1C)=O N1(C(C2(CC)CC2)=O)CCC(O)(CNC(=O)C(c2ccc(Cl)s2)C)CC1 C1(CC=C)(NC(c2cc(CN(C)C)c[nH]2)=O)CN(C(c2conc2CC)=O)C1 N(C1COc2ccccc21)C(CC(C(F)(F)F)NC(Cc1c(C)nccc1)=O)=O c1(C(C(N2CCC(N(C(Cc3ccn(CC)n3)=O)C)C2)=O)(C)C)cccc(F)c1 c1(CS(Cc2nnc(C(C)(C)C)o2)(=O)=O)cccc(Cl)c1 O=C1NC2(C(=O)NC3CC(NC(C4CCCC5(CCC5)O4)=O)C3)CC3CC1C2C3 CCC(C)C(C(=O)NCC1CC(O)CN1C(c1csc(C)c1)=O)NC(C)=O c1(NC(c2c(NC(C3C(C(=O)OC)C3)=O)cc(C)cc2)=O)c(C)ccnc1C#N c1(C(=O)NCC(c2ccccc2)NC(C(C)(CO)OC)=O)ccc([N+](=O)[O-])[nH]1 c1(C(N(CCCNC(CSCC)=O)C)=O)nc(N(C)C)nc(=N)[nH]1 c1(N(C)Cc2ncn(C)n2)ccc(S(=O)(=O)NCC2CCCC(CO)C2)cn1 C(=O)(C(CC)C(=O)N1CCCC1C1(O)CN(C(c2cnc[nH]2)=O)C1)OCC c1(C(N2C(CNC(c3cc(CC)no3)=O)CC2)=O)cn(C(C)C)nc1C(F)(F)F c1(C(=O)NCCN(C(C)C(=O)NC)CCOC)cccc2ccncc12 C(=O)(C(Cc1cscn1)NC(C1CC(CCC(=O)O)CO1)=O)OC(C)(C)C CCCCCC(=O)NC1CCC1NC(=O)COC(=O)NCC(=O)NCC N1(C(C(C2CC2)OCC)=O)CCC(C(N2CC(C#N)C2)=O)C1CC N1(C(CNC(=O)OC)=O)CCC2CN(C(C34CSCC3C4)=O)C2C1 N1(C(c2c(C)nc[nH]2)=O)CCN(C(=O)C(C)N(CC(F)(F)F)C)C(COC)C1 N1(C(C(=O)NC)=O)CC2(C1)CN(C(=O)C(=O)C1CCCC1)CC2CO CC(C)CC(O)C(=O)N1CCC2CC12C(N1CC2(CC=CC2)C1)=O C1(CC(N2CC(O)(CNC(C3C=CC=CC=C3)=O)C2)=O)CCCC(F)(F)C1 c1(C(=O)NCCCN(C(c2c(C)nc(C3CC3)o2)=O)C)coc2ccc(Cl)cc12 N1(C(C(C)OCOC)=O)CC(NC(=O)NCc2cnn[nH]2)C(c2ccccc2)C1 C1(NC(CS(N)(=O)=O)=O)COCCN(C(c2cccs2)=O)C1 c1(C(=O)NCC2C=CC(NC(c3c(C)nco3)=O)C2)ccc(F)c2[nH]ccc12 C1(C(=O)NC2CCN(C(C3(N(C)C)CCCC3)=O)C2)CCOCC12CCCCC2 c1cc(Cl)nnc1O.Cc1ccccc1NC(=S)N CCN=C(NCC1CCCN1S(=O)(=O)CC)NCC1CC2(C1)CC2F CCC(CC(=O)OC)NC(=O)C(O)CCNC(=O)COc1cccnc1 N1(CC)CC(C(=O)NCC2C(C)CCN2C(c2n[nH]c(C)n2)=O)CC1=O c1(CNC(C2CCN(C(C(C)(C)N(C)C)=O)C2)=O)ccc(OCC(F)(F)F)cc1 Cc1ccc(Br)c(C(=O)NCC2COCCN2C(C2CC2(C)C)=O)c1F c1(NC(C(CC)OC(=O)CC2COC2)=O)ccc(F)cc1F c1(C(N2CCNC(=O)C23CCC3)C(=O)NC(CC)C)ccc([N+](=O)[O-])c(Cl)c1 c1(C(N(CC(CNC(c2c(COC)cco2)=O)C)C)=O)c(O)cccc1Cl C1(NC(C(C)Cc2ccc(Cl)cc2)=O)COCCN(C(=O)CCOCC(F)F)C1 N1(C(c2ccc(OC(F)F)nc2)C(=O)NC(CC)(C)C)CCC2OC(=O)OC2C1 c1(SCC(N2CC(C)C(NC(=O)COC3CC3)C2)=O)nc2ccccc2s1 c1(CC(=O)NCCN(C2CCCC2)C(C2C(COC)C2)=O)ccc(O)c(Cl)c1 C1(NC(c2cc(C)ncn2)=O)CC2CN(C(c3csc(C(F)(F)F)c3)=O)CC12 C(CC(=O)N1CCC(C#N)(CC)CC1)(CC(C)C)NC(C(C)NC(CC)=O)=O C1(O)(CNC(CCC(N)=O)=O)CCN(C(c2ccsc2)=O)CC1 C1(C(N(C2CCN(C(c3coc(C)c3)=O)C2)CCC)=O)Oc2ccccc2C1C Cc1ncc(C(N2CCOC(C3CN(C(c4cnc(S)nc4)=O)C3)C2)=O)c(=N)[nH]1 [N-]=[N+]=NCCCCC(=O)NC(Cc1ccco1)C(=O)NCC(=O)NC1CCCC1 c1(CC(=O)NC2CCN(C(CSCC=C)=O)C2C(C)C)c(C)nn(C)c1C C1(NC(C2(OC)CCOC2)=O)CCCN(C(=O)Cc2cccc(Br)c2)C1 c1(OCC(=O)NCCC2CN(C(C3C(C)(COC)C3)=O)C2)c(C)occc1=O c1(OCC(n2cc(CCCNC(c3nc(NC)sc3)=O)nn2)C)ccc(C)cc1 C(CCC(=O)NC(C)C(C)NC(c1cnc(-c2cccs2)s1)=O)NC(=O)OCC C1(O)(CCNC(C2(C)CNC(=O)C2)=O)CCN(C(C2CCCCC2)=O)CC1 c1(Cn2cc(C3CCN(C(C(CN(C)C)O)=O)C3)nn2)ccc(N)cc1 C1(C(N(CCCF)CC)=O)CC(NC(=O)CCc2ncccn2)C(O)C1 c1(C(C(=O)NCCCN(C(c2cc(Br)n[nH]2)=O)CC)C)ccccc1Cl Oc1ncnc2ccc(-c3noc(-c4nc5ccccc5o4)n3)cc12 c1(C(N2CCC(n3cc(C(=O)NCC#CCCO)nn3)C2)=O)cnc(CO)cn1 N1(CC2N(C(=O)OC(C)(C)C)C(C)(C)SC2)CCC(C2CCNCC2)C1 C(=O)(CC(C)CC(=O)OC)NCc1cn(CC(N2CC(OCCCCC)C2)=O)nn1 c1(C(=O)NC(C)C(C)NC(c2n[nH]cc2[N+](=O)[O-])=O)cccc2ncn(C)c12 c1(NC(=O)CCNC(=O)Cc2ccsc2)c[nH]nc1Cl CCC(C)(C)C(O)C(=O)N1CC2CCC2(CCC(C(=O)NC(=O)OC)(C)C)C1 C(C)(C)(CC(F)C(=O)NCC(C)(C)CO)NC(C(CN(C)C)O)=O C#CC1(O)CCN(C(=O)C(C)(CO)NC(=O)C(F)C(C)CC)C1 C(=O)(C1=CCN(C(=O)CC2CC3CC3C2)CC1)NCC1(O)CCC(C)C1 N1(C(c2nn[nH]c2Cl)=O)CCC2CN(C(c3ccc(-c4ccon4)cc3)=O)C2C1 C(=O)(CC1=CCOCC1)NCCCC(C(=O)N(CC)CC1CC1)O c1(C(N2C(CN(C(=O)C(CO)C(C)(C)C)C)COCC2)=O)c(F)ccc(N)c1F c1(C(=O)NC2CCC(F)(CNC(C(CC=C)C)=O)C2)ncc(C)cc1Br C1(C(N(C(C(C)SC)C)C)=O)C(C2CC2)CCN1C(C1Cc2ccccc2C1)=O c1(C(N2CC(C(C)NC(C(C(=C)Cl)(C)C)=O)OCC2)=O)ccc2c(c1)CC(=O)N2 C1(C(N(C(CCNC(Cc2cccc(C)c2)=O)C)C)=O)CC1C1CCCC1 N1(C(COC(C)=O)=O)CCCC2(CCCCC2NC(c2nc(Cl)sc2C)=O)C1 C1(CCC(=O)NCCC2CC(NC(CN(C3CCC3)C)=O)C2)CCC(=O)N1 c1(NCCC(N2CCCCC2)=O)cc(=NCc2ncc[nH]c2=O)[nH]cn1 Cc1cc(NC(=O)C(C)N(C(=O)C(O)CC(C)C)C)cc(C)c1O CCCCC(O)CC(=O)N1CCC(C)(C(=O)NCCN(C(C)C)CC)CC1 N1(C(CC2N(CC)CCOC2)=O)C2CCCC1CN(C(C1CCS(=O)(=O)C1)=O)C2 c1(C(=O)NC2(C3N(C(c4c(COC)cco4)=O)CCC3)CC2)cnncc1C c1(C(C)N(C(CNC(C2CC(C(C)(C)C)C2)=O)C2CC2)C)nn[nH]n1 c1(C(C(=O)NC(C)(C)C)N(CC(CCC)C)C)ccc(F)c(C)c1 N1(CCNC(C(C)N(C(=O)C=Cc2ccc[nH]2)C2CC2)=O)CCCOC1=O C#CC1CCCN(C(=O)C(C2CC=CCC2)NC(C2CCC2C#N)=O)CC1 c1(NC(C2CCCC(O)C2)=O)cnc(CN(CCCN(CC)CC)CCO)c(Cl)c1 C1(CC)CN(C(=O)CCN(C(=O)Cc2cn(C)cn2)C)CCN1C C(=O)(CC(O)CC(C)(C)C)NC1(CC(N2C3CN(C(C)C)C(C3)C2)=O)CCC1 C1(CNC(CCCNC(=O)NCC#C)=O)CN(C(=O)CCCN=[N+]=[N-])CCC1C c1(OC)ccc(CN(CC(C)NC2CCC(C)CC2)C)c(OC)c1.C1(C)=CCC1 CC1CC(NC(c2cc(C#N)on2)=O)CCN1C(c1ccc(Br)o1)=O CC1(CO)CCC(N=c2[nH]c(=NCc3cncs3)[nH]c3c2SCC3)CC1 c1(C(N2C(CCNC(C(C(CC)O)C)=O)COCC2)=O)ccc(C#N)nc1O C(=O)(C(CC=C)C(C)C)NC(CCC=C)C(=O)N(C1CN(C(C)C)C1)C c1(C(=O)NC2C(NC(C(C)C#N)=O)CCC2)cc(C(F)(F)F)cc(O)n1 C1(NC(CC2CC(=O)C2)=O)CCN(C(c2csc(Cl)n2)=O)CC12CCC2 C(CNC(=O)Cc1csnn1)(CC(F)(F)F)NC(C(N1CC(C)C1)C)=O C1(CC(=O)NCCC2(C(=O)NC(CC)C3CC3)CCCC2)CCN(C)CC1 N1(C(=O)NC2C(F)(C(=O)OC)C2)CCN(C2CCSC2)CC1 C(CNC(C1CCC1C(F)F)=O)(CC(F)(F)F)NC(=O)COc1ccccn1 C12(C(N(C3CC(N4CCCC4)C3)CCOC)=O)CC(c3cccs3)(C1)C2(F)F c1(CC2(CC(=O)N(CC(C)(C)NC(COCC(=C)C)=O)C)CC2)ccccc1 N1(C(CC(C)F)=O)CCC2CN(C(c3csc(-c4cnc[nH]4)n3)=O)CC12 C1(NC(C2(COC)CC(F)(F)C2)=O)CN(C(c2cn(C)[nH]c2=N)=O)C2(CCC2)C1 N1(C(=O)CC2CCCN(C(c3ccc(O)cc3)=O)CC2)CCC2(CCCC2)C1 Cc1cc(CC(N2CCC(C(C)NC(C3CC(O)C3)=O)C2)=O)ccc1Cl C(=O)(C#CC1CCCCC1)NC(C(=O)Nc1cn(CC)c(=O)cc1)COC(C)C CC1CCOC(C(=O)NC(C2CCCN2C(=O)CCNC(=O)CO)C)C1 c1(C(N2CCC3(NC(c4nn(C)c(O)c4)=O)C(C2)C3)=O)ccc(Cl)c(N)c1Cl CCCC(O)C(CO)NC(=O)C=CC(C)NC(=O)CCN(C)C1CC1 c1(CC)ccc(C(=O)N(CC(C)NC(=O)Cc2nc(=N)[nH][nH]2)CC)cc1CC c1(C(=O)NC(CC)(C)CNC(c2ccc(O)nc2Cl)=O)cc(C)c(C)nc1C C(=O)(C1=CCCC1(C)C)N1CCN(C(c2c[nH]c(=NC)s2)=O)CC1CO C(CCCC(=O)N(C(CNC(=O)CC1CCCCC1O)CC)C)OCC CCN=c1ccc(C(N2CC(NC(c3cc(C)c[nH]3)=O)CC3(CC3)C2)=O)c[nH]1 C(c1ccc(S(N)(=O)=O)cc1)=CC(=O)N(C(C)CNC(C1C(C)C1C)=O)C CN1CCC2CC(NC(=O)CCc3cnc(C4CC4)o3)CCC12 Cc1cc(C(N2CC(O)(CCNC(=O)Cc3cnnn3C)C2)=O)c(C)cn1 c1(C(N2CC(OC)(CNC(C3CCSC(C)C3)=O)C2)=O)cc2ccccn2n1 C(=O)(C1CCc2nccn21)N1CC2(CC(NC(C3CN(CCC)C(=O)C3)=O)C2)C1 C1(C2CCN(C(=O)CC3CCC(=O)NC3=O)C2)(NC(c2c(C)coc2)=O)CC1 C12(C(N3CCC(NC(CNS(CC)(=O)=O)=O)C(F)C3)=O)CCOC1CCOC2 C1(N(C2(C(N(C)C)=O)CC2)C(C2CC=CCC2)=O)CCN(C(=O)C=CCF)O1 N1(C(c2c(C)cn(C)c2)=O)CC2CC(C(=O)Nc3ccc(F)nc3)C(C2)C1 C(=O)(C1CCCn2nccc21)NC1CC(C(C)NC(=O)CS(=O)(=O)N(C)C)C1 N1(C(C2C(C)CCO2)=O)CCCC2C(NC(=O)CCc3n[nH]c(=N)s3)C(C)(C)C12 c1(OC(C)C)c(C(=O)N(C)Cc2ccnc3[nH]ccc23)cc(Cl)cc1Cl c1(N(C(c2cncn2CC)C(=O)NCC2CCOC2)CCOC)ccccc1C N1(CC)CCCC(C(N2CCOC(CNC(c3cc(C)nn3C(F)F)=O)C2)=O)C1 CS(=O)CCC(=O)NC(C1CCCC1)CNC(c1scnc1C1CCCC1)=O c1(C(N(CC#C)C2CC2)=O)ccn(CCNC(=O)Cc2ccc[nH]2)c1 CCCCC(O)C(=O)N1CCCC1(C)C(=O)N(C)Cc1ncc(C)o1 C1(CC(=O)NC(CC)CN(C)C(c2ccoc2CC(N)=O)=O)C(=O)ON=C1C C1(N(C(C(C2CN(C(C(C=C)C)=O)C2)OC)=O)C)CCOC(C)C1 c1(C(C(=O)NCCC2(NC(C3CC4CC4C3)=O)CC2)CO)ccc(Cl)cc1 CC(C)S(=O)(=O)CC(=O)N1CCCC1CCNC(c1cc(C(F)(F)F)cs1)=O c1(SCC(=O)NCC2CCC(NC(C3(CC4CC4)CC3)=O)CC2)ccc(Cl)cc1 N1(C(C2(CCC)CC2)=O)CCC2(CCCN2C(C2(CCC)CCC2)=O)CC1 Cn1cc(S(C)(=O)=O)c(C(=O)NCCCNC(c2ccc(C3CC3)cn2)=O)n1 Cc1cn2c(C(=O)NCC(C)N(C)C(c3ccnc(S)c3)=O)c(Cl)nc2s1 C(=O)(C#CC1CCC2(CC1)OCCO2)N1CC(C)(NC(C(C)C(F)F)=O)C1 c1(N2CC(NC(C3(C(C)C)CCC3)=O)CC(F)(F)C2)ncnc2c(Br)c[nH]c12 C(=O)(C1Cc2ccc(F)cc21)N(CC(C)(C)NC(C1CCc2nncn2C1)=O)C c1(CSC)ccc(S(=O)(=O)NC(=O)NCCCC2COC(C)(C)C2)cc1 c1(C(=O)NC(CC)(CNC(C2CCCCN2C)=O)CC)n[nH]c2c1CCOC2 Cc1ccccc1C=CC(N1CCC(NC(C2(C)CC=CCO2)=O)C1)=O C12(CNC(c3csc(Br)c3)=O)CCC1CN(C(=O)C(O)CN1CCCC1)C2 c1(C(=O)NCCCN(C(=O)C(c2cnn(C)c2)C)CCC)cnc(O)c(Cl)c1 c1(C(C(=O)NC(C)C(C)(C)C2C(CC(C)C)C2)=O)ccc(F)c(F)c1 C1(C(N2CC3(CC(NC(C4C(CCC)C4)=O)C3)C2)=O)CCCC(C)(C)CC1 c1(CC(=O)NCCNC(COc2c(C)c(Cl)ccc2)=O)cnc2n1CCOC2 c1(C(=O)NC2CCC(C)N(c3ncc(Cl)c(O)n3)C2)cc2cc(F)ccc2s1 CC1(CNC(C2COCCO2)=O)CCCN(C(C2CC3(CCO2)CC3)=O)C1 C1(CNC(c2cccc(OCOC)c2)=O)C2CCC1CN(C(=O)C(C)(F)F)C2 C1(C(CC)C)CCN(C(c2csc(C(=O)O)n2)=O)CC1.C12(C)CC(C1)S2 c1(NCCCCCC)ccc(S(=O)(=O)N2CCC(OC)CC2)c(Cl)c1 c1(C(C(N2C(CNC(CSCCC)=O)CC2)=O)N(C)C)c(F)cccc1Cl c1(SC)nccc(N2CC3C(NC(c4cnoc4-c4ccco4)=O)C3C2)n1 N1(C(=O)OC(C)(C)C)CCOCC12CCN(C(=O)Nc1c[nH]c3ncccc13)C2 N1(C(c2ccc(C(C)C)cc2)=O)CCCC(C)(C(N2CCCC2C#N)=O)C1 CC1CC(CO)CCN1C(C12CCC(NC(c3ccn(C)n3)=O)(CC1)C2)=O N1(C(CC=CC=C)=O)CCC2(CCOCC2)C(CNC(=O)Cn2[nH]cnc2=N)C1 C1(C(=O)NC2CC(CNC(C3CCS3(=O)=O)=O)C2)(OC)CCC12CCC2 C(CC1=CCCCCC1)NC(C1C2(CCN(C(C3=C(C)OCC3)=O)C2)C1)=O C1(CC(=O)NCC(CC=C)NC(c2cnc(N(C)C)nc2)=O)COC(C)(C)C1 c1(CCC(=O)NCC2(F)CC(NC(=O)CC3CCC(=O)N3)C2)ccc(Cl)nc1 C1(C(N(CC#C)C)=O)CCCC1CNC(c1cnc(OC)s1)=O c1(CC)c(C(=O)NCC2CC(COC)CN2C(=O)CC)nnn1CC.C(C)=O c1(NC(C2CC3(C2)CN(Cc2cnccc2C(F)(F)F)C3)=O)nccc(Cl)c1I N1(C(c2c(C)[nH]c(C#N)c2)=O)CC(C(=O)NC(C)C(C)C)CC12CCC2 C(C)(N=c1nc(Cl)[nH]n2c(Br)cnc12)c1ccc(OC)cc1OC c1(CN2C(C(N(CCOC)C)=O)CCC2)cncc(N2CCCC2)n1 C1(NC(c2ccc(C)nc2C)=O)CCN(C(=O)Cc2cccnc2O)CC(O)C1 Cc1cc(Br)ccc1S(=O)(=O)NC12CC(C(=O)N=c3cc(Cl)cn[nH]3)(C1)C2 N(C(=NCc1ccc(C(F)(F)F)cn1)N1CCC(CN(C)C)C1)C(=O)OC(C)C c12ccc3nc(ccc3c1)NC2.C(=O)(C(COC(F)(F)F)N(C)C)OC C1(C(=O)NC2(CC(=O)NC(C(CC)C)CN(C)C)CCC2)CCC(=O)N(C)C1 c1(C(=O)NCCC2CCCN2C(C2CC23CC3)=O)cc([N+](=O)[O-])cc(Cl)c1Cl Cn1c(S)nc2cc(C(=O)NCCCNC(C3CCC3CF)=O)ccc2c1=O CN1CCN(c2nnc(-c3ccon3)s2)C(CNC(c2cc(F)cnc2O)=O)C1 N1(C(c2cnc(C)cn2)C(=O)NCC(=C)C)CC(C)CC1(C)C c1(CC(=O)NCC2(O)CCN(C(COC(C)=O)=O)C2)cncc2ccccc12 C1(NC(C2C(OC(C)=O)C2)=O)CC2CCC(C1)N2C(c1oc(CO)nc1C)=O c1(CC)nc(C)[nH]c1C(=O)NC1CCCC(NC(c2cc(C#N)no2)=O)C1 N(C1CN(C(c2coc(CO)c2)=O)Cc2ccccc21)C(c1cc(C)c(C)[nH]1)=O C1(C(=O)NC(CCC)C(N)=O)CN(C)CCN1C(=O)COC1CCOCC1 c1(C(N2C(CC(=O)NCC(C)(C)C(N)=O)CCC2)=O)ccc2ncoc2c1 S(=O)(=O)(c1ccc(C(N2CC(NC(=O)COCC3CC3)C2)=O)cc1)NC CC1CC(=O)NCC1C(N1CCN(C(C2CCCC(O)C2)=O)C(CCO)C1)=O C#CCCCC(C)C(=O)NC(CC(F)F)C(=O)NC1CCN(CCC)C1 C1(C(C)C)CN(C(=O)CCc2ncccn2)CCN1C(=O)CN1CCCS1(=O)=O C1(C)(C(=O)NCC(N(C(COCC=C)=O)C)C2CC2)Cc2ccccc2NC1=O C(=O)(C1=CCCCCC1)N(C)CC1N(C(CC(C)O)=O)CCCC1 N1(C(=O)CCc2cnccn2)CCN(C(c2cnn3c2CCCC3)=O)C2CCC12 C1(C(=O)NCc2cncc(C(=O)NC(CO)C3CCC3)c2)CCC(=O)NC1 C12(C(=O)NCc3nccc(C(=O)NCC4(CC)CC4)c3)C(=O)C3CC1C2C3.CN C1(NS(Cc2ccc(C)cc2)(=O)=O)CCCCN(Cc2ccc(O)c(C(=O)O)c2)C1 N1(C(c2c(C)ccnc2O)=O)CCC2(CC1)CC2NC(c1ccc(O)nc1C)=O N1(c2c(C)cncn2)CCC2(CCCN(C(C3CCCC4CCCN34)=O)C2)C1 c1(CNC(C2(C=C)CCC2)=O)cnn2c1CN(C(c1cc(C)on1)=O)CC2 C(=O)(CCCCCNC(=O)COCCOC)NCC(=O)N(CCC(F)(F)F)CC c1(CNC(CC(=C)C)=O)nnc2n1CCN(C(c1cnc3sccn13)=O)C2 Cc1coc(C)c1C=CC(N1CC(CNC(C2CC2C#N)=O)C(O)C1)=O CC(C)CC(C(=O)NCC1CCOC1)N(C(=O)CC1CC2(CC2)C1)C C(=O)(CC(C)C(=O)NCC1CCC1C(=O)NCC(CC)(CC)CC)OCC N1(CC(c2ccccc2)OC)CCCC(C(C)NC(=O)C(C)(C)CO)C1 c1(C(N2CCC(NC(CC3(C)CC3(Cl)Cl)=O)C2)=O)nc(O)nc(O)c1F C1(C(N2CC(O)(CCNC(C3CCC=CCC3)=O)C2)=O)CCC(=O)N1C1CC1 C=C(C)CC(C(=O)N(CCCNC(c1cc(OCC)ns1)=O)C(C)C)NC(C)=O c1(C(=O)NC23CC(C(N4CC(O)C(F)C4)=O)(C2)C3)c(F)ccc2[nH]ccc12 C(=O)(C(CC(F)F)C1CCC1)NCCOC1CN(C(COc2cc(C)on2)=O)C1 N1(C(C2(C#N)CCCO2)=O)CC2CC(C1)CN(C(=O)CCc1cc(Cl)cs1)C2 N1(c2cc(SC)nc(SC)n2)CCC(NC(=O)COCC2CCCO2)C12CCC2 Cc1ccc2cc(C(N3CCC(c4nnc(S)o4)CC3)=O)cnc2c1 c1(C(N2CCC(C(CO)NC(C3CCOCC3)=O)CC2)=O)cnc(Cl)c(I)c1 c1(C(=O)NC2CC(C)N(C(=O)CN(CC(C)(C)C)C)CC2)c(O)cc(F)cc1F N1(C(C=CCC2(NC(CNC(=O)OC)=O)CCC2)=O)CC2(CCC(O)CC2)C1 c1(-n2ncc(C(=O)NCC3N(C(COC4(C)CCCC4)=O)CC3)c2)ncc(Cl)cn1 Cn1cnn(CC(=O)NCC2CN(C(=O)CN3CSCC3=O)C2)c1=O C=CC(C)(O)CC(=O)NCC1(CNC(c2nccc(Cl)c2C)=O)CCCCC1 C1(C)(C(=O)NC2CCC(CNC(C3(OC)CCOCC3)=O)CC2)CCC(=O)CC1 C1(CNC(c2n(CCCC)nnn2)(C2CCC2(F)F)C)CC2CCC1CC2 CC(C)=C=CC(=O)NC(C(=O)NC(c1n[nH]c(CO)n1)C)C1CCOC1 C1(C(=O)NCc2c(CNC(C3(C)COCCO3)=O)cccc2)CC12CCOCC2 C1(NC(=O)COCC2CCCC2)CC2(C1)CC(CNC(C1C3CNC(=O)C13)=O)C2 N1(C(CC(C)(C(F)F)N(C)C)=O)CCC2(CCCCN(C(c3csnn3)=O)C2)C1 c1(N)cn2c(n1)CCC2.N1(C(C=C(C)Cl)=O)CC(F)C1 c1(N(CC=C)Cc2ccncc2)cc(Cl)nc(Cl)n1 N1(C(c2n(CCC)ncc2)=O)CCC(C(=O)N(CC)CC2CCCN2C)=C(F)C1 C(=O)(C1=CS(=O)CCC1)NC1C(NC(C(C)CN2CCCCC2)=O)C1 c1(NC)ccc(C(=O)NC2CC(N(C)C(C3CC(C(F)(F)F)C3)=O)C2)c(Cl)c1 CCS(=O)(=O)c1ccc(-c2cnc(C(=O)Nc3c(F)cc(I)cc3F)nc2)cn1 C1(NC(C(c2ccc(C)cc2)F)=O)CC(O)CN(C(=O)CCCN2CCCC2)C1 c1(C(=O)NC(CCCNC(COCC)=O)c2ccccc2)c2c(nn1C)CCC2 N1(C(=O)CC2(O)CCC2)CCC2CCN(C(=O)COc3cccc(Cl)c3Cl)C2C1 c1(CC)nc(C)sc1C(=O)N(C)CCOCCN(C(=O)Cc1ccccc1F)C c1(C(=O)NC(C)(CNC(C2CCNC2=O)=O)C2CC2)nc(C2CC2)n2ccccc12 c1(C(N2CC(NC(C3CCCC(CC(F)(F)F)C3)=O)(CO)C2)=O)ccccc1F c1(C(=O)NC2CC(CNC(CCC(C)OC)=O)C2)ccc(Br)cc1N C1(CC)(NC(=O)CCNC(N)=O)CCCN(C(=O)CC2(C)CCCCC2)C1 O(P(=O)(CCSCC1(O)CCCCCC1)OCC)CC c1(C(=O)NCCN(C2CCCCC2)C(C(C)C2CCC2)=O)cc(Cl)cc(Cl)c1F CC1(C)CCN(C(=O)C(C#N)CCCc2ccccc2)CC1NC(=O)C=CBr c1(C(=O)OC)ccc(NNC(=O)C(C)NS(=O)(=O)c2cccc(Cl)c2)cc1 N1(C(C(CC(F)F)NC(c2cc(C)ncn2)=O)=O)CCCCCCCC1 C1(NC(C2(C#C)CCCC2)=O)CC2(CCN(C(=O)Cc3cccc(CC)c3)C2)C1 n1(CC)nc(C)c(C(=O)NCCC2CC(NC(=O)C3=CCCCO3)C2)c1C CC1CN(C(=O)CC2CC2(Cl)Cl)CC1(C)CN(C(=O)CN1C(=O)CCCC1=O)CC C(=O)(CC(C)(C)SC)N(CC=CC(=O)N(CC(CC)O)CC)C c1(CNC(C(CC)(C)CC)=O)nc(C(F)(F)F)n2c1CCCC2 c1(C(N(C)Cc2nnc(C)o2)=O)ccc(O)c(Cl)n1 C(=O)(C(CO)C(C)(C)C)N1CC(N(C(CS)=O)CCC)C(O)C1 N1(C(c2cnc(CCCC)s2)=O)CCOC(C)(CNC(C2(CO)CCCO2)=O)C1 CC(CCNCc1ccccc1OCC(F)(F)F)C(F)F CC1(C)CCCCCC1NC(C1CCCCC1)=O c1(C(=O)OCC)[nH]cc(C)c1C(=O)NC1CN(C(C2(C)CS(=O)(=O)C2)=O)CC1C CC1=C(C(=O)N2CCOC(CCNC(c3cncc(Cl)c3Cl)=O)C2)CCCO1 c1(NCCOCCOCCOC)nc2ccccc2nc1NC1CC(F)(CO)C1 C1(CNC(c2onc(C)n2)=O)CCC(NC(=O)C(C)CF)CC1 C1(N(C)C)(SCC)CN(C(=O)C(C)CN(C(=O)C=CC(=O)NC2CC2)C)C1 Cc1ccc(C)c2[nH]c(C(=O)N(CC(O)CNC(C3CNC(=O)N3C)=O)C)cc12 C1(CNC(COC2CCC(C)CC2)=O)CC2(CC2)CN1C(=O)C(C)N(C)C C1(CC(NOCCCC)=O)CCC(C(OC)OC(C)(C)C)CC1 c1(C(=O)NC(C(C)(C)C)CNC(C2CC2C(F)F)=O)cc(F)c(F)cc1Cl C1(C(=O)NCCN(C(=O)C=C(C)Cl)CCC)CCC(C(C)C)NC1=O N1(C(Cc2cc(C)no2)=O)CCC(C)C(CC(=O)NC2(C)CCSC2)C1 Cc1cccn2ncc(C(=O)NC(C)CCN(C(=O)C=C3CC3)C)c12 C(=O)(CC(CC(N)=O)CC(C)C)NCC1N(C(C(CC#C)CC#C)=O)CC=C1 n1(CC(=O)NC2CC(N3CCNCC3)C2)ccc(C(=O)O)n1 N1(C(C2C(=C)C2)=O)CCC(CNC(c2cscc2C(F)F)=O)CC1C c1(C(=O)Nc2cnc(C(=O)Nc3cn[nH]c3)s2)cc2ccc(Br)cc2[nH]1 C1(NC(C(C)n2cnnn2)=O)CCCC2CN(C(=O)C(O)CC(C)(C)C)CC12 c1(C(=O)NC2(C(=O)O)C(C)SCCC2)cncc(P(C)(C)=O)c1 C12C3CN(CC13)C2.C1(C(=O)NC(c2cn(CC)nn2)CCC)(OC)CCN(C)C1 c1(CC)cc(C(=O)OCc2ccc(Sc3ccc(Cl)cc3)cc2)cc(CC)c1 C1(CNC(CCCNC(C)=O)=O)COCC2(CCN(C(=O)C=CC=C(Cl)Cl)CC2)O1 c1(C(N2CC3CCN(Cc4cocn4)C3C2)=O)cc(I)ccc1[N+](=O)[O-] c1(CC(N2CC(COCC)(NC(=O)C=CC3CCOC3)C2)=O)cccnc1O N1(C(C(CC)=CCCC)=O)CC2(CC2)CC1C(N1CCC(CC)CC1)=O N1(C(CCC=C=C)=O)CCC2CN(C(C34C=CC(CC3)C4)=O)CC2C1 C1(NC(C2CC(SC)C2)=O)CCN(C(C2(C(N3CCCC3)=O)CCC2)=O)C1 c1(C(N2CC(C)C(C)(CNC(C3CC3(F)F)=O)C2)=O)csc2c1CCC(C)(C)C2 N1(C(c2ccc(OC)cc2)=O)CCN(C(c2cc(Cl)c[nH]2)=O)C2CC12 C1(NC(=O)NC(Cc2cccnc2)CO)COCC1C(=O)O c1(C(=O)NCC2C(CNC(=O)COC(F)F)C2)cncc(N2CCCC2)c1 Cc1cc(=O)n(CC(N2CC3CC(CNC(c4ccon4)=O)C3C2)=O)cn1 C(c1ccc2c(c1)NC(=O)CO2)=CC(=O)NCC(CC)NC(CSCCC)=O c1(CC(=O)NC(CC)(C)CNC(c2ccsc2OC)=O)ccc2c(c1)CCCO2 CCCC(C(=O)NCC(C)S(C)(=O)=O)NC(c1cc[nH]c1C)=O c1(CNC(C=CC(C)NC(C(C)NC(C)=O)=O)=O)nc(C)c(C)[nH]1 N1(C(c2c(NC)nccc2)=O)C(CNC(=O)CN2CCOCC2)CC2COCC12 C1(C(=O)NC(COC)COC)(CC)CCCN(C(=O)CP(C)(C)=O)C1 C1(C(=O)NCc2ccc(CCNC(=O)OC(C)(C)C)cc2)CCCCC12CCC2 C(=O)(C(CNC(C)=O)C(C)C)NCC(CC(=O)NC(CCC)C(=O)N(C)C)C c1(NCC(=O)NCC2C(CNC(C=CC=CC)=O)C2)ccc(C)cc1 C1(CC(NOCCCOC)=O)CC(C)(C)CN1C(=O)Cn1c(O)nnc1O N1(C(=O)NCc2cnc(C(C)C)s2)CCCCC1C(C)O Cc1cccc2ncnc(N3CC(NC(c4cncn4C(C)C)=O)CC3C)c12 C(CC(=O)O)(c1cccnc1)NCC(CO)NC(=O)OC(C)(C)C c1(C(N(CC(C)NC(=O)C=CC2CCOC2)C)=O)cnn(C2CCC2)c1 c1(CC)cc(Br)ccc1C(N1CC(NC(c2cc(I)ccc2F)=O)C(O)C1)=O C(=O)(CC(F)(F)C(F)(F)F)N1CCC(N(C(c2ccnc(C)n2)=O)C)C2(C1)CC2 C1(NC(c2c(C)nn(C)n2)=O)CCC2CCN(C(c3cnsn3)=O)C1C2 c1(C(N2CC(C(C)NC(C3CCN(C)CC3)=O)C2)=O)cc2n(c1)CCCC2 N1(C(CCCC)=O)C2CCC1CN(C(c1cncc(N(S(C)(=O)=O)CC)c1)=O)C2 CC1(C)CN(C(c2cnc[nH]2)=O)C1Cn1cc(CNc2ccc(Cl)cc2)nn1 N1(C(C2C(C)CCO2)=O)CCC(C2CC2)C1C(=O)NCc1ccncc1 CC1CN(C(C2(C)CC2(F)Cl)=O)CC(C)N(C(c2n[nH]c(C3CC3)n2)=O)C1 c1(CNC(CCNS(NC)(=O)=O)=O)ccc(C)cc1.C1(=O)CC2(CC2)CNCN1 CC1c2cc(Br)ccc2CCN1CC(=O)NCC1CCc2ccccc21 N1(C(C)=O)CC(C2CN(C(=O)C(C(C)C)NC(=O)C(C)(C)C)C2)C1 N1(C(C(CC)N2CCCC2=O)=O)CCC(CN2CCC(F)(F)C2)CC1 CC1Cc2cc(S(=O)(=O)NC(=O)C(c3cc(F)ccc3Br)C)cc(Cl)c2O1 C1(C)(CC)CC(C(=O)NC(C)CNC(c2ccc(NC(=O)NC)s2)=O)CCO1 CC1CCN(C(c2cccnc2C(F)(F)F)=O)CC1CNC(C1(C)CCCO1)=O n1(CCOC)ncc(C(=O)NC2CN(C(=O)CCCN3CCCC3)CC2F)c1C N1(CCCC)CCOCC1C(=O)NCC(C)NC(=O)CCc1ccc(C)s1 c1(C(C(=O)NC2CCCC2)C)cn(C)nc1C1(NC(COC)=O)CC1 N1(C(C2C3CN(C(c4ccc(OCCC)cc4)=O)CC32)=O)C2CCCC1COC2 C1(OC)(CNC(C23CC(C2)C3)=O)CN(C(C2CN(C(C)C)C2)=O)C1 c1(C(N2CCC(C)(CNC(=O)CSc3ccncc3)C2)=O)cnn2c1OCCC2 N1CCCCC(C2CN(C(=O)CCSC)C2)C1.C=C=CCC=O C(=O)(C(O)CC(C)(C)C)N1CCCCC(C(=O)NC2CCN(CCC)CC2)C1 C#Cc1ccc(CCNC(N2CCN(c3cncc(Br)c3)C(=O)C2)=O)cc1 C1(c2ccccc2)(NC(=O)Nc2cc(C(C)C)no2)CCCOC1 CC1CCC(N(C(c2cn(CCNC3(C)COC3)nn2)=O)C2CC2)CC1 N1(C(CC)=O)CCOC(C)(CNC(c2c(Cl)csc2Cl)=O)C1 c1(C(=O)NCCC(C)N(C)C(C2CC3CCC2O3)=O)cc(Cl)c(Br)[nH]1 c1(OC)c(CC2CN(C(=O)NC3(CCS(N)(=O)=O)CCC3)CCO2)cc(Cl)cc1Br S(=O)(=O)(CC(=O)NCCC(C)(C)NC(C1CC1c1ccoc1C)=O)NC C1(C)(c2nnc(-c3cc(C)n(C)n3)o2)CCC(C)CC1 N1(CC(C)C)CCC(C(=O)NC(C2CN(C(C3(CF)CCOCC3)=O)C2)C)CC1 C1(CNC(=O)Cn2cnnc2)CC2CCCC2N1C(=O)CSC1CCS(=O)(=O)C1 c1(OC)ccc(C(=O)NCC2CC(C)N(C(c3ccccc3C)=O)C2)c(OC)c1 N1(C(CC(CC)CC)=O)CCN(C(=O)C(C)Cn2ccc(C)n2)CC(O)C1 c1(OC)ccc2c(c1)C(NC(=O)C(N1CC3CC(O)CC1C3)=O)CCC2 c1(C(N2CCN(C(Cc3ccc(C)cc3)=O)C(C)C2)=O)c(C)ccc(C)c1N C(=O)(CC(C)(C)C(=O)N(CC(C)NC(c1cncc(Cl)n1)=O)C)OC C1(CNC(CC(CN(C)C)(C)C)=O)CC2CCCCC2N1C(C1CCC1)=O c1(C(C(CC)=O)=O)cncc(NC(C2(C)CC2)=O)c1.C12(CC1)CC(=O)NC2.N.OC c1(C(=O)NCC(CNC(c2cccc(C3CC3(F)F)c2)=O)O)cc(F)ccc1O c1(C(N2C3(C(=O)NCCCC(C)(C)CO)CC(C2)C3)=O)cncc2[nH]ccc12 c1(NCc2ncc(OC)nc2)nccc(=NCc2cccnc2Br)[nH]1 C1(OC)CCCC(CNC(=O)CCN(C)C(c2nc(C)oc2OC(C)C)=O)C1 Cc1nn(C)c(C)c1C(=O)C(=O)N(C)CCOCCN(C)C(c1cnsc1)=O c1(C(N(C2CC(NC(C3(C(F)F)CC(F)(F)C3)=O)C2)C)=O)cnc2n1CCC2 C1(OC)CCCC(NC(=O)CC2(N(C(=O)C=C3CCCCC3)C)CC2)C1 CS(=O)(=O)c1ccsc1C(=O)NCCCCC(CO)NC(=O)Cc1cnsc1 C(=O)(CCN(OC)C(=O)C1CCN(C(C2CC(OC)C2)=O)C1C)OC CC1CN(C(C2(C3CCCCO3)CC2)=O)CCC1CNC(C1(C(N)=O)CC1)=O C1(CN(C(C2(CC#C)CCOC2)=O)C)CC(F)CN1C(=O)CCC(=O)NCC C(=O)(C(O)C(CCC)NC(C1CCS1(=O)=O)=O)NC1(C#C)CC(F)(F)C1 C=CC1(CC(=O)NCCC(C)CCO)CN(C(C2(OCC)CCCC2)=O)C1 C1(CNC(C(C)(C)C)=O)CN(C(C2CCCCCC2)=O)CCC1C(F)(F)F N(C1CCc2cccnc21)C(C12C(NC(c3c(C)nccn3)=O)C3CC1C2C3)=O N1(C(c2cc(CNC(c3cccc(C)c3O)=O)no2)=O)CCCC2C(O)C(C)(C)C12 Cc1c(C(N2C(C(=O)NCC(F)CO)CC2C)=O)cccc1C#N C1(NC(C2CCCCC2)=O)CCCC12CCN(C(c1cc(Br)cs1)=O)C2 c1(C(N2C3(CNC(C4CCCC(C)C4)=O)CC(C2)C3)=O)csc([N+](=O)[O-])c1 Cc1ccc(CCC(=O)NC2CCC(NC(C3SCCCS3)=O)C2)cn1 C1(C(N(c2cn(C)cn2)C)=O)CCCN(C(=O)CN2CCCCC2)C1 N1(C(CNC(CC(C)C)=O)=O)CC(NC(C2CC=CC2)=O)CCC1C C1(N(C(C(C(C)O)N(C)C)=O)C)CCCCN(C(c2ccc(O)cc2)=O)C1 Cc1cc(Br)c(NC(C2(C)CCN(C(c3ccncc3)=O)C2)=O)cc1[N+](=O)[O-] CC12CCCCC1CN2C(C1CCN1C(=O)CC(F)(F)F)=O N1(C(COCc2cc(C)no2)=O)CCC(N(C)C(c2c(C)n[nH]c2C)=O)CC1 c1(OC)cc(C=CC(N2CC=CC(NC(=O)C(Cl)=CCl)C2)=O)ccc1O N1(C(C2CCCC(OC)C2)=O)CCN(C(=O)CCn2cnnn2)CC1CO c1(NC)ccc(C(N2CCCC2CNC(=O)C(O)C2CCCC2)=O)c(C)c1 C1(C(C(=O)NCc2cccs2)N(C)Cc2cn(CC)nc2)CCC2(CC1)CC2 N1(C(C)=O)CCOC(C(=O)Nc2cccc(-c3cc(C(=O)N(C)C)no3)c2)C1 C1(C(=O)NCC2C(NC(c3cn(C)nc3C(F)F)=O)C2)CCC2(CCC2)O1 c1(C(N2CC(C)C(NC(=O)C=CC(C)(C)C)C2)=O)cc(Br)ncc1F C1(C(=O)NC(C)CN2CCN(C)CC2)CC12CCN(C(c1cnns1)=O)CC2 N1(C(C=CC)=O)CCC(C2(NC(c3cccn3CCC)=O)CC2)C1 Cc1cc(C(=O)NC(C)CC2CCN(C(=O)CC(C)(C)F)C2)ccc1C(N)=O C1(CNC(C2C(C)COCC2)=O)CC2(C1)CC(N)CCO2 c1(OCCOC)cccc(C(=O)NC2CC(CO)N(C(=O)CC(F)F)C2)c1 N1(C(=O)NCC(N2CCCC2)C)CCCN(C(=O)Cc2nn[nH]c2Cl)CC1 CC1CCC(F)(C(=O)N(CCC(N2CCCCCC2CO)=O)CCO)CC1 N1(C(C(CN(C)C)NC(CSCC#C)=O)=O)CC2CCC1C(O)C2O C1(NC(c2cncc(CC)c2)=O)CCCN(C(=O)Cc2ccnn2C)CC1 c1(C(=O)NCC(O)CCNC(C2(F)CCC2)=O)cnc2ccc(F)cn12 N1(C(C(CC)CC)=O)CC(CNC(c2ncc(F)cc2F)=O)C(C)(C)C1 N1(C(c2ncn(C)c(=O)c2)=O)CC2(C1)CN(C(c1csc(Cl)c1)=O)CC(C)(C)O2 N1(C(C(c2cc(C)oc2C)C)=O)C2CCC1C(CNC(c1cc(F)n(C)n1)=O)C2 C1(C(N(CCC(C)NC(=O)C(C)(C)n2cnnn2)C)=O)CC12CCOCC2 CC(C)(C)C(CNC(C1CC2(CCC2O)C1)=O)C(=O)NCCc1ccc(O)cn1 c1(C(=O)OCc2ccc(O)cc2)cnn2c1OCC2 N1(C(CN(C)C(=O)C2CC2)=O)CC2(CCN(C(c3csc(Cl)n3)=O)CC2)C1 C(=O)(CC(C)CN(C)C)NCC(CC)NC(=O)CCc1ccc(C(C)C)cc1 C1(CNC(c2ccc(OCC#C)cc2)=O)CN(C(C2CCCN2C)=O)CC12CC2 c1(C(Cn2cccn2)NC(C(=O)N(C23CC(C2)C3)C)=O)ccccc1 C1(OC)CN(C(=O)CCCNC(=O)C(C)(C)n2cnnn2)CC12CC2 S(=O)(=O)(c1c[nH]c(C(=O)O)c1)N1CCC(C(C)O)CC1 c1(C(=O)NCCCCC2CCCN(C(C(C)(C)SC)=O)C2)cnc(O)n(C)c1=O C1(OC)(CNC(=O)Cc2cncn2C)CCN(C(=O)C(c2ccc(F)cc2)=O)C1 Cc1csc2ncc(C(N3CC4CCN(C(=O)CC5CCCO5)C4C3)=O)c(=O)n12 C1(NC(Cc2n(C)ccc2)=O)CC2CCC1(C(=O)NCCCC(C)(C)O)C2 N1(C(c2ccc(C)c(Cl)c2Cl)=O)CC2COCC(C1)C2NC(=O)C(Cl)=CCl C(=O)(CC(C)CC(C)(C)C)N1CC(O)(CNC(C(C)N(C)C)=O)C1 C=CCCC(C(=O)OC)NC(C1(CC=C)CCN(C(=O)C(F)=CCC)C1)=O c1(CCC(=O)N(C)CC2N(C(CC(CC)C)=O)CCCC2)cccc(C#N)c1 C1(C(=O)NC(CC)CNC(c2cc(Cl)c(Cl)s2)=O)CCc2nncn2C1 Cc1cnc(CN2CC(C(N3CCCCC(C)C3)=O)CC(F)C2)c(F)c1 c1(C(N2C(C)CC(NC(c3cc(CCC)[nH]n3)=O)C2)=O)coc2c(C)cccc12 CN1CCN(C(C2CCCN(C3CCC(=O)NC3)C2)=O)CC1 c1(C(=O)OCC)c(C)sc(CNC(CC2CCCN2C)C2CC2)c1Cl N1(C(C2CCC3CC3CC2)=O)CC2CCCC(C1)N2C(C1CCS(=O)(=O)N1)=O c1(CC)cc(C(N2CC=CC2CNC(C2CN(C(=O)NC)C2)=O)=O)ns1 Cc1[nH]c2ccc(F)cc2c1C(N1CCCN(C(=O)Cc2cnccn2)CC1)=O c1(CN2CCN(C3CN(C(C4C5COCC45)=O)C3)CC2)ccc(O)cc1O O=S(=O)(c1ccc(N2CC3C=CCC3C2)c(Cl)c1)NCC(O)CN1CCCC1 CC1CN(C(C2(S(N)(=O)=O)CC2)=O)CCC1NC(=O)CC1CC(O)C1(C)C C1(CNC(c2c(OC)ccs2)=O)CN(C(C2C3(CC3)C23CC3)=O)CC2(CCC2)O1 C1(CCC(N2CC(NC(CC(=O)OCCC(C)C)=O)C2)=O)CCCCCC1 N#Cc1cccc(CNc2ccc(-c3ccc(F)s3)nn2)c1 Cc1sc(C(N2CC(C3(NC(c4n[nH]cc4F)=O)CC3)C2)=O)c(C)c1C c1(NC)ccc(C(=O)NC(C(=O)NCCC(O)C(F)F)c2cccs2)cc1 C1(CCNC(C(C)(O)C2CCC2)=O)CSCCN1C(c1cccnc1N)=O N1(CC(N2CC(N(C(C3(C(=O)OCC)CCOC3)=O)CC)C2)=O)CCCC(C)C1 c1(-c2cc(C)c(O)c(C)c2)ccc2ncc(C(N3CCOCC3)=O)n2c1 C1(C(N(CCCN(C(c2ncn(C3CC3)n2)=O)CC)CC)=O)CC(C(C)C)=NO1 Cc1nc(C(=O)NCC(C(C)C)NC(c2cc(Cl)c(Cl)[nH]2)=O)c2ccccn12 Cn1c(C(N2CCCCC2C2(NC(C3C(Cl)(Cl)C34CC4)=O)CC2)=O)cnc1S C1(CCC=C)(C(=O)NCC2(C)CCCO2)CN(C(=O)CC2OCCCO2)C1 CC1C(NC(C2CCC3CC23)=O)CCCN1C(c1cnc(Cl)cc1Cl)=O C1(C(=O)NC(COC)C)C2CCCC1CN(Cc1c(Br)cc(Br)c(O)c1Br)C2 S(=O)(=O)(CCCNC(C)(C(C)(C)C)c1nnnn1C1CCOC1)NC c1(C(=O)NC(CNC(C(CC)OC)=O)C2CC2)cc2nc(Cl)ccc2o1 CC(C)C(C(=O)NCCc1ocnc1CO)C(C)NC(C1CC(OC(F)F)C1)=O CC1(C)CC(CNC(c2nnn3ccccc23)=O)CN(C(C2(C)CCCS2)=O)C1 Cc1ccc(C)c(S(=O)(=O)NC2CN(Cc3ccc(Br)c(Cl)n3)CC2(F)F)c1 C1(C(C)NC(c2ccn(C(F)F)n2)=O)CCCN(C(=O)C=C2CCCC2)C1 N1(C(C(C2(O)CCC2)NC(CC2ON=C(C)C2)=O)=O)CC(O)CC1C(N)=O c1(C(=O)OC)ccc(C(=O)NCC2CCCCCN2C(c2cnn[nH]2)=O)cc1Cl C(=O)(CCCCCCNC(C1CC1C1CCCO1)=O)N1CCC(C#C)CC1 c1(OCC)ccccc1C(=O)N(C(C)CNC(=O)C(F)(F)c1ccccn1)C c1(C(N(CCN(C(=O)CCCC(C)(F)F)C)C)=O)n[nH]c2c1CCOC2 N1(C(CSCCC#N)=O)CC(C2(NC(C3(Sc4ccccc4)CC3)=O)CC2)C1 C(c1ccc(Br)cc1)=CCCNC(c1c(C)nccc1)=O c1(C(=O)NCC2(NC(C=CCC)=O)CC3CCC2C3)cccc2c1COC2 C#Cc1cccc(C(=O)N(C)CCN(C)C(c2cc(O)nc(OC)n2)=O)c1F C(=O)(C(C)CN(C(=O)C=C(C)C1CC1)C)NC(C#C)CC CC1CCC(NC(=O)CCCSC(C)(C)C)CN1C(c1cc(C(F)F)ncn1)=O C1(CC(=O)OC2CC2)CCN(C(N(C)CC2CCC2C(=O)OC(C)(C)C)=O)CC1 C12(C(=O)NCc3nccc(C)c3)CC(CO)(CN1C(C1CC3COCC3C1)=O)C2 C1(CCOC)(NC(=O)C(c2cn(C)nn2)NC(=O)CC2OCCC2C)CCCC1 c1(NC2CC(C)N(C(C3(CN(C)C)CC3)=O)C2)cc2nncn2cn1 c1(OC)cccc(Cl)c1CNC(N1CCC(C)C(NC(=O)OC(C)(C)C)C1)=O C(=O)(CC(C)CN=C(NCC1(O)CCN(C)C1)NC1CCCCC1)OC C1(CC#C)(C(=O)NC23CC2CN(C(=O)CCc2cnc[nH]2)C3)CCCCO1 C1(NC(c2cc(-c3ccncc3)ccn2)=O)CC2CN(C(=O)CSC3CC3)CC2C1 C1(CNC(C2(CC)CCCCO2)=O)CC(C(=O)Nc2cc(C)ccc2O)=NO1 C1(CNC(CC(C)(C)C#N)=O)CN(C(c2ccnc(O)c2)=O)C2(CCOCC2)C1 Cc1nc(C(N2CC(NC(c3ccccc3OC(F)(F)F)=O)C3CC23)=O)c(C)s1 c1(CNC(c2cccc(C(=O)NC(C(=O)OCC)C)c2)=O)cncc(OCC)n1 Cc1cc(=NCCOc2ncccn2)[nH]cc1S(=O)(=O)NCC(C)C(F)(F)F C#Cc1ccc(NC(C2CCCCC2C)=O)cc1C#N N1(C(c2cnc(SC)n2C)=O)CCC(NC(C2CC2C)=O)C(F)C1 C1(CC(=O)NC2C(CCOC)C2)CN(C(=O)CCc2ccc(C)o2)CCC1C C(=O)(C(F)C(=O)N1CCN(CCNC(=O)CCc2ccnn2C)CC1)OCC Cn1cc(Cl)c(CC(=O)NC2CCCCC2NC(=O)C(O)C(F)F)n1 C1(NC(c2sccc2F)=O)C2CC1CN(C(C1COCCC1(F)F)=O)C2 CN=c1[nH]cc(C(=O)NCC(C)C(=O)NCCc2c(C)n[nH]c2C)s1 c1(N2CCN(C(C3CCCN(CCC)C3)=O)CC2C)nc(Cl)nc2[nH]cnc12 c1(NC(C2(F)CCN(Cc3cccc(C#N)n3)C2)=O)cccc2c(Cl)cccc12 c1(C(=O)NCC(C)NC(=O)C2=CCCC2)cc2ccnn2cn1 c1(C(=O)NC2(C(N3CCC(OCC)C3)=O)CC(O)C2)cnncc1O c1(OC)ccc(CN2CC(C)(CNC(=O)COC3CCOC3)C2)c([N+](=O)[O-])c1 Cc1cc(C(=O)NCC23CC2CN(C(=O)C#CC2CC2)C3)ccc1F C1(NC(C(C2CC2)OCC)=O)(CO)CCCN(C(=O)C(C)C(F)F)C1 C1(C)(CNC(CC2CCCC(C)O2)=O)CC(F)(F)CN1C(c1cnn[nH]1)=O CCC(C)C(O)CC(=O)NCC(C)(C)C(=O)N(C1CCC1C)C C1(F)(C(=O)NC(C2CCOC2)CNC(c2c(SC)cn(C)n2)=O)C(C)(C)C1(C)C Cc1ccc(S(=O)(=O)NC(CCC(N)=O)C(=O)NC2CCCCC2(F)F)c(F)c1 C1(CC=C)CC(O)CCN1Cc1ccc(C)cc1C CCCC(CC)C(=O)NC1CCCCC1CNC(c1ccc(F)s1)=O N1(C(Cc2c(C)cco2)=O)CCC(CO)(NC(C2CC23CC3)=O)CC1 C(Cn1nnnc1C(C(C)(C)C)c1ccccc1)(C(C)C)OC.C1CCS1 c1(OCC)cc(NCC2CC(NC(C3CC3F)=O)C2)nc(C)n1 Cc1nc(Br)ccc1-n1cc(-c2csnc2C)nn1 N1(C(c2c(C)snn2)=O)CC(NC(c2cn(C)cc2C(F)(F)F)=O)CC(O)C1 c1(CC(=O)NC2C(CNC(C3N(CCC)CCC3)=O)CC2)nc2ccccc2s1 Cc1cc(N2CCOCC(CNC(=O)CCCC3CCC3)C2)nc(S(C)(=O)=O)n1 C1(C(N2CC(CNC(c3cncc(CC)c3)=O)C(C)C2)=O)CCN(C)C(=O)C1.C1CC1 c1(C(N2CCN(C(CC(CCC)C)=O)CC2CCO)=O)cc(F)c(C#N)c(F)c1 C1(C(N2CCC(CC)C2)=O)COC2(C1)CN(C(C1CC(O)C(F)C1)=O)C2 CC(C)CCC(F)C(=O)NCC(CC1CC1)C(=O)NCCCn1cnnn1 c1(C(=O)NCC(C)CN(C(=O)Cc2cncn2C2CC2)C)n[nH]c2c1CCOC2 N1(C(c2c(CC)ccs2)=O)C2CCC1CC(NC(=O)CC1C=CCC1)C2 Cc1cccc2cc(C(=O)NCC3(N(C(=O)CC4CC4(C)C)C4CC4)CC3)oc12 CC(C)CC(C)(C)C(=O)NC1CCCC1NC(c1ccccc1CO)=O C1(NC(CC(C)F)=O)CCC(NC(c2nccnc2N)=O)CC1 C(=O)(C(C)CO)N(C(C(=O)NCCOC(C)C)C1CC1)C N1(C(c2cc(OC)c(Br)nc2)=O)CCC(C)(C)C(NC(C2CCC2)=O)C1 CCCC(CC1CCCC1)C(=O)NC1CN(C(=O)C(COCC)N=[N+]=[N-])C1 C1(NC(C(CC=C)OC)=O)COC2(C1)CN(C(=O)CC1OCCO1)C2 c1(CC(=O)NC(C2C(C(=O)Nc3cccc(OCC)c3)C2)C)cc(C)ccc1F N1(C(CC2CCC(C)CO2)=O)CC2CC(C1)CN(C(C13CSC(C1)C3)=O)C2 c1(C(=O)NC2(CCC(=O)NC3C(CC)CCC3)CCCC2)cnc2c(c1)COC2 c1(OC)ccccc1C(CNC(=O)C(C)CO)NC(c1sccc1OC)=O Cc1ccc(CN2CCCC(CCC(=O)NC(CO)C(C)C)C2)cc1C C1(C(N2CCCC(C=C)C2)C(=O)NCC(=C)C)Cc2ccccc2C1 c1(C(N2CCC(O)C(C)C2)C(=O)NC(c2ccccc2)C)ccc(F)c(I)c1 C1(NC(c2cnc(COC)s2)=O)CCC(C)(CNC(=O)CC(F)(F)F)C1 Cc1cc(Cl)c(Cl)cc1C(=O)NC1CN(C(=O)C(O)CC(C)C)C2(CCC2)C1 N(C1CCCc2occc21)C(C1C(C=CC)CN(C(=O)Cn2cnnc2)C1)=O C1(C2CCCN(C(=O)CN(C)C)C2)(NC(CN(C)C(c2ccncc2)=O)=O)CC1 c1(C(=O)NCC2CC(NC(C3CCC(O)C3)=O)CCO2)ncc(Cl)cc1Cl C1(NC(C2CCNC2=O)=O)CC=CCC1C(N1CC(Cc2ccoc2)C1)=O C=C1CCN(C(C2COCOC2)=O)C(C(N2CCC(OCCO)C2)=O)C1 N1(Cc2c(C)nc[nH]2)CC2(CCOCC2)C1C1CC1 c1(C(=O)NC(CNC(=O)C=Cc2ccco2)C2CC2)cc2c(s1)CCC2 N1(C(c2c(C)cccc2N)=O)CC(C)(CNC(C23CCC2C3)=O)CC1(C)C c1(C(=O)NCCN(C(C(n2c(C)ccn2)C)=O)C(C)C)cnc(=NCCF)[nH]c1 C1(C(=O)NC(C2CCCC2)CNC(=O)Cc2cc[nH]c2)CCS1(=O)=O c1(C(=O)NC(CNC(C=C(C)c2ccsc2)=O)(C)CO)ccc(S(C)(=O)=O)[nH]1 c1(CNC(c2scc3c2OCCO3)C)c(Br)sc2ccccc12 C(=O)(C1=CS(=O)CCC1)N1CC(C)C(CNC(C2(C)CNC(=O)C2)=O)C1 C1(NC(C)CCO)COC2(CCN(c3ncc4[nH]ccc4n3)CC2)C1 C1(C(=O)NCC(CC2CC2)CO)(CNC(=O)Cn2ncnn2)CCCC1 N1(C(C(C=C)(F)F)=O)CCOC(C)(CNC(=O)Cc2cnc(C3CC3)[nH]2)C1 CCC(C)(C)CC(=O)N1CCOCC(C(N2CC(C)(OC)C2)=O)C1 CCCC(CNC(c1cc(C)nn1C)=O)C(=O)NC1CC12CC(OC)C2 C1(CC=C)(CNC(=O)Cc2cnoc2)CCCN1C(=O)C(O)CCN(C)C Cc1nc(C(=O)NCC2(F)CC(CNC(=O)Cc3cnn(C)c3)C2)c(C)s1 c1(C(=O)NC2CCCC(N(C(=O)Cc3cncnc3)C)C2)cc2nnn(C)c2s1 CN1N=C(C(=O)N2CCC3CCN(C(c4ccc(=N)[nH]n4)=O)C3C2)CCC1=O c1(C(N2N=C(C=O)CC(C)C2)=O)cnc2ccc(Br)cc2c1 C(CC(=O)N1CC(O)CCO1)C1N(C(=O)Cc2ccccn2)CCC1 c1(CNC(=NC)NCC2C(F)(F)C23CC3)ccccc1Cl.C12CCN(C1)C(=O)N2 c1(N(CCC#N)C)ccc(S(=O)(=O)NCC2COCO2)cc1 Cc1ncc(NC(C2C3CN(C(C4CC5CCC4O5)=O)CC23)=O)cc1F c1(OC)ncc(-c2sccc2C)cc1C(=O)Nc1sccc1C(C)=O C(CCC(C(=O)N(C)Cc1cocn1)NC(c1cc(CCO)on1)=O)OC C(=O)(C1=CCN(C(=O)C(F)C2CCOC2)CC1)N(C)CCn1cncn1 CC1CC2CC2CC1C(=O)NCC1CN(Cc2ccc(SC(F)(F)F)cc2)C1 S(=O)(=O)(c1ccc(Br)cc1NC1CCC(CCO)CC1)N1C(C(CC)O)CCC1 c1(C(=O)NC(CNC(c2cccc(CC)c2F)=O)C2CC2)ccn2cccc2c1 N1(CC(=O)N(C2CCN(C(COCC(=C)C)=O)C2)CC)CCN(C)C(=O)C1 C12(C(=O)NCc3c(C)noc3)C(NC(c3ncc(F)cc3F)=O)C3CC1C2C3 CCCC(F)(F)C(=O)NC1CCC(CCC(=O)NCc2cn(C)nc2OC)C1 C1(CC(=O)N(C2CCN(C(=O)C(C)C(=O)OC)C2)CCC)(COC)CCCCC1 c1(C(=O)NCC(C)NC(C=Cc2ccc(SC)s2)=O)ccc2nc(O)n(C)c2c1 c1(C(N(CCC)CCNC(=O)C(C)OCC(C)C)=O)cnsc1C C#Cc1cc(C(=O)NCC(C)(O)CNC(=O)C(C)(C)N(C)C)cc(F)c1 C(=O)(C(C)CC(N)=O)N(C1CCN(C(=O)CCSc2ccc(F)cc2)C1)CCC C1(C(=O)NCCC(C)NC(c2c(C(=O)OCC)c[nH]c2)=O)CCN(C)C1C c1(CC(=O)NC2(CNC(C(CC)O)=O)CCOCC2)cc(F)c(F)cc1F CC(C(=O)NCC(C1CCC1)NC(C1CC(=O)C1)=O)S(C)(=O)=O C(=O)(CCCCCn1cnnn1)N1CC2C(CCNC(CCC3(C)CC3)=O)C2C1 c1(C(=O)NCC2CN(C(Cc3cc(C)sc3)=O)CC2C)n[nH]c2c1CCOC2 C1(CC(=O)NCc2cnc(C)s2)CC(NC(C23CC(F)(C2)C3)=O)C1(C)C c1(CC)ccccc1CC(=O)NCC1CN(C(C2CC2CC(C)C)=O)CC1O c1(C(C(=O)OC)(C)NC(C2CN(C(C)C)C2)=O)cn2cccc(F)c2n1 Cc1cc(C(=O)NC2CCC(C)(N3CCOCC3)CC2)nnc1O c1(C(N(CCCNC(c2nccc(OC)c2F)=O)C)=O)nc2n(c1Cl)CCCC2 C1(CCNC(CSc2cn(C)nc2)=O)CN(C(C2CCC(O)C2)=O)CCO1 N1(C(CC=CC=C)=O)CCCC(C)(C)C1CNC(C1CCC(C)(C)OC1)=O Cc1nsc(N)c1C(N1CCC(C(C)NC(=O)C#CC2CC2)CC1)=O C(=O)(C(C)(C)CCCO)N(C)CC1OCCN(C(Cc2onc(C)n2)=O)C1 Cc1ccc(Cl)c(F)c1C(=O)NC1CC(C(=O)O)C2OC(C)(C)OC12 N1(C(COCC#C)=O)CCC2(CC2NC(c2cccc(OC)c2F)=O)C1 c1(C(=O)NCC2C(NC(c3nc(CC)sc3)=O)CC2)cc(COC)cn1C c1(C(=O)NCCC2CN(C(CN(C)C)=O)C2)ccc([N+](=O)[O-])c(S(N)(=O)=O)c1 c1(C(=O)NCC(CNC(C(C)OCCOC)=O)O)sc2ncccc2c1Cl Cc1nc(O)c2cc(C(=O)NCC3CC3NC(C3CC4CCC3O4)=O)ccc2n1 C(C(CC(F)(F)F)NC(C1CCC1(C)C)=O)NC(C1(CC#C)CCC1)=O N1(C(CC2(C=C)CN(C(C3CC34CCCCC4)=O)C2)=O)CC2CCC1C(O)C2O c1(C(N(C2CCN(C(=O)Cn3nccn3)CC2)C)=O)cc(C(F)(F)F)cc(O)c1 CCCCCC(O)CC(=O)NCCC(C)NC(=O)COCCC n1(CC(=O)NCCC2(NC(c3cc(C)no3)=O)CCC2)nc(C)c2c1CCCC2 CCCCC(CC)CC(=O)NCCN(CCOC)C(c1cc(Cl)nn1C)=O Cc1ccc(C(N2CCCC(C(=O)NC3CN(C)CCC3O)C2)=O)cc1O C(=O)(C(F)CC(C)(C)NC(=O)C1=CCN(C)C1)NCc1c(C)csc1 C1(n2cc(C(C)O)nn2)CN(C(=O)C(N2CCC(C)C2)=O)CC1C C(CCCCCCC(=O)NC(CNC(C1CCC(C)(C)O1)=O)C(C)(C)C)SC C1(CCNC(=O)COC(C(c2ccc(C(F)(F)F)cc2)CC)=O)CCCCC1O c1(C(=O)NCCN(C)C(C2(C(F)(F)F)CC(O)C2)=O)ccncc1N(C)C C1(NC(C=C(CC)C)=O)CN(C(=O)CCc2cnoc2)C2(CCCCCC2)C1 C1(NC(c2ccc(F)cc2Cl)=O)CC(C2CCN(C(=O)C3=C(Cl)CCCC3)C2)C1 CCCC(CC(=O)NCCCNC(=O)NC)NC(=O)C=Cc1ccsc1 CCCC(CCCNC(c1ccc(CN(C)C)o1)=O)N=c1nc(C)[nH]s1 C(=O)(C1CCc2c[nH]nc21)NCC(CCOC)NC(c1ccc(F)c(C)c1)=O N1(C(=O)NC(C)Cc2ccncc2)CCC(F)(C(c2ccccc2)=O)C1 CC(CS(C)=O)C(=O)NC1C2CC1N(C(c1cc(N3CCCC3)nc(Cl)c1)=O)C2 c1(CC(=O)N(C(CN2CCCC(CC3CC3)C2)=O)C)cn2ccccc2n1 c1(C(=O)NCC2CCC(NC(c3c(C)ncs3)=O)C2)nc(O)c(C)s1 N1(C(c2c(C(=O)OC)csc2)=O)CCC(NC(=O)CSC)C2(CCC2)C1 C1(C#N)(C(N(CCN(C(=O)CCOC2CCC2)C(C)C)C)=O)CCCOC1 C(=O)(C1CCc2ccc(OC)cc21)NC(C)CN.CCCOCCNC(C)=O n1(CCC(=O)N2CC(C3CCCNC3)C2)cc(Cl)cn1 Cn1[nH]c(C(=O)NC2(CN(C(=O)CC3CC(CF)C3)C)CC2)nc1=O N1(C(c2c(C)nc(O)cc2)=O)CCC2(NC(=O)Cc3ccco3)CCCC12 C12(CCSC1)C(=O)N2.C(CC(=O)NC1CC1)N(C(=O)CC1OCCO1)C C1(C(N(CCC(=O)NC2(CN(C)C)CCCC2)C2CC2)=O)CCC2(CC2)C1 CC1(C)C=C(C(=O)NC(C)(C)C=CC(=O)NCCC2CCC(C)(C)O2)C1 N1(C(c2c(OC)csc2)=O)CCC(O)C(C(N2CCCCC2C)=O)C1 c1(C(N2C(CNC(CC)=O)CCCCC2)=O)ccc2[nH]c3c(c2c1)CN(C)CC3 c1(C(N(CC(C)NC(C2CN(CCOC)C(=O)C2)=O)C)=O)sc(C#N)cc1Cl C1(C)(C(N2C(C)CC2CO)=O)CCN(C(=O)C(F)C2CCCC2)CC1 C1(NC(c2c(C)onc2-c2ccccc2Cl)=O)CCN(C(=O)C(F)F)CC1F N1(C(CC#N)=O)Cc2ccccc2CC1CNC(C1CC(=O)N(O)C1)=O C(=O)(C(C)S(N)(=O)=O)NC(C1(C(N2C(CSC)CCC2)=O)CC1)(C)C n1(CC(=O)N(CCCC)CC(=O)NCc2ccccc2)c(C)ccc1C c1(COC)ccc(C(=O)N(C2CCN(C(=O)CO)CC2)C)cc1OC C(=O)(C1=CCCSC1)NC(C(C)O)C(=O)N(C1(CCO)CC1)C C=CC(C)CC(=O)NC(C1CC=CCC1)C(=O)NCc1cc(C(C)C)on1 C1(CN(C(C2CCCC2F)=O)CC)CCCCN1C(=O)CCSCC(N)=O C(=O)(C1=CCCC1C)NCC(C(=O)Nc1cn(C)nc1Cl)OC CC(F)(F)CC(=O)NC1CCC(CNC(c2ccc(NC=O)cc2)=O)CC1 S(=O)(=O)(c1cccc(=NC(C)Cc2ccc(SC)cc2)[nH]1)NC(CCC)C1CC1 c1(C(N(C)CC2N(C(COCCC)=O)CCC2)=O)cc(O)cc(=O)o1 N1(CC(=O)OC)CCN(C(=O)NCCCN2C(c3ccccc3)C(C)CC2)CC1 c1(CNC23CC(C(=O)Nc4cnc(CC)nc4)(C2)C3)ccc2ncsc2c1 N1(C(c2cnc(C)[nH]c2=N)=O)CC2(C=C(C(=O)NC(c3nccs3)C)CO2)C1 c1(C(N2CCN3CCOCC3C2)=O)cc(F)ccc1[N+](=O)[O-] c1(C(N2CC(F)CC(C(=O)NC(C)(C)CO)C2)=O)cc(F)c2cc[nH]c2c1 C1(C(=O)NCC2(COC)CN(C(=O)CC(O)CN(C)C)C2)C2CC(=O)CC12 N1(C(c2nc(C(C)OC)oc2)=O)CCCC(O)(CCNC(c2cnns2)=O)C1 N1(C(CNC(CCC)=O)=O)CCN(C(=O)CC(C(=O)OC)OC)CC(CO)C1 N1(C(C=CC)=O)CC2CCC1CC2NC(=O)CC(C)(C)O N1(C(c2nc(CCC)oc2)=O)CC(NC(C2CCC=CO2)=O)CC2(CC2)C1 c1(C(=O)NCCCC(C)NC(C2CC3C=CC2C3)=O)cnn2cc(C#N)cnc12 N1(C(c2cn(C)nc2)=O)CC(CNC(=O)Cc2cccc(OCC#N)n2)C(O)C1 C1(C(N(CC(C)C#N)C)=O)CC2CC1CC2NC(=O)CCC(N)=O n1(CC(=O)NCC2C(CNC(c3c(N)cn(C)n3)=O)C2)cc([N+](=O)[O-])cn1 C=CC(CC)C(=O)N(C)CC1CCN(C(C2CC(OCC)C2)=O)CC1 C1(C(=O)NCC(C(=O)NC2C=CCC2)N(C)C)(OC)CCOC1 c1(C(N2CCCC(CNC(C(C)c3ncco3)=O)C2)=O)cc(Cl)cc(Cl)c1 c1(C(=O)NCC(C)CNC(c2ccnn2CC(F)F)=O)cccc(Br)c1 N1(C(C(CC=C)C)=O)CCCN(C(=O)CCOCC(F)(F)C(F)(F)F)CC1C N1(C(c2cc([N+](=O)[O-])n[nH]2)=O)CCN(C(c2ccno2)=O)C2(CCC2)C1 N1(C(C2(CC)CCOC2)=O)CCCC2(CCCN2C(c2cnn(C)c2C)=O)C1 C(C(=O)NCC1(F)CCN(C(=O)Cc2c(C)cnn2C)C1)(C(C)C)NC(C)=O Cc1cccc(Cc2nc(-c3nccs3)nn2-c2ccc(Cl)nc2)c1C Cc1ccc(C(=O)NC2CC(C)CN(C(c3ccnc(C)c3C)=O)C2)cc1Cl C1(C(N(C2CCCOC2)CC)=O)COC(CNC(=O)CCCOC(C)=O)C1 C#Cc1c[nH]nc1C(=O)NCc1cncc(C(=O)O)c1 C(=O)(CS(=O)(=O)C(C)C)NCC1C(CNC(C2(OC)CCCCC2)=O)C1 c1(CC)cnc(O)c(C(N2CCN(C(=O)CN(C3CC3)CC)CC2C2CC2)=O)c1 CC(C)C(C)CC(=O)NC(C1CN(C(=O)C(O)CN(C)C)C1)C n1(CC)nc(C)c(C(=O)N(CC(C)N)C)c1C.c1(C=O)n[nH]c(Cl)c1Cl C(=O)(C(CC(F)(F)F)NC(=O)Nc1cccnc1OC)OCCCC C(=O)(CC(F)(F)F)NCCCCCN(C)C(C1CC1c1ccccc1Br)=O n1(CCCn2c3ncnc(CC(=O)NCC(=C)Cl)c3nc2)c2ccccc2c(=O)c2ccccc12 C(CCN=c1ccnc(SC)[nH]1)NC(C(CC)F)=O c1(C(=O)NC2CN(C(C3CC3c3cccnc3)=O)C2)cnc2c(F)cccc2c1 N1(C(C2CCN(C(C)=O)C2)=O)CC2CC2(CNC(c2csc(C)n2)=O)C1 C1(C)CCN(N(C2CC2)NC(CN(C(=O)OCC)C)=O)C1.C1(F)(C=O)CCOC1 C1(C(N(CCOCCNC(c2c(CC)c[nH]n2)=O)C)=O)C(O)C(=O)N(C)C1C C12(C(N(C(C#C)C)C)=O)CC(NC(C3CCCSC3)=O)(C1)C2 c1(CC(=O)NCCN(C(=O)C2=NOCC2)CC)cc(C(F)(F)F)cc(Cl)n1 CCCCC(C)C(=O)NCCOCCOCCNC(=O)Cc1csc(CCC)n1 N1(C(C2C(C)C2C)=O)CC2(CCC(CNC(c3cc(C4CCC4)no3)=O)O2)C1 c1(C(=O)NCC(CC)NC(=O)CCCc2ccc(C)s2)cnccc1C n1(CC(OCC)OCC)cc(C(=O)N(C)CCN(C)C(C2CC(C)CO2)=O)nn1 CCC(CN(CCN(C)C)C(C1CC=CC1)=O)CC C(=O)(C1CCCc2nc[nH]c21)NCc1nc(O)cc(CNC(C(C=CC)O)=O)n1 Cc1nc2ncnn2c(C)c1CC(=O)NC1CN(C(c2csc(O)n2)=O)CC1C c1(CC(N2CCC(OCCNC(c3c[nH]nc3F)=O)C2)=O)ccc2c(c1)OCO2 C1(NC(c2ccnnc2)=O)CN(C(=O)Cc2ccc(Br)s2)CCC1CO C1(C(=O)O)(NC(c2cnc(-c3ncccn3)s2)=O)CCNCC1 c1(N(C)C)cccnc1NCC=CCl.c12ccc(cc1)C(=O)NC2 C(c1ccc(F)cc1)=CCC(=O)NC(CNC(c1cc(SC)oc1)=O)C(C)C N1(C(CC2(C)CC2)=O)CC2(CC(NC(c3cn(C4CC4)nn3)=O)c3nccn32)C1 C(=O)(C(F)CC(CC)CC)NCC1C(OC)CN(C(=O)COCC(C)C)C1 c1(C(N2CC(C)N(C(=O)CCC3CCCCO3)CC2)=O)nncc2c1CCCC2 C(C(O)CC(=O)NC1COCC1CO)NC(Cc1n(C)nnc1)=O N1(C(c2c(C)cc(F)cn2)C(=O)NC2CCOC2)CCN2C(=O)C(C)CC2C1 S(=O)(=O)(c1ccc(NCCOC)c(Br)c1)NCC(OC)NC1CCN2CCCC12 C(=O)(C1=CCC(NC(C2CC(C3CC3)=NO2)=O)C1)NCCCSC c1(C(=O)NC(CC)CNC(=O)C(CO)NC(=O)C(F)(F)F)cc2sc(C)cc2s1 N1(C(C(=O)Nc2c(C)c(Cl)ccc2)CC2CCCC2)CCC(=O)N(C)CC1 N1(c2cc(O)nc(=N)[nH]2)CCC2(CC1)CC2C(=O)Nc1ccc(OCCO)cc1 C(CC(=O)NOC1CCCC1O)N(CC=C)C(C1CCOCC1)=O c1(CCC(N2CCOCC(NC(C(N)=O)=O)C2)=O)ccc2c(c1)OCCO2 C(=O)(CS(=O)(=O)CC(=O)N1CCC(O)(C(C)NC(c2ccoc2Cl)=O)C1)OC N1(C(c2c(C)noc2)=O)CCC(C(N2CC(F)(C3CC3)C2)=O)C(O)C1 C(=O)(C1=CCSC1)N1C(CCNC(C(C)OCCC(C)C)=O)CCC1 c1(C(C)C)cnn(C)c1C(=O)N(CC(O)CNC(=O)C(C)(C)CO)C C1(OC)CC2CCC1CC2C(=O)NCC(C)NC(=O)C=Cc1nccs1 c1(NC(CN(c2cccc(F)c2)C(CCNC(=O)C=CCl)=O)=O)ccccc1Br C1(C(=O)OC)CCC(NC(=O)OC(C)(C)C)CN1C(=O)NCc1cn(C)nc1I N1(C(CCc2c(C)cccc2)=O)CCC2(CC2NC(C2CCCC(=O)N2C)=O)C1 S(=O)(=O)(CC#Cc1ccccc1)NC(C1CC(C)OC1=O)=O C1(NC(Cc2ccn(C(C)C)n2)=O)CCC2CN(C(c3sccc3F)=O)CC2C1 C1(C(NC[Si](C)(C)C)=O)CC2CC2N1C(=O)C=Cc1ccsc1 N1(C(C2OCCC(C)C2)=O)CCC2(CCCN(C(c3cnc(C#N)s3)=O)C2)C1 CCN=C1NCCOCCN1.C(CCC)NOC n1(CC(=O)NC2CC(NC(Cc3cc(C)nn3C)=O)C(O)C2)nc(O)ccc1=O Cc1ccc(C)c(NC(C2CCC2=O)=O)n1 C1(SCC(=O)NCC(CN(C)C(C2(c3ccsn3)CC2)=O)O)CCCCO1 CN1CC2CCN(C(C3CCN(C(c4nn(C)cc4Cl)=O)CC3(C)C)=O)CC2C1 c1(C(N2CC(NC(C3(C#N)CC4CC4C3)=O)C2)=O)cc2c([nH]1)CCCC2 CC(C)C(C)C(=O)N(CCC(C(C)C)NC(c1ncoc1C1CCCO1)=O)C c1(COC)ccoc1C(=O)NC(C)C(C)NC(c1ncccn1)=O n1(CC)ncn(NC(=O)c2cc(C)nn2C(F)F)c1=O.C12CCCC1CNC2=O Cc1cc(C(=O)NCc2cc(C(N3CC4CC4C3)=O)co2)c(C)s1 C(=O)(C1=CCCOC1)N(C(C)CN(C)C(c1cnc(N(C)C)s1)=O)C N1(C(CSCCN(C)C)=O)CCN(C)CC1CNC(=O)CCc1nncs1 CCC(CC)(CC)C(c1ccccc1)N(S(=O)(=O)CC(C)OC)C C1(C(=O)NC)CCN(C(=O)C(CC=CC(=O)O)NC(=O)CC2CCOCC2)C1C N1(C(c2ccnnc2)=O)CCC2(CC1)CC(C(N1CC(F)(F)C(F)(F)C1)=O)C2 N1(C(C2CCCC(NC(c3cccnn3)=O)C2)=O)CCCCCC1CO Cc1oc(Cl)nc1C(=O)N(C1CCN(C(=O)CC2CCOC2C)CC1)CCO Cc1cc(C#N)cnc1N1CCC(C)C(NC(C2CC3C=CCC(C2)C3)=O)C1C C1(OC)CC(C(=O)NCC2CN(C)C2)N(C(=O)CC2CCC(=O)N2C)C1 C(C)(CNC(=O)C(O)Cn1cncn1)(CC(C)C)NC(c1nc(C)n(C)c1)=O C12(C(N(CCC(=O)N(C)CC3(C#N)CC3)CCO)=O)CCC(CC1F)C2 C1(C(=O)NC(C)COC(F)F)(NC(=O)C(c2cncnc2)C)CCCC1C C1(C(N2CC(C)C(CC(N3CCC(F)(CF)C3)=O)C2)=O)C2CC3C(C2=O)C13 c1(C(C)=O)ccc2sc(C(N3CC(O)CC3c3ccc(F)cc3F)=O)c(C)c2c1 C1(CC(=O)NC2CC(C)(CNC(c3cnc(C)[nH]3)=O)C2)CCCCC1O c1(C(=O)NC(CC)CNC(=O)COC(F)(F)C(F)(F)F)c(C)[nH]cc([N+](=O)[O-])c1=O C1(C(N2CCC(O)(C(CNC(c3c(C)n[nH]c3)=O)C)C2)=O)CN2CCN1CC2C C(=O)(CC(=O)NCC(C1CC1)NC(=O)Cc1cncn1C)OC N1(C(CC2CCCN(C)C2)=O)CC2CC(NC(c3cncnc3)=O)C(C2)C1 Cc1ncnc(C(=O)NCCC(C)N(C)C(C2CC(=O)NC2(C)C)=O)c1C C(CC(C)(C)C)N(C(C(C)N(C)C(C1CCCOC1)=O)=O)CC1CC1 CC(C)CC(C(=O)N(C(C)C)C1CC1)ONC(=O)C(C)(O)C1CC1 C1(CNC(C2(NC(C(CC)C)=O)CC(F)C2)=O)CCOCC1C C(=O)(N=c1cc(Cl)nc(O)[nH]1)Nc1ccc2cnn(CC)c2c1 N1(C(C(CC(=C)Cl)NC(C23CCC(C2)C3)=O)=O)CCn2nc(C)cc2C1 N1(C(C2C(C=C)C2)=O)CC2CC(NC(=O)COc3c(C)cccc3C)C2C1 CC(C)C(C)C(=O)NC1CCCCC1CNC(=O)C=CI c1(OCCN(C)C)cncc(C(=O)NC(C)(C)C(O)c2ccccc2)c1 c1(NCC2(CNC(c3cc(C)c(C)s3)=O)CCC2)ncnc2cnn(C)c12 C1(N(C)C(c2cnn(-c3cccc(F)c3)c2)=O)CN(C(=O)C(N)=O)CC12CC2 N1(C(c2cc(C)cc(OC)c2N)=O)CCCC2C1CCCN2C(C)=O C(=O)(N=c1cc(OC)n(C)[nH]1)C1C2(CCN(C(c3nc(OCC)oc3)=O)C2)C1 C(=O)(C1CCCCc2ccccc21)NCCOCCCNC(CN(C(C)C)C)=O C1(CC(=O)NC(CC)CNC(c2cnc(O)o2)=O)CC2(CCO1)CC2 c1(C(N(CC(=O)NCCN2CCCC2=O)C)=O)cc2cccnn2c1 c1(NC(C(c2cccc(Cl)c2)CC)=O)ccc2c(c1)oc(=O)n2C C1(NC(c2ccnc3c2CCC3)=O)CN(C(=O)CN2CCSCC2)C2(CCC2)C1 Cc1ccc(C(=O)NCCNC(N2CCCC(Cc3ccc(F)cc3)C2)=O)cc1 C1(C(C(=O)NCCC)N(C2CCC2)C2CC2)CCC2COCCC2C1 c1(C(N2C(C(=O)NC(CC)C(C)(F)F)(COC)C=CC2)=O)c[nH]c2cnccc12 N1(C(C(C)N2CCC2)=O)CCC2CN(C(=O)C3=CC(C)(C)C3)C2C1 C(=O)(C(CC)CCOC)NC(CCNC(CNC(C(CC)CC)=O)=O)C C1(C(=O)NC2C(C#C)CCC2)CC2CC1CC2NC(c1ccn(C(C)C)n1)=O C1(CNC(=O)C=CC2CCCO2)COCCN(C(c2ccc(Cl)nc2)=O)C1 C1(NC(C2C3(CN(C(=O)OC(C)(C)C)C3)C2)=O)CCC2(CC1)CC2C#N C=C1CCC(C(=O)NC2CCC(CC(=O)Nc3cnsc3)C2)CC1 C(=O)(C1CCOc2c(F)cccc21)N1CCCCC(NC(C(=O)NC2CC2)=O)C1 N1(C(C2CCN(C)C2)=O)CC2CCCC(N(C(=O)CC=C(Cl)Cl)C)C2C1 N1(C(C2N(C)CCCC2)=O)CCC2(CC(NC(=O)C=CCF)C2)C1 C1(C(=O)NCC(C)(F)F)CC(NC(c2ccc[nH]2)=O)C12CCC2 C1(CNC(C(CC)(C)CC)=O)CCN(C(=O)Cn2cnc(Br)c2)CC1(F)F C1(C(=O)NC2C(NC(c3ccn(C)c3)=O)COC2)CCOC1(C)C c1(OC)cc(C(=O)NCC(C)NC(=O)CCC(=O)c2cccs2)nn1C C12(C(=O)NC3C4CC(NC(CC(C)SC)=O)CC43)CC1COC21CCC1 c1(C(=O)NC(CCC)C2CC2(C)C)coc2c1C(=O)NCCC2 c1(COC)cc[nH]c1C(=O)NCCn1cc(C(=O)NCC2CC3(CC3)C2)nn1 C(=O)(C(O)CCCNC(c1c(OC)noc1C)=O)N(CC(CC)OC)C N1(CC)OCC(NC(C2CCC2NC(c2ccnc(O)c2)=O)=O)C1=O N1(C(c2csnn2)=O)CCCCC1C1CCCN1C(C1CCC(=C(F)F)CC1)=O CCS(=O)(=O)c1cccc(C(=O)NC2CC(n3cc(C4(O)CCC4)nn3)C2)c1 C(CC(C(=O)NCCn1ncnn1)NC(=O)C(c1cnn(C)c1)=O)=CC CC1(C)CC1(C(=O)NOCCC1CC1)NC(=O)Cc1ccon1 c1(NC(c2ccncn2)C)ccnc2ccnn12 N1(C(CN(C2CC2)CC)=O)CC2CCCC(C1)N2C(=O)C1=NOC(C)C1 c1(C(=O)NCC(CNC(c2ncccn2)=O)F)c(Cl)sc2nnsc12 C1(C2CCC2)(C(=O)NCC2(C)CCCN(C(C(C3CCC3)OC)=O)C2)CC1(F)F C1(CCC)CC(C(N2CCC(OCCNC(=O)COC(C)CC)CC2)=O)CCO1 c1(CC)conc1C(=O)NC(C(=O)N(C)Cc1ncnn1C)C1(O)CCC1 c1(C(=O)NCC(CC)NC(C2(C#C)CCC2)=O)cnn2c1NCC(C)C2 [N-]=[N+]=NC1(C(=O)NC(c2ccc(Br)cc2)CO)COC1 c1(-c2nc(C3OCC(C)C3)on2)ccc(-n2cccn2)cc1 CCCCC(CC)C(=O)NCC1(NC(=O)C(C(C)(C)C)C2CCCC2)CCCC1 C1(N(C(C(CN(CC)CC)F)=O)CC2CC2)CCN(C(=O)C(C)C(F)F)CC1 N1(C(C)=O)CCCC1C(=O)NCC12CC(NC(c3ccnn3CC3CC3)=O)(C1)C2 C1(NC(C2=NOCC2)c2n(C(CC)(C)C)nnn2)CC(C2CC2)(C2CC2)C1 c1(OC)ccc(C(=O)NCCNC(C2CCN(C)C(=O)C2)=O)c(Cl)c1 c1(CC(=O)NC(C2CCCC2)CNC(C(C)=CC)=O)cc(F)ncc1Br N1(C(C(CCC)O)=O)CC(C2CCCCN(C(=O)CC3CCC(=O)N3CC)C2)C1 C(C(C)(C)C(=O)NCc1ccc(SC(F)(F)F)s1)(OC)OC C1(NC(c2cc(CNC(C)=O)sc2)=O)CCCCC1F c1(C(N2CC(NC(C3(C=C)CCC3)=O)C(OC)C2)=O)c(Cl)nc2cc(Cl)ccn12 N1(C(=O)CC2C=CCC2)CC2CCN(C(c3c[nH]cc(F)c3=O)=O)C2C1 N1(C(COC(C(CC(=C)C)NC(C)=O)=O)=O)CCOCC12COCCN(C)C2 CC(C)CC(C)C(=O)N1CCCC(C)(CNC(c2cc(CO)ccc2Cl)=O)C1 CCC(CC(=O)N1CCC2C(NC(c3cccc(OC)n3)=O)C12)SC C1(C)(CNC(C2CC(NC(C3C(COC)CC3)=O)C2)=O)CCCO1 C1(C(=O)NCC2CN(C(=O)Cc3ccccc3)CC2(F)F)(OC)CCCCCC1 c1(C(=O)NC(CNC(c2c(C)cc(CC)o2)=O)C)sccc1S(C)(=O)=O c1(C(N2CCN(C(C(CCC)NC(N)=O)=O)C(CO)C2)=O)cnn2ccn(C)c12 Cc1cnc(NCC2(C)CCN(C(C3CCCCS3)=O)CC2)nc1S(C)(=O)=O C(=O)(C(C)(C)C(C)O)N1CC(OC)C(NC(=O)Cc2ncccc2C)C1 c1(C(C(=O)N(C(CNC(CCOCC#C)=O)C2CC2)C)C)ccncc1C C1(NC(=O)NC2C(CCC(=O)OC)CCC2)CC(=O)N(c2ccccc2OC)C1 CC1CNc2c(C(=O)NCC(C3CC3)NC(=O)COC3(C)CCCC3)cnn2C1 N1(C(C=CC=CC)=O)CC2(CC(C(=O)NCCSC)CO2)C1 n1(CCC)cc(C(=O)N(CCN(C)C(c2cc(CC)cs2)=O)C(C)C)cn1 N1(CCC)CCC(C(=O)NC23CC2CN(C(=O)C(CN(C)C)CC)C3)CC1 N1(C(CC2(CC(=O)OC)CCC2)=O)CCCC(CNC(C2(COC)CC2(F)F)=O)C1 c1(C(=O)NCc2c(F)cc(C)c(F)c2)c(F)cncc1C1=CCN(C)CC1 C1(CC(=O)N(c2ncn(CC(=O)OC(C)=O)c2)CC(C)CC)CC(C)(C)CCO1 C=C=C(C)CC(=O)N1CCC(F)(CNC(=O)CCn2cncn2)C1 N1(C(c2cc(CCCC)no2)=O)CCCCC1Cc1cn(CCCC(=O)O)nn1 N1(C(CCCCCC#N)=O)CCC2(CC1)CC2(CO)CNC(C1CCCCS1)=O CCC(CCC(=O)N1CCN(C(C2CN(CC)CC2N(C)C)=O)C(CO)C1)OC C1(CNC(Cc2c(C)n(C)cn2)=O)CN(C(c2csc(O)n2)=O)C(C)(C)C1 c1(C(N2CC(CC(=O)NC(C(=O)NC(C)C)C)OCC2)=O)ncc(F)cc1F C(=O)(CC1=CCCCC1)N1CCCCC(CCC(=O)NC2(C)C(C)CCCC2)C1 C1(C(=O)NC(CCC)C(F)(F)F)C(C2CC2)CCN1C(=O)CN1CCNC(=O)C1 C1(C(=O)OCC)(C(=O)NCCCOCc2nccs2)CCc2ccccc2O1 c1(NCC(=O)NCC(NC(C(COC)C)=O)OC)c(C(F)(F)F)ccnc1OC c1(NCc2ccc(CC)cc2)cccc(S(=O)(=O)N(C)CNC(C)=O)c1 N1(C(C(Cc2ccccc2)OC)=O)CCCC(CNC(c2cc(CF)on2)=O)C1 C1(CC(=O)NCC(C(=O)NC)(C)C)CN(C(=O)C(COC)OC)CC12CC2 C12(NC(C3(C(=O)OCC)CCC3)=O)CC(NC(c3cnccn3)=O)(C1)C2 N1(C(CCNC(N)=O)=O)CCC(CO)CC1.N12CCN(CC1)C(=O)C1CC1C2=O C(=O)(C(O)CC(C)(C)C)NCCC1N(C(CCCCCN(C)C)=O)CC(F)(F)C1 Cc1cc(C(=O)NC(C2CN(C(c3cc(C)[nH]c3C)=O)C2)C)n(C)n1 CCC(C(=O)NCC(F)CNC(=O)C=CSC)OC1CCCC1 CCCC(CNC(=O)CCC1(C)CN(C(C2CCOC(C)(C)C2)=O)C1)CCO N1(C(C2C(C(C)C)CCC2)=O)CC(C2CC2)(C(=O)N(C)CC2(F)CCC2)C1 C1(NC(C(CCCCC)F)=O)CCC2(CCCN(C(c3ccc(Cl)o3)=O)C2)C1 CC(CN1CCCC(C)C1)N=c1ccnc(N(C2(CCO)CCCC2)C)[nH]1 C#Cc1cccc(OCC(=O)NCC=CCNC(=O)C(N2CCCCCC2)C)c1 CCC(C(=O)N1CCC(CNC(c2sc(CC3CCCC3)nc2C)=O)C1)C(C)C C1(CNC(=O)CCF)COCCN(C(=O)CC2CC3CC3C2)C1 N1(C(C(c2ccc(Cl)cc2)C)=O)CCC(C)C(NC(=O)Cc2ccc(F)cn2)C1 C=CC(C)CCNC(c1occc1CNC(=O)C(c1cnn(C)c1)O)=O N1(C(CN2CC(C)(C)C2)=O)CC2(CCC(CNC(C3CC=CCO3)=O)O2)C1 c1(NC(c2ccc(Cl)c(C#N)c2)c2n(C(C)(C)C)nnn2)ccc2nncn2c1 N1C2CCC1(c1cn(C3C(C=C)CC3)nn1)CC2.C(=O)(C(C)CCCOC)OC c1(CNC(=O)C(O)CN2CCCC2=O)cc(F)ccc1Cl.C123CC(C1)(C2)NC3=O C1(NC(c2c(C)nn[nH]2)=O)CC(NC(=O)COCCC(C)C)C1(C)C CN=c1ccc(C(N2CCCC(CN(C(=O)C(O)CC(C)C)C)C2)=O)c[nH]1 C12(NC(CC3CCN(OC)CC3)=O)CCC(CNC(C3(Cl)CC3)=O)(CC1)OC2 C1(CC(=O)N(CCC(=O)N(C(C(=O)NC)C)C)C)CCCCN1C c1(C(=O)NCC2C(CNC(C3N(CC)CC3)=O)C2)ccc(S(=O)CC#N)cc1 C(=O)(C1=NNC(=O)CC1)NCC1(CNC(c2cccc(NC)n2)=O)CC12CCC2 c1(CN(C(C(CC)C)=O)C)cccc(CNC(C2(CC)CC2(F)F)=O)c1 CC(C)C(C(=O)N1CC2(NC(C34CCCC3(C(N)=O)C4)=O)CC1C2)n1ccnc1 c1(C(=O)NCC2(C)C(C)CN(C(C3(C)CCC3)=O)C2)cc(C#N)c2n1CCCC2 N1(C(C2CCC(CNC(C3(CC)CCC3)=O)O2)=O)CC2(CCCC2)C1 n1(CCC(=O)OC)cc(CC2(O)CN(C(C3(CCS(N)(=O)=O)CCC3)=O)C2)nn1 N1(C(C2(CC)CC2)=O)CC(C)N(C(C2(C)CCC2)=O)C(C)C1 n1(CC)nc(C(=O)OC(C)C(=O)Nc2ccc(CC#N)cc2)c2c1CCOC2 C(=O)(CC(C)(C)C#N)NC(C)CNC(=O)CNc1ncccn1 c1(CC)cc(Cl)ccc1C(=O)NCc1ccnc(C(=O)O)c1 C(=O)(CS(C)(=O)=O)N1CC(C(C(=O)NCCNC(C)=O)O)C1 C1(C(=O)NCC2CCN(C(C(COC)C)=O)C2(C)C)Cc2cccnc2C1 Cc1nc2cccc(C(=O)NC(C)CCNC(=O)C(c3cccnc3)O)n2n1 CCCC(C)C(=O)NCCOCCOCCNC(=O)CC1CCC(O)C1 C1(C)(CNC(c2cn(CCC)nn2)=O)CCN(C(=O)CC(=O)NC)CC1 c1(CN(C(c2ccc(C(F)F)o2)C(=O)NCc2ccc(Cl)s2)CC)ccccc1 C1(C)(C)CC(=O)OCc2cn1nn2.C1(NC(=O)OC(C)(C)C)CC(CC#N)C1 C1(C(=O)NC2C(C(N3CCN(CC=C)CC3)=O)CCC2)CCN(OC)CC1 C1(NC(c2c(C)cccn2)=O)CN(C(C2Cc3nnc(C)n3C2)=O)CC(F)(F)C1 C1(CC)CC(O)CN1C(=O)CN(C(=O)Cn1[nH]cnc1=N)C(C)C C(=O)(C1=CCN(C)C1)NCCC(C)NC(c1cnc(CC)o1)=O CC1=C(C(=O)N2CCCC(NC(=O)C=C3CCN(C)CC3)C(F)C2)CCCO1 CC1CN(C(c2nncn2C2CC2)=O)CC1CNC(=O)C(F)=CC1CC1 Cc1nn(C2CC2)cc1C(N1CCC(CO)(NC(C2CC(F)(CO)C2)=O)C1)=O N1(C(C(COCC)NC(C2CC2(C)C)=O)=O)CCC2C(=O)NCC2C1 N(C1CCCc2c(Cl)ccc(Cl)c21)C(=O)C(N1CCOC(C(F)F)C1)=O N1(C(C2C3CN(C)CC32)=O)CCC(NC(=O)C(c2ccccc2)O)C(F)C1 N1(Cc2n(C)cnc2)CCN(C(c2cccnc2S)=O)CC1 C1(C(C(=O)NCC(C)N(C)C(C2CC2(Cl)Cl)=O)C2CC2)CCCCC1 C=CCC(C)(CC=C)NC(=O)C(CC)N(C(=O)C(F)F)C n1(CC)nc(C)cc1C(=O)N(CCC(C)NC(=O)C(c1ccnn1C)O)C c1(OC)noc(C2CC2)c1C(N1CCC(N(C(=O)CCC2CCCO2)C)CC1)=O c1(CC(N2C(CCNC(CCC3C(C)C3)=O)CCC2)=O)ccc2c(c1)CCCC2 c1(C(CNC(c2n[nH]cc2Br)=O)NC(CC=C=C)=O)ccccc1F N1(C(CC(CCC)(C)O)=O)Cc2ccc(CNC(c3n[nH]cc3CC)=O)cc2C1 C(=O)(C1CC=Cc2ccccc21)N1CCCC(F)(CNC(=O)Cc2cnns2)C1 c1(C(N(C2CC(C#N)C2)CC(=O)NCCc2cnc(C)[nH]2)=O)cc[nH]c(=N)n1 c1(CC)oc(C(=O)O)cc1S(=O)(=O)NC(C)C(=O)Nc1ccc(F)cc1 C12(CCCCC1)CC(=O)NC2.C1(C(=O)OC)(C(=O)N(C)C)CNC1 C1(C(N2CCN(CC(C)NC(c3ccc[n+]([O-])c3)=O)CC2)=O)(OC)CC2CCC1C2 CC(CC(=O)NC1(CF)CCN(C(=O)CN2CCCCC2=O)C1)C(F)(F)F c1(SC)ccsc1C(=O)N(CC(C)NC(=O)CCc1nc[nH]n1)C(C)C C1(CCNC(C2C=CCCC2)=O)CN(C(c2sccc2Cl)=O)CCO1 c1(CCCN2C(C)(CO)CCC2)ccc(F)c(F)c1 CC(O)CC(C)N=c1cc(NCc2ccc(CO)c(F)c2)nc(C(F)(F)F)[nH]1 N1(C(C2(C)CCCN(C(C3(C)CC3)=O)C2)=O)Cc2ccc(F)cc2C1 N1(C(C(C2CC2)OCC)=O)CCOC2(C1)CN(C(C1CC1C(F)F)=O)C2.C1(C)CC1 N1(C(c2c(C)cc[nH]2)=O)CCCC(NC(C23CC(C2)C(C)(C)O3)=O)CC1 C12(C(=O)NC3(COC)CC=CC3)CCC(CC1)N(C(=O)CC1(O)CCCOC1)C2 O=C(CC1NC(=O)c2ccccc21)NCC1CCN1C(c1cc(O)no1)=O C1(C(=O)NCCC(=O)NC)CCN(C(C2CC(C(C)C)C2)=O)CC1 C#CC1(NC(C2(CC)C=CCN2C(=O)C=C(C2CC2)C2CC2)=O)CCCCC1 CC1(C)CC(CNC(c2cncc(F)c2Cl)=O)CN(C(=O)CCCS(N)(=O)=O)C1 Cc1cc(C(=O)N(CC(C)O)CCNC(=O)C(C)(F)F)cc([N+](=O)[O-])c1Cl c1(C(=O)NC(CN(C(=O)CC2CC2(Cl)Cl)CC)C)cc(N)ccc1[N+](=O)[O-] S(=O)(=O)(c1csc(C(=O)N(CC(C)NC(=O)Cn2ncnn2)C)c1)NC N1(C(C(C)SC)=O)CCc2c(CNC(=O)C(N3CCCCCC3)C)cccc2C1 c1(OCCOC)ccc(CN(Cc2ccccc2)Cc2nc(C)no2)cc1 Cc1ccc2c(cnn2C)c1-c1csc(NC(C2CC23CCOC3)=O)n1 CC1(C#N)CCC(N=c2cc[nH]cc2S(=O)(=O)NCC2CN3CCN2CC3)CC1 CC(C)CC(=O)N(CCCC1CCNCC1)CCO C1(c2n(C3C(F)(F)C3)ncc2)NC(=S)N(C2CC2)C2=C1C(=O)NC2c1ccccc1 Cc1cccnc1C=Cc1nc(C(=O)NNC(=O)Cn2cnc3ccccc23)no1 C(=O)(C(CN(C)C)C(C)C)N1CC(OC)C(NC(C2(n3cccn3)CCC2)=O)C1 c1(CC(=O)N(C2C3CN(C(CC4CN(C)C4)=O)CC32)C)c[nH]c2cc(F)ccc12 c1(C(=O)NCC2N(C(C=CC=CC)=O)CCCCC2)cc2cccnc2o1 N1(C(C(N)=O)=O)CC=CC(NC(C2(O)CCC2)=O)C1 c1(-c2cc(OC)cc(COC)c2)ccc2nnc(C(N3CCOCC3C)=O)n2c1 c1(C(N2CC(O)(C(C)NC(=O)C(C)n3cncn3)C2)=O)cc(CO)n(C)n1 C(CO)(CCCCNC(=O)C(F)=C1CCCC1)NC(=O)CCC1CCC(O)CC1 C(CC(C)C)(C(=O)N1CCC(F)C(F)C1)ONC(=O)C1(CC(C)C)CC1 c1(C(C2CC2)NC(CN(CCOC)C(c2cnn(CC)c2)=O)=O)ccc(C)cc1 CC(C)CC(O)C(=O)NCCC1(O)CCCN(C(=O)C(F)(F)COC(C)C)C1 C1(C(=O)NCC23CC(NC(c4cnc(C)s4)=O)(C2)C3)CCCN2CCCCC12 C(=O)(C(O)C1=CCCCC1)NCC(CNC(c1ccn(CC(C)C)n1)=O)CO C(=O)(CC(C(F)(F)F)NC(=O)C(C1CCCCC1)F)NC1(CC=C)CCCCC1 c1(CC(=O)OCC2(COC)CCC2)cccc(F)c1Nc1ncccc1OCC c1(C(=O)NCC2CC(OC)CN2C(C2OCCC2C(C)C)=O)cc2occc2[nH]1 C1(NC(C(C)(C)OC)=O)CN(C(=O)C(C(C)C)n2ccnc2)C(C)(C)C1 c1(C(=O)NCC(CC=C)NC(c2c(Cl)cnn2C)=O)ccccc1CC C(=O)(C#CC(C)(C)C)NCCCN(CC(=O)OC)C1CC1 CCCCCCC(C)C(=O)NC1CN(C(=O)C=Cc2cnc(C)s2)CC12CCC2 C1(C(N2CCN3CCOCC3C2)=O)CC2CCCCC2N1Cc1ccccc1Br C(=O)(CC(C)(C)CCC)NC(C1(O)CCN(C(C2(CC=C)CCOC2)=O)CC1)C CC(C)CC(O)C(C)C(=O)N1CC2(CCC2NC(=O)CCCn2cncn2)C1 N1(C(C(C)(C)OCC)=O)CC(NC(=O)CP(C)(C)=O)C2(CCC2)C1 C1(C)(CC(N2C(COC)CC2)=O)CCN1C(c1cnnn1C)=O N1(C(CCC2N(C(c3c(C)cc[nH]3)=O)CCCC2)=O)CCOCC(O)C1 C1(NC(CNC=O)=O)CN(C(=O)CCC2CCOC2)CC1Cc1ccccc1 Cc1cc(CN=c2[nH]c(C(=O)NCCCN3CCCC3)cs2)cc(Br)c1 CC1(C)CC(NC(c2c(F)cccc2Cl)=O)CN(C(=O)C(C)(O)C2CC2)C1 Cc1cc(Nc2cccc(C(F)C(F)(F)F)n2)c2ccc(F)cc2n1 N1(C(C(CCC(C)C)=O)=O)Cc2n[nH]cc2C1C(=O)NC1CCn2ncnc2C1 c1(N(C)C)nc(Cl)c(C(N2CCOCC2CNC(=O)CCc2cnc(O)[nH]2)=O)s1 C=CCC(C)(C)CC(=O)NCC(C)CN(C)C(C12COC(CO)(C1)C2)=O N1(C(C(=O)N(C)C)=O)CCCC(CNC(=O)CNC(c2ccncc2)=O)C1 N1(CCN(C(c2cccc(C)c2)=O)CC)CCC(S(=O)(=O)F)CC1 CC1CC(C(=O)NC2(CNC(c3cc(O)nn3C)=O)CCC2)CCN1C C1(CCNC(CSCC(C)C)=O)CCN(C(=O)C(C)(C)n2ccnn2)CC1(F)F c1(OC)ccccc1OCC(N1CCC(NC(c2scnc2Cl)=O)C1)=O C1(CCC=C)(C(=O)Nc2cscc2C)CN(C(=O)CCOCC(F)F)C1 CC1(C)CN(C(c2ccoc2)=O)CC(CNC(C2(C)CCCS2(=O)=O)=O)O1 C=CC1CCCN(C(=O)C(CCSC)NC(=O)COCCOC)C1 C12(C(=O)NCC(CC)NC(C3CCC(=O)N(C)C3)=O)CCCN1CC(OC)C2 C1(CC)CN(C(c2cnc(Cl)c(C)c2)=O)CCN1C(c1cc(I)ccc1C)=O C1(C(N)=O)COCCN1C(C12CC1CN(Cc1ncccc1F)C2)=O C1(CC)CCC(C(=O)N(C)CC2COCCN2C(C2CCOC2)=O)CC1 c1(C(N2CCC(C)(CNC(=O)C(F)C3CC3)C2)=O)cc2ccccc2s1 c1(CC(=O)NCC(C)N(C(c2c(CC)onc2)=O)CC)cn2cc(F)ccc2n1 CCCCC(O)C(C)C(=O)N(C1CC(CC(N2CCC2(C)CCO)=O)C1)CC c1(C(N(CC(C)O)CCNC(=O)CC(C)(C)C)=O)cnn2c1OCC2 C(c1c(Cl)cccc1Cl)=C(C)C(=O)N(CCCNC(=O)CCc1cn(C)nn1)C C1(C(=O)NCC2C(NC(c3cccc4c3COC4)=O)C2)CCc2ccccc2C1 c1(C(N(C)CC2CN(C(c3scc(OC)c3)=O)C2)=O)ccc(F)c(N(C)C)c1 c1(CNc2ccc(C(C(F)F)F)cn2)cccc2ncnn12 N1(C(Cc2c(C)n[nH]c2C)=O)CC(NC(C2CC(CF)C2)=O)C(C)(C)C1 N1(C(C2C(C(=O)OCC)CC2)=O)C(C(N2CCC(O)(CC)C2)=O)CCC12CC2 c1(C(=O)NCC2(O)CCCN(Cc3c(C)ccc(O)c3)C2)cccc(C#N)c1Cl c1(C(=O)NC(C(C)NC(c2nc(CC)sc2N)=O)C)c(C)nn(C(C)C)c1C c1(C(N(CCCN(C(CC2C(C)C2)=O)C)C)=O)cn2c(n1)COCC2 N1(C(C(=O)OC)C)CCOCC(C(=O)N(c2ccc(C)cc2)C(C)C)C1 C1(C)(C(=O)NCCCCC(C)NC(C(C)CCO)=O)CCN(C)C1=O c1(CNC=O)ncn(CC2CNCCO2)n1.c1(C2(C(=O)NC)COC2)ccccc1 c1(C(=O)NC2C3CC(CNC(CC(=C)C)=O)(C3)OC2)ccc2c(c1)CC(C)O2 C1(CNC(C(CC(=O)OC)C)=O)CC2CCC1N(C(=O)CC1COCCN1C)C2 Cc1[nH]c2ccccc2c1C(=O)NC1CCC(CNC(C2CCCC2(C)O)=O)C1 C1(OCC(=O)NC(CN(C(c2c(CC)scc2)=O)C)CC)CCCCCC1 c1(C(=O)NC2C(NC(C3NC(=O)OC3)=O)CCCC2)cc(C2CC2)nc2ccnn12 C1(C(=O)NCc2c(CC)nccn2)CCCC(NC(=O)C(C)OC2CC2)CC1 c1(C(=O)NCC(CCC)CCC)c(Cn2cc(CC(C)O)nn2)nn2c1CCC2 c1(C(N2CCCC(CCNC(=O)C(O)C(F)F)CC2)=O)cc2ccc(F)cc2o1 C1(NC(C(C=C=C)C)=O)CN(C(c2cccnc2SC(F)F)=O)CC12CC2 c1(CC2(C(=O)NC3CCCC(N(C(C(C)N(C)C)=O)C)C3)CC2)ccc(F)cc1 C1(CNC(C(C=C)C)=O)CC(C)N(C(c2cn(C(C)C)cc2C)=O)C1 C1(NC(=O)CC2CCC3CC3C2)CC2(C1)CN(C(=O)C=Cc1cncc(O)c1)C2 CN1CCC(CC(N2CCC(CNC(=O)CN3CC(C)(C)C3)C2)=O)C1 c1(C(N(CCOCCCNC(C(CC)(C)CO)=O)C)=O)n[nH]c2ccc(C)cc12 N1(C(C(C(C)C)F)=O)CCC2(CCCC2CNC(=O)C=C2CCCC2)CC1 C(=O)(CC(O)C(C)(C)C)N1C(CCN(C(C2CC(=C)C2)=O)C)CCCC1 Cn1c(O)nc2c(C(=O)NC3CCC(P(C)(C)=O)C3)cccc12 Cc1nnc(NC2CCCCC2CNC(c2n[nH]cc2Br)=O)c(C#N)c1C c1(C(C(=O)NCCCF)N(C)Cc2cncs2)ccc(F)c2c1CCC2 C1(C(=O)NC(C)CCCNC(=O)COCC(C)(C)C)CC2(C1)NC(=O)NC2=O CCCCCCC(F)C(=O)NCCC1(C)CCN(C(=O)Cc2ccc(F)cc2)C1 C(c1cccc(O)c1)=CC(=O)NC1CC2CC1N(C(c1cc(O)nc(O)n1)=O)C2 C1(CC(=O)NC(CCC)CO)CCCN(C(=O)CN2CCOCC2)C1 O=C(CC1CC(C(F)(F)F)CO1)NNC(=O)N1CCC(c2cc[nH]n2)C1 O=C(CCC(F)(F)F)NC(C1(O)CCCCC1)C(=O)NC1(CF)CCCC1 Cc1cc(Br)cc(CN2CCC(N(C)C(c3cnc(O)c(Cl)c3)=O)C2)c1O C1(CC)CC(CC(=O)N(C2CCCC2)CCNC(=O)C(C)=C2CCCC2)CCO1 C1(C(=O)NC2(CC=C)CN(C(=O)Cc3n[nH]c(=NC)s3)C2)CCN(C)C(=O)C1 C1(CNC(C(C(C)C)SCC)=O)CCCCCN1C(=O)C1=CCCOC1 c1(OCCCOC)ccc(C(N2CC(NC(C3(CO)CCC3)=O)C3CC23)=O)cn1 N1(C(C2C(C)(Br)C2)=O)CC2(C1)C(NC(=O)Cc1cccc(F)c1)CCS2(=O)=O N#Cc1cncc(NC(=O)CC2CN(C(=O)C(c3cccc(Br)c3)O)CCO2)n1 C1(CC=C)(NC(C2CC2(C)C(F)F)=O)CCN(C(=O)CSc2nncn2C)C1 c1(OC)nn(C)cc1NC(C1COCCN1C(=O)CCc1cnn[nH]1)=O C=CC1(C(=O)NC23CC4CC(CC2C4)C3)CCN(C(=O)C#CC2CC2)CC1 c1(CN(C(C(=O)NC2C(C)CSC2)=O)C)nnc2n1CCNC2=O c1(CN(C)CC2CCN(C(CC(C)C3CC3)=O)C2)ccc(-n2ccnc2)cc1 c1(CC(N2CCC(N(C)C(C3CCN3S(C)(=O)=O)=O)C2)=O)cc(F)cc(Cl)c1 c1(C(=O)NCC(CC)(C)NC(c2cnsc2)=O)cc(C)c(C)cc1Cl c1(C(=O)NC2CC(C)N(C(c3ccn(O)c(=O)c3)=O)CC2)cnn2ncccc12 C1(C(=O)NCC(C(CC)C)OC)CCC2(CCOCC2)N(C(=O)OC(C)(C)C)C1 Cc1ccc(NC(=O)OC(C)(C)C)cc1CNC(=O)CCC(=O)c1cccnc1 C1(C(N2CCC(Nc3ncnc(O)c3Br)C2)=O)CC2(C1)CS(=O)(=O)C2 Cc1scc(C(N2CCC(C)(NC(=O)CCCC3CCCO3)C2)=O)c1C C12(NC(COCC(C)C)=O)CC(CNC(=O)COCC(c3ccccc3)C)(C1)C2 C(=O)(CCCN(C)N=O)NCCCN(C(=O)Cc1cnn(C)c1)C(C)C N1(C(=O)NC(C(C(C)C)CO)(C)C)CC(CO)CC12CCOCC2 Cc1ccc(CC(=O)NCC2CCN(C(=O)CSc3nncs3)CC2)cn1 C1(C(N(C(C)CN(C)C)CC)=O)CCN(C(=O)CCOCC(C)C)C1C Cc1ccc(C=CC(=O)NC2CCCC2NC(c2ncoc2C2CC2)=O)cc1C c1(C(N(C2CC(=C)C2)C)=O)conc1CNC(C1(CCC)CCC1)=O C1(CNC(C(C)SC)=O)N(C(c2cccc3oncc23)=O)CCCC1(C)C c1(C(=O)NCC2CC(C(C)C)OCC2)ccc(S(=O)(=O)NC2(C3CC3)CC2)cc1 N1(C(c2c(C)cncc2)=O)CCC2CCC(C1)N2C(=O)CN1CC2CC2C1 CCCC(C)(CCC)C(=O)N1CCOC(CC(N2CC(CO)C(O)C2)=O)C1 c1(CCC(=O)NCC(CO)NC(CC2C(C)C2)=O)nc(-c2cccs2)no1 c1(C(=O)NC(C(C)NC(CC(n2ccc(C)n2)C)=O)C)ccc2c(c1)OCCO2 c1(C(N2CC(NC(C3CCCO3)=O)CC(C)(C)C2)=O)ccc2c(O)n[nH]c2c1 C1(CCNC(CCCOCC=C)=O)CN(C(c2cnc(CC)s2)=O)CCS1(=O)=O C=CCC(C)(C)CC(=O)NC1CCN(C(=O)CCCc2ccc(Cl)cc2)CC1F Cc1ccc(NC(=O)NC2CCC2c2ccccc2)nc1C1CC1 c1(OC)ccc(C(=O)NC2CC2CNC(=O)CN2CCC(C)C2)cc1O c1(C(N2C(CNC(c3c(C)cn(C)n3)=O)CC3(CC3)C2)=O)ccc2cccnn12 c1(NC(C2C(NC(c3cn(C)nc3C(F)(F)F)=O)C2)=O)cc(Cl)c(Cl)cc1I CCC(CC)(C(=O)NCC1(NC(=O)Cn2cnnc2)CCC1)OC C1(NC(c2c(C)nc(CC)o2)=O)CN(C(c2ccc(C)cc2O)=O)C2(CCC2)C1 c1(NC(C2CC(NC(C3CCCO3)=O)C2)=O)cc2ccccc2c(Br)n1 Cc1cc(C(N2CCN(C(c3c(C)cnn3C)=O)CC2C)=O)c(O)c(C)c1 C(=O)(C1=CC2(CN(C(C3CCC(F)C3)=O)C2)OC1)NCCc1n(C)cnc1 C(=O)(CC(C)CC(C)C)NC1C(NC(CCCc2nnc(C)n2C)=O)CCC1 C(C(CCC)C(=O)N(CC(C1CC1)OC)C)NC(COCC(=C)C)=O N1(C(c2c(OC)ccc(OC)c2)=O)CC(C)CN(C(=O)CSCCN(C)C)CC1C c1(CNC(C23CC(C(=O)Nc4cnc(Cl)cn4)(C2)C3)=O)ccc([N+](=O)[O-])cc1 C1(NC(c2c(Br)ccc(N)c2)=O)CC2CCC(C1)N2C(C1CC2(CSC2)C1)=O N1(C(c2c(C)sc(O)n2)=O)CCCN(C(c2cc(N)cc(O)c2)=O)CC1 N1(C(CSC)=O)CCOCC1CC(=O)NCCNC(C1COCCN1C(C)=O)=O N1(C(CSCCCC)=O)CCC(CNC(C2(OC)CCOC2)=O)C1C(C)C c1(C(N(C(C)C)CCNC(C2CC2c2ccccc2)=O)=O)cc(C(F)F)nn1C CC1=C(C(=O)NC2CCN(C(=O)Cc3ccc(F)cn3)C(C)C2)CCS1(=O)=O CC1(C)CCCCC1CC(N1CCSCC1CCNC(=O)C(C1CCCCC1)O)=O c1(CN(S(=O)(=O)CC2CCCC(C(F)(F)F)O2)C)c(F)cccc1F C(=O)(C1CC(=O)Nc2cc(F)ccc21)NC1(C)CN(C(C2COC(=O)N2C)=O)C1 c1(NC(C)C)cncc(C(=O)NCC2(C)CCN(C(c3cc(CF)on3)=O)C2)c1 c1(C(N(CCCCCNC(COC(CC)C)=O)C)=O)cncc(CO)c1 O=C1CC(C(=O)NCc2n[nH]cc2C(N2CC3CCCCC3C2)=O)C2(CCC2)C1 c1(CCC(=O)NCC2(O)CCN(C(c3cc(F)cs3)=O)C2)ccccc1Cl C12(CNC(C3(OC)CCCC3)=O)CC(CN(C(=O)CC3CC(SC)C3)C1)C2 CC1(C)CCCC(C(=O)NC2CC(C(N3CC(F)(F)CC3C(N)=O)=O)C2)C1 C1(NC(C2CC(OC)C2)=O)CN(C(=O)CC(C)c2ccccc2)CC12CC2 Cc1cc(C(N2CCC(C(C)NC(=O)COCC3CC3)C2)=O)ccc1O C(=O)(C(O)C(C)(C)CC)NC(CN1CCN(C(C(CC=C)(F)F)=O)CC1)C N1(C(CCC(=O)OC)=O)CCc2c(NC(=O)Cc3[nH]cnc3C)cccc2C1 c1(C(=O)NC2C(NC(C3(C)CCCCC3)=O)CCC2)cccc(C#N)c1 C1(C(C)NC(C(COC)O)=O)CN(C(=O)Cn2cnnc2O)CCO1 c1(C(N2CC(COC)(CNC(=O)C(CO)N(C)C)C2)=O)cc2n(n1)CCCO2 CC1(C(=O)NCC2(CNC(c3cscn3)=O)CC(F)(F)C2)COC(=O)C1 CCC(CC(=O)NC(c1n[nH]c(CC)n1)C)NC(C1CCN1CC)=O C=CCC(CNC(c1cc(C#N)cn1C)=O)C(=O)N1CCC(C(=O)OC)O1 Cc1sc(C(=O)NC2(C3CCCN3C(c3cc(O)n(C)n3)=O)CC2)nc1O Nc1ccc2nc(N3CC4CC(NC(=O)Cc5cnoc5)CC3C4)sc2c1 CCCC(C)CCN=c1ccnc(NC(c2nccn2CC)C)[nH]1 N1(C(C(CN(C(c2c(CC)cncc2)=O)C2CC2)C)=O)CCC2(CC1)CC2 Cc1cc(=O)n(C)nc1C(N1CC(Oc2ccc(Cl)c(F)c2)C1)=O C12(C(=O)NC3(C#C)CC3)CC(C)(CN1C(=O)C(C(C)C)SC)C2 C1(C(N2CCC(O)(CC)C2)=O)CN(C(C2CC3CCC2CC3)=O)CC12CCC2 c1(C(C)C)cc(C(N2CCN(C(=O)C(F)C(C)(C)O)CC2C)=O)cc(F)c1 O(NC(=O)C(C)N(C)C(c1c[nH]nc1CC)=O)CCC C1(C(N2C(CCNC(=O)C(F)=CC3CC3)CC(F)(F)C2)=O)CCc2nn[nH]c2C1 CCCC(CNC(c1ccnc(C)n1)=O)C(=O)N(C)CC1(OCC)CCC1 Nc1cc(C(N2CCOC(CNC(C3Cc4nncn4C3)=O)C2)=O)cnc1Cl C(=O)(C1CCCc2sccc21)NC(C(C)NC(C(C)C)=O)CO C=C(C)CCC(=O)N1CCN(CC2CCCN(C(C3CC3C(C)C)=O)C2)CC1 N1(C(CN(C(C(COC)OC)=O)CC2CC2)=O)CC2(CCC(=O)O2)C1 CC(C)P(=O)(CC(=O)NCCC1CN(C(C2CCn3ncnc3C2)=O)C1)C(C)C N1(C(C(=Cc2ccc(F)cc2)C)=O)CCC2(C1)CN(C(=O)Cn1nnc(=N)[nH]1)C2 N1(C(C(C)n2cnnn2)=O)CCC(CCNC(=O)C(c2cccc(O)c2)C)CC1 c1(NC(C2CCN(C(C(COC)OC)=O)C2(C)C)=O)cccc2cccnc12 C=C1CON(C(=O)COC2CC(NC(=O)C(C)(CCC)OCC)C2)C1 C1(NC(=O)COCC2CC2)CCCCC1.C12CC(C1)NC2C C1(CC)(NC(=O)NCc2cnn(-c3ccccc3)n2)CCCN(C(C)=O)C1 C1(C(=O)OC)CN(C(=O)Nc2cc(C)ccc2Br)CCC1(F)F c1(C(=O)NCC2(C(N)=O)CN(C(c3cnsn3)=O)C2)ccc2c(c1)C(=O)NC2 N1(C(C(CSC)C)=O)CCCC2(C1)CN(C(C1(C#N)CCCOC1)=O)C2 c1(N(C)CCOCCNC(c2ccc(S(N)(=O)=O)o2)=O)nc2c(F)cccc2o1 CC(C)C(C#N)C(=O)NCC1CN(C(=O)CCCNC(=O)C2CC2)CC1C c1(OC(C(C)(C)OC)=O)ccc(NC(C2C(C(=O)OC)C2CC2CC2)=O)cc1 Cc1ncc(C(=O)NCc2cc(C(=O)NC(C)Cc3nncn3C)no2)c(=N)[nH]1 N1(CC(N2CC(NC(=O)OCC)C2)=O)CCN(C)CC1.C12CCCN1C2 Cc1cc(C(F)(F)F)c(C(N2CC3(C2)CN(C(C2(C)CC=CC2)=O)C3)=O)c(O)n1 CCC(C)(C(=O)Nc1ccc(NC(C2CC3(CCCC3)CO2)=O)c(C)c1)C(F)F c1(C(N2CC(O)(C(C)NC(C(C)C3CCCC3)=O)C2)=O)ccc([N+](=O)[O-])cn1 Cn1cncc1C(=O)NC1(CO)CN(C(C2CCNC2=O)=O)C1 c1(C(C)=O)cc(-c2csc(NC(=O)CCC3CC3)n2)n(C)n1 C12(CNC(C(C(CC)C)C)=O)CN(C(=O)C3=COCCO3)CC(F)(C1)C2 CCCCCC(O)C(=O)NC1CC(NC(C2(C(C)C)CCC2)=O)C1 Cc1cn2ccnc(C(=O)NCCC(C)N(C(=O)CN3CCC3C)C)c2n1 C(c1nccs1)=CC(=O)N(C(CC)CNC(C1(c2ccsc2)CC1)=O)C N1(C(CC2N(CC)CCOC2)=O)Cc2ccccc2C1CNC(=O)C(C)COC c1(C(N2CC(CN(C(C(CCC)OCC)=O)C)OCC2)=O)cc(Cl)c(Cl)cc1N N1(C(c2c(C)cccn2)=O)CCC(NC(c2cccs2)=O)C(C(C)C)C1 C(=O)(CC(C(F)(F)F)NC(C1CCOC1(C)C)=O)N1CCC(CCCC)C1 C1(NC(c2c(F)ncc(OC)c2)=O)CCCC12CN(C(=O)CCCSC)C2 c1(C(N2CC(C(=O)Nc3ccc(F)c(Cl)c3)C2)=O)cc2cccc(Cl)c2s1 O=C(CCCCO)NCC(=O)NC1CCCC1.C12CCCC1NCC(=O)NC2 C1(C(=O)NC2(CC)CCOC2)C2CC3C(C2NC(=O)CCCNC(N)=O)C13 c1(OC)cc(NC(C2CCC3(CCC3)CN2)=O)c(C)cc1C c1(CC(C)Nc2nccc(N3CCSC(C(F)(F)F)C3)n2)ccc(C#N)cc1 N1(C(N)=O)CCCC1C(=O)NC1CC(CCNC(=O)C(c2ccccc2)O)C1 CC1OCCCC1C(=O)NCC1C2CC1N(C(c1cnccn1)=O)C2 N1(C(C(CC)C)=O)CCOC(CNC(=O)CC2CC3(COC3)C2)C1 C12(C(=O)NCC3(F)CCC(NC(C4CC(C)OCC4)=O)C3)CCC(O)(CC1)CC2 c1(C(=O)NC(C(=O)N(CCCCO)CC)c2ccoc2)coc(N(C)C)n1 N1(C(C2(COC)CC2)=O)CCCC2(CCN(C(=O)C#CC3CCCOC3)C2)C1 c1(CC(=O)NCCN(C(=O)C(C)C(F)(F)F)CC(C)O)cc(O)nc(O)n1 CCCCCCCCNC(N1CC2CC2(CN(C(c2ccc(Cl)cn2)=O)CC)C1)=O c1(C(C(=O)NCCCOC)N(CC(C)OC)C(C)C)cc(C)cc2c1CCC2 N1(C(C2CC(F)CN2Cc2cc(C(F)(F)F)ccc2Br)=O)Cc2ccncc2C1 c1(-c2ccc(C(=O)NCC(CNC(c3c(CC)scn3)=O)O)s2)ccc(Cl)cc1 C(=O)(C1Cc2ccc(F)cc21)N(CCCNC(=O)Cc1ccoc1)CCO c1(CC(=O)NC2C3CC2CN(C(=O)CC2C=CCC2)C3)ccc2c[nH]nc2c1 CS(=O)CCC(O)C(=O)NCC1CN(C(=O)CC2(C(F)F)CC2)C1 c1(C(N(C)CC2OCCN(C(C(CCC)O)=O)C2)=O)nn(C)c(=O)cc1C CN1N=C(C(=O)NC(c2ccnn2C)C(=O)NCC2(C)CCOCC2)CCC1=O C(=O)(C#CC1(C(F)(F)F)CC1)NCC(CNC(c1cc(C)ncc1)=O)O C1(C(=O)NC(C=C)(C)CC)CCC(NC(=O)CC2(C)CCCCC2)CC1 Cc1ccc2c(c1)CN(C(C1CCC(NC(=O)CC3(C#N)CC3)C1)=O)C2 C1(CC)CN(C(=O)CCc2ccc(F)cc2F)CCC1NC(c1csc(O)n1)=O C1(C(=O)NC(C#C)(C)C2CCCO2)CCC(CNC(=O)CCc2nc[nH]n2)C1 c1(C(=O)OC)c(F)cccc1NNC(=O)c1ccc(Br)c(F)c1 C1(C(=O)NCCCN(C(C2(CO)CCCO2)=O)CC2CCCC2)(OC)CCCC1 c1(NC(C2CCC(C(CC)(C)C)CC2)=O)cc(C(=O)OC)ccc1P(C)(C)=O C(=O)(C(C)S(=O)(=O)Cc1ccc(C#N)cc1)N1CCC(N(C)CC)CC1 c1(C(=O)NCCN(C(=O)C(C)(C)F)CC)cc(-c2ccccc2)oc1C CC1(C)CN(C(c2n[nH]cc2Cl)=O)C(CNC(=O)C(C2(O)CCCC2)F)CO1 c1(C(=O)NC2CC(C)(NC(=O)Cn3cnnc3O)C2)c(F)cc(Cl)cc1F C(=O)(C(C)(C)CC(F)(F)F)NCC(c1c(C)ncs1)n1cc(C2(CO)CC2)nn1 C(=O)(C(CC(=C)C)NC(C1CCC(=O)N(C)C1)=O)NCC(C#C)CC C1(CC)CCN(C(=O)C=CC(C)NC(c2ncoc2C2CC2)=O)CC1 c1(CC)cncc(Cl)n1.C12(COC1)C(=O)NCCOC1CN(C1)C2=O N1(C(c2scc(C)c2)=O)CCCC1C1CCCN1C(=O)CCN(C)CCO c1(C(N(C)CCNC(c2cc(-c3cn(C)nn3)on2)=O)=O)nn(C)cc1Cl C1(NC(CCC=C)=O)CCC(C(=O)Nc2cnc(C(C)C)nc2)CC1 C12(C(=O)NCC(=O)NCC(=O)NCCCc3ccccc3O)CCCCC1C2 c1(C(=O)NCC2CCC2C(=O)NCC2CCCO2)cccs1 C(=O)(C1Cc2c(Cl)cccc21)N1CC2C(NC(=O)CC3CCC3)(C2)C1 c1(NC(N(C(CC)C)C)=O)cnn(CCOC)c1 C1(C)(CNC(C2(C(=O)OCC)CCC2)=O)CN(C(=O)C(O)C(C)CC)CC1C Cn1ncc(C(=O)NC2CCC2NC(=O)C(O)C2CC2)c1Br N1(C(C(CN(C)C)O)=O)C2CCC1(CNC(C1CCC(=O)N1)=O)CC2 C1(CNC(CC2C(C(=O)OCC)C2)=O)CC(F)CN1C(c1ccsc1C)=O Cc1nnc(O)c(C(=O)N(C)CC2(NC(=O)C(C)SC(F)(F)F)CC2)c1C c1(C(=O)NC2C(NC(c3cc(OC)nn3C)=O)COCC2)cccc2nccn12 C1(C)(CCC)CCCN(C(C2(C)CN(C(=O)Cc3cnnn3C)CC2C)=O)C1 C1(CC=C)(CNC(=O)C(=O)Nc2ccnn2CC2CCOC2)CCOCC1 C1(CCCC)CCC(N=c2[nH]c(Cl)nc3c2CC(C)CC3)C1 CCC(C#N)C(=O)NCCC1CC(NC(=O)C=Cc2cn(C)nn2)C1 C1(CC(=O)OC)C2CN(C(C3(N)CCC4CC34)=O)CC12 c1(C(=O)NCC(C)CN(C)C(C2(O)CC2(C)C)=O)ccccc1N(C)C c1(C(N2CC(CNC(c3cncc(C)n3)=O)C2)=O)nc2n(c1Cl)CCCC2 c1(C(=O)NC2CN(C(C=COCC)=O)C(C)(COC)C2)cc2ccccc2o1 C(=O)(C1CCc2cccc(OC)c21)NCC(C)(CO)NC(CS(=O)(=O)NCC)=O N1(C(C=Cc2cccc(OC)c2)=O)CC(NC(=O)CC2(C#N)CC2)C(C2CC2)C1 C1(C(=O)NC(C(C2CC2)OC)C)CCC=CC1NC(=O)Cn1cnnc1 N1(C(C2C(N(C)C)CC2)=O)CCCN(C(C2CC3C=CC2CC3)=O)CC1 N1(C(C(CC2CC2)OC)=O)CCCCC(NC(c2ccc(CNC(C)=O)o2)=O)C1 C1(CN(C(=O)C(O)c2cnc[nH]2)Cc2cnn[nH]2)CCOC1=O CC1CCN(C(=O)COCCCF)C1C(N1CCC1)=O C(=O)(C1CCCc2sccc21)N1CC(C)(NC(c2onc(C)n2)=O)C1 CC1CC(CO)CN(C(C2CCCN(C(=O)Cc3ccns3)C2)=O)C1 C(=O)(CC(O)CC(C)C)Nc1ccc(C(=O)NC(CCC)C(F)(F)F)cn1 Cc1cc(CC(=O)NC2CCCCC2C(=O)NCc2cn[nH]c2)nn1C C(=O)(C(O)C1=CCCCC1)NCCC(CC)(C)NC(c1cc(CC(=O)OC)on1)=O C1(NC(c2cnn(CC)c2Cl)=O)CC2CN(C(=O)CC3CCN(C)CC3)CC2C1 N1(CC(C)O)CCN(C(=O)CCCn2cc(CCN(C)C)nn2)CC1 Cc1ccc(CCC(=O)NC2CCN(C(=O)C=C3CC3)CC2C)cc1C C1(CNC(C(CCCOC)C)=O)CC2(CCC2)CN1C(C1CCCN1C=O)=O c1(OC)cscc1C(=O)NC1(C(=O)NOCCCCC2CC2)CC1 c1(C(=O)NC2CC(NC(C(C)NC(c3ccc(F)cc3)=O)=O)C2)cn2ccnc2s1 C(=O)(N1CCC(C(=O)NOCC2(O)CCOC2)O1)C1(C)CC1CC1CC1 N1(C(c2c(N)non2)=O)CCC(C2CCN(C(=O)C(=O)NCC(F)F)C2)C1 c1(CCN2CCCC(C(=O)NC(C3(C)CCOCC3)=O)C2)c[nH]c2ccccc12 c1(C(=O)NCCC(C)CCNC(=O)C=Cc2ccco2)cc2c(s1)CC(C)(C)C2 N1(C(c2cc(C)sc2)=O)CCC(C)(CCNC(C23CC(CF)(CO2)C3)=O)C1 C1(CC)CN(C(=O)CCc2cnoc2)CCC1NC(=O)CCN1CCOCC1=O C(=O)(CCC(=O)NC(C(C)NC(c1csc(O)n1)=O)C(C)C)NCCCOC Cc1noc(NC(C2CN(C(c3cccc(=O)n3C)=O)CCN2)=O)c1C#N S(=O)(=O)(C=Cc1ccccc1)NC1CCC(NC(c2ccsc2)=O)C1 N1(C(c2c(C)nns2)=O)CC2(CCC2)CC1CNC(c1ccc(CCO)cc1)=O N1(CCC#C)CCC(C(N2CC=CC2CNC(C2CC2(C)C(F)(F)F)=O)=O)CC1 CC(CC(=O)NCCC(N)=O)NC(=O)Nc1ccccc1 N1(C(C(CC)(C)CO)=O)CCCC2(CCN(C(=O)CC(C)(O)C(F)(F)F)CC2)C1 C(=O)(CC(CN(C)C)C(F)F)N(C1(NC(CN(C(C)C)C)=O)CC1)C C(CC(CC)C(=O)N1CC=CCC1C(=O)NCC1CCC(C)C1)=CC C(C(=O)NC(CNC(c1cccc(SC)c1)=O)C1CCC1)(C(C)(C)C)OC N1(C(=O)C2=C(Cl)CC2)CCCC(C2CN(C(=O)COCCO)C2)C1 c1(CC(=O)NCCN(C(c2cnc(C3CC3)[nH]2)=O)C2CC2)ccc(F)cc1 N1(CCC)C(=O)CCC1C(=O)N(C)CC1CCCCN1C(c1coc(CO)c1)=O C1(CC)CCN(C(c2cnn(CC)c2)=O)C1C(=O)N(CC)Cc1cn(C)nn1 N1(C(COCCC#C)=O)CCC2CCN(C(=O)CCCCCCCSC)CC2C1 C1(NC(CC2(C)CC2(F)F)=O)C2CC3CN(C(c4cc5occc5s4)=O)C1C3C2 CC1CN(C(C2(CNC(C3CC(O)C(F)C3)=O)CC3(CC3)C2)=O)CC(CO)O1 c1(CCC)cc(C(N2CC(CNC(=O)CCc3nncn3C)CC2C)=O)n(C)n1 c1(C(=O)NCCCN(C)C(C2(CF)CCC2)=O)cncc(C(F)F)c1 C(CC(F)F)(C(=O)NC(C)CN1CCOCC1)N(C(Cc1c(C)nccc1)=O)C C(C)(c1ccccc1C)=CC(N1CC(OCC)(CNC(c2c[nH]cc2Br)=O)C1)=O N1(C(CCOCCOC)=O)CCN(C2CCN(C(C3CCC(=O)N3)=O)CC2)CC1 c1(C(N2CC(CNC(C(CC)(C)F)=O)OCC2)=O)ccc([N+](=O)[O-])cc1Cl C1(C(N2CCCC(CCNC(C(C)=C(C)C)=O)CC2)=O)CC2CSCC(C1)C2 C(Cc1cc[nH]n1)(C(=O)NCCC1COCC1O)NC(C=CCOC)=O C=CCN=C(NCC1CCOC1(C)C)N1CCC2(OC)CCCCC2(OC)C1 c1(C(N2CC(N(C(c3cnc(OC)c(Cl)c3)=O)C)C2)=O)c(Cl)cccc1[N+](=O)[O-] C1(CC(=O)NCCC2CCC2)CC2(C1)CN(C(=O)COC1CCCC1)C2 N1(C(C(C)OC)=O)CCC2(CCCCC2NC(c2cc(C)no2)=O)C1 C(CCCCCN=[N+]=[N-])NC(C(C(C)NC(C1C(C)(C)C1(F)F)=O)(C)C)=O C1(O)(C(C)NC(=O)CCc2cn[nH]c2)CCN(C(=O)C(N2CCC(O)CC2)C)C1 CCC(O)C(C)(C)C(=O)N1CCC(CNC(c2sccc2F)=O)(OC)C1 c12ncc(Cl)c(n1)C(=O)NC2.C1(COC)CN(Cc2ccc(N(C)C)s2)CCS1 C(=O)(C1=NOC(C(=O)NCC(C)(C)NCc2cnoc2)C1)OC(C)(C)C c1(C(=O)NCC2CC2CNC(=O)C=C2CCCCC2)ccccc1-n1cncn1 C1(C(N2C(COC)C=CCC2)=O)CCN(C(=O)C(C)O)C1(C)C O=C1Cc2cc(C(N3CC(NC(c4cc(Br)c[nH]4)=O)C(F)C3)=O)c(Cl)cc2N1 N1(C(Cc2cc(CC)oc2)=O)CCCC(n2cc(CCC(=O)N(C)C)nn2)CC1 CCC(CC(=O)NC1(CNC(c2sccc2-n2ccnn2)=O)CCC1)C1CC1 C12(C(N3CC(C)C(O)CC3)=O)CCCC1CCN2C(=O)CNC(=O)CN(C)C CC1N(C(C2(CNC(=O)CCc3cccn3C)CCCO2)=O)CCCC12CCC2 CC12CC(NC(=O)CC3CCCCC3)(C1)C1(CN(C(c3cccnc3)=O)C1)O2 c1(C(=O)NC(C)CN(C)C(c2ccc(F)o2)=O)c(Cl)cc(Cl)cc1Cl N1(Cc2cccc(N(C)CCO)c2)CCC(C)(CNC(c2nccs2)=O)CC1 C(CCOCCO)(C(=O)NC1CC(O)(CO)C1)NC(C1CCC(F)(F)C1)=O C1(C(=O)NCCCN(C(=O)Cc2ccnc(O)c2)CCC)CC2CCC1C2 c1(NC2N(C(CCNC(CCOCC)=O)=O)CC(OC)C2)cccc(OC)c1C c1(C(N2CC(C(N)=O)(CNC(COC(C)C)=O)C2)=O)ccc2nc[nH]c2c1F c1(OC)cc(OC)c(OC)cc1CN(c1cc(NCCN(C)C)ncn1)C N1(C(=O)C=CCN2CCCC2)CCN(C(=O)CNC(=O)NC2CC2)C2CC12 Cc1cccc(C(=O)NC2CC2C(N2CCC(O)C2)=O)c1 Cc1ncn(C)c(=O)c1C(=O)NCC1CC1CNC(C1(C#N)CC2(CCC2)C1)=O C1(C2CCCCO2)(C(=O)NC2C(C)CN2C)CCOCC1 CC1(C)CN(C(=O)Cn2ccc(O)nc2=O)CC(CNC(C2CC3CC3C2)=O)O1 N1(C(C(C)OCc2cccnc2)=O)CCC2CN(C(C3(CO)COC3)=O)CC12 CC(CCC(=O)NC1CC(NC(C2CN(C)C(=O)N2)=O)C(O)C1)N(C)C C1(NC(c2cn(Cc3cccs3)nn2)=O)Cc2ccccc2N(C(=O)C2CC2)C1 CCCCC(C)C(=O)N1CC2(C1)CN(C(c1ccc(NS(C)(=O)=O)cc1O)=O)C2 C1(C(N2C(CC(=O)NC3CCC(N(C)C)C3)CC(O)C2)=O)CCCC12CCC2 N1(C(=O)CO)CCCC2(C1)CN(c1ccnc3cc(Br)nn13)CCO2 Cc1cc(Oc2ccc(I)cc2)cc(-c2nnc(C(N3CCOCC3)C)o2)c1 C1(C(=O)NC2(COC)CN(C(=O)C=CC3CC3)C2)(OC)CCSCC1 C(=O)(CC(F)(F)C(F)F)NC(C1CCN(C(c2ccc(C=C)cc2)=O)CC1)(C)C N1(C(CC(=O)NCC)=O)CC2COCCC2(NC(=O)Cc2ccc(F)cc2C)C1 N1(C(C(=O)NCCC)c2cnn[nH]2)CC2(CCOCC2)CC1CC(=O)OC Cc1cnn(CC(=O)NC2CCC(NC(c3cscn3)=O)C2)c1 c1(C(=O)NC2C(NC(C=C(C)C(F)F)=O)CC2)ncnc2c1CCC2 C1(C(=O)NCC(c2ccccc2)OC)CN2CCN1CC2C.C1(C(=O)N)(CO)CCC1 CCCCC(C)CC(=O)NC1C=CC(C(=O)NC(C)CCC)C1 Cc1nc(O)c(C(N2CC(NC(C3CC4CCC(C3)C4F)=O)C2)=O)nc1C n1(C2CN(c3c(Br)cnc(C)n3)C2)ccc(=NC(=O)C2(c3cccs3)CC2)[nH]1 C=CC(C)(CC)C(=O)NC1CN(C(c2ccc(C)c(F)c2)=O)C1 C=CCCCCCNC(N1CCOCC1c1nc[nH]n1)=O C(=O)(CCCCC(F)(F)F)NCC(C)NC(=O)C(CO)NC(=O)OC(C)(C)C C12(C(N(CCCCO)CC)=O)CCN(C(c3nc(O)sc3C)=O)CCC1C2 c1(C(N(CC(CC)NC(=O)CNS(=O)(=O)N(C)C)C)=O)cccc(Cl)c1C c1(C(N2CCC(F)(CNC(C3(CC)CC3)=O)C2)=O)cccc2nccn12 c1(C(C(=O)NC(C(C)NC(CC2CC(=C)C2)=O)CO)C)ccc(OC)cc1 C(C1=NOC2CCCC12)NC(C(C1CN(C(CCC=C)=O)C1)O)=O C1(C(=O)NCC2C(CNC(COc3cccc(CC)c3)=O)C2)OCCOC1(C)C C(=O)(C(C)(C)CCF)N1CC2C(C(=O)NCCC(C)N3CCC3)(C2)C1 c1(C(=O)NC(CN(C(CCSCCC)=O)CC)C)ccccc1Cl.C12CCN1C2 C1(C(=O)NC(c2nc(C(N3CCC3C3CCC3)=O)co2)C)(CO)CC=CC1 c1(OC)ccccc1-c1ncc(C(=O)NC2CC2CNC(C2OCCC2C)=O)s1 CC(C)(C)C(CNC(c1ncn(C(C)(C)C)n1)=O)NC(C1CC2(C1)CC2F)=O N1(C(C(c2ccc(Cl)cc2)C)=O)CC2(C1)CN(C(=O)C(C)(C)S(C)(=O)=O)CCO2 C#CC1(C(=O)NC2CCOC2=O)CCN(C(=O)COC)C1 c1(NC(CCCCCNC(C(C)(CO)OC)=O)=O)cnc2ccnn2c1 N1(C(C(c2nc(C)sc2)=O)=O)CCC(C)C1CNC(=O)CCOCC(F)F CCCC(O)C(=O)N(C1CCC(NC(=O)C(C)(F)F)CC1)C CC1CCCC2CCCN(C(=O)C(=O)NC3CCN4CCCC4C3)C12 c1(OC)cnc(Cl)[nH]c1=NC(=O)C1CC1Nc1ncncc1I c1(N(C(CNC(C(=Cc2cccs2)C)=O)C)C)ncnc2[nH]ccc12 C12(CNC(c3cc(C)nnc3)=O)CC(CO1)N(C(C13CSCC1C3)=O)C2 CCC(C)CC(C)C(=O)N1CCC(C(C)(O)CO)C1 c1(C(N2CCCC(C)(NC(COCCC)=O)C2)=O)nn(C)c(=O)c2ccccc12 CCC(CCC(=O)NCCc1ccc(O)cn1)NC(=O)Cc1cnnn1C CCCN(OC)C(=O)CC(CCC)NC(=O)C(N)CC(C)C C(=O)(C(C)(C)C(=O)N1CCC(NC(=O)C=C2CCN(C)C2)C(O)C1)OCC Cc1c(C(N2CC(=C(F)CNC(=O)C(F)C(F)(F)F)C2)=O)oc2ccc(F)cc12 C1(CC#C)(C(=O)NCC(=C)CCNC(=O)CCC2CCCOC2)CCOC1 Cc1n[nH]cc1CN(C)C(c1ccoc1CNC(C12CSCC1C2)=O)=O C1(NC(c2nc(C(C)OCC)sc2)=O)CCN(C(c2cocn2)=O)CC12CCC2 c1(C(N(C(CC)C(=O)NC2CC2)C)=O)ccnc(OC)n1 C(CC(CC)C(=O)N1CC(CC(F)C(N2CC3C(C(N)=O)C3C2)=O)C1)=CC C1(C(N(CC(O)CO)CC)=O)CC2CN(C(c3cccn4cncc34)=O)CC2C1 Cc1nc(C(N2CCCC2CN(C(=O)CN(C)C(=O)C2CC2)C)=O)nn1C c1(CC(C(C(=O)NCCN(C(CCC(C)C)=O)C)F)C)c[nH]c2ccccc12 c1(CC)ncc(C(N2CCC(NC(c3csc(C#N)n3)=O)CC2C)=O)c(C)n1 CC1CN(C(=O)NC(c2ccc(F)cc2)c2cnn(C)c2)CCN(C)C1 N1(C(C(C)(C)C2CC2)=O)CCSCC1C(=O)NCc1ncc[nH]1 C(C(CO)(CO)NC(C1OCCC1(C)C)=O)NC(C1(CC)CC1)=O c1(OC)ccc2c(c1)CCC2(O)CNC(=NCC1CCC1)NCC1OCCO1 c1(C=O)nc2sc(C)cn2c1C.C12CN(CC1O)N2C.C(C=O)OCCSC C1(NC(CSC)=O)CN(C(c2cc(O)nc3c2CCCC3)=O)CC12CCOCC2 CC(CC(N)=O)C(=O)N1C(CNC(=O)CCc2cn(C)nn2)CC2CC12 C(C)(CCCCNC(c1cccc(SC)n1)=O)NC(C1(CC#C)CCOC1)=O N1(C(C(C)OCCOC)=O)CC2CC(NC(c3ccnc(C4CCC4)c3)=O)CC1C2 N1(C(CC(CN(C)C)O)=O)CCN(C(c2ccn(C3CCC3)n2)=O)C(C(F)F)C1 n1(CC(=O)NCC(CC)N(C(CC(CC)C)=O)C)cc(F)ccc1=O c1(SC)cccc(F)c1C(=O)NCCC(C)NC(c1c(Cl)cnn1C)=O N#Cc1c(NC(C2CC23CCN(C(C2(O)CC2)=O)C3)=O)cccc1F N1(C(c2cc(SC)c(C)o2)=O)CC(C)C(NC(=O)CC2(O)CCC2)C(C)C1 N1(CCC(N2CC(C(C)NC(C3C(C(=O)OC)CC3)=O)C2)=O)CCN(C(C)C)CC1 c1(C(N(C(C)CCNC(=O)CNS(C)(=O)=O)C)=O)ccc(-c2cnco2)cc1 C(=O)(C1=CC2CCCC12)NCC1CCN(C(c2c[nH]c(=NC)s2)=O)CC1 C1(CCOC)CN(C(=O)C2=NOC(C(C)(C)C)C2)CCN1C(=O)CS(N)(=O)=O C1(NC(C(C2(O)CCOCC2)(C)C)=O)CC2CCC(C1F)N2C(C1CCSC1)=O N1(CC(=O)NCC2(C(C)(C)O)CN(C(C(CC)F)=O)C2)CCN(C)CC1 c1(C(N2CCCC(NC(C3CC4CC4C3)=O)(CO)C2)=O)cc2c(nn1)OCCS2 c1(OCC)nc(N2CC3C(C(=O)Nc4ccc(C5COC5)cc4)C3C2)ncc1Br C=CCC(C)(C)CCN(C(=O)C(c1cccs1)NC(C)=O)C Cc1ccc(C(=O)OCC2CC=CCC2)nn1 C1(NC(C2C(C)N(C(C3CC3c3ccco3)=O)CC2)=O)CC2(CCCCC2)C1 Cn1c(C(=O)NC2CC(NC(C3(CO)CCCO3)=O)C2)cnc1S CC(O)C(C(=O)NC1CCC1)NC(C1CC1C(N)=O)=O c1(COC)c(Cl)ccc(C)c1OCC(C(c1cccc(Br)c1)=O)N(C)C C1(CCNC(C2CC3CCC2C3)=O)CSCCN1C(c1ccc(Cl)nn1)=O c1(C(=O)NC2C(NC(C(c3ccccc3)N(C)C)=O)C2)c[nH]c2cccc(Cl)c12 C(=O)(C1=CNS(=O)(=O)N=C1C)N(CC(C)O)CCNC(C(C)OCC#C)=O C1(C(N2C(CNC(C3C(C)(C)C3C#N)=O)CCC2)=O)CC(=O)CC(=O)C1 C1(NC(CCc2ccn(C)n2)=O)CN(C(=O)Cc2cnn(C(F)F)c2)CC1F Cc1ccc(CC(=O)NC2CCN(C(c3cc(O)nc(Cl)c3)=O)CC2F)c(C)c1 c1(C(=O)NC(CC(C)C)(C)CNC(C2CC=CCO2)=O)ccc2cncn2c1 O=C(C1c2c[nH]nc2CN1C(=O)CC1CCCCO1)N(C1CC1)CC1(F)CCC1 N1(C(C(C=C=C)C)=O)CC2(CNC(C3(F)CCC3)=O)CC1(COC)C2 N1(C(CSCC(C)C)=O)CCCC(CN(C)C(c2cc(C(N)=O)cn2C)=O)C1 c1(C(=O)NCC(CN(C(=O)CC2CCC(C#N)C2)C)(C)C)cn(C)nc1Br Cc1cc(C(=O)NC2CC(O)CN(C(c3ccccc3C(C)C)=O)C2)cc(C)c1 N1(C(C(C)=C(CC)C)=O)CC2(COC(CNC(c3nccn4ccnc34)=O)C2)C1 C1(C(N2C(C(=O)Nc3ccc(OC)nc3C)CC3CC32)=O)CCc2ccccc2C1 C1(CNC(C(C)c2cccs2)=O)CCCCN(C(C2(C#N)CCOCC2)=O)C1 c1(C(=O)NCCN(C(C)C)C(C2CCOC2C)=O)nnc2n1CCCC2 c1(N2CCCC(C(C)(C)C)CC2)nc2ccsc2c(=NCC2(CO)CCCOC2)[nH]1 c1(C(=O)NCC(CC(C)C)NC(CS(=O)(=O)NC)=O)ccc2c[nH]nc2n1 c1(OCC(N2CC(NC(c3nc(CC)oc3)=O)C(C)C2)=O)c(C)cc(C)cc1C c1(C(N2C(C(CNC(C(C)(C)F)=O)(C)C)CCC2)=O)cnc2cc[nH]c2c1 CCCC(O)CC(=O)NCC12CC(NC(=O)CN3CC=CC3)(C1)C(C)O2 CCN=C(NCCc1cnc(Cl)c(C)c1)N1CCC(O)C1 C(CCC(C)NC(c1cccnc1)=O)NC(C(c1ccccc1)C)=O c1(C(=O)NC2CC(NC(CC3(COC)CC3)=O)C2)cc(OC)ns1 C1(CNC(CC(CC)C2CC2)=O)N(C(=O)C=CC(=O)NC2CC2)CCCC1(C)C C=Cn1nncc1C(=O)NC(COCC)C(=O)NCCC1COCCO1 N#CC1CCCC(CC(=O)NC2C3CC2CN(C(=O)Cc2ccc(Cl)cc2)C3)C1 c1(NC(CC)CC)ccc(Cl)nc1N(C(=O)C(=O)Nc1ccccc1C)CCC c1(NC(c2ccc(F)c(F)c2Br)=O)ccc2oc(Cl)cc2c1 Cc1ccc(C=CC(=O)NC(C2(O)CN(C(C3CCC(=O)N3)=O)C2)C)cc1C Cc1cc(C(N2CCC(C(CO)NC(=O)CCc3cnn[nH]3)CC2)=O)c(C)s1 N1(C(C(C)=C2CCC2)=O)C2CCC1CC(NC(C1CC1c1ccccc1Cl)=O)C2 C(=O)(CS(=O)(=O)C1CC1)N1CC(CN(C(C(Cc2ccccc2)OC)=O)C)C1 C(CNC(=O)CC=CC(C)(C)C)(CC(F)(F)F)NC(C(C1CC1)OC)=O c1(CS(=O)(=O)NC(C(=O)OC)(C)C2CC2)cc(Br)sc1Br C1(Nc2c(C(=O)OC)scc2)CC2CCC(C1C)N2C(c1cnoc1NC)=O c1(CC(=O)NCC(CN(C)C(C2C=CCS2)=O)O)cncnc1O N1(C(c2cnc(OC)s2)=O)CCC(C2CC2)C1C(=O)NC1C2CCC3C(C2)CC13 C1(C)(NC(C=CC(C)NC(C2CC3CCC3C2)=O)=O)C(C)(C)C1(C)C c1(CC)nc(C)c(CC(=O)NC(C)CCCNC(=O)C(C)C#N)c(C)n1 C1(C(=O)NC(C2CCN(C(=O)OC(C)(C)C)CC2)C(F)(F)F)CC(O)C12CCC2 c1(CC)ccc(C(c2nnnn2C(C)C)NCCCC2CCOCC2)cc1 C1(C(N2C(C)(C(=O)NCCCN(C)C)C=CC2)=O)CC2(CCC2O)C1 CCCC(C(=O)OC)C(=O)NCC(C)N(C(=O)COc1cccc(Cl)c1)C c1(C(N(C)CC2(O)CCN(C(C3(CF)COC3)=O)C2)=O)nc(O)nc(O)c1F CCCCCCCCOCC(=O)NCC1(NC(C2CC2C(=O)OC)=O)CCCC1 C1(NC(c2c(C)nccc2)=O)CN(C(=O)CCc2ccncc2)C2CCCCC12 N1(C(=O)OC(C)(C)C)CCC2C(NC(=O)Cn3cccc3)C12 c1(C2(C(=O)O)CCN(C(c3cn(C(C)C)nn3)=O)C2)cc(Br)ccc1F C(=O)(CC(O)C(C)C)N1CCC(OCC(=O)NCc2nc(C)c(C)s2)C1 N1(C(C2CC(C)=C(C)CC2)=O)CC2(CCCC2NC(=O)C(C)OC2CCOC2)C1 N1(C(c2c(C)oc(C#N)c2)=O)CCC2(CC1)CCN(C(=O)C1=CCN(C)C1)C2 CCC(O)C(C)(C)C(=O)N1CCC(N(CCO)C(c2cc(N)ccc2Cl)=O)C1 c1(C(=O)NC2C=CC(CC(N3CCC(OC)C3)=O)C2)nccc(C)c1N CCC1(CNC(C2CN(c3ccccc3)C(=O)N2)=O)OCCc2ccccc21 C=CCC(CC(=O)N=CC(=O)NC(C)COC)OCC N1(C(C(CC)(CC)OC)=O)CC(NC(=O)CCCCCOC)C(C2CC2)C1 Cc1cccc(C(O)C(=O)NCC(c2ccccc2)NC(C2CCCN2C)=O)c1 N1(C(c2c(C)noc2)=O)CC2CC1CN(C(=O)C(C(C)C)n1ccnc1)C2 C(CCC(=O)NCC1CCCN1C(C1CC2CC2C1)=O)N(C(C)=O)C CC(C)(CCCNC(c1sccc1F)=O)NC(=O)COc1ccccc1C(N)=O C1(NC(CCCN=[N+]=[N-])=O)CCN(C(c2c(F)ccc(O)c2F)=O)C12CCC2 N#Cc1ccc(C(N2CCC2CC(=O)Nc2ccc(C3CC3)cc2)=O)nc1 C(=O)(C1Cc2ccc(Cl)cc21)NCC(C)NC(=O)C=Cc1ccccn1 CCCCC(CNCc1cccc(C#N)c1F)CCC c1(C(=O)NCC(C)NC(=O)CCN(c2ccccc2)C)cc(S(N)(=O)=O)cn1C C(=O)(C(C)(C)C(=O)NCC1CC(C)(C)CN1C(=O)C(CC(C)C)N(C)C)NC CN1C(=O)C2CC1CCN2C(=O)CC1CC2(C1)CN(C(c1ccc(F)s1)=O)C2 Cn1nncc1C(=O)NCCCOCCNC(c1cnc(C2CCCCC2)s1)=O C1(COC)(NC(c2cc(Cl)cnn2)=O)CCN(C(=O)CCCn2cccc2)C1 C(=O)(C(=O)CCC(C)C)NC1C(CC)CN(C(=O)COC2CCOCC2)CC1 C1(CC)CN(C(c2cc(C)ccc2I)=O)CCN1C(c1cnc(Cl)s1)=O c1(C(N2CCC(O)(CNC(C3CCCOC3)=O)C2)=O)cccc2cc(Cl)ccc12 c1(C(CNC(CSC)=O)NC(=O)C(O)CF)ccc2ccccc2c1 C(CCN(C1CCCCCC1)N1CCCC12CCS(=O)(=O)CC2)OCCOC c1(N(C)C)cc(Br)ccc1CN1CC2CC1CN2C(c1ccnn1C(C)(C)C)=O C#Cc1ccc(NC(c2cn(CC)nn2)c2nnnn2CCCSC)cc1Br C1(C(=O)NCC(=O)NC(CN(C(c2cncnc2)=O)CC)C)CCOCC1 C1(NC(C2(COC)CC2)=O)CCC12CCN(C(c1nsnc1NC)=O)CC2 C#CCCCCC(c1nnnn1C1COC1)Nc1cccc(CCC(F)(F)F)c1 C1(C(F)(F)C(=O)NC2CC(NC(=O)Cc3cnsc3)C2)(OC)CCOCC1 C1(NC(C2(S(C)(=O)=O)CC2)=O)CN(C(c2ncn3ccccc23)=O)CC2(CC2)C1 C12(CNC(c3cnn(C)c3Cl)=O)CC(C1)C(NC(=O)C(O)c1ccsc1)CO2 CN=c1[nH]c(=NCCS(=O)(=O)N2CCCC2)[nH]c(=NC2CC2)[nH]1 Cc1cc(C(=O)NCC(C)(CO)NC(C2CC(n3cccn3)C2)=O)ncc1F c1(C(C(N2CC(OCC)(CNC(c3cc(F)c[nH]3)=O)C2)=O)(F)F)cccc(C)n1 c1(C(N2CC(NC(C3(O)CCC3)=O)CC(O)C2)=O)cccc2ccccc12 C(=O)(C(C)CC(=O)OC)NCC(CC)NC(c1ccc(OC)nc1C)=O C1(NC(C(C(COC)C)C)=O)CC12CCN(C(c1cnnn1C1CC1)=O)CC2 N(C1CN(C(C23CC2C3)=O)CCc2ccccc21)C(C(CC)OC)=O C1(C(=O)NCC=CCNC(C(C2CCCC2)OCC)=O)CC(C(F)(F)F)CO1 N(C1CN(C(=O)CC2CC2)Cc2ccccc21)C(C1(C(C)C)CCCCC1)=O c1(NC(C2CCC(CN(CCOC)C)C2)=O)c(C)nn(-c2ccc(F)cc2)c1C C(c1cnc(C)nc1O)=CC(=O)NC1CCN(C(c2cn(CC)nn2)=O)C12CC2 C(=O)(C(=O)N=S(C)(C)=O)NCC1CC(C)N(C(=O)CCC(C)(F)F)C1 c1(OC)ncc(F)cc1C(=O)NC(C)(C)CNC(=O)C(C)c1ccon1 CN1CCC(CO)(CNC(=O)C(CCC2CC2)NC(c2coc(C(N)=O)c2)=O)C1 c1(C(N(CCNC(=O)CCc2cccnc2Cl)CC)=O)c(C)cccc1C c1(CC)ccc(C(=O)NCc2cc(C(=O)NCCC=C(C)C)on2)s1 C1(NC(c2ncoc2C2CC2)=O)CCCC(CNC(C2CC(O)C2)=O)C1 c1(CCC(=O)NC2C3CN(C(C4OCC(C)(C)C4)=O)C2C3)cc2ccccc2o1 c1(C(N2C3C(NC(=O)C=CC=C(Cl)Cl)C(CC3)C2)=O)cc2c[nH]cnc-2n1 N1(C(CC2(C)CCC2)=O)CCC(O)(CCNC(c2ccc(F)cc2)=O)C1 C1(NC(C2C(C)C2C)=O)CCOCC1C(=O)NC1(CCO)CCCCC1.CCO C(=O)(C1=Cc2ccccc2C1O)N1C(CNC(c2cc(OC)no2)=O)CCC1 CCCCC(=O)C(=O)N1CC(NC(=O)Cc2ccc(OC(F)F)cc2)C(O)C1 CC1CC(NC(C(=O)N(C)Cc2ncccc2F)=O)CN1C1CC1 Cc1nn(C)cc1C(=O)N(C1CC2CNC1C2)CCc1cnc[nH]1 c1(CCC=C)ccc(C(=O)NCC(C)(O)CNC(C2CCCOC2)=O)cc1 C1(NC(CNC(=O)OCC)=O)C2CN(C(C3C4CCC3(c3ccco3)C4)=O)CC12 CCC(C)(CO)C(=O)NCC1CCN(C(c2cc(O)ccc2C(C)C)=O)C1(C)C C(CCO)N(C(C)C1CC1)CCNS(C)(=O)=O c1(C(=O)NCC2(OC)CN(c3ncc(C#N)cc3F)C2)sc2nccn2c1C N1(C(CC(C)(C)OC)=O)CCC(C2(NC(=O)C(C)O)CC2)C1 c1(CN(C)C(=O)NCC2(Cl)CC2(F)F)nc2c(s1)CCCC2 c1(CNC(C(C2CCCOC2)OC)=O)cccn1C(c1ccncc1)C C(=O)(C(C#N)(CC)CC)N1CC(CC(N2CC(C#C)C(OCC)C2)=O)C2(C1)CC2 c1(N2C(CC(=O)NC(COCC)(C)C)CCC2)c(COC)nc(CC)n1CO CC1=C(C(=O)NC2C=CCN(C(=O)CN3CC4CC4C3)C2)CCC1 C(CC(N)=O)(C(=O)NCc1cn(C)nc1O)NC(CCC=C=C)=O c1(CC(=O)NC2CC2CNC(C2(c3cccs3)CC2)=O)ccc(O)nc1 O(NC(=O)CCCC(C)(C)NC(C1CC(OC)(OCc2ccncc2)C1)=O)CC c1(COCC(=O)NCC(C)NC(c2ccc(CCC)s2)=O)cccc(OC)c1 c1(C(=O)NCCCCNC(C(CSC)C)=O)ncccc1C(F)(F)F c1(C(=O)NC2C(NC(C3CC(=C)C3)=O)CCOC2)cc(=N)[nH]c(Cl)n1 c1(C(N2CC(CNC(C(COC)O)=O)C(C)(C)C2)=O)cnc2[nH]cc(C)c2c1 Cc1cc(C(N2CCC(c3ccon3)C2)C(=O)NC2(C)CC2)cs1 c1(CC)cc(C(=O)NCC(C)CN(C(=O)CC(C)OC)C)n[nH]1 c1(COCCNC(CC(CN(CC(N)=O)C)O)=O)ccc(C#N)c(C)n1 Cc1c(C(=O)NC(C)(CNC(=O)CSC(C)C)C(C)C)cnn1CCC(C)C N1(C(C2C(CNC(C(C)n3ccnn3)=O)CC2)=O)CCN(C(C)(C)C)CC1 N1(CC)CC2CCCC1C2CC(c1cn(CCC2CCCC(C)C2)nn1)C c1(C(=O)NC(C2CCCN(C(c3cc(F)n[nH]3)=O)C2)C)ccc2nsnc2c1 C(=O)(CS(=O)CCC(F)(F)F)N(CC(C)C)C(c1cc2ccccc2o1)C C1(NC(c2c(CC)nccn2)=O)CCC2(CC1)CC2NC(=O)Cn1ncnn1 N1(C(c2c(CC)c[nH]n2)=O)CCCC2(C1)CN(C(=O)CN1OC(C)(C)CC1=O)C2 C#Cc1cccc(N(C(=O)C(C)N(C(=O)CCC(C)N(C)C)C(C)C)C)c1 N1(C(C(c2n(C)ccc2)=O)=O)CCOC2(CCN(C(C3CC(F)(F)C3)=O)C2)C1 c1(C(=O)OC)cc(NC(=O)C(=O)Nc2ccc(SCC(N)=O)cc2)c(C)cc1F c1(C(=O)NC(CN(C(CC(c2ccc(F)cc2)C)=O)C)C)ccc2ncnn2c1 c1(C(N2CCN(C(C(c3c(C)cncc3)C)=O)CC2)=O)cc(Br)cc(N)c1C Cc1ncc(NC(C2CCCCC2CNC(=O)C(C)CN(C)C)=O)c(C)n1 c1(OC)cc(Cl)c(I)cc1NC(=O)CCCNC(=N)N c1(C(=O)NC2(C(F)F)CC(NC(C(C)Cc3cnc[nH]3)=O)C2)ccsc1C#N CC1C(NC(c2ccc([N+](=O)[O-])s2)=O)C(C)CCN1C(=O)Cn1cccc1 CC1(C)COC(NC(=O)COC(=O)CCCn2cc(C3CC(F)(F)CNC3)nn2)C1 N1(CCNC(CS(=O)(=O)NC)=O)CCCN(C(=O)CCN2CCCC2)CC1 C(=O)(CC(F)(F)C(C)C)NC1CC2CN(C(C=C(C)C(C)(C)C)=O)C1C2 C1(NC(C(CC)(F)F)=O)CCC2CC1CN2C(=O)C(=Cc1ccccn1)C CC1CN(C(=O)CCCCCNC(C2CCNC(=O)C2)=O)C(C)(C)C1 C(CC1=CCN(Cc2cncs2)CC1)NC(C(c1c(C)noc1C)C)=O c1(N(CC(CC)C)C)nnc(-c2ccc(Br)s2)n1CCCCCCSC CC1(CNC(C2(CO)CC2(F)F)=O)CCCN1C(c1cccc(C2CCC2)c1)=O C1(CC(=O)NCC23CC(NC(C4CCCC(=O)N4)=O)(CO2)C3)C=CS(=O)(=O)C1 c1(C(C)(F)F)ccc(C(=O)NCC2(CCNC(C34CCCC3C4)=O)CC2)cc1 C1(C(=O)NC(CC)CNC(=O)CSc2cccs2)CCc2nc(O)[nH]c2C1 C(=O)(C(C)(C)C)NCCOCCC1CC(C(=O)OC(C)(C)C)C1 C1(CCNC(c2c(C(=O)OC)coc2)=O)C(C)CCCN1C(c1c[nH]nc1F)=O c1(C(=O)NC(CC(C)NC(=O)C=CI)C)c(Cl)cnn1C c1(CNC(CC)=O)cn(C2CCN(C(=O)C(C)(C)c3ccno3)C2)nn1 c1(C(N(C2CCCCC2)CCC(=O)OCC)=O)cc2n(c(=O)c1)CCS2 n1(CC)cc(CCNC(C2(NC(c3coc(C)n3)=O)CSC2)=O)nn1.N c1(N2CC(CC(N3CC(C)(O)C3)=O)OCC2)ncnc2ccc(Br)cc12 N1(C(C(CO)N(C)C)=O)CC(F)(F)CC1CCNC(c1cc2n(c1)CCC2)=O c1(C(=O)NC2(CN(C(=O)Cc3c[nH]ccc3=O)C)CC2)cc2c(Br)cccc2[nH]1 N1(C(c2cccc3nc(O)[nH]c23)=O)CCCC2(CNC(C3(F)CC3)=O)CCCC12 CC(N=c1cc2n([nH]1)CCOC2)c1nc(Cl)ccc1Cl C1(NC(=O)COC(F)F)C=CCN(C(=O)CNc2ccc(O)cc2)C1 Cc1cc(=NC(=O)C2CCCN(Cc3cccc(OC(F)(F)F)c3)C2)cc(C)[nH]1 C1(C(N2CC(C)N(C(C34CSC(C3)C4)=O)CC2)=O)COc2ccc(Cl)cc2C1 C(C1=CCN(C(c2scnc2Cl)=O)CC1)NC(C1C(C)C1C)=O c1(C(N(C)CC2N(C(CCC=C)=O)CCOC2)=O)c[nH]c2ncnc(O)c12 C12(NC(C(CC(C)C)O)=O)CCCCC1CN(C(c1nc3cnccc3s1)=O)C2 c1(C(=O)NC(C(C)NC(=O)Cn2nccn2)C)cnc2sccn2c1=O N1(C(C(CC#C)O)=O)CCC2CN(C(=O)CNC(=O)OCC=C)CCC12 C1(NC(c2n(C)c(S)nn2)=O)CC2CCC1N(C(c1ncc(F)cc1F)=O)C2 C1(NC(c2n(C)ncc2Br)=O)CCCCCN(C(=O)CC2COC(C)(C)C2)C1 N1(C(C2CCC3(CCC3)O2)=O)CC2CCC(C1)N2C(=O)CCC1CCCOC1 c1(NC(COCCOCCOCC#C)=O)c(O)cccc1Cl Cc1c(CNC(C2CC(C)N2C(=O)CCCCN(C)C)=O)cccc1O C#CCCCCCC(=O)NC1(C)CCC(NC(=O)C(C)CO)CC1 C1(C)(C(=O)NC2CCCCN(C(c3c(CC)non3)=O)C2)CC2(CC(O)C2)C1 C1(NC(c2cnc(C(C)C)[nH]2)=O)CCCC(NC(=O)C(F)(F)c2ccnn2C)C1 CC(C)(C)C(O)C(N)C(=O)N1CCCC(c2nc(=N)[nH][nH]2)C1 C(CC(CC)C(=O)N1CC(C(=O)NOCC(C)(C)C)CC(C)C1)=CC N1(C(C2C(O)CCN2C(C2CC=CCC2)=O)=O)CC2CCCCC2C1 C12(Nc3nc(CC)cc(CC)n3)CCCC1CN(C(C1(COC)CC=CC1)=O)C2 c1(NCC(c2ccccc2)SCC)cc(Br)cc([N+](=O)[O-])c1C c1(CNC(=O)C(N2CC(F)(F)CC2c2ccccc2)=O)c(O)ncnc1O C1(CCN2CCC(OC)C2)CC(C)N(C(=O)OC(C)(C)C)C(C2CC2)C1 C1(NC(C2OCCN(C(CCCOCCC)=O)C2)=O)CCCCC1C#N c1(C(N2CC(CNC(=O)CCCc3nccs3)C3C2C3)=O)ccc(O)c(Cl)n1 C(CCSC)(C(=O)NC(C)CCC=C)NC(CCC#C)=O c1(CNC(C2C(NC(=O)CC34CCCC3C4)COC2)=O)cccnc1Cl C1(CNC(c2c(CC)c[nH]n2)=O)C2CN(C(=O)CC3CCC(=O)CC3)CC12 S(=O)(=O)(c1cc(Cl)c([N+](=O)[O-])cc1F)NC(c1cccc(NS(C)(=O)=O)c1)C CC(C)S(=O)(=O)CC(=O)N(C1CCC(NC(C2CCc3cncn3C2)=O)CC1)C CCC(Cc1cccc(C)c1)C(=O)NCCNC(=O)CCn1cccnc1=O N1(C(CNC(C)=O)=O)CCCC(N(C(=O)CCN(c2ccccc2)C(C)=O)C)C1 C1(CNC(CN(CCC#C)C)=O)CN(C(=O)C(O)CCSC)CC1F c1(C(=O)NCC(CC)NC(=O)CCCCSC)cc([N+](=O)[O-])cc(=O)n1C C(=O)(C(F)CC(C)(C)NC(c1cccn2ccnc12)=O)N1CCCC(=C)C1 N1(C(c2c[nH]c(=NC)o2)=O)CCCC1C1CCCN1C(=O)CN1CCCCC1 C1(C(N(CCCC=C)C)=O)CCC(O)CN1C(c1cnc(=N)[nH]c1)=O C1(C)(C(=O)NCc2ccc(SC)o2)CCCN1C(c1ccsc1C#N)=O CC1CC(NC(=O)C2=NNC(=O)C2)CN(C(c2cc(=N)[nH]cc2Br)=O)C1 c1(NC(C2C(Nc3cc(C)ncn3)C2)=O)nc(C)c(C)cc1Br N1(CCCOCC)CC2CN(C(c3cnn(C4CCC4)c3)=O)CC2C1 N1(C(C2C(CCC)C2)=O)CC(N(C(=O)CCSCc2ccccc2)C)C(O)C1 C1(NC(CCN(c2ccccc2)C)=O)CC2(CCN(C(=O)CSC(F)F)C2)C1 C(C(CC(=O)N1CC(C)(NC(c2ccc3oncc3c2)=O)C1)C(F)(F)F)N(C)C c1(C(N)=O)ccc(C(=O)NC2CC(NC(C3CCCC3c3nc(S)n[nH]3)=O)C2)o1 C=CCC(C(=O)NC1CC1CNC(=O)C(COC)OC)NC(C)=O.C(C)(C)(C)O C1(N(C)C(C2COCCO2)=O)CCC(NC(c2sccc2C#N)=O)CC1 N1(C(c2cccc(SC)c2)=O)CCC2CCN(C(c3cnc(C)n3C)=O)C2C1 N1(C(c2cc(C(=O)NCC)no2)=O)CCC(C)N(C(=O)COc2cn[nH]c2)CC1 c1(CC(C)NCC(c2cccc(C)c2)OC)c(F)cccc1Cl C1(C(=O)NC2C(NC(C(CNC(C)=O)(C)C)=O)COC2)CCC(N=[N+]=[N-])CC1 Cc1nc(O)ccc1C(=O)NCc1cc[nH]c1C(=O)N(CCCCO)C1CC1 C1(CC(N2CC(NC(c3nc(C)oc3)=O)C(C)C2)=O)OCCCC1(C)C O=S(=O)(NCCc1cccc(C(F)(F)F)c1)N1CCC2CNCC2C1 C1(CN(C)C(c2cc(CCCO)on2)=O)CCCN1C(c1ccc(C(N)=O)[nH]1)=O c1(NC(C23C(CN(C(C4(Br)CC4)=O)C2)C3)=O)cc(Cl)ccc1[N+](=O)[O-] N1(C(C2C(C)(C)COC2)=O)CC2(C=C(C(=O)NCCC34CCCC3C4)CO2)C1 C(=O)(CCCC(=O)NC1CC(F)(CNC(C2CCC3(CCC3)C2)=O)C1)N(C)C N1(C(c2cnc(C3CC3)nc2)C(=O)NC(CC)C)CC(N(C)C)C(C)C1 c1(CC)cc(C(=O)NCc2nc(C(=O)NCC34CCCCC3C4)cs2)ccn1 N1(C(C2C(C)CCC2)=O)CCOC2CN(C(=O)C=Cc3ccc(O)cc3Cl)CC12 Cc1ccc2nc(C(=O)NCc3ncc(-c4ccc(C)c(C#N)c4)cn3)sc2c1 C1(CS(=O)(=O)NC)CCCN(c2ccnc(N(C)Cc3ccc(Cl)s3)n2)C1 Cc1ncn(C)c1C(C(=O)NCc1cccs1)N(C1CCC1)CC1CCCO1 C=CC1(C(N2CC(OC)CC2CNC(C2COCCO2)=O)=O)CCCCC1 Cc1cnc(N(C2CCCNCC2)C(c2ccc(CO)o2)=O)nc1 CCCCC(O)CC(=O)N1CCOC(CCNC(c2ncc([N+](=O)[O-])n2C)=O)C1 c12ccnc(n1)CC(=O)N2.C1(c2cn(C3(CN(C)C)CC3)nn2)CC2C=CC1O2 NS(=O)(=O)c1ccc(C(N2CCOCC2CNC(=O)C2=CCC2)=O)c(Cl)c1 c1(CC(C)C)cc(C(=O)N(C2(C(O)CO)CCC2)C2CC2)no1 N(C1CCCOc2ccc(F)cc21)C1(c2n(CCCC)nnn2)CCOCC1 C1(NC(Cc2cc(OC)c(C)cc2)=O)CN(C(C2CCCS2)=O)CCC12CCC2 c1(C(N(C2CCN(c3cc(CC)cnn3)C2)CCC)=O)ccc2c(c1)OCO2 CC1CC(C)(NC(=O)C=CCN(C)C(C2CNC(=O)N2)=O)C1 c1(OC)ccc(Cl)cc1C(=O)NCCC1CC(NC(C2CC23CCCOC3)=O)C1 C1(C2CCOCC2)(C(=O)NC2CCC(NC(=O)C(c3cccc(Cl)c3)O)C2)CC1 C1(C(=O)NC2(CN(C)C(C3(C)CC4CC4C3)=O)CC2)CCCC1C1CC1 c1(C(N(CC(C)O)CCNC(=O)C(C)C2(O)CCC2)=O)scnc1Br c1(C(=O)NCC2N(C(C3C(CC)C3)=O)CC(O)C2)cc(Br)ccc1OC Cc1ccccc1CNC(c1nnnn1-c1cccc(Br)c1)CC1CCCCC1 N1(CC(=O)NC(C2CCN(C(=O)CC3CCOCC3)C2)(C)C)CCSCC1 C(=O)(CCC(CF)CF)N(CC(=O)NCCC1CCOCC1)CC#C C(=O)(CCCC(F)(F)F)N1CC(C)C(CNC(c2nc(Cl)cc(N)c2Cl)=O)C1 CC(CC(=O)NC(c1noc(C2CC2)n1)C1CC1)c1cnn(C)c1.C1C(=O)N1 c1(-c2ccc(Cc3nc(C(CC)(O)CC)on3)s2)cn2ccsc2n1 c1(COC2CN(C(c3cnc(-c4ccccn4)s3)=O)C2)cccnc1 c1(C(=O)NCC(CC(C)C)NC(C2CC3OC2C2CC32)=O)onc2ccccc12 C(=O)(C1=CC2C=CC1C2)N1CC(C2(NC(c3cc[nH]n3)=O)CC2)C1 C#CC1CN(C(c2cncn2C)=O)CCN1C(c1ccc(OC)cc1OC)=O c1(C(N2CCC(C)C(NC(=O)CSc3nnnn3C)C2)=O)ccc2nccn2c1 c1(C(N(C(C(=O)NCCC(C)SC)=O)C)C)cc2ccccc2o1.N1(C)CCOCC1 CC(C(CCc1ccccc1)NC(=O)CCOC1CCC1)NC(=O)CCC1CC1 N1(C(c2cnc(C(C)O)s2)=O)CC2(C1)CN(C(=O)CC1NC(=O)NC1=O)CCO2 C1(NC(C(C)NC(CC)=O)=O)CC12CC(NC(c1cnn(C3COC3)c1)=O)C2 c1(C(=O)NC(CN(C(CCC(=O)NC)=O)C)(C)C)nc(C)c(C)cc1N N1(C(C2C(OC(C)(C)C)C2)=O)CC2(C1)CN(C(=O)C1=CCCOC1)C2 c1(C(NOCC2CC(=C)C2)=O)oc(CNC(c2ccc(CC)s2)=O)cc1C N1(C(C(C)SC(C)C)=O)CCC(F)(CNC(=O)C=Cc2ccc(C(N)=O)o2)C1 N1(C(CC2(C=C)CC2)=O)CCN(C(=O)C(n2cc(C)cn2)C)C(CC(F)(F)F)C1 c1(N2CCC(c3c(C)ncs3)C2)nccc(=NC(C)c2ccoc2)[nH]1 N1(Cc2ncc(OC)cn2)CCP(C)(=O)CC1.N1CCC(N(C)C)C(=O)NC1=O C(c1ccc(N(C)C)cc1)=CC(N1CC(O)(CN(C(c2scc(C)c2)=O)C)C1)=O C1(C)(NC(C(COCC)C)=O)CCN(C(C2CCCS2)=O)CC1 C1(NC(c2cncc(C)n2)=O)CC2CCC1N(C(c1sc(CO)nc1C)=O)C2 C1(NC(c2cc(COC)on2)=O)CN(C(=O)CC2CC3(CCC3)C2)C2CCCC12 C1(C(=O)NC2C3C=CC(C3)C2CO)CC2CCC(C1)N2C(=O)C1=CCCCO1 C1(CC(C)NC(CCOCCCC)=O)CCN(C(=O)C(C2(O)CCCC2)F)CC1 C1(C(=O)NC(CC)CN(C(=O)CN(C)C2CC2)CC)C2COCC12 c1(C(=O)NCC(=O)NCC(=O)N(C(C)CO)C)ccc(C#N)o1 N1(C(CS(=O)(=O)N(CC)CC)=O)CC2CN(C(c3cn(C)nc3C)=O)CC(C1)O2 C(C1c2ccccc2CCN1C(C1(OC)CC1)=O)NC(C1CCC(CC)O1)=O c1(C(=O)NC2CC(C)CN(C(=O)C(F)CC3CCCC3)C2)ccc(N=[N+]=[N-])cc1 C1(O)(CC(N2CC3CC(O)C2C3)=O)CCN(Cc2cc(-c3cccs3)[nH]n2)CC1 Cc1nc(O)ccc1CN(C(C1(c2ccccc2)CC1(F)F)=O)C(C)C C1(C(N2CCC(OCCNC(c3cccc(C)c3)=O)C2)=O)CCN2CCOCC12 C1(C(N2C(CN=[N+]=[N-])CCC2)=O)CN(C(=O)C=CCO)CC1(F)F NS(=O)(=O)c1cc(C(=O)NCCCCNC(=O)C=CC2CCCC2)c(Cl)o1 N1(C(C(C)C2CCCC2)=O)CC(CC(N2CCC(C(C)(C)C)CC2)=O)C2(CC2)C1 Cn1cc(C(N2CCN(C(=O)C(C)(F)F)C3CCC23)=O)c2cccc(Cl)c12 c1(CC(=O)NCCNC(CC(CC)CN(C)C)=O)ccn2cncc2c1 C1(C(C)(C)NC(c2cc(C(C)C)no2)=O)CCN(C(C2CCOC(=O)N2)=O)CC1 C(C(C(C)C)NC(C1CCN(C(=O)Cn2ccc(C3CC3)n2)C1)=O)OC N1(C(CC(CCC)C)=O)CCOC2(C1)CN(C(=O)C1=C(C)OCCS1)C2 C(=O)(C1Cc2ccccc21)N(C(C)CNC(c1c(C)nc2sc(C)cn12)=O)CC CC(C)C(O)C(F)(F)C(=O)NCCC1(CNC(=O)C(c2ccccc2)C)CC1 C(=O)(C(C)CC(F)(F)F)NCC1(NC(C=Cc2c(C)n[nH]c2)=O)CCCC1 C1(C(=O)NCc2cccc(OC)c2)CCC(C)CN1C(c1cc(C)sn1)=O C1(CN(C(C2CC(=C)C2)=O)C)CCCC(NC(=O)CCCc2ccc(Cl)cc2)C1 N1(C(c2c(C)ncs2)=O)CC(F)(F)CC1CNC(=O)C(C)S(N)(=O)=O n1(CC(N2CC(NC(=O)CC3CCC(O)C3)C(O)C2)=O)cnc2c1CCCC2 CC(O)(C(=O)NC1COCC1CNC(C1(CO)CCC1)=O)C(F)(F)F c1(C(C)C)nc2cc(NC(C3(C)COCCO3)=O)ccc2o1 c1(CCC(=O)NCC2CCN(C(C3CC34CC(F)(F)C4)=O)C2)ccc(F)c(F)c1 C1(C)(NC(C(CCC)O)=O)CCCN(C(=O)CCCOc2ccc(C)cc2)C1 C(=O)(C1CCCc2ncccc21)N(C(C)CNC(=O)CCC(C)(C)F)C C1(=C(C(=O)NCCCOC=C)F)CCN(CC2CCC(C)CO2)CC1 Cc1nc(C)n(CC(=O)NCCC2(O)CCN(C(C3(C#N)CCCO3)=O)C2)n1 C12(NC(C3(C(F)F)CC(=C)C3)=O)CCN(C(c3cccc(OCC)c3)=O)CC1C2 N1(C(c2c(C#C)cn(C)n2)=O)CC2=C(C1)CN(C(c1cc(Cl)c[nH]1)=O)C2 c1(C(c2n(C(CC)C)nnn2)NCC2(S(C)(=O)=O)CC2)ccc(C)cc1Cl c1(C(=O)NC2(C)CCC(NC(C(C=C=C)C)=O)CC2)cccc2cnsc12 C1(CNC(C2C(C(=O)OC)C=C2)=O)CC2(CCN(C(c3cccn3C)=O)C2)CO1 Cc1ccc(C)c(OCCCC(=O)NC2CC3(C2)CC3NC(=O)CS(C)(=O)=O)c1 N1(C(C2CN(C(C(CCSC)(C)C)=O)CC2n2ccnn2)=O)CC2(C1)CC(C)(O)C2 c1(CC)nn(C)cc1C(=O)NC1CCC(C(=O)NCCC2CCCC(C)C2)C1 N1(C(C2CN(C(C)C)C2)=O)CCCC(C)(CNC(=O)CCCN=[N+]=[N-])C1 c1(-c2cn(CCCCNC(=O)C(C3CCOCC3)F)nn2)ccc2ncsc2c1 CC(CCCC(=O)NCCCCC1CC1C)NC(=O)Cc1cc[nH]c1 c1(C(=O)NC(COC)CNC(=O)CC2C(C)C2(F)F)ccc(C)cc1 c1(OC)ccc(CCC(=O)NCCCN(C(c2occc2C)=O)C(C)C)c(F)c1 Cn1cncc(C(N2CC(NC(C3CCOC3)=O)CC(F)C2)=O)c1=O C1(C)(C(=O)NCCN(C(C(C)OCc2c(C)cccc2)=O)C)CCC12CCC2 c1(OC(N2CC(OCCCC(=O)NC)C(n3ccnn3)C2)=O)cc(Br)ccc1C C(=O)(CCC(C)(C)[N+](=O)[O-])NCCNC(c1cc(C2C(C)C2)on1)=O C1(NC(C(N2CCCC3CC23)C2CC(C)C2)=O)CCC(F)(F)CC1 C1(NC(=O)C(F)C2CCC2)COC2(C1)CN(C(C13CCC(CC1)CO3)=O)C2 C=CC(CC)C(=O)NC1CC(CNC(c2ccc[nH]2)=O)CC1O C(=O)(C(CCC1CC1)NC(C1C=CCS1)=O)NC1(C)CC(O)C1 Cc1cncnc1C(=O)NC1CCC1C(=O)NCC(C)(C)C(N)=O c1(C(=O)NCC2C(=O)N2)cc(C)n(C2CC2)c1C.C(CC)OC C1(NC(Cc2onc(C)n2)=O)CCN(C2CCN(C(=O)C(F)CC3CC3)C2)CC1 CC(C(=O)N1CC(CCNC(C2(Cl)CC2)=O)C1)N(C)C Cc1c(C(=O)N(CC(CO)(CO)NC(=O)Cc2ccccc2F)C)cncc1Cl CC1=C(CN2CCOCC2c2ccc(Cl)c(Cl)c2)S(=O)(=O)CCO1 C1(Cc2nc(-c3cccc(-n4c(CCC)ncc4)c3)on2)CCC(F)(F)CC1 c1(C(N(C)Cc2scc(C)c2)=O)cc(CNC(=O)C(C)(C)C2CCOC2)nn1C c1(C(=O)NCC2CCCC(NC(CCCOCC)=O)C2)cc2cccc(F)c2o1 N1(Cc2c(C)nn(C(C)C)c2)CCCNC(=O)C(F)(F)C1 c1(C(N2CCC(O)(CN(C(C(CC)SC)=O)C)C2)=O)ccc2ncc(=O)[nH]c2c1 C1(CNC(C2(CCC)CCNC2=O)=O)CN(C)CCN1C(=O)Cc1nc[nH]n1 N1(C(c2c(CNC(C=CC(=O)N(C)C)=O)nnn2C)=O)CCCC(N=[N+]=[N-])C1 c1(C(=O)NC2CC(NC(c3cccc(Br)c3CO)=O)C2)c[nH]c2ccc(Br)cc12 N1(C(C2CCC(=C)CC2)=O)C2CCC1CN(C(C1CC1C1CCOCC1)=O)C2 CC1SCCC1N=c1nc(N(C)Cc2cn(C)cn2)c2c([nH]1)CCCC2 c1(C(=O)OC)cc(C(=O)NCC(F)CNC(=O)CC2(C)CC2)cc([N+](=O)[O-])c1 C(CC(C(C)(C)C)NC(C1(c2ccccc2Cl)CC1)=O)N(C(CC(C)SC)=O)C C1(NC(C2=C(C)CCC2)=O)CCOC2(CCN(C(c3cc(CO)[nH]n3)=O)CC2)C1 N1(Cc2c(C)nc(C)s2)CCS(=O)(=O)C(CCNC(c2cc(C)n(C)n2)=O)C1 c1(N(C(CC(=O)O)c2ccncc2)C)nccc(CNCC2(C(F)(F)F)CC2)n1 C1(C(C(=O)NCC2(CO)CCCC2)F)CCN(C(c2ccoc2)=O)C1 CC1CCCC(C)N1C(=O)CN1CC2(CCN2C(=O)COCC2CCCO2)C1 c1(OC)cc2nc(NC3CCCN(Cc4cccs4)C3)nc(O)c2cc1OC CCC(CC(F)(F)F)NC(=O)CC(CNC(=O)Cc1cnoc1)C1CCC1 c1(C(=O)NCC(C2CCCC2)NC(C(CC=C)(C)C)=O)ccc2oc(=N)[nH]c2c1 c1(C(=O)NC2CC(NC(c3n(CC)nnc3)=O)C2)c(F)ccc(C#N)c1F c1(C2(C)COC2)cn(CCCC(=O)NC(C2CCC2)C2CC2)nn1 c1(C(=O)NC2(CO)CN(C(c3ccc(OC)s3)=O)C2)cnnc(C)c1 C1(CN(C)C(c2cncc(C3CC3)c2)=O)COCCN1.C1(C=O)COCCN1C C1(CNC(Cc2c(C)noc2Cl)=O)CN(C(=O)C(=O)N(C)C)CC1(C)C c1(NC(N(C(C=NOC)=O)CCCNC(=O)CSC(C)C)=O)ccc(Cl)cc1 N1(C(C2CN(C)C(=O)C2)=O)CC2C=CC1C(C(=O)Nc1ccc3nsnc3c1)C2 N1(C(c2c(CC(=O)OC)scc2)=O)CC2CCN(C(=O)CCC(C)N(C)C)C2C1 CCC(CCOC)C(=O)N1CCC(COC)(NC(=O)Cc2cncnc2O)C1 Cc1ccc(C(=O)OCc2cn(CCN3CCOCC3)nn2)c(Cl)c1 C1(NC(CCc2ccc(CC)cc2)=O)CCN(C(C2CC23CC3)=O)CC1F C12(C(=O)NCC3(F)CCN(C(=O)COc4ccsn4)CC3)CCCCN1CCC2 Cc1ocnc1C(=O)NC(c1ccccc1)C(=O)N(C)CC1(CC(C)C)CC1 N1(C(C(n2cc(Cl)cn2)C)=O)CC2CCCC(C1)N2C(=O)C(C#N)CC1CC1 C1(CCNC(C2NC(=O)OC2)=O)CN(C(C2(CO)CCOCC2)=O)CCO1 C1(NC(C2(C)CCCC2)=O)CCN(C(=O)Cc2cccc(N)c2N)CC1F CCC(CC(C)C)C(=O)N1CC(C(=O)NCC2CCC2CO)C(F)(F)C1 CCC(C)(CC)C(=O)N1CCOC(CNC(C2(C#N)CC3(CC3)C2)=O)C1 C(C(=O)N=c1ccn(CC2CCOC2)[nH]1)Oc1c(C)cc(Cl)cc1 CC(C)C(=O)C(=O)NC(c1ccccc1)CNC(C1CC(F)C1)=O CC1CCC(=CC(=O)NCC2CC2CNC(c2cn(CC3CC3)nn2)=O)C1 Cc1ncc(C(=O)NC(C2(CNC(C3CC34CCSCC4)=O)CC2)C)c(C)n1 c1(SC)cc(O)ccc1NC(=O)CCC1CCCN1C(=O)Cc1ccccc1O C1(C)C(C)C(=O)N1C1CC1.c1(OCC)cc(C(=O)NCCC(C)C)on1 C1(C(=O)OC)CCCC(C(N2CC(OC)C(n3ccnn3)C2)=O)C1 CCCC(C)C(=O)N1CC2C(CNC(=O)C(=CC3CCCCC3)F)C2C1 C1(NC(C2N(C(C3CCC(C)O3)=O)CC3CC32)=O)CC2(CCC2)C1O Cc1nc(N2CCCC(CNC(c3ccno3)=O)CC2)c(C)c(Cl)n1 C=CCCCCCCCC(=O)NC1CN(C(=O)Cn2ncn(C)c2=O)C(C)(C)C1 N1(C(c2c(F)ccc(O)c2F)=O)CCCC2(NC(C3CC(O)C3)=O)CC2C1 N1(C(C=CC(C)NC(=O)C2=C(Cl)CCOC2)=O)C2CCCC1CN(C)C2 c12ccc(cc1)-c1n[nH]c(n1)CC2.C(c1cccnc1)=C(COCC)C c1(-c2nc(CCC(C)(C)C)nn2Cc2ccccc2)ccc(F)cc1C(F)(F)F C=CCN(OC)C(=O)C(F)CC(C)(C)NC(c1ncccc1Cl)=O CCC(C)(COC)CNC(=O)COC(C)(C)CNC(=O)CCCCSC C1(F)(C(=O)NCCCCCSC)CCCN(C(=O)CSc2nc[nH]n2)C1 N1(C(CC(C=C)(C)C)=O)CC(C)CN(C(c2cnn(CC(F)F)c2)=O)CC1C Cc1ccc2ncc(C(=O)NC3CN(C(c4cnc(N)c(Cl)c4)=O)C3)cc2c1 CCCC(CNC(C1(C#N)CCC1)=O)C(=O)NC(C(C)C)C(C)C Cc1nn(CC(F)F)cc1C(=O)NC1CCC1NC(C1(O)CCC1)=O c1(C(N2CCC(NC(C3CCN(C)S3(=O)=O)=O)C2)=O)cc(N)c(F)c(F)c1Cl CC1C(NC(=O)C2=CCC2)CCN1C(c1cc(C2CC2)cs1)=O C1(NC(CC(CCC)C)=O)CC(C(=O)N(c2ccccn2)CC(C)C)=CC1O c1(C(N2CC(C)(CCC(N3C(C(N)=O)CC3)=O)C2)=O)cc2ccccc2[nH]1 N1(c2ncnc(C)c2Br)CCC2CCC(C1)N2C(C1CCOCC1(C)C)=O C1(N(C(C=CCCC)=O)C)CN(C(c2sccc2CO)=O)CC1O c1(NC(=O)Nc2ccc(CC)cc2)ccc(NC(C2(C)CC(CC)C2)=O)cc1F c1(NC(N(CC(C)NC(=O)OC(C)(C)C)C)=O)ncccc1Cl C1(c2cn(C)nc2)CN(C(=O)C(O)C2CC2)CCN1C(c1cc(C(N)=O)co1)=O N1(C(CN(C(C)=O)C)=O)CCC(C2CC2)(NC(=O)CN2CCN(C3CC3)C2=O)C1 n1(CCOC)nc(C(N2CC(N(C(=O)Cc3nc[nH]n3)C)C(F)C2)=O)ccc1=O N1(C(=O)NC2C(C(C)(C)C)C2)CCC2CC(O)CCC2C1 c1(C(C(=O)NCC=C)N(C)Cc2ccc(NC(C)=O)cc2)ccc(Cl)cn1 O=C(O)C1CCCc2nc(C(N3CCC4(CCO4)CC3)=O)cn21 C1(C(=O)NC2C(C(C)(C)C)C2)C2CC(O)C(C2)N1C(C1CC2CCCC2C1)=O C1(NC(c2cc(CC)n[nH]2)=O)CC(NC(C2(CC)CC(F)(F)C2)=O)C12CCC2 CC(c1ccccc1C)=CC(=O)NCC1CC(O)CN1C(=O)C(O)CC(F)(F)F C1(C(=O)NCC2(COC)CCC2)CN(C(c2c[nH]nc2C)=O)CCO1 C(CN=c1[nH]ncs1)NC(CNC(CS(=O)(=O)N(C)C)=O)=O Cc1ccc(NC(=O)CC2CC(F)CN2C(=O)C(=O)C(C)C)c(F)c1F N1(c2c(C#N)cncn2)CCC2(CC1)CC(Nc1cccc3c1CCO3)C2 CCCC(C)(C)CC(=O)NCC(=C1CN(C(=O)CCNC(=O)OC)C1)F C1(C(=O)NCCCCNC(c2ccc(C(N)=O)nc2)=O)OCC2CCCC12 CC1=C(C(=O)NC2CCC2NC(C2(N(C)C)CCCCC2)=O)CCC1 C=CCCCC(C(=O)NCC(C1CCCCC1)O)NC(C1CC(=O)N(C)C1)=O N1(C(c2cnc(CC)s2)=O)CCN(C(c2cc(C3CC3C)on2)=O)C(CCO)C1 C1(O)(CNC(=O)Nc2ccccc2OC2CC2(F)F)CCOCC1 C(=O)(CCC=CBr)N(CCC)CCNC(=O)Cn1ccc(C(F)F)n1 c1(C(=O)NCC(CO)NC(CNC(C)=O)=O)cc2c(ccn2C)s1 C1(CC(=O)NCC2CN(CP(C)(C)=O)C2)Oc2ccccc2NC1=O C1(C#N)(NC(CCCC#C)=O)CCN(C(=O)Nc2cc(F)ccc2C)C1 C=CC1(C2(C(=O)NCC3CCN(C(c4c(C)cnn4C)=O)C3)CCC2)CCC1 CCCC(CCC)=CC(=O)NC1(CO)CCN(C(=O)C(C)(C)n2cnnn2)C1 c1(C(CNCCCN(C(CCC(C)C)C)C)O)nc2ccccc2[nH]1 c1(C(N2CC(CNC(=O)CN3CSCCSC3)C2)=O)cccc2occc12 C1(C(=O)NCCC2CN(C(=O)CCC(F)(F)F)CCO2)CC2(C1)CC2(F)F N1(C(=O)Cn2cc(CC3CCCCO3)nn2)CCOC(c2ccc(Cl)cc2)C1 c1(-c2cn(C(C(=O)NCC3CN(S(CC)(=O)=O)C3)C)nn2)ccn(C)c(=O)c1 c1cc2c(C3CN(CCS)CCO3)[nH]nc2cn1 N1(C(CC2(C)CC2(Cl)Cl)=O)CC2CCC2(CNC(C2(C(N)=O)CC2)=O)C1 C(CCCCCC(=O)NCCC1CCC(C)(C)O1)NC(c1ccc(CC)nc1)=O c1(C(=O)NCC2(F)CC(NC(CC(C)C)=O)C2)cccc(C(C)C)c1F C(=O)(C(C)(C)CCS(C)(=O)=O)NCC1OCCN(C(C=C(C)c2cccs2)=O)C1 c1(OC)ccc(C=CC(=O)N(C2CCN(C(C3CC(SC)C3)=O)C2)C)c(OC)c1 CN(CC(=O)c1cccnc1OC(F)F)N1CCN(c2ccc(O)nc2)CC1 N(C1CCCc2occc21)C(C1(n2cnnn2)CCOCC1)=O C(=O)(C(F)(F)CCSc1ccccc1)NCCC(C)NC(CSCC(C)C)=O c1(C(N2C(C)C(C(=O)NCC(C)(O)CCO)CCC2)=O)ccc2ccoc2c1 n1(C(C)C)ncc(C(=O)NC(C)CCc2nccs2)c1Cl c1(C(C(=O)NC(CNC(C2(CC(=O)OC)CC2)=O)CO)C)ccc(Br)s1 c1(CC(=O)NCC(CC)NC(c2ccc[n+]([O-])c2)=O)nccc2ccccc12 CC(=NOCC#N)C(=O)N1CC(CNC(C2NC(=O)OC2C)=O)CC1C C1(C(N(C(C)(C)CO)CC)=O)(OC)CCN(Cc2ccn(C3CCCC3)n2)CC1 C1(CNC(c2csc([N+](=O)[O-])c2)=O)CC2(CCN(C(=O)CC3CC(F)C3)C2)CO1 C(=O)(CS(=O)(=O)N1CCN(C2COCC2C)CC1)OC.N(C)C(C)=O C12(C(N3CC(CNC(=O)CCc4ccsc4)C(O)C3)=O)CCC(CC1F)C2 N1(C(c2cc(Br)ccc2C)C(=O)NCCOC)CCC(F)(F)CC1C C#CCC(CC(=O)NC(C)CCC(=C)C)NC(=O)CCOC(C)=O C(=O)(C#CC1CCCO1)N1CC(O)CC(NC(c2cc(=O)cc[nH]2)=O)C1 Cc1nc(O)ccc1C(=O)NC(C)C(C)NC(c1ccc(CS(N)(=O)=O)cc1)=O c1(C(=O)NCCn2cc(C(N3CC(CC#C)OCC3)=O)nc2)ccc(C)c(C)n1 C1(C)(C(=O)NCC(C)(C(C)C)NC(CCc2c(C)nccc2)=O)CCC(=O)NC1 C1(C(=O)NCC23CC(NC(C4NC(=O)C(F)C4)=O)(C2)C3)CCCC(F)(F)C1 C1(C(N(c2nocc2Cl)CC)=O)CCCCN1C(=O)COCCSC CC1(C)CCC(CC(=O)NCC2C3CN(C(C4(C#N)CCCOC4)=O)CC23)CC1 c1(CC)n[nH]c(=NCCC2CCN(C(=O)C(c3cc(F)cc(F)c3)O)C2)s1 C1(NC(c2n(C)ncc2Cl)=O)CCN(C(c2ncc(Br)cn2)=O)C12CC2 C(CC(C)C(=O)NCC1CC(O)CN1C(c1[nH]c(O)nc1C)=O)=CC C1(=O)C(C)C(C)N1.C(c1ccccc1)=CCN(C(=O)COCC(=O)NCC)CC c1(CNC(C(C)(C)O)=O)cc(Cl)ccc1OC(F)F c1(C(=O)NCCCN(C(C(CCC)O)=O)C(C)C)ccc(OC)cc1Br CC(C)(C)CC(O)CC(=O)NC1CC(C)(NC(=O)COCc2nccs2)C1 C12(NC(c3ccc(C)s3)=O)CCC(CN(C(c3csc(C)c3C)=O)C1)C2 CC1CN(C(=O)Cc2ccon2)CCC1NC(c1cc(Cl)ccc1C(F)(F)F)=O C1(OC)CCCC(CC(=O)NCC(C)CNC(c2ccc(C3CC3)cc2)=O)C1 N1(C(CCNCCCCC)=O)CC2CCN(C(=O)CN(C)CCOC(C)=O)CC12 c1(C(=O)NC2C(NC(c3c(C)nsc3)=O)CC2)cccc(-c2nnco2)c1 C(C(C(=O)NCC1CC1[N+](=O)[O-])NC(=O)CCOCC1CC1)N(C)C C1(C(=O)NC2C=CCN(C(c3ccc(OC)s3)=O)C2)Cc2ccncc2C1 C12(C(N(C(CC#C)C)C)=O)CCCC1CN(C(=O)C(C)(C)C#N)C2 c1(OC)cc(Br)ccc1CC(=O)NC1C=CC(C(=O)Nc2ccc(Cl)cc2O)C1 C1(F)(CNC(=O)C=CC(=O)NC2CC2)COCCN(C(C2COC(=O)C2)=O)C1 c1(NC(N(C)CC2C(OC)CC2)=O)cncc(-c2ccccc2)n1 C12(C(N3CC(N(C)C(C4CCCC45CC5)=O)C3)=O)CC(CO)(C1)OC21CCC1 C1(CNC(=O)CC2COCCO2)CC2CCC1N(C(c1ncnc(O)c1Cl)=O)C2 C1(NC(c2cc(CC)no2)=O)CC(C(=O)NCCCNC(=O)OC)CC1O c1(SC)ccc(C(=O)N(C)Cc2c(C)sc(C)c2Br)c(Br)c1 Cc1ccc(NC(=O)C(C)(O)C(F)(F)F)c2[nH]ncc12 Cc1nn(C)c(C)c1CC(=O)NCC1(C)CCC(NC(=O)C(O)C2CCC2)CC1 N1(C(C(F)=C(C)C)=O)CC(NC(c2coc(C(C)C)n2)=O)CC(F)C1 c1(C(=O)NC(C2CCN(C(C3CCCC3O)=O)CC2)C)snc2ccccc12 C(C1=NOC2CN(C(c3nnc(O)cc3O)=O)CC12)NC(C1(SC)CC1)=O c1(C(N2C(C(=O)NCc3ccc(Cl)c(O)c3)COCC2)=O)c(F)ccc(F)c1F Cc1c(NC(c2c[nH]nc2CCNC(=O)C(C(C)O)N(C)C)=O)cnn1C c1(CCC(=O)NC2(CO)CCN(C(=O)C=CC3CC3)CC2)c(F)cccc1Cl C1(C(=O)OC(CCC)CC)CCC(F)(C(=O)OC(C)(C)C)C1 c1(C(N2CC3(CCN(C(C4CC45CCCOC5)=O)C3)C2)=O)cnn2c1CCCC2 C1(CC(N)=O)COCCN(C(=O)C(c2cc(C3CC3)c(O)nn2)=O)C1 c1(NCCC2N(C(=O)C=CBr)CCC2)ccnc2ncnn12 N1(C(COC2(C)CCC2)=O)CCC(CCNC(C2OCC2(C)C)=O)CC1 C1(NC(c2nncc(C)c2)=O)CCC2CN(C(=O)CCc3cnn[nH]3)CC2C1 C1(C(=O)NCC2CCC(NC(c3ccc(C#C)o3)=O)C2)CC(=O)NC1(C)C N1(C(C2C(=C)C2)=O)CCC(N2CCC(CNC(=O)C(N)=O)CC2)CC1 N1(CC(=O)NC2CCC(NC(C3(CC)CC3)=O)C2)CCC(=O)NC1=O C(=O)(C1=CS(=O)(=O)CCC1)NCC(C)NC(C1(n2cccn2)CCC1)=O C1(CNC(CC(C)(C)OC)=O)CN(C(c2ccc(C)nc2O)=O)C2CCN1C2 c1(-c2c(C)cc(C#N)cc2)ccc2c(C(=O)N(C)CCN(C)C)nsc2c1 C1(C(=O)OCC)CCC(NC(=O)C(=O)NC2C=CC2NCCc2ccccc2)C1 CCC(C)C(O)C(=O)NCC1C2CN(C(=O)CC(F)(F)CC)CC12 C1(C(=O)NCCCNC(c2cccc(F)c2)=O)CC(c2cccc(Cl)c2F)=NO1 C1(C)(CNC(COCC)=O)CC(F)(F)CN1C(C1CCc2n[nH]cc2C1)=O c1(C(=O)NC2(C)CCCN(C(CNC(CC)=O)=O)C2)ccc(S(=O)(=O)CC)cc1 c1(CN2CCC(C)(CNC(c3ncn(C)c3)=O)C2)cc(Br)ccc1Cl C1(C(=O)NC2CCN(C3CC3)C2)(CNC(=O)CCOC2CC2)CC12CCC2 c1(C(=O)NC2(CC=C)CCN(C(C3CCC(=O)O3)=O)C2)cc2ccccc2cn1 Cc1cccn2cc(CNC(=O)OC(C)(C)C)nc12.N12CCC(C1C1CC1)C2=O C(=O)(CC(C)(C)C#N)N1CCC(C(C)(C)CNC(=O)C=CC(=O)N(C)C)CC1 Cc1cc(C(=O)NCC2CCCN2C(c2ccc(-c3ccco3)s2)=O)nc(C)n1 c1(C(=O)NC2C=CCN(C(C3C=CCC3)=O)C2)occ2c1CCC2 c1(N(CCNC(=O)Cc2ncsc2Br)CC)ccc(C(=O)OC)cc1 c1(C(N2CCCC(N(C(=O)CN(C3CCSC3)C)C)CC2)=O)cc(F)cc(F)c1 Cc1c(-c2cnc(CNC(c3ncnn3C)=O)nc2)cccc1F N1(C(C2N(CC)CC2)=O)CC(CNC(=O)CC2CCC(C)(C)O2)C(C)C1 CCC(C)C(O)C(=O)NCC1(NC(c2nnn(COCC)c2N)=O)CCC1 c1(C(N(C2C(C)CC2)C)=O)cnc(C2CC2)nc1.c1(C(C(=O)NC)SSC)cccnc1 c1(C(=O)NC2CCC(CNC(c3cc(Cl)c(Cl)[nH]3)=O)CC2)ccc2cccnn12 CS(=O)c1cccc(C(N2CC=C(CNC(C3CC4CC4C3)=O)CC2)=O)c1 C1(CC)CCN(C(=O)CC(C)C2CC2)C(C(=O)NC2CC(CCF)C2)C1 C1(CNC(c2ccn(CC)n2)=O)CN(C(=O)CSCC(C)C)CCC1C c1(CNC(CCCCC#C)=O)nnc2n1CCN(C(=O)C(O)CCCC)C2 C1(C(NOCC(=C)Cl)=O)CCCC1CNC(=O)C(C)SC(C)C c1(C(N(CCCCNC(C2CCCCC2(C)C)=O)C)=O)c(F)ccc(O)c1F N1(C(C(CC)OC)=O)CCN(C(c2ccn(CC)c(=O)c2)=O)CC1CN(C)C c1(C(=O)NCCC2CCCN(C(C(C)CN(C)C)=O)C2)cn(C)c(=O)n(C)c1=O N1(C(=O)CCN(C2CC2)Cc2ccccc2Br)CC2CNCC2(CO)C1 C#Cc1cn(C)nc1C(=O)N(C1CCCC(NC(c2cncs2)=O)C1)C CC(C)(C)C(O)C(=O)NCC1C2CN(C(c3ncc(Cl)cc3O)=O)CC12 C(=O)(CC(C)(O)C(F)(F)F)N1CC(C(C)NC(c2ccccc2F)=O)OCC1 N1(C(C(C)n2ccnn2)=O)CCOCC(NC(=O)C(O)CC(N)=O)C1 C1(NC(c2nnc(CC)s2)=O)CCCN(C(=O)CCc2cc(C)[nH]n2)CC1 C1(NC(CN(C2CCC2)C)=O)CCOCC1NC(=O)CCn1cnccc1=O c1(COC)nc(C)c(C(N2CC(F)CC2C(C)(C)O)=O)s1.c1(C=O)cnn(CCl)c1 c1(OC)ncccc1CCNC(=O)NC1CCCC(C(F)(F)F)C1 C1(CNC(CCN(C(=O)CSc2cccnc2)CCOC)=O)CC(C#N)C1 C1(C(N2C(C)(C(C)C)CC2)=O)CCCCN(C(=O)C(C)S(C)(=O)=O)C1 N1(C(C(CCC#C)O)=O)C2CCCC1CN(C(C1(Cc3ccccc3)CC1)=O)C2 c1(C(=O)NCC(CNC(c2cc(C)[nH]n2)=O)(C)C)ccc2c(n1)CCC(C)(C)C2 c1(C(=O)Nc2ccc(O)c(F)c2)cnc2ccncc2c1 c1(CC)ncccc1C(=O)NC1CN(C(C2(O)CCSC2)=O)CC1O c1(N(C(=O)C(O)C2CCN2C(=O)COC2CCOCC2)C)cccc(CO)c1.C1CC1 N1(C(c2ccc(CCCCC)o2)=O)CCC(O)(C(C)CNC(C2(CO)CC2)=O)C1 C1(C2CCN(C(=O)C(C)C(C)(F)F)C2)(NC(c2ccc(CC)c(Cl)c2)=O)CC1 C=CCC(CC(=O)N1CC2CC2C2CC12)NC(C1CC(OC)(OC)C1)=O C=CCC(C(=O)NCCn1cc(-c2ccc(C(=O)O)cc2C#N)nn1)C(C)(C)C c1(C(N(C(=O)CC2CN(C(=O)OCCC#N)C2)C)C2CC2)ccccc1 N1(C(C(CC=CC)C)=O)CCC2CN(C(=O)C=Cc3ccco3)CC2CC1 c1(NC(=O)NC2CCN(CC(F)F)C2)cccc(N2C(=O)CCC2=O)c1 C(CC(=O)NOC1CCCCC1)NC(CC)=O.C1CCOC(=O)C1 Cc1nc(C2CC2)ccc1C(N1CCOCC1CN(C(=O)Cc1nc[nH]n1)C)=O c1(C(N2CCSC(C(N3CC4COCC4C3)=O)C2)=O)c[nH]c2nccc-2c1 CC1(C(N2CCC(C)(NC(=O)CC3COC(=O)C3)C2)=O)CNC(=O)C1 c1(C(C)C)nccc(CNC(CCO)c2nccs2)n1 C1(NC(c2n[nH]c(C)c2O)=O)C2CC1CN(C(=O)Cc1cc(F)ccc1Br)C2 C1(C(=O)NC2CCN(C(c3c[nH]nc3C)=O)C2)(OC)CS(=O)(=O)C1 c1(N2C(CN(C(C(CC)N(C)C)=O)C)COCC2)ncnc2c1ncn2C C1(CNC(c2cccc(CF)c2)=O)CN(C(c2occc2C)=O)CCN1OC c1(OC)ccccc1C1(CNC(C2CCC(N3CCCC3)CC2)=O)CCC1 Cc1cccc(C(=O)NC2CN(C(=O)C(C(C)C)N3CCCC3=O)CC2O)c1Cl C(CN=c1[nH]c(=N)[nH]c(=NCC(C)NC(=O)OC(C)(C)C)[nH]1)N(CC(C)C)C Cn1cc(C(=O)NCCN(C(C2C=CC=CC=C2)=O)C2CC2)c(-c2ccco2)n1 C1(C(=O)NC2(C)CCCN(C(=O)COCCF)C2)OCC2CCCC1C2 c1(C(=O)NCC(CNC(c2cc(C)nn2C)=O)O)nc(O)c2ccccc2c1C CC1(C)CCCN(CC2CCc3ncnn32)C1C(N)=O C1(C(N(CC(C)(C)NC(c2nn(CC)c(C)c2)=O)C)=O)CN2CC3CC2(CO1)C3 CCC#CCN=c1nc(N2CCCC(N3CC(O)C3)C2)c2ccccc2[nH]1 Cc1cc(CNC2CC3(C2)CC(NCc2cccnc2)C3)cc(O)n1 N1(C2C(=O)N(c3ccc(OC(F)F)cc3)CCC2)CCCC2(COCCO2)C1 Cn1cc(C(F)(F)F)nc1C(N1CCC(C(C)(O)CNC(C2(O)CC2)=O)CC1)=O N1(C(C(C(C)C)NC(Cc2c(C)n[nH]c2C)=O)=O)CC2CCCCC2C1 S(=O)(=O)(c1ccc(F)cc1F)N(C)CCNC1CCC1(F)F c1(C(N2C(CNC(C3CC(OC)C3)=O)CCCCC2)=O)ccc([N+](=O)[O-])cc1 N1(C(CC(C)(C)O)=O)CCn2nc(CNC(c3snc(O)c3Cl)=O)cc2C1 CC1(C)CC1(C)C(=O)NCCC1(CNC(c2cc(Br)n[nH]2)=O)CC1 c1(CC(=O)N(C2CN3CCC2CC3)CCO)ccc(S(=O)(=O)N2CCOCC2)s1 N1(C(C(C)C2(O)CCC2)=O)CCC(C(=O)NOCc2ccccc2F)CC1(C)C C(C(=O)N1CCC(F)(c2cn(C(C)C(=O)N(C)C)nn2)C1)(C(F)(F)F)OC(C)=O c1(NC2(CNC(C)C(=O)NC)CCOCC2)nccc(Br)n1 C#CCC(C)(C(=O)NCCOCC(N)=O)N(C(=O)C(C)C1CC1)C1CC1 Cc1nn(C)c(C)c1COC(=O)C(O)Cn1cncn1 c1(C2C(C(=O)NCC(C)NC(Cn3c(C)cc(C)n3)=O)C2)c(Cl)cccc1Cl Nc1nc(Cl)ccc1C(N1CC2CC1C2NC(c1ccc(Br)o1)=O)=O Cc1ccc(C(=O)NC2CCCCC2NC2CN(c3ncncc3F)C2)nc1O C1(CNC(C2(CC#C)CCCC2)=O)CC(C)(C)CN1C(C1CC1C(C)O)=O CC1CN(C(=O)CC2CCCC2NC(c2ccncn2)=O)CC(C)(C)O1 c1(C(=O)NC2CCN(C(c3c(CC)noc3)=O)CC2O)cn2c(n1)CCC(C)C2 N1(C(C(C)OCCC=C)=O)CCCC1C(C)(C)NC(C1CCC(F)C1)=O C1(C(N2CCC2Cn2cc(Cn3cccn3)nn2)=O)C2CCCOC12 C1(C(=O)Nc2c(C)cccn2)CN(C(c2cc(F)c(F)cc2I)=O)CCC1(F)F C(=O)(C1CCCc2sccc21)NCCN1CCN(C(C2C(C)C2C)=O)CC1 Cc1cc2c[nH]nc2cc1C(=O)NC(C)(CNC(c1cnn2ccsc12)=O)CO CCCC(O)(CCC)CC(=O)N1CCN(C(=O)CCCC(F)(F)F)C(C)C1C CC(C)C(F)C(=O)N(C1CCOCC1)C.C12CN(CC1c1ccc(F)cc1)C2 n1(CC)nc(C(=O)NC2CCCCC2CC(=O)NCc2cc(C)nn2C)cc1O C1(NC(C=CCOC)=O)CCN(C(c2cnc[nH]c2=N)=O)C(c2ccccc2)C1 C1(C(=O)NCC(C(C)C)Nc2cc(Cl)nc(C3(C)CC3)n2)CNC(=O)CC1C N1(CC(N2CC(C)(NC(CNC(CCNC(C)=O)=O)=O)C2)=O)CCCCC1=O C1(NC(CC(CNC(c2nnn(CC)c2C)=O)C)=O)CC2(C1)CN(C)C2 C(=O)(CC(C)C(F)(F)F)N(CC(CNC(c1n(CC)nc(C)c1)=O)C)C CC(CC(F)(F)F)C(=O)N(CCCNC(=O)C(F)(F)C(C)(C)O)C Cc1c(C(=O)NCC23CCC(CC2)N3C(=O)C(O)C2CC2)c(C(F)(F)F)nn1C Cc1nc(Cl)ccc1CC(N1CCC(C(C)NC(=O)C=CC2CCCO2)CC1)=O c1(CC)cc(C(=O)NCC2CCC(NC(=O)Cc3csc(COC)n3)O2)nn1C N1(C(c2c(C(C)C)cco2)=O)CCC2(CC1)CC2NC(=O)CN1CC=CC1 C1(CCOC)(NC(=O)CC2CCC(=O)N2)CCN(C(=O)C(F)(F)C(C)C)CC1 N1(C(=O)CN2CCCC2=O)CCCC(C2CN(CCC3CCOC3)C2)C1 c1(NC(CC(C)(C)c2nn[nH]n2)=O)ccc(S(C)(=O)=O)cc1 C(=O)(C1=CC(O)C(C(=O)N(C)C)C1)NCCOCCNC(C)C c1(C(C(=O)N(CC(OC)OC)CC2CC2)(C)C)ccc(Br)c(C)c1 C=CC1CCC1C(=O)NC(C1CCN(C(c2ccn(CCCCC)n2)=O)C1)(C)C c1(OC)ccc([N+](=O)[O-])c(C(N2CCC(NC(c3cnns3)=O)C(CO)C2)=O)c1 C12(NC(c3cn4cc(C)nc4s3)=O)CCOCC1CN(C(C1(C(F)F)CC1)=O)C2 C(=O)(CC(C)CC(C)C)NCCC(C)N(C(c1ccc(C#C)cc1)=O)C C1(NC(C2(CC(=O)OC)CC2)=O)(COC)CCN(C(C2(F)CCCCC2)=O)CC1 CCCCCC(CC)C(=O)N1CCCC(NC(c2ccc(CC3CC3)s2)=O)CC1 C12(CNC(c3ccns3)=O)CCCCC1N(C(c1ccc(F)nc1)=O)CC2 C#CCCCC(C)C(=O)NC(C1(C(=O)NC(C)CCOC)CC1)C C1(C(=O)NOC2CCCC2)CCN(C(=O)c2cnc(S)nc2)O1 c1(CNC(C(C)C)=O)nnc2n1CCN(C(=O)Cc1ccc(Cl)cc1)C2 c1(C(=O)NCCC2CCC(NC(COCC)=O)C2)ccncc1Br c1(NC(C23CC2CN(Cc2cc(B(O)O)co2)C3)=O)nc2cc(Cl)ccc2s1 C=CC(C)(O)CC(=O)N1CC(CNC(=O)C(C)(C)C2CCOCC2)C(O)C1 Cc1cc(C(=O)NCc2ccc(C(=O)NCC3(F)CCOC3)cc2)cnc1C C12(CC)CCC(C(N3CCC(CNC(c4ccncc4F)=O)(OC)C3)=O)(CO1)C2 C#Cc1ccc(NC(=O)Nc2n[nH]cc2C(=O)OC(=O)C2CC2)cc1 C(=O)(C(F)(F)C(F)(F)F)NCC1C(C(=O)Nc2ccc(CO)nc2)CCC1 N1(C(C=COCC)=O)C2CCC1CN(C(=O)CC1CCC(=O)O1)C2 c1(OCCC)ccccc1CN1CC2C(C1)N2C(C1CCC(F)(F)C1)=O C1(C(=O)NCCCC(C)(C)O)CC2(CC2)CN1C(C1CC2(CCO1)CC2)=O C(=O)(CS(=O)(=O)C(C)C)N1CC(F)CC(NC(COc2cc(C)cc(C)c2)=O)C1 c1(C(N(CC(C)NC(C2(C#N)CC2)=O)C)=O)ccc(Cl)c(Br)c1F C1(C(=O)NC(CC)CNC(c2cc(C)c(C)s2)=O)CCCN(S(N)(=O)=O)C1 CC1(CNC(C2CCC(=O)N2)=O)CCN(C(c2ccsc2N)=O)CC1 N1(C(C=CCC)=O)CCCCCC1CNC(c1c(Cl)cncc1Br)=O C1(NC(C)=O)COCCC1NC(c1ccc(-c2ccccn2)nc1)=O C1(NC(COCc2ccc(C)s2)=O)CCOCC1NC(=O)Cc1cncnc1O C12CCN(C1)C(=O)C(O)COCCOCCN2C.c1(COC)ccccc1.CC C#Cc1cccc(C(=O)NCCC(C)NC(C2CC3(C)CC2CO3)=O)c1 N1(C(C(C2CC2)SC)=O)CCN(C(c2csc(C)n2)=O)C(C2CC2)C1 Cc1cnc(Cl)cc1NC(C1(C)CCN(Cc2ccc(F)c(O)c2)CC1)=O CC(CC(C)(C)O)N1CCC(CNC(C2(c3ccc(F)cc3)CCCC2)=O)C1 C(CCCC(=O)N1CCC(O)C1C(C)(C)C)N(C(C(C)SCC)=O)C C=CCCCCN=c1nc2ncn(CC)c2c(NCC(C)C(=O)N(C)C)[nH]1 Cc1cc(C(=O)NC2(CNC(=O)CNC(=O)CC(F)(F)F)CC2)nc(O)n1 c1(C(=O)NCC2(NC(C(CCOC)C)=O)CCC2)ccc2[nH]c(=N)oc2c1 N1(C(C2CCCC(C)CC2)=O)CCCN(C(c2ncccc2C2CC2)=O)CCC1 C(=O)(C1=CCCCCC1)NCC1N(C(C2CC(C)OC(C)C2)=O)CC=C1 N1(C(C2C(CNC(C(C(C)C)OC)=O)CCC2)=O)CCC2(CC1)CN(C)C2 C=CC(CCC)CC(=O)N(C1CN(C(c2ccc3c(c2)COC3)=O)CC12CC2)C c1(C(N2CC3CC(NC(=O)C(O)C4CC4)CC(C3)C2)=O)cnc(O)c([N+](=O)[O-])c1 CC(F)CN=c1nc2c(cnn2C)c(NCC2CCCC2N2CCCS2(=O)=O)[nH]1 C1(CC)CN(C)CCCN1C(C1CC(O)CN1C(=O)C(Cl)Cl)=O C=CC1CCN(C(=O)CC2CC3(C2)CN(C(=O)Nc2cc(C)ccc2C)C3)CC1 CCC(CNC(=O)C(F)(F)c1cccnc1)(CC)NC(=O)CCN(CCO)CCO C1(C(N(C(C2CC2(F)F)(C)C)C)=O)CCC(n2cc(-c3ccccn3)nn2)CC1 C1(CNCCc2[nH]nc(COC)n2)CC12CCOc1ccccc12 C1(CCCC(CCC)NC(=O)NC(=O)OC(C)(C)C)Cc2nn[nH]c2C(C)C1 c1(CC(N2CCN(CC(=O)NC(CC)C(C)O)CC2)=O)cc(C)ccc1C CC(C)(C)C#CCCNC(C1COCCN(C(=O)C=CC(F)F)C1)=O N1(C(CC2(C)CCCCC2)=O)C2CCC1CC(CNC(=O)C=CC1CCOC1)C2 c1(C(=O)NCC(N2CCN(C(C3CCCCS3)=O)CC2)C)cc(O)ccc1F C12(CNC(CCCCSC)=O)CCC(C1)N(C(=O)Cc1cc(F)ccc1F)C2 Cc1cccc2cc(C(=O)NCC(n3cc(C4(C(C)C)COC4)nn3)C)[nH]c12 c1(C(=O)NC2CC(C)N(C(c3csc(=N)[nH]3)=O)C2)cccc([N+](=O)[O-])c1 c1(C(=O)NCC(C)O)c[nH]c2ccc(-c3cccc(NC(N)=O)c3)cc12 c1(C(=O)NC23C(CN(C(CS(CC)(=O)=O)=O)C2)C3)cc(F)c(C#N)c(F)c1 C1(CNC(C#CC(C)C)=O)(CO)CCN(C(=O)C(C)COc2ccccc2)CC1 C(=O)(C=C1SCC(=O)N1C)N1CC(OC)(CNC(c2nncs2)=O)C1 CC(C(=O)NC1CN(C(=O)C(C)(C)n2cccn2)C1)C(F)(F)F c1(OC)c(CNC2CCS(=O)(=O)C2C)cc(Cl)cc1Cl c1(C(=O)NC(CCC)CO)coc2c1CN(C(=O)CN(C)C1CC1)C2 N1(C(C(CC)(CC)CO)=O)CCCC2CN(C(C3CC(C)CC(C)C3)=O)CCC12 c1(C(N(CC(C)NC(=O)C(c2nc(C)cs2)C)CC)=O)cc2c(ncn2C)[nH]1 C1(C)(CNC(CSC)=O)COCCN(C(c2c(C)noc2-c2ccccc2)=O)C1 C(CC(F)(F)F)NC(c1cn(CC2CCCNC2)nn1)=O c1(OC)cncc(C(=O)N(CC(=O)NCc2csc(C)n2)C2CC2)n1 c1(OC(C(=O)NCC2CC(NC(c3c(C)nsc3)=O)C2)C)cccc(Cl)c1 C1(NC(c2cc(C)nnc2O)=O)CCCCN(C(=O)C(C)(Cl)Cl)CC1 N1(C(c2c(COC)ocn2)C(=O)NC2CCC2)CC2(CCCCC2)CC1C C1(C(N2CC(C(N)=O)(CNC(C3(C)CCCCC3)=O)C2)=O)Cc2ccccc2O1 C1(NC(C=C(C)CNC(=O)CCC(N)=O)=O)CCOC12CCCC2 c1(C(=O)NCCCCCN(C)C(C2CCCOC2)=O)nn(C)cc1Br c1(C(=O)NCC(CNC(C2CC2c2cccs2)=O)OC)cc(O)cc(Cl)c1 CCCCC(CNC(c1occc1Cl)=O)NC(C1CCC(C)(C)C1)=O n1(C(CC)C)nc(C(=O)NCC2CCCN(C(=O)CCOCC(F)F)C2)cc1C C(=O)(C(C1=CCCSC1)N1CCCC(c2ccccc2)(CO)C1)NCCCOC CCCC(CNC(=O)CCOCC)NC(c1cc(=N)[nH][nH]1)=O CCC(CC(=O)N1CC(CC(C)NC(c2sccc2S(N)(=O)=O)=O)C1)C(F)F c1(C(N2CCC(O)(C(C)NC(CCc3cc(C)no3)=O)C2)=O)ccc(N)c(N)n1 c1(C(=O)OC)sccc1C(=O)NCC1(O)CN(C(C2(CN(C)C)CC2)=O)C1 C(C(C(=O)N1CC(C(C)NC(c2cn(CC(F)(F)F)nn2)=O)C1)N(C)C)OC N1(C(CCSCC(=O)OC)=O)CC2(CCC2)CC1CNC(=O)CC(C)NC(N)=O C1(NC2C(C)OC(C)C2)CCC2CN(C(=O)OC(C)(C)C)CC2O1 CC1(C)CN(C(=O)C(c2ccoc2)NC(c2ncc[nH]2)=O)C2CCCC12 Cc1cc(F)cnc1C(=O)NCCNC(C1CC2(CC(=O)C2)C1)=O c1(C2(C(N3CCC(O)(CCNC(CC=CCC)=O)C3)=O)CC2)ccc(C#N)cc1 C1(N(C(=O)Cn2cc(CO)nn2)C)CCC(NC(c2cnc(OC)nc2)=O)CC1 c1(C(=O)NC2C3(NC(CCC(C)(C)C)=O)CCC(C2)C3)scc2c1CCCC2 CC1(C)CC(NC(C2CN(C(=O)CC3OCCCO3)CC2C2CC2)=O)C(C)(C)O1 C(=O)(C1CCCn2cncc21)NCC(CCCC)NC(=O)CCOC C1(CC(=O)N(CC(=O)NCc2cc(C)no2)C)CCCCC12CCC2 N1(c2cc(C)[nH]n2)CCN(C(=O)NC2CCCC(c3cc(C(F)(F)F)[nH]n3)C2)CC1 N1(C(c2cc(C(N)=O)[nH]n2)=O)CC2CC(C1)CN(C(C1CCC3CCC13)=O)C2 C1(CC(=O)NCC(CN(C(=O)C(C)(O)C2CC2)C)(C)C)CCCC(F)(F)C1 C1(CNC(=O)C=CCF)CCC2(CCC2)C1NC(=O)COc1ccccc1[N+](=O)[O-] Cc1cc(N2Cc3c[nH]nc3C2)nc(N2CCCC(CO)C2)n1 Cc1ccc(Cl)c(OCC(=O)NCC2(F)CC(NC(=O)C(=O)N(C)C)C2)c1 C12(CNC(C(C=CCCC)O)=O)CC1CN(C(c1cnn(CC)c1Cl)=O)C2 C1(CC(=O)OC)CC(O)CN1C(=O)NC(c1ccncc1)C12CC(C1)C2 C1(NC(c2ccccc2-c2ccncc2)=O)CCCCCC1(F)F c1(C(=O)NC2(CN(C)C(C3CC4CCC3O4)=O)CC2)cc(=O)n(C)o1 C1(C#N)(CC(=O)N(C)CCOCCN(C)C(c2cccc(Cl)c2)=O)CCOCC1 CC1CC(C(N2CCCC(N(C)C)C2)=O)N(C(c2ccc(CO)o2)=O)C1 Cn1ncc(CNC(=O)CCc2nncs2)c1C(=O)NC1CC(O)C1 C(=O)(CCCCCn1cc(CCN2CCOCC2)nn1)N(C)Cc1cnccn1 Cc1cc(Cl)ccc1-n1nc(CCC(C)C)nc1C1CCCN1c1ncccn1 c1(C(=O)NC2CCN(C(c3ccc(CSC)o3)=O)C2)ccc2cnccc2n1 c1(CC(=O)NCCCCn2cc(C3(OC)CCOC3)nn2)ncc(C)cc1C CC(C)C(O)CC(=O)N(CCNC(c1csc(NC(N)=O)n1)=O)C(C)C N1(C(C2CCC(=O)N(C)C2)C(=O)NCCCSC)CCc2cc(CO)ccc2C1 c1(C(=O)NC(C(=O)NCCC)C)ccnc(CNC(=O)CN2CCCCC2)c1 N1(Cc2c(C)n(C)n(-c3ccccc3)c2=O)CCCn2nncc2C1 c1(C(N(CCCCCCNC(CC2C(OC)CC2)=O)C)=O)ccc2c(n1)CCO2 Cc1cccc(C(CNC(c2c(C)n[nH]c2C)=O)NC(=O)CC2(C)CCC2)c1 c1(C(N2CCN(C)C(CNC(C3CCCO3)=O)C2)=O)ccc(Cl)c(F)c1N CCS(=O)(=O)N1CC(C(=O)NCCC2(NC(=O)C(C)c3ccsc3)CC2)C1 CN1CNC(=O)C12CCN(C(c1ccc3c(n1)COCC3)=O)CC2 N1(C(C2CC(O)(CC#C)C2)=O)CC2CCC2(CNC(c2ncn(C)n2)=O)C1 C=CCCCC(=O)NC1(C)CN(C(C2(c3ccccc3)CC(C)C2)=O)C1 N1(C(CNC(C2CCCC3(CC3)C2)=O)=O)CC=C(C(=O)NC2CC2)C1 N1(C(C2C(C)=C2)=O)CCC(CF)(NC(c2ccc(C3CCOC3)s2)=O)C1 C1(F)(CNC(C(C)SCC)=O)CCN(C(c2cc(C3CCCCC3)n(C)n2)=O)C1 C(C)(C(O)C(C)C)NC(c1c(CNC(c2c(C)snc2)=O)c[nH]n1)=O C(=O)(C(C)(C)Cc1ccc(Cl)cc1)NC1(CCNC(CSC)=O)CC1 c1(C(=O)NC2CN(C(C(CCCC)NC(N)=O)=O)C2)nccc2ncccc12 CC1CC(NC(c2cc(O)cc(O)n2)=O)CN(C(C2(C)CC2Br)=O)C1 c1(OCC(=O)NCC(CC)(C)NC(C2CNC(=O)N2)=O)c(F)cccc1F N1(C(=O)OC)CCC(O)C(C)(CNC(=O)CN2CCC2NC(=O)CNC(C)=O)C1 Cc1cc(COC(=O)CCN2CCCC(OC(C)(C)C)C2)cc(C)n1 Cc1ccc(F)cc1C(N1CCC(C)C(C)C1)C(=O)NC1(C)CC1 c1(C(C)C)ccc(C(N2CC(F)(CNC(C3CCC3C)=O)C2)=O)c(F)c1 N1(C(CC(=C=C)C)=O)CCC(C)C(CNC(C2(COC)CCCCO2)=O)C1 c1(N2CC(=O)NCC2)ccc(NC(C2C(F)(F)C23CCC3)=O)cc1Cl N1(C(C=CC)=O)CC(NC(c2cnc(C(C)(C)C)[nH]2)=O)C2(CCCC2)C1 C1(NC(CC2(N(C)C(c3csc(F)c3)=O)CC2)=O)CC2CCC1O2 C1(NC(C(CSC)OC)=O)CCCC(NC(c2cncc(C(F)F)c2)=O)C1 C1(C(N(C2CCN(C(=O)C=Cc3cc[nH]n3)C2)CCC)=O)C(C)(C)C1(F)F C(=O)(C(C)CCC(C)(C)C)NCC1N(C(c2c(OC)cc(C)cc2)=O)CC1 N1(C(=O)CCOC2CCC2)CC2CC1CN2C(=O)C=Cc1cncs1 C1(CNC(c2ccc(OC)nn2)=O)CC2(CC2)CN1C(=O)C(C)(F)F c1(OC)ccc(OC)c(C(=O)NC2CC(CNC(=O)C=CC=C(Cl)Cl)C(O)C2)n1 C(=O)(C(N)CC(C)(C)O)N(C)CCc1cccc([N+](=O)[O-])c1 c1(OC)ccc(O)cc1NC(C1CC(N(C)C(c2[nH]cc(C)c2C)=O)C1)=O c1(C(=O)NC2CCN(C(c3c(C)[nH]nc3Cl)=O)C2)nccc2cccnc12 C(c1ccccc1-n1cccn1)=CC(N1CCC(NC(=O)Cc2ccon2)C1)=O N(C1CCCc2ccc(Cl)cc21)C(CN1C(C)CNCC1)=O c1(C(N(C(C(=O)OCC)C)C)=O)csc(CNC(C2(C#N)CC2)=O)c1 C1(NC(C(COC)(F)F)=O)CC2CCC(C1)N2C(=O)CC1CCCCCC1(F)F C(C(CN=c1[nH]n(C(C)C)cc1[N+](=O)[O-])C(F)(F)F)NC(c1c(C)ocn1)=O C1(O)(CC(=O)NN2CCCCC2)CCCC1.C1(C2CNC(=O)CN2)CCCCC1 C1(C(=O)NCc2cncs2)CN(C(=O)CC2CCCC3CC23)CCO1 C1(O)(CNC(c2c(CC)cns2)=O)CCN(C(C2C(C)(C)C2(F)F)=O)C1 N1(C(CC=C=C)=O)CCCCCC1CNC(=O)CC1(OC)CCCC1 CC1CN(C(C2CCCC(=O)N2)=O)CC1CC(=O)NCC1(CCO)CC1 C1(C)(NC(C2(CCNC(c3cn(CC)nc3)=O)CC2)=O)CCC(=O)N(C)C1 c1(CN(C)Cc2n(CC)ccn2)nc(N2CCOCC2)[nH]c(=N)n1 N1(C(C(C#C)(C)C)=O)CCN(C(=O)Cc2cc[nH]n2)C2(CC2)C1 CC1CCC2(CCN(C(=O)CN(C(=O)CCc3ncccn3)C)C2)C1 C1(CNC(c2nccc(C)c2F)=O)CN(C(=O)CSc2cn[nH]c2)C2(CCC2)C1 C1(OC)CCC(NCC2(c3noc(C)n3)CC2)CC1 c1(NC(CNCCC(=O)N(C(CC)C)CC)=O)ccc(C)cc1C c1(NC(c2nccc(CNC(c3ccc(C)nc3)=O)c2)=O)cnn(C)c1C#N C(=O)(C(CC(C)C)NC(c1ccc(F)c(C)c1)=O)N1CCC(SC)C1 c1(-c2onc(C(C)NC(=O)NCCC3SCCS3)n2)ccc(Br)cc1 C1(NC(c2ccc(I)c(Cl)c2)=O)CC12CCN(C(C13CC(C1)C3)=O)CC2 C=C1CCN(C(C2CC(C)N(C)C2)=O)C(C(=O)NCc2[nH]ccc(=O)c2O)C1 N1(C2CCN(C(C(C)CF)=O)CC2)CCN(C(=O)C=CC2CC2)CC1=O c1(C(N(CC(C)NC(c2nnc(S)n2C)=O)C)=O)cc2cc(Cl)ccc2o1 N1(C(=O)NC2CCN(c3cc(O)nc(O)n3)C2)COC2CCCCC2C1 N1(C(=O)NC(c2nnnn2C)C)CCCC(O)(CNC(C2CC2C2CC2)=O)CC1 C(=O)(C(CC)CC(C)C)NC(CCCC(=O)NCc1c(COC)noc1)C c1(C(=O)NCCC2CC(NC(CC(CN(C)C)O)=O)C2)ccn2cc(C)nc2c1 c1(OC(C)C)ccc(CC(=O)NCC2(F)CC(NC(c3ccsn3)=O)C2)cc1 N1(C(COC(C)(C)C)=O)CC2CCC1C1CN(C(=O)C=Cc3ncc[nH]3)CC21 CC1(C)CC(CNC(C2(C3CC3)CCC2)=O)N(C(=O)CCCn2ccnc2)C1 c1(CNC(C(COCC)NC(CC=CC=C)=O)=O)ccc(O)cn1 c1(CSCCC(=O)OC)ccc(NC(=O)C(=O)Nc2cccc(I)c2)cc1 Cc1nncc(C(=O)NC(C)C(N2CC(C)C2(C)C)=O)c1C c1(C(=O)NCC2(CCNC(c3ccc[nH]3)=O)CC2)nccc2c(F)cccc12 c1(C(C)(C)C(=O)N2CC(CO)(NC(=O)CS(=O)(=O)N(C)C)C2)ccc(F)c(F)c1 c1(C(=O)NCCC2CCN(C(c3c(CC)occ3C)=O)C2)cc(C)ccc1C C1(CNC(COC2(C)CCC2)=O)CC(CNC(c2csc(C(C)(C)C)n2)=O)CO1 Cc1cc(O)c(Cl)cc1C(=O)NC(C)CN(C)C(c1ccc(Cl)[nH]1)=O N1(C(CCOCC)=O)CCC(F)(CNC(C2CC(O)(CC)C2)=O)C1 C1(C(=O)NCCCN(C(c2nc3cnccc3s2)=O)CC)CCc2nn[nH]c2C1 CC1(C)CC(CNC(=O)Cc2cc[nH]c2)CN(C(=O)CC2COCC2(C)C)C1 C1(c2nn[nH]n2)(CNC(C2(COC)CC2)=O)CCOCC1 C(=O)(C(C)CC(F)(F)F)N1CCOCC(NC(c2nccc(C)c2)=O)C1 C1(C(N2C(CC(=O)NC)CC2)=O)CC(O)C(O)CC1CNC(=O)C(C)(C)CC#N c1(CC(c2ccccc2)=O)csc(=NCC2C3CCOCC23)[nH]1 c1(C(=O)NC2CC(C)N(C(c3cc4c(ccn4C)s3)=O)C2)cc2occc2n1C Cc1cc(C(=O)NC(C)CC(=O)NC2CCCC2)nn1-c1ccccc1 C(=O)(C1=CC(c2ccccc2)=NS(=O)(=O)N1)NCC(C(C(=O)OC)C#N)=O N1(C(C2C(N(C(C3OC4CCC3C4)=O)CCO)CCCC2)=O)CC=CC(O)C1 C1(CNC(C(C2(C)CN(C(C(CC)n3cncn3)=O)C2)F)=O)(CO)CC2CC2C1 CCCCN=C(NCC1CCNC(=O)C1)N1CCN(CC(C)C)CC1 c1(NC(C=C)=O)ccc(Br)cc1NC(=O)Nc1ccc(Sc2ccncc2)cc1 N1(C(Cn2c(C)cnc2)=O)CCCC1(C)CNC(C1(C(C)C)COC1)=O c1(N2CC(C(C)NC(=O)C=Cc3cn[nH]c3)C2)nccc(-c2ccccc2F)n1 C(=O)(C1=CCCCCC1)N(C(c1ccccc1)CNC(c1cccc(O)n1)=O)C CCCC(F)C(=O)N1CC2CC2(C(=O)NC(c2ccccn2)CO)C1 C1(NC(c2cc(C)c(F)cn2)=O)CCN(C(c2ccc(Cl)cc2Cl)=O)CC1(C)C N#Cc1cscc1C(=O)NC12CC(NC(=O)Cn3cnnn3)(C1)C2 C1(NC(c2nsnc2O)=O)(CO)CCN(C(c2cc(C(F)F)ccn2)=O)C1 C1(S(N)(=O)=O)(C(=O)NC2CCCN(C(C(F)OC)=O)C2)CCC1 c1(C(=O)NC2(CCOCC)CC2)nnc(O)cc1C.C12(CC1)CC(=O)NC2 N1(C(COCCCCC)=O)CCCC(N(C(=O)CC2C=CCCC2)CCOC)CC1 C#Cc1cnn(C)c1C(=O)NCC1CCC(C)N(C(=O)Cn2nc(C)nc2C)C1 C1(NC(C(C)OCC(C)C)=O)COCCC1NC(=O)CCC1CC1 C1(CC)CN(C(=O)CC2CCCCO2)CCC1CNC(c1c[nH]cc(C)c1=O)=O N1(C(c2ccc(Cl)c(F)c2)=O)CCC2(CCN(Cc3cc(O)cc(Br)c3)CC2)C1 Cc1cc(C(=O)NC2CCC(CNC(=O)CC(C)(C)O)C2)nn1C N#CC1(C(=O)NCC2(CN=[N+]=[N-])CC2)CCc2ccccc2C1 c1(C(=O)NC2CN(C(C(CC=CC)CC)=O)C(C)C2)cc(Br)c([N+](=O)[O-])[nH]1 N1(C(CC2(OC)CN(C(c3ccc(Cl)s3)=O)C2)=O)CCC(CO)CC1 C=CCCCC(C(=O)NCC(F)F)NCC(=O)NCC1CC1.C1(CC(=O)OC)(N)CC1 C(=O)(C1=C(c2c(OCCC)nnn2C)CCCCCC1)N1CCC(C)C(C)(C)C1 C1(C(N2CCC(CSC)C2)=O)CC(CC)CCN1C(=O)CCc1cncn1C Cc1cc(C(=O)N(CCNC(C2(C)CC3CC3C2)=O)C2CC2)c(O)c(C)n1 C=CC(O)C(=O)N(C1CCC(NC(c2ccc(C(=O)OC)[nH]2)=O)C1)C C(=O)(C1=Cc2cc(F)ccc2OC1)NC1CCN(C(C=C2CCN(C)C2)=O)CC1 C1(C(=O)NC2CCN(C(C3(CC=C)CCOCC3)=O)C2)CCCC2(CCC2)O1 c1(C(=O)NC2CC3(CC(C)C3)C2)nc(Cl)c(=O)[nH]c1N C1(C(=O)NCc2c(C(=O)NCCC(CC)O)c[nH]n2)OCC2CCCC12 Cc1nccc(C(C(=O)NC2COC2)NC(C2CC(OC(C)(C)C)C2(C)C)=O)n1 N1(C(=O)NC(COCC=C(C)C)C)CCOCC1C1CCOCC1 Cc1cc(C(=O)N(C2CC(C#N)C2)CC(=O)NCCN2CCCC2=O)c(C)s1 C12CN(CCO1)C2.C1(C(=O)O)CCCN1Cc1cn(Cc2csc(Br)n2)nn1 Cc1cc(F)c(NC(=O)NCC2CC2Cc2ccccc2)c(F)c1 Cc1nc2ncccc2cc1CCC(=O)NCC#CCNC(=O)CCCCSC Cc1ncc(CC(=O)NCC(C)NC(C2CC3(CC3)C2)=O)s1 C1(C(N(C)CCO)=O)CCCC(NC(C2(F)CC=CCC2)=O)C1 c1(C(C#N)N(C)Cc2conc2C2CCC2)ccccc1C(F)(F)F N1(C(CC(COC)C)=O)CCN(C(=O)CCCCCC#N)CC(CO)C1 CC1SCCCC1C(N1CC=CC1(C)C(=O)NCCN(C)C)=O c1(NC(c2nnnn2C2CCC2)C)[nH]c(=NCc2cocn2)nc2c1ncn2C C(=O)(C(C)(C)C1=CCN(C(=O)C(O)CN2CCCC2)C1)N1CCC(C)(C)C(O)C1 C#CC1CCN(C(C2C(NC(=O)CN3CC(C)(C)C3)C2)=O)C1 C(=O)(CC1NC(=O)c2ccccc21)N1CC(CNC(C(COC)O)=O)C(C)C1 Cc1nc2c(o1)CCCC2CC(=O)N1CC(NC(c2ccc[nH]2)=O)CC(F)C1 C(=O)(CS(=O)(=O)C1CC1)NCC1(C(C)NC(C)=O)CC1 C1(C(N2CC(C(N)=O)(CNC(C3(CC)CC3(F)F)=O)C2)=O)CC(C)CCO1 C(CCC(C)NC(c1cnc(C(C)(C)C)o1)=O)NC(C(=O)NC(C)C)=O C1(CNC(c2nc(CC)sc2)c2nnnn2CCCSC)CCCC(F)C1 Cc1nn(C)c(C)c1CC(N1CC2(CC2C(=O)NCc2sccc2F)C1)=O c1(C(=O)NC2C(NC(C(CCCC)CC)=O)C2)cc2cccc(OC)c2o1 C(=O)(CS(=O)(=O)CCO)N(C)CC1CCCN(C(=O)CC2CC3(CC3)C2)C1 C(N=c1nc(C2CCOCC2)[nH]s1)C12OCC(CNC(c3ccon3)=O)(C1)C2 Cc1ccc(C)c(C(N2CCN(C(=O)C=Cc3ccc(F)cc3F)CC2)=O)c1O c1(C(=O)NC(C(CO)NC(c2oc(CC)c(C)c2)=O)C)coc2c1COC2 c1(CCCNC(CCN(C(CCOCCOC)=O)C(C)C)=O)cccnc1 N1(C(CCCc2onc(CC)n2)=O)CCCN(C(C2CNC(=O)N2)=O)CCC1 C1(CC=C)CCCCN1C(C1CSCCN1C(c1cc(C)nn1C)=O)=O C=C(C)c1cn(CC2CCCN(C(c3ccc(CNS(C)(=O)=O)o3)=O)C2)nn1 CC1CC(CC(=O)NCCCC2CCCCC2)CN1C(c1cnsc1)=O N1(C(=O)OC(C)(C)C)CCC(C(F)(F)F)(CNCC2CC2(F)F)C1 Cc1cc(C(F)(F)C(=O)NCC(O)CCNC(C2CCCN2N=O)=O)cnc1Cl C(=O)(CC(C)C(=O)OC)NCc1c(C(=O)NCc2c(CC)n[nH]c2)cccn1 C1(C(N2C(CNC(c3n(C=C)nnc3)=O)CCC2)=O)Cc2cc(Br)cnc2C1 CC(C)C(C)(CNC(=O)CSCc1cscn1)NC(=O)CC1CCCC1O C1(c2ccc(COC)cc2)CCCN(Cn2nc(-c3cccc(C)c3)sc2=S)C1 N1(C(CCC#C)=O)CCCC2CCN(C(c3cnc(CC)cn3)=O)CC12 C1(CNC(c2c(CCC)nsc2N)=O)CC2CCC1N(C(c1cncn1C)=O)C2 c1(C(N2CC(CNC(C3N(C)C(=O)CC3)=O)C2)=O)nnc2ccccn12 C1(CC(=O)NC2CCC(F)(CNC(c3c(C)ncn3O)=O)C2)(OC)CCOCC1 N1(C(COC)=O)CCCC(C2CN(C(=O)Cc3ccccc3C#N)C2)C1 C1(OC)CC2(CCC(C(=O)NCC(C)CN(C)C(c3n[nH]cc3Br)=O)CC2)C1 C1(OC)CCCN(C(=O)C(C2CCN(C(=O)C(=O)NOC)CC2)C)CC1 Cc1occc1CC(=O)NCCOCCCNC(=O)C(c1ccccc1)O C12(CC)CC1CN(C(C1(c3cscc3Br)CCCO1)=O)C2 c1(C(N2C(CNC(CCCC=C)=O)CC(COC)C2)=O)cc(O)ncc1F Cc1ccsc1C(=O)NCC1CC(F)(CNC(C2CC2(c2ccccc2)C)=O)C1 N(C(=NCCCCS(C)(=O)=O)NCCOC)CC1CCn2c(C)cnc2C1 C(CN=C(NCCF)N1CCC2CCCOC2C1)N(C)C(=O)OCCS.C(C)(C)(C)O C1(NC(=O)C(c2cc(F)ccc2F)=O)CCCC(NC(c2cc(O)cs2)=O)CC1 CC1CCCN(C(=O)C(C2CC2)NC(=O)CS(C)(=O)=O)CC1 C1(NC(CC2CC(SC)C2)=O)C2CC(NC(c3ccc(Cl)cn3)=O)CC12 C(C1CCC(C)CC1)=C(C)C(N1CC(NC(c2c[nH]cc2Br)=O)C(C)C1)=O C1(C(=O)N(CCCNC(=O)Cn2cc(Br)cn2)C)(COCC)CCCC1 C1(NC(C2C(C3CC3)C2(F)F)=O)CN(C(=O)C=CBr)C2(CCCCC2)C1 Cc1ccc(CSCCC(=O)NCC2CCN2C(=O)Cn2nc(C)nc2C)cc1 CCC(CC)CCC(=O)N1CC2CC(C(=O)NCc3ccc(OC)cc3)CC2C1 N1(S(CCOc2ncc(C(=O)NCC)cn2)(=O)=O)C2CCC1CC(NC)C2 c1(CNC(C2N(C(C(CC)n3cncn3)=O)CC2)=O)nnc(O)n1C CC1CC(NC(C2CCCCCC2)=O)CCN1C(c1cc(F)c[nH]1)=O Cn1cc([N+](=O)[O-])c(NC2CCCCC2CNC(c2ccccc2CO)=O)n1 c1(-c2n(-c3ccn(CC)n3)nc(-c3ccsc3)n2)cc(F)ccc1F C1(CC)CN(C(=O)C2CC2)CCN1C(=O)COc1cc(F)ccc1Br c1(C(=O)OCc2sc(-c3ccccc3)cc2Br)cc2n(c1)CCOC2 S(=O)(=O)(CCC(F)(F)F)NC1CCN(C(=O)CC2CC3CCC2C3)C1 C1(CN(C(CCOCCC)=O)C)CCCCN1C(C1C2CCOCC12)=O c1(-c2nc(CCCOC)nn2-c2ccc(OC)nc2)ccc(F)c2[nH]ccc12 N12CC3CC(CC(C3)C1)NC(=O)C1C(C1)C2=O.c1(SC(C)C(=O)ON)ccccc1 c1(C(=O)NCC(CC(C)O)C)nc2ccc(C(F)(F)F)cn2c1N C1(C(=O)NCc2scc(C(N(C3CC(OCC)C3)C)=O)c2)OCCCC1(C)C c1(NC(=O)Nc2ccc(C(=O)NCCCCl)cn2)cnnc(O)c1Cl C1(C(=O)NCCN(C(Cc2cn(CC)nc2)=O)C)CCCCC1(F)F c1(N(C)C)nc2cccc(C(=O)NCCC3CN(C(C4CC45CC5)=O)C3)c2o1 C1(C)(NC(C(CCC)=CCC)=O)CCN(C(=O)C(O)Cc2ccc(F)cc2)CC1 c1(C(=O)NCC(C2CC2)NC(C2COC2)=O)cc(Cl)c(Cl)s1 C1(c2ccn(C)n2)CCN(C(C2CCN2C2CCNCC2)=O)CC1 Cc1occ(-c2ccccc2)c1C(N1CCC(N(C(=O)CC2CC23CC3)C)C1)=O CC(C)(CNC(N1CCC(C(=O)O)C1)=O)Cn1cc(CCCC#N)nn1 Cc1c(C(=O)N(C(C)CCNC(C2CCC2)=O)C)csc1Br N1(C(c2n[nH]c(CC)c2Cl)=O)CCC2CN(C(c3ccc(F)c(C)c3)=O)CCC12 c1(C(=O)NC2CN(C(C(C)=C3CC3)=O)CC2C)ccc(Br)cc1[N+](=O)[O-] CC1CC(C(=O)N2CCC(C)(CC(=O)NC3CCCCC3(C)C)C2)=NO1 C(C(=O)Nn1nnc2c1CCCC2)(C(C)(C)C)NC(c1c(C)cns1)=O CC(O)(CNC(=O)CCN(C(C1CC=CCC1)=O)CC1CC1)CCO C(=O)(CCC(C)CN(C)C)NCCC(CCNC(c1nn(CC)c(C)c1)=O)C C(=O)(C(C#N)C(C)(C)C)N1C(C)CC(CNC(c2nc(OCC)oc2)=O)C1 N1(C(C2OCC(C)C2)=O)CCC(CNC(=O)C(C)(C)N(C)C)C(F)(F)CC1 c1(C(=O)NC2C(COC)N(C(C3CC3OC)=O)CC2)oc2ccc(C)cc2c1C CC1CN(C(=O)Cc2csnn2)CC1(C)CNC(=O)C(C)(C)Oc1ccccc1 N1(C(c2n(COC)ncc2)=O)CCN(C(C2C(OC)CCCC2)=O)CC12CC2 c1(CNC(CC(C)SC)=O)cccc(NC(c2ccnn2-c2ccncc2)=O)c1 N1(C(c2nc(C)[nH]n2)=O)CCCCC1CN(C)C(C1(c2ccncc2)CCC1)=O CC1OCC2(CCC(CNC(=O)C(CO)NC(=O)C(F)(F)F)O2)C1C N1(C(C2(COC)CCCC2)=O)CCC(NC(=O)CC23COC(C)(C2)C3)C(C)(C)C1 C1(C)(C(N(C)CC2(O)CN(C(C(c3cccc(F)c3)C)=O)C2)=O)CCSCC1 N1(CC)CCC(N(C)C(C2CC(CNC(=O)C=CC3CCOC3)C2)=O)C1 N1(C(C(COC)(C)OC)=O)CC2(CC(CNC(=O)CCc3ccn(C)n3)C2)C1 CCC(CC)C(=O)NCC(=O)NCC1CCCC1NC(c1cc(OC)ns1)=O N1(C(CSC)=O)CC(O)(C(C)NC(=O)CCOCC2CCCO2)C1 c1(C(=O)NC(CNC(C(CCCC)CC)=O)CO)ccc2c(c1)COCO2 N1(C(c2ccc(F)cc2)=O)CCC2CCCN(C(c3cc4[nH]ccc4s3)=O)C2C1 C1(C(=O)OCC23CC(C2)C(C(F)(F)F)N3)CCCCC1Sc1ccccc1 n1(CC#C)cccc1C(=O)NC(C1CCCN1C(c1cnc(CC2CC2)s1)=O)C N1(C(CC)=O)CCC(C(C(C)C)NC(C2CC3CCC3C2)=O)CC1 C1(CNC(Cn2c(C)c(Cl)cn2)=O)C(C2CC2)CCN1C(=O)C(N=[N+]=[N-])C(C)C C(CCCCNC(=O)C(F)F)N(C)C(c1sccc1NS(C)(=O)=O)=O C1(OC)CC(CNC(=O)COC2CCCC2)N(C(c2[nH]c(C3CC3)nc2C)=O)C1 C12(NC(C3CCC(OC)C3)=O)COC(CNC(=O)CCc3cccc(F)c3)(C1)C2 C1(CC(=O)NCCC2(OC)CN(C(=O)C(F)=C(C)C)C2)CCCC(O)C1 N1(C(c2c(C)n(C)cn2)=O)CCC(NC(c2ccccc2F)=O)C(O)C1 C1(C(N2CC(CNC(c3ccc(C)o3)=O)CC2(C)C)=O)C2COC(C)(C)OCC12 C1(C(=O)OCc2cn3ccsc3n2)CC(O)(C2(O)CCC2)C1 N1(C(C(CNC(c2cnc(C)s2)=O)(C)C)=O)CC(C)OC(C)(C)C1 c1(C(N2CCC(NC(C3CCSCC3)=O)CC2)=O)ccc2cnnc(O)c2c1 S(=O)(=O)(c1cc(Cl)ccc1OCC1CCC1)NC(C)(CO)C1CCCO1 CC1(C(N2CC(CCNC(=O)C(=Cc3cccnc3)F)C2)=O)CC2(CCC2)C1 c1(CC(C)N(C(NOCC(=O)OCC)=O)C)ccc2sccc2c1 Cc1cnc2cccc(C(N3CC(NC(=O)Cn4cncn4)CCC3C)=O)n12 c1(C(=O)NC(C2CCCN(C(CCC(=O)NC)=O)C2)C)ccc(F)c(F)c1F c1(NC(C2(C)CCN(C(C(CC)(C)C)=O)C2)=O)cccc(C#C[Si](C)(C)C)c1 N1(C(C2C(C=C)C2)=O)CCN(C(c2c(C)cccc2F)=O)CC1CS(C)(=O)=O N1(CCCNC(C2CCC(C(N)=O)C2)=O)CCN(C(=O)CCc2ccco2)CC1 N1(C(CN2CCN(CC)CC2)=O)CCC(C)(NC(c2nnn(C)c2N)=O)CC1 c1(CC(=O)N(C)CC2COCCN2C(=O)C2=CSCS2)c(Cl)cccc1Cl N1(C(Cc2cc(CC)on2)=O)CC(N(C)C)C(CNC(=O)CC2CC(C)=NO2)C1 n1(CCNC(C=CC(CC)C)=O)ccc(C(=O)N(CC)CC2COC(=O)N2)c1 CC1=C(C)CC(C(=O)NCC(O)CCNC(=O)CC23CCC(CC2)CC3)CC1 C1(N(C(CN(CCCC)C)=O)C)CCN(C(C2CC2C(=O)OC)=O)C1 c1(C(=O)NC(CC=C)CNC(=O)Cc2cncs2)c(C)nc2ncnn2c1C CN1CCN(C(=O)CCOCC2CC2)C(C(=O)NC2CC2c2ccccc2)C1 C(=O)(CC(O)CC(C)(C)C)N1CCC(=C)CC1C(N1CCC1(C)CC)=O c1(CCNCc2n(CC)c(-c3ccccc3)nn2)cc(F)c(OC)cc1Cl NC(=O)CCCC(=O)NCC1(NC(c2ccc(C3CC3)cc2F)=O)CCCCC1 C(CC(C)(C)C)(C(=O)NCc1nc(C(C)C)no1)NC(CN(CCOC)C)=O N1(CC(=O)NCCCC(C)NC(=O)CCSC2CCCC2)CCCCS1(=O)=O C1(CNC(CCC)=O)CC(NC(=O)C=C(C)c2ccco2)CCO1 C1(C(=O)NC2CC(F)(CNC(c3n(C(CC)CC)ncc3)=O)C2)CCCS1(=O)=O Cc1ncnc(C(=O)NC2CC=C(C(=O)NCC3C4CCCC34)C2)c1C Cc1ccc(O)cc1C(=O)NC1CCC(CNC(=O)C#CC(C)C)CC1 Cc1csc(C=CC(=O)NCC(C(C)C)NC(=O)COc2ccon2)n1 c1(CC(=O)NCC(C)C)cc(Br)nn1C.c1(CCC(=O)N)nc(C)n[nH]1 Cc1cc(C)c(C(N2CC(C)(CNC(C3(C)CCCC3)=O)C2)=O)c(Cl)n1 c1(C(=O)NCCCN(C(C(C)=C2CC2)=O)CC2CCCC2)c(Cl)cc(Cl)nc1N C(C(F)(F)CN(C(=O)C(CC1CCCC1)NC(=O)COC1CCC1)C)OC c1(C(=O)OCC)cc(C(=O)NCC2CN(C(c3ccon3)=O)C2)no1 c1(C(=O)NC(C)(C)CNC(C23CCCC2CC3)=O)cccc2nc[nH]c12 C1(NC(c2noc(CC)c2C)=O)CCCC12CN(C(=O)CC1COC(C)(C)C1)C2 CON(CCC(=O)NCC1CC2(CC2)CO1)C(=O)CCC1CCCN1C C1(c2cn(C(CNC(COCCCOC)=O)C)nn2)CN(C(C)=O)CC(C)(C)C1 C1(CCOC)CN(C(=O)CCC(=O)c2ccccn2)CCN1C(C1CC(F)C1)=O Cc1cc(F)cnc1C(=O)NCCCCCCNC(=O)CC(C)(C)O N1(C(C2CCN(C(C(C(C)C)O)=O)CC2)=O)CCCC2CC1C2(C)C CC(C)CC(C(=O)NC(C)CNC(=O)Cc1coc(C(F)F)n1)N1CCCC1=O c1(C(N2CCC(CC)(CO)C2)C(=O)NC(CC)C)ccc(N2CCCCC2)cc1 c1(CC(=O)NC2CN(c3nnc(CCOC)s3)CC2(C)C)cnn2ccccc12 c1(C(=O)NC(CN2CCN(C(C=CC=CCC)=O)CC2)C)cc2cn[nH]c2cn1 c1(C(=O)NC(C)C(C)(C)NC(c2ccc(O)cc2)=O)cn2c(n1)COCC2 N1(C(CCSCC(C)C)=O)CCCC2(CCCN2C(C2OCCOC2C)=O)C1 c1(C(C)C)nnc(C=CC(=O)N(C)CCN(C(C2(F)CCCC2)=O)C(C)C)o1 C1(F)(CNC(=O)Cc2cnns2)CCC(CNC(=O)C(F)(F)c2ccncc2)C1 C1(NC(c2ccccc2CO)=O)CCC2CN(C(=O)CCOC3CC3)CC2C1 N1(C(c2cnc(C)s2)=O)CCC(C=CC(=O)NC2CC(=O)N(C)C2=O)CC1 c1(C(N(C)CC2CCCN(C(C(C)C#N)=O)C2)=O)cc2cccnc2cc1F C1(C(=O)NC(c2ncc(C)[nH]2)CC)CCCN(C(C2CC3(CSC3)C2)=O)CC1 CCCC(C(=O)N1CCN(CCC)CC1)NC(c1cccc(C)n1)=O CC(CN(C)C)CC(=O)NCc1cn(CC(=O)NC(c2ncccc2F)C)nn1 C1(CNC(C(CC)C)=O)CCCCN(C(=O)CCc2c(C)nc(C)nc2O)CC1 c1(N(C)CC2CCS(=O)(=O)C2)ncccc1S(=O)(=O)N(C1COCC1O)C c1(C(=O)NC2(CNC(=O)C3=CC4CCCC34)CC2)c[nH]c2cc(Cl)ccc12 S(=O)(=O)(c1cc(C)ccc1C)CN1CC(NC(CCSC)=O)C(C#N)C1 C1(C)(CN2CCCC(CN(c3ccccc3)C)C2)CCC(F)(F)C1 c1(CNC(C2(C)CCCN2Cc2cc(Cl)nc(Cl)c2)=O)ccc(C#N)cc1F CCCCC(C)C(=O)NC1(COC)CCCN(C(c2c[nH]c(Br)c2)=O)C1 c1(OC)cccc(NC(=O)COCc2cn[nH]c2)c1.C1(=O)CO1 C(=O)(C(CC(N)=O)NC(C1CC12CCC2)=O)N1C(C)(CCO)CC1 C1(C(=O)NCCC2CN(C(C=C(CC)CC)=O)C2)CCC(NC(=O)C2CC2)CC1 C1(C(c2n(CCC)nnn2)Nc2cccc3c2CCO3)CC(C)(C)OC(C)(C)C1 N1(C(c2ccc(N)c(F)n2)=O)CCC(C2CC(NC(=O)Cc3cn[nH]c3)C2)C1 N12CCC(C)(C)C(C1)NC(=O)c1c(cccc1C)OCC2=O.C12(SC)CC(C1)C2 CC1=C(C(=O)N2CCCC(NC(=O)C3=CCC3)CC2)Cn2nnnc2N1C c1(C(N2CCC(CC=C)C2)C(=O)NC2CC2)ccc2nc(C)ccc2c1 CCC(C(=O)NC(c1cn(C2COC2)nn1)C)C(F)(F)F C#Cc1ccc(OC)c(C(=O)NCC(C)(CNC(=O)C(C)(CO)OC)OC)c1 C1(NC(=O)C=CBr)COCCN(C(c2cccc(F)c2Cl)=O)C1 c1(C(=O)NC(CC)CN(C)C(c2cc(C)no2)=O)cncc(C(=O)OC)c1 c1(N2CC(NC(C(c3ccccc3)C)=O)C(O)C2)nccc(C#N)n1 c1(CNC(CCNC(CC)C2CC2)=O)ccc(Sc2cccs2)cc1 C(=O)(C(CC)C(F)(F)F)NC(CC(N1CCC(C#C)CC1)=O)C1CC1 C1(CC(=O)NC(c2nc(C(=O)NCC3CCCC(C)C3)co2)C)C(C)(C)C1(C)C c1(C(N(CCN(C(C(CC)COC)=O)C)C)=O)c(Cl)c(C)nn1C Cc1cc(C(C)C(=O)NC2CN(C(=O)C(C)CCO)C2)cc(C)c1 c1(OC)cncc(CNC(=O)CN(C(=O)C(C)C#N)C(C)C)n1 C(C)(CC(=O)NCCC1CCC(NC(=O)Cc2cccnc2)C1)OC C1(NC(C(CC)O)=O)CCOCC1NC(c1cccnc1OCC)=O c1(C(=O)N(C2CC2)CC2CCCN2C(=O)C=CC(F)(F)F)cn2ccsc2n1 CC1(C)CCCCC(C(N2CC(NC(c3ncccc3O)=O)C2)=O)C1 c1(CN(C(Cc2ccccc2Br)CO)CC=C)c(Br)nn(C)c1C N1(CC2N(S(CCC)(=O)=O)CCC2)CCN(C(=O)OCC2OCCOC2C)CC1 c1(C(N(CC(C)NC(CCC=C)=O)CC)=O)ccc2c(Br)cnn2c1 C(=O)(C(C(C)C)n1cncn1)N(CCN(C(=O)C(C)(C)C)CCOC)C1CC1 C1(OC)CCCC1C(N1CCCC1CNC(=O)C=CC1CCCO1)=O N1(C(CCCOCCC)=O)CCC2CC2(NC(c2cc(OC)cnn2)=O)CC1 c1(C(=O)NC(CCOC)CNC(=O)CCCc2nccs2)cccnc1Cl c1(C(=O)NC2C(NC(c3n(C)c(S)nn3)=O)C2)cnc(O)c2cccnc12 C1(CC#C)(C(=O)NCC2CC2[N+](=O)[O-])CCN(C(c2sc(F)cc2C)=O)C1 CC1(CNC(=O)Cc2cscn2)CCCN(C(=O)CCC2NC(=O)NC2=O)C1 c1(C(=O)NCC2C(C)(C)C(=O)N2)cccc(S(=O)(=O)N2CCSC23CCC3)c1 c1(C(N2C(c3cn(Cc4c(C)c[nH]n4)nn3)CCCC2)=O)cc(=O)n2ccsc2n1 Cc1c(C(N2CC3(CCN3C(=O)CC3CCCC(O)C3)C2)=O)sc2nnc(S)n12 C1(NC(Cc2ccc(C)s2)=O)C(C)CCN(C(c2cc(O)cc(N)c2C)=O)C1C c1(C2N(C(=O)Nc3occ(C)n3)CC2)ccc(C)c(OC(F)F)c1 Cc1ccc(C(=O)NC(C(=O)N(C2CCOC2)CCO)C2CC2)o1 C=CCC(CC)N=c1nc(N(C)Cc2nocc2CC)c2cnn(C)c2[nH]1 c1(C(CNC(c2n(CCOC)nnn2)c2ccoc2C2CC2)C)ccccc1Br c1(C(c2n(CC)nnn2)NCCc2ccns2)cc(OC)cc(OC)c1Br c1(CC(=O)NC(CCN(C(C2C(=C)C2)=O)C)C)sc(C2CC2)nc1C Cc1cc(=NC(=O)C2CCCC23CN(C(=O)CCc2ccsc2)C3)[nH][nH]1 N1(C(CC2N(C)CCCC2)=O)CC(CNC(c2cc(C(F)F)no2)=O)CC1(C)C C1(C(=O)NC(CC)C)CC2(CCN1C(C1C=CC1C(=O)OC)=O)CC2 N1(C(CC2C(C)OC(C)C2)=O)CCCC(N(C)C(c2ccc([N+](=O)[O-])s2)=O)CC1 C1(NC(Cc2cnc(C)s2)=O)CN(C(c2cc(F)c(N)cc2F)=O)CC(C)(C)C1 C12(CNC(C3CCCC3)=O)CC(CCO1)N(C(c1cccc(CO)c1)=O)C2 c1(NC(c2c(O)ccc(C)n2)=O)cccc2c1C1CN(C(=O)OC(C)(C)C)CC1O2 C1(OC)CC2CC(C(=O)NCCN(C)C(C3(C(=O)OC)CC3C)=O)CC12 C1(CNC(C(CCOC)C)=O)CC(NC(=O)C(=O)NC2CC2)C12CCC2 N12CCC(C3CC3)C1C2=O.c1(OCC)cc(OC)nc(NC2CC2)n1 c1(OC)cnncc1C(=O)NC1CCC1C(=O)NCCc1ccnc(C)c1 CN1C(=O)CCCC1C(=O)NC1(CNC(C2(C3CCCO3)CC2)=O)CCCCC1 CCCC(C(=O)OC)C(=O)NCC1CC1CNC(=O)CC1CCC1 C1(CCOC)(NC(=O)CC2(C)OCCO2)CCN(C(=O)C=C=C(C)C)C1 c1(C(=O)NC2C(NC(C3(C)CC3)=O)CCCC2)cc(Cl)c(Cl)c(Cl)c1 c1(NC(C(CO)NC(C2CCC(OC)CC2)=O)=O)ccc2nncn2c1 C(C(C)(CC)C(=O)NCCn1ccc(=O)cc1)NC(C(CCC)NC(N)=O)=O N1(C(C2(SC)CCC2)=O)CCC(F)(F)C(CNC(=O)CCCc2ccccc2)C1 C(CCC(=O)NC(C(=O)NCC(=O)NC1CC1)C1CCCC1)OC(C)(C)C c1(C(=O)NCC2(F)CCCN(C(c3nc(=N)[nH]cc3)=O)C2)ccnc2cc[nH]c12 N1(C(c2nc(COC)sc2)=O)CC(C)CN(C(c2cc(Cl)no2)=O)CC1C C1(C(=O)NCC(C)NC(=O)C(C)c2ccsn2)CC(F)(F)C1 c1(C(C)O)cccc(-c2ccc(CN3CCN(c4ccc(Cl)cn4)CC3)cn2)c1 C(=O)(C1CCCn2ncnc21)N1CCCC(CNC(C(C(C)C)(C)C)=O)CC1 N1(C(c2cccc(Cl)c2OC)C(=O)NCCCCCC)CC2OC(=O)N(C)C2C1 N1(C(c2cc(CCC)[nH]n2)=O)CC(NC(=O)CC2CC=CCC2)CC(C)C1 N1(C(c2nc(COC)oc2)=O)C2CCC1CN(C(=O)CCC=CBr)C2 C12(SC)CCC(CN1CS(C)(=O)=O)C2.c12csc(n1)CNC(=O)C2 C(=O)(C(C)(C)C(=O)NCC1C2CN(C(=O)CC3COCCO3)CC12)OCC C=CC(C)(CCOC)C(=O)N1CC2(CNC(C3CC34CCCC4)=O)CC1(CC)C2 C1(CCC)CCCN(C(C23CC2CN(C(=O)C(CC)SC)C3)=O)CC1 c12ccc(cc1)CCNC2=O.C1(NS(C)(=O)=O)CCCC1Cc1ccccc1 c1(C(=O)NC2CCCN(C(c3c(C#C)c[nH]n3)=O)C2)cnc(C)cc1Cl Cc1ccc(C(CNC(C2CCCSC2)=O)NC(C2CC(C)(C)C2)=O)cc1 C1(F)(CNC(C2CCCO2)=O)COCCN(C(=O)C=CCN2CCOCC2)C1 C1(COC)CC(CNC(C2CC23CC(O)C3)=O)N(C(c2ccccc2Cl)=O)C1 c1(C(=O)NC(CCNC(c2c(CC)nc(C)o2)=O)(C)CC)ccc(OC)c(C)c1 Cc1ccc(NC(C2(C)CCN2C(c2cc(C(F)(F)F)cc(Br)c2)=O)=O)c(Br)n1 C(CC(C(=O)N(C)Cc1nc(C)ns1)NC(c1nn(C)cc1C)=O)=CC c1(C(C(=O)N(CCNC(=O)CN(C)C(N)=O)CC)C)c(F)cccc1F N1(C(C(CC)C)=O)CC(NC(c2ccc3nncn3c2)=O)CC(F)(F)C1 C(=O)(C(C)CC=CC)N(CC(=O)NC(CC=C)CC)CCC O=C(CCCCSc1ccccc1)NCCC(O)CNC(=O)CCn1cccn1 CC(CC(C)(c1ccccc1)NC(=O)CCCC(=O)N(C)C)C(=O)O CC1CCc2onc(-c3nc(-c4cccc(Cl)n4)nn3C3CCSC3)c2C1 c1(C(=O)NC(C)CNC(C2COC(=O)O2)=O)ccc(C(=O)N(C)C)cc1 c1(C(=O)NCCSC2CC(OC)C2)cc(C)n(-c2ccc(C3CC3)cc2)c1C Cc1cccc(CNC(=O)CCN(CCCO)C(c2cccnn2)=O)c1O.C1CC1 Cc1cc(C(N2CC3(CC(CC(=O)N(C(C)C(C)N(C)C)C)C3)C2)=O)ccc1O N1(C(CCc2ccc(C)cc2)=O)CCC(C(=O)NCC2CC(C(C)C)C2)=C(F)C1 Cc1ccc(C(=O)NCC2(F)CCCN(C(C3(N(C)C)CC3)=O)C2)c(C2CC2)n1 C1(C2CN(C(=O)C=C(C)Cl)C2)(NC(C2CC(C(F)(F)F)(OC)C2)=O)CC1 N(C1CCOc2cc(Cl)ccc21)C(N1C2CN(C)C(C2)C1)=O c1(N2CCC(CCOC)CC2)nc2c(c(=NCC3CCOC(C)C3)[nH]1)CCC2 C=CCC(C)(O)C(=O)NC(c1ccccc1)C(=O)NCCC(O)C(F)F c1(C(=O)NCC(CNC(CC2N(CC)CCOC2)=O)O)cc(F)ccc1F C1(C(N(CC(C)N(C)C(c2coc(O)n2)=O)C)=O)COCOC1 CCC(C(=O)N1CC(N2CCN(C(=O)Cn3nnc(C)n3)CC2)C1)C(C)(C)CC C(C(C)(C)CNC(c1cn(C2CC2)nn1)=O)N(C(=O)C(C)N(C)C(C)=O)CC c1(C(=O)NCC(C(=O)NCCNC(N)=O)OC)ccc(Cl)c(Cl)c1 CCC(CC)C(C(=O)N(C(CC)CC(N1CCC(O)C(CO)C1)=O)C)N(C)C C12(C(=O)OC)CC(C(N3CCCC3c3nn[nH]n3)=O)(C1)C2.C12CCN(C1)C2=O Cc1c(C(N2CCC(NC(=O)C(C)(C)CCl)C(F)C2)=O)ccnc1Cl Cc1cc(F)cnc1C(=O)N(C1CCN(C(C2CC(C)(F)C2)=O)CC1)C C1(C(=O)NCCC2CCCCN2C(=O)C=Cc2cscn2)CCOCC12CCC2 Cc1ccc(CNC(=O)CC2CC(C)N(C(C3CC(N(C)C)C3)=O)C2)cc1O c12oc3ccccc3c1COCCNC2=O.C1(NC(=O)C2CC2)(CF)CCC1 Cc1nc(NC2CCN(C(=O)CC3CCOCC3)C(C)C2)cc(C(F)(F)F)n1 N1(C(C2N(C(c3c(NC)cccc3)=O)CCCC2)=O)CCN2CCCCC2C1 c1(C(=O)NC(C2CCN(C(=O)C=CC3CCCC3)C2)C)ccc(Br)cc1O c1(OC)cc(C)c(C(=O)NC(CNC(=O)C2=CCCS2)C2CCC2)cc1OC CC(C)(CCCNC(=O)CNC(=O)C1CC1)NC(=O)CNCC1CCOCC1 C1(O)(C(C)NC(C(CC=C)C)=O)CCN(C(=O)COc2cncc(Cl)n2)CC1 c1(C(N2CCCC(CN(C(=O)CC3CCCO3)C)C2)=O)ccc(C2CC2)nc1O c1(C(N2CCC(C)C2C(N2CCSCC2)=O)=O)cc(O)cc(F)c1 C1(CNC(C(CC)c2cccnc2)=O)CCC(C)(C)CN1CCC1CCCCC1 c1(C(N2CC3=C(CN(C(C(CCSC)O)=O)C3)C2)=O)ccc(F)c(C)c1C#N S(=O)(=O)(c1ccc(NC2CSC2)cc1Br)NCCC1CC(C)(C)C1 CCC(CCC(=O)NC(C)(COC)CC)NC(C1CC1c1ccco1)=O c1(C(=O)NC(CC=C)CNC(=O)Cc2ncc(C)o2)cc(C)c2[nH]cnc2c1 C12(C(N3CC(NC(C(C)OC)=O)(CO)C3)=O)CC(C)(C1)OC2C N1(C(c2c(C)ccs2)=O)CC(C(N2CCSCC2C2CC2)=O)C2(CCC2)C1 O=C(C1=CC2CCCCC12)NCCN(C(=O)COCC(F)F)Cc1ccccc1 c1(C(=O)NCCC(CNC(=O)CC2CC(F)(F)C2)O)cc(Cl)ccn1 Cc1cc(C(N2CC(NC(c3ccc(C)s3)=O)CC(C)C2)=O)n2ncnc2n1 N1(CCNC(N2CC(F)(c3ccccc3)C2)=O)CCOC(c2ccccc2)C1 C1(CC)C(C(=O)NC(C2CCCCC2)CO)CCN1C(C1COCC1C(N)=O)=O C1(C(=O)Nc2ccc(SC)cc2)CCC(C)N(C(=O)Cc2cc(F)ccc2F)C1 C(=O)(C1=CCCCO1)N1CCC(NC(c2c(C)nn[nH]2)=O)(CO)C1 c1(N(CC(C)NC(=O)CN2CC3CC3C2)C)ccnc(C2CCCC2)n1 Cc1cc(C(=O)N(C)CC2CCCN2C(c2cscn2)=O)ns1 CCCCC(C(=O)N(C)CCOCCNC(=O)Cc1cncn1C)C(C)C N1(C(C2(COC)C=CCC2)=O)CCN(C(=O)C(O)C2CCCC2)C(CCOC)C1 c1(C(=O)OCC)cnn(C)c1C(=O)N(C)CC1CCN(C(C2CC2(Cl)Cl)=O)C1 C1(CC(C)NC(=O)CC2(O)CCC2)CN(C(=O)COC2CCC2)C1 CC(C)C(C)(O)C(=O)NCCn1cc(C(=O)NOCCOC2CC2)nn1 N1(C(CCC(C)OCC)=O)C2CCC1CC(N(C(=O)C(=CC1CCCC1)C)C)C2 N(C(=NCc1ccccc1F)NC1CC(C(=O)OC(C)(C)C)C1)C(CC)CC Cc1ncc(F)c(N2CCN(C(C3CC(=O)N3)=O)C3CC23)n1 Cn1c(C(=O)NC2CC2NC(C2CC=CCC2)=O)nnc1S c1(CC(=O)NC2(C)CC(NC(CC(C)(C)O)=O)C2)c(F)cccc1F c1(N2CC(CNC(c3[nH]ccc3-c3cccs3)=O)OCC2)ncnc2[nH]ccc12 C(=O)(CCC(CF)CF)NC1C2CC(C(=O)NC(C)(CO)C3CC3)C(C2)C1 C#CCCCCCCC(=O)NC1CCCN(C(=O)CC(O)CCC)CC1 C(C(O)CC(=O)NC1CCC(=O)NC1)NC(C=C(CC)CC)=O C#CCC(C(=O)N(C(C)CNC(c1snc(O)c1Cl)=O)CC)C1CC1 C(N=c1[nH]c(=N)[nH]c(=NCC(F)(F)CC2CC2)[nH]1)C1N(C)CC(O)C1 c1(C(=O)NCC2CCCCC2NC(c2cnns2)=O)nc2cncnc2nc1O CC(C)C(C)C(=O)NC1CCOC1C1CCN(C(C2(O)CC(F)(F)C2)=O)CC1 c1(C(N(C)CC2N(C(C=CC=CC)=O)CCOC2)=O)ccc(F)c(Br)c1 C12(C(N(c3ccn(C)n3)CC)=O)CC(CN(C(C3CCCCC3C)=O)C1)C2 S(=O)(=O)(c1ccc(F)cc1)N(C)CCNC1CN(C(=O)CC(F)(F)F)CCN1 N1(C(C(C2CCOCC2)C)=O)CCOCC(CNC(=O)CC2CC(CF)C2)C1 C1(c2nnnn2CCCF)(Nc2ccc(C(=O)NC)c(F)c2)COCC(C)(C)C1 Cc1cc(=NC(=O)C(=O)N(C)C[Si](C)(C)C)[nH]n1C1(CCN=[N+]=[N-])CC1 N1(C(c2cc(CC)ncc2)=O)CC(C(=O)NCC(C)(C)CC)CCC1(C)C CCC(C)C(C(=O)NCC1(C(N2CC3C=CC3C2)=O)CCC1)N(C)C c1(C(=O)NC(C(C)NC(C2C(CC(C)C)C2)=O)CO)ccc(N2CCCC2)c(F)c1 c1(C(N2CC(C(C)NC(C(C)(C)NC(=O)NCCC)=O)C2)=O)cnn(C)c1CC N1(C(=O)OC)CCCC1C(=O)NC1(C(=O)NC2CC2)CC(O)C1 N1(C(C(F)OC)=O)CCN(C(=O)CCSC)C(CC(C)(C)C)C1 C(=O)(C1=C(F)CN(C(=O)C(C)(F)F)CC1)N1CC(C)C(CCO)C1 Cc1ccc(NC(C2OCCC2CNC(c2ccccc2)=O)=O)cc1C Cc1ccc(C(=O)NCC2C(C(=O)NCC3CCOC3=O)C2(C)C)nc1O N1(C(CCC(=O)NC)=O)CC(C(=O)O)C2(C1)CN(C(=O)C(c1ccccc1)O)C2 c1(C(=O)NCC#CCNC(C2C(C)(C(F)F)C2)=O)ccc(-c2nnc(O)o2)cc1 N#Cc1c(NC(C2CC(F)CN2C(=O)C2=NNC(=O)CC2)=O)cccc1Cl C1(CCC)CN(C(=O)C(CC)N(C(=O)CCc2nc(C)no2)C)CC1CO C(C(C)(CC(C)C)NC(=O)C(c1ccc(C)cc1)C)NC(CCC(=O)NCC)=O CCCCC(CC)C(=O)N1CC(CN(C)C(c2ccc(F)o2)=O)C1 C(CC(=O)N1CC2CCC1CC2)(C(F)(F)F)NC(C(C(=O)OC)C)=O c1(OCC(=O)N(C2CCN(C(c3cc(CC)oc3C)=O)C2)C)ccc(Cl)cc1Cl N1(C(C2=NOC(C)C2)=O)CC2(CCN(C(=O)CC3CCOC3)CC2)C1 C1(C(=O)NCCC2OCCN(C(C3(C)CS(=O)(=O)C3)=O)C2)CCC2(CCC2)CO1 c1(C(=O)NCC2N(C(C3ON=C(C)C3)=O)CCCC2C)ccc([N+](=O)[O-])cc1Cl C(=O)(C1CCc2nccn21)NC(C(=O)NCC(CC)(C)CC)C(C)OC Cc1ccc(NC(C2CN(C(C3CCCC34CCC4)=O)CC2F)=O)c(O)n1 c1(OC)cc(C(=O)NC(c2ccc(SC(C)C)cc2)C)ncc1Br c1(CNS(=O)(=O)c2nc[nH]n2)cc(F)c(F)c(F)c1F C12CCN(C1)C2=O.N1(CCNCCC(=O)OCC)CCOCC1 N1(C(C=CC)=O)CCN(C(c2conc2Cc2ccccc2)=O)CCC1C N1(C(C2CC(C)C2)=O)CCN(C(=O)CC2CN(C)C2)C(C2CC2)C1 C12(CCNC(c3c(C)nc(CCC)o3)=O)CCC(C1)N(C(C1(SCC)CC1)=O)C2 C1(C(=O)NC(c2ccc(C)s2)C)CCn2cncc2C1 CCCCC(CCC)N=c1[nH]c2c(c(=NCc3cn(C4CC4)nn3)[nH]1)CSC2 CC1CN(C(=O)CC(C)(C)c2ccc(F)cc2)CC1NC(c1cc(C#N)cs1)=O c1(OC)ccc(NC(=O)CN(C)CC23CC2CCN3)cc1NC(C)=O C1(C(=O)NC2(CCCC)CC2)COCCN(C(c2ccnc(OC)c2)=O)C1 N1(C(C(C(CC)CC)C)=O)CCC(NC(=O)Cc2c(C)cnn2C)CC(C)(C)C1 CC(C)C(C(=O)N1CCCCCC1CNC(=O)C(C(C)O)N(C)C)C(C)C C#Cc1cccc(C(=O)NCCC2CN(C(=O)COC3CC3)CC(C)O2)c1F C=C=C(C)CC(=O)N1CCC(N(C(C2(N3CC4CC4C3)CC2)=O)CC2CC2)CC1 Nc1cnc(C(N2CCC(O)(CCNC(c3cnncc3O)=O)CC2)=O)c(Cl)c1 C1(COC)CN(C(=O)C(C2CCOCC2)F)CCN1C(c1nc(Cl)cs1)=O C(=O)(CN=c1ccc(Cl)n[nH]1)N1CCN(C(CS(CC)=O)=O)C2(C1)CCC2 C1(C(=O)NCC(CC)N(C)C(c2[nH]nnc2C)=O)CC2(CCO1)CC2 c1(OC)ccc(C(N2CC(C)(NC(C3CCCC(F)C3)=O)C2)=O)cc1 Cc1cc(O)cc(C)c1NC(=O)CC1CC1CNC(C1CC1Cl)=O Cc1ccc(C(N2CC(NC(c3cncc(F)c3)=O)C(C#N)C2)=O)c(C)c1 CC1(C)CCC(CO)N(C(C2CN(C(=O)Cn3cnnn3)CC2(F)F)=O)C1 C1(C(N2C(C)CCCC2)=O)CC12CCN(CC(=O)Nc1cc(C#N)ccn1)CC2 CC1(C)OC2(CNC(C3(C)C=CCC3)=O)CC1(NC(C1CC1(C)C)=O)C2 N1(C(CSCCCC)=O)CCN(C)C(CNC(=O)COC2CCOC2)C1 N1(C(C(C)SCCCC)=O)Cc2ccccc2C(NC(c2cnc(S)[nH]2)=O)C1 C1(CNC(c2nn(CC)nc2C)=O)CC2(CC(NC(c3cc(OC)no3)=O)C2)C1 C1(NC(C2(COC)CC(F)(F)C2)=O)CCN(C(c2sccc2F)=O)CC1O C(=O)(C(O)CCCc1ccccc1)NCCCN(C(C1N(CC)CC1)=O)C N1(C(Cc2ccc(OCC)cc2)=O)CC2OCCN(C(=O)C(O)CC(C)C)C2C1 C=CC(CC(=O)N1CC(NC(c2csc(C#N)c2)=O)C(O)C1)c1ccccc1 c1(C(=O)NCCNC(c2cccc(OC)n2)=O)cccn(C2CC2)c1=O C1(NC(C2CCCC23CC3)=O)CN(C(c2ccoc2Cl)=O)CC1O C#CCCCC(C)C(=O)N1CCCC1C(=O)NCCc1ncc(C)o1 c1(OC)ncc(Cl)cc1C(=O)NC1CC(CNC(=O)C(C)c2ccco2)CC1O c1(C(N2C3C(NC(CCNC(C4C(C)C4)=O)=O)C(C3)C2)=O)ccc([N+](=O)[O-])c(C)c1 O=C1CC(CC(=O)NCC2CCCN2C(c2cnns2)=O)CCCN1 C1(NC(c2cc(SC)oc2C)=O)CCSC12CN(C(=O)C(c1ccccc1)F)C2 N1(C(c2nnc(CC)s2)=O)CCN(C(=O)C(CC(C)C)OC)C(CO)C1 C1(C(N2C(C)CCCC2)=O)CC(c2ccccn2)=NO1 N1(C(C=CC)=O)CCCC(C2CCN(C(=O)C(CC3CC3)CC3CC3)C2)C1 c1(OCC)ccc(CNC2CC(C(N3CCC(CSC)C3)=O)C2)cc1OC C1(CN(C(C2CCC2(F)F)=O)CC)CCN(C(c2ccc(Sc3nc[nH]n3)o2)=O)C1 C(C(C(C)(C)C)NC(=O)CCc1ncccc1C)NC(C(=O)NCC)=O CCC(C(=O)N1CC2CCC2(NC(c2nnc(O)cc2O)=O)C1)C(C)C CC1OC2(C)CC1(C(N1CCC(CNC(c3ccnc(F)c3Cl)=O)C1(C)C)=O)C2 C1(NC(=O)CCN2CCCC2)CCN(C(c2ncn3c2CCC3)=O)C12CCC2 c1(C(N(CCC(C(C)C)NC(COC(CC)C)=O)C)=O)ccnc(F)c1OC c1(OC)ccc(CC(N2CCC(C)C2CNC(=O)CS(N)(=O)=O)=O)cc1O c1(OC)ccc(S(C)(=O)=O)cc1C(N1CC2CN(Cc3coc(C)n3)CC2C1)=O c1(C(=O)OCC2CC3(CCCO3)C2)nc(O)c(C(c2cccc(C)c2)=O)cc1C N1(C(CCCSC)=O)CCC(NC(c2cnccc2C(C)(C)C)=O)C(F)C1 C1(NC(C(C)SC(C)C)=O)CCN(C(=O)CCNC(=O)CO)CCC1(F)F C(C(O)CC(=O)N1CC(F)CC1CN(C)C(c1cc(CO)n(C)n1)=O)N(C)C C1(C(N2CC(CC(=O)NCCc3cscn3)OCC2)=O)CC2(CCO1)CC2 N1(c2cc(COC)ncn2)CCN(C(c2cc(Cl)ccc2Cl)=O)CC1C1CC1 C1(C(=O)NCC(CN(C)C)(C)O)CCCC(NC(=O)C=Cc2ccncc2)CC1 c1(CC)cc(C(N2CC(NC(c3cc(F)c[nH]3)=O)C(F)C2)=O)cc(C)c1 c1(C(=O)NC2C(NC(c3nc(C(C)C)sc3)=O)COC2)ccnc2ccccc12 O=C(C(F)C(F)(F)F)NCc1ccc(NC2(C3CCCO3)CC2)cc1 N1(C(C(C)C(C)(C)C)=O)CC(NC(c2ccccc2[N+](=O)[O-])=O)CC(C)(C)C1 c1(CCCC(=O)NCC2CC(F)(CNC(CC(=C)Br)=O)C2)nnc(C)n1C c1(OC)c(Cl)ccc(C(N2CCCN(C(=O)CC3C=CCC3)C(CO)C2)=O)c1F C1(NC(CNC(C2C(C)C2)=O)=O)CC2C(NC(C3CCC4(CC4)C3)=O)C2C1 c1(C(=O)NC2CC(NC(C(CC)n3cccn3)=O)C2)nn(C(C)C)cc1Br c1(CC)cccc(C)c1NC(=O)Nc1ccc(Cl)nc1OC C(=O)(CCCCCC(C)O)NCC1CC(O)(CNC(c2cc(CC)nn2C)=O)C1 C1(C(=O)NCC=CCC(=O)NCC(CO)OC)CNC(=O)N1 C1(F)(C(=O)NCC2C(C)(C)C2CO)CCCN(C(=O)CC2CCC(=O)N2)C1 c1(C(=O)NCC(C)(C2CC2)NC(c2cnccn2)=O)c[nH]nc1-c1ccccn1 c1(C(=O)NCC2CC(CNC(CCC)=O)OC2)cc(F)c2[nH]nnc2c1 c1(CC)cn2c(C(=O)NCCC3CN(C(=O)C(C)=O)CC3C)cccc2n1 N1(C(C(C)(C)C#N)=O)CCC2(CC1)COC(CNC(=O)C=CC1CCOC1)C2 CCC1=C(C(=O)NC(C(C)NC(c2cc(Cl)c[nH]2)=O)C(C)C)SCCO1 C1(C)(C(N2CCC(C)(CNC(C(C)=C(CC)C)=O)CC2)=O)CCC(=O)N(C)C1 C(=O)(C(CN(C)C)C(C)C)NC(C(N1C(CC)(CC)CC1)=O)Cc1ccco1 c1(C(N2CC(O)CC2COC)C(=O)NCC(=C)C)c(Cl)ncn1C c1(C(=O)NC2CC3CN(C(CCOC)=O)C(C2)C3)cccc2cccc(OC)c12 N1(C(C(C)SCCCC)=O)CCC2CN(C(=O)C(CSC)OC)C(C)C12 CC#CC1CCN(C(=O)CC(CNC(c2cc(C#N)[nH]c2C)=O)OC)C1 c1(C(=O)NC(CNC(c2cnn(CCC)c2Cl)=O)(C)CO)ncnc2c1CCC2 C1(C)(C(=O)NCCC(=C)C)CCN(C(=O)C=C(C)c2ccccc2)CC1 CC1OC2(C(N3CC4CC(NC(c5cnnc(O)c5)=O)C3C4)=O)CCC1CC2 C(c1nc2ccccc2o1)=CC(=O)NC1CCN(C(C=C(CC)C)=O)CC1CO c1(SCC(CC)N(C)C)nnc(-c2ccc(OC)cc2)n1CCC#N N1(C(c2c(SC)scc2)=O)C2CCC1C(CNC(=O)C(O)CC(F)F)C2 Cc1ccc(C23CC(C(=O)NCCc4cc(C)n(C)n4)(C2)C3F)cc1 n1(C(C)C)ncc(F)c1C(N1CCCC(C(C)NC(=O)C=Cc2ccco2)C1)=O c1(C(N2C(CNC(C3CCCO3)=O)CC(C)(C)C2)=O)cc(Br)c2c(c1)OCO2 C12(C(=O)NCC3N(C(CCC(C)(F)F)=O)CC3)CCOC1CCOC2 N1(C(CCOCCCOC)=O)CC2CCC(C1)N2Cc1ccc(C)cc1F N1(C(c2cnc(C(C)C)s2)=O)CCC(C)(NC(c2n[nH]c(C(C)(C)C)n2)=O)C1 N1(C(CCC(C)OC)=O)CCN(C(c2ccc(C)cc2N)=O)CC1C1CC1 c1(CNC(C(C(C)SC)O)=O)c(C)nn2c1CN(C(=O)CCCSC)CC2 c1(C(=O)NCC2CCC(NC(Cc3cc(C)on3)=O)C2)c(Cl)ccc(F)c1C N1(C(C2N(CC)CC2)(C)C)CCC(C)(CC(=O)NCC(n2ccnn2)C)C1 N1(C(c2c(C)nccn2)=O)CCCC12CCCN(C(=O)Cc1ccc(Cl)cc1)C2 C1(C(F)(F)F)(C(=O)OC)CCN(C(=O)NCCc2occc2C)CC1 CCC(C(=O)N(C1CCN(C(C2(C)CCCCC2)=O)C1)CCO)C(C)(F)F C1(CC(=O)N(C(CC#C)C)C)CC(C)N(C(=O)CSCCC)C1 C1(NC(C2CC3CC3C2)=O)CN(C(=O)Cc2csnn2)CC1C(F)F C1(NC(C23CC(C)(C2)C3)=O)CCCN(C(=O)C(=O)NC2CCCN(C(N)=O)C2)C1 C12(NC(C3N(C(=O)NC(C)C)CCC3)=O)CC1CN(C(=O)CC(O)CN(C)C)C2 C1(F)(CNC(C2CCCN(C(C)=O)C2)=O)CCCN(C(=O)CCC(C)C#N)C1 CC(C)CN(CC1CCCC1)N(Cc1ccsc1)CCOC C=Cn1nccc1C(=O)NCC1CC(NC(=O)CCNC(=O)CO)C1 C1(O)(C(=O)NC(CCC)CNC(c2c[nH]nc2Cl)=O)CCC(C)(C)CC1 C1(NC(C2CC(O)(CC#C)C2)=O)CN(C(=O)Cc2ccsn2)CC(C)(C)C1 C1(CNC(=O)CO)CC(CNC(c2coc(C(F)F)c2)=O)CO1 C1(NC(c2cc(C)on2)=O)CCN(C(C2CCC=CCC2)=O)CCC1CO c1(CC(=O)NC2(CN(C)C(C3CCCC(F)(F)C3)=O)CC2)cc(Cl)cc(Cl)c1 c1(C(=O)NCC2CC(NC(=O)CCF)C(O)C2)cccc2c1COC2 C1(C(C)(O)CNC(=O)CCc2cnc[nH]2)CCCN(C(=O)CP(C)(C)=O)C1 c1(C(N2C(CCNC(c3n(C)ncc3)=O)COCC2)=O)cnc2c[nH]nc2c1 CC1CCC(NC(C2CCC(=O)N2)=O)CN1C(C1CC(C)(C)CN1C)=O c1(C(=O)NCC(CO)NC(c2c(C)occ2)=O)ccc(F)c(C)c1N C1(NC2C(c3cn(C)nc3)CCC2)CC2(C1)CC2CNC(=O)OC(C)(C)C N1(C(C(CN(C)C)O)=O)CC(NC(c2csc(C(F)(F)F)n2)=O)C(O)C1 CC(C)CC(CNC(=O)C(C1(O)CCCC1)F)NC(c1cc(Br)cs1)=O c1(OC)ccc(O)cc1C(=O)NC1SCCC1C C1(C2CC2)(CNC(C(CCCC)N(C)C)=O)CCN(C(c2cc(C)c(C)[nH]2)=O)C1 OC1CC2(CC(NCc3sccc3Br)C2)C1 N1(C(c2ccc(C)nc2N)=O)CC23CCCCC2(C1)CN(C(C1(F)CC1C)=O)C3 c1(SC)ccc(Cc2cc(-c3ccccc3)cs2)cc1.N12CC(F)CC1C2=O c1(NC2C(NC(c3c(CC)nc[nH]3)=O)CS(=O)(=O)C2)cc(C#N)nc(C)n1 CC(CCCNC(c1cc(Cl)cs1)=O)NC(=O)Cc1nc(C(C)C)n[nH]1 C1(NC(CC(CCC)CC)=O)CC2CCCC(C1)N2C(C1CCS(=O)(=O)N1)=O C(c1ccccc1Cl)=CC(=O)NCC(C)(C)CNC(C1CC1CF)=O C1(NC(CCOCC#C)=O)CCC(C)(NC(=O)C(F)Cc2ccccc2)CC1 N1(c2cc(NCC(c3ccc(F)cc3)C)ncn2)CCc2ncn(C)c2C1 CCCC(C)(CC)C(=O)N1CCN(C(=O)CCn2cnnn2)C(COC)C1 C=C1Cn2c(C(N3CCN(C(c4c(C)ccn4C)=O)CC3CC)=O)nnc2S1 c1(CC(N2CCCC(C)(NC(c3c(CC)nns3)=O)C2)=O)ccc2nsnc2c1 C1(C(=O)NCC(CNC(=O)CCCn2ccnc2)O)CCCC2(CCOCC2)O1 c1(CC(=O)NC(CCNC(C(COC)N(C)C)=O)C)ccc2c(c1)COC2 C12(C(=O)NC(C)CCC3CCCO3)CC(CO)(CN1C(c1ccns1)=O)C2 C1(NC(C(C)=C(C)C)=O)CC2(CCN(C(c3cccc(C4(C)CCO4)c3)=O)C2)C1 C1(CC)CN(C(c2cccc(Cl)c2Br)C(=O)NC2CCCCC2)CC(C)O1 C1(C(N2C(CN(C(c3snc(C)c3N)=O)CC)CCC2)=O)C2CN(C)CC12 C12(SC(C(c3ccc(-c4ccc(OCC)cc4)cc3)=O)C)CC(C1)C(CO)CO2 c1(C(=O)NC2(C3CCCN3C(=O)CC3CC4(CC4)CO3)CC2)ccc(Cl)nc1O C1(C(C)C)CN(C(c2nc(Cl)cs2)=O)CCCN1C(c1cc(C(C)(C)C)c[nH]1)=O N1(C(CC2(N(C)C)CCCC2)=O)CCC(CCCNC(C2CCOC2)=O)CC1 C1(CC=C)(NC(C2OCCC2C)=O)CCN(C(c2sccc2NS(C)(=O)=O)=O)C1 C1(C(=O)NC2(CCCNC(C3C(CC)CCC3)=O)CC2)CC(F)C(=O)N1 Cc1nnc2n1CCN(C(=O)C(CNC(C1C=CCCC1)=O)CC(C)C)C2 c1(C(C)NC(=O)C(=O)NCc2cc(Br)ccc2O)nc2ccccc2n1C(F)F CC1CCOC(C(=O)NC(CO)CCCNC(C2CCC(=O)C2)=O)C1 C1(N(C(=O)Cc2c[nH]nc2O)C)CCCN(C(=O)C(O)C(F)F)C1 n1(CC)cc2ccc(C(N3CC(CNC(c4cnccc4OC)=O)C3)=O)cc2n1 c1(CNC(=O)NCC)ccc(S(=O)(=O)NCC2(CC(F)(F)F)CC2)cc1 C1(CC(=O)NCC(CCC)C)CN(C(c2cccc(CC#N)c2)=O)CC12CC2 CC(C)C(O)C(C)(C)C(=O)NC1CC(CNC(c2ccc(F)c(F)c2)=O)C1 Cc1cc(-n2ccc(C(=O)NCCC(C)(C)O)n2)ccc1Cl CC1(C)CCC=C1C(=O)N1CC2CCCC2(NC(=O)Cc2ccccc2Br)C1 N1(C(C(C2CCOCC2)OC)=O)CCN(C(=O)CCCN=[N+]=[N-])C(C2CCC2)C1 C(=O)(C1CS(=O)(=O)c2ccccc21)N(C1CCCC1)CCNC(c1csnn1)=O C12(CNC(c3cnc(OC)s3)=O)CN(C(C3CCCC(=O)C3)=O)CC1CCO2 CN1CC(O)CC1C(=O)NCC1(CCNC(=O)CN2CCC(F)(F)C2)CC1 c1(C(=O)NC(CC)CNC(=O)C(C)CC2CC2)noc2cc(F)ccc12 c1(C(=O)NC(CC)CN(C(=O)CCC2(C)CC2)CC)cccc(Cl)c1O N1(C(CSCC(C)C)=O)CC2CCCC(C1)N2C(=O)CNCc1ccccc1Cl CCCC(C(=O)NC(Cn1ccnn1)C(=O)NCCCCS(C)=O)OC c1(C(=O)NC(c2ccc(F)cc2)C(=O)NC)cn2c(n1)CCCC2C(=O)O N1(C(CCOCCOC)=O)CCc2c(ncn2C)C12CCN(CC1CCOC1)C2 N1(C(c2occ(C)c2)=O)CCN(C(=O)CCC2OCCO2)CC1CO C12(C(=O)NC(CN(C(Cc3ccc(C)cc3)=O)C)(C)C)C3C4C1C1C2C3C41C C(=O)(CC(C)(CC)C(=O)OC)NCc1cccc(NC(C(F)=CC)=O)c1 C#CCC(CC(=O)NC(C1CSC1)C)NC(=O)CSCCN(C)C c1(CN2CC3N(C(c4cccc(O)n4)=O)C3C2)c[nH]c2ncc(Br)nc12 Cn1nc2c(c1C(=O)NC1CCCCC1NC(c1ccc(=N)[nH]n1)=O)CCC2 N1(C(C(C)=CC2CC2)=O)CC(F)(F)CC1CCNC(=O)Cc1scnc1C c1(C(CNC(C2C(C)C2)=O)NC(=O)CC2(N(C)C)CCC2)ccccc1Br c1(OC)cc(C(=O)NC2CN(C(C3CCCC3)=O)C2)cc(Br)c1OC(C)C c1(C(N(CCCNC(C2(C)CCCN2C)=O)C)=O)cnc(S(C)(=O)=O)s1 c1(C(=O)NC(CNC(C(C)N2CCC2)=O)C2CCC2)cc(C(N)=O)co1 c1(C(=O)NC2C(NC(C(C)NC(c3ccoc3)=O)=O)CC2)cc(Cl)cnn1 C1(CC)CC(C(=O)NCCN(CCOC)Cc2noc(CCCO)n2)CCO1 C(=O)(C1Cc2ccc(F)cc21)N1CCN(C(C(COCC)C)=O)CC12CCC2 C1(C#CC(=O)N2CCC(C(C)(O)CNC(=O)Cc3cc(C)on3)CC2)(CC)CC1 C1(NC(C(=O)NCC2CC(COC)C2)=O)CC(C)(C)CN1 C1(NC(c2cc(Cl)c(Cl)[nH]2)=O)CN(C(=O)C(F)F)CCC1c1ccccc1 c1(C(=O)NCCNC(CCCc2scc(C)n2)=O)cc2c(F)ccc(F)c2[nH]1 C1(NC(CCOc2ccc(C)cc2)=O)CCN(C(c2ncc(F)cn2)=O)CC1C C1(CCC(=O)OC)CCC(C(=O)NCC(C)(O)CNC(=O)C(C)C)O1 C(=O)(C1CCc2c[nH]nc21)NC(CC=CC)C(=O)O C1(NC(=O)CC2CC=CCC2)CC(F)CN(C(c2cc(Cl)ccc2O)=O)C1 N1(C(C(CC2CN(C(C=C(CC)CC)=O)C2)F)=O)CC(O)CC(C)(C)C1 c1(NC(C23N(C(C(C)NC(CC)(C)C)=O)CCC2C3)=O)cnc(C)c(C)c1 N1(C(C)C(N2CC(O)(C(C)NC(=O)CCn3cnnn3)C2)=O)CCCCC1=O c1(CNC(c2ccccc2)C2(NC(COCCCCC)=O)CC2)n[nH]c(C)c1Cl Cc1cc(C(=O)Nc2cccc(NC(c3cc[nH]c3C(C)C)=O)c2)cn1C c1(OC)cc(CNc2ccccc2N2CCC(CO)C2)ncn1 CC1CCC(CNC(=O)C=C2CCC2)N(C(=O)CN(c2ccncc2)C)C1 c1(C(=O)NC(CC(C)C)C(F)F)c2ccccc2nn1C CCCC(C(=O)OC)C(=O)N1CC(NC(c2cc(C(C)C)[nH]n2)=O)C(N=[N+]=[N-])C1 N1(C(C)C)CCCC1C(=O)NCCOCCN(C)C(c1ccccc1)=O.CO N1(C(C2ON=C(CC)C2)=O)CC(N(C(=O)C(c2ccccc2)=O)C)C2(CC2)C1 CN1CCOC(C(=O)N(CCCNC(C2CNC(=O)N2)=O)CC2CCCC2)C1 c1(CNCc2nc(-c3ccc(OCC)cc3)oc2C)cc(Br)cc(Cl)c1F CC(C)C(CNC(=O)CCCn1ccnn1)C(=O)N1CCC(C(C)C)(N(C)C)C1 N1(C(CSCCC)=O)CCC2(CCN(C(c3cc(Cl)ccc3OC)C)C2)C1 N1(C(CNC(CNC(C)=O)=O)=O)CCC(F)(CNC(c2cscc2Cl)=O)C1 C(c1ccc(C)cc1)=CCC(=O)NCCN(C(=O)CCC(C)N(C)C)CCOC N1(C(C2C(C(=O)OC)C2)=O)CCC(n2cc(-c3csc(C(=O)O)c3)nn2)C1 C(CCC(C)C(=O)N1CCC=CC1C(=O)NCCCC(=O)NO)OC C1(F)(CNC(c2c(CC)nc(C)[nH]2)=O)CCCN(C(C2(C3CC3)CC2)=O)C1 CCC(C(=O)NCCCC(C)NC(C1(C(N)=O)CC1)=O)C(C)C O=C(CCCC(F)(F)C(F)(F)F)NC1CCN(C(C2(F)CCC2)=O)CCC1CO N1(C(c2c(C)nccc2)=O)CCC(C)C(NC(c2cc(C)n(CC(F)F)n2)=O)C1 C1(NC(CN(C)CC)=O)CC2CN(C(c3cc(C)nn3C)=O)CCN2C1=O c1(C(=O)NCCCCN(C(CS(=O)(=O)NC)=O)C)cc(F)ccc1C(F)F c1(C(=O)NCC(C2CCCC2)NC(=O)CCc2cnn[nH]2)cc(Cl)ccn1 c1(C(=O)NCCCCCNC(C2N(CC)CC2)=O)cnc(C(F)(F)F)cc1C C1(C(=O)NC(C)COC(F)F)CCN(c2ccccc2C(F)(F)F)C1=O c1(NC(C2CC(=O)C2)=O)ccc2cnn(Cc3ccccc3)c2c1 N1(C(CC=C=C)=O)CC(NC(=O)CCc2ccccc2OCC)CC2(CCC2)C1 C(=O)(C#CC1CCCOC1)N(CC(C)N(C(c1c(C)c(Br)cnc1)=O)C)C c1(C(N2CCC(N(C(CC)=O)C)C2)=O)cccc2c1CCCCC2 c1(C2(C(C)C(N3CCOCC3C3(C)CC3)=O)CC2)ccc(Br)cc1 C1(NC(C2(C=C)CCC2)=O)CCCCC1NC(=O)CCN(C(CC)CC)C C1(C)(C(=O)NCCC2OCCN(C(CC(C)(C)OC)=O)C2)COCC1(F)F C(N=c1nc2[nH][nH]cc-2c(O)n1)C1(NC(Cn2ccc(C)cc2=O)=O)COC1 N(C1CCc2cc(CNC(C3(C#N)CC(=O)C3)=O)ccc21)C(C1(C)CC1(Cl)Cl)=O C=CC1(C(=O)NCCC2(O)CN(C(c3ccc(CCC)[nH]3)=O)C2)CCC1 N1(C(c2n(CC)ncc2Cl)=O)CCN(C(c2nccc(Cl)c2C)=O)CC1CO N1(C(C2CCCS2(=O)=O)=O)CCCC2(CCCCN2C(=O)C(O)O)C1 c1(C(=O)NC2CN(C(c3[nH]cc(CC)c3)=O)CC2C(F)F)cccc2[nH]ccc12 C1(CC)C(=O)N(C)CCN1C(C1CN(C(c2cc(C)cs2)=O)CCC1(C)C)=O CCCCC(C)CCC(=O)N1CCC2CCCC12C(=O)NCCCc1nncs1 N1(C(C(C)Cc2ccncc2)=O)CC2CC(NC(=O)CN3CCCCCC3)C2C1 c1(C(=O)NCC(CNCC(=O)NC2CCC2c2nc[nH]n2)F)cc(Cl)ccc1Cl C1(CNC(c2cn(CCNC(c3cccc(F)c3O)=O)nn2)=O)CC2CCCC2C1 C#CCC(CC(=O)NC1CC2(CCCO2)C1)NC(c1cc(Cl)c[nH]1)=O CCC(C)(C#N)C(=O)NC(CC(=O)N(CC(C)C(C)C)C)C(C)OC N1(C(CNC(c2cn(-c3ncc(Br)s3)nn2)C)=O)CCN(C(=O)C2CC2)CC1 c1(C(N2C(C)(CNC(C3C(C)(C)C3)=O)CCC2)=O)cc(Br)cnc1N c1(CC)[nH]nc(C(=O)NC2CC3CC2CN(C(=O)C(CSC)OC)C3)c1[N+](=O)[O-] c1(NC(c2ccn(C3CN(C(C(C(=O)OCC)OC)=O)C3)c2)=O)cc(C)cc(F)c1 C1(NC(CCCCOCC)=O)CC=C(C(=O)NC2(C)CCC(C)(C)C2)C1 N1(C(C2(O)CC(C)(C)C2)=O)CCCC(CCNC(c2cccnc2F)=O)CC1 C1(NC(c2ccc(=O)oc2)=O)CCN(C(=O)CC2CCCCC2O)C12CCCC2 Cc1cc(=NCCCCC#N)[nH]c(=NCCOCCS(N)(=O)=O)[nH]1 c1(C(=O)NC2(CO)CN(C(COCc3cc(C)no3)=O)C2)cc(Cl)c(C)cn1 C1(C(N2CC(O)(CNC(CCCC(C)O)=O)C2)=O)CS(=O)(=O)CC(=O)N1 C(=O)(C1=CCc2ccccc21)N1CC(N(C(C(CC(C)C)OC)=O)C)C(C)(C)C1 C(=O)(C(CO)C(C)(C)C)NC1(C(N2CCC(C(C)(C)C)C2)=O)CCCC1 Nc1nccnc1C(N1CCCCC1CC(N1CCC(CO)CC1)=O)=O N1(C(c2cc(CC)no2)=O)CC(CC(=O)NOCCCOC)C(C)C1 C1(C)(C(N2CCC(C(N3CCN(C(=O)OCC)CC3)=O)CC2)=O)CNCCC1O Cc1cc(NC(C)CCNC(=O)COCc2cc(C)on2)n2nc(C)cc2n1 N1(C(CN(C(C(CC)C)=O)C)=O)CCN(C(C2C(C)(C)C2(F)F)=O)CC1 CC1CC=C(C(=O)N2CCC2CNC(=O)Cn2ccc(Br)n2)CC1 C1(NC(c2cccc(Br)c2Cl)=O)CCN(C(=O)NCCCl)CC1O C(C)(C)(CC(F)C(=O)N(C)CC1(N(C)C)CCC1)NC(c1cncc(C)n1)=O C1(CNC(=O)CCC2CCCC2)CC2CCC1N(C(c1c[nH]nc1Br)=O)C2 c1(OC)ccc(CC(=O)NCC2CC(NC(=O)CC=C(C)C)C2(C)C)c(F)c1 C12(CNC(CN(C(COC(C)C)=O)C(C)C)=O)CCC(CC1)CC2 Cc1cc(C(C)C(=O)NCCCCN(C)C(C2C3CCC(F)(F)C23)=O)cc(F)c1 c1(CC(=O)NC2CCN(C(C=CC)=O)CC2O)nnc(O)c2ccccc12 Cc1cc(-n2cc(CNC(=O)C(C)C3(c4ccccn4)CC3)nn2)cc(C)c1Br C1(C(=O)NC2CN(C(c3c[nH]c(=NCC)s3)=O)CC2(C)C)CCCC2C1C2(F)F N1(C(C(CC)COC)=O)CCCC(C)(C)C1C(=O)NC1CCC2CCC12 C12(C(=O)NCCc3ccc(C(=O)NCc4cnc[nH]4)cc3)CC=CCN1CCC2 N1(Cc2ccc(OC)c(SC)c2)CCC2(CCC(O)C2)C1 CCCCC(O)C(=O)N1CCOCC(NC(c2cc(C(=O)OCC)n(C)n2)=O)C1 C1(NC(c2c(CC)nc(CC(C)C)cc2)=O)CC(N=c2nc(C3CC3)[nH]s2)C1 CCCC(C)(O)CNC(=O)CN(C1CCN(C(C2CCCN2C(C)=O)=O)C1)C c1(C(N(C2CCN(C(=O)CCC(C)(C)O)CC2)CC)=O)ccc2c(c1)OCCO2 Cc1ccnn1C(C)C(=O)NC1CC(CNC(c2csc(CC(C)C)n2)=O)C1 Cc1cc(C(N2CC3CC2C3C(=O)NCc2ccccc2F)=O)nc2nccn12 O=C(CCCCC(F)(F)F)CO.C12(CCS(=O)(=O)C1)c1noc2n1 C1(NC(CC2(OC)CN(C(CCSCC)=O)C2)=O)CCCN(C)C1C c1(C(N2CCC(CNC(CCC(=O)NC)=O)C2)=O)sc(C#N)cc1Cl C(CCCCCC(C)C)n1cc(C2N(C(CC(C)(C)OCC)=O)CCCC2)nn1 N1(C(Cn2ncc(C)c2)=O)CC2CCN(C(C3COCC3C(F)F)=O)CCC2C1 c1(C(=O)NC(CCCNC(CCC#C)=O)C)cc([N+](=O)[O-])c(C)cc1Cl c1(C(=O)NC2CN(C(C(CC)O)=O)CC2C(F)F)cc2c(nc1O)CCCCC2 C1(NC(CCn2nc(C)c(C)c2C)=O)CC12CCC(NC(=O)C=C1CC1)CC2 n1(CC(=O)NC(C2CN(C(C3CC3c3ccco3)=O)C2)C)nnc(C2CC2)n1 C=CC(C)(CCOC)C(=O)NC(C)C(=O)NC(C)CCC1CC1 C(=O)(CC(C)(C(F)(F)F)N(C)C)NC1CC(C)(NC(CCCCOC)=O)C1 C1(NC(C(C)OCC2CCCO2)=O)CN(C(c2c(F)cncc2Cl)=O)CCC1F c1(NC(CC)=O)ccccc1C(=O)NCC1CN(C(C2(C)CC=CCO2)=O)C1 N1(C(C(=O)NCCC2CN(C)CC(C)O2)=O)CC(c2ccccc2)C2CCCC12 c1(-c2nn(CC)c(C(F)(F)F)c2)ccc(N(C)C)cc1F C(c1ccc(C)cc1)=C(C(=O)NC(CN(C(c1ccc(CC)nc1)=O)CC)C)C CCCC(C)(O)C(=O)NCCCN(C)C(C1(C)CCN(C(C)=O)C1)=O c1(OCC)ccc(CC(=O)NCC2CC2NC(c2cnc(OC)cn2)=O)nc1 Cc1[nH]nc2c1CCC(C(=O)N(CCCCNC(C1CC3COCC3C1)=O)C)C2 C1(OC)CN(C(=O)C(F)(F)c2cnccn2)CCC1NC(C1CCSC1)=O C(=O)(CC(C(C)(C)C)NC(=O)CC1(CSC)CC1)NC1(CC)CC(C)(C)C1 c1(CS(Oc2c(C(N3CCC(=C)C3)=O)nc(C)o2)(=O)=O)noc2c1CC(OC)CC2 Cc1ncc(C(=O)NCC2CCN(C)C2)c(Cl)c1Br c1(C(=O)NCCOCCCNC(C(CCSC)O)=O)ccc(S(C)=O)cc1 C1(C)(NC(C=C(C)CN2CCOCC2)=O)CCN(C(c2ccno2)=O)C1 N1(C(c2c(C)ncs2)=O)CC(NC(c2ccsc2Br)=O)C(O)C1 c1(-c2nc(CCCCCCNS(C)(=O)=O)on2)ccc(F)c(S(C)(=O)=O)c1 CC1CC(C(=O)NC2CC3(C2)CC(O)C3)CCN1C(=O)CCc1cn(C)cn1 N1(C(c2c(OC)noc2C)=O)CCCC(CNC(C2CC(C3CC3)=NO2)=O)CC1 CC1(C(=O)NCC2(O)CC(NC(C3(N4CCOC4=O)CC3)=O)C2)CC=CCC1 c1(C(N2C(C(=O)Nc3c(CC)cc(Cl)cc3)CSCC2)=O)ccn2ccccc12 c1(OC)ccc(CN2C(C(N3CCC(N4CCCC4)CC3)=O)CC3CC23)cc1F c1(C(=O)NCC(C2CC2)NC(C#CC2(C)CC2)=O)ncn2cc(Cl)ccc12 c1(C(N2CC(NC(c3[nH]cc(CC)c3)=O)C(F)C2)=O)nccn2nccc12 C1(c2ccc(C)cc2O)NC(=S)N(c2cccc(Br)c2)C2=C1C(=O)NC21CCOC1 c1(OC)ccc(F)c(C(N2CCCC(C(=O)Nc3ccnc(Br)c3)C2)=O)c1 N1(C(C2(CC#C)CCN(C(=O)CCCSC)C2)=O)CC(=O)NC(=O)C1C C1(C(N2CC(NC(CC(C)C3CCCC3)=O)(CF)C2)=O)CC(F)(F)CS1 CCC(C(=O)N1CCOCC1CNC(c1c[nH]nc1C(C)(F)F)=O)C(C)C N1(C(C(C)(C)NC(C)=O)=O)CC(CC(N2CCC3C(CO)C23)=O)C2(CC2)C1 c1(NCC(=O)NC)nccc(=NC(C)c2nc(O)n[nH]2)[nH]1 N1(C(C2CCC(C)O2)=O)CC2CCC(C1)N2C(c1cscc1C(F)(F)F)=O N1(C(c2c(Cl)cc(C)c(C)c2)=O)Cc2ccccc2CC1CNC(=O)CC(C)F Cc1c(O)ccc(C(=O)NCC2CCN(C(c3ccc(Cl)nc3)=O)C2)c1C C1(CNC(C(C(C)C)OC)=O)CC2CCC1N(C(=O)CN1CCCC1=O)C2 N1(C(c2c(CNC(CC(C(C)C)C)=O)cc[nH]2)=O)CCC(O)CC(C)(C)C1 CP(C)(=O)C(CC(=O)NC1CC(O)CN(C(C2CC(O)C2)=O)C1)C(F)(F)F N1(C(CNC(CCCCC)=O)=O)CCCCC(NC(=O)C(=O)Nc2ncc[nH]2)C1 C(CC(=O)NC1CC(=O)N(C2CC2)C1)(C(F)F)NC(C1(OC)CCC(C)C1)=O C1(C(C)NC(C(C)N(CCC)C(c2nccn2CC)=O)=O)CN(C)CCO1 C1(C(N(C2CCC(CNC(C(CC)(F)F)=O)CC2)C)=O)CCc2nccn2CC1 Cc1cc(C(=O)N(C)CCOCCCN(C(=O)C(F)n2cccn2)C)ccn1 c1(C(=O)NC(CC)CN(C)C(C2CC=CCC2)=O)ccc(N2CCC2)cc1 C1(NC(C2CC(CCC)C2)=O)CCC(NC(C2CC3C=CC2O3)=O)CC1 C1(NC(COCCN(C)C)=O)CS(=O)(=O)CC1NC(=O)C=CC1(C)CCOCC1 N1(C(CC2ON=C(C)C2)=O)CC(C)CC1C(=O)NC(c1cccnc1O)C CN1CCC(C(=O)NCCCSC(F)F)(NC(=O)C(F)=CC2CC2)C1 C#Cc1ccc(C(=O)NC2CC3CC2N(C(=O)C#CC2CC2)C3)cc1C C1(N(C(C2N(C(CNC(CCC)=O)=O)CSC2)=O)C)CCCCC1(C)C N12CCC(CC1)C2=O.CC1(C(=O)OC)CN(C(=O)Nc2cc(CN)cs2)C1 C(=O)(CCC(=O)NCc1cc(C(=O)NCc2cnco2)n[nH]1)NCC c1(OCOC)cc(Br)ccc1CNCCCCCN N1(C(C(C=C)O)=O)CCCC2CN(c3ncccn3)CCC12 C1(NC(CN(CC)CC)=O)CC(OC)CN(C(=O)CC2CCC(=O)N2C)C1 C1(CCC)CC1C(=O)NCCCOC(C)C.C1C(=O)N1CC=C Cc1cc(-n2cccn2)nc(NC(=O)NCCCN2CCCC2(C)CO)n1 c1(CNC(C2(SC)CC2)=O)cn(CC(C)(C)CNC(=O)Nc2ccccc2)nn1 c1(C(=O)NCC(C2CC2)NC(c2cn(C)nn2)=O)ccnc(-n2cccc2)c1 C1(C(N(CCCNC(C(C#N)c2ccccc2)=O)CCO)=O)CCNC(=O)C1 c1(C(=O)OC)nc(NC2CC3CN(C(c4c(C)nn(C)c4Cl)=O)CC23)ncc1Cl N1(C(c2cc(OC)c(Cl)cc2)=O)CCC2C(CCN2Cc2ncc[nH]2)C1 C1(C(=O)NC2CN(C(Cc3n[nH]c(=NC)s3)=O)CC2C)CCn2c(cnc2C)C1 CC1(C)Cc2cccc(C(=O)OCC(=O)NCC34CCCC(C)(C3)OC4)c2O1 N1(C(C)=O)CCC(C)(NC(=O)C(O)CN2CCCC2)C1.N12CCC(C1)C2=O c1(C(=O)NCCC(CC)(C)NC(C2CCCC2C2CC2)=O)cc(F)cc(C)c1N CCCCC(=O)C(=O)NCC(C)NC(=O)CCNC(=O)COC C1(N(C(c2c(C)scn2)=O)C)CCCC(N(C(=O)Cn2cc(C(F)F)cn2)C)C1 c1(CSCC(=O)NCC#CCNC(C2C(C)(C(=O)OCC)C2)=O)ccc(F)cc1 CC1CCN(C(C23CC(CO2)C3)=O)CC1NC(c1cccc(=S)n1O)=O C1(CNC(=O)C=CCO)CC2COCC2N1C(=O)C(O)CC1CCCCC1 N1(C(CC)=O)CCN(C(=O)C(c2cc(Cl)ccc2OC)(C)C)CC1C(F)F N(C1CN(C(=O)CCCC2CC2)Cc2ccccc21)C(CC1C(=O)NCCC1)=O c1(CC)cccnc1C(=O)NCC(C1CCCN1C(=O)CN1CCCC1=O)(C)C Cc1cn2c(C(=O)NCC(C3CC3)NC(C3(C4CC4)CCCO3)=O)c(C)nc2s1 CCS(=O)(=O)CC(=O)NCCCCCN(C(=O)C(C)(C)C1CCCO1)C c1(ONC(C2(C(N(OC)CCO)=O)CCSC2)=O)cccc2cncn12 CC1=NOC2(C1)CC(C(=O)NCCN1CCN(C(c3nc(O)c(C)s3)=O)CC1)C2 c1(CNC(=O)CC2CCSCC2)nccc(Br)c1Br CC1CN2CCN1C(C(=O)NCC1CCN(C(=O)CCCC(N)=O)C1)C2 N1(Nc2ncc(C#N)cc2F)CCC2(CCCC2NC(c2coc(Br)n2)=O)CC1 c1(C(=O)NC2CN(C(C3C(C(C)C)CCO3)=O)CC(C)C2)c(F)cc(F)cc1F C1(SC)CCN(C(c2nc(C)co2)C(=O)NCC2CCOC2)CC1 C1(CNC(C2CN(C)C2)=O)(CO)CC12CCN(C(=O)CC1COCCN1C)CC2 C1(NC(Cc2c(C)scc2)=O)CC2CCC1(NC(=O)CCCNC(=O)C1CC1)C2 C1(CC(=O)NCC=CC(=O)NC(C2(CO)CCC2)C)CCCC2CC12 N1(C(C2(c3cc(C)on3)CC2)=O)CCN(C(C2CC3CCCC3C2)=O)CC1CO CCCCCCC(F)C(=O)N1CC(N2CCN(C(=O)C3=CCSC3)CC2)C1 C1(C(N(C)CC2CCC2)=O)CN(C(c2ccc(CO)cn2)=O)CCO1 c1(C(N(CCN(C(C2(CC)COC2)=O)C)C)=O)ccc2ccnc(O)c2n1 C1(NC(C(C)CC(F)F)=O)CN(C(=O)Cc2cc(Br)cs2)C2(CCC2)C1 Cc1cc(C)c(C(=O)NCC2(NC(=O)C=Cc3cc[nH]n3)CC2)c(S)n1 C#CC1CCC(C(=O)NC2CS(=O)(=O)CC2NC(c2[nH]c(=N)ccc2C)=O)CC1 N1(C(CN(CC#C)C(c2ccn3ccccc23)=O)=O)CCC2CCC(C2)C1 CC(C)(C)CCC(F)C(=O)NC(CC1CCC1)C(N1Cc2cc(F)ccc2C1)=O N1(C(C(Br)=C(C)C)=O)CC(CNC(c2cc3n(n2)CCO3)=O)CCC1C C1(C(=O)NCC#CCC)CCCCCCN1C(c1ncc2ccccn12)=O c1(C(C(=O)NC2CCCN(C(c3cc(C)oc3)=O)C2)C(C)C)ccc(C#N)cc1 c1(C(C)C)nc(N(C)CC2CCCS2)cc(N2CCC(c3ccccc3)CC2)n1 N1(C(C(N2CC(C)OCC2)=O)=O)CCCC2CCC(C)CC12 c1(C(N(CCNC(Cc2cc(C)sc2)=O)CC2CC2)=O)cc2oc(Br)cc2[nH]1 c1(C(N(C)CC2CCN(C(c3cc(Cl)no3)=O)C2)=O)cc2ccc(F)cc2s1 c1(C(N2CC(F)CC(NC(CC(COC)(C)O)=O)C2)=O)ccc2c(c1)C(=O)OC2 C1(NC(CC(CCSC)O)=O)CCN(C(c2cnc(C3CC3)nc2)=O)CC1(C)C Cc1ncncc1C(=O)NC1CC2(C1)CC2NC(c1n[nH]cc1F)=O C1(CN2CCC(C(=O)NCCc3cn(C)nc3)C2)COC(C)(C)O1 c1(CCC(N2CCC(CNC(c3ccc(C(C)=O)[nH]3)=O)C2)=O)ccc(Cl)c(F)c1 CCC(C)(C)C(O)C(=O)N1CCC(C)C(NC(c2cc(C(N)=O)c[nH]2)=O)C1C Cc1cn2cc(CC(=O)NCCC3CCCN3C(=O)CN3CCNC3=O)nc2s1 C(C(C)(C)C(=O)NC1CCC1NC(c1cc(I)on1)=O)OC c1(CC)ccc(S(=O)(=O)NC2CN(Cc3cccc(OC)c3)CC2(F)F)cc1 CC1CCCN(C(=O)C(=O)NCC2CCN2C(C2CCCN2C2CC2)=O)C1 N1(C(c2c[nH]c(=N)s2)=O)CCC(NC(c2ncccc2Cl)=O)C(CO)CC1 C1(CNC(c2cc(CCC)oc2C)=O)CCCN(C(=O)C(C(C)C)OC)CC1 C(=O)(CC(C)CC(C)C)N1CCC(NC(c2n(COC)ncc2)=O)C(CO)C1 C12(CNC(C=CC(CC)C)=O)CCCC(CN1C(c1cccc(C)c1C)=O)C2 c1(C(C)C)ccc(CC(=O)NCC2CN(C(=O)CCCC3CCC3)CC2O)cc1 C(=O)(C1Cc2ccc(F)cc21)NC(CC=C)CNC(c1ccc(C)nc1CC)=O c1(C(=O)NC(C(=O)NCc2cnc(C)[nH]2)C2CC2)ccc([N+](=O)[O-])o1 c1(C(N(C2CC2)Cc2ccc(C)o2)=O)ncn2c1CCC2 Cc1ncc(Br)cc1NC(=O)C(O)C(F)F C(=O)(C(=O)N=c1cc(-c2ccccc2)o[nH]1)Nc1c(C)cc(Cl)cc1 CCCCC(C)C(=O)NCC12CCC1CN(C(c1cc(CN(C)C)c[nH]1)=O)C2 C(=O)(C(C)(O)CCC)NC(CCC)C(=O)NC(c1ncc[nH]1)C Cc1c[nH]c(CC(N)=O)c1C(=O)NCC(C)NC(=O)C(C)Cc1ccc(F)cc1 c1(C(N2C(C(N)=O)CC2C(=O)O)=O)nc(C2CC2)c(Br)cc1Br C1(COC)CCCCN1C(=O)C(=O)NC1CCCNC1=O c1(-c2cccc(C)c2O)ccc2c(c1)c(C(N1CCC(=O)C(C)C1)=O)cn2C C1(NC(CN(C(=O)C=Cc2cscn2)CCC)=O)CCCC1(C)O c1(CC(=O)NCCN(CC(C)O)C(c2cnns2)=O)nccn1C CCS(=O)CC(=O)NC1CN(C(c2c[nH]nc2I)=O)CC1C C(N=c1[nH]c(N2CCC(c3nncs3)C2)nc2c1SCC2)c1cccc(CC)n1 C(C(C)(C(C)C)NC(C1CCN(C(C)=O)C1)=O)NC(C(C)(C)OC)=O C(=O)(C(C)(C)c1cscn1)NCC(C)NC(c1cnc(CC(C)(C)C)s1)=O C1(NC(c2c(C#C)c[nH]n2)=O)CC1C1CCN(C(=O)CCOCCCOC)CC1 Cn1nc(C(N2CCC(CCC(=O)N3CC(n4cccn4)C3)C2)=O)cc1O N12CC3CCN(C3C1)C(=O)c1c[nH]c(c1)C2=O.c1(COC)c(C)cc(C)cc1C C1(c2nn[nH]n2)(CC)CC1C(C)C.C12(CC1)C(=O)N2C1CC1 c1(C(N2C(Cn3cc(CC(C)(C)C)nn3)CCC2)=O)ccc2c(n1)CCCC2 N1(C(CCCCOCC)=O)CCC(NC(=O)CCSCC(N)=O)C(O)C1 C1(NC(CSCCCC)=O)COCCN(C(=O)CCC2COC(C)(C)O2)C1 N1(C(C2(CSC)CC2)=O)CCC(NC(c2cccc(CC)c2)=O)C(F)C1 c1(N2CC(COC)OC(C)(C)C2)nc(=NCC2CC23CC3)[nH]c2c1SCC2 C=CCC(CC(F)F)C(=O)NC1(CO)CN(C(c2c[nH]c(=N)o2)=O)C1 N1(C(C(CC)C)=O)CC(CNC(c2cn(CC3(CC)COC3)nn2)=O)C(O)C1 C1(CNC(c2cc(C)ns2)=O)CC(C)(C)CN1C(c1nn(C)c(Cl)c1Cl)=O C1(C2N(Cc3cn(CC(=O)OC)nc3)CCC2)CCC(C)CC1 CC1CN(C(=O)Cc2ccoc2)CC1CC(=O)NCC(c1ccccc1)F Cn1cc(Br)c(C(N2CC(C(=O)O)C(O)C2)=O)n1.C1COCCOCCOCCO1 CC1CCCC(O)(C(=O)Nc2ccc(SCc3ccc(Br)cc3)cc2)CC1 CN1CCn2cc(C(N3CCOC(CNC(=O)CCP(C)(C)=O)C3)=O)nc2C1=O N1(CC)C(=O)CCC1CC(=O)NCC(CO)NC(c1n[nH]cc1OC)=O c1(-c2n(C)nc(CCC(F)(F)F)n2)cc2ccccc2n1CC(F)F c1(N2CCC(CC)(CO)C2)nc(NCC(C2CC2)OC)c2ccsc2n1 N1(C(c2c(CCC)n[nH]c2)=O)CCOC(C(=O)N(c2ccccc2)C)CC1 Cn1cc(C(=O)NCC(CNC(=O)CC2(n3ccnc3)CC2)S(C)(=O)=O)n(C)c1=O C1(CC)(CC)CCCN1C(=O)C(C)NC=O.C12(C)CC(C1)NC2=O C1(NC(C(C2CCN(C(c3c(OC)n[nH]c3)=O)C2)C)=O)CCc2ncnn2C1 n1(CC(=O)NCC2C3CN(C(C(CC)(C)O)=O)CC32)c(NC)nc2ccccc12 CCCS(=O)(=O)C(C)C(=O)N(C1CN(C(c2ccc(Cl)c(F)c2)=O)CC1(C)C)C c1(C(N2CCCC(C)(C(=O)NCCNC(C)=O)C2)=O)cn2c(Cl)cccc2n1 N1(C(c2c(C(C)C)ocn2)=O)C(C)CN(C(=O)C(C)N2CCC2)CC1C C1(CNC(CC2(C)CC2(F)F)=O)CC(O)CN1C(C1CC1c1ccc(O)cc1)=O Cc1cc(C(=O)NCC2(F)CCN(C(C3CCCCCCC3)=O)CC2)nc(C)n1 c1(C(=O)NCC(Cn2cc(C(CC)O)nn2)(C)C)cc2c(C)n[nH]c2cn1 C12(CNC(Cc3cc(C)no3)=O)CN(C(C3CCCCS3)=O)CC1CCO2 N1(C(C2(OC)CCS(=O)(=O)C2)=O)CC2CCCC(C1)N2Cc1cnsn1 N1(C(C(C)(C)F)=O)CC(CC(=O)NC2CCCC2O)C2(CC2)C1 Cc1cccc(CCC(=O)NC2CCC2CNC(=O)CC2CCC23CCC3)c1 C(C(CC(C)C)C(=O)N1CCOCC1C1CCC1)NC(c1cncc(C)n1)=O C1(CNC(=O)COC(F)(F)F)CCC2(CCC2)C1NC(c1cccc(O)c1Cl)=O CCCC(O)C(=O)NCCCC(C)NC(=O)C(F)=CC1CC1 C=CCC(C)(CC)C(=O)NCC(CO)NC(=O)CSC C1(C(=O)NC2(CC)CC(C)(C)C2)CCN(C(=O)C(C)OC(C)(C)C)CCO1 C1(OC(=O)NC2(N(C(C)(C)C)C3CC3)CSC(C(F)(F)F)C2)CCC2CCC1C2 C1(C(N2CCC(CC(N3CCC(c4cccc(F)c4)CC3)=O)C2)=O)CC2CCC2C1 Cc1c(C(N2CCCC(O)(C(=O)O)C2)=O)cccc1Cl c1(C(N2CCCC(CC(=O)Nc3cn(CC)nc3C)C2)=O)ncc2[nH]ncc2n1 C(C(C)(C)CC(=O)N1CCC(CNC(=O)C(C)(C)c2cc[nH]n2)C1(C)C)N(C)C N1(C(c2c(C)cno2)=O)CCCC12CCN(C(c1ccnc3[nH]c(O)nc13)=O)C2 C1(C(=O)NCC2CN(CC)C(=O)O2)CC2CCC(C1)N2C(=O)CCC1CC1 CC(CC(=O)N(C)CCN(C)Cc1nncn1C1CC1)N1CCOC1=O NC(=O)CC(N=c1ccnc(NC2CC3CCCCN3C2)[nH]1)c1ccc(Cl)cc1 CC1C(NC(=O)Cn2cccnc2=O)C(C)CCN1C(=O)C(C)(C)F CC(C)CC(CC(C)C)(c1nnnn1-c1ccccc1)NCCCO c1(CNC(CNC(CC(C)C)C#N)=O)cc(F)cc(Br)c1 Cc1ccc2c(=NC(C)c3ccc(Br)cn3)[nH]c(=NCC(C)CO)[nH]c2c1 CC1CN(C)C(=O)CN1C(=O)CCC(C)NC(c1cncc(F)c1)=O N1(C(CCN(C(C2CC(C)(O)C2)=O)C2CC2)=O)CC2(COC(=O)C2)C1 C=CC(C)CC(=O)NCC1(OC)CN(C(c2cc(C3CC3)cs2)=O)C1 c1(-c2c(OC)cccc2)nc(=NCC2CCCN2C(c2cscc2C)=O)s[nH]1 C1(CCC)CC(C(=O)NCC2CC2NC(=O)C(C)NC(C)=O)C1 c1(OC)cccc(CN2CCCC(C(=O)NCCC3CCCCO3)C2)c1C C1(COC)(NC(=O)CC(F)(F)F)CCCN(C(c2ccccc2C(C)(C)C)=O)C1 C(CC)(CCC(=O)N(CC(O)CF)C)NC(c1[nH]cc(C(C)=O)c1)=O N1(C(C(C(C)C)OC)=O)CCC2(CCN(C(c3ccc(F)nc3)=O)C2)C1 N1(C(C2(C)CCNC2=O)=O)CC2(C1)CN(C(=O)C=Cc1cn[nH]c1)CCO2 c1(C(N2CCN(C(C3CCCCC3)=O)C3CC23)=O)ccc2c(O)nnc(O)c2c1 c1(NC(=O)NCCCN2C(=O)CCC2=O)cc([N+](=O)[O-])n[nH]1 CC(C)CC(O)CC(=O)NCc1ccc(C(=O)NC2C3CCC(=O)C23)c(F)c1 C1(NC(CCn2c(C)cc(C)n2)=O)CC2CCC1C(NC(c1coc(Cl)c1)=O)C2 C1(NC(c2cc(CC)nc(O)c2)=O)CC2(CCCN(C(C3CC3COC)=O)C2)C1 Cc1cc(C(=O)NC(CNC(C2CCCC2O)=O)C(C)(C)C)nn1CCO CC1CCN(C(c2cn(CCCF)nn2)=O)CC1NC(C1(C)CC1(F)F)=O n1(CCC(=O)NC2CN(C(C=CCC)=O)CC2(C)C)c(C)nc2ccccc12 c1(C(C)=O)ccc(C(=O)NC2CC(C(C)NC(=O)C(C)n3ccnc3)C2)nc1 CC(C)(CC1CCOCC1)C(=O)NCC1(CNC(=O)C(F)CC2CCCC2)CC1 C1(C2CN(C(=O)CN3CSCCSC3)C2)(NC(c2c(C)cc(C)s2)=O)CC1 N1(C(CN(c2ccccc2)C)=O)CC(NC(=O)C(CC(N)=O)N(C)C)C(C)(C)C1 c1(C(=O)NC(CNC(Cc2cc(C)sc2)=O)C(C)(C)C)cnc2ncnn2c1C C12(NC(CCNC(=O)NC)=O)CC(C1)N(C(c1sncc1Cc1ccoc1)=O)C2 c1(C(N2C3CN(C(c4c(OC)nsc4)=O)CC2C3)=O)ccc2cncn2c1 C1(C(=O)NCCCC(C)NC(=O)CO)CC2(CCC2)C1 C(=O)(CC(C)C(=O)NCC(C)(F)CNC(C1CN(C)CCO1)=O)OC C1(COC(C2CC(C(=O)OC)C2)=O)CCCOC1.C1CC(=O)NC(=O)N1 N1(C(C2CN(C(C)=O)C2)=O)C2CCC1C(C(=O)Nc1cccc(Cl)c1C)C2 C1(OC)CN2CCCC2(C(=O)NCC(C(C)C)N2CCOCC2)C1 C(c1ccc(Cl)cc1)=CC(=O)NCC1C2CN(C(C3C(C)(C)CCO3)=O)C1C2 c1(OCC)n[nH]cc1C(=O)NCCCCCNC(=O)C(C)OCC1CC1 C#Cc1ccc(C(=O)NC(CNC(=O)C(C(C)C)N(C)C)C2CCC2)c(C)c1 O=C(CC1CC1C1(C(=O)OC)CC1)NOCC1(C(=O)O)CCSC1.c1(C)ccccc1 C1(CCNC(=O)Cn2nccn2)CCCCN1C(c1ncncc1Cl)=O C(CCCCC(=O)N1C2CCC(C2)C1CC(N1CCC(n2ccnc2)C1)=O)OC N1(C(c2c(C)nc(CC)o2)=O)CCC(NC(c2cc(NC)on2)=O)C(CO)C1 c1(CNC(C)COC(F)(F)F)cc2cc(OCC(F)F)ccc2nc1Cl c1(C(=O)NC(CNC(C2(COC)CC2)=O)(C)CC)ccc(F)cc1[N+](=O)[O-] C1(NC(c2cc(CCO)on2)=O)C=CCN(C(=O)C=Cc2ncco2)C1 c1(CONC(C(C)(O)c2n(C)ccn2)=O)ccc2ccccc2c1 c1(C(=O)NCCN(CCC)C(C2(F)CCOC2C)=O)cc(C)nn1C(C)(C)C c1(CCNC(C2(C)CSC2)=O)ccc(CNC(=O)CC2CCC(=O)N2)cc1 C1(C(=O)NC2CC3(C(NC(C4(C)COC4)=O)C3)C2)CC(F)(F)CCC1(C)C c1(C(N2CC(C)N(C(=O)Cn3[nH]cnc3=N)CCC2)=O)cnc2sccn2c1=O CC(C)=C=CC(=O)NCC1CCC(C(=O)NCCSC(C)C)CC1 C(=O)(CCN=c1cc(C)[nH]c(=NCC2CC3CCCCC3O2)[nH]1)NC(CC)C C1(C(=O)NCCN(C)C(C2CC3(CCC3)CO2)=O)CC(C)(C)CCO1 C1(CC(=O)NCC(CCNC(=O)CSc2ccncc2)O)CC2(CCC2)CO1 C=CCC(C(=O)NC1(CNC(c2cn(C)cc2C)=O)CCOCC1)OC C(=O)(CC(O)CC1CC1)N1CCC(OCC)C1 N1(C(COCCOC)=O)CCC(NC(c2c(SC)cccc2F)=O)C1(C)C c1(C(N(CC(CNC(CC(C)(C)OC)=O)O)C)=O)cnc2cc(Br)ccn12 C(C(C)(C)CCNC(=O)C=CC1CCC1)NC(CCN(C(CCC)C)C)=O c1(-c2cn(CCN(C(C34COCC3C4(F)F)=O)CC)nn2)ccccc1[N+](=O)[O-] CC1(C)CCCC(C(N2CCC2(C)CC(=O)NC2CC3CCC(C2)S3)=O)C1 c1(C(N(C(CNC(C(C=C)(C)CC)=O)C)C)=O)c[nH]c2c(Br)cccc12 c1(OC)c(Br)cc(OCCCN2CCC(N3CCCCC3)CC2)cc1Br C1(C(=O)NCCCCCO)CC12CN(C(C1CC(O)CN1)=O)C2 CC1C(C)N(C(C2CC(C(=O)C3CC3)C2)=O)CCN1C(=O)Cc1ccc(O)c(F)c1 C1(C)(CNC(CCOC)=O)CCN(C(=O)C(C)Cc2ccc(N)cc2)C1 c1(C(N(C(C)CCNC(c2coc(O)n2)=O)C)=O)cccc(C2(F)CC2(F)F)c1 C1(CCOC)(NC(C2CCC3(CC3)C2)=O)CCN(C(=O)CCOCC2CC2)C1 C1(OC)CC(NC(c2cscn2)=O)CN(C(=O)C(C)(O)c2ccccc2)C1 C1(NC(CC=CCCCCC)=O)CCC1(C)C.C1(NC(C=C)=O)CC(N(C)C)C1 C1(C(=O)NCC(CC=C)(C)C)CN(C(=O)C(C)OCOC)CC1(F)F C1(NC(C(C)CN2CCCCC2)=O)CCN(c2nnc(C(F)F)s2)C12CCC2 Cc1ncc(C(=O)NC(C2CCCN(C(C3(S(C)(=O)=O)CC3)=O)C2)C)cc1N CC1(C)CCC=C(C(=O)NC2CN(C(c3nc(C4CC4)cs3)=O)CCC2(C)C)C1 C12(CNC(c3nc(C)nc(O)c3)=O)CCCC(CN1C(=O)Cc1csnc1C)C2 C1(CN(C2C(C)(C)CO2)CCO)CCN(C(=O)C(c2ccccc2F)(F)F)CC1 C1(C(=O)NCCN(CC(C)O)C(=O)Cc2csc(S)n2)Cc2nncn2C1 C(CC(C(=O)N(C)C(c1cc(Br)cs1)c1cccs1)NC(=N)N)SC N1(C(CCC#CC)=O)CC2(CC(CNC(c3ccc(OC(C)CC)cc3)=O)C2)C1 C1(c2nnnn2-c2cccc(F)c2)(NCc2nnn(C)n2)CCC2C3C=CC(C3)C12 C1(C(=O)NCc2c(C(=O)NCC3C(C(=O)OC)C3)[nH]cc2)CC2(CCO1)CC2 C(CC1=CCOCC1)NC(C(CCC)NC(=O)CCOC(C)C)=O C(CC(C)(C)NC(c1cc(-c2ccc(C)o2)on1)=O)NC(C1CC(SC)C1)=O C(CCCCCNC(C1CCCCC1)=O)N(C)C(c1ccc(C2CCOC2)s1)=O c1(C(=O)NC2(C(=O)NCc3cc(C)nc(C)c3)CSC2)cc2cccn2cn1 C1(CCC(=O)NC(c2ccco2)C)CCCCN(C(=O)CCCF)C1 C12(NCC3(COC)CN(C(C4(c5ccccn5)CC4)=O)C3)CCCC1CC(=O)C2 C#Cc1cc(C(N2CCC(NC(=O)CN(C)CC)C2)=O)cc(Br)c1 Cc1cc2c(cc1Br)N(C(C(=O)NCC1CC1(C)C)C1COC1)CCO2 c1(C(=O)NC(C(C)NC(=O)CC(F)(F)Cl)C)cc(C(F)(F)F)cc(N)c1 c1(C(=O)NC(CNC(CCC)=O)C2CCC2)ccn2ccnc2c1 CC1CC2(CC(C(=O)N(CCCCC(=O)N3CCOCC3C)C)C2)C1 C(=O)(CCC(C)(C)F)N1C(C2CCN(c3ncc(C)cn3)C2)CCCC1 CC(C)CCC(O)C(=O)NC1CC2CC1N(C(c1cccc3oncc13)=O)C2 c1(N2CCC(CN(c3cncc(F)c3C)CC)CC2)ncc(C(F)(F)F)cc1Cl N1(C(CC)=O)CCC(CNC(=O)CCNC(c2ccccc2OC)=O)(OC)C1 N1(C(CCCNC(=O)OC)=O)CCCN(C(=O)CN2CCC(C)CC2)CC1CO N1(C(C2C(C)(C)CC2)=O)CCn2c(CNC(C3(C)C=CCCC3)=O)nnc2C1 c1(OC)ccc(CN2CCN(C(c3ccon3)=O)C(CC#N)C2)c2ccccc12 c1(C(=O)NCC(CNC(C(C)OCC(F)(F)F)=O)CO)cnc2ncccn12 C1(C(=O)NC2CC(CNC(CN(CCC#C)C)=O)C2)CN2CCN1C(C)C2 N1(C(c2nn(CC)c(C)c2)=O)CCC12CN(C(c1cc(CC(C)C)c[nH]1)=O)C2 C1(CCCC)CN(C(C2CC2C(=O)OC)=O)CCN1C(=O)CP(C)(C)=O c1(OCC)oc(C)nc1C(N1CC(CNC(=O)C=CC2(C)COC2)C(O)C1)=O C1(OC)CCN(C(=O)C=CCC(C)(C)NC(=O)CCCn2cncn2)CC1 c1(CC(CNC(=O)NCCC2CC3C=CC2C3)CO)ccccc1F c1(CNC(CCc2ccn(C)c2)=O)cc(F)c(Br)c(F)c1 C#CCCC(C(=O)NC12CCCN(CC1)C2)NC(=O)C=C(CCC)CCC c1(C(N2C(CCCC)CN(C(=O)C(C)O)CC2)=O)ccc(Cl)c(Cl)c1OC c1(OC)cccc(NC(=O)CNC(=O)CNC(c2cc(C)sc2N)=O)c1 c1(CC)cscc1C(=O)NC1(CNC(c2cnsc2C)=O)CCOC1 CC(C)CCC(F)C(=O)N1CC(NC(C2CCC(CO)CC2)=O)CC(F)C1 C(C)(CNC(c1c[nH]nc1-c1ccoc1)=O)(C(C)C)NC(Cc1c(C)nc[nH]1)=O C(CC(=O)NCCC(Cc1ccccc1)NC(C1CCC1)=O)(C(N)=O)NC(C)=O c1(C(=O)NCCN(C(CCCc2ccc(C)s2)=O)C)cccc(CO)c1C O=C1CC(NCCO)CN1Cc1cn(CC2CC2)nn1 O=C(NOCC(N1CCCCC1C#N)=O)C(F)(F)CCc1cn(CC2CC2)nn1 C=CC1(CC(=O)NC2CC(NC(=O)C(C)c3cccs3)C2)CCOCC1 Cc1ccccc1C(=O)NC1CCC(CC(=O)NOCCOCCF)C1 Cc1ccc(C(N2CC(C(C)NC(C3C=CC=CC=C3)=O)C2)=O)cn1 C1(C(N(CC(=C)C)C)=O)CC2CC1CC2NC(C1(CO)CCCCO1)=O C(c1ccccc1OC)=CC(=O)NCC1CN(C(C(c2ccc(CC)s2)=O)=O)C1 Cc1c(O)c(=O)ccn1CC(=O)NCCCN1CCN(c2nccn2C)CC1 C1(NC(C2(COC)CCN(C(=O)C(C)CC(N)=O)C2)=O)CC2C(C1)C2(F)F c1(C(N2CCC23CN(Cc2csc(Br)c2)C3)=O)ccn2cnnc2c1 c1(NC2CCN(C(Cn3ccc(C)n3)=O)C(C)C2)ncnc2c1nnn2C(C)C c1(C(=O)NCCCCNC(c2ccn(C3CC3(F)F)n2)=O)cscc1F CCCCCC(C)(C)C(=O)NC(C)CNC(=O)CCc1cccnc1F Cc1ccnc(Cl)c1CN1CC(C)(C(=O)NC2CC2c2ccc(Br)cc2)C1 C1(C(=O)OC)CCN(C(=O)CC2CCC2C)CC1.C1(=O)CO1 c1(C(N(C)CC2CCCN2C(=O)CCF)=O)cc2cccc(Br)c2[nH]1 CCC(CC(=O)N1CC(NC(c2nnsc2C(F)F)=O)C(C)C1)c1ccccc1 N1(C(C2C(C)=C2)=O)CCN(C(C2CC3(C2)CC3(F)F)=O)C2(CCC2)C1 Cc1ccc(NCCC(N2CC(NC(c3cnncc3O)=O)CC2C)=O)cc1 c1(N2CCC(N(CCC)C(c3oncc3C)=O)CC2)ncc([N+](=O)[O-])cc1C N1(C(c2cc(CNC(C=CCCC)=O)sn2)=O)CC(C2CC2)C1C1CC1 C(C(N)=O)(C(=O)O)NC(CONC(Cc1ccn(CCC)c1)=O)=O c1(OCC(=O)NCC(CC)N(C(=O)CC2CC(OCC)C2)C)cccc(C)c1 C1(C(N2CC(C(N)=O)C2)=O)CCCCN(C(C2C3CCC2(C(F)(F)F)C3)=O)C1 C1(NC(CC23CC(C)(OC2)C3)=O)CCC2CCN(C(C3(C)CCCO3)=O)C1C2 S(=O)(=O)(c1ccc(C)cc1C)NC(N(C1CCCCC1C)CC)=O c1(CCC(=O)NCC2C3CC2N(C(=O)C=Cc2ccoc2)C3)ccc(F)cc1F N1(C(c2cnc(C(C)C)nc2)C(=O)NCC=C)CC(C(F)F)CC1(C)C c1(C(N(CCN(C(=O)CCCC(F)F)C)C)=O)cc(Br)c2c(c1)OCO2 c1(OCCOC)ccccc1NC(N1CCC(c2ccn(C)n2)CC1)=O C(=O)(C1=Cc2ccccc2C1O)N1CCC(NC(CCC(=C)Cl)=O)(CC)CC1 c1(C(=O)NC2CC(C)(NC(CC3C(C)CCO3)=O)C2)ccccc1O N1(C(c2ccc(C(C)=O)cc2)=O)CCC(NCc2cn[nH]c2)C(F)C1 C1(OC(C)C)CC(NC(C2(NC(C3CC3(C)C(F)F)=O)CC2)=O)C1 c1(N2CCCC(CCC)CC2)nc2c(c(=NC(C)C3CC3)[nH]1)SCC2 C1(CNC(C(C(C)C)N(C)C)=O)CC2CN(C(c3cc(O)cc(Cl)c3)=O)CC12 c1(C(=O)NCC(C)NC(c2c(C)nc(C(C)OC)s2)=O)ccc(C(N)=O)cc1N c1(NCCNC(C(CC#C)(C)NC(C)=O)=O)ccc2c(c1)C(=O)C(=O)N2 c1(C(N2C(CNC(C(C)C3(O)CCC3)=O)CCC2)=O)coc2c1CS(=O)(=O)C2 n1(CC)cc(Br)c(=NC(=O)N2CCCC2c2nnc(C)o2)[nH]1 N1(C(C(C)n2cccn2)=O)CCCC(CC(=O)Nc2ccccc2Br)C1 C1(NC(c2cc(OCC)n[nH]2)=O)CC2CCC1N2C(=O)CC1CCCC1(F)F N1(C(C=CSC)=O)CC2(CCC(CNC(=O)CNC(=O)NC3CC3)O2)C1 C(C)(CCCCCO)NC(C1(C2N(C(c3nc(C)oc3C)=O)CCC2)CC1)=O C(CN=c1[nH]c(=N)[nH]c(=NCCCC2CCCO2)[nH]1)c1nc(C)nc(O)c1 C1(NC(c2cc(C(C)=O)sc2)=O)CC(NC(=O)C=C2CCOCC2)C12CCC2 c1(C(=O)NC2CN(C(C3(SCC)CC3)=O)C2)cccc(CC)c1F c1(C(=O)NC2C(CNC(CC=C)=O)C2)nn(C(C)C)nc1Br CCC(C#N)(CC)C(=O)N1CCCCC(CNC(=O)Cn2nc(C)n(C)c2=O)C1 c1(C(=O)NC(CC2CN(C(C3C(CCOC)C3)=O)C2)C)cccc(Cl)c1OC N1(C(c2cc(C)cc(OC)c2O)=O)C2CCCC1CN(C(=O)CN=S(C)(C)=O)C2 Clc1cnc(N2CCN(c3noc(-c4ccccc4Cl)n3)CC2)c(Br)c1 N1(CC(CNC)O)CCN(C)CC1.c1(OC)ccc(C(C)(C)N)cc1 c1(SC)cc(-c2nc(C)nn2C2CCC2)cc(Cl)n1 C1(NC(C2(C)CC=CC2)=O)CCCCN(C(=O)CCN2CCCC2=O)CC1 C(=O)(CCC(=O)N(C)C)NC(C1CCCN(C(=O)C(C2CC(F)(F)C2)O)C1)C CCC(CNC(C1CCN(C)C1)=O)(CC)NC(c1ccc(C(N)=O)nc1)=O N1(C(CN(C)C(N)=O)=O)CCC(C2CC2)(NC(=O)C(C2CCOCC2)O)C1 c1(C(N2CC3C(NC(C(C)S(N)(=O)=O)=O)CC(C3)C2)=O)cnn(C)c1S(N)(=O)=O CCC(CC)C(C(=O)N1CC2CC2C1C(N1CC2C(CO)C2C1)=O)OC C=CC1CCCC(NC(=O)CCC(C)NC(=O)C(C)(COC)COC)C1 C1(CNC(c2cc(CC(C)C)[nH]n2)=O)(NC(=O)CC(C)(F)F)CC(F)(F)C1 c1(CSCC(=O)Nc2ncc(-c3ccccc3F)o2)ccccc1Br CCS(=O)(=O)CCn1c(N(CC(C)C)C)nnc1CSc1nccs1 C(CCC(=O)NC1CCC(CCC(=O)N(C2CSC2)C)C1)=CC(C)C Cc1cc(C(=O)NCC2N(C(=O)CS(N)(=O)=O)CCCC2(C)C)c(N)c(Cl)n1 c1(OC)cc(C(=O)NC2CC(C)N(C(C3CCC(C)CC3)=O)C2)cc(N)c1N C1(NC(C2CC(OC)C2)=O)CCN(C(=O)CCSC2CCCC2)C(C)C1 C#Cc1ccc(C(N2CC(CNC(=O)C(F)(F)C(F)(F)F)OC(C)C2)=O)cc1C C12(NC(C3CC(C)OCC3)=O)CC(C)(C1)OC21CN(C(c2ccc(O)cn2)=O)C1 n1(CC(=O)NC2C(C)(C)CN(C(=O)C(O)C(F)(F)F)C2)ncn2cccc2c1=O O=C1CCc2cccc(C(N3CCOC(C(N4CCC5(C4)CC5(F)F)=O)C3)=O)c21 C1(N(C(CC(=C)C)=O)CC)CCCN(C(c2cnoc2-c2ccccc2C)=O)C1 CN1CCN(C(=O)CC2CCCOC2)CC1CNC(c1ccnc(Cl)c1Cl)=O c1(C(=O)NC2COCC2CNC(C2CC23CCCC3)=O)sc2ncccc2c1Cl N1(C(CC(CC)C)=O)CCC2(CC1)CN(C(C1CCN(c3nncs3)CC1)=O)C2 C1(c2cn(C)nc2)CN(N2CC3CCCCCC3C2)CC1NC(N)=O CC(C)C(O)C(=O)NN(CCOC(C1CCCCN1S(C)(=O)=O)=O)C1CC1 c1(C(N(C(CN(C(c2c(CC)nco2)=O)C)C)C)=O)cc2nc(C)[nH]c2cc1F N1(C(C(=O)NC(C)CC2CCCNC2)=O)CCC(C(C)(C)C#N)CC1 c1(CN(c2ccc(OC)c(C)c2)C)cc(Br)cc(C)c1F C1(COC)CCN(C(=NCCc2ccc(F)cc2)NCC(c2nc(C)cs2)C)C1 C(=O)(C(CN=[N+]=[N-])NC(c1cnsc1)=O)N1CCN(CCC#C)CC1 c1(C(N(CCC(C)OCCC)C)=O)cnc(NC(=O)C(=O)NCC(F)(F)F)cn1 c1(OC)ccc(C(C)C(=O)NC(C)CCNN2CCCCC2=O)cc1F N1(C(c2cccc(N)c2)=O)CC2CC(NC(C3Cc4cccnc4C3)=O)CC1C2 C12CC3CN(CC13)C2.c1(C(=O)OCC)cccc(OCC)c1.C12CCC1CN2.N C(CCC(=O)O)(C(=O)N1CC2CCC2(CO)C1)NC(=O)OC(C)(C)C n1(CC)cc2ccc(C(=O)NCCN(C(=O)C=CCF)C)cc2n1 N1(C(CC2(C(=O)OC)CC2)=O)CC(O)(c2cn(COC(=N)O)nn2)C1.c1(C)nccs1 O=S(=O)(c1ccc(Br)s1)N1CCCC(NC2(c3ccccc3)CCC2)C1 c1(C(=O)NC2CCCN(C(C3ON=C(C)C3)=O)C2)c(C)c(C)cc(C)c1C C1(CN(C)C)CN(C(C2OCCC2CNC(c2nocc2Cl)=O)=O)CCO1 c1(CC(=O)NCC(CN(C)C(C2CC2c2ccco2)=O)O)nc2c([nH]1)CCCC2 C1(C(N2CC(O)(CC=C)C2)=O)CNC(=O)CN1C(=O)CSCC(N)=O C1(CC(=O)N(CC(CC)NC(c2cnc(C(N)=O)cn2)=O)C)CCCCC(=O)N1 n1(CC)ncc(C(=O)NCC(C2CCOC2)NC(c2cnc(Cl)[nH]2)=O)c1Cl c1(CC)cnc(CNC(=O)CC2CCN(c3nc(COC)ns3)C2)o1 c1(-n2c(CNC(c3n(CC=C)nnn3)C3CCSC3)ncc2)ccc(F)cc1 Cc1ccc(Cl)c(C(N2CCCC(NC(c3csc(-c4nc[nH]n4)n3)=O)C2)=O)c1 CCC(F)(F)C(C)(C)C(=O)NC1CCCC(NC(=O)C(=Cc2cnc[nH]2)C)CC1 C(=O)(NNC(=O)C(C)(C)CCCCNC(C1SCCC1C)=O)c1c(CC)ocn1 Cc1ncnc(C(N2CCN(C(c3cc(C4CC4)[nH]n3)=O)C(C(F)F)C2)=O)c1C c1(NC(C2CN(Cc3cccs3)CCO2)=O)ccc(I)c(Br)c1 C(=O)(C1Cc2ccccc21)NCCCCCNC(C(CNC(C)=O)(C)C)=O C(C1=CCN(C(c2ccc(C(F)F)cc2)=O)CC1)NC(C1CC12CC(O)C2)=O Cc1ccc(F)c2oc(C(=O)NCCN(C(c3ccnc(S)c3)=O)C3CC3)cc12 c1(C(=O)NCCn2cc(C(N3CC=CC3)=O)nn2)ccc(O)cc1 C=CC(C)C(=O)NC1CC(CCNC(=O)CNC(=O)CN(C)C)C1 c1(C(=O)OC)cc(C)cnc1NC(=O)CCC1(OC)CCCCC1 C12(NC(C3CC(N(C)C)C3)=O)CCCC1CN(C(=O)CC1CCCCC(=O)N1)C2 c1(NC2CN(C)C2)[nH]c(=NCc2c(Br)cccc2Br)nc2scnc12 C#CCCN=C(NCC1(CC2CCC2)CC1)N1CC(C)CC(C)C1 N1(C(C2N(C(COCC3(C)C=CCCC3)=O)CCC2)=O)CC2CCC(C1)C(=O)O2 c1(CC)cccc(C(=O)NC(C2CCN(C(c3[nH]ccc3C)=O)C2)C)c1 C1(C(N2CC(OCC(=O)NCc3n(CCC)ccn3)C2)=O)CC2(CC(=O)C2)C1 c1(CC(=O)NCC(C)NC(c2cc3cc[nH]c3cn2)=O)ccc2c(c1)CCOC2 N(C)(C(=NCc1cc(C)on1)NCc1cc(F)cc(Cl)c1)CC1CCN(CC)C1 c1(C(=O)OC)cnccc1CC.C1(C)(C=O)CCCN1C(=O)C(C)N=[N+]=[N-] Cc1cc(=N)[nH]cc1C(=O)NCC(C)(C1CC1)NC(c1cccs1)=O c1(CN2CCN(CC(=O)NC3CCCCC3(F)F)CC2)cc2ccoc2cn1 N1(C(C2CCC(=O)N2Cc2ccc(Sc3ccccc3)cc2)=O)CC(=O)NC2(CC2)C1 CCC(CO)CCNCc1cc(CC(C)C)ncn1 C1(C(N2C3CC(=C)C(C3)C2)=O)C(C2CC2)CCN1C(=O)CCC(=O)OC Cc1cc(S(N)(=O)=O)ccc1CNC(=O)NCCc1cnnn1C c1(C(=O)NCC2C(NC(c3nnn(CC)c3C)=O)C2)cncc2ccc(F)cc12 Cc1cc(Br)cc(C(=O)NC(C)(C)CN(C)C(C2CCC(F)C2)=O)c1F C1(C(=O)NCC#CCC)C(CC)CCN1C(=O)Cc1csnn1 C1(C(C(=O)N(C(C)CCNC(c2scnc2C)=O)C)OC)CCC(F)(F)CC1 c1(C(=O)OC)cn(C)nc1CCC(=O)NCC(CNC(=O)C1=C(Cl)CC1)CO C(CN=C(NCCC1(F)CCCCC1)NCC1CC1)=CC N1(C(CC(CN(C)C)O)=O)CCc2[nH]nc(CNC(C3(C)CC=CCO3)=O)c2C1 CC(C)CCCCC(=O)N1CCCC(CNC(C2(C)CC(C)C2)=O)CC1 CCC(O)C(C)C(=O)NCC1C2CC1N(C(c1cc(F)ccc1C(F)(F)F)=O)C2 C1(N=[N+]=[N-])(C(=O)NCc2c(C)cc(C)s2)CCN(C(C2CN3CCC2CC3)=O)C1 C12(NC(C3CC4(C3)CC(F)C4)=O)CCCC1N(C(c1ccc(O)cc1)=O)CC2 c1(C(C(=O)OC)N(C(=O)CCCNC(N)=O)Cc2ccco2)ccc(Br)cc1 Cc1cncc(CC(=O)NC(C)(CNC(C2CC2(F)F)=O)CO)c1 N1(C(CC(C(C)C)c2ccon2)=O)CCC(O)(C2CCC2)CC1 C1(C2CC2)(CNC(C(c2n(C)cnc2)O)=O)CCN(c2ccc(C(F)(F)F)cn2)C1 N1(C(C(C)SC)=O)CC2CC(NC(=O)CCCc3nc4ccccc4o3)C(C2)C1 C12(NC(=O)CCn3cnccc3=O)CCCC1N(C(C1CSC1)=O)CC2 c1(C(=O)OC)ccc(F)c(C2CC(OC(c3ccc(OC)c(Cl)c3)=O)C2)c1 CC(C)C(O)CC(=O)NC1CN(C(=O)C(O)C(C)C)CC1O N1(C(=O)Cc2ccns2)CCCC2(C1)CN(C(c1n[nH]cc1[N+](=O)[O-])=O)CCO2 c1(C(=O)NCC(CC(C)C)NC(c2nccnc2O)=O)ccnc2cc[nH]c12 C=C(C)CC(C)C(=O)NCC(C)(CO)NC(=O)CC1(O)CCOCC1 c1(C(=O)NCC2(NC(C3C4CCCOC34)=O)CCOC2)cn2ccnc2cn1 C1(C(=O)NC(C2CC=CCC2)C(=O)NCCCSCC)CCCC1O c1(CN2CC(c3n(C)cnn3)C3(C2)COC3)cc(CN)cc2c1CCC2(C)C N=c1cc(C(N2CCC(NC(=O)C(Cl)=CCl)C23CC3)=O)c(Br)c[nH]1 C(=O)(C1=CCCCC1)NCC1C(CNC(C(C)CC2CC2)=O)C1 CC1CC(N=c2ccc3c([nH]2)CCCC3=O)CCN1C(=O)CN(C)C(=O)C1CC1 C1(C(N)=O)CCC(NC(C2CCCCC2c2ccccc2)=O)CC1 Cc1[nH]nc2ncc(C(N3CC(C(=O)O)C(c4ccsc4)C3)=O)cc12 C1(C(=O)NCC(C)NC(=O)C(c2ncccc2Br)(F)F)CC(C2CC2)=NO1 C1(NC(Cc2c(C)ncs2)=O)CCC(S(C)=O)C1 c1(NC2CCC(CC(=O)NCC3CN(CC)C3)CC2)ccc(C(=O)OC)c(N)c1 N1(C(C(C)n2ccnc2)=O)CCC2C1CCCN2C(c1cc(Cl)cc(F)c1Cl)=O c1(C(=O)NC2C3(CC(NC(COCC=C)=O)C3)C2)ccc(N)cc1C Cn1ccc(=O)c(C(=O)NCc2nc(-c3cnccn3)no2)c1 CCCC(C)(CCC)C(=O)N1CCC(NC(c2cnc(O)o2)=O)C(O)C1 C1(C(=O)Nc2cncc(OC)c2)CN(C(c2cnccc2C#N)=O)CC12CCC2 CC1CN(C(c2c(F)cccc2Cl)=O)CCCN1C(C1CCCC1(F)F)=O CCCCCC(C)(C)CNC(c1nnnn1CCC)c1ncnn1C(C)(C)C c1(NC(C(C2CCOCC2)OC)=O)cccc(CNC(=O)C(C)c2ccsc2)c1 C1(CNC(c2cccc(N(C)C)c2)=O)CC(C)(C)CCC1NC(=O)CSC1CC1 C12(C(N(CC(C(N3CCCC(COC)C3)=O)(C)C)C)=O)CCC(CC1)CC2 C(C(=O)NOCC(=O)NCCCCC)(C(C)O)NC(C)=O N1(C(C(CCC)NC(=O)CC2CC2C2CC2)=O)CC(C)OCC1C N=c1[nH]cncc1C(N1CC2C(NC(c3cn(-c4cccnc4)nn3)=O)C2C1)=O C12(CNC(c3ccnnc3)=O)CCC1CCN2C(=O)COc1cc(F)cc(Cl)c1 C(=O)(C(C)(CC)C(=O)NCCC1(O)CN(C(c2ncc(F)cn2)=O)C1)OCC c1(CC(CCOC)NC(C2CCOCC2)CC)ccc(F)cc1F CC1(C)CCCCC1NC(N1CCC(=CC(N2CCOCC2)=O)CC1)=O c1(CC(=O)NC(C)CCNC(=O)C(C)N2CC2)ccccc1Cl n1(CC)nc(C(=O)NC2(CNC(=O)CCc3cnn(C)c3C)CC2)cc1C C1(CNC(C2(COC)CC2)=O)CCC2(CN(C(c3nnc(O)nc3O)=O)C2)O1 c1(C(N2Cc3c(C(=O)OCC)ncn3CC2)=O)cc(F)cc2cc[nH]c12 N1(C(c2cc(OC)no2)=O)CCN(C(C2(C)CS(=O)(=O)C2)=O)CC(C)(C)C1 C(=O)(CCCCCS(N)(=O)=O)N(CC(CN(C(=O)CCn1cnnn1)C)O)C Cc1cccc2c1OC(C(=O)NCC(C)(O)CNC(=O)CNS(C)(=O)=O)C2 c1(CC)ccccc1OCC(N1CC(NC(=O)CC2CCC(=O)N2C)C(C)C1)=O Cc1nc(O)ccc1C(N1CCCC(CNC(c2c(Br)noc2C)=O)C1)=O c1(C2(C(=O)NC3(COC)CCN(C(C(CC)C)=O)C3)CC2)cccc(Cl)c1F CC1CC(C(=O)NCC2CN(C(c3snc(O)c3Cl)=O)C2)Cc2nn[nH]c21 N1(C(CCN(C)CC)=O)CCC(C)(CNC(c2ccc(C)cc2N)=O)CC1 N1(C(CC(=C=C)C)=O)CC(NC(=O)C=Cc2nc(C)cs2)CC2(CC2)C1 Cc1c(Cl)ccnc1C(=O)NCC1(CNC(=O)CC2CCOC2C)CCCC1 C(=O)(CCC[N+](=O)[O-])NC(C)CNC(c1ccn(C)c1)=O C1(C(=O)OC)CCCCCC1NC(Cn1cc(C2(CC)CCC2)nn1)=O C1(N=c2[nH]c(=N)[nH]c(=NC(C)COCC3CCC3)[nH]2)(CC)COC1 N1(C(c2cncc(C)n2)=O)CCC2CN(C(C3CCC34CCC4)=O)C2C1 C1(S(N)(=O)=O)(C(=O)NC2C(CNC(Cc3cnc(C)s3)=O)CCCC2)CCC1 CN1CCN(C(=O)C(O)C2CN(C(C3(C)CCC4CC4C3)=O)C2)C(CO)C1 c1(C(N2C(CC(=O)NCc3c(CC)nn(C)c3)CC(O)C2)=O)ccc([N+](=O)[O-])o1 C12(NC(C(CCC)NC(N)=O)=O)CC3CCC(C1C2)N3C(=O)CN(C)C(C)=O N1(CC(=O)NCC(C)(C2CC2)NC(C2CC=CCC2)=O)CCC(OCCF)CC1 c1(C(=O)NC(C)C)cncc(=NC(c2ccc(F)c(F)c2)c2ccccc2)[nH]1 c1(C(C)C)ncc(C(=O)NC2CCC(NC(=O)CCN3CCCCC3C)C2)cn1 c1(C(N2C(C)C(C)N(C(c3cscn3)=O)CC2)=O)cnn2c1OCC(C)(C)C2 S(=O)(=O)(c1cnc(NC2CCCCC2O)cc1C)NCc1ccc(C)cc1F C1(C(C)NC(=O)CC2CC(C(F)F)C2)CN(C(c2nccnc2N)=O)CCO1 C(=O)(C(C)C(O)CC(C)C)NC(C(N1CCN(CC=C)C(=O)C1)=O)C C(CC(CNC(=O)C(C)n1cccn1)NC(=O)CNC(c1cnoc1C)=O)OC C1(CC)CCN(C(C2CNC(=O)N2)=O)C1C(=O)NC(C(C)C)c1ncc[nH]1 c1(C(=O)Nc2ccc(O)cn2)cn2c(n1)CN(C(c1cncs1)=O)CC2 C=C1CC2CC1CN2C(c1ccc(C(F)F)o1)C(=O)NCCCF C(C)(C)(C(C)NC(C(C)c1cccs1)=O)N(C)Cc1ccsc1.C1(=O)CN1 Cc1cccc(C(F)C(=O)NCCCCNC(=O)CN(C)C(N)=O)c1 c1(CC(=O)NC(CN(C)C(C2CCCC(C)(C)C2)=O)(C)C)cc(F)c(F)cc1F Cc1c(C(=O)N(C(C)(C)CC(=O)NCCC2CCC(C)O2)C)cncc1F N1(C(C2N(C(C)=O)CC(O)C2)=O)CCN(C(C2CCCCC2)=O)C(C)C1 Cc1nn(C)c2c(NCC3(C)CCOC3)nc(N3CC=CC3)nc12 N1(C(c2ccc(C)c(C)c2O)=O)CC2CCCC(C1)N2C(=O)C(C)(C)S(C)(=O)=O n1(CC(=O)NCC2(C)CC(NC(c3c(C)noc3)=O)C2)ccc(=O)c([N+](=O)[O-])c1 Cc1cc(C(=O)NCc2ccsc2C(=O)NC2CCOC2(C)C)ccc1C#N C(=O)(CC(CC)c1ccccc1)N1CCC(N(C(=O)Cc2ccno2)CC#C)C1 c1(CC)ncncc1C(N1CC(O)(CNC(=O)CC2CC2(C)C)C1)=O C1(CCN(C(C(C)OCCN(C)C)=O)C)CCN(C(=O)CCS(C)=O)CC1 c1(-c2nc(CCCC(=O)N(CCCC)CCCO)on2)cncc(F)c1 c1(C(N(CC(C)NC(Cc2c(CC)con2)=O)CC)=O)cccc(OC)c1F c1(CC(=O)NC(c2ccccc2)CNC(C(C)(CO)OC)=O)ccc(Cl)cc1F C1(CC)(NC(c2ccc(O)c(N)n2)=O)CCN(C(c2cccc(F)c2C)=O)CC1 Cc1ncc(C)c(=NCCC2CCCCN2C(=O)CCCc2ccccc2)[nH]1 C1(CCNC(CC2CC(C)(C)C2)=O)CCCN(C(c2cccc(Cl)c2N)=O)CC1 c1(C(N2CC(NCc3ncn(C)c3)C2)=O)ccccc1S(=O)(=O)N1CCCCC1 c1(CCCc2cc(C)[nH]n2)nc(-c2ccco2)nn1C1CCOC1 Cc1cc(O)cc(O)c1CNC1CC(C(N2C3COCC2C3)=O)C1 c1(C(N2CC(CNC(C(CC)F)=O)C2)=O)ccc(Br)cc1N1CCOCC1 C(=O)(C(C)(CCC)CCC)N1CC2C(C(N(C(=O)C(F)(F)F)CCCC)=O)(C2)C1 C1(C(=O)NCC2(NC(CCOCCC)=O)CCC2)CC(O)C(F)C1 C1(C(N2C(C3CCN(C(CNC(N)=O)=O)CC3)CCC2)=O)Cc2cccnc2C1 N1(C(C2(C)CC(F)C2)=O)CC2CN(C(C3CC4CCCC(C3)C4)=O)CC2C1 C(=O)(C(F)(F)C(C)(C)O)N1C(C2CCN(C(c3cc(SC)oc3C)=O)CC2)CCC1 C1(NC(CCCCCCCC)=O)CCOC12CCN(C(C1(OC)CC1)=O)CC2 C1(NC(Cc2c(C)ccnc2)=O)CCCC(NC(c2cc(Cl)c(Cl)[nH]2)=O)CC1 C1(CC)(NC(=O)Cn2cc(CN3CCN(C)CC3)nn2)CCSCC1 c1(C(=O)NC2(c3ccccc3)CCN(C(C)=O)C2)ccc2c(c1)B(O)OC2 C1(CNC(C2C=CC=CC=C2)=O)CCCCN1C(=O)CC1CC2(COC2)C1 C=CCC(C)(C)CC(=O)NC1CN(C(c2cncc3n[nH]cc23)=O)CC1C(F)F N1(C(C(COCC=C)c2ccccc2)=O)CCC(c2ccc(C)cc2)CC1C c1(CC(=O)NCCn2cc(C(=O)NC3(C#C)CC3)nc2)ncccc1C c1(C(=O)OC)c[nH]c(=NCC2CCCCN2C(=O)C(C2CC2)OC)s1 C(C(C)(C)CNC(=O)CC1(O)CCOC1)N(C(=O)CC1CC2(CC2)C1)C N1(C(Cn2c(C)nnn2)=O)CC(C(N2CCN3CCCC3C2)=O)C2(CCC2)C1 Cc1ccc(C(N2CC=CC(NC(C3(C(F)F)CCCC3)=O)C2)=O)cc1 N1(C(CCSC)=O)CCN(C(=O)Cc2nc(C)sc2C)CC1c1cn[nH]c1 CC(C(=O)N1CCC(NC(c2cnn(CC3CC3)c2)=O)C12CC2)S(N)(=O)=O CC(C)(C(=O)N1CCC(C)(NC(c2ccc(N)cc2Cl)=O)C1)C1=CCSCC1 c1(C(=O)NC2CC(C)N(C(C3CC=CCO3)=O)CC2)cn2cccnc2n1 c1(OC)nn(C)cc1CNC(C1CN(C(=O)C(C)C2CCCC2)C2CC12)=O N1(C(C2CCC(C)O2)=O)CCCC12CCN(C(c1cc(C3(C)CC3)on1)=O)C2 c1(CCC(=O)NCC(O)CNC(=O)C(=O)Nc2ncc[nH]2)ccncn1 c1(OC)c(C(=O)NC2COCCN(C(=O)C(C)c3ccco3)C2)c(C)nn1C CCC(C)(C)C(O)C(=O)NC1COCC1NC(=O)C(C)(C)CN1CCOCC1 C(=O)(C(CCF)NC(=O)CCCn1cncn1)N(CC(=O)NC(C)C)C C1(C(=O)OC)CCN(C(c2cc3c(-c4nn[nH]n4)cccc3[nH]2)=O)CC12CCC2 c1(C(N2CCC2C(N2CCC(c3ccc(Cl)cc3)C2)=O)=O)n[nH]c2cccc(F)c12 C(C(C)(CC(C)C)NC(=O)C#CC1CC1)NC(c1c(CC)nco1)=O C(=O)(C1=NOC(C)(C)C1)N(CCC(C(C)C)NC(Cc1ccc(C)cc1Cl)=O)C CC1CN(C(C2CCOCC2)=O)CC1CNC(C1(C)CC1(F)F)=O C1(C(=O)NC(C)C(C)NC(c2cnc(S)[nH]2)=O)CCC(=O)NC1 CC(C)CCN=C(NCC1CC(=O)N(C(C)C)C1)N1CCC2CCCC2C1 c1(C(N2CC(CNC(=O)CCC(N)=O)CC(C)(C)C2)=O)ccccc1P(C)(C)=O CCCCC(CNC(C1CCCOC1)=O)NC(c1ccc(CC)nc1)=O c1(C(N2CCN(C(C(CC)C(C)C)=O)CC2C)=O)c(C)nc(C)nc1C Cc1cc(C)c(NC(C2(F)CCCN(C(C3CCN(C)C3)=O)C2)=O)cc1O C12(C(=O)NCCC(CNC(c3cnc(OCC)s3)=O)O)CC3CC1C2C3 C#CCC(C)C(=O)NCC1CCC1NC(C1CCCC1C(C)C)=O c1(OCC(=O)NCC(CC)NC(C2(C#N)CC=CC2)=O)c(C)cc(Cl)cc1C N#Cc1ccc(S(=O)(=O)N2CCCc3n[nH]cc3C2)cc1F C1(C(=O)NC(CCN(C(c2ccc(NC)cc2)=O)C)C(C)C)CN2CCN1CC2 C(=O)(C(C)(C)C(=O)N1CC2(C1)CN(Cc1ccc(C(C)C)cc1)C2)OC C1(CNC(c2nc(C(=O)OC)sc2)=O)CN(C(c2cc(CO)[nH]n2)=O)CC12CC2 CCC(C)(C)C(O)C(=O)NC(C)CCCNC(=O)Cc1ccsc1 c1(C(=O)NC(C(C)C)C(=O)NCC2CC2c2ccco2)cc2n(n1)CCC2 C1(C(=O)NC2CC(C(N(CC(C)C)C(C)C)=O)C2)CCCCCN1C N1(C(c2cnc(S(C)(=O)=O)s2)=O)CCCC12CCN(C(=O)Cc1cscn1)CC2 Cc1cccc(C(N2CCCCCC2CNC(c2ccnn2C)=O)=O)c1N C(=O)(CCCC(F)(F)F)NCC12C(CN(C(c3c(OC)ncc(Cl)c3)=O)C1)C2 N1(C(c2cc(Cl)cc(Cl)n2)C(=O)NCC=C)CCOc2ccnc(Cl)c2C1 N1(C(c2nc(CC)on2)C)CCC(CC)CC1.c12nc(cs1)CCNC2=O c1(OCCC)ccc(C(=O)NC(C)CCNC(c2cc(C3CCC3)no2)=O)cc1 c1(CC)nn(C)c(CC(=O)NC2CC(CNC(=O)C(O)C(C)SC)C2)c1Br C1(NC(C(CCC)=CCC)=O)CCN(C(c2ccc(CC)c(N)c2)=O)CC1F c1(C(=O)OCC)cnc2cc(Cl)c(Cl)cc2c1OCCc1noc(CC)n1 C(CC(=O)NC1CCN(C(=O)C(F)=CC2CC2)C12CC2)(C(N)=O)NC(C)=O N#Cc1cccc(CN2CCOCC(C(=O)Nc3cc(Cl)ccc3F)C2)n1 C(CCCCCC(=O)N1CCc2sccc2C1)NC(C1(CC#C)CCCC1)=O N1(C(C2C(C)N(C)CC2)=O)CC2CN(C(c3ccccc3Cl)=O)CC2(C)C1 c1(C(N2CC(C)(C)C2COC)C(=O)NCCCCCC)nc(C)n(C)n1 C#CCC(C(=O)Nc1cnc(SC)nc1)NC(C1CC1Cl)=O CCCC(CC)C(=O)NC1CCCCC1CNC(=O)Cc1c(C)noc1Cl N1(C(Cn2c(C)ccn2)=O)CCN(C(=O)CC(C)F)C(CC2CC2)C1 C1(NC(C2C(=C)CC2)=O)(CNC(c2cc(Br)no2)=O)CCCC1 c1(OC)cc[n+]([O-])c(C(=O)NCC2CC(NC(c3cc(C(N)=O)[nH]n3)=O)C2)c1 c1(C(=O)NCCN(c2cnc(OC(C)C)cn2)CCC)nc(C)c(C)s1 C1(CNC(c2cc(CC)n(C)n2)=O)CCC2CN(C(=O)C(O)CSC)CC12 C#Cc1cnn(C)c1C(=O)NCC1CCCCN1C(=O)C(COC)N(C)C c1(CC(=O)N(CC2CCN(C(CC3C(CC)C3)=O)CC2)CC)ccc(F)c(Cl)c1 c1(C(N2CC(CF)C2)=O)ccc(CNC(C2CCOCC2)=O)o1.C1C(=O)N1 c1(OCC)c(C)cc(C(=O)NC2CC(NCc3ccccc3F)C2)cc1C C1(C(N(C)C)=O)CC(NC(=O)C(=O)NCc2cncc(C3CC3)c2)C12CCC2 CCCC(C#N)C(=O)N1CC(CN2CCN(C(=O)CC3CC3(Cl)Cl)CC2)C1 CC1(C)CCCC1CNC(=O)C=CCNC(=O)COCCN(C)C N1(C(COCCCC(C)C)=O)CCC(n2cc(C3(C(=O)O)CC3)nn2)CC1 CC(C)CCC(C(=O)NCC(C)CC1CCC1)NC(C12CCC(C1)C2(C)C)=O c1(C(=O)NCCN(C2CCCC2)C(COC(CC)(C)C)=O)cc(Cl)c(Cl)n1C C=CC(C)(CC)C(=O)N(CC(C)(C)NC(=O)C=Cc1ccnn1CC)C C(=O)(CCS(=O)(=O)C1CCCC1)NC1C(NC(=O)COC2CCCCC2)CCC1 c1(C(=O)NCCC(C)N(c2ncnc(CO)n2)C)ccc(O)nc1 C(C(C(C)C(C)C)NC(c1cn(CCO)nn1)=O)NC(CCOCC(C)C)=O C1(O)(C(C)NC(c2n(CC=C)ccn2)=O)CCN(C(=O)CC2CC3CCC2C3)C1 C1(C(=O)NCC2(C)CC2)CCN(C(=O)C2C3CC(=O)CC23)O1 C(CCN=c1cc[nH]c(=NCCCCC2CCCC2)[nH]1)N1CCNCC1 C1(NC(c2c(C)cccc2)=O)CCN(C(=O)CC2CCCCCC2)CC1C(C)C C12(CC3CCC1CC3)NC(=O)C1C(OCC1)C(=O)NC2.c1(CC)ccccc1O C(=O)(C(C)(C)C1=CCSCC1)NC1CCN(C(CCC(CCC)CC)=O)CC1F N1(C(COCCC(C)C)=O)CC2CCN(C(c3cc(CF)on3)=O)C(C2)C1 C1(C)(CNC(C(CC)COC)=O)COCCN(C(=O)C(F)(F)c2ccccn2)C1 N1(C(c2cc(C)cc(Cl)c2)=O)CC2CCCC2(NC(c2ccn(C)c2C)=O)C1 N1(CCN(C2C(C)C2)C(=O)CC)CCC(n2[nH]c(CN(C)C)nc2=S)CC1 c1(C(=O)NC2(COC)CN(C(CC3CC(CC)C3)=O)C2)cnc2ccncc2c1 C(=O)(C1c2c[nH]nc2CN1C(=O)C1=C(Cl)CCCC1)Nc1cncc(OC)c1 CC1(C)OCCOC1CNC(=O)NC1CC12CCCCC2 C1(C(N(C2CCCN(C(C(CC)CC)=O)C2)CCO)=O)CC(=O)NC(C)C1 c1(C(=O)OC)c(F)cc(CN2CCOC(C(=O)NCC3(F)CCC3)C2)cc1F c1(OC)cccc(C(=O)OCCS(=O)Cc2nc(-c3ccncc3)no2)c1 c1(C(N2CCC(n3cccc3)C2)=O)csc(-c2ccoc2)n1 C(CCC(C(=O)NCc1ccccc1OC)N(C(C)COC)C)OCC c1(C(N(CC(=O)NC2CC2)C)=O)cc2c(nn1)CCC2.C1(=O)COCCN1 N1(C(CC(C)(C)NC(=O)CC=C(Cl)Cl)=O)CC2CC2(C(=O)OC(C)(C)C)C1 Nc1ccc(Cl)cc1C(=O)NC1COCC1CNC(C1CC1c1cn[nH]c1)=O C1(C(=O)NCCC(C)(C)NC(c2c(CCC)n(C)nn2)=O)C2CCC(F)(F)C12 c1(C(=O)NC2C(CC)N(C(=O)C(C)=C3CCCC3)CC2)[nH]c2ccccc2c1Cl c1(CC)nccnc1C(=O)NCCC(O)C(=O)NC1CCCC(CO)C1 C(=O)(C(CCc1ccccc1)NC(=O)C(C#N)C=Cc1ccccc1)OCC C1(NC(C(C)n2cncn2)=O)CC2(C1)CN(C(=O)C(C1CCOCC1)O)C2 Cn1nc2cc(Br)ccc2c1CN1CCC(NS(=O)(=O)c2cccc(F)c2)CC1 c1(NC(=O)NC(Cc2ccoc2)CO)csc2c1CCCC2 Cc1ccc2c(=NC(C)c3csnn3)[nH]c(N3CCC4(CC4C(N)=O)C3)nc2c1 Cc1cc(CCC(=O)NCCC2(NC(=O)C(C)CF)CCC2)cc(C)c1 C(=O)(CC(C(C)CC)NC(C1CCSCC1)=O)NC(CCC=C)(C)C c1(C(=O)NC2(C)CSC2)nocc1C1CC1 c1(C(N2CCC(NC(CC(C)F)=O)C2)=O)ccc(NCCON)cc1 C=CC(C)(C)C(=O)NCC1CCN1C(C1CCCN(Cc2ccc(O)cc2)C1)=O O=C(C1COc2ccccc21)NC1(C2CCN(C(C3CC34CCOC4)=O)C2)CC1 c1(C(N(CCC)CCNC(C2CCC(C)(C)CO2)=O)=O)ccnc(S(N)(=O)=O)c1 c1(C(N(C)Cc2ccsc2)=O)nnc(S)s1 CC1CCCC1(C)C(=O)NCCc1cn(CCN(CCCF)CCO)nn1 C1(CCCC)CN(C(=O)CN(C)CC)CCN1C(c1ccoc1C)=O.C1(=O)CN1 C1(CC(=O)NCc2c(C)cns2)CN(C(=O)Cc2ccccn2)CCC1C n1(CC(=O)NC(C)CCNC(=O)CC#N)cc2ccccc2n1 N1(C(C(C)NS(CC)(=O)=O)=O)CC2CC(CNC(C3OCCCO3)=O)C2C1 c1(C(=O)NCC2CN(C(C3CCC(C)(CC)O3)=O)C2)cc(N)c(C)c(N)c1 N1(C(CC(=C)C)=O)CCC(CCNC(c2scc3c2CCCC3)=O)C(F)(F)CC1 C(=O)(C1SCCc2ccccc21)N1CC(N(C(=O)CCc2cnoc2)C)C1 C1(CNC(c2cnc3ncccn23)=O)CCN(C(=O)C(O)C(F)(F)F)CC1(F)F C1(C(=O)NC2C(NC(c3c(N)c(Cl)ccc3)=O)CC2)CCOCC12CCC2 c1(C(=O)NCCNC(C(C2CCCC2)OCC)=O)cc(O)cc([N+](=O)[O-])c1 C1(C(=O)NCCN(C2CC2)CC)C(C)OCCN1C(=O)CC1CCC(C)CO1 N1(C(CC=CC=C)=O)CCN(C(=O)Cc2cc(OC)cc(C(F)(F)F)c2)C2CC12 Cc1ccc(C(C)(C)C(N2CCC(CO)(NC(c3ccsn3)=O)C2)=O)cc1 Clc1ccc(C2(NCc3cnc(C4CC4)nc3)CCOCC2)cc1Cl c1(N2CCC(CNC(CSCCCC)=O)C(C)C2)nc2cc(C)ccc2o1 CCC(CC(=O)N)C(F)F.c1nc(=N)[nH][nH]1.C1CCCC2CN1C2 CC(N=c1cc[nH]cc1S(=O)(=O)NCc1csnn1)c1cccc(Cl)c1 N1(C(C(C2CC2)OC)=O)CC2(CCC(CNC(c3cccc4sccc34)=O)O2)C1 C(=O)(C1=CCCCCC1)NCC1C(CC)CN(C(=O)CC2C=CS(=O)(=O)C2)CC1 Cc1ccccc1-n1cc(C(N2CCN(C(N)=O)CC2)C2(N(C)C)CC2)nn1 C1(C(=O)NC(n2cc(CN(C)CCOC)nn2)C(C)C)CC(c2ccccc2)=NO1 C1(CC(N2CCCC(C)C2)=O)N(C(c2ccn(C3CC3)n2)=O)CCC1(C)C C(Cc1cn[nH]c1)(C(=O)NOCC)NCc1cn(-c2c(CC)n(C)cc2)nn1 C(C(=O)NC1C=CC(C(N2CC(OC(F)F)C2)=O)C1)(C(C)C)SC C(=O)(C1CCCc2nnn(C)c21)NC1CN(C(c2c(CC)n[nH]c2)=O)CC(F)C1 C1(C(N2C(CC)C(CO)CC2)=O)Cc2c(C)cccc2O1 c1(C(=O)NC(CNC(C(C#N)C2CC2)=O)C2CCC2)ccc(-n2cccn2)cc1 Cc1c(Cl)ccc(C(=O)NCC2C3CN(CCC4CCCCCCC4)CC23)c1Cl C1(CN(C(=O)CC(c2cccs2)C2CC2)C)CCN(CC(C)(C)C)CC1 C(=O)(C1=Cc2ccccc2C1O)NCCN(C)C(c1cccc2nc(O)[nH]c12)=O C=CC1(CO)CCN(C(C2C=CCCN2C(c2cc(Cl)ns2)=O)=O)CC1 N1(C(C(C(C)OC)NC(C(C(C)C)SCC)=O)=O)CCC2(C1)CN(C(C)=O)C2 Cc1nc(C(C)C)ncc1C(=O)NCC(C1CCC1)NC(=O)C(Cl)=CCl c1(CSC)cccc(C(=O)NCC2(NC(=O)CN3CCOC3=O)CCCCC2)c1 N1(C(C=C(C)C(F)F)=O)CC2C(CN(C(=O)CC(C)N(C)C)C)C2C1 C1(C(=O)NCC(C)(CO)NC(C=C(CCC)C)=O)CCN(C)S1(=O)=O C(CCCCF)NC(CCN(C(=O)Cn1cc(CO)nn1)C)=O N1(C(N2CCC(O)(c3ccccc3)C(O)C2)=O)CC2CCCCC2C1 C1(NC(C(CO)N(C)C)=O)CN(C(c2cnc(C(N)=O)s2)=O)CCC1CO Cc1n[nH]c(=NC(=O)c2ncn3c2CCCC3)n1C C1(CNC(C(C)OCCCC)=O)CCN(C(c2ccnnc2)=O)C12CC2 CCN=C(NCC1CCC1)NCc1cccn1CC1OCCC1C CC1OC2(CNC(N3CCOC(c4cccc(C(F)(F)F)c4)C3)=O)CCC1C2 c1(C(N2CCCC(N(C(C=COCC)=O)CC)C2)=O)cn2ccn(C)c(=O)c2n1 N1(C(CN(CC(C)C)C(c2cccc(CC=C)c2)=O)=O)C2C=CCC1CCC2 c1(C(=O)NCCCCC(C)NC(C2CCS(=O)(=O)C2)=O)c(N)nn2ccccc12 CN=c1ccc(C(N2CCSC3CCC23)=O)c[nH]1 C1(NC(C2(C)CC3CC3C2)=O)CN(C(=O)CCC2CC(F)(F)C2)C2(CCCC2)C1 c1(NC)cncc(C(=O)NCc2cc(C(N3CCC(N(C)C)C3)=O)n(C)n2)c1 C1(O)(CNC(C=CC=CCCCCC)=O)CCN(C(=O)CC2CNC(=O)C2)C1 C1(NC(Cc2ccc(C)nc2)=O)CC2CN(C(C3(C4CCC4)CC3)=O)CC12 C1(C(C)OC)CCN(C(=O)C=CC2CCCN2C(c2n[nH]c(=N)[nH]2)=O)CC1 N1(C(c2ccc(C#C)o2)=O)CCC(C2CC2)C1C(N1CCCOC(C)C1)=O C1(CC)(CNC(=O)CC2C=CC(NC(C3CCOC3)=O)C2)CC(C)(C)C1 C(=O)(CS(=O)(=O)C1CC1)NC1CC(NC(c2c(COC)nn[nH]2)=O)C1 N1(C(C2NC(=O)OCC2)=O)CCC(C(F)(F)F)C(N)C1 C1(NC(c2c(CC)non2)=O)CCN(Cc2ccn(Cc3ccccc3)n2)CC1 C=C1CC(C(F)(F)F)(C(N2CC(O)(CNC(C3CCCCS3)=O)C2)=O)C1 C1(O)(C(N2CCCC(NC(c3occ4c3CCC4)=O)C2)=O)CC2(CCOCC2)C1 c1(CN(C(C2(CC)CN(C(c3ccsc3C)=O)C2)=O)C)cccc(C)c1 c1(C(N(CC(C)NC(C2(c3nccs3)CC2)=O)C)=O)cnccc1N(C)C Cc1ccc(C)c(C(N2CCN(C(c3cn(CCO)nn3)=O)C3CC23)=O)n1 N1(C(CC=CC)=O)CCC(c2ccccc2)(NC(=O)C(CC)OCC)C1 C1(C(CNC(c2c(SC)csc2)=O)O)CCN(C(=O)C(CCO)N(C)C)CC1 c1(C(N(C(CCNC(COC(CC)C)=O)C)C)=O)c(F)ccnc1Cl Cc1nn(C)c(C)c1C(=O)NC1CCCCC1C(N1CCCC(CCCO)C1)=O C(=O)(C(F)CCC(C)C)NCC1CCN(C(C2CC(CC)OCC2)=O)CC1 O=C1CC(C(=O)N2CC3(C2)CN(C(c2cc4c[nH]nc4s2)=O)C3)c2ccccc21 Cc1nc(N2CCC(NC(c3sccc3C(C)C)=O)C2)ccc1C#N Cc1ccc2c(CCC(N3CC(F)(CNC(C4CC4(C)CF)=O)C3)=O)c[nH]c2c1 CC(O)C(C)CNC(=O)C(CC1CC1)NC(=O)CC(C1CC1)C1CC1 CC#CCC(C(=O)NCC1CC2CCCC2C1)NC(c1cccc(C)c1)=O C1(C(C)(C)C)CC(CNC(C2(F)CCCC2)=O)CN(C(=O)Cc2ccsn2)C1 C(=O)(CCC1=CCCCC1)NC(CC(=O)NCC1(C)ON=C(C)C1)C C1(NC(C(CO)OC)=O)COC2CN(C(=O)CC3CCSC3)CC12 C1(CNC(c2cncc(SC)c2)=O)CCCCCN1C(c1cn(CO)nc1C)=O N1(CC(COCC(C)C)O)CCC(C)(NC(c2cnc(Cl)c(Cl)c2)=O)CC1 C1(C(=O)NCCC2(NC(C(=O)NCCOC)=O)CC2)CS(=O)(=O)CC12CC2 CC(N=c1[nH]c2cc(Cl)ccc2s1)C1CCCN(C(=O)C(O)C2CCC2)C1 Cc1ccc(C(N2CC(NC(c3c[nH]c(=N)o3)=O)C3(CC3)C2)=O)c(C)c1 CC1=C(C(=O)NCC2CC3(CC(NC(c4cnc(S)nc4)=O)C3)C2)CCC1 CCC(C)(C)CCCC(=O)N1CC(C)N(C(=O)C(C)OC2CCCCC2)CC1C CC1CCC(OC(=O)C=C(C2CC2)C2CC2)C=C1Br Cc1ccc(C)c(C(N2CCC(NC(=O)C(C)(C)n3ccc(C4CC4)n3)C2)=O)c1C N1(C(CC=CC)=O)CCN(C(c2ccnc(C3CCC3)c2)=O)C(C(F)F)C1 C1(O)(CNC(CN(CC(C)(C)C)C)=O)CC(C)(C)C1.C12(C)CC(C1)NC2=O c1(C(C)NC(c2c(C)n(CC(F)(F)F)nc2)=O)ccc2c(c1)CC(=O)N2C c1(CC)ncc(C(N2CC(NC(C3CC34CCOCC4)=O)CC(F)C2)=O)c(O)n1 c1(C(N2C(c3ncc(C)s3)CCCC2)=O)cc(O)c(Br)c(O)c1 CC1CN(C(=O)C(F)CC2CCOC2)CC1NC(C1CCNC(=O)C1)=O Cc1nc(C=CC(N2CCCC2(C)CNC(c2ccncc2)=O)=O)cs1 C(=O)(CC(C)n1ccc(C)n1)NC1(CCCNC(COCCCCC)=O)CC1 c1(C(=O)NC(CCCCNC(C(C)(C2CC2)OC)=O)C)ccn2ncccc12 c1(C(=O)NC(C2CCOCC2)C#C)cc2cccc(Br)c2nc1C C1(C(C)(F)F)(C(=O)NC2(C)CN(C(C(C)NC(N)=O)=O)C2)CCOCC1 C=C(C)CCCC(=O)NCC1CC1CNC(=O)C(C)(C1CCOCC1)OC Cc1cnc(NC(c2cccc(Cl)c2Cl)C)c(S(=O)(=O)N2CCC(CO)CC2)c1 c1(C(=O)NCCCCN(C(C2(C(=O)OC)C=CCC2)=O)C)cccc2ncsc12 C(=O)(C(F)(F)CC(C)C)N1CCC(O)(C(C)NC(c2cccc(OCC)c2)=O)C1 N1(C(C2CC=C(C)CC2)=O)CCC2(CC1)CCN(C(C1COC(=O)O1)=O)CC2 N1(C(c2c(C)snc2)=O)CCc2cc(-c3cn(C4CCOC4)nn3)ccc21 c1(COc2ccc(OCC)cc2)n[nH]c(=NC(CO)C(C)C)n1Cc1ccccc1 C(CCC(C(=O)NCc1[nH]cnc1C)NC(c1ccsc1OC)=O)OC C1(C)(C(=O)NC(CC)CN(C(=O)C(F)=C2CCCC2)C)CS(=O)(=O)C1 C1(NC(C2CCN(CC#C)CC2)=O)COCCN(C(C2CC3CCC2O3)=O)C1 c1(OC)ccc(C(=O)NCC2(F)CC(NC(C3CCCS3(=O)=O)=O)C2)nc1Cl c1(CNC(CC2CCC(NC(C3C(C(C)C)C3)=O)C2)=O)noc(C(N)=O)n1 C(=O)(CC1NC(=O)c2ccccc21)N1CCC(NC(CNS(NC)(=O)=O)=O)CC1 c1(C(N2C(CNC(CCS(C)(=O)=O)=O)CC3CC32)=O)ccc2ncccn12 Nc1ccc(C(N2CCCC2CCNC(C2CCCC(C(N)=O)C2)=O)=O)cc1O N1(C(c2c(C)c(Br)no2)=O)CC2CC(NC(=O)COc3cccnc3)C2C1 c1(C(N2C(C(C)NC(=O)CC3CCC34CCC4)CCC2)=O)cnn2ncccc12 c1(OC)ccc(C(N2CCN(C(=O)COc3cccnc3)C(CO)C2)=O)c(C)n1 N1(CC)CCC(NC(c2ncoc2CNC(=O)C(C)(O)C2CCC2)=O)C1 N1(C(C2CN(C(=O)C=CCO)CCO2)=O)CC(F)(F)CC1CO CCC(C)C(O)C(=O)NC1CCC(C(N2CCOC(CC)C2)=O)CC1 CCC(C)(C)CC(=O)NCC(C)(F)CNC(=O)C=Cc1ccsc1 CCC(C)C(C(=O)NC1CCC(CNC(C2(CC(C)C)CCCC2)=O)CC1)OC c1(OC)cc(C(=O)N(CC(O)CN(C(=O)C2=CSCS2)C)C)n(C)n1 C1(C(N2CCCC2CO)=O)CN(C(c2cnccc2-c2ccccc2)=O)CCO1 C(C)(C(C)(C)C(=O)N1CCCC(OC)C1C)NC(c1n(CC)nnc1)=O c1(C(N(c2csc(NCC(N)=O)n2)C(C)=O)=O)cc(Br)ccc1NC(COC)=O N1(C(COC(C)=O)=O)CCC(NC(c2cc3c(cn2)CCCC3)=O)C12CCCC2 C1(O)(CNC(C23CC(NC(CNS(NC)(=O)=O)=O)(C2)C3)=O)CCCC1C Cn1nc(C(=O)NCCC2CCCN2C(=O)CC2(C)CC2(F)Cl)cc1CO c1(C(=O)NC2CCC(NC(C=C(C)Cl)=O)C2)ccc(Cl)c(F)c1O c1(C(=O)NCC(C2(O)CCN(C(c3nn(C)cc3N)=O)C2)C)ccc[n+]([O-])c1 C1(C(N(C)Cc2onc(C)n2)=O)CN(C(c2[nH]ccc(=O)c2C)=O)CC1C1CC1 C(CO)(CCC(C)C)N(C(C(CCSC)NC(CCC#C)=O)=O)C(C)C CCCCCC(C)(CC)C(=O)NCC(C(C)C)NC(C1(C)CCC(C)C1(C)C)=O N#Cc1ccc(CNC2CCCCC2NC(=O)CCC2CCOCC2)nc1 C1(C(=O)NCCC(C)N(C)C(c2coc(C(F)F)n2)=O)CC2(CCOCC2)CO1 c1(OCC)cccc(C(=O)NC2CCN(C(=O)C(C3CCC3)OCC)C2C)c1N Cc1nc2cccc(C(=O)N(CC(C)NC(=O)C=Cc3cncnc3O)C)c2s1 N1(C(c2c(C)oc(Cl)n2)=O)CCCOC(CCNC(C2CCO2)=O)C1 C1(C(N2CC(C(C)NC(c3cc(C4CCCC4)no3)=O)C2)=O)C(F)(F)C12CC2 C1(OCCC)CCCN(C(C2CN(C(=O)C(C(C)C)N(C)C)CC2C)=O)C1 Cc1c(C=CC(=O)NC2(CCCNC(C3COC(C)C3)=O)CC2)cnn1C C1(CNC(CCN(CCCCC)CC)=O)CCN(C(=O)CS(C)(=O)=O)C1(C)C c1(C(=O)NCC(CNC(c2c(C#N)cn[nH]2)=O)O)cc2c(nc1O)CCOC2 CCC(C)CCC(=O)NCCN(C(=O)CC1(C)CCOCC1)C1CC1 N1(CC)C(=O)CCC1C(N1CC2C(NC(c3c(CO)noc3C)=O)C2C1)=O C#CC1CCCN(C(=O)CCOCCN(C(=O)C=CC(=O)OCC)C)CC1 C(CCF)(C(=O)NCCCNC(=O)OC)NC(C(CC)=CCCC)=O N1(C(CC)CO)CC2(C1)CN(S(=O)(=O)C(F)(F)F)C2.CC(=O)OCCO C1(C2CC2)(CNC(C(C=C)O)=O)CCN(C(c2cc(CC)nnc2C)=O)C1 C(=O)(C(C(C)C)C(C)C)NC12CC(CNC(CCCCOCC)=O)(OC1)C2 CC(C(=O)NC1(CCCNC(c2ccc(-c3ccccc3)[nH]2)=O)CC1)P(C)(C)=O C1(NC(CC(C=C)(C)C)=O)CN(C(=O)C2=CCCOC2)C2CCCCC12 C1(C(=O)NCC(C2(O)CN(C(=O)C3=CCCCC3)C2)(C)C)CC2CCCC2C1 N1(C(c2cnc(OC)nc2C)=O)CC(NC(=O)CCCCCF)C(C2CC2)C1 c1(CC)cc(C(N2CCCOC(CNC(C3CC4(CSC4)C3)=O)C2)=O)cc(O)n1 c1(C(=O)NCCNC(C2CCCC3(CC3)C2)=O)cc2c(Br)cncc2s1 C1(N(C(=O)CC2C=NN(C)C2=O)C)CCCN(C(C23COCC(C2)C3)=O)CC1 C1(C(N2C(CN(C(CNC(CC)=O)=O)C)CCC2)=O)CCCN1N=O c1(CC(C)(C)C)noc2ncc(C(N3CCN(C(=O)C(F)F)C(CF)C3)=O)cc12 C1(C(N2CCC3(CCC3)C2)=O)CCN(C(=O)c2cccc(Cl)c2)O1 C1(SC)CC(C(=O)N(CCC(=O)NCC2(CC3CC3)CC2)C2CC2)C1 c1(OC)cccc(C(N2CCC3(CC3C(=O)NC3CS(=O)(=O)C3)C2)=O)c1OC c1(C(N(CCC(C)NC(c2cn(CCC)nc2)=O)C)=O)sc2ccsc2c1C CC(C)(CN=c1[nH]nc(C#N)s1)NC(c1csc([N+](=O)[O-])c1)=O N1(C(C2(C)CC(F)C2)=O)CCCCC(CNC(c2ccc(SC(F)(F)F)o2)=O)C1 N1(C(CCC#CC)=O)CCC(C)(C(=O)NCC(C)COCC)CC1 C(=O)(CC(C)(O)C(F)(F)F)N1CC(C)(CNC(c2c(CC)ocn2)=O)OCC1 C1(C(N2C(CNC(CC=C)=O)CCC2)=O)CCC(C(F)(F)F)CC1 C1(CCS(N)(=O)=O)CCCN1N1CCCC(c2nc3ccc(Br)cc3[nH]2)C1 C1(NC(CC)=O)CC(O)CN(C(C2(NC(=O)OC(C)(C)C)CC2C)=O)C1 c1(OC(C)(C)C)ccnc(CNCC23CC(CCO2)C3)c1 c1(OC)ccc2c(c1)CCC2C(=O)NC1CCC(NC(c2nocc2C)=O)CC1 C1(CC)CCCCC1C(=O)N(C1CCN(C(c2ccncc2)=O)CC1)CCO C(=O)(CCC(F)(F)C(=O)NC1CCC(C)N(C(c2cccnc2O)=O)C1)OCC C(CC(C)C(=O)NC(CNC(C1(c2ccn(C)n2)CC1)=O)CC)=CC N1(C(C(C)C#N)=O)CC(O)(C2CCN(C(=O)COc3c(F)cccc3F)CC2)C1 c1(C(=O)N(C)C)ncccc1O.C(=O)(CCOCCCN)N(C)CCNC C1(C(N2CCN(CCn3cc(C(CC)OC)nn3)CC2)=O)CC2COCC(C1)C2 CC1CCN(C(=O)Cc2ccsc2Cl)C1CNC(C1(C(C)(F)F)CCOCC1)=O c1(OCC)ccc(S(=O)(=O)NCCc2c(F)cccc2Cl)cc1C(C)C C=CC(C)CC(=O)N1CC(N(C)C)C(CNC(C2(C(C)(F)F)CC2)=O)C1 N1(C(=O)CC2CCCCO2)CC2CCC1CN2C(c1coc(C(F)F)n1)=O CC(C(=O)NC1CC(O)CN(C(=O)Cc2cnccc2Cl)C1)S(N)(=O)=O c1(C(=O)O)cccc2nc(CNCC3(COc4ccccc4)CCCO3)[nH]c12 S(=O)(=O)(c1ccccc1C#N)N(C)Cc1nc(Br)cs1 C1(C(=O)OCC)CCN(C(=O)C(Cc2ccc(C)cc2)NC(C)=O)C1C N#Cc1cnn2cc(C(=O)NC3CCCN(C(c4ccccn4)=O)C3)cnc12 C1(C2CC2)(C(N2CCC(NC(C)=O)C2)=O)CN(C(=O)CSCCC#N)C1 c1(C(=O)NC2CN(C(C34OC(C)(C)C(C3)C4)=O)C2)cnn2ncccc12 N1(C(c2c(OC)nccc2)=O)CCOC2(C1)CN(CCN=c1cc(C)nc[nH]1)C2 CC(C)CC(CNC(c1ccn(CCNC(C23CC(F)(C2)C3)=O)c1)=O)CO C(=O)(CCCCC(C)=O)N1CC(C)(COC)C1 C1(NC(CC(C=C)C)=O)CN(C(=O)C=CC=C(Cl)Cl)CCC12CCOCC2 CC(O)(CC(=O)NC1(C)CC(NC(c2cccc(N)c2)=O)C1)c1ccccc1 c1(NC(N(C)C)=O)ccnc2ccc(C(N3CCCCC3CS(C)(=O)=O)=O)cc12 c1(C(=O)NC2CN(C(c3cccc(I)c3Cl)=O)CC23CC3)c(O)cc(O)cc1O C=CCC(CNC(=O)C(F)CCCC)C(=O)NC(c1cc(C)no1)(C)C CC(C)C(F)(CNC(C1C=CCS1)=O)C(=O)N1CC(C)(O)C1 C1(CNC(COC(C)C)=O)C2CN(C(=O)C(c3ccc(F)cc3)F)CC12 c1(C(C(=O)NC2CC(NC(c3ccc(OC)nn3)=O)C2)O)cc(F)c(F)c(F)c1 CC1(C)CN(C(c2ccccc2Br)=O)CC(C)(C)C1NC(=O)C1=NOCC1 c1(OCCC(=O)N(C)CC2CCCN(C(C(CC#C)C)=O)C2)ccc(F)cc1Cl C(=O)(C1OCCc2ccccc21)N1CCCCC(NC(c2ccco2)=O)C1 C1(O)(CCNC(C=CCN(C)CC)=O)CCCN(C(=O)C(C)C2(O)CCC2)C1 C1(C(N(CCCC(=O)NC)C)=O)CCC(C)N(C(=O)CCC2CC2)C1 C=CCCCCCCCCC(=O)NC1CN(C(=O)C(C)n2cccn2)CC1SC CC1(C)CC(C(=O)NCCNC(C2CCCN(C(=O)CC(F)(F)Cl)C2)=O)CCO1 C(C(C)(C)C(=O)NCC1(CO)CCN(C(C2CC=CCO2)=O)C1)OC CCC(C)CCC(=O)NCCn1cnc(C(=O)NCC2(Cl)CC2(F)F)c1 N1(C(CC(=O)OC)=O)CCC(C2CCCN2C(=O)C(C2CCC2)OC)CC1 N1(C(COCC)=O)CCC2(CCCC2C(N2CCC(C)(C)C2)=O)C1 C1(CNC(CCc2ccc(N(C)C)cc2)=O)CCOC2(CCCC2)C1 C1(C(C(=O)N(CCNC(C=CSC)=O)C(C)C)C)CCC(C)(C)CC1 c1(C(N(C2CCCCC2NC(=O)Cn2cc(Br)c(=N)[nH]2)C)=O)cnncc1O N1(C(C)=O)CCCC1C(=O)N(C1CC(NC(=O)C(C)C2CCOC2)C1)C N1(CCC)C(=S)NC(c2ncoc2C2CC2)C(C(=O)OC)=C1c1cccc(C)n1 C(=O)(C(C(C)NC(C1CCC2(CCC2)O1)=O)C(C)C)NC(C#C)(C)C C1(C)(Cc2cn(CC(C)NC(=O)CC3CCCOC3)nn2)Cc2ccccc21 C(=O)(CS(=O)(=O)C1CCCC1)NC1CC(NC(c2ccc(C#C)c(C)c2)=O)C1 C1(C)(CNC(c2cc(OC)ncc2)=O)CCCN(C(C2CC=CCO2)=O)C1 N1(C(C2(NC(C(C(CC)C)O)=O)CCCCC2)=O)CCOC2COCC12 N1(C(c2ccc(C)n2C)=O)CCC(NC(=O)CC2CCOC2)C(F)(F)CC1 N1(C(CCOC)=O)CC2CCCC(CNc3nccc(C)n3)C2C1 N1(C(C2(C)CCSCC2)=O)CCCC(CO)(NC(=O)C=Cc2ccncc2)C1 C(=O)(CCCCCN(C(=O)CC(C)(C)C)C)NC(c1cccnc1N(C)C)C CC(C)CC(C(=O)N1CCC(n2cc(C(c3nn(C)cc3Br)=O)nn2)CC1)N(C)C C1(NC(COC(CC)C)=O)CCCCN(CC(c2ccccc2)O)C1 N1(C(C2C(C)C2)=O)CC(O)(C(C)NC(c2csc(-c3cnc[nH]3)n2)=O)C1 Cc1c(C(=O)NC(C2CCCN2C(=O)CCSCC(N)=O)C)ccn1CCO Cc1nn(C)c2c(N3CCN(C)CC3)nc(N3CCC(n4ccnc4)C3)nc12 N1(C(c2n(CCC)ncc2)=O)C2CCC1CN(C(C1CCOCC1)=O)CC2 C(=O)(C(C)CCCCCC)NC(CC#C)C(=O)NCC=CCl N1(C(c2ncn(CC)n2)=O)C2CCC1C(F)C(NC(c1coc(Cl)n1)=O)C2 Cc1cc(=NC(=O)C(=O)NCC2CC2(C)C)[nH]n1CC1CC1 C(C(C)(C(=O)N1CC2C(NC(c3coc(Br)c3)=O)C2C1)OC)OC c1(C(N2CCC(N(C(C(C)NC(C3CCC3)=O)=O)C)C2)=O)cccc2cnnn12 Cc1cccc2c1CCC2NC(c1ccc(OC(F)(F)F)cc1Cl)=O c1(CC)c[nH]nc1C=O.c1(C(N(C(CCN2CCCC2)C)C)=O)ccncn1 N1(C(C2CC(OC)C2)=O)CCC(NC(=O)C(C)Cc2cccnc2)C(O)C1 C1(C(N2CCC(NC(C3CC3Sc3ccccc3)=O)C2)=O)CCN(CCF)CC1 c1(C(=O)NCC(C2CC2)NC(c2nc(COCC)sc2)=O)sc(CC2CC2)nc1C C1(C)(CC(=O)NC(C(C)C)CNC(C2CCOC2)=O)CC(F)(F)C1 Cc1cc(N(C)Cc2ncoc2C(F)F)nc(N(CC(C)(C)C)C)n1 C(CCC(=O)NC1CCCC1NC(C1CCN(CC(F)(F)F)C1)=O)=CCC=C c1(C(N(CC(C)NC(=O)CCc2ncccn2)CC)=O)cccc([N+](=O)[O-])c1Cl C1(CNC(=O)C(O)c2cnc[nH]2)C2CC1N(C(c1cccc(C(F)F)c1)=O)C2 c1(N2C3CC(CC(NC(c4c(CCC)n[nH]c4)=O)C3)C2)c(C)cncc1[N+](=O)[O-] c1(CNC2CCC(NC(=O)CCc3cc(Br)ccc3Br)C2)cc(Cl)cc(Cl)c1Cl c1(CCC(=O)N(CC)Cc2cccnc2)ccc(Br)c(Cl)c1 c1(C(CC)C)nccc(N2CC(C)(NC(=O)Cc3ccnn3C)C2)n1 c1(N2CCCC(CNC(c3cn4c(n3)CCC4)=O)CC2)nc2ccccc2s1 Cc1cc(C(N2CCN(C(=O)C(C)C(C)(C)C)C3CC23)=O)n2nc(C)c(C)c2n1 c1(C(=O)NCC(CC)NC(c2cc(C)ncc2C)=O)ccn2c1CSCC2 N1(C(C(C#N)=CC(C)C)=O)CCC2(NC(=O)C(Cl)=CCl)CCCC12 C1(C)(NC(C2CC(CNC(C(COCC)C)=O)OC2)=O)CCCOC1 N1(C(C2C(C=C)C2)=O)CCN(C(c2cc3cccc(F)c3o2)=O)CC(C)(C)C1 C1(C(CC)=O)CCC(C(=O)N(C2CC2)Cc2cn(Cc3cnnn3C)nn2)CC1 c1(C(N(C)CC2CCCN(C(C3C(C#C)C3(C)C)=O)C2)=O)cnc(C)c(N)c1 NC1CN(C(=O)COCCOCC2CCOC2)CC12CCC2.C1CO1 CCCCCCCCCC(=O)NC1C2CCN(C(=O)C(=O)C(C)(C)C)C12 C1(NC(c2cnc(Cl)s2)=O)CC2CC1N(C(c1ccc(-c3ccco3)s1)=O)C2 C12CCC(CC1)NC2=O.C(=O)(C(C)(C)C1CCC1)N(CC(=O)NC1CC1)C C1(C(C)C)CN(C(C2(C)CCCN(C(C3CN(C(N)=O)C3)=O)C2)=O)CCCO1 c1(COC)nc(Cl)cc(=NC2CN(C(C3CCCN3C=O)=O)CC3(CCC3)C2)[nH]1 O=C(C1=CCCN(C(=O)COC2CC=CC2)C1)Nc1cccc(C2CC2)c1 N#Cc1cc(I)ccc1NC(C1CC1C(=O)Nc1cc(C(F)(F)F)n[nH]1)=O Cc1[nH]c(=N)nc(O)c1CC(=O)NCC(C)CNC(=O)CC1CCC(F)(F)CC1 C1(C(C(=O)N(CC=C)CCOC)C)CCN(C(c2n[nH]cc2Cl)=O)CC1 c12ccc(C)cc1OCCc1cccc(c1)NC(=O)NC2.C(C(=O)N(C)C)NC c1(C(=O)NC2C(C=C)CN(C(C3(C)CCCCO3)=O)C2)nccn2cc(C)nc12 C1(C(=O)NC(CCC)C2CCCC2)CCN(C(=O)C(C)CC#N)C(C)(C)C1 CCCC(CC)CC(=O)N1CCCC(C)(CNC(c2cccc3scnc23)=O)C1 C#CCC(C)(C(=O)NC(c1ccc(O)cc1)C)NC(=O)C(C(C)C)SC c1(N(C)CC2CN(C(=O)OC(C)(C)C)CCC2C)ncnc(N)c1N.C(C)(C)(C)O c1(C(N(C(C(N2CC3C(C2)C3(C)C)=O)C2CC2)C)=O)cccc(F)c1F c1(C(N2CCN(C(=O)CCCn3ccnn3)C3C2C3)=O)cncc2nc[nH]c12 c1(NCC(N2C(CN(C(=O)CC3CCCOC3)CC)CCC2)=O)cc(C)nn1C c1(CNC(c2c(C)scn2)c2nnnn2-c2ccccc2)cccc(C(N)=O)c1 C1(OC)CC(NC(C2CC3(CC3)C2)=O)CN(C(c2cc(C)ccc2C2CC2)=O)C1 N1(C(COC)=O)Cc2ccccc2CC1CNC(c1nc(C)no1)=O C1(CNC(=O)NCC2CCC(C)(C)O2)CCCC(F)(F)C(=O)N1 c1(C(=O)Nc2scc(-c3c(C)cc(O)cc3)n2)cc(F)c(F)c(Br)c1F C(C)(CCC(=O)N1CCOC(CCNC(c2cnn(C3CCC3)c2)=O)C1)SC c1(-c2cn(CC3N(C(C(C4CCOCC4)SCC)=O)CC3)nn2)cncc(C)n1 c1(C(=O)NCCOCCCNC(C(C)c2cccs2)=O)ccc2c(n1)OCCO2 c1(NC(c2cc(OC)ns2)C)cc(NC2CC2C2CCC2)ncn1 N12CCCC(C1)C(=O)N(C)C1CC(C1)N(C)C2=O.C(=O)(CC1(C)CC1)NC1CC1 c1(CC)ccc(C(=O)NCC2CC(C(=O)NC3CCOCC3)C2)[nH]1 N1(C(C(CO)OC)=O)C2CCC(C(=O)NCC(C)(C)C(F)F)C1CC2 C1(C(N(CC(C)C)CC(=O)NC2CC(O)(C(=O)OC)C2)=O)COCC(C)O1 N1(C(c2cc(C(N)=O)co2)C(=O)NC)CCCN(CC#N)CC1 C(=O)(C(CC(C)C)NC(=O)C=Cc1ccco1)NC(c1ccc(C)cc1)C CC1(CNC(=O)C=CBr)CN(C(c2ncc(F)cc2N)=O)CCO1 Cc1cc(=NC(CCO)C2CCCCCC2)[nH]c(C)c1C#N CCC(C)C(=O)NC(c1ccccc1)C(=O)NCCC1(C)CCOC1 c1(N2CC(CC=C)(NC(C3CCCCC3O)=O)C2)nc2c(cc1C#N)CCC2 C#CCCCCC(=O)N(C1C2CN(C(c3ccc(CSCCC)o3)=O)CC12)C C=C(C)C1CN(C(C2CC3(CCN(C(C4CN(C)C(=O)N4)=O)C3)C2)=O)CCO1 C1(C)(C(=O)OC)CN(C(=O)CC2(NC(=O)CC3(C)CCOC3)CCC2)C1 N1(C(=O)CC2(O)CCC2)CC2(CC2C(N2CCC(n3ccnn3)C2)=O)C1 Cc1ccc(C)c(NC(C2(NC(c3cc(C)c(C)[nH]3)=O)CC2)=O)c1 C(=O)(NNc1cc(C)ccn1)c1c(CNC(c2ccccc2)=O)ccc(C)c1 C1(OCC=C)CCN(C(C2CC(CNC(=O)CCC=C(C)C)C2)=O)C1 N1(C(C(=C(C)C2CC2)F)=O)CCCCC1CCNC(C1CC(C)CCO1)=O C12(CNC(=O)CSC(F)F)CCC(CC1)N2C(=O)C(=O)Nc1ccc(Cl)cc1 C1(C)(CC(=O)NCC(C(C)(C)C)NC(=O)CCc2csc(=N)[nH]2)CCS(=O)(=O)N1 C=C(C)CCC(=O)N(C1CCCN(C(=O)C(O)CSC)C1)C C1(C(=O)NC2CC(CCNC(C(CN(C)C)N(C)C)=O)C2)CCc2nn[nH]c2C1 N1(C(C(C2CC(F)(F)C2)OC)=O)CCCN(C(c2c(C)noc2C(F)F)=O)CC1C Cc1cn(CC(N2CCC2(C)C(N2CCOC3CC23)=O)=O)c(=O)nc1O Cc1nc(C(=O)N(C2C3CN(C(c4cc(C)c(Cl)s4)=O)CC23)C)c(C)o1 C(=O)(CS(=O)c1ccc(Cl)cc1)N1CC(CNC(C(CC)CC)=O)C(O)C1 CN1C(=O)Cc2cc(S(=O)(=O)N3CCCC3C(F)F)ccc21 CCC(C)(C)CCCC(=O)NC(CO)C(=O)NC1CC2C=CC1C2 c1(CNC2CC(C)(C)OC2)cccc2c1CNCCO2 c1(NC)nc(C)ccc1C(=O)NC(C1CCCN(C(=O)CCOCC(F)F)C1)C C1(C(N(C(CC(=O)OC)C)C)=O)CCN(C(=O)CC23CCCC2C3)C12CC2 c1(C(=O)NC(CNC(C2(C#C)CCCC2)=O)(C)CO)cncc2[nH]ccc12 N1(C(C(C)(C)C)=O)CC2CCCC2(CNC(C2CC(=O)N(C(C)(C)C)C2)=O)C1 c1(C(N2CC(CN(C(=O)CC(C)(C)O)C)C3(C2)CC3)=O)[nH]nc2c1COC2(C)C C1(C(=O)Nc2cc(C)nn2C(C)C)C2CC(CC2F)N1C(=O)C(Cl)Cl C1(C(=O)NCCCC2(NC(c3cn(C)nc3)=O)CC2)CCC(C)(C)OC1 N1(C(C(C)=C2CCCC2)=O)CC2N(C(c3cccc(Cl)c3)=O)CCC2(C)C1 Cc1cccc(C(N2CCC(NC(=O)CC3CC(C(F)F)C3)C(F)C2)=O)c1Cl c1(SCC(N2CCCC(NC(C3CC4CC4C3)=O)C2)=O)ccc(F)cc1 C(CC)(CCCC(=O)Nc1ccc(F)nc1C)NC(C=CCCC)=O N1(C(C2CN(C(C)C)C2)=O)CCC2(COCC(CNC(=O)C3=CCCC3)O2)C1 Cc1cc2c(C(N3CCCN(C(C4(O)CCC4)=O)CC3C)=O)nccn2n1 c1(C(=O)N(CCCNC(C2CC(n3cnnc3)C2)=O)C2CC2)coc(C2CCC2)n1 N1(C(=O)C2COc3ccccc32)Cc2ccccc2Sc2ccccc21 N1(C(CCSCCCC)=O)C2CCCC1CC(NC(=O)CC1CCC3CC3C1)C2 S(=O)(=O)(c1cccc(C(C)(C)C)c1)N(C1(CC(F)F)CC1)C c1(CC(=O)NC2C3CN(C(C4(C#N)CCCC4)=O)C(C3)C2)ccc2c[nH]nc2c1 C1(=O)CCCC(=O)OC(C)CC(=O)NCC(C)N1C.C1(C(=O)N(C)C)CCCCC1 c1(C2CN(C(C(C3CCCC3)NC(C)=O)=O)C2)ccccn1.C12CN(C1)C(=O)N2 C1(O)(CNC(CN(C(=O)CC2CCOCC2)CCOC)=O)CCOC1C c1(C(c2nnnn2CC(F)F)NC(c2ccn(C)c2)C)cc(Br)ccc1Cl c1(OC(C(=O)Nc2ccnn2CC=Cc2ccccc2)(F)F)ccccc1F c1(C(N(C2CCN(C(C3CC3F)=O)CC2)CC(C)C)=O)nnn2c1CSCC2 c1(C(N2CC(C)C(NC(c3nc(O)nc(O)c3F)=O)C2)=O)cc(Cl)cc(Cl)c1O C1(OC)CC12CC(CS(=O)(=O)NCC(=O)NCCNC(=O)OC(C)(C)C)C2 N1(C(c2c(C)ncc(Br)c2)=O)CCCN(C(=O)C(C)CO)C(C)C1 CC(F)CC(=O)NC(C)CCN(C(=O)CN(C(=O)OC(C)(C)C)C1CC1)C c1(OC)ccc(Cl)cc1CN1CCCOC(CNC(c2ccc(Cl)cc2C)=O)C1 C1(NC(C2C(C)C2)=O)CCCC12CN(c1cc(Cl)nc(CS(C)(=O)=O)n1)C2 c1(C(N2C(C(N3CCCC3CF)=O)CC(O)C2)=O)cc([N+](=O)[O-])n[nH]1 Cc1cc([N+](=O)[O-])cnc1N(C1CCCN(C(c2cncn(C)c2=O)=O)C1)CCO C1(C(=O)Nc2nc(C3CCCC3)ns2)CCCC(Cc2ccccc2)C1.C(=O)(C1CC1)N c1(OCC(CNCCCCC(C)N(S(C)(=O)=O)CC)O)ccccc1OC CCCC(CC)C(=O)NCC(C)(CC(C)C)NC(c1ccc(C2CC2)c(F)c1)=O c1(C(=O)NC(CC=C)CNC(c2scnc2CC)=O)ccnc(-n2cccn2)c1 c1(C(C(=O)NCC(CN(C(C=CC)=O)C)O)C)ccc(C(F)F)cc1 c1(C(=O)NCCN(C(CN(CCOC)C)=O)Cc2ccccc2)ncncc1Cl c1(OC)cc(OCCNC(=O)Nc2c(Cl)cccc2Cl)ccc1Br N1(C(c2cnc(CC)s2)=O)CCOCC1CNC(=O)C(C1CCOCC1)F C1(C(N(CC(CC)NC(=O)Cc2cncc(O)c2)C)=O)CCC2(CCCCC2)C1 C(c1c(F)cccc1F)=CC(=O)NCC(CN(C(=O)CC1CCOC1)C)O N1(C(CN2CCC(C)C2)=O)C2CC=C(C(=O)NCCc3cscn3)C1CC2 CC1CON(C(=O)c2csc(-c3cccc(C(O)C(F)(F)F)c3)n2)C1 C1(COC)(CNC(=O)C(C)NC(=O)C(C)(C)OC(C)=O)CCCO1 Cc1ccc(C(C)(C)C(=O)NCC2(NC(C3CCC4CCC34)=O)CC2)cc1 N1(C(c2cc(OC)n[nH]2)=O)CC(NC(C2CNC(=O)N2C)=O)C2(CCOCC2)C1 Cn1c(C(=O)NC(C)(C)CNC(=O)CCC2CCCC(O)C2)cc2sccc12 c1(C(=O)NCC(CO)NC(C(=O)NCCOC)=O)cnc(O)n1C N1(C(c2c(OCC)oc(C3CCOCC3)n2)=O)CC2(C(=O)OCCNC)CCC1C2 N1(C(C2N(CC)CCC2)=O)CCCC12CCN(C(c1occc1Cl)=O)C2 CC(N=c1[nH]c2ccc(O)cc2s1)c1ccc(N2CCCC(C)C2)cc1 C#CCC(CC(=O)Nc1cc(CO)cc(F)c1)NC(c1ncoc1CC)=O C(=O)(CCCC(C)(C)C)N1CC(O)(CCNC(c2ccc(CC)[nH]2)=O)C1 C(=O)(C(CNC(=O)Cc1cc(C)on1)CC1CCCC1)NCC(CC)C c1(C(=O)NCC(CC)NC(C2(C)C(CC)CCC2)=O)cc(C)nnc1O C(CC(=O)N1CCC(CN(C)C)(OC)C1)(C(C)(C)C)NC(CCOC)=O C=CCC(C(=O)N1CC(O)C(O)CO1)NC(c1ncn(CC)n1)=O c1(C(N(C2CCN(C(C34CCCC3C4(F)F)=O)C2)CC)=O)ccc(C)c(Cl)c1 N1(C(CN(C)CC)=O)CCC(CO)(NC(C2CCCS2)=O)C1 Nc1cn[nH]c(=NCCCOc2cc(Cl)cc(Cl)c2)c1 N1(C(CC=C(C)C)=O)CC(NC(=O)Cc2csc(S)n2)CC(C)C1 CC(CCNC(=O)CC1CCCOC1)CCNC(c1cc(=O)n(C)o1)=O c1(C(N(CCNC(C2C(C)OCC2)=O)C)=O)ccc2c(Br)cccc2n1 c1c(F)ccnc1F.O=C1CCCN1Cc1cn(CC2CCCO2)nn1 Cc1nn(C)c(C)c1C(=O)NC1(C)CN(C(=O)COCCCF)C1 Cc1nc(C)c(C(C)NC(=O)COC2CC(NC(=O)CCC3CCC(C)O3)C2)[nH]1 C(=O)(N=c1[nH]nc(-c2ccc(C)cc2)s1)N(CCNC(C)=O)C1CC1 N1(C(c2ccc(OC)s2)=O)CCC(O)(CCNC(c2sc(C)cc2Cl)=O)CC1 c1(C(N2C(CNC(CCC(=O)N(C)C)=O)CC2)=O)cc2c(F)cc(F)cc2[nH]1 C1(CNC(C2(COC)CCCCC2)=O)CCC(C)N(C(=O)Cc2sccc2C)C1 c1(C(=O)NC2CN(C(CC(C=C)(C)O)=O)CC2C)cccc([N+](=O)[O-])c1OC N1(C(C(NOC)=O)=O)CCN(C(C23COCC2C3)=O)CC(C)C1 C1(CNC(C(COC)O)=O)CC2CCC1N2c1cc(C(C)(C)C)nc(Cl)n1 CCCC(C)(O)CC(=O)N1CCC(CNC(C2CN3CCN2CC3)=O)C(O)C1 Cc1cccc([N+](=O)[O-])c1.C1(N(CC(=O)Nc2ccc(F)cc2)C)CC2(CCN(C(C)C)C2)CO1 c1(CC)nc(-c2cc(-c3ccccc3)ccn2)nn1C1CCCOC1 C1(CC(=O)NC(c2ccccc2)CNC(=O)CCC2CC2(F)F)CCCC(=O)N1 c1(-c2ccc(CNCCCCCOC)o2)cc(CN2CCCC2)ccn1 c1(C(=O)NC2CC2NC(=O)C(O)Cc2ccc(F)cc2)cccc2ncccc12 c1(C(N2CC(COC)N(C(=O)C(C)N3CCC3)CC2)=O)c(C)cc(C)nc1S C1(C)(CNC(C2C(C=C)OCC2)=O)CCN(C(c2nocc2CC)=O)CC1 CN1CC(NC(C2CCC2CNC(=O)CN2C(=O)CCC2=O)=O)CCC1=O C1(C(C)Cn2cc(CC(=O)O)nn2)CCCN(C(=O)CN2CSCC2=O)C1 C(=O)(C1CCCc2nncn21)NCC(CC)NC(c1csc2cc(Cl)cnc12)=O C#Cc1ccc(CC(=O)NC2CC(O)CN(C(=O)CCc3ccon3)C2)cc1 c1(CCC(=O)NC(CNC(CC2C(C)CCC2)=O)C)cccc(F)c1F C1(NC(C2N(S(C)(=O)=O)CC2)=O)COC2(CCN(C(=O)COCC(F)(F)F)C2)C1 c1(C(N2CCC(CNC(c3ccc(F)cc3)=O)C23CC3)=O)ccc2c(n1)CCO2 c1(CN2CC(NC(C3CC(C)(C)C3)=O)C2)cc(C(=O)CBr)ccc1O C1(C(CNC(C(C)N(C)C)=O)(C)O)CCN(C(c2c[nH]ccc2=O)=O)CC1 Cc1cc(C(=O)NCc2ccc(CNC(C3(C#N)CC(C)C3)=O)cc2)cnc1O N1(CC)CC(C(N2CCC(NC(c3cscn3)=O)CC2)=O)CCC1=O Cc1nsc(C)c1C(=O)NCC1CC(F)(CNC(=O)CC2CCCO2)C1 C1(C(=O)NCC=CC(=O)NC(C)(C)CF)CCC2(CC2)C1 C=CCC(C(=O)NC1CC(C(F)F)(NC(=O)CC2NC(=O)NC2=O)C1)C(C)C N1(C(c2ccc(C)nc2)=O)CCCOC(CCNC(C2C3CCCCCC23)=O)C1 c1(CNC(CNC(CC)=O)=O)ncccc1CNC(c1cc(C(C)(F)F)on1)=O C(=O)(C(F)C(C)(F)F)NCCCCCN(C(C)C)C(C1CC12CCSCC2)=O N1(C(COCC(=O)Cl)=O)CCC2(CCN(C(=O)COc3cccc(Cl)c3)C2)C1 [N-]=[N+]=Nc1ccnc(NCC2CCN2)c1 c1(C(CNC(=O)CC2CNCC2O)N(C)C)ccccc1Cl C1(C(=O)NCC(C2CCC2)NC(c2cncc(C)n2)=O)CCC(F)(F)CC1 N1(C(C(c2ccc(C)cc2)C2CC2)=O)CC2CC1CN2C(=O)CC1CCOC1 C1(CNC(c2c(C(=O)OC)scc2)=O)CCN(C(=O)CC(C)F)CC1C C1(C(N2CCC(C(=O)OC)C2)=O)CC(C)(C)CCN1C(=O)C(C1CCOCC1)O Cc1cc(C(C)C)ccc1C(=O)OCC1CCN1C(=O)OC(C)(C)C C(CCCN=c1[nH]c2ncc(Cl)cc2s1)NC(c1cncc(CC)c1)=O c1(CC)ccc(C(=O)NCCCCCCNC(C2CCNC2=O)=O)cc1Br Cc1cc(C)c(OCC(=O)NC2CCC2NC(C2(C)CCNC2=O)=O)c(C)c1 C1(n2cc(CC3N(CC)CC3)nn2)CC(C(=O)OC)N(C(=O)C(CSC)OC)C1 Cc1csnc1C(=O)NCC=CCC(=O)NCC(c1ccnn1C)O C1(C(=O)NC(C=C)C2CCC2)CC=CCN1C(=O)C(COC)N(C)C C1(NC(Cn2ncc(C#C)c2)=O)CN(C(=O)CSC)C2(CCCOC2)C1 C(C(C)C)(C(O)C(=O)NCC(C)(C)CNC(c1cc(Cl)ccc1O)=O)OC c1(C(=O)NC2CC(CNC(c3cc(CCC)on3)=O)CC2O)ncc(N)cc1Cl c1(C(=O)NC2(CF)CCN(C(=O)CCNc3cncnc3)C2)cnc(Cl)c(Cl)c1 N1(C(C2N(C(c3c(C)n(C)nc3)=O)CC(=O)C2)=O)CC2CC1CS2=O C1(F)(C(=O)NC(C(CC)C)CO)CCN(C(c2cccc(C#N)c2)=O)CC1 C1(CC(=O)Nc2[nH]nc(C3CCN(C(CCC#C)=O)CC3)n2)CCOCC1(C)C O=C(C1CCCc2nccn21)NCC1(F)COCCN(C(c2cncnc2)=O)C1 c1(C(=O)NCCCCC(C)NC(=O)CC2COCCO2)ccc(Cl)c(Cl)c1N c1(OC)ccc(C2(NC(=O)C(C(C)C)N(C)C)CCOC2)cc1OC c1(C(=O)NCCN(CC(C)O)C(c2c(C)n(C)nn2)=O)cnc2n1C(C)CCC2 Cc1csc(=NCC(=O)NCC(C)(C)CNC(c2cc[nH]n2)=O)[nH]1 C(C1=NOC2COCC12)CNC(COC1CCN(C(C(CCCC)O)=O)C1)=O C1(C(=O)NCC2N(C(C(C3CC(F)(F)C3)OC)=O)CC=C2)CCCCC12CCC2 c1(CC)ccc(F)cc1C(=O)NC1CN(C(=O)C(O)CC(N)=O)CC1C(F)F C(=O)(C1CCCCc2ccccc21)NCC1(O)CN(C(Cc2cc(C)no2)=O)C1 c1(C(=O)NCC2CCN(C(C(c3ccc(F)cc3)CC)=O)C2)cccc(N)c1C C1(C(=O)NCCNC(c2cc[nH]n2)=O)CN2CCCC1C2 N1(C(C2C(=C)CC2)=O)CC2CC2(CNC(c2cncc(C(F)F)c2)=O)C1 c1(OC)ccc(CNC2CC2C(=O)NCc2cc(Br)ccc2F)c(F)c1 Cc1cc2ccc(C(=O)NC(CO)CCCCNC(=O)CCC3CC3C)cn2c1 c1(CC)oc(C(=O)NC(C)(C)CCCNC(=O)CC2CCC23CCC3)cc1C c1(C(N(C2CCNC2=O)C)=O)cc(O)ncn1.C12(CC1)CC(=O)N2C C(CCCC(=O)NC1CCC1NC(=O)C(c1cccc(CC(C)C)c1)C)OC c1(OC)cc(C(N2CCC(NC(c3ncc(F)cc3C)=O)C(C)C2)=O)cc(Cl)n1 C(C(COC)C(=O)N(C)CC1CCCC(NC(c2ccn(C)n2)=O)C1)OC c1(C(=O)NCC(C#C)CC)cccc2ccc(O)nc12 C1(NC(CSC(C)(C)C)=O)CCC(CNC(c2nc(C(F)(F)F)cs2)=O)C1 C(CCC(=O)NC(C)CNC(C1CC(F)(F)C1)=O)NC(=O)OCC N1(C(C(C)NC=O)=O)CCC(C2(C(=O)N(CC(N)=O)C3CC3)CCOCC2)CC1 N(C(=NCCC(C)=O)NCC1CC1c1cc(F)cc(F)c1)C1N(CC)CCC1 C1(NC(C(C)c2ccco2)=O)CCC(O)CN(C(=O)C=CCF)C1 N1(C(c2cc(C)nc(O)n2)=O)CC2CC1CCC2NC(=O)Cc1nncn1C CC(C)C(C(=O)NCC(C)(C)CN(C(=O)C(O)C1CCC1)C)N(C)C c1(C(C)(C)C)cncc(C(=O)NC2COCC2NC(c2c[nH]c(=N)o2)=O)c1 N1(C(C(C)OCCC(C)C)=O)CCC(NC(=O)C2=CC(C)(C)C2)C2(CCC2)C1 C(=O)(C(F)(CNC(=O)COCCCN(C)C)C(C)C)NCC(C#C)CC1CC1 N1(C(C=CC2(C)COC2)=O)CC2CC(O)C1C2NC(c1cccc(Cl)c1O)=O c1(C(N2C(CNC(C(CC=C)NC(C)=O)=O)C(C)CC2)=O)n[nH]c2ccccc12 N1(C(CC2(C)CCCN(C(C3C4CNCC34)=O)C2)=O)Cc2ccc(F)cc2C1 c1(C(=O)NC2C(CNC(c3c(OC)scc3)=O)CCC2)ccccc1C(N)=O c1(C(=O)NCCCNC(C2C3CS(=O)(=O)CC23)=O)cc(Br)c2occc2c1 c1(C(N2CCC(CC(C)NC(C(CC)SC)=O)CC2)=O)cc(N)c(Cl)cn1 n1(C(C)C(=O)N(C2CCOCC2)C)cnc2ccccc12 N1(C(C(CC(C)C)OC)=O)C2CCC1CC(CNC(c1cc(C(F)F)no1)=O)C2 C(=O)(C(CCOCCO)NC(=O)CNC(N)=O)NCC(CC)(C)Cl CC1CN(C(C2CC(F)(F)C2)=O)CCN1C(=O)C(F)(F)C1CCOCC1 N1(C(C(CNC(Cc2c(C)occ2)=O)C)=O)CCC(CO)C1(C)C CC(C)C1=NOC(C(=O)NCCCCC2CN(C(C3CC4C=CC3C4)=O)C2)C1 c1(OC(C(=O)N(c2c(OC)ccc(F)c2)C)C)ccc2c(c1)CCC2 C1(C(N(C)C(C2CC(O)CN2)=O)=O)CCN(C(c2cccc(Cl)n2)=O)CC1 C1(CNC(CC2CC(C)C2)=O)(CNC(=O)CC2OCCCO2)CCCC1 CC(C)CC(C)CC(=O)NCC(C)(C)CCNC(=O)C=CC(C)(C)SC C1(C(N(CCNC(c2n(CCOC)ncc2)=O)C2CC2)=O)CCC(C)(C)CO1 CC(C(=O)NC(C)(CNC(=O)CCOc1ccccc1)C1CCC1)P(C)(C)=O C1(NC(c2ccc(C)cc2O)=O)CC2CC1CN(C(=O)CS(=O)(=O)CC1CC1)C2 CCC(CC(=O)NCC1CN(C(c2ccsn2)=O)C(C)(C)C1)C(F)F C12(CC(N3C(CNC(c4coc(C5CC5)n4)=O)CC(O)C3)=O)CCC(CC1)CC2 C(c1cccc2ccccc12)=CC(=O)NC1CN(C(C(F)=CCC)=O)C2C1C2 c1(C(=O)NCC2(N(C(=O)Cn3cncn3)C)CC2)ccc(Cl)nc1 N1(C(C(CCC)OC)=O)CCCC(NC(c2cnn(CCN(C)C)c2C)=O)C1C C1(C(=O)NCCc2ncc(-c3ccccc3)[nH]2)CCC2CNCCN12 S(=O)(=O)(CCC(=O)NCCNC(=O)CN1CC=CC1)NC CS(=O)(=O)c1ccc(C(=O)NC2CC(CNC(C34CCC(CC3)C4)=O)C2)[nH]1 Cc1nnc2n1CC(C(=O)NC1(CNC(c3cc[nH]c(=N)n3)=O)CCCC1)C2 n1(CC)ccc(S(=O)(=O)Nc2ccc(N3CCCC4CCC34)nc2)n1 c1(C(=O)NC(CCNC(CCC=CC)=O)C)ccnc(Br)c1N C1(NC(C(c2ccc(Cl)s2)C)=O)CCC(C)(CNC(=O)C=Cc2ccoc2)C1 CCC(C(=O)N1CC(O)(C2CCCN2C(=O)C(C)OCCN(C)C)C1)N(C)C c1(OC)cc(C#N)ccc1-c1noc(-c2cc3scnc3[nH]2)n1 C1(C2CCCC2)(C(=O)NCC2N(C(c3c[nH]c(=NCC)s3)=O)CCC2)CCNC1=O C(C)(C)(CC(=O)NC1(C2CCCN2C(=O)CCN2CCCC2=O)CC1)OC N1(C(c2n(CCC)nc(C)c2)=O)CCC2(CCC(NC(=O)CCCOC)CC2)C1 N1(C(C2CC(C(F)(F)F)(OC)C2)=O)CCN(C(c2nn(C)cc2N)=O)C(C)C1 CC(C)C(CCNC(=O)C(C1CC1)N(C)C)NC(=O)CN1CC=CC1 C=Cc1ccc(NC(C2CCN(C(c3ccns3)=O)C2c2cccnc2)=O)cc1 C(C(C)(C)C(=O)NCC1CCCN1C(c1cnn(CC(F)F)n1)=O)OCC CCCCC(CNC(=O)Cc1cccnc1C)NC(=O)CC1CCCC1 CC(CC(=O)NC1C2CCCCC12)C(C)(C)NC(c1cccc2ccnn12)=O c1(-n2ccc(CC(=O)NC(C)C(CO)N(C)C)n2)ccc(F)c(F)c1 C1(O)(CC(=O)N(C(CNC(c2cncc(C)n2)=O)C)C)CCCN(C)C1 c1(C(N(C(CN(C(C2(SC)CCC2)=O)C)C)C)=O)cc(F)c(F)c(Cl)c1F C1(C#CC(=O)N2CCC(N(C(=O)CC(C)(C)O)CC3CC3)CC2)(CC)CC1 c1(CN2CCC(N(C(C3CCC(C(C)C)CC3)=O)C)C2)ccccc1[N+](=O)[O-] Cc1ccc(C=CC(N2CCN(C)CC2CNC(=O)Cn2cc(Cl)cn2)=O)cn1 c1(OCCC)ccc(CNC(C(=O)O)C(C)OC)cn1 c1(CC(N2CCN(CCNC(C(CC)COC)=O)CC2)=O)ccc(Cl)c(C)c1 C(=O)(C(=O)N=c1ccn(-c2ccc(Cl)cc2Cl)[nH]1)Nc1c(C)nsc1 C(CN=c1ncc(C(F)F)c[nH]1)N(C(=O)C1=CC2CCCC12)CC c1(NC(c2ccccc2)COC)[nH]c(=NC2CCCCCCC2)nc2scnc12 c1(C(=O)NCC2N(C(C(C)SCCCC)=O)CCC2)cc(C(F)(F)F)cnc1C N1(C(C(CC)SC)=O)C(CNC(=O)CC2CC(=O)NC2=O)CC2COCC12 c1(C(=O)NC(CNC(C2CCCN2C2CC2)=O)CO)cc(F)cc2ccncc12 C(C)(C)(C(C)CC(=O)NCCC(CO)C(C)C)NC(c1cncc(C)n1)=O n1(CC(=O)NC(C)CCCNC(c2ccon2)=O)cc(C#N)c(O)nc1=O C(CC1=CCN(C(C2CC23CC(F)(F)C3)=O)CC1)NC(C1(CC#C)CCCO1)=O C1(OC)CC2CC(NC(=O)C(C)N(C(=O)CCn3cccc3)C)CC12 C1(CCN(C(C(F)=CCC)=O)C)CCCCN1C(=O)CC1CCC(=O)N1C c1(CC(=O)NC2C(NC(CCC(C)(C)C)=O)CCC2)c[nH]c2cnccc12 C1(NC(c2scc(CC)c2)=O)CCCCC12CCN(C(c1cc(C#N)on1)=O)C2 c1(C(=O)NC2(C)CC(NC(CC3CC(=C)C3)=O)C2)noc2c1CCCC2 C1(NC(CC2CC(NC(C(C)SC)=O)C2)=O)CCc2n[nH]cc2C1 C1(C(=O)NC(CC)(C)CNC(=O)CCC)CCCCN1C(c1cc(C2CC2)on1)=O C1(C(=O)NC(C(N)=O)CO)(NC(c2ncncc2Cl)=O)CC(F)(F)C1 CCCCS(=O)(=O)CC(=O)N1CC2CC1CN2C(c1[nH]nc([N+](=O)[O-])c1Cl)=O Cc1ccccc1-c1nc(-c2cc(CC(C)C)on2)n(CCOC(C)C)n1 c1(CCC(=O)NCC(CC)NC(COC(CC)CC)=O)nc(C)c(C)[nH]1 N1(CC(=O)NC)CCN(CCCNC(c2ccc(C)cc2F)=O)C(C)C1 c1(C(=O)NC2(C)CN(C(c3c(COC)cco3)=O)C2)ncn2c1COCC2 C1(C2CCOCC2)(C(N(C2CN(C(Cc3c(C)nc[nH]3)=O)C2)C)=O)CC1(F)F C(=O)(C1CCc2ccccc21)N1C(C=CC(=O)NCC(C)(O)C2CC2)CCC1 C1(NC(C2CCCSC2)=O)CCC2(CC1)CN(C(C1CN3CCN1CC3)=O)C2 c1(CCC(=O)NC(CC=C)CNC(=O)C(C)O)cc(OC)ccc1OC Cn1nc([N+](=O)[O-])c(Cl)c1C(=O)NCC(C1CCOC1)NC(=O)C1=CCCOC1 c1(C(N2CCCC(C(=O)NC(C(=O)OCC)C)C2)=O)c(C)nc2ccc(F)cn12 CC1CCC(C)(C(N2CC(CN(C(=O)CCCC#N)C)C2)=O)C1 C1(C)(CCC)CN(C(C(=O)Nc2ccccc2OC)C2CCOC2)CCO1 c1(COC)ncc(C(=O)NC23CC(C2)N(C(c2ccc(Cl)cc2)=O)C3)cn1 N1(C(c2cc(CCC)c(C)s2)=O)CC(NC(C2CC=CCO2)=O)C(C)(C)C1 N1(C(C(CC=C)OC)=O)CCC2(CC1)CC2C(=O)NC1CCCOC1 CC(C)C(F)C(=O)NCCC1CC(NC(c2csc(Br)c2Cl)=O)C1 N1(C(Cc2c(C)non2)=O)CCN2CCN(C(=O)CCc3cscn3)CC2C1 C1(CNC(CCSCC)=O)(NC(=O)CN2CCCCC2C)CCCCC1 c1(C(N(C2CCN(C(C3C(C)C3C)=O)C2)CC)=O)cc(F)c(C)cc1Cl N1(Cc2c(C)n[nH]c2)CC(NC(=O)CC2CCC2)C(C#N)C1 C1(C(N(C2CN(C(C3(OC)CCC3)=O)C2)C)=O)CC(=O)CO1 c1(OC(C)C)nc(C(N2CC(CCNC(=O)COCP(C)(C)=O)C2)=O)cc(O)n1 c1(C(=O)NC2CN(C(Cc3c(C)con3)=O)CC2C)csc2c(F)cccc12 C1(C#CC(=O)NC2CC(O)(CNC(=O)C3=CCCCC3)C2)(CC)CC1 N1(C(C(C(=C)C)(C)C)=O)CC2CCC(C(N3CCSC(C)C3C)=O)(C2)C1 c1(C(N2CCN(C(c3ccccc3)=O)C(CO)C2)=O)cc(Cl)c(F)cc1F N1(C(=O)CC2C=CCC2)CCC2CN(C(c3cc4c(s3)CCC4)=O)C2C1 c1(NS(C)(=O)=O)ccc(CCNC2CCCC(N3CCCC3)C2)cc1 N1(C(c2nc(COCC)sc2)=O)CC(C)CN(C(=O)C2=CCOC2)CC1C C(=O)(C(CC)C(=O)NCCC(C)NC(=O)C(C)(C)c1cscc1Cl)OCC C=C1CC(C(=O)N(C)CCN(C(C)C)CC)(CNC(C2CNC(=O)C2)=O)C1 C1(C(=O)NCCC2(C)CCN(C(COCCC)=O)C2)CC2CCC(C1)O2 Cc1cnc(C(=O)NCC(C2CC2)NC(c2ccc[n+]([O-])c2)=O)c(Br)c1 c1(C(N2C(C(=O)NCC(=O)N(C)C)CC(OC)C2)=O)ccc(C)c(C)c1I n1(C(C)C)ccc2cc(C(=O)N(C3CCN(C(C)C)CC3)CCCO)ccc12 C(=O)(CS(=O)c1ccc(Cl)cc1)N1CC2(C(NC(CCCC#CC)=O)CC2)C1 Cc1cccc(-c2cc(C(=O)NCC(C)(C)CNC(=O)C(C3CC3)N(C)C)on2)c1 C12(C(=O)NCCCCCNC(C(C)O)=O)CC3(F)CC(F)(C1)CC(F)(C2)C3 c1(CC(N2CCC(C)C2CNC(=O)CNC=O)=O)csc2ccc(Cl)cc12 CC1(C)OCCOC1C(=O)NCC1CCCCN1C(=O)C(c1ccc(Cl)cc1)=O C1(NC(C(C)=C2CCCC2)=O)C=CCN(C(C2CC(=O)N(C(C)(C)C)C2)=O)C1 c1(C(=O)NCCOC2CN(C(COC(C)(C)C)=O)C2)c[nH]ccc1=O N1(C(C(CCCCC)O)=O)CCOC2CN(C(C3CCC4(CCCC4)C3)=O)CC12 C(C(C)CC(C)C)N(C1CCCCC1)CCCCCC c1(C(N2CC(C(C)NC(=O)CC3(C)CC3)OCC2)=O)ccc2n[nH]cc2c1Cl c1(OC)ccccc1NC(=O)C(C)N(C1CCN(CC2CC(O)C2)CC1)C C1(CC(=O)NCCN(C(c2cnn(CCF)c2)=O)CC)CN2CCN1CC2 N1(C(C2(OC)CCN(C(CC(CCC)C)=O)C2)=O)CCCCCCC1C C(C)(C(CCc1ccccc1)N(C(=O)CCCCC1CC1)C)NC(C=NOC)=O C1(C(N2CC(CCNC(=O)C(C)n3ccnc3)(OC)C2)=O)(CO)CCCCO1 C1(NC(c2c(COC)ncs2)=O)CC(CO)N(C(c2scnc2Cl)=O)C1 c1(OC)ccccc1C(C)C(=O)NCC1CC(NC(=O)C(=O)NC2CC2)CC1O Cc1c(CNC(C2C3CC3CN2C(=O)CC(O)CN(C)C)=O)nnn1C N1(C(COc2ccn(C)n2)=O)CCC(NC(C2CS(=O)(=O)C2)=O)CC(O)C1 C1(C(=O)NCC(C)(C2CC2)NC(C2CN(C(N(C)C)=O)C2)=O)CCOC1=O c1(NC(CC)C(C)C)cc(N(C)CCN(c2ccc(=N)[nH]c2)C)ncn1 CC1CCCCC1C(=O)N(CC(O)CN(C(=O)CNS(C)(=O)=O)C)C CC1CCN(C(=O)C(=O)N(C)C)CCN1C(c1cncc(O)c1Cl)=O c1(C(N(C2CCN(C(C=CCCC)=O)C2)CC)=O)ccc(=O)n(O)c1 N1(C(CCC#C)=O)CCC2(CC2NC(=O)CCNC(c2ccccc2)=O)C1 N1(C(C(c2n(C)ncc2)O)=O)CC2=C(C1)CN(C(c1ncc3ccccn13)=O)C2 C1(C(N2CC(C(C)NC(=O)C(F)(F)C3(O)CCCC3)C2)=O)(COC)CCCO1 C1(CC)CN(C(C2(NC(c3cc(C(C)=O)c[nH]3)=O)CCC(C)(C)C2)=O)CCCO1 c1(OC)c(Cl)cc(C(=O)NC2CCCN(C(=O)CN3CC=CC3)C2)nc1Cl C1(NC(C(C)OCC)=O)(CF)CN(C(=O)COCC2CCC2)C1 c1(CC(=O)NCCNC(C2(C)CC=CCO2)=O)ccc([N+](=O)[O-])cc1Cl C1(CNC(COCCCC)=O)C(C2CC2)CCN1C(c1cc(Cl)ccc1C)=O c1(C(N2CCC(N(C(CC=C=C)=O)CCO)C2)=O)cccc(N2CCOCC2)n1 C#CCCCC(C(=O)NC(C)(C)CC)N1CCC(OCCN(C)C)C1 c1(CNC(c2ccc(OC)cc2)CC)ccc2c(c1)CCCN2C N1(C(=O)CCc2ccc[nH]2)CC2CCCC2(C(N2CC(F)(C3CC3)C2)=O)C1 Cc1nc(NC2CCCc3sccc32)c(Cl)cc1C#N.C(=O)(C(F)(F)F)N1CCC(=O)OCC1=O N(C1CCc2cccnc21)C(C(CC(C)(C)C)NC(=O)Cc1cc[nH]c1)=O C1(NC(=O)CN2C(=O)CCC2=O)CCCCN(C(c2cocn2)=O)C1 c1(CN(CCNC(c2c(CC)ncs2)=O)CC2CC2)cccc(OC)c1 C1(O)(CNC(C(C)Oc2ccccc2)=O)CCCN(C(=O)CNC(N)=O)C1 N1(C(c2cc(C)sc2C)=O)CC(C2CC2)(C(=O)NCCc2ccncc2)C1 C(=O)(CC(F)(F)C(F)(F)F)NCC1N(C)CCN(C(C(COC)C)=O)C1 c1(CNC(C2CCCCN2Cc2c(F)cccc2F)=O)c(F)c(F)cc(F)c1F C(=O)(C(CCC1CC=CCC1)N1CCN(c2ccc(OC)nn2)CC1)NCC=C C1(N(CCCC)C(=O)CC2CC2(C)C)CCN(C(=O)Cn2ccnc2C)CC1 c1(CC(=O)NC2C(CNC(CCSCCCC)=O)CC2)c[nH]c2ccc(F)cc12 C=CC(CC)CC(=O)N1CCCC(CC(N2CC(OC(=O)N(C)C)C2)=O)CC1 C1(NC(c2c(COC)cco2)=O)COCCN(C(C2C(Cl)(Cl)C23CC3)=O)C1 C1(NC(COCCC#C)=O)CC2CC(C1)N(C(=O)C=CC(c1ccccc1)=O)C2 c1(C(=O)NC2CN(C(C=CC(=O)OCC)=O)CC2O)cc2scc(Cl)c2[nH]1 c1(C(C(=O)NCC(CO)NC(c2c(CC)con2)=O)O)ccc(F)c(Cl)c1F C1(C(c2n(C)nnn2)Nc2ccc(SCCO)cc2C(N)=O)CCC2(C1)CC2(F)F c1(Cn2c(-c3c(C)occ3)nnc2N2CCOCC2)cc(SC2CC2)cc(F)c1 C1(NC(C2(OC)CCSCC2)=O)CCN(C(C2CC3CC3C2)=O)CC1(C)C CC(C)S(=O)(=O)CC(=O)NC1CC1c1cn(-c2cncc(C(=O)O)c2)nn1 CN(C1CCc2c(F)cccc21)C(=O)CC1CCCC1(F)F C1(n2c(-c3scc(-c4c(C)nn(C)c4)c3)ncc2)CC(C)(C)CCC1=O C=C(C)CC(C(=O)NC1CS(=O)(=O)CC1NC(c1sc(C)nc1C)=O)OC CC(C)C(F)(CNC(C1C2CC(=O)CC12)=O)C(=O)NC(C)Cc1cccnc1 c1(C(N2CC(C)(C)C(NC(C3CC(C#N)C3)=O)C2)=O)cc2cc(Br)cn2cn1 C1(NC(C(C)SC)=O)CN(C(c2c(C)nc(C)n2O)=O)CC2(CCC2)C1 C1(C(=O)NC(C)CCCNC(C2(c3cc[nH]c3)CC2)=O)CCCN(CC(F)F)C1 c1(N2CCN(CN3C=C(OCC)N=CC3)C(C#N)C2)ncnc2ncc(Br)cc12 C(=O)(C1=CCSC1)NC1CC(C)(C(=O)NCC(C#C)OC)C1 N1(C(C(CSc2ccccc2)NS(CCCC)(=O)=O)=O)CCc2cc(N)ccc2C1 C1(O)(CCNC(c2cc(C)oc2)=O)CCCN(C(c2cncc(O)c2)=O)C1 CCC1CC(=O)O1.C1(C2CCCC2)CCCO1.CC(C)(C)OC(=O)NCC1CCC1 C1(N)CCC(n2nnnc2C(COC)(C2CC2)NCC2(CC(C)C)CC2)C1.CO C1(NC(CC(C)(C)F)=O)CCC(C)(NC(=O)CCc2ccccc2O)CC1 CCCC(CCC)CC(=O)N1CCC(NC(=O)CCN2CCCS2(=O)=O)C1 c1(OC)cc(C(=O)Nc2cnc(Cl)c(C(F)F)c2)c(-c2cncn2C)cn1 N1(C(c2cnn(CC)c2Cl)=O)CC(NC(C2CC(C(N)=O)C2)=O)CC(F)C1 C1(CC)CN(C(=O)Cn2cc(CCCOC(C)=O)nn2)CC(C)S1(=O)=O N(C1CCc2cc(CNC(n3ccc4ccccc34)=O)ccc21)C(=O)CC1CC1 N1(C(C(COC(C)C)NC(C(CSC)(C)C)=O)=O)CCCN(C)CC1C c1(C(=O)NCC(C)NC(=O)CS(C)(=O)=O)nnn(C2CC2)c1C(F)(F)F C1(CNC(C(C)SC)=O)CCCN(C(=O)C=Cc2ccsc2C(F)(F)F)C1 C(=O)(CCCC(O)c1ccccc1)NCC1CCN1C(C1CCOC(=O)N1)=O C(=O)(CCC(C)(C)C#N)NC1C(=O)NCC1(C)C.C12CC(C1)C(=O)N2C C(C(C)CC(=O)N1CCC(OCCNC(c2n[nH]c(C3CC3)n2)=O)C1)OC c1(NC(CCN(C)Cc2ccncc2)=O)cc(C#N)ccc1F c1(CCCC)ccc(C(=O)N(C2CN(C(=O)CSC3CC3)C2)C)cc1 c1(C(=O)NCc2cc(C(N3CCC(O)(CC)C3)=O)ncc2)ccc(C)c(O)n1 C(=O)(C1CCCn2c(C)nnc21)NCC1(F)CN(C(c2nn(CC)nc2C)=O)C1 CC12CN(C(=O)CN3CCOC3=O)C(C(=O)NC3(C(=O)C4CC4)CC3)(C1)C2 c1(C(=O)NC(C)CC(=O)NCCC2CCCC2)cc([N+](=O)[O-])c[nH]1 N1(C(=O)OC2N(C)CCN(C(=O)OC(C)(C)C)C2)CCC(C)(O)C(C)(O)C1 N1(C(C(CSC)O)=O)CCCCC1C1(NC(c2cccc(F)n2)=O)CC1 Cc1ccc(SCC(=O)NCC(C)(CO)NC(C2CC3(CC3)C2)=O)c(C)c1 N1(C(c2cnnc(Cl)c2)=O)CCCC(C2CCN(C(c3cc(Cl)on3)=O)C2)C1 C1(NC(c2csnc2C2CC2)=O)CN(C(=O)CC2=CCCCC2)CC2(CC2)C1 C(=O)(C(C)(C)C(C)(F)F)NCC(C)(C)OCC(=O)NC(COCC)C(C)C C1(NC(c2cc(C)c(Br)o2)=O)C2CC1CN(C(C1CCSCC1)=O)C2 c1(C(=O)OC)csc(C(N2CC(C)C(F)C2)C(=O)NCCCSC)c1Cl Cc1ccccc1CC(C)C(=O)NCC#CCNC(C1(C(=O)NC2CC2)CC1)=O C1(NC(C(C(C)C)NC(C)=O)=O)CCN(C(=O)Cc2cc(C)cc(C)c2)C(C)C1 C1(NC(c2nc(COC)sc2)=O)CC2CN(C(=O)C(F)(F)C3(O)CCC3)CC12 CCCC(CNC(=O)CCc1csnn1)NC(C1CCN1C)=O C(=O)(CCC(=O)OC)N(CCNC(C1(COC)C=CCC1)=O)C(C)C Cc1ncc(CNC(=O)C(C)CN(C(=O)C(=C2CCCCC2)F)C)o1 c1(OC)cc(NCC2CCCCC2NC(=O)C(F)CC2CCCCC2)ncn1 N1(C(CC2CCCC(NC(C=CC(CC)C)=O)C2)=O)CCCC2(CCC2)C1 C1(C(=O)NCC(c2ccccc2F)NC(=O)CCC2CC2)CCCCCC1 C1(NC(c2ccc(OC)s2)=O)CC(NC(=O)C=CSC)C12CCC2 Nc1c(C(=O)NCCC2CCN(C(=O)C=Cc3cnc[nH]3)C2)ccnc1Br C12(NC(c3ccccc3)C3(NC(C4C(C)(C(C)C)C4)=O)CC3)CC(F)(C1)C2 c1(C(N2CC(CCC)N(C(c3nnn(C)n3)=O)CC2)=O)ccc2snnc2c1 CCC(C)CCCCC(=O)NCC1CCC2(CN(C(c3c(Cl)cnn3C)=O)C2)O1 C=CC1CCN(C(=O)CC2CC(F)CN2C(=O)C(COC(C)C)N(C)C)C1 C=CCCCCC(=O)N(CC(CC)NC(=O)COc1ccccc1C(C)C)C C1(C(=O)NC(CC(=O)OC)c2ccccc2)CSCCN1Cc1cccc(C)c1 C1(C(=O)NC2CC(NC(c3cc(=N)[nH]cc3Br)=O)C2)CS(=O)(=O)CC(=O)N1 N1(C(c2cnc(C(C)C)s2)=O)CCC(C)(C)C(NC(C2(F)CCCCC2)=O)C1 CC(C)CC(C(=O)N(C(C)C(=O)NOC1CCCCC1)C1CC1)C(N)=O n1(C(C)C)ncc(Br)c1Cn1nnn(C2CCCC(C(C)C)C2)c1=O C#Cc1ccc(Br)c(C(=O)NCC(C)NC(C2CCN(C)S2(=O)=O)=O)c1 C1(N(C(C(C(C)C)O)=O)C)CC2CCC(C1)N2C(c1ncccc1F)=O C(=O)(N=c1cc[nH]cc1F)C1CCCC(NC(c2cccc(O)c2O)=O)C1 N1(C(CC(C)C(F)F)=O)CC(CNC(c2cn3c(n2)CCC3)=O)CC12CCC2 N1(C(C(CC)(C)C)=O)CC2CCOCC2(NC(c2cc(CO)ccc2OC)=O)C1 CCCC(C)(O)CNC(C1(CCNC(=O)Cc2coc(C)n2)CCC1)=O c1(C(=O)NCC2CC(OC)CN2C(c2sc(C)nc2C)=O)ncc(C#N)cc1Cl c1(C(N2CC(C(C)NC(C3CS(=O)(=O)C3)=O)OCC2)=O)ccc2nc[nH]c2n1 N1(C(CC2CC(C)(C)C2)=O)CCCC(C)(CNC(C2CC23CCCC3)=O)C1 c1(C(N2CC(NC(CC(C)n3cccn3)=O)CC2(C)C)=O)ccc2occc2c1 c1(C(=O)NC2CC(CCNC(C3(COC)CC=CCC3)=O)C2)c(N)sc(C)c1C NC(=O)CCCCC(=O)NC1CCC(C(=O)NCCCNC(=O)C2CC2)CC1 N1(C(C=CC(C)(C)SC)=O)CCC2C(NC(=O)CC3CN(C)C3)C2C1 S(=O)(=O)(c1c[nH]ccc1=NCCC1CCCO1)NC1C(c2cn(C)nc2)C1 Cc1cnc(C(N2CC(C(=O)NCC(F)Cl)C(C)C2)=O)c[n+]1[O-] c1(C(=O)NC23C(CN(C(C(C)Oc4ccc(Cl)cc4)=O)C2)C3)cnc2n1CCC2 C#CCC(C(=O)NC1CC1CC(C)C)NC(=O)CCc1cscn1 C1(C)(NC(C2(O)CC(CNC(CC(C)N3CCCC3=O)=O)C2)=O)CCSCC1 CN1CCCC12CCN(C(=O)C1=C(F)CN(C(=O)CCn3cccc3)CC1)C2 C(=O)(C1=NOC(C)(C)C1)NCC1CC(C)N(C(c2ccsc2Cl)=O)C1 n1(CC(=O)NC2C(NC(C3(C)CCC3)=O)CCC2)cc([N+](=O)[O-])cn1 N1(C(c2cn(C)nc2)=O)CCC(NC(=O)CCc2cc(Cl)cs2)C12CCCC2 c1(C(N2CCC(O)(CN(C(CSC)=O)C)C2)=O)ccc2cnccc2n1 C(=O)(CCCCCS(N)(=O)=O)N(C)CC1(O)CN(C(C2CC2(Cl)Cl)=O)C1 CC(C)CCCCCN=c1[nH]c(=NCCn2cccnc2=O)[nH]c2ccccc12 C=C(F)C1(CC(=O)N(CCNC(=O)C(C2CCC(C)CC2)CC)C2CC2)CCC1 CC(c1cnn(C)c1)=CC(=O)NCC1CC2(CC2)CN1C(C1CCCS1(=O)=O)=O N1(C(C(CC)OC2CCCC2)=O)CCCC2C1CCN2C(=O)C1=CC(C)(C)C1 C1(C(N(CCCNC(=O)CCc2ccco2)C)=O)CCCN(S(C)(=O)=O)C1 C1(NC(C2CCC(C)O2)=O)COC2(C1)CN(C(c1cc(Cl)on1)=O)C2 C(=O)(C(O)C(F)(F)F)N1CC2C(C(=O)NCC3(C#N)CCCC3)(C2)C1 c1(C(=O)NC2(CC=C)CCN(C(=O)COCC(C)C)C2)cncc2cccnc12 CC(C)(C)CC(O)C(=O)NCC1(F)CC(NC(=O)CC2CCCC2(F)F)C1 C1(=O)C(CC(C)C)n2cc(nn2)C2CN1CCO2.c1(CC)onc(C)c1CO CC1CN(C(C2(CC(F)F)CCC2)=O)CC(C)C1NC(c1cc2sccc2s1)=O Nc1ccc(-c2noc(-c3cnc(-c4cccs4)o3)n2)c(Br)c1F c1(C(=O)NCC(CNC(CCn2c(C)nc(C)n2)=O)O)cnn2c1OCC(C)C2 CCC(C)(C)CCCC(=O)NCC(Cc1ccccc1)CO N1(C(CCNC(c2ccc(F)cc2)=O)=O)CC2CC(O)CC(C2)C1 C(CCC(C)CC(=O)Nc1ccc(NC(=O)CCS(C)(=O)=O)cn1)=C(C)C C(=O)(CCC(CF)CF)N1CCCCC(NC(c2n(CCOC)ncc2)=O)C1 c1(C(N2CCC(O)C(CC(C)C)C2)C(=O)NCCCC)ccc2cccnc2c1 C1(NC(C2(NC(C(C(C)C)C3CCC3)=O)CC(F)C2)=O)CCC(C2CC2)C1 C(N(C)N1CCN(S(C)(=O)=O)C2(CCCC2)C1)c1ccc(SC)cc1 C(CC(C)C)(C(C(=O)NC1CCC1)N(C1CC1)C(c1nc(C)no1)C)OC CCCC(C(O)C(=O)NCCN(C(C)C)C(C)C)NC(=O)C(F)OC(F)(F)F C=CCC(C)(C)C(=O)NC(C1CCCN(C(c2conc2C)=O)C1)C c1(C(CC2(OC)CCC2)=O)ccc(S(=O)(=O)Nc2ccn3nccc3n2)cn1 c1(C(=O)NC(C2(O)CN(C(c3c(C)nsc3N)=O)C2)C)csc2cc(Cl)cnc12 C1(N(c2cnn(C)c2)CC)CCCN(C(=O)C(N)=O)CC1 c1(CN2C(CNC(=O)Cc3ccc(F)cc3C(F)F)CC2)n[nH]c2c1COCC2 C1(C(=O)OC)CC2(CCCC2)CN1C(c1cc(Cl)cc([N+](=O)[O-])c1)=O C12(CNC(c3ccc[nH]3)=O)CC(C1)C(NC(C1CCCC(F)(F)C1)=O)CO2 CCC(N=c1[nH]c(N2CCC(C)C(F)(F)C2)nc2c1CCC2)c1cccc(Cl)c1 CN1CCC(=CC(=O)NCCC(O)CNC(c2ccccc2CO)=O)CC1 c1(C(=O)NCCC2N(C(C3CC(CC)C3)=O)CC(F)(F)C2)ccc2sncc2c1 N1(C(C2(OC(C)C)CCC2)=O)CC(NC(c2scnc2Cl)=O)CC(O)C1 c1(CC2NCCN(c3nc(=N)[nH][nH]3)C2)ccc(F)cc1[N+](=O)[O-] c1(C(N2CC(CNC(C=C(C)c3cccs3)=O)C(C)C2)=O)c(C)ccc(C)c1O CC1=NS(=O)(=O)NC=C1C(=O)N(C(C)CNC(c1c(C)cc(F)cc1C)=O)C CCC(C(=O)N(CCNC(c1c[nH]nc1C(F)F)=O)C(C)C)OC C1(CNC(CC=CCC)=O)CC(C(=O)NCc2cnc(C)s2)=NO1 C(CC(C)C)(C(=O)N(CCOCC(=O)NCC(C)(C)C)CCN(C)C)OC C1(C(N2C(CNC(c3ccc(C(F)(F)F)o3)=O)CC2)=O)Cc2ccccc2O1 c1(N2CCCC(NC(c3cscc3Cl)=O)CC2)ncnc2cccc(F)c12 NC1CCC(CC(N2CCC2C(=O)NCCOc2ccccc2)=O)CC1 c1(N2CC(CN(C(C=C(C)c3cccs3)=O)C)OCC2)cc(C)nc(C(C)C)n1 CC(=O)n1cc(CN2CCSC(C(=O)Nc3nnc(C)n3C)C2)c2cccnc12 n1(CC(=O)NCC2(c3ccccc3)CC2)nc(C(=O)O)c2ccccc2c1=O N1(C(CN2CCC(OC)C2)=O)CCOC(C)(CNC(c2ncc(C)cc2F)=O)C1 Cc1ccnc(-n2cc(C3CC(NC(C45CC(I)(C4)C5)=O)C3)nn2)n1 c1(C(=O)NC(C(=O)NCC(=C)CC)COC)cncc(F)c1C CC1(C)C(CNC(C23CCC(C2)C3)=O)CCN1C(c1cc(O)cc(F)c1)=O C(=O)(C(C)(C)CC(=O)N1CCOCC1CC(=O)NCCCCCCO)OC C1(CC(=O)NC2CN(C(C=C(CCC)C)=O)CC2(C)C)Cn2ccnc2NC1=O Cc1ncnc(O)c1C(=O)NCC1CC(C)(C)CN1C(c1ccoc1)=O C1(C(=O)NCC2(CO)N(C(c3cc(CC)no3)=O)CC2)CC(=O)N(C(C)C)C1 N1(C(C2C=CC2C=O)=O)CC(C)(OCC(=O)NOC2COCC2O)C1.CO N1(C(C=CC(CC)=CC)=O)CCCC2(CCCCC2NC(=O)CC(C)C)C1 C1(C(=O)NC2CC2c2ccsc2)CCc2ccccc2C1=O O=C(C1=C(Cl)CCCC1)NCC1(CNC(=O)C2CC2)CCCCC1 CCC(CC)CC(=O)NCCCOCCNC(=O)C(C)C(C)c1ccc(Cl)cc1 C(=O)(CC(F)(F)CC)N1C(CCNC(C=CC(CC)=CC)=O)CSCC1 N1(C(C23CC(C(=O)OC)(C2)C3)=O)CC2CC1CCC2NC(C1(Br)CC1)=O CC(CCC(=O)N(CCO)C1CCC1)NC(=O)Cn1cnnc1O CC(CS(C)=O)C(=O)N(C)CCNC(C1(CCF)CCOCC1)=O Cc1cc(C(=O)NCc2nc(CO)cs2)c(O)cc1F.c1(C(=O)N)cc(CO)c(C)o1 N1(C(C=CC)=O)CC=C(C(C)(C)C(=O)N2CC(CSC)C2)C1 CC12CCC(n3cc(COC4CCCNC4)nn3)(CO1)C2 C(CN=c1cc(Cl)nc(CS(C)(=O)=O)[nH]1)(C1CC1)NC(CC1C(C)(C)CCO1)=O N1(C(C2CCN(C(C)=O)C2)=O)CC2CC(C1)C2NC(=O)C(C(C)C)n1cnnn1 c1(C(=O)NC(C)C(C)(C)NC(=O)C(C)C(C)(F)F)ccc([N+](=O)[O-])c(Cl)c1 c1(OC)cc(C(=O)NC(C)CCNC(=O)C(C2CCCCC2)O)cc(N)c1O N1(C(c2scc(COC)c2)=O)CCC(NC(=O)CCCSC)C(F)(F)CC1 N1(C(CC2C(C)C2(F)F)=O)C2CCC1CC(CNC(c1nnc(S)n1C)=O)C2 C1(C(=O)NCC2C(C)CCN(C(C(C(CC)C)OC)=O)C2)CN2CCN1C(C)C2 C1(C(=O)NCc2nn(CC)nc2C)CCN(C(c2ncnn2CC)=O)C(C)(C)C1 C1(NC(CSC)=O)CCCC1(C)NC(=O)CCCn1nc(C)nc1C c1(-c2nnc(CNC(=O)NC(c3nc[nH]n3)CC)s2)ccccc1F n1(C(C)C)cc(CNC(=O)CC2CC(NC(=O)C(=O)C3CCCC3)C2)cn1 C1(CNC(C(CCC)(C)O)=O)CN(C(C2CC(=O)N(CC)C2)=O)CCC12CCC2 C1(C(=O)Nc2cn(CC(=O)OC)nc2)CC(NC(=O)CC(F)(F)F)CCO1 N1(C(C=Cc2ccc(C)s2)=O)CC2CCN(C(C3CC3c3ccnn3C)=O)CC12 N1(C(c2cc(C)n(CCO)n2)=O)CCN(C(c2ccsc2)=O)CC1CS(C)(=O)=O C1(F)(CNC2CC(NC(c3cnc(SC(C)(C)C)[nH]3)=O)C2)CCCOC1 Cc1nn(C)cc1C(=O)NC1CC(C)N(C(=O)CCc2c(C)noc2Cl)C1 N1(C(CN(C(COC)=O)C)=O)CC(C)C(C)(CNC(=O)CC2CCOC2)C1 CCCCC(C)C(=O)N1CC(C(=O)NCC(C)COCC)C2(CC2)C1 N12CCC(CC1)C2=O.C1(NC(=O)NCCOC)CCN(Cc2ccccc2)C1=O CC1CN(C(=O)C(O)C(C)(C)C)CCCN1C(C1CCN(C(=O)C2CC2)CC1)=O Cn1cc(NC(=O)CC2(NC(c3cccc4c[nH]nc34)=O)CC2)c(O)nc1=O C(=O)(C(CCC(C)C)NC(=O)C(F)C1CCC1)NCc1cccc(CC)c1 C1(O)(CCNC(=O)COc2ccccc2)CCCN(C(c2cccc(=O)o2)=O)C1 N1(C(C2(CC#C)CCCC2)=O)CCCC(CNC(c2cc(C(F)(F)F)cs2)=O)C1 C1(C)(CN(C2(C3CCCO3)CCC2)C(C)=O)COCCN(C(C2CCOCC2)=O)C1 C1(CNC(C=CSC)=O)CCCC2(CN(C(c3n[nH]c4c(C)cccc34)=O)C2)O1 N1(C(C2(C)CCCN2Cc2ccc(I)cc2O)=O)CCC2(CC1)CC2 c1(-c2cnc(-c3c(C)ccs3)s2)cc(C)c(N)cn1.C1(C=O)C2CC1NC2 CC1(CNC(c2cccc(C3CCC3)c2)=O)CCCN1C(=O)Cc1ccsc1Cl c1(NC(C2N(C(c3c(CC)ncs3)=O)CCC2O)=O)ccc(Br)cc1I c1(C(N(CCCNC(CN(C(C)C)C)=O)C)=O)cc([N+](=O)[O-])ccc1OC(F)F N1(C(C(C)Cc2ccnn2C)=O)CCCCC(NC(c2c(O)cccc2Cl)=O)C1 c1(C(=O)NC(C2CC(C)(C)C2)C(=O)OC)cc(-c2cccc(F)c2)n(C)n1 CCC(C)(CC)C(=O)N(CC(C)NC(=O)C(C)(C)Oc1ccc(Cl)cc1)C N1(C(C(c2ccc(OCCO)cc2)NC(CNC(C)=O)=O)=O)CCCC2OCCC12 C1(C)(C(C)C)C=CCN1CC(=O)Nc1ccc(F)cc1 c1(CNC(=O)C=CC2CC2)ccc2c(c1)CCC2NC(=O)C1CCc2c[nH]nc21 c1(OC)ccccc1-c1ncsc1C(C(=O)Nc1nc(C(F)(F)F)nn1C)OC C(CCCCCNC(C1CC1C(C)(C)C)=O)N(C)C(C1(CF)COC1)=O N1(C(c2c(C)snn2)=O)CCC(C)(C)C(C(=O)NC(C)(CO)CCF)C1 c1(C(=O)NC2CC(NC(CC(c3ccc(C#N)cc3)C)=O)C2)ncnc(O)c1F c1(C(=O)NC)cccc(C(N2CC=CC(NC(=O)C3=COCC3)C2)=O)c1 C1(CC(N2CC(C)C(CCNC(C3(O)CCOC3)=O)C2)=O)CCC2(CC1)CC2 N1(C(C(CCC)C)=O)CCC(CNC(C2CC2C(F)(F)F)=O)C12CCC2 [N-]=[N+]=NCCCCCCC(=O)NC1CC2CN(C(=O)CCN3CCC(F)C3)CC12 CC(C)C(F)C(=O)N1CCOCC1CN(C)C(C1CN(C)CCO1)=O Cc1cc(Br)cc2cc(CN3CCC(C)(C(=O)O)C3C)[nH]c12 C1(C(=O)NCCN(C(=O)CCC2CCCN2C)CCOC)(CF)CC2(CCC2)C1 Cc1ncn(C)c(=O)c1C(=O)NCCC(C)CCNC(c1cc(O)cs1)=O N1(C(c2c(C)scn2)=O)CCC(O)(CCNC(=O)CCC2CCCN(C)C2)C1 C1(N(C(c2c(C)onc2)=O)CCO)CCCN(C(=O)CCC2CCN(C)CC2)C1 N1(C(CC2C(C)CCC2)=O)CC2CCN(C(C3CN4CCCN3CC4)=O)CC2C1 c1(-c2scc(CC(=O)NC(C3CN(C(C=CSC)=O)C3)C)n2)ccc(F)c(F)c1 Cc1ccncc1NC(N1CCN(C(=O)C(O)CN2CCCC2)CC1)=O C1(CNC(CNC=O)=O)CCC2CN(C(c3ccc(O)cc3Cl)=O)CCC2C1 n1(CC(=O)NC2CC3CCC2(CNC(=O)CCCC(F)F)C3)cc(F)ccc1=O N1(C(c2cc(CC(=O)OC)on2)C(=O)NCC)CCN(C)C(c2ccccc2)C1 C1(C(N2CCN(S(C)(=O)=O)CC2)=O)CN(C(=O)Sc2ccncc2)CC(F)(F)C1 c1(N(C)C)ncccc1CNC(N1CCCC1c1ccc(Cl)cc1)=O CC(C)CC(Cc1ccccc1)C(=O)NCC1CC(NC(=O)C(C)C(C)(F)F)C1 c1(C(N2C(CCC(=O)NCc3cccc(F)c3)CCC2)=O)ccnc(CO)c1 C12(CNC(C3CC34CC4)=O)CC(CO1)N(C(c1cncc(Cl)n1)=O)C2 C1(NC(c2cnn(C)c2N)=O)CC2(C1)CN(C(C1CCC1C(C)(C)C)=O)C2 C1(O)(CC(=O)N(CC(CC)NC(=O)CN(CC)CC)CC)CCCN(C)C1 CC(C)CC(C(=O)N(C1CCCC(O)C1)C)NC(=O)COCCF C1(C(N(C2CC(NC(=O)CC3CCCC3)C2)C)=O)CN(S(=O)(=O)N(C)C)CCO1 C1(CNC(c2cncc(C(F)F)c2)=O)C2CN(C(=O)COC3CCCOC3)CC12 C(=O)(CC(C)(C)CC)Nc1ccc(CC)nc1.C12CCOCC1Cc1cn2nn1 N1(C(C(C)SC)=O)CC(C)CCC1CNC(C1(C2CC2)CC1)=O CCCCS(=O)(=O)CC(=O)NCC(C)NC(=O)Cc1ccc(OC)cc1OC C1(C(=O)NCC=Cc2ccc[nH]2)CCCC1CNC(=O)C(F)(F)C1CC1 CCCC(F)C(=O)N(CC(C)C(=O)N(C)CCN(C)C)C C(C)(CNC(C1CCOC1C1CC1)=O)(CC(C)C)NC(c1c(SC)csc1)=O C(CCNC(c1cccc(=O)o1)=O)(C(=O)NCC1COCCO1)OC c1(C(=O)NCC(CNC(c2ccc(CC)s2)=O)F)cc(C)nc2c1CCCC2 C=CCCC(C)(C)C(=O)NCc1nc(C(=O)NC(CN2CCCC2)CC)co1 C(=O)(C(F)C(=O)NCCCC1CCCCN1C(c1c[nH]c(Br)c1)=O)OCC C(CN(C)C)(CCO)NC(CN(C(=O)CCC1(C)N=N1)C(C)C)=O c1(C(N(CCNC(C(COC)O)=O)C(C)C)=O)cnn(-c2ccc(F)cc2)c1C c1(C(N2CCN(C(c3cc(C)c(C)[nH]3)=O)C(C)C2)=O)nn2cccnc2c1Cl c1(C(C(=O)NC2(CN(C)C(C3CC34CC4)=O)CC2)C)ccc(Cl)c(Cl)c1 c1(N2CCCC(CNC(c3cc(F)cc(F)c3)=O)CC2)ncnc2c1COC2 N(C1CCCn2ccnc21)C(C(CC=C)CNC(=O)C(C(C)C)NC(C)=O)=O N1(CC(=O)N(c2cc(O)ncn2)CCOC)CCCS1(=O)=O c1(C(=O)NCC(CC)(CC)NC(=O)CC2CC2(Cl)Cl)ccc(NC)c(F)c1 CC(C(=O)NC(CC1CC1)C(=O)N(CC(C)(C)C)C)S(C)(=O)=O Cc1c(C(=O)NC2CC2CNC(=O)CCC2CCOC2)ccc(Br)c1F C(C(=O)NCCC1(NC(=O)CCC(=O)N2CCC(O)CC2)CCC1)(C(C)C)OC c1(CCNC(C(CSCC)NC(c2cnccn2)=O)=O)ccc(F)cc1 CCCCC(C(=O)N(C(C)C(=O)N1CC(n2cc(C)cn2)C1)CC(C)C)C(C)C c1(C(=O)NC(C)CCNC(=O)C(c2cncc(F)c2)C)ccc(S(N)(=O)=O)cc1 c1(NC)ccccc1C(=O)NC1(C(F)F)CC(NC(c2cnn(C)c2)=O)C1 c1(OCC=C)ccc(C=NC(=O)CC2(COC(CNCCO)=O)CC2)cc1.C(C)=C c1(N2CC(CO)CC(C(C)(C)C)C2)nc2cccnc2c(=NC2CC(=O)N(C)C2)[nH]1 c1(CN(S(CC(=O)OC)(=O)=O)c2ccn(C3CNC3)n2)cc(Cl)c(Cl)c(Cl)c1 N1(C(=O)NC2(CCCN3CCCC3)OCCO2)CCN(C(c2ccsc2)=O)CC1 CC1(C)CC(N=c2nc(N3CCCCCCC3)c3cc(F)cc(F)c3[nH]2)CCO1 c1(C(N(C(C)CNC(=O)CC2(C)CC2)C)=O)ccccc1Cl N1(C(CSCC)=O)CCC2(CC1)CN(Cc1sc(CC3CCOCC3)nc1C)C2 C(CC(=O)NCC(C)C(C)(F)F)(C(F)(F)F)NC(c1c(OC)ccnc1)=O c1(C(=O)NC2CC(NC(c3cccc(NC(=O)NC)n3)=O)C2)ccc(F)c(C)c1 c1(N2C(CC(CC)NC(C3CCCC4CC34)=O)CCC2)ncc([N+](=O)[O-])c(C)n1 C=CC(C)(O)CC(=O)NCCC1(OC)CN(C(=O)CC2CC3CCC2C3)C1 C1(C(=O)NCCCN(C)C(c2ccc(N3CCCC3)cc2)=O)CC(C2CC2)=NO1 c1(CCNC(C2CCCC(NCc3ccc(O)nc3)C2)=O)ccc([N+](=O)[O-])cc1 C(CCC)(CCCC)NC(CC1(C=C)CN(C(=O)C(F)(F)CCC)C1)=O C12(NC(CP(C)(C)=O)=O)CCN(C(c3cncs3)=O)CC1C2 C1(C(=O)NC2CN(C(C(N3CCNC3=O)C)=O)C2)CCc2nc[nH]c2C1 N1(C(C(C)=C2CCC2)=O)CC2(C1)CN(C(=O)CC1CSC1)CC2CO N1(CCCN2C(C)(C(C)C)CC2)C(=O)CNC(C)(C)C1=O N1(C(C2C(C#C)C2(C)C)=O)CCN(C(=O)C=C(C2CC2)C2CC2)C(CCOC)C1 c1(C(=O)NC2CC3CC2CN(C(c2cncnc2)=O)C3)cnn2cccc(Cl)c12 c1(-c2cn(C3CC(NC(c4ccncc4)=O)C3)nn2)cc(F)cc(F)c1 N1(C(CCN(C(=O)C(C2CC2)OC)CC)=O)CCC(O)CC1 C1(CC(=O)NC2CCOC2C2CC2)COCCN1C(=O)COc1ccsc1 C(=O)(C(C)(C)C(O)C(C)C)N(CCCCCC(=O)NCCCC(C)C)C Cc1cc(C(=O)NC(C(=O)NCCC(F)F)C2CCCO2)oc1C Cc1cc(C(N2CCC(O)C(NC(C3(C(F)(F)F)CC3)=O)C2)=O)cc(C)n1 CN(C)S(=N)(=O)N1CCCC1C(N1CCn2ccnc2C1)=O C1(C(N2C(CNC(C(C)SC(C)C)=O)CC(F)C2)=O)CC2(C1)CC(F)C2 c1(C(N2CCOCC(CNC(C3CC4(CCC4)CO3)=O)C2)=O)cnc(O)cc1O C1(CCC(=O)NC2C(C(=O)OC)CC2)CCCN(C(=O)CC2CC(N(C)C)C2)C1 c1(C(N2CCC(Cc3ccccc3Cl)CC2)C(=O)NC)cccc2cnccc12 c1(OC)ccccc1OCCC(=O)NC1(CN(C(=O)CCSC(C)C)C)CC1 C(CCN=c1nc(N2CCS(=O)(=O)C(CO)C2)c2c([nH]1)CCCCCC2)NC.C1CO1 COn1cnc(C)c1C(=O)NC1CN(C(=O)CNc2ccccc2Cl)CC1F N1(C(CCN(C)C(c2c[nH]nc2C(F)F)=O)=O)CCC2(CCOC2=O)C1 C1(C(N2C(CC(=O)N(C)Cc3nccn3C)CC(F)C2)=O)CCCC2(CC2)C1 c1(C(=O)NCc2c(-c3scc(C(=O)OC)c3)c[nH]n2)ccc2nc(Cl)sc2c1 C1CCN=C2NC(=NC=C2Br)N1.C#CCCCOCCOC C1(NC(C2C(C)(C)C2)=O)CC2(NC(=O)C=C3CCSCC3)COC1C2 CC1CN(C(C(=O)NC2COC2)C(C2CC2)C2CC2)Cc2c[nH]nc21 c1(C(N2CCC(CNC(C3(C)CCOC3)=O)C2)=O)c2c(cc3c1CCC3)CCC2 c1(C(N2CCC(C3CCCO3)CC2)=O)ccc(-n2cccn2)cc1 C1(CC)(NC(=O)C(C)SC)CCN(C(C2CC(C)(C(C)(C)C)C2)=O)CC1 N1(C(C=Cc2ccc(C)o2)=O)CCC(C)N(C(=O)CCc2ccn(C)n2)CC1 Cc1cc(OCC(=O)NC2C3CN(C(C4CNC(=O)CC4C)=O)CC23)ccc1Cl C1(C(=O)NCC2OCCN(C(C)=O)C2)CC2CC(CN2)O1 C1(C(N(C)CC2C(C)C2)=O)CCCC(NC(=O)C(C)(C)CF)C1 c1(C(CC(=O)NCC(C)CNC(c2cc(Cl)no2)=O)C)c[nH]c2ccccc12 N1(C(c2cc(C)sn2)=O)CCC(CC(C)NC(C2(O)CCOC2)=O)CC1 Cc1cc(O)ncc1C(N1C2CC1CN(C(=O)Cn1cnc(=N)[nH]1)C2)=O C1(C(=O)OC)CC2(CC(NC(C3(F)CCN(Cc4ccc(F)c(O)c4)C3)=O)C2)C1 c1(C(=O)OCC#CC(C)C)ccccc1OCc1cccnc1 CCC(CC)CC(=O)NC12CCC(n3cc(CN4CCC4CO)nn3)(CC1)C2 C1(NC(C(C=C)(C)C)=O)CCN(C(=O)Cc2c(F)cncc2Cl)CC1F c1(NS(CC2(OCC)CCC(F)(F)CC2)(=O)=O)cc(Cl)c2c(c1)OCO2 N1(C(C(C(C)C)OCC)=O)CC2(CCNC(=O)Cn3nc(C)nc3C)CCC1C2 Cc1cn(C)nc1C(=O)N(CCCNC(=O)C(C)CO)CC1CCCC1 C1(S(N)(=O)=O)(C(N(CCC)CCNC(=O)CCOc2ccccc2O)=O)CCC1 C1(C(=O)NC2(c3ccc(F)cc3)CC2)CC2CC2N1C(c1cc(Br)no1)=O c1(N2CC3C(CNC(CCCOCCC)=O)C3C2)cnc2ccccc2n1 Cn1nnnc1C(C)(CCC1CCCC1)NCCCOc1ccncc1 C(=O)(C1c2c[nH]nc2CN1C(=O)Nc1nc(-c2ccc(C)cc2)c(C)s1)NC CC(C)(C)C(CC(F)(F)F)C(=O)OC1CCCC1=O.C1(=O)CO1 c1(C(N(CC(CC)NC(C(C)OCC=C)=O)CC)=O)cncc2nc(C)[nH]c12 N1(S(C)(=O)=O)CCCC(c2nc(Cc3ccns3)no2)C1 Fc1ccc(-c2nc(C3CCC3c3ccccc3)n(C3CCC3)n2)c(F)c1 N1(C(c2cc(C(C)=O)sc2)=O)CCC(NC(=O)CC2CCN(C)C2)C(F)C1 N1(C(c2ccn(CC)n2)=O)CC(OC)CC(NC(c2cnn(CC(C)C)c2)=O)C1 c1(CCC(=O)NC(CNC(c2cn(C)nc2)=O)C2CCC2)ccc(N(C)C)cc1 C(=O)(CC(F)(F)F)NCCN(C(=O)COc1ccccc1)CCC.C(=O)(C=CCF)N C=C=CCC(=O)NCCN(CCCN(C)C)C(c1cc(-c2ccn(C)n2)on1)=O C#CCC(CC#C)C(=O)NCC1CC(CNC(c2cc(N)cc(F)c2)=O)C1 c1(CCn2c(C(CCCSC)NCCC=C=C)nnn2)cccc(F)c1 c1(C(=O)NCC(C)NC(=O)C(c2ccc(Cl)cc2)(F)F)ccc(CO)cn1 C1(C(N2C(CN(C(Cc3cn(C(C)C)nc3)=O)C)CCC2)=O)NC(=O)OC1C CC(CCNC(C1(CF)CCC1)=O)CCNC(C1(F)CC1c1ccccc1)=O c1(OC)c(C(=O)NC2CN(C(C3CCCC(C)C3)=O)C2)cc(Cl)cc1Cl N1(C(C)NCCn2nnnc2C2(C(=O)OC)CCC(C#N)C2)CCC2(CCCO2)CC1 n1(CCC(=O)NCCC(=O)NC(CC)COC)ccnc1C CC(CS(C)=O)C(=O)N(CCNC(c1cccc(NC(N)=O)c1)=O)C1CC1 C12CCCC1NC(=O)C2.c12sccc1OC2=O.C1(CN(CC)CC)CCC1 N1(C(C(C)SCC)=O)CCN(C(c2cn(CC)nn2)=O)C2CCCC12 Nc1ccc(C(=O)NCC2CCCN2C(c2coc(C(F)(F)F)n2)=O)nc1N c1(CNC23CC(CC(=O)NCC4OCCN(C)C4)(C2)C3)ccc([N+](=O)[O-])cc1 C(=O)(C1=CCCOC1)N1CC(C)C(CCNC(=O)CCc2cccc(Cl)c2)C1 C=CCCC(F)(F)C(=O)N(C)CCN(CC(=O)O)C CC(C)CC(C)(C)C(=O)NC(C)C(C(C)C)NC(c1ccccc1F)=O C(=O)(CCC(=O)Nc1nccs1)NCC(C1CCC1)NC(c1ccc(CC)s1)=O CS(=O)(=O)c1ccc(CNC2CC(C(=O)Nc3cc(Br)ccc3C(N)=O)C2)cc1 N1(C(C)=O)CSCC1C(=O)NCCC1(NC(=O)Cc2ncc(C)s2)CC1 N1(C(c2nnn(C)n2)=O)CC(NC(c2nnc(Cl)cc2N)=O)C(C)(C)C1 CC1CC(CNC(c2cc(=N)[nH]n2C)=O)CN1C(c1cnn(C2CC2)c1)=O C1(F)(CNC(c2cccc(CF)c2)=O)CCN(C(c2cn3ccnc3s2)=O)CC1 C1(CC#C)(C(=O)N(C2CSC2)C)CCN(C(c2ccncc2Cl)=O)C1 N1(CCC(=O)NCC(C2N(C(C=CCSC)=O)CCC2)(C)C)CCN(C)CC1 c1(OC)ncc(Cl)c(=NCC2(O)CCCN(C(C3C(C)OC(C)C3C)=O)C2)[nH]1 N1(C(COCc2cc(C)on2)=O)CCCC(N(C(=O)C(C)C(C)C)CCF)C1 CCC(CC)(CC)C(=O)NCC(C(=O)NC(c1csnn1)C)N(C)C C1(CC(=O)N(CC)CC2CC2(C)C)CCCN1C(=O)CCC1CC1(F)F Cc1cccc(CCNC(=O)C(C)NC(c2c(C)nsc2C)=O)c1 CCC(F)(F)CC(=O)NCC(C(=O)NCCn1ccc(=O)cc1)N(C)C.CC c1c(F)cccc1F.c1(NC(C2(C)C(C)(C)C2)=O)cccnc1C(=O)OC CC(C)CC(C)CC(=O)NCC1(F)CCN(C(C2(C)CCNC2=O)=O)C1 O=[N+]([O-])c1ccc(S(=O)(=O)NCCc2ccccc2Oc2ccccn2)s1 C1(C(N(CCN(C(C=CCCC=C(C)C)=O)C)C)=O)CCCC1P(C)(C)=O C1(NC(c2csc(C3CC3)n2)=O)C2CN(C(c3cncnc3C3CC3)=O)CC12 c1(NCC2CC(F)(CO)C2)cc(NCC(N2CCC(O)CC2)C)ncn1 Cc1ncc2n1CCN(C(=O)CC=CCNC(C1CC(=O)CCO1)=O)C2 C1(C(N2CCCC(NC(=O)CCc3ncc[nH]3)CC2)=O)CCc2nc(O)[nH]c2C1 CCCC(F)C(=O)N1CCCC1CNC(C1(OCC)CCCCC1)=O N1(C(C(C=C)(C)CC)=O)CCC2C(C1)NC(=O)CN2C(=O)C1=CCC1 N1(C(C(CC)COC)=O)CCC(CNC(=O)CCCC2CCC2)C(F)(F)C1 CC(C)(CCNCCNC(=O)C(=O)Nc1nnnn1CC(F)F)S(C)(=O)=O N1(C(C(CCC)C)=O)CC(CNC(c2cccc[n+]2[O-])=O)OC2CCCC12 N1(C(CCCCN(C(C)=O)C)=O)CC2CCN(C(C3(C)CCC3)=O)CCC2C1 c1(C(=O)OCC)ncnc2ccc(OC)cc12.N12CCC3C(CCN3CC1)C2 C1(NC(c2c(OC)nccc2)=O)CC2CCC1N2C(=O)Cc1csc(C)n1 N1(C(C(CSC)(C)C)=O)CC2CC(NC(c3cc(C4CC4)ccc3Cl)=O)C1C2 C(CCN=c1ccnc(NCCNCCCN2CCOCC2)[nH]1)OC C1(CNC(CCOCCN(C)C)=O)CCC(C)(C)CN1C(C1CCNC1=O)=O Cc1cc(Br)cc(CNC2CCC(C(C)(C)C)C2)c1OC(F)F c1(SCC(=O)N(C2CN(C(=O)CC3CCCCO3)CC2F)C)cccc(F)c1 N1(C(C(C2CC2)OCC)=O)CCC2(C1)CN(C(=O)C#CC1(C)COC1)CCO2 C1(C(N(C(C(=O)N(CCF)CC)C)C2CC2)=O)CC(C)CC(=O)N1 Cc1nc2ccccc2c(C)c1C(N1CC(NC(=O)C(F)(F)C2CC2)CC1C)=O c1(C(=O)NCC(CC(C)C)(C)NC(=O)COCCCF)occ2c1CCOC2 CC1CC(C(=O)NCC2=CCN(C(=O)COCC3CCOCC3)CC2)CC(C)C1 C1(O)(C(=O)NCC2C(CNC(c3c[nH]c(=N)s3)=O)C2)CCSCC1 C1(C(=O)NC2(CC(=O)NCC3=CCCCC3)CC2)CCC(C2CC2)C1 c1(CC)conc1CC(=O)NC1(CNC(=O)C(C)Cc2cnco2)CCOC1 c1(C(=O)OC)cc(=NC(CNC(C2(O)CCCC(C)CC2)=O)C(C)C)[nH]c(Cl)n1 N1(C(CCC(=O)OCC)=O)CCN(C(c2c(C)nc(SC)nc2O)=O)CC1C#N CN1CCC(O)(CNC(=O)CC2(F)CCN(C(=O)C(C)(C)N(C)C)C2)C1 CC(C)(C)C(CO)C(=O)NC1CCCC1NC(c1c(Br)cnn1C1CCC1)=O c1(C(N2CC3C(NC(C4CC(O)(CC#C)C4)=O)C(C3)C2)=O)cc2c[nH]cnc-2n1 C1(CC)CCN(C(=O)OC(C)(C)C)C1C.C12(CSC1)NC2 CC12CC(CNc3nccc(N4CCC(C)(CC#N)C4)n3)(CO1)C2 c1(OC)cc(C(=O)NCC2CCCC2NC(c2cc(C)ns2)=O)sn1 C1(NC(CC2N(C(C)=O)CCC2)=O)CC(F)CN(C(c2cnn[nH]2)=O)C1 C1(C(=O)NC(CC#C)C(=O)NCCC)CC2C=CC1CC2.C1CCCC1N(C)C CC1(C)OCCC1C(=O)NC1CCCC1CNC(c1csc(=N)[nH]1)=O C=C1CCC(C(=O)NC(C(=O)NCc2cccc(Cl)c2)C2CC2)CC1 c1(CC)ncncc1C(N1CC2CC2(CNC(=O)Cc2csnn2)C1)=O C(=O)(CCC1=NNC(=O)CC1)N1CC(NC(C(CC)CC)=O)C2C1C2 C(=O)(C(O)(C(F)(F)F)C1CC1)N1CCC(CNC(=O)CC2CCC2)C(O)C1 C1(NC(=O)CC(F)(F)F)CC(F)CN(C(=O)Cc2cncc(O)c2)C1 N1(C(=O)OC(C)(C)C)CCCC1C=CC(N1CCOCC1C(C)(C)C)=O c1(OC)cc(OC)c(C(N2CCC(NC(C3CC3(C)C)=O)C(OC)C2)=O)c(N)c1 C1(C(=O)NC(CC)CNC(=O)Cc2cnn(C(C)C)c2)CN2CCCCC2CO1 c1(C(=O)NC2C(CNC(c3c(C)n(C)nc3)=O)C2)cc2c(C)c(Cl)ccc2[nH]1 c1(C(C)NCC2CCN(c3ccc(OC)cc3)CC2)ccc(F)cc1Br C1(C(=O)NC(C(CO)NC(CCC#C)=O)C)CCCOC1C(=C)C c1(C(N2C(CNC(C3C(=C)C3)=O)(CO)CCC2)=O)ccc(OC)c(Cl)c1F c1(CC)nc(=N)[nH]cc1C(N1CC(NC(c2ccncc2F)=O)C2CC12)=O C(C)(CCNC(=O)Cc1cnoc1)NC(C1C(=C)C1)=O c1(SCC(N2C(CNC(c3cnc(CC)[nH]3)=O)CCC2)=O)ccc(Br)cc1 Cc1cnc(C(=O)NCCC(C)NC(=O)COCCN(C)C)cc1Cl Cc1ccc(C(CN2CCCCC2)Nc2ccc(-n3cnnn3)cc2)cc1 Cc1ccc(C(N2CC(c3ccccc3)Nc3ccccc32)=O)c2c1cnn2C O(S(=O)(=O)c1ccccc1S(=O)(=O)N1CCCC1)C1CN(C(C)COC(F)F)C1 c1(OC)cc(CN=c2[nH]c(CN3C(CO)CCC3C)cs2)cc(O)c1O C1(NC(c2c(C(=O)OC)scc2)=O)CCCC2CN(C(c3ccn(C)n3)=O)CC12 N1(C(C(CC)C)=O)CCC(c2ccccc2)(CNC(=O)COc2ccsc2)CC1 c1(NC(C2CC(CC(=O)NCC3(OCCO)CCC3)C2)=O)ccc(Br)nc1 C(=O)(CC1=CCN(C(C2(C)COC(=O)N2)=O)CC1)N(C(C(C)SC)C)C c1(C(N(CCOC)CCNC(=O)C2=NOC(C)C2)=O)cc2c(s1)CCCCC2 c1(C(=O)NC(CCNC(c2nc(OCC)sn2)=O)C(C)C)ccc(S(N)(=O)=O)o1 CC1(C)CN(C(c2nn[nH]c2Cl)=O)CC1NC(C1CCN(c2nccs2)CC1)=O C1(NC(CCSCC)=O)CC2(CCCN(C(=O)C(C)=C3CC3)C2)C1 c1(C(=O)NC2CC(C)(NC(C(CCCCC)O)=O)C2)cccc2nc(C)[nH]c12 c1(OC)ccc(CCCC(=O)NC(c2ccc(Cl)cc2)CC(=O)O)cc1F C=CCCCCC(=O)N1C2CCC1C(CNC(=O)CS(=O)(=O)N1CCCCC1)C2 c1(C(=O)NC(CNC(C2CS(=O)(=O)C2)=O)CO)c(C(F)(F)F)cccc1Cl CC1(C)CCCN(C(c2cccnc2N)=O)C1CNC(C1CCC2CC12)=O N(C(=NCCCN1CCOCC=C1CCO)NCC)Cc1c(F)cc(C)cc1F c1(C(N2CCC(O)(CN(C(=O)C=C3CCC3)C)C2)=O)cnn2ccc(O)nc12 C1(CC)C(NC(=O)COC2CCOC2)CCCN1C(=O)CCCCOC CC1(CNC(C2(CC(F)(F)F)CC2)=O)CCN(C(=O)C=CC=C(Cl)Cl)C1 c1(CN2CC3C(C(=O)Nc4cc(OC)c(Br)nc4)C3C2)ccc([Si](C)(C)C)cc1 Cc1ccc(C=CC(=O)NC2(C3CCCCN3C(C3CCC3(C)C)=O)CC2)o1 Cc1cc(O)c(F)cc1NC(C1COCCN1C(c1ccc2cc[nH]c2c1)=O)=O C(=O)(C(C#N)C(C)C)NC(C(=O)NC1C(OCC)CCC1)CCF N1(C(c2c(CC)[nH]nc2Cl)=O)CCC(C)(C)C(CNC(C2CCN(C)CC2)=O)C1 c1(C(N2C(CCC(=O)N(C)C3CC3)CCC2)=O)ccnc(Br)c1F CCC(CC)C(F)C(=O)N1CC2C(CC(=O)N(CC(C)SC)C)C2C1 N#Cc1cc(CNC(C2CC3(C2)CN(Cc2cc([N+](=O)[O-])cs2)C3)=O)ccc1F N1(C(C2C(CNC(C=CCOC)=O)C2)=O)CCC(c2ncco2)C1 Cc1cc(Br)c(NC(C2CN(Cc3ccc(O)c(F)c3F)CCC2O)=O)nc1C C(C(CC(=O)O)NC(=O)C(c1ccccc1Br)C1CCC1)SC c1(C(=O)NCC(C2CC2)NC(C=Cc2c(C)cccc2)=O)ncc(C#N)cc1Cl C(=O)(CC1OC(=O)c2ccccc21)N(CCC(C)NC(c1scnc1Cl)=O)C N1(C(c2cnsc2)=O)CCC2(CCCC2NC(=O)C(O)(C2CC2)C2CC2)CC1 CC(C)C(C)(C)C(=O)NC1C2CCC(C2)C1C(N1CC(O)(C(F)(F)F)C1)=O N1(C(C(CCC)OC)=O)CCCN(C(C2CC3CCC(C2)C3=O)=O)CC1C c1(C(=O)NCCCC(CCC)NC(c2ccco2)=O)cnn2ccc(OC)cc12 CCC(C)CCCC(=O)N(CC(C)(C)CNC(=O)C(C(C)O)NC(C)=O)C c1(C(=O)NCC(CNC(C2N(CC)CCCC2)=O)(C)OC)ccc(C#N)c(C)c1 c1(CC(C)C)ccccc1C(=O)NC(C12CCC(CC1)C2)C c1(N2CCC(NC(CC(CCC)C)=O)C(F)C2)ccc2c(n1)CCC2=O C#Cc1ccc(F)cc1C(=O)NC1(C)CC(NC(=O)C(c2cccn2C)=O)C1 c1(NC(c2c[nH]n3c2nc(=O)c2ccccc32)=O)nc2ccc(Cl)c(Cl)c2s1 c12ccc(cc1)CSCC(C)(CC)NC2=O.CCC(O)C=O C1(CN2CCN(C(c3cccnc3)C(C)C)CC2)CCCC2(C1)CC2(F)F N1(C2CCCN(C(C3C(C(N)=O)C3)=O)C2)CCN(C(=O)C(O)C2CCC2)CC1=O c1(N2CCC(CC=C)(NC(=O)C(c3ccccc3Cl)C)C2)ccncc1[N+](=O)[O-] Cc1nn(-c2ccc(F)cc2)cc1C(=O)NCCCNC(c1n[nH]c(C)c1C)=O CCCC(O)C(=O)NCC(c1ccccc1)CNC(=O)C=CC(C)(C)SC CC1(C)CC(O)(C(=O)NCCNC(c2ccnc(C(C)C)n2)=O)C1 c1(C(N(C)CC2CCN(C(c3ncoc3C3CC3)=O)C2)=O)cnc2ccoc2c1 CC(C)CC(C(=O)NCC1CC(C)C1)ONC(c1cc(Cl)cn1C)=O N1(C(C)C)CCOC(C(=O)NC(C2CCN(C(=O)COc3ccsc3)CC2)C)C1 c1(OC)ccc(Br)c(CC(=O)NC2CCCC2NC(C2CCOC2)=O)c1 C1(C=C)(C(=O)NC(CC=C)CNC(c2nc(C)n(C)n2)=O)CCOCC1 c1(OC)ccc(CO)cc1C(=O)NCCC1CCN(C(=O)Cc2cccnc2)C1 C1(O)(CN(C(C(=O)NC(C)C)=O)C)CCCN(C(C2(CO)CCCC2)=O)C1 C12(C(N3C(CNC(C4N(CCC)CCC4)=O)CC3)=O)CC3CC(C1)CC(O)(C3)C2 CC1CC(CC2(C)CC(CNn3cc(-c4cccnc4F)nn3)C2)CCS1 N1(Cc2ccccc2)CCCN(C(=O)Nc2cc(C)c(Cl)nc2)C(C)C1 c1(CC(N2CC(SC)C(NC(C3(CC(F)F)CC3)=O)C2)=O)ccc(O)c(F)c1 c1(NC(C2CCCCCN2C(C2CCCN2C2CC2)=O)=O)cccc2[nH]ccc12 C1(NC(c2cccc(Br)c2F)=O)CN(C(C2CC23CCC3)=O)CC2CC12 N1(C(CCCCSC)=O)CCN(C(=O)CSC2CC2)CC1CO C1(N(C(=O)Cc2csc(S)n2)C)CCCN(C(c2cc(Cl)n[nH]2)=O)CC1 c1(C(=O)NC(C=CC(=O)NCC2(SC)CCC2)C)cc2ccccc2[nH]1 N1(C(C(CN(C)C)(F)F)=O)CCN(C(=O)CC(=O)Nc2nccs2)C2CC12 CCC(C(O)C(C)C)NC(C1(CC)CCN(C(=O)CCCC(C)=O)CC1)=O C=CCC(C(=O)N1CCC(CF)(NC(C2CC2C2CCCO2)=O)C1)c1ccccc1 C1(C(=O)OC)CC(OC)CN(C(c2nc[nH]c2CNC(C)=O)=O)C1 N1(C(C(CCC#C)O)=O)CC2CC(NC(=O)CCCCCOC)CC1C2 O(C=C(C#N)C(=O)NCC1CCN(C(=O)C2=C(Cl)CC2)CC1C)CC C#CC1CCCC(N=c2[nH]nc(-c3ccc(Br)cc3)n2C2CC2C)C1 C(=O)(C(F)CC(C)(C)C)NC1CC=C(C(=O)NCC(c2ncn(C)c2)O)C1 Cc1ccn(C)c1C(=O)NCC(O)CNC(c1cccc(N2CCCC2=O)c1)=O C(=O)(CCCCCNC(c1cc(CO)n(C)n1)=O)NCC(CC(C)C)N(C)C CC(C)CCC(C(=O)NCC(F)C(C)(C)O)NC(C1(C)CC(C)C1)=O C1(C(=O)NC(C(=O)N(C)CC2CC(=C)C2)CCOCC)CC2(C1)CC(C)C2 c1(C(=O)NCC2(F)CCCN(C(C3C(=C)CC3)=O)C2)c[nH]c2cc(Cl)ccc12 C(=O)(CCS(C)(=O)=O)NCCN(C(c1nc(CC)sc1)=O)CCOC C1(C(=O)NC(C(CO)NC(c2c(OC)nsc2)=O)C)CC(C)OC(C)C1 C1(CNC(c2cccc(NC(C)=O)n2)=O)CC2(CO1)CN(C(c1cnoc1)=O)C2 CC1(C)CN(C(c2cccc(CF)c2)=O)CC1NC(=O)C(c1ccccc1Cl)O Cc1cnc(C(=O)N(C2CCN(C(=O)COc3cccnc3Cl)C2)C)cn1 c1(C(N2C(CCNC(c3n(C)nnc3)=O)CCCC2)=O)ccc2c(c1)NCC2 c1(C(=O)NCCN(C(C(CC)COC)=O)C2CC2)cnn2c1OCC1(CC1)C2 C1(C(N2C(C(N(CCCC)CC=C)=O)CC(O)C2)=O)COCCC1(F)F.C=CCO N1(C(c2ncc(OC)cn2)=O)CC(NC(C2CCCCO2)=O)C(C)(C)C1 N1(C(c2ccc(C)[nH]2)=O)CCCC12CCN(C(=O)C(F)(F)C1CC1)C2 C(C(C)(C)CC(=O)NC(CO)CC(C)(C)C)NC(c1cn(CC=C)nn1)=O N1(C(c2n(C)nc(O)c2)=O)CC2(C)CN(C(c3csc(S)n3)=O)CC2(C)C1 C1(C(=O)OC)CCCC12CN(C(=O)CC(C(F)F)NC(=O)OC(C)(C)C)C2 Cc1nn2c(C(=O)NC(C)CN(C)C(c3ccc(C)n(C)c3=O)=O)c(C)nc2s1 CCC(CNC(=O)C(CC1CCC1)NC(c1c[n+]([O-])c(C)cn1)=O)C(C)(F)F N1(C(C2(n3cc(CC=C)nn3)CCOCC2)=O)CC(=O)N(C)CC1C C1(C(C)NC(c2cnc(C(C)C)[nH]2)=O)CCCN(C(=O)C(C)(C)OC(C)C)C1 N1(C(c2cc(C)n(C)n2)=O)CC2(CCC2)CC1C(=O)NC1COC(C(C)C)C1 C1(N(C(c2c(C)cn(C)c2)=O)C)CCN(C(=O)CCCC(C)C)CC12CC2 C1(CC(=O)NCC=CCSC)(NC(c2ccoc2)=O)CCC1 Cc1c(C(=O)NC(CNC(=O)C(C)(C)C2CCCO2)C2CCC2)cnn1CCO N1(C(CCCC(CC)CC)=O)CCC2(C=C(C(=O)NC(C)Cn3cnnc3)C2)C1 N1(C(c2c(CC)oc(C)c2)=O)CCOC(C(N2CCN(CC)CC2C)=O)CC1 c1(C(=O)NCCC2N(C(CC(C)C(F)F)=O)CCSC2)cccc2nn[nH]c12 N1(C(c2ccnc3cc[nH]c23)=O)CCC2CN(C(C3CC3(F)Cl)=O)CC2CC1 C12CN(CC13CC3)C(=O)CCC(C)(C)NC(=O)N2.C1(C(=O)OC)(CO)CCCC1 c1(OC)cccc(CC(=O)N(CCCN(C(=O)COc2cccc(C)c2)C)C)c1 Cc1ccc([N+](=O)[O-])c(NC(C2CN(C(=O)CN(C)C)CCC2O)=O)n1 S(=O)(=O)(c1ccc(N2CCC(NC3CCCCC3)CC2)nc1)N(CC(C)CO)C C(c1ccc(O)cc1)=CC(N1C(CCNC(c2c(C)scc2)=O)CCCC1)=O c1(C(C)NC(C2N(Cc3c(C)scn3)CC(F)(F)C2)=O)ccc2ncsc2c1 c1(NC(c2ccnn2C)CC)ncc(C)cc1S(=O)(=O)NCCC(C)C(F)F c1(C(N2C(C(=O)NC(C3CCCCC3)C)CC3CC32)=O)occ2c1CCC2 c1(C(N2CCN(C(C(C=CC)O)=O)CC(O)C2)=O)ccc2nc(C)[nH]c2c1 C1(CNC(CCC#C)=O)C(C)CCN1c1cc(C(F)(F)F)ncn1 CC(C#N)CCC(=O)N1CCCCNCC1.C(=O)(N(CCN)C(C)C)O CCCCC(O)C(=O)N1C(CC(N2CCCCC2CCOC)=O)C2CCCC12 CN1C(=O)CN(C(=O)CC2NC(=O)CNC2=O)CC1=O C=CCC(CC)C(=O)NC1(C(=O)NCCC(C(C)C)N(C)C)CCOC1 c1(C(=O)NCC(C)NC(C=CC(C)(C)SC)=O)cnn2c1CN(C)CC2 C1(N(C)Cc2ccc(C(=O)OC)[nH]2)Cc2ccccc2C1OC C1(CCNC(=O)C(F)CC2CC2)CCN(C(C2(Cl)CCC2)=O)CC1 C=CCCC(F)(F)C(=O)N1CC2CCC2(CNC(C2CC(C)(C)CN2C)=O)C1 C(CC(O)C(=O)N(CCNC(C1CC12CC(O)C2)=O)CCc1ccccc1)SC C1(C)(COC)CCCN(C(C2CN(C(C3(N(C)C)CCCC3)=O)CC2CO)=O)C1 C1(C(=O)NC2CC(NC(c3sc(C)c(Br)c3)=O)C2)CC2(CCOC2)C1 C12(C(=O)NCCc3c(C)n[nH]c3)CCN(C(c3[nH]ccc(=O)c3C)=O)CCC1C2 O=C1Nc2ccc(Br)cc2CCC1Sc1ccc(Cl)cc1 c1(C(N2CCC(O)(c3cn(CCOC(C)=O)nn3)C2)=O)cc(F)cc2c1CCC2 C(C)(CCC(C)(C)C)NC(CSCCNC(CCCCOC)=O)=O Cc1nc(CCNC(=O)CC2CN(C(=O)CCNC(=O)C=CCl)C2)c(C)c(O)n1 c1(CNC(Cc2c(SC)cccc2)=O)nc(C)ccc1F C1(C(=O)NC)C2CN(C(=O)NC3CCN(C4CCCCC4)C3)CC12 C1(N(C(CSCCC)=O)C2CC2)CC(C(=O)N(CC(C)C)CC)C1 C(Cc1ccccc1)(C(=O)N1CC(O)C1)NC(=O)OC(C)(C)C c1(C(C(=O)NCC2CC(F)(F)CN2C(=O)COC(F)F)=O)ccc(F)c(Cl)c1F C=CC(CC)CC(=O)N1CCC(N=[N+]=[N-])(C(=O)NCCCCN(C)C(C)C)C1 N1(C(CCCC#N)=O)CCCC(CC(=O)NCC2(c3ccccc3F)CC2)CC1 c1(OC)csc(C(N2CCN(C(=O)CC3CCCC3)CC2)=O)c1OC C(=O)(C(C)CC(C)CC)N(C1CN(C(=O)C2=COCC2)C1)CC#C c1(C(=O)NC2CC(F)(CNC(C3(F)C(C)(C)C3(C)C)=O)C2)ccc2cccnn12 c1(OC)cc(C#N)ccc1NC(=O)Cc1cc(F)c(C)cc1F C1(NC(CC(c2c[nH]c3ccccc23)C)=O)CC2CCC1N(C(C1(C)CC1)=O)C2 c1(C(N2CCC(C(C)NC(Cc3cc(C)sc3)=O)C2)=O)cc([N+](=O)[O-])cnc1C c1(C(=O)OCC(C)(C)C)nc(=NCC2(OCC)CCCCC2)cc(C(N)=O)[nH]1 Cc1oc(Cl)nc1C(=O)N(CC(N1CCCC(C)C1)=O)CC(C)C N(C1CCOc2ccccc21)C(c1cccnn1)C(=O)NC1CCOC1 c1(C(=O)NCCCCCN(C(=O)CCCC(N)=O)C)ncc(C#N)cc1Cl Cc1ccc(-n2nnnc2C(CCc2ccccc2)Nc2nc(C)c(C)[nH]2)cc1 C1(NC(C(C)Sc2ccccc2)=O)CC2CC(C1)N(C(=O)Cc1cscn1)C2 C(=O)(C(C)N(OC)C(=O)C1C=CCN(C(=O)CC2CC(=O)NC2=O)C1)OC C(c1cncc(OC)c1)=CC(=O)NCC1C(NC(c2ccc(COC)[nH]2)=O)CC1 C1(NC(C(C)(C)C)=O)CC(F)CN(C(C2CC3C=CC2C3)=O)C1 c1(C(=O)NC2C(C)N(C(C3CC=CC3)=O)CCC2)cc2c(cn1)OCCC2 c1(CC(=O)N(CCN(C(=O)C(c2cc(Br)co2)=O)C)C)cnn(C(F)F)c1 N1(C(C2(CNC(C3C4CC5C(C4)C35)=O)CCCCC2)=O)CC2C=CCC(C2)C1 c1(C(=O)NC(Cc2cc(C)[nH]n2)C)ccc(C(F)(F)F)nc1O Cc1cc(C(=O)NCC2CCCN(C(C34CCC3C4)=O)C2)nn1-c1ccccc1 C(=O)(C1CNC(=O)c2ccnn21)NC1CC(NC(c2c(OC)ccc(C)n2)=O)C1 c1(CCC)c(C(=O)NC(CN(C(=O)C=C2CCC2)C)CC)[nH]c(C)c1C(=O)OC C1(CNC(NC(COC)C)=NCCC2(O)CCOCC2)COc2ccccc2C1 Cc1c(C=CC(=O)NC2(CNC(c3ccnn3CC#N)=O)CCOC2)cnn1C C1(C)(CNC(c2cc(CNC(C3C(C(C)C)OCC3)=O)[nH]n2)=O)CC=CCC1 C(=O)(CS(=O)(=O)c1ccc([N+](=O)[O-])cc1)NC(C(C(C)C)NC(CCSCC)=O)C c1(C(N2C(CCNC(c3ccc(CO)o3)=O)CCCC2)=O)cc2sccc2s1 CC1=NOC(C)(C(=O)NCC2CCC2C(=O)NCC2(C3CC3)CCCO2)C1 C1(F)(CNC(C2CCOC2)=O)CCCN(C(c2cnn3c2OCC3)=O)CC1 Cc1cccc(C(F)C(N2CCSCC2CCNC(=O)C=CBr)=O)c1 Cc1[nH]nc(C(C)C)c1C(N1CCC(C)(CNC(c2cc(C(N)=O)c[nH]2)=O)C1)=O OCCC(N=c1ccnc(NC2CCCOC2)[nH]1)c1cccs1 Nc1ccc(Br)cc1C(=O)NCC1CCCC(NC(=O)Cc2cccnc2)C1 c1(C(N(C)CCOCCC(=O)Nc2cnn(C(F)F)c2)=O)ncccc1O N1(C(CCN(C)CCO)=O)CCC2(CC1)CC2C(=O)N(C1CCCC1)C N1(C(C(CCC2CC2)NC(=O)C(F)CC2CCOC2)=O)CC(F)(F)C(F)(F)C1 C1(NC(CCN(C)CCO)=O)CN(C(=O)C2=CCCCO2)CCC12CCC2 N(C(=NCCC)N(C)Cc1ccccc1Cn1ccnc1C)C(C=C)C CC1(CNC(=O)CSC2CC2)CCCN1C(=O)CN1CCCOC1=O C1(NC(CCCOC)=O)CC2(CCCCN2C(=O)Cc2ccc(Cl)cc2)C1 CCC(O)C(C)C(=O)N1CCC(C)(CNC(C23CC2C3)=O)CC1 CC(C)C(C(=O)NC1CCCCC1CNC(C1(C(=O)N(C)C(C)C)CC1)=O)C(C)C CC(C)C(C)(O)C(=O)NCc1nc(C(=O)NCC(C)Cn2ccnc2)co1 Cc1cc(C(C)NC(=O)CC2(O)CCOC2)ccc1C#N C(=O)(CS(=O)(=O)CC(C)C)NCC(CC=C)NC(C1(CCOC)CC1)=O N1(C(CCN(C)CCO)=O)CC(F)CC1CN(C(=O)CN1C(=O)CNC1=O)C Cc1cc(C#N)ccc1C(=O)NC(Cc1cn[nH]c1)C(N1CCCC(CF)C1)=O c1(CC(=O)NN(CC(=O)CCC2(CN)CCCC2)S(C)(=O)=O)cccc(C)c1.CO CN1C(=O)CCC1CC(N1CSCC1C(=O)NC(CO)CO)=O Cc1ccc(O)cc1NC(C1(CNC(=O)C=CC(F)(F)F)CCCC1)=O c1(C(N2CCC(c3ccc(C)s3)CC2)C(=O)NCCC#N)ccc2c(c1)CCC2 Cc1ccc(C)n1CCC(=O)NCCC1CCN(C(C2CCCCCC2)=O)CC1 C(=O)(C(F)(F)CCc1ccccc1)N(CCC)CCNC(c1scc(C)c1C)=O C(=O)(C1=NOC(C)C1C)NCCCC(C(=O)NCCOCC=C)O C1(C(=O)NCCCC(=O)N(C)CC2(OC)CCCC2)(OC)CCCCC1 C1(C(N2C3C(NC(c4cc(C5(C)CC5)n[nH]4)=O)C(C3)C2)=O)CC2(C1)CC1(CC1)C2 c1(SC)ccc(Cl)c(C(=O)NC2CC(F)(CNC(=O)CC3CCCS3(=O)=O)C2)c1 CCC(C)C(O)C(C)C(=O)NCC1CCC(C(N2CC(O)C(F)C2)=O)CC1 N1(C(C(C2CC2)OC)=O)CC=CC1CNC(=O)C(C)(C)c1ccn(C)n1 C(CC1CC1)(CC(=O)N1CCC1)NC(CSCC(N)=O)=O c1(CC(C)NC2CC(=O)N(CC3C(O)C(O)CN3C)C2)cc(Br)ccc1F C1(NC(C(CSC)(C)NC(C2C(C)(C)C2(F)F)=O)=O)CCCCCC1C CN1CC(C(=O)NCCCNC(c2nn[nH]c2Cl)=O)CCC1=O CCCCCC(F)C(=O)NC(CCCC)CC(=O)NCC1CC(F)(F)CO1 CCC(CC)(C(=O)N1CC2CCC(C(=O)NC3CCSC3)(C2)C1)C(C)C C(=O)(C1=CCCOC1)NC1C(CNC(Cc2ccc(OC)nc2)=O)CC1 C1(CC(=O)NCC(CN(C(CC(CC)SC)=O)C)(C)C)CCC(F)(F)CO1 N1(C(=O)OC(C)(C)C)CCC(CC(=O)Nc2ccc(F)c(F)c2)C(F)(F)CC1 c1(C(=O)NC(C#C)(CO)CO)n[nH]c2c1CN(C(=O)CN(CC)CC)C2 CC(C)C(C)(O)C(=O)NC1CCN(C(C2CCCN2C2CCOCC2)=O)CC1 CCCCC(F)C(=O)N1CCN(C(=O)CC(C)(F)F)CC1CC CCC(CC(=O)N1CC2(CCN(C(C3COC4COCC34)=O)C2)C1)C(C)C C1(O)(C(C(=O)NCC2(CC(=O)NCCn3cc(C4CC4)cn3)CC2)F)CCCC1 C(=O)(C1CCc2c(Cl)cccc21)NCC(CN(C(c1cc(SC)oc1)=O)C)C N1(C(c2cccc(C#N)c2)C(=O)Nc2ccc(OC)cc2)CCS(=O)C(C)(C)C1 C12(C(N3CCC(=C)C3)=O)CC(CN(C(C3CCCSC3C)=O)C1)C2 N1(C(C23OC(C)C(C2)C3)=O)C2CCC1CN(C(c1c[nH]c(=N)o1)=O)CC2 C(=O)(C(=O)CCC(C)C)N1CC(O)(CNC(C2=CC(C)(CC)C2)=O)C1 C(=O)(C(CC)CCCC)N1CCC(C(N(CCCSC)C)=O)(CF)C1 N#Cc1ccc2c(c1)CCCC2Nc1ccc(C(F)F)cc1 C(=O)(C(C)S(N)(=O)=O)NCC1CN(C(c2c(C(C)C)noc2)=O)CC1C CN1CCN(C2CC(C(=O)NCC3CC(N(C)C)C3)C2)CC1 Cc1nc2c(N3CCCC4(NC(C5CC5(Cl)Cl)=O)CC4C3)ncnc2s1 C(=O)(CCCC(F)(F)CO)N1CC(O)(CN(C(C(C)NC(CC)(C)C)=O)C)C1 C1(NC(c2cc(C)[nH]c2)=O)CCC(N(c2ccc(C(F)(F)F)cn2)C)CC1 c1(OC)csc(C(=O)N(CCCCNC(c2cc(-c3ccco3)c[nH]2)=O)C)c1 c1(OC)cc(Cl)c(C(N2CCC(C(C)NC(c3csnn3)=O)CC2)=O)cn1 CC(C)C#CC(=O)NC1(C)CCN(C(=O)C(c2ccc(Cl)cc2)(F)F)C1 S(=O)(=O)(c1c(Cl)cccc1Cl)NC1CN(C(c2ccc(F)c3ccoc23)=O)C1 c1(OC)cccc(COC(C)C(=O)N(CC(C)NC(c2cnccc2Cl)=O)C)c1 c1(C(CC)(C)C)ccc(C(=O)N(C2CN(C(c3cnsn3)=O)CC2F)C)cc1 C1(C(=O)NC2CCC(N(C(=O)CNC=O)C)CC2)OCC2COCCC12 CN1N=C(CC(=O)N2CC(CNC(=O)CC3(O)CCOC3)CC(C)(C)C2)CC1=O N1(C(C2CN(CCC)C(=O)C2)=O)CCCC(C)(CNC(c2cnc(C)[nH]2)=O)C1 C1(C(=O)NCC2C(NC(CCc3scc(C)n3)=O)C2)CC2C=CC1C21CC1 c1(C(N2CC(NC(C(n3cnc(C#N)n3)C)=O)C2)=O)ccc(F)c(C(C)(C)F)c1 N1(CC(C2CCCNC2)(C)C)CCC(O)(Cc2ccccc2)CC1 C(=O)(C(CC(C)C)NC=O)NCC(C#C)C(C)C.C1(N)C(C)(C)C1(F)F Cc1ccn(CC(=O)N(C)CC2CCN(C(C3C4COCC34)=O)CC2)c(=O)c1 N1(C(Cc2c(OC)cccc2Cl)=O)CCC2(CC(=O)NC2=O)C1 C(=O)(CCCCF)N(C1CCN(C(=O)C(c2ccccn2)O)CC1)CC#C Cc1nc(C=Cc2cnn(CCC(=O)N(C)C)c2)nc2c1cnn2C N1(C(COCC#C)=O)CCCC(C)(CNC(=O)Cn2ccnc2)C1 C1(NC(C2CC(=O)C2)=O)C2CC(CN(C(=O)CCCc3ccsc3)C2)C1CO N#Cc1ccc(=NCC(=O)NC(CNC(=O)CCC(F)(F)F)CO)[nH]c1 C=CCCCCCCNC(=O)C(Cc1cnc[nH]1)NC(C1CCCC(CF)C1)=O C1(SCCCC)(NC(CSCC(=O)N)=O)CCC1.c1(C)ccco1.C12CC1NC2=O c1(N2C(C)CC(CNC(C3(CCOCC)CCC3)=O)C2)ncnc(Cl)c1[N+](=O)[O-] C(C1(C)CCOCC1)=CC(=O)NCC(N(C)C(c1ccnc(O)c1)=O)C1CC1 N1(C(C(CC)NC(C)=O)=O)CC(C)(C)CC1CNC(c1cn(C)nc1C1CC1)=O c1(NCC2(C)CCCN(C(=O)COc3cccc(F)c3)C2)ccnc2[nH]cnc12 Cc1ccc(C(=O)NC2CC3CN(C(C4CC(O)C4)=O)CC23)c(F)c1F CC1CN(C(=O)Cc2cn[nH]c2)CC1CC(=O)NCC1CCCC1O c1(NC(C(C)N(C(=O)C=CC2CCOC2)C2CC2)=O)cnccc1CO C1(C2CN(C(c3cccc(C)c3N)=O)C2)(NC(C2CC(CC)C2)=O)CC1 C(CCCCC(=O)N1CC2CC(NC(c3cnn(C4CC4)c3Cl)=O)C1C2)OC CC1=C(C(=O)NC2CN(C(=O)CCOc3c(C)cccc3C)CC2O)CCO1 C1(C(=O)OC)CC(NC(=O)Nc2cccc(N3CCOCC3)c2)CCN1 C1(C(C)=O)CCCN(Cc2ccccc2)C1C.c12cccc(c1)SCC2=O C(=O)(C1=C(Cl)CCC(C)C1)NCC1N(C(CCCC#C)=O)CC(C)(C)C1 C1(C(=O)NCc2nc(C3CNC3)cs2)CC2CC1(c1ccnn1C1CC1)C2 c1(C(N2CCC(C)(NC(c3c(C)coc3C)=O)C2)=O)cc2c(Cl)cccc2s1 C1(NC(C2(C#N)CCCC2)=O)CN(C(c2ccnnc2)=O)CC2(CCC2)C1 C#CCC(C)(C(=O)NCC1(CC)CCOC1)NC(C)=O Cc1ccc(F)c(NC(=O)NCC2CN(C(c3ccc(C)c(O)c3)=O)C2)c1 c1(OC)cc(C(N2CCCN(C(c3cc(Br)oc3C)=O)CC2)=O)cc(C)n1 N1(C(C(C)(C)F)=O)CCN(C(c2ccc(O)nc2Cl)=O)C2CCCCC2C1 C(=O)(CCCC(=O)NC(C)CCCNC(C1CCN1C1CCCC1)=O)OC Cc1cc(N2CCCC2CN(C(=O)C(C)Oc2ccccc2)C)nc(C)n1 c1(OC)nccnc1C(=O)NCC(C1CCOC1)NC(c1ccccc1O)=O N1(CC#C)CCCC1C(N1CC(C(C)NC(=O)C(c2cscn2)N(C)C)C1)=O C1(NC(C=CC)=O)(CC)CCCN(C(=O)C(C)N(C)C)C1 C(CC(=O)N1CCC(NC(c2cc(C)n(C(C)C)c2C)=O)C1)(C(N)=O)NC(C)=O C(CC(=O)NC1CC(N(C)C(C2C=CCC2)=O)C1)SCCCC N1(C(CC2C(C)CN(C(C3(C(N)=O)CC3)=O)C2)=O)CCOCC(C)(C)C1 CCN=c1cc(C(=O)NC2CN(C(c3coc(C(N)=O)c3)=O)CC23CC3)cc[nH]1 c1(OCC(=O)NC2CC(NC(C(c3cccc(F)c3)C)=O)C2)ccc(CO)cn1 C1(C(N2CCCC(C3CCCN3C(c3nc(Cl)cs3)=O)C2)=O)CCC2(CC2)C1 N1(CC(=O)N(CC(C)OCCOC)C)C(=O)CCC1=O.c12ocnc1C(=O)N2 N1(C(c2c(C)ccnc2)=O)CC(C(=O)N(CC(C)O)C)CC1(C)C c1(CCCCC)nc(C(=O)NCCCC2CCCN2C(C2CCC(=O)O2)=O)cs1 N1(C(c2cc(Cl)ncc2Br)C(=O)NC(C(=O)OC)C)CC(C)S(=O)C(C)C1 C1(c2nnnn2-c2ccccc2)(Nc2cccc(C(C)C)c2)CCN2CCCC12 N1(C(CC2(C(=C)F)CCC2)=O)CCCN(C(C2CCS(=O)(=O)CC2)=O)C(C)C1 C(=O)(CC(C)P(C)(C)=O)NCCC1(O)CCN(C(c2c(NC)cnc(Cl)c2)=O)C1 CS(=O)(=O)C1CN(C(=O)C(O)C2CC2)CC1NC(c1cc(-c2ccco2)no1)=O N1(C(c2c(C)ccc(C)n2)=O)CC(NC(=O)CC2CCC2(C)C)C2(CCC2)C1 C1(NC(=O)CCC2CCCC2)CC2CC1N(C(=O)Cc1cnns1)C2 N1(C(c2cnn3c2CN(C)CC3)=O)CCC2(CCCN2C(c2cc[nH]n2)=O)CC1 Cc1ccc(CC(=O)NCCC(C)N(C)C(c2ccc(CO)c(F)c2)=O)cc1Cl N1(C(C=CSC)=O)C2CCCC1CC(NC(C1CCCC3(CC3)C1)=O)C2 C1(NC(C(C2CCC2)OCC)=O)(CF)CCN(C(=O)CCCc2ncco2)C1 C1(C)(C(=O)NC2CN(C(C(CCC)(C)O)=O)CC2F)Cc2ccccc2C1 Cc1cc(C(=O)NCC2(C)CCC(NC(=O)C(C)C(C)(F)F)CC2)cc(C)c1C c1(C(N2CCC(O)(CCNC(C3CCC3)=O)C2)=O)nnn2ccccc12 C1(C(=O)NCCC2(NC(=O)C3=CCCCO3)CCC2)CCn2c(O)nnc2C1 C#CC1(C(=O)NC2CC(C)CC(C)(C)C2)CCN(C(=O)CC2CCC(C)C2)CC1 c1(CCC(=O)N(C2CCN(C(c3ccco3)=O)C2)CCO)ccc2c(c1)CCO2 N1(C(CSc2cn(C)nc2)=O)CC2(NC(c3cn(C(C)(C)C)cn3)=O)CCC1C2 C1(C(=O)NCC(C)=CC(=O)NCC2COCCO2)(CO)CC(C)(C)C1 c1(C(=O)NC2(C(=O)NCC)CC2)cnn2c(C)cc(C)nc12 C1(C)(O)CCOCC1.c1(NC(=O)NC(CNC(C(C)NC(N)=O)=O)C)cccc(Cl)c1 CC1(C(N2CCC(C3CCCCN3C(=O)CCc3cn[nH]c3)C2)=O)CC2CC2C1 C(=O)(C(CCC(C)C)NC(C)=O)NCCC1(OC)CN(C(c2cnco2)=O)C1 c1(OC)cccc(C2(C(=O)NCC(C)(C(C)C)NC(C3C4CCC34)=O)CC2)c1 c1(OC)cccc(NC(C2CC(CNC(=O)COCC(F)F)C(O)C2)=O)c1C c1(C(=O)NCCN(C(CC=C=C)=O)C)ncc(F)c2ccccc12 c1(C(=O)NC2C(C)N(C(=O)CSCC#N)CCC2)n[nH]c2c1CCCCC2 Cc1onc(C2CCCC2)c1C(=O)NC1CCCCC1NC(=O)C=CCO C1(N(C(Cn2cc(CNC(c3c(C)nco3)=O)nn2)=O)C)CCCC1(C)O C1(n2cc(CCCCNC(Cc3cn(C)nn3)=O)nn2)CCCC1(C)O N1(C(=O)Cn2cnnn2)CCC(F)(C(=O)NCCCOC2CC2)CC1 C(=O)(C1CCc2cccc(O)c21)N1CCC(CCNC(C(C=C)O)=O)C1 CCC(C)CC(C)C(=O)N(C(C)CNC(c1ccc([N+](=O)[O-])cc1)=O)C N1(C(COCC(C)(C)C)=O)CC(=O)NCC1C(N1CCSC2(CC2)C1)=O C1(NC(C2(C#N)CCOCC2)=O)CN(C(=O)CCNC(=O)CO)C2(CCOC2)C1 c1(CC(=O)NC(CCN(C(C(CSC)OC)=O)C)C)c(C)nc(C)nc1O c1(C(N(C)CC2OCCN(C(C(CCOC)C)=O)C2)=O)cccc(C#CCO)c1 N1(C(CCc2cc(C)[nH]n2)=O)CCC2CN(C(C3CCN3C)=O)C(C)C12 c1(C(N2CCC(C)C2C(=O)NC2CCCC(O)C2)=O)cc(=O)n(C)cn1 CCC(O)C(C)(C)C(=O)N1CC2(CC(NC(=O)CC(C)(C)COC)C2)C1 Cc1cc(C(N2CC(C(C)NC(C3(CO)CCOCC3)=O)C2)=O)cnc1C(F)F C1(F)(CNC(C2(C(=O)NC)CC2)=O)CCCN(C(=O)CCCCCC#N)CC1 C(=O)(C#CC1CCCC1)N1CC(C=C)(CC(=O)NCC(F)Cl)C1 C1(C(=O)NC2C(CNC(C(C(=C)C)(C)C)=O)CCC2)CC2(CCOCC2)C1 c1(C(=O)OC)ccc(C(N2CCC(N)CC2C)=O)c(F)c1 C1(C(=O)OC(C)(C)C)(CO)CCN(C2CCN(CCCCCC(=O)O)CC2)CC1 c1(C(N(C2CCN(C(C(C)n3cccn3)=O)C2)C)=O)cc(C#N)c[nH]1 CC(C)(C)CC(O)CC(=O)NCC1OCCC1C(=O)NOCC1(C)CCC1 Fc1ccccc1-n1nnnc1C(c1cc(C2CC2)cs1)NCC1C=CCCC1 Cc1cn(CC(=O)NCC2CC(O)(CNC(=O)C(Cl)=CCl)C2)c2ccccc12 S(=O)(=O)(c1ccc(NC2CC(CO)C2)c(Br)c1)N1CC(CC)OCC1C N1(C(C=CC(C)NC(=O)COC2CC2)=O)CC2(C)CC1CCO2 c1(C(C(=O)NC2COC2)N(CCOC)CCF)cc(OC)cc(OC)c1Br C(=O)(C1=CCCOC1)N(CCOCCC(N1C(COC)CC(C)C1)=O)C N1(C(c2ccc(OCC)cc2)=O)CC(NC(c2coc(N(C)C)n2)=O)CC1(C)C CC(O)(CNC(c1cn(CCO)nn1)=O)CNC(c1cn(C2CC2)cn1)=O C1(C)(C(N2CCC(CCNC(CC=C=C)=O)C2)=O)CCN(C(C)=O)CC1 n1(CC(N2CC(CNC(C3(CF)CC3)=O)C3(CC3)C2)=O)nc2c(n1)CCCC2 CC1(C)CC(NC(=O)C(c2ccc(F)cc2)O)CN(C(=O)C(F)=CC2CC2)C1 c1(-c2cn(C(C)C(=O)N3CCC3C(=O)O)nn2)ccc(C(C)(C)C)cc1 C1(C(=O)Nc2ccc(C)cc2O)C2C(CN1C(c1cc(O)cc(O)c1)=O)C2(C)C c1(NC(C2CC(N(C(=O)COCC(F)(F)F)C)C2)=O)ccc([N+](=O)[O-])cc1C#N CC1CCCC1(C(N1CCC1CN=[N+]=[N-])=O)NC(c1ccsc1C#N)=O C(C(C)(C(C)C)NC(=O)CNC(c1ccncc1)=O)NC(c1c(C)nns1)=O c1(CC(=O)NC2CC(N(C(c3ccn(CCOC)n3)=O)C)C2)nnc(S)n1C CCC(CC)CCCC(=O)NC12CC(C(=O)NC(C)C(C)(C)CN(C)C)(C1)C2 c1(C(=O)NCC(CC)(CC)NC(CSCC=C)=O)ccc2nc(C)n(C)c2c1 c1(CC(=O)NCC(CC)NC(c2cc(C)ccc2O)=O)cc(OC)cc(Br)c1 N1(C(CC(CC)C(C)C)=O)CCCCC2(CCN(C(C3(C#N)CCOC3)=O)C2)C1 CC1(C)OC(=O)CC1C(N1CCC1CNC(c1cccc(Br)c1F)=O)=O c1(NCCN(C)CC2CCNCC2)cc(=O)c(O)co1 Cc1ccc(C(=O)NC2C=CC(CC(=O)NC3(c4nc[nH]n4)CC3)C2)cc1 c1(C(=O)NC2CC(F)(CNC(C(C)(C)CO)=O)C2)cc2cccc(Cl)c2s1 C=C(Cl)CCC(=O)NC(CNC(c1cc(Cl)cnn1)=O)CC(C)C c1(C(=O)NC2CCN(C(C3(C)COCCO3)=O)CC2O)ccc([N+](=O)[O-])cc1Cl C1(NC(CCOCC)=O)CN(C(C2CCC(N=[N+]=[N-])C2)=O)CC2(CC2)C1 C1(C)(CC)CCC(C(N2CC(F)(C(=O)NC3COCC3N(C)C)C2)=O)O1 c1(C(=O)NC2CN(C(CS(CC)(=O)=O)=O)CC2C)cc2cc(Cl)ccc2o1 N1(C(C2COCC3(CCC3)O2)=O)CCOCC12CCC2 N1(C(CC(C=C)C)=O)CCCC(N(C)C(c2ccc(CCO)cc2)=O)CC1 c1(NC(CC(=O)NC2(COC)CN(C(C=CCC)=O)C2)=O)ccc(C)c(C)c1 N1(C(COCc2nnc(C)s2)=O)CC2CCN(C(c3nnc(O)nc3O)=O)C2C1 C(CCN=c1[nH]c(=NC(C)C(C)C)[nH]c2cccc(F)c12)c1c(C)ncs1 C(C1CCCCC1)=CC(=O)N(C)CC1(CNC(=O)Cc2coc(C(F)F)n2)CC1 N1(C(C(CC(C)C)C)=O)CC23CCCC2(C1)CN(C(c1occc1C1CC1)=O)C3 C1(NC(C2CC(=O)NC2)=O)CN(C(=O)CN2CCNC2=O)C2CCCC12 N1(C(C(C)O)=O)CC2CCN(C(c3csc(C(=O)C4CC4)n3)=O)CC12 c1(C(N2CCC(NC(C3(CCC)CC3)=O)C(C)C2)=O)n[nH]c2c1CCSC2 C(=O)(C=CS(=O)(=O)CC)NC(CC)CNC(=O)CC1CCCCN1C N1(C(C2(CNC(c3ccc(C(F)F)o3)=O)CCCO2)=O)CCOC(CCF)C1 Cn1cc(CC(=O)NCC2CCCC2NC(=O)Cn2cnnn2)cn1 N1(c2ncc(CCC)cn2)CC2CCN(Cc3cc(F)ccc3[N+](=O)[O-])CC2C1 CC1ON=C(C(=O)N2CC(NC(c3c(F)ccc(O)c3F)=O)C3CC3C2)C1C CCCC(CCC)C(=O)NC1CC(CNC(C2CCCCO2)=O)C1 N1(C(Cc2c(C)con2)=O)CCC2CCN(C(=O)C3=CCSC3)C2C1 c1(CCc2ccc(C)o2)nc(-c2ccc(Cl)cn2)nn1-c1nc(Br)nn1C N1(C(c2cc(C(=O)OC)on2)=O)CC2CC(NC(C3CCOC(C)C3)=O)CC1C2 Cc1ccc(Cl)c(C(N2CCC(C(O)CNC(C3COC(C)C3)=O)CC2)=O)c1 N1(C(c2n(CCC)ccc2)=O)CC(NC(C2CCCCCS2(=O)=O)=O)C2(CC2)C1 Cc1cccc2c1CN(C(=O)Cc1ccccc1NCc1c(F)cccc1Br)C2 c1(NC(=O)CNC(=O)OCC(N2CCc3ccccc32)=O)n[nH]c2ccc(F)cc12 c1(C(N(C2CCCN(C(=O)C=C3CC3)CC2)C)=O)cc2nc(=O)ccn2[nH]1 N1(C(CSC)=O)CCCC(C2(NC(C3CC34CCC4)=O)CC2)C1 c1(OC)cccc(C(N2CCN(C(c3ccc(C)c(F)c3)=O)CC2CO)=O)c1N Cc1ccc(F)c(C(=O)NCC#CCNC(=O)CC2=CCCC2)c1O c1(C(N2CC(C#N)C(NC(C3CCCO3)=O)C2)=O)cccc2nc[nH]c12 c1(C(N2CCC(N(C(=O)CC3CCCC(O)C3)C)C2)=O)ccn2nccc2c1 c12c(C)nc(nc1O)SC(=O)CC2.c1(CC(CCSC)CO)ccc(F)c(F)c1 C1(NC(c2cnn(C)c2Cl)=O)CC2CCC1(N=c1[nH]nc(-c3ccccc3)o1)C2 C1(CC(=O)N(C)Cc2cccs2)CCN(C(C2CCC(=O)O2)=O)C1(C)C C1(NC(C(CCC)C)=O)CC(O)CN(C(=O)CCc2cccnc2F)C1 C1(NC(Cc2cc(C)[nH]n2)=O)CCN(C(=O)Cc2cccc(F)c2F)CC1CO C(c1ccccn1)=C(C)C(=O)NC1(C2CCCN2C(C2C=CCS2)=O)CC1 C1(CCCCNC(CSCC=C)=O)CCN(C(=O)C(C)(C)C#N)CC1 C(=O)(C(O)C(C)(C)CC)N1CCN(C(COCCC)=O)CC1C1CCCC1 C1(C(N(C)CC2CCN(C(c3n(C(C)C)ccc3)=O)C2)=O)CCS(=O)(=O)C1(C)C CC1C(NC(C2(O)CCSCC2)=O)CCCN1C(c1cccc(CF)c1)=O CC1(C)CCCC(CC(=O)NC2CC(C)(NC(=O)CNS(=O)(=O)C3CC3)C2)O1 C1(C(C)C(=O)N(C)CCn2cncn2)CCN(C(C2CC3C=CC2O3)=O)CC1 c1(C(N2CCCC(NC(C3(C=C)CC3)=O)CC2)=O)cc2ccccc2s1 N1(C(C(=O)NCC)=O)CCN(C(c2ccn(CCO)c(=O)c2)=O)CC1COC CCC1(CNC(=NCC(C)CC)NCc2nnc(C)s2)OCCc2ccccc21 Cc1ccc(NC2(NCCN(C)C(=O)OC(C)(C)C)CCCCC2)c(I)c1F C1(CC(=O)N(CCC(C(C)C)NC(C2CCOC2)=O)C(=O)CO)CCC(C)(C)CO1 Cc1cc(=NCC2(F)COCCOC2)[nH]c(NC(CC2CC2)C2CC2)n1 Cc1cccc(CNC(C2CCC(n3cc(C4(CO)CC4)nn3)C2)=O)c1F CCCCCCCCCCC(=O)N(C)CCNC(C1(OC)CC1)=O C(C(=O)NCc1ccsc1C(=O)NC(c1nn[nH]n1)C1CC1)(C(C)C)SC N1(C(C(C(CC)O)C)=O)CCC2CN(C(c3cc4nc(C)sc4[nH]3)=O)CC2CC1 c1(C(=O)NCCOC2CCN(C(C(C)N(C)C)=O)C2)cc2ccccc2cn1 CCC(CCCC(=O)Nc1cnccc1C)NC(C1(F)CCC1)=O CCC(CC(F)(F)F)C(=O)N1CCCCC1CNC(c1c[nH]nc1C1CCC1)=O C(=O)(C(CNC(C1(C(C)(C)O)CCC1)=O)C(C)(C)C)NC(c1ccccc1)C c1(C(CC)C)cn(CCN(C(C)CNC(=O)C2CC2)C(C)=O)nn1 c1(OC)ccc(F)c(CN2CC3CN(Cc4c(C)cccc4Cl)CC3C2)c1OC N1(C(c2c(OC)ccnc2)=O)CCC(CC(=O)NCC(O)C(N)=O)C1(C)C c1(CC(N2CC(O)(CCc3cn(CCC(C)C)nn3)C2)=O)ccc(Cl)nc1 Cc1cnc(F)c(NC(=O)N(CC(C2CCOC2)O)C)c1 CCC(C)C(C(=O)NC12CC(C)(C1)C2)N(C(=O)CC1CC2C=CC1C2)C CCCCCC(CC)C(=O)N1CCC(C)(NC(c2ccc(OC)nc2F)=O)C1 N1(CC)CC2(CN(C(=O)C(C)(C)C3CCCN3C(C)=O)C2)C1 C(=O)(C(F)C(C)C)NCCn1ncc(C(=O)NCc2n(C(C)C)cnc2)c1 C(=O)(C1CCCn2cnnc21)NC1C(C(C)C)N(C(=O)Cn2nnc(=N)[nH]2)CC1 C(CCCCCC(=O)N1CC2(COC(=O)C2)C1)SCC C(=O)(C(=O)C(C)(C)C)N(CC(N1C(CN(CC)CC)CCCC1)=O)C C12(C(=O)NCC3CC(NC(CN(c4ccccc4)CC)=O)C3)CC=CC(C1)OC2 C1(C(=O)OC)OC(C(=O)NCCN(C(c2ccnnc2)=O)C(C)C)CC1C C12(NC(CCC(=O)NC)=O)CN(C(=O)CCCn3cncn3)CC1CS(=O)(=O)C2 N1(C(CN2C(C)CC2)=O)CC2CC2(NC(c2ccc(C(=O)N(C)CCO)cc2)=O)C1 C(C)(c1ccccc1C)=CC(N1C(CNC(C2CCCSC2)=O)CC(OC)C1)=O C1(NC(c2csnc2Cl)=O)CC(=O)N(C2CN(C(=O)C(O)Cc3cnc[nH]3)C2)C1 c1(C2C(n3cc(CNc4cn(CC)nn4)nn3)C2)ccc(F)cc1F CCCCCCC(C)C(=O)NCC1=CCCN(C(=O)CN(C)C)C1 Cc1cnn(CC(=O)NCC(C2CC2)N(C(=O)C=C(Cl)Cl)C)c1 c1(NC(C2(O)CCN(C(C(C=CC)O)=O)C2)=O)cc(OC)ccc1C C1(C(N2CC(C)N(C(=O)CC3NC(=O)NC3=O)CC2)=O)CCc2nc(O)[nH]c2C1 N1(C(c2cnc(C(C)OC)s2)=O)CC2CC1CN2C(=O)C=Cc1cc(F)c[nH]1 N1(C(CCNC(N)=O)=O)CCCOC(CCNC(=O)COCC2CCCCC2)C1 C1(CC(=O)N(C2CN(C(=O)Cn3cc(Br)cn3)C2)C)C=CCCC1 N1(C(c2cc(C(F)F)no2)=O)CC(OC(C)(C)C)C(NC(c2csc(O)n2)=O)C1 c1(SCC)cccc(CC(N2CCN(C(=O)C(C)C(=O)OC(C)(C)C)CC2)=O)c1 CP(C)(=O)c1ccc(C(=O)NC2CCN(C(C3OCCCO3)=O)C2)cc1 C1(Cc2cn[nH]c2)C(=O)NOCC(=O)N1.CCC(C)N(CC)CC CC(C)(C)S(=O)CCCN=C(NCCOc1ccccc1)NCCc1ccoc1 c1(OCC)c(NC2(c3nnnn3C)CCC2CC(C)C)occc1=O N1(C(CC(C=C)c2ccccc2)=O)CC2(CCN(C(C3(C#N)CC(C)C3)=O)C2)C1 C(CCC(C)C)(C(=O)NCC1(CO)CC1(C)C)NC(C=CC)=O C1(CNC(C2CC3(C(NC(C(NOC)=O)=O)C3)C2)=O)Cc2nccn2C1 C(CC(CC)C(=O)N1CC(O)(CNC(=O)COc2cn[nH]c2)C1)=CC c1(OC)cc(SC(C2(CCC)CS(=O)(=O)CC=CC(c3occc3C)=C2)C)c(F)cc1O Cc1cc(C)c(C(N2CCCN(C(=O)C=Cc3ccc[nH]3)C(CO)C2)=O)c(S)n1 C=CCCCCC(=O)NC12CCN(C(=O)CCCCCF)CC1C2 c1(C(C)NC(CCCOC)c2nnnn2C(C)C)ccc(OC)c(C)c1 N1(C(C(CC)SC)=O)CCCC(F)(CNC(=O)C=C(Cl)Cl)C1 N1(C(CC2CC(C)C2)=O)CC2CC1(C(=O)NC1CCOC1(C)C)C2 c1(C(=O)NCC(C)(CC)NC(C(COCC)C)=O)cncc(C(=O)OC)c1C C1(C(=O)NCC2CCN(C(Cc3nnc(C)o3)=O)CC2)CCCNS1(=O)=O C(=O)(C(C)(F)C(F)(F)F)N1CC(O)(CCNC(C2N(S(C)(=O)=O)CCC2)=O)C1 C1(CC(=O)NC(CNC(C2CCCCN2C(N)=O)=O)CO)CC(=O)NC1=O C1(N(C(COCCCC)=O)C)CCC(NC(=O)CN2CC(C)(OC)C2)CC1 Cc1nccnc1C(=O)N(C1CCCN1CC(=O)NC1CCCC1)C(C)C C12(CCNC(C3(CC)COC3)=O)CCC(C1)N(C(=O)Cc1ccc(F)c(F)c1)C2 c1(N2CCCC(CCNC(c3c(C)ocn3)=O)CC2)nc(Cl)nc2c1SCC2 CC1(C)OCC2CC12C(=O)NC1COCCC1NC(c1csnc1Br)=O CC(CC(=O)N1CCCC1Cn1c(C(N(CC(=O)O)C)=O)ccn1)CC(C)(C)C C1(CNC(c2ccc(SCC)nc2)=O)CN(C(=O)CC(C)(F)F)CCC12CCC2 C(=O)(C1=NN(C2CC2)C(=O)CC1)NC1C(C)CN(C(C2CCC2)=O)CC1 Cc1c(C(N2CCC(OCCNC(C3CCCN3C(C)C)=O)C2)=O)ccn1C Cc1cnc2c(C(=O)NCC(C)(C)CNC(=O)CSC(F)(F)F)cccn12 CCC(CC(F)F)C(=O)N1CCC(N2CCN(C(c3ccc(N)cn3)=O)CC2)C1 C(=O)(C(C)(C)C(C)(C)O)NC1CC(CCNC(C(C)OCC)=O)C1 c1(C(=O)NC2CC(C)(CNC(C(CC=CCC)C)=O)C2)ccnc(Cl)c1OC c1(OC(C)C(N2CCCC2C(C)(C)CNC(=O)CCF)=O)ccccc1C#N c1(-c2c(C(N3CCOCC3)=O)n[nH]c2)cccc(N2CCOCC2)c1 C(C)(C)(CC(=O)OCC)NC(C=CC=CC)=O.c1(C2C(=O)N2)ccccc1 C=CC(C)(CC)C(=O)NC1CCC1NC(=O)Cc1ccc(Cl)cn1 c1(C(C(=O)OCC)OC(c2c[nH]nc2CC)=O)ccccc1Cl C(=O)(C1=C(Cl)CCC(C)C1)NC1COCCN(C(c2c(OC)ccnc2)=O)C1 c1(NC2(C(=O)OCC)CC3(CCCC3)C2)nccc2oc(I)cc12 c1(CNC(C2(C=C)CCC2)=O)cnn(C)c1C(=O)NC(C1CCCCO1)C C1(C(N(CC(C)(C)CNC(=O)CC2CCCO2)C)=O)CCCC2(CCC2)O1 c1(CC(=O)N(CCCNC(=O)Cc2cc(Cl)ccc2O)C)nc2ncccn2n1 CCC(CC)CC(F)C(=O)N1CC(C(=O)NC2CC23CCCCCC3)OC(C)C1 N1(C(C(C)C(F)F)=O)CCC(C2(NC(=O)COCC3CCCO3)CC2)CC1 c1(C(N(CC(C)NC(c2cc3sccc3[nH]2)=O)CC)=O)cccc2c1OC(C)C2 S(=O)(=O)(c1cc(C)cnc1NCC1CCC(F)C1)N(C1(COC)CCC1)C N1(Cc2c(OC)cccc2)CCC(NC(=O)C(C2CCC(=O)N2)C)CC(C)(C)C1 C1(OC)CN(C)C(C)(C(=O)NC2CN(C(=O)CCc3cncs3)C2)C1 CCCC(C)(O)CC(=O)NC1CCN(C(=O)C(=O)NC2CC2)C1 C(=O)(C1CCCc2nnn(C)c21)N(CC(CN(C(c1onc(C)c1C)=O)C)O)C C=CCC(CC(C)C)C(=O)N1CC2CCCN(C(=O)CCC3CCCCO3)C2C1 Cc1cc(OCC(N2CCC(CN(C)C(c3cc(C(C)(C)C)no3)=O)C2)=O)no1 C(=O)(C(O)C(F)(F)F)NC1C(CNC(=O)CCCNc2ccccc2)CCCC1 N1(C(C(CC(CC)C)NC(c2ccc(C(C)C)o2)=O)=O)CCCC(C2(C)CC2)C1 N#Cc1cc(C(N2CC3(CCC(C(=O)NCC4(C(F)(F)F)CC4)O3)C2)=O)ccc1Br C1(C(=O)NCC)CN(C(=O)C(C)(C)C2CCOC2)CC12CC2 C(CCC(F)(F)F)N(C(=O)CCCN(C)C(C1CCCOC1)=O)C C1(CNC(N2CCC3CC2CO3)=O)CCC2(CCOC2)O1 C1(OC)CC(NC(=O)CC2CC(=O)NC(=O)C2)CN(C(c2ncnn2C)=O)C1 c1(C(=O)NC2(C3CN(C(C4C(C)C4C)=O)C3)CC2)cccc2c1C(=O)OC2(C)C C1(NC(CC2N(C(CC3N(C)CCC3)=O)CCC2)=O)CCC2CCC12 CC1CCCn2ncc(C(=O)NCC3CC(NC(c4cncs4)=O)CC3O)c21 CC1Oc2ccc(NC(=O)Nc3ncc(C4CC4)s3)cc2NC1=O n1(CC(C)O)cc(C(=O)NC2C=CCN(C(c3ncc[nH]3)=O)C2)ccc1=O C1(CNC(Cc2c(C)occ2)=O)CN(C(=O)Cn2cnc(=N)[nH]2)CC1C C1(CC=C)(NC(C2CC23CCCC3)=O)CCN(C(=O)CS(=O)(=O)NC)CC1 C1(C(N2CCN(C(C=C(CCC)C)=O)CC2)=O)CN(CC)C2(CCC2)C1 C1(NC(CCC2(C)CN(C(C3CCCC(=O)CC3)=O)C2)=O)CCOC12CCCC2 c1(C(N2CCCC(N(C(=O)CCN3CCCC3)C)C2)=O)ccc(N(C)C)c(F)c1 C1(C)(C(=O)NCCC2CC(NC(c3ccn(CC)n3)=O)C2)CC2CC2C1 c1(-c2ccc(CCCC)s2)ccc(C(N2C(C(=O)O)CC2C(C)C)=O)cc1 C1(NC(c2cc(F)n[nH]2)=O)CC(C2CCN(C(=O)CC3CC=CC3)C2)C1 CC(C)CCCCC(=O)NCCCN(C(C1CNC(=O)O1)=O)CC1CCCC1 C1(CNC(=O)CSc2cncs2)COCCN1C(=O)C(F)=C1CCCC1 N1(C(C(CSC)O)=O)CCCCC1CCC(N1CC(F)(F)C1C1CC1)=O CC1CCC(C)(C)N1C(C1CCN(C(=O)CC2CCC(C)(C)O2)CC1)=O C(=O)(CC1NC(=O)c2ccccc21)N1CC(CCNC(c2c(N)nccc2)=O)C1 CCC(CC(=O)N(CCCN(C)C)CCNC(=O)C(C1CC(F)(F)C1)O)C1CC1 c1(NC(C2CCN(CCC)C2)=O)[nH]c2ccc(C)cc2c1CNC(=O)C1CC1.CCO c1(C(=O)NCC(CC)NC(C2CC3(CC3)CO2)=O)cncnc1C1CC1 C1(CCNC(C(C)N(C(=O)CC2C=CCC2)CC)=O)CC(C)=NO1 c1(-c2n(C(COC)C)nc(C(C)C)n2)cc(Br)c2cccnn12 CC(C(=O)NCC1CC1C(=O)NCCN1CCC1)C(C)(C)C CC1CN(C(C2CC3(CCO2)CC3)=O)CCC1NC(c1cnc[nH]1)=O c1(CC2N(C(C)C(=O)O)CCN(Cc3ccccc3Cl)C2)ccc2c(c1)COC2 N1(CCN(C(CCN(CC#C)C(C2CC2Cl)=O)=O)C)CCCC1=O C1(NC(c2ccc(C)nc2)=O)C2CCC(C2)C1C(=O)Nc1ccc(N(C)C)nc1 N1(C(C2(C)CCOC2)=O)CC2(CCN(C(=O)C(N3CCCC3)C3CC3)CC2)C1 CC(C)(C)CC(C(=O)NCC1CCCCO1)NC(c1cccn2ccnc12)=O c1(C(C(=O)NC2(C)CC2)N(C2CCOC2C)CCOC)cc(F)ccc1C c1(C(N2C(C(C)NC(=O)C(=O)NCC(F)F)CCCC2)=O)nnc(O)nc1O C1(C(N(CCCO)C)=O)CC2CC2N1C(c1cc(C2CC2)on1)=O Cc1ncccc1CCC(=O)NCC1(F)CC(NC(C2CCCN2N=O)=O)C1 C(CN=c1[nH]c(N2CCc3cncnc3C2)nc2cccc(F)c12)SCC CC1CN(C(c2cn(CCNC(=O)Cc3ccoc3)nn2)=O)CC(C)O1 CCCCCC(C)CC(=O)N1CC2(CCC2CNC(=O)COCC2CCC2)C1 C=CCCCC(=O)N1CCCC1(CC=C)C(=O)Nc1cncnc1C C1(C(N)=O)(NC(C2C(NC(CC(C)O)=O)COC2)=O)CCCCC1 C(=O)(C(C)C(CC)CC)N1C(C(=O)NCc2c(CC)noc2C)CCCCC1 C(C(C)(C)CC(=O)NCCC1CCCN(C(=O)CCC(C)(C)C)CC1)OC C1(N(C(c2c(CC)ocn2)=O)C)CCCN(C(C2(C)CC(F)(F)C2)=O)CC1 N1(C(CCCCN(C)C)=O)CC2(CC(C(=O)NC(c3cnn(C)c3)CO)CO2)C1 N1(C(C2CC(OCC)C2)=O)CC(O)CC1(C)C(=O)NCCc1ncn(C)n1 c1(CC(=O)NC2C3CN(C(C(C(C)C)SC)=O)C2C3)cc(C)cc(C)c1 c1(C(=O)NCCCC(=O)NCC(C2CCC2)NC(CC#N)=O)ccc(Cl)cc1 C1(NC(C2CCCC(C)(C)C2)=O)CN(C(=O)CC2CC(=O)C2)Cc2ccnn2C1 N1(CCNC(c2n(CC)ccn2)c2nnnn2CCCSC)CCC(F)(F)CC1 c1(NC(C(C)C2CCOC2)=O)cnc(O)c(F)c1 N1(C(C2N(C)CCOC2)=O)CCC(C2(O)CN(C(C3CC4(C3)CC4F)=O)C2)CC1 c1(C(=O)NC(CCC)CC(=O)NCc2n[nH]c3c2CCC3)ccc2cnoc2c1 CON1CCC(C(=O)NC(C2CN(C(c3ccc([N+](=O)[O-])[nH]3)=O)CCO2)C)CC1 N1(C(C(COC(C)C)(C)C)=O)CC2CC(NC(c3ccc(C(N)=O)nc3)=O)C1C2 N1(C(COCCOC)=O)CCC(C(=O)NC2(OC)CCSC2)CC1C C1(CC(=O)NC2CC(CNC(C(N3CC(C)C3)C)=O)C2)CCC(=O)C1 c1(C(=O)NCC23C(CN(C(c4scc(COC)c4)=O)C2)C3)cnc(Cl)c(N)c1 c1(C(N(CCC)CCNC(c2cncc(OC)n2)=O)=O)cc(OC)nc(C)c1 C(=O)(C1=C(Cl)CCCC1)NCC(CCC)NC(c1ccn(CC)c(=O)c1)=O c1(OC)cc(NC(=O)NNC(=O)Cn2c(C)csc2=O)c2ccccc2c1 N1(C(COCCCC#C)=O)CC2CN(C(=O)Cc3cccc4c3OCO4)CC2C1 N1(C(C2CC3C=CC2C3)=O)CC2CN(Cc3ccc(C(F)(F)F)cc3Cl)CC2C1 C1(CC)CCC(C(=O)NCC(C)(C)NC(c2cc(C)ns2)=O)C1 C(CCCCN(C(C1CC1c1ccccc1)=O)C1CC1)NC(c1cncs1)=O C(CN=c1cc[nH]c(=NCCCC2CC2)[nH]1)c1cc(Cl)cc(Cl)c1Cl c1(C(=O)OC)cc(N2CCC(C)(NC(c3ccc(Cl)s3)=O)C2)nc(C)n1 c1(CNC(N2CC(O)CC2C(=O)NC2CC3CNC2C3)=O)cc2ncccc2[nH]1 CC1CC(C(=O)N(CC(=O)N(C)C)C)N1C(=O)COc1cn[nH]c1 c1(N2CCC(C)(NC(c3nccc(SC)n3)=O)C2)ncnc(Cl)c1C(C)C N1(C(c2n(C)cnc2)=O)CCN(C(c2ccc(C(C)(C)C)s2)=O)C2CCC12 C1(C(N(C)Cc2n(CC)cnn2)=O)C=CCCN1C(=O)CC=CC(C)(C)C N1(C(CCC(CC)C)=O)CCC2(CCOCC2)C(CNC(=O)CN(C)CCO)C1 c1(C(=O)OC)ccc(C(C(=O)NC2CCOC2)N(C)CC2CC(O)C2)o1 C1(C2CC2)(COC)CN(C(=O)C(CN(C)C)NC(=O)C(C)CC2CC2)C1 C1(NCC2(COC)CCOCC2)CCCCC1N=[N+]=[N-] N1(C(=O)OC(C)(C)C)CCCC12CC(NC(=O)CC1CCCCC1O)C2 c1(C(=O)NCC(CNC(C(C)(C)SC)=O)(C)O)cnc(C(F)(F)F)nc1 Cc1nn(C)c(C)c1C(N1CCCC(CNC(=O)CN2CCC(C)(C)C2)C1)=O N1(C(C2CCCC(OC)C2)=O)CCOC2(CCCN(C(C3CNC(=O)O3)=O)C2)C1 N1(C(c2cc(C(C)C)[nH]n2)=O)CC2CC(NC(C34CCCC(C3)OC4)=O)CC1C2 N1(C(C(C)CC2CCCCC2)=O)CCC2(CCC2CNC(c2ccns2)=O)CC1 C1(C(N(CCC)CC)=O)CC(=O)CN1C(c1cc(CC)sn1)=O C1(C(=O)NC2C(CNC(C3CCC(=C)CC3)=O)C2)CCOC2(CCOCC2)C1 c1(C(=O)NC2CN(C(=O)Cc3c(F)cccc3F)CC2O)c(F)cc(F)cc1Cl Cc1nnc(O)c(C(=O)NC2CC(NC(c3c[nH]nc3C3CC3)=O)C2)c1C N=c1[nH][nH]c2ccc(-c3nc(-c4nnc(C(F)F)o4)nn3C3CCS(=O)(=O)C3)cc12 C1(O)(C(N2C(CNC(C3CC4CCC3C4)=O)CCC2)=O)CCCCCC1 S(=O)(=O)(c1c[nH]ccc1=NCC(CO)C1CCC1)N(CCC(O)C(C)(C)C)C C#CC1(C)CCCN(C(c2ncc(C(=O)OC)s2)C(=O)Nc2ccccc2Cl)C1 CC1(C#N)CN(C(=O)C(CO)NC(c2ccc(Cl)o2)=O)C1 Nc1[nH]c(=O)c(Cl)nc1C(=O)NCC1CCCCC1NC(c1cnns1)=O c1(NC(C2CC(O)CN2c2ccncn2)=O)c(Cl)cccc1Cl N1(C(N=c2cc(C)n(CCO)[nH]2)=O)CCc2cc(F)cc(F)c2C1 n1(C(C)(C)C(=O)NC2CCC(CNC(C3CC(C#N)C3)=O)C2)cc([N+](=O)[O-])cn1 C(C)(CC(C)NC(=O)C(F)(F)C1CCCCC1)NC(C1(C(C)C)CC1)=O C1(C(N(CC(=O)NCCCO)CCOCCO)=O)C2CCC(=O)C12 N1(C(=O)CCc2cscn2)CC2(C(=O)NCC=CCl)CC1CO2 c1(CNC(C2N(C)CCOC2)c2nnnn2CCF)cccc(C(F)(F)F)c1Cl c1(CNCC2(C(=O)Nc3ccc(Cl)c(Cl)n3)CC2)cc(F)ccc1Cl C1(NC(c2ncc(Cl)cc2Br)c2n(CC)nnn2)CCOC2(CCCC2)C1 C1(NC(CCNC(C)=O)=O)CCCN(C(=O)Cc2ccccc2C)CC1F c1(C(C)NC(C(c2cnn(C)c2)NC(=O)OC(C)(C)C)=O)ncc(F)cc1F C1(C(=O)NC(C2CCCCC2)CNC(C2(CCCC)CC2)=O)CC2CC2CC1C C(=O)(CC(C(N)=O)N(C)C)NC(C(C)N(CCC(C)C)CCC)=O c1(OC)cc(N)ccc1C(=O)NCC(CO)NC(=O)C(C(C)C)N1CCCCC1 N(C1CCc2cccc(Br)c21)C(=O)NC12CC(n3cc(C(C(C)C)O)nn3)C1C2 C=CC(C)CC(=O)N(C)CCN(C)C(C1C(c2ccncc2)C1(C)C)=O C1(O)(CNC(c2n(C)c(S)nc2)=O)CCCN(C(C2CN3CCN2CC3)=O)C1 C1(O)(C(C(=O)N(C)CC2(CN(C)C)CC2)F)CN(C(c2cnsc2)=O)C1 C(CCC(=O)N1CCC(C(=O)NCCCN(CC(C)C)C)O1)NC(C)=O N1(C(CC)=O)CCCCC1C(=O)N(CC1CCN(CCC2CC(C)=NO2)C1)CC C(=O)(C(C)CC(F)(F)F)NC1CN(C(C2CC(C(C)C)C2)=O)C(CO)C1 c1(C(N2CCCC(N(C(=O)CC3C(C)(C)C3(C)C)C)C2)=O)ccnn(C)c1=O CC(C)(C#N)CC(=O)N1CCC(O)(CCNC(=O)CCOc2cccnc2)C1 C1(N(C(CONC(C2(C(C)=O)CCC2)=O)=O)C)CCCC1C n1(CC)c(C(=O)NCC(C)(CO)NC(=O)CCCn2cccn2)cnc1O c1(CC(C2CCN(NCC3(O)CC3(C)C)CC2)C)ccc2c(c1)CCC2 C12(C(=O)OC)CCC(C(=O)NCCC3(O)CN(C(C4CCCO4)=O)C3)(C1)C2 c1(CCC(N2CCC(N(C(=O)CC3CC3)CCO)C2)=O)ccc(Br)c(F)c1 c1(C(N2C(CCNC(C34OC(C)C(C3)C4)=O)COCC2)=O)ccc(F)c(Cl)c1F C(=O)(CS(=O)(=O)CCC(F)(F)F)NC1CC(C)N(C(=O)C=CS(C)=O)CC1 Cc1cc(NC(=O)NCC2CC(NC(=O)OC(C)(C)C)C2)nc(Br)c1 N1(C(CSC)=O)CCC(C2CCCN2C(=O)Cc2cc(C(F)(F)F)nn2C)CC1 N1(C(CNc2n(C)cc(-c3ccc(C(F)F)cc3)n2)=O)Cc2ccc(F)cc2C1 c1(OC)cccc(C(F)(F)C(=O)NC2CCCC2NC(=O)Cn2nnnc2C)n1 C1(NC(C(C)(C)OC(C)C)=O)CN(C(=O)CC2CCC(C)(C)O2)CC2CCCC12 N1(C(C2C(C)C2)=O)CC(CNC(=O)CC2=NNC(=O)C2)C2(CCOCC2)C1 N1(C(c2ccc(CC(=O)OC)cn2)=O)CCCc2ccc(C(=O)OC)cc2C1 c1(C(=O)NCCNC(N2CCCCCC2)=O)ccc(F)cc1C(F)(F)F C#CCC(CC(F)F)C(=O)N1CCC(CC=C)(C(=O)NCC2CN3CCC2C3)C1 N1(C(C(=O)N(C)C)=O)CC(NC(=O)CCCOc2cccc(F)c2)C(C(F)F)C1 c1(C(N(CCN(C(C)=O)CC)CC)=O)ccc(Nc2ccc(C)cc2F)cc1C c1(C(N(CC(CNC(C(CSC)OC)=O)O)C)=O)cc(O)nc(N(C)C)n1 Cc1c(CCC(N2CCC(C)(NC(=O)C(C)Cn3cccn3)C2)=O)cnn1C CC1CN(C(C2(CCF)CCC2)=O)CC1(C)CNC(c1cc(Br)sn1)=O N1(C(c2cccc(OCCC)c2)=O)CC(NC(C2CC(O)CN2C)=O)C(C)(C)C1 C#CC1(CNC(=O)CC2CN(C(=O)Cc3ccccc3O)CCO2)CCOCC1 N(C(=NCCCCCCSC)NCc1noc(C)n1)CC1C(OC)CCC1 C(=O)(CCCCCC(C)O)NCC(C(C)(C)C)NC(c1c(CC)[nH]c(=N)s1)=O C1(NC(C2C(OC)C2)=O)CN(C(c2ccc(C)c(C)c2Cl)=O)Cc2nccn2C1 N1(C(C2(COC)C=CCN2C(=O)Cc2ccsc2C)=O)CC=C(CO)CC1 CC(C)CC(CNC(=O)C(CC1CCCC1)NC(c1ccoc1)=O)CO C1(C(N2CCC(OCC(=O)NCCC=CC)C2)=O)CCC(O)CN1C C1N=C(NCC2(CO)CC2)NC2CC12.C1(NS(C)(=O)=O)CCCCC1 n1(C(C)C)cnc(C(=O)NC2(CC(=O)NC3CC3c3ccnn3C)CC2)n1 C=CCC(CC)C(=O)NC1CCCC1NC(c1cc(OCC)n[nH]1)=O c1(-c2cn(C3CCC(C(=O)Nc4n(C)nnc4)CC3)nn2)ccc(Cl)c(F)c1 CC1CC(NC(C2(C(F)(F)F)CCC2)=O)CCN1C(=O)CCC1CC1 C(=O)(C(CC(=C)Cl)NC(C1CCC(F)CC1)=O)N(CCCC=C)C O=C1OC2CCN(C(c3onc4c3CCCC4)=O)C1C2 c1(OC)ccnc(F)c1C(N1CCCC(CNC(c2ccn(COC)n2)=O)C1)=O CN1CC(O)CC1(C)C(=O)NCc1cc(C(=O)NCC2=CCCC2)on1 C1(N(C(CC(C)OCc2ccccc2)=O)C)C2CN(CCC3CCCO3)CC12 N1(C(CC2CC(NC(C(n3ncc(C)c3)C)=O)C2)=O)CCCC2(CCO2)C1 C1(C(=O)NC(CNC(c2c(C)nn(C(C)(C)C)c2)=O)C2CC2)CC(C)(C)CN1C c1(C(N(CC(CNC(C(c2ccnn2C)C)=O)O)C)=O)cc2c(nn1)CCCC2 C1(C(=O)NC(CCCC=C)C2CC2)CC12CCN(C(=O)C1=CCSC1)C2 C1(C(N(CCCN(C(C(C2CCCCC2)OC)=O)C)C)=O)C(C#N)C1(C)C c1(C(N2CCCC(N(C(COCCCC)=O)CCF)C2)=O)cnn2ncccc12 CC1CN(C)C(C)CC1CCNC(=O)CN(C(C1(C)C=CCCC1)=O)C1CC1 Cc1ccc(Br)cc1CC(=O)NC12CC1CN(C(=O)C(C)Cc1ccco1)C2 N1(C(CC2(OCC)CC2)=O)CC(NC(c2ccn(C)c2)=O)CC(O)C1 C=CCCC(CC(C)C)C(=O)N1CCC2(C1)CN(C(c1cnnn1C=C)=O)C2 c1(CC(=O)N(CC(CC)NC(c2nc(C3CC3)no2)=O)C)cccc(C)c1C C1(NC(CNS(C)(=O)=O)=O)CCOC1CNC(=O)CCCc1ccsc1 c1(C(=O)NC2CCCC(NC(C3N(C)C(=O)OC3)=O)C2)nccc2ncncc12 N1(C(C(CCC)OC)=O)CCN(C(C2CCCC2OC)=O)CC1C1CCCC1 C=Cc1ccc(C(=O)NCC2COCC2NC(=O)C(CCOC)OC)cc1 CC(C(=O)NCC1CCC2(CN(C(C3(C(C)(F)F)CC3)=O)C2)O1)C(F)(F)C(F)F c1(NCC(CNC(COCCCC(C)C)=O)O)ncnc2sc([N+](=O)[O-])cc12 C1(C2CC2)(C(=O)NC2C(C(=O)OC)CC2)CN(C(=O)C(C)N=[N+]=[N-])C1 CCCCS(=O)(=O)NCC(=O)NC(CN(C(=O)Cc1csc(CC)n1)CC)CC c1(C(N2CCC(CNC(C(CC)(CC)CC)=O)C2)=O)cnc2ccc(C)cc2c1 C(c1ccccc1C)=CCN(CC(N1CCN(CC)CC1)=O)CC(C)C N#Cc1cc([N+](=O)[O-])ccc1C1CCN(Cc2cn(C3CCNC3=O)nn2)CC1 c1(NC(N2CC3C(C)C3C2)=O)cc2c(cc1Br)OCCO2 c1(OCCC)nc2ccccc2cc1C(N1CC2CC1(CNC(=O)CSC)C2)=O C1(NC(C2CCOC2)=O)(CNC(C2CCC(O)CC2)=O)CCCCCC1 Cc1ccc2c(C(=O)NCC3(F)COCCN(C(=O)CNC=O)C3)ccnc2c1C c1(NC(CCc2c[nH]c(=N)[nH]2)=O)cnc2ccccn12.C12CC3CCC1N3C2=O CC1CN(C(=O)COCCCF)CC1C(N1CCC(C(C)(C)C)CC1)=O N1(C(C=C(C)C(F)F)=O)CCC(N(C(=O)CC2CCC(C(F)(F)F)O2)CCO)C1 c1(NC(=O)NC2CC(=O)N(c3cc(Cl)cc(Cl)c3)C2)[nH]cc2c1CCCC2 C(=O)(C1=CC2(CCOC2)C1)NC(CC(C)NC(c1c(C)nc(CC)nc1C)=O)C C1(NC(=O)OC(C)(C)C)CCc2[nH]c(=NCCC(C)(C)C3CC3)sc2C1 c1(C(=O)NC2C(NC(c3c(CC)n(C)nc3)=O)COCC2)cccc2ncnn12 CCCCC(C)C(=O)N1CCC(N(C(=O)CCc2ncccn2)CCC)C1 N1(C(Cc2cnc(C)s2)=O)CC(C(=O)N(CC(=O)NC(C)C)C)C2(CC2)C1 c1(C(=O)NCC2C(NC(C(C)OC)=O)CC2)ccc(O)cc1C(F)F CCCC(CNC(C1CC(=O)C1(C)C)=O)C(=O)NCc1cnc(C)n1CC C1(NC(C2CC=C(C)CC2)C)CCCN(S(N)(=O)=O)C1 C(CC1CC1)(C(=O)NC1CCSC1)NC(=O)CCC1CC1 C1(CC)CN(C(c2ccc(CNC(=O)C(=O)NC(C)C)o2)=O)C(CC)CO1 N1(C(CCCC(C)C)=O)CCCN(C(=O)COCC(C)(C)C)C(C)C1 C1(CC(=O)NCC(C)(C2CC2)NC(CC(C)c2ccncc2)=O)CC(C)(C)CO1 C(CC(CNC(=O)C(C)NC(=O)NC)NC(=O)C(CO)N(C)C)OC C(CCCOC)(C(=O)N(CCF)CCOC)NC(C(C=C)CC)=O C12(C(=O)OC)CCC(CC1)N(CCC(=O)Nc1cc(Cl)ccc1Cl)C2 Cc1c(C(=O)NCCC(C)NC(c2sccc2F)=O)nn2c1CCCC2 C(CC1C(=O)N(C)N1)OCC.c1(CC2CC3(CSC3)C2)cccc(C)n1 c1(C(N(C2(CC(=O)NC34CCCCC3C4)CC2)C)=O)ccc(O)nn1 CC(C)CC(C)(CNC(C1CCC(C(C)C)CC1)=O)NC(=O)C(O)CC(N)=O N1(CC2CN(C(C(=O)N(CCO)CC)=O)CC(C)C2)C(=O)c2ccccc2C1=O C1(NC(C(C)OCC)=O)CCCN(C(=O)Cc2cc[nH]c2)CCC1 N1(C(COC(CC)CC)=O)CC=CC(C(=O)NCC2(O)CC2)C1 C=CCCC(=O)NC(CNC(c1csc(CC2CCC2)n1)=O)CCOCCSC C=CCCC(O)CNC12CC(n3cc(CNC(C4CCCC45CC5)=O)nn3)C1C2 c1(C(=O)OC)c(NC(C2CC3CC3N2Cc2cncc(Cl)c2)=O)cccc1Br Cc1ccc(CCC(=O)NC2CCC2C)o1.C12(CCCC1)C(=O)NCC2 CC1(C)CC(O)(CN2CCC(F)(CCCCn3nnnc3C(F)(F)F)C2)CO1 C1(OCC)CCCC1NCC(C1CCCCC1)(C)C#N c1(C(c2n(CC)nnn2)NCCCCF)cccc([N+](=O)[O-])c1C c1(C(=O)NC2C(NC(c3cn(CC=C)nc3)=O)CCC2)cc[n+]([O-])cc1 C1(NC(C(CC#C)O)=O)CCCCN(C(=O)CC2CSCCO2)C1 C1(CNC(CNC(=O)NC)=O)CCN(C(=O)CC2CCCC(F)(F)C2)C1(C)C C(=O)(CC(C(F)F)NC(c1ccnnc1O)=O)N1C(CC)CC(C)C1 C1(O)(CC(=O)NC2C3CN(C(C4CCC(NC(C)=O)CC4)=O)CC32)COC(C)(C)C1 CC1CN(C(=O)CCCC2CCC2)CC(C)N(C(c2cc(N)cc(F)c2)=O)C1 N1(C(C(C2CCOC2)OC)=O)CC2(CCN(CC3CCCCCC3)CC2)C1 c1(C(=O)NCC=CC(=O)NCC(CO)OC)cc(C2CC2)oc1C C1(CC)CCN(C(=O)CC(C)(C)N(C(=O)CCOCC(F)F)C)CCO1 C(C)(C)(CC(=O)N1CCOC(C2CN(C(=O)CN(C)C(C)C)C2)C1)OC C(=O)(C(C)(C)C1=CCS(=O)(=O)CC1)NCC1C(NC(C(=O)NCC)=O)CCCC1 N1(C(C(C)CCO)=O)CC(F)(F)CC1(C)CNC(C1CSCCS1)=O N1(C(C(CCC)OC)=O)CC2CCC(C(=O)NCC3C(C)(C)C3(C)C)(C2)C1 C1(CNC(=O)C(N2CCCC(N3CCCOCC3)C2)=O)C(F)(F)C12CC2 C#Cc1cc(Nc2nc(F)ccc2NC(=O)C2CC2)ccc1Cl C1(NC(C(C)OCC)=O)CC2CC(NC(=O)CCc3ccccc3)CC12 CN1CCN(C(=O)C2=CCSC2)CC1C(=O)NCC12CCC(CC1)CC2 C(=O)(C1=NOC2(CCOC2)C1)NCC12C(CN(C(CNC=O)=O)C1)C2 C1(N(C(C(F)OC)=O)C)C2CN(C(C3(F)CCCC3)=O)CC12 CCC(C)(CC)C(=O)NCC1CC(NC(C2(C3CC3)CC2)=O)C(O)C1 CCC(C(=O)NC(C)CC1CN(C(=O)CNC(=O)CCC(C)C)C1)C(C)C N1(C(c2sccc2Br)C(=O)Nc2ccc(OC)cc2)CC2CCC1C(O)C2O N1(C(CCC(C)SC)=O)CC(C)CN(C(=O)Cc2c[nH]c(=N)nc2O)CC1C C1(NC(CC(C)N(C(c2cnn(CC)c2C)=O)C)=O)CCC2(CCC2)C1 N1(C(CCCOCCC)=O)CCC2(CC1)CCN(C(C1CCCN1C)=O)CC2 C1(C)(CC(=O)N(CCOCCN(C(=O)C(C2CC2)C2CC2)C)C)CCCO1 CCCCC(C)(F)C(=O)N1CCC(CNC(=O)CC2CCCCC2O)C(C)C1 CCC(C(=O)NC1CC(NC(c2cc(O)nn2C)=O)C1)C(C)(F)F N1(C(CC(C)C)=O)CCC(NC(=O)CN(C)C(c2ccsc2)=O)C1(C)C c1(C(N2C3C(NC(C(C4CC4)OC)=O)CC(CC3)C2)=O)nn2cccnc2c1Cl c1(OC)ccccc1C(N1CC(O)(C(C)NC(=O)COc2ccc(F)cn2)C1)=O S(=O)(=O)(c1ccc(Br)c(Cl)c1)NC(C)C(=O)NCCc1ccccc1F C1(C)(NC(c2c(C)cco2)=O)CCCN(C(=O)CC2NC(=O)NC2=O)C1 C12(CNC(c3n(C(C)(C)C)ncc3)=O)COC(CNC(C3CC3(F)Cl)=O)(C1)C2 N(C(=NCCF)N1CCC(c2nncs2)C1)Cc1cc(COC)no1 Cc1cc(C(=O)NCC2CCN(C(C3CCC(=O)O3)=O)C2)c(Br)cn1 c1(NC)cc(C(=O)NC(CNC(c2occc(=O)c2OC)=O)CO)cc(Cl)n1 C1(NC(=O)NCC23C(C)(C)OCC2C3)CCc2c[nH]nc2C1 c1(C(C(=O)NC2COC2)N(C(c2ccncc2)C)C)cc(F)nc(F)c1F c1(C(=O)NC2(OC)CCC(C(=O)O)CC2)c(C)oc(C)c1S(N)(=O)=O c1(C(=O)NCCC(C)(C)NC(Cc2c(C)ncs2)=O)[nH]cc2c1CCCC2 N1(CCC(=O)NC(CCC)C(=O)OC)CCCC(F)(F)C1 c1(C2(NC(=O)NCC3C(SC)COC3)CC(F)C2)ccccc1F Cn1ccc2cc(C(=O)NCC3CN(C(C4CC4CN(C)C)=O)C3)cnc12 c1(C(=O)NC2CC(N(C(C(C3CCOCC3)C)=O)C)C2)cccn1C C1(NC(C2C(C)C2)=O)CC2CC1N(C(C1(c3ccc(F)cc3)CCCCC1)=O)C2 c1(C(OC)NC(=O)N(CCC#N)C)ccc(F)cc1C(F)F c1(NC(C2(CN(C(CC(C=C)c3ccccc3)=O)C)CC2)=O)ccc(N)c(O)c1 c1(C(=O)NC(C(C)NC(C2CCCN2C(N)=O)=O)CO)cc2n(c1)CCSC2 N1(C(C(C(CCC)NC(=O)C(C)SC(C)C)O)=O)Cc2cccc(F)c2C1 CC1(CNC(=O)Cc2ccc(CO)cc2)CCCN1C(c1ccsc1Cl)=O Cc1cc(C(=O)NCC(C)NC(=O)CC(C)(C)C#N)cc(C)c1F C1(C(=O)NC2(c3ccc(F)cc3)COC2)CC2CC1C1CC21 c1(C(N2CCC(NC(c3c(CC)ncs3)=O)C(O)C2)=O)cc(F)cc2ccoc12 C1(c2cccc(NC(C(=O)Nc3ncc(C)cn3)=O)c2)CCC(C)C1(C)C C1(NC(=O)NCCSC)COCCC12CN(C(=O)OC(C)(C)C)C2 N1(C(CCC=CC(C)C)=O)CCC(C(=O)NCCc2ocnc2CO)C1C CC(C)(C)CCCCC(=O)N1CC=C(CC(=O)N2CCC3CCCCC3C2)CC1 C1(CNC(c2ccc(OC)o2)=O)CC(NC(=O)CCc2ccc(Cl)nc2)C1(C)C c1(N(CC(F)(F)C(F)(F)Br)Cc2ccc(OCCCCC)cc2)ccc(C#N)n1C c1(N(c2ccc(F)c(Cl)c2)C)ncnc2c(Br)nn(C)c12 c1(OC)cccc2sc(NC(CN(C)C)CC(C)C)nc12 C1(NC(C(C=C)O)=O)CCN(c2cc(C)nc(CC)n2)C12CCCC2 C(=O)(C(C)CCCCCC)N1C(C)(C(N2C(CC#C)COCC2)=O)C=CC1 c1(C(=O)NCCC(C)(CC)NC(C(CC)OC)=O)cnc(OC)nc1C(F)(F)F c1(OC)ccc(-c2ccc3c(c2)CN(C(c2ncccc2C)=O)C3)c2cn[nH]c12 N1(C(Cc2ccc(C(=O)OC)cc2)C(=O)OC)CCCN(c2ccccc2C)CC1 N1(C(C2(OC)CC(C)(C)C2)=O)CC2CCC(C(=O)NCc3ncco3)(C2)C1 C1(CC(=O)Nc2c(OC)nn(C)c2)CC2(C1)CN(C(c1ccsc1Cl)=O)C2 CCCCCCCCC(=O)N1CCN(C(C2CC3(C2)CC(O)C3)=O)CC(C)C1 c1(OC)n[nH]cc1C(=O)NCC=CCNC(C1CCC1C)=O N1(C(c2cnc(OC)s2)=O)CC2CC2(CNC(=O)CCC2CCC(C)O2)C1 N1(CC(CCC(=O)NC)C(=O)OC)CCn2c(-c3cccs3)nnc2C1 n1(CCCNC(=O)COC(=O)CO)cc(-c2cccnc2)nn1 C=Cc1cncc(C(=O)NC(C2CCN(C(C3CCC(C)(C)CO3)=O)CC2)C)c1 c1(CC(=O)N(CC(C)NC(c2ccnc(F)c2F)=O)C)cc(F)cc(F)c1 S(=O)(=O)(c1nc(N2CCCOCC2)ccc1Br)N1CCN(CC(C)(C)F)CC1 C1(C(C)NC(c2n[nH]cc2NC(N)=O)=O)CCCN(C(=O)OC(C)(C)C)C1 c1(C(=O)NC2C(C)(C)C(CNC(=O)CSC(F)F)C2)cc2sccc2[nH]1 c1(C(=O)NC(CCNC(C(c2cc(C)sc2)(F)F)=O)C)cc2c(Cl)cccn2n1 C(=O)(CCCCCC#N)NCC1N(C(Cc2ccc(OC)nc2)=O)CC1 C1(O)(C(C)NC(C2CC2c2ccc(Cl)s2)=O)CN(C(C2CC(O)C2)=O)C1 CC(C)CC(O)C(C)C(=O)NCCC(C)(C)NC(=O)C1=C(Cl)CCCC1 N1(C(CNC(C)=O)=O)CCCCC(CNC(=O)CC2CCN(OC)CC2)CC1 C1(CC(=O)NC)CN(C(=O)Cc2c(C)cccc2Cl)CCN1C(=O)C(F)OC C(CNC(C1CC1[N+](=O)[O-])=O)(CC(F)(F)F)NC(c1c(Cl)cc(C)s1)=O C1(C(C(=O)NC)F)CCN(C(c2cnn(C(F)F)c2)=O)C1 C(=O)(C(F)(F)C(C)(C)O)N1CC(CCC)N(C(=O)CSCc2cccnc2)CC1 C1(C(=O)NC(C)C(C)(C)C#N)CCCCCN1C(=O)CCCN(C)C C1(N(C)C)COCCN(C(=O)Cn2cnc(C(N)=O)n2)C1 c1(C(=O)NCC2N(C(C(n3ccc(C)n3)C)=O)CC2)cccnc1OCCO N1(CCN(C(c2ccc(CC)o2)=O)C)CCN(C(=O)C(c2cnn(C)c2)=O)CC1 C1(OC)COc2c(NC(=O)N(C)Cc3ccc(SC(F)(F)F)cc3)cnn2C1 N1(C(c2c(C)nc(C3CC3)o2)=O)CCCC(C2CC2NC(=O)CNS(N)(=O)=O)C1 Cc1c[nH]c(C(=O)NC(C)(C(=O)NCC(C)S(N)(=O)=O)C2CCC2)c1C C(=O)(C1=CC(O)C(NC(=O)CC2CC(C)(C)CO2)C1)N(C(C)CO)CC C1(C(=O)NC2CCCC2CNC(c2cnc(Cl)s2)=O)(COC)CC1(F)F c1(N(C2CCCSC2)C)nc(=N)[nH]c(=NC(CF)c2ccc(F)cc2)[nH]1 C1(c2nnnn2C2CCC2)(NC2C(CC(=O)OC)CNC2)CCN(C)CC1 Cc1nc2n(n1)CCC(C(N1CC3CC1(c1cn(C4CCCC4)nn1)CO3)=O)C2 Cc1cc(C(=O)NCC2CC3CCC2N3C(c2ccc[nH]2)=O)c2c(C)noc2n1 N1(C(c2n[nH]c(C)c2Cl)=O)CC(N=c2[nH]cnc3cnn(C)c23)CC2(CCC2)C1 C(=O)(CC(C(C)=O)N1CCC(n2ncc(N)c2C(F)F)CC1)OCC C1(C(N(CC(CC)C)C)=O)(CCOC)CCN(C(c2ncc(C)cc2C)=O)CC1 C1(N(C(C(C)Cc2ccccn2)=O)C)CCCCC1N(C)C(c1cnc(Cl)s1)=O c1(C(=O)NC(CCNC(CCCNC(C)=O)=O)C)cc(Cl)c2cc(Cl)ccc2n1 CCC(C)(CNC(=O)CC1CCC(NC(=O)C(C)=NOCC#N)C1)C(N)=O C(CC1CCC1)(C(=O)N=c1ccn(C(C)(C)C)[nH]1)NC(Cc1cc(CC)no1)=O C1(NC(c2c(C)nc(C)[nH]2)=O)CCCC(NC(C2(CS(N)(=O)=O)COC2)=O)CC1 C1(C(=O)NC(C(C)C)C(C)NC(=O)C=Cc2ccnn2C)CCC2(CC1)CC2 c1(CN(C(=O)Cn2cc(CN)nn2)Cc2c(OC)nccc2)c(C)cccc1Cl CCN=c1[nH]c(C(N2CCCC(C)(CNC(C3CC3CCOC)=O)C2)=O)cs1 N1(C(c2ccnc(C)c2Cl)=O)CCC2(CC1)CC2NC(=O)CCc1nncs1 C(=O)(CCC(N)Cc1ccccc1)C1C(CC(=O)OC)C1 c1(C(=O)NCC(C)NC(c2cnc(SC)s2)=O)cc(C(N)=O)cc(F)c1 C(=O)(C(C)(C)CC(=O)N1CCC(CNC(=O)C(C)OCC2CC2)C1)OC C(c1ccc(CC(C)C)cc1)=CC(=O)NCCCCN(C(CCCCOC)=O)C C1(C(=O)NCCC2CCN(C(c3cn(CC)nn3)=O)CC2)CCC2(CCC2)C1 CC1(C)CCCCCC1NC(c1ccc(C(F)(F)C(F)(F)F)s1)c1nnnn1C c1(C(C(=O)NCC(C)CN(C(=O)Cc2cscn2)C)C)cncnc1 C1(C(=O)NCc2c(CC)nco2)CN(C(=O)COCC2CCOC2)CCC1(C)C C(C(CC1CC1)C(=O)NC1CC(O)C1)NC(CC1(C)CCC1)=O C1(C(=O)NC(C2(O)CCN(C(C3(O)COC3)=O)C2)C)CCC2(CCC2)CO1 C(=O)(C(CCc1ccsc1)NC(c1c[nH]cc1CCO)=O)OC c1(C(N(CCOC)CCNC(c2c(C)cnn2C(C)C)=O)=O)cc(C)nc(O)n1 C1(CNC(c2cc(C)no2)=O)CCN(C(=O)C(C)NS(C)(=O)=O)CC1C c1(C(=O)NCC23C(CN(C(CCCCC#C)=O)C2)C3)sc2[nH]cnc(=O)c2c1C Oc1ncnc2c1CCN(N1CCCC(c3n[nH]cc3I)C1)CC2 N1(C(CCC(C)C)=O)CCN(C(C2CC3(C2)CC3F)=O)CC2(CC2)C1 Cc1cc(C2CCCN2C(C2(C(=O)N(c3ccccc3Br)C)CC2)=O)ccn1 c1(C(N(C2CCCN(C(=O)CC3CCCCO3)C2)CC)=O)cnn2c(C)cccc12 n1(CC(=O)OC(C)(C)C)ncc(Cl)c1C(=O)NC1CCC(NS(C)(=O)=O)CC1 C(=O)(C(CC)C(=O)NCC1CCCN(C(C2CCCCO2)=O)C1)OCC C(C(C)(C)C(=O)N1CCC(CCC(=O)N2CC(CF)C2)C1)OCC CCCC(CC)C(=O)NC1(C(=O)N(C)CC2(F)CCCC2)CC(CO)C1 C#CCC(C(=O)NCCC1CCCN(C(c2nnccc2C)=O)C1)C1CC1 C1(C(=O)NC(CC#C)C(=O)NC)C2CC3C(C2NC(C2CC(C)=NO2)=O)C13 N1(C(C2CCC(C(=O)OC)CC2)C(=O)NCC)CCOc2c(OC)cccc2C1 N1(C(c2cnc(SC)[nH]2)=O)CCC(NC(c2nnccc2C)=O)C2(CCC2)C1 N1(C(CNC(CC(C)(C)C)=O)=O)CCCC2CN(C(c3sccc3F)=O)CCC12 c1(NC(C(CC)N(CC)CC)=O)ccc(N=S(C)(C)=O)s1.C12(CCC1)C(=O)N2 c1(CNC(C(N2CCCC(C(=O)OCC)C2)=O)=O)oc2ccccc2c1Cl CCCCC(CC(=O)NCC1(O)CCCC1)NC(=O)C=CC1CCOC1 c1(C2(C(=O)NC3C(CNC(C(C)N4CCCC4)=O)CCC3)CC2)ccc(O)cc1 C1(CC(=O)NC2CCN(C(c3c(CCC)n[nH]c3)=O)C2)(OC)CCCCC1 c1(CCN(C)C)cccc(C(=O)NCCCN(C(=O)CCC2CCCC2)C2CC2)c1 C(C(CCCC)NC(=O)C=CC(=O)NC1CCOCC1)NC(C(F)=CCC)=O C12(OC)CCC(C(N3CCC(CCNC(=O)CC4CC(=O)NC4=O)C3)=O)(CC1)C2 c1(C(N2C(CC(=O)Nc3cc(N(C)C)ncn3)COCC2)=O)cc(Cl)ccc1Br C1(NC(c2cc(-c3ccc(Cl)cc3)ns2)=O)C2CN(C(=O)CC3C=CCC3)CC12 N1(C(c2cn(CCOC)nn2)=O)CCCC(CO)(NC(C2CCC2(F)F)=O)C1 C(=O)(C(O)CC(C)(C)C)NC1(CC=C)CCN(C(=O)CC(C)(C)O)C1 N1(C(=O)CC2CCC2)CC(C2CN(C(C3CC34CC(F)(F)C4)=O)C2)C1 N1(CC)CCCN(C(=O)C(C2CN(C(C3CCS3(=O)=O)=O)C2)OC)CC1=O C1(Cn2cc(CCCCC)nn2)CN(C(c2cnc(C)cn2)=O)CCO1 N1(C(CCCCCN(CCCC)S(C)(=O)=O)=O)CCCCC1C1CN(C2CCC2)C1 N1(C(C2C3CN(C(CCC(C)OCC)=O)C2C3)=O)CC2COCC(C2)C1 C(=O)(C(CCC)CC(C)C)NC(CCCC)CNC(c1cnccn1)=O c1(C(N(C2CCN(C(C(CC(C)C)F)=O)C2)C)=O)ccc2c(c1)C(=O)C(=O)N2 c1(-c2nnc(-c3ccc(C4(c5cccc(Br)c5)CC4)cc3)o2)csc2cncn12 N1(C(C(C)N2CCC2)=O)CCCC(NC(c2ccc(F)c(Cl)n2)=O)CC1 C1(NC(c2c(CC)occ2C)=O)CS(=O)(=O)CC1NC(c1cc(F)ccc1O)=O CC1CCCN(C(=O)C(O)CCNC(C2CN3CCN2CC3)=O)CC1 Cc1nc2c(s1)CC(C(=O)NC1(C3CCCN3C(c3csc(=N)[nH]3)=O)CC1)CC2 CCC(O)C(F)(F)C(=O)N1CC(NC(c2cnc(C3CCC3)nc2O)=O)C1 C1(C(N2CCC(C)(CNC(c3c(C)noc3N)=O)C2)=O)OCCN(C)C1=O c1(C(=O)NCCC(=C)CNC(C2CC2CC(C)C)=O)ccc2nonc2c1 c1(C(N(CC(C)CNC(=O)C(=O)NCC2CC2)C)=O)cn2c(n1)CCC2 c1(C(=O)NC2CC(C(C)NC(Cn3ncc(CC)c3)=O)C2)n[nH]cc1[N+](=O)[O-] c1(C(=O)NC(C)CNC(c2ccc(N)cc2)=O)cccn2nnnc12 C1(CNC(C2(C)CCCOC2)=O)CN(C(=O)CCOC2CCC2)C2(CCC2)C1 c1(C(N(C(CNC(C2C3CC4C(C3=O)C24)=O)C2CC2)C)=O)ccc2cnnn2c1 N1(C(=O)C=CCc2ccccc2)CC2(C1)CN(C(C1(c3cccc(F)c3)CC1)=O)C2 c1(C(C(N2C3C(NC(C=CC(=O)OCC)=O)C(C3)C2)=O)C)cc(F)cc(F)c1 Cc1nn(C)cc1-c1ccc(NC(c2cc(Cl)sc2Cl)=O)cn1 Cc1cc(C)c(C(=O)NC2CC(CNC(=O)CCn3ncn(C)c3=O)C2)cc1C C1(C(=O)NCC(=O)NC2CC2)CC12CN(C(c1ccn(C3CCCCO3)n1)=O)C2 N1(C(CCN(CCCCC)C)=O)CCC(C2(NC(=O)CCCNC(C)=O)CC2)C1 Cc1cc(C(=O)NC(CNC(c2ccnn2C2CCCC2)=O)C2CC2)ncc1N C1(CCCC)CN(C(C2CC2C2CC2)=O)CCN1C(=O)Cc1csc(Cl)n1 C1(C(=O)NC(C(CO)NC(c2nc(C)sc2)=O)C)CCC(C)(C)OC1 c1(C(N2CCCC2c2cc(C)nn2C)C(=O)NCCC)sc2ccccc2c1C N1(C(CNC=O)=O)CCC2(CCOC2)C(CNC(=O)CCN2C(=O)CCC2=O)C1 Cn1ncc2c1CC(C(=O)NCC(C1CCC1)NC(C1C3COCC13)=O)CC2 N1(C(c2c(C)n(C)nn2)=O)CCN(C(=O)CNC(c2ccccc2)=O)C(C)C1 c1(C(=O)NCc2ccc(C(N3CC(C4CCCO4)C3)=O)s2)ccccc1C1CC1 c1(C(=O)NCCCN(C(c2cccc(CC)n2)=O)CCO)cc(O)cc(=O)o1 Cc1ccc(C=CC(=O)NC2CC2NC(C2CCC(OC(C)C)CC2)=O)c(C)c1 CC1(C)CC(CNC(c2scnc2Br)=O)N(C(=O)CN2CCCC2=O)C1 CCC(CNC(c1ncn(C)c1C)=O)(CC)C(=O)N1CCC(CN(C)C)C1 N1(C(C(C#C)(C)C)=O)CCN(C(c2cc3c(s2)CCC3)=O)C(C(F)F)C1 Cc1nc2ccccn2c1CN1CC2CCCC2C1 N1(C(c2cnn(C)c2F)=O)CCN(C(C2CCN(CCF)CC2)=O)C2CC12 N1(C(C(CC=C)C(C)C)=O)CC=C(C(C)(C)C(=O)N2CC3CC(C2)C3(C)C)C1 N1(C(Cn2c(C(C)C)ncc2)=O)CCCN(C(=O)Cn2cncn2)CC1 c1(-n2cc(CN3CC(CNC(CC4CCC(=O)C4)=O)C3)nn2)cc(F)ccc1Cl C(=O)(CC(C(C)C)NC(C1(CCC)CC1)=O)NC(C=C)C(F)(F)F CCC(CNC(C1C(CN=[N+]=[N-])C1(C)C)=O)(CC)NC(=O)C(C1CCC1)OC c1(C(=O)NCC2CC(F)(CNC(C3CCN(C)C3=O)=O)C2)cccc2sncc12 C1(CNC(CS(CC)(=O)=O)=O)CC2OCCC2N1C(c1ccc(C)c(C)c1)=O N1(C(CCC(CC)NC(=O)CC2CCOC2C)=O)CCCC2CC1C2(C)C CCCC(O)C(=O)N(C)CC1CCN(C(C2(C)CCSCC2)=O)C1 c1(N2Cc3c(ccc(Cl)c3)C2)nc(=NCC2CN(c3ccccc3)C2)[nH]c2c1CCC2 C12(CCNC(CCCNC(C)=O)=O)CCC1CN(C(c1c[nH]c(=N)nc1C)=O)C2 N1(C(CC2CCC(C)C2)=O)CCC2(CC1)C(NC(=O)CC1CN(C)C1)CS2(=O)=O Cn1c(CC(=O)NC(Cn2ccnn2)C(=O)NCc2nccs2)nnc1S c1(SC)cn(C)nc1C(=O)NC1CN(C(=O)C=Cc2cocn2)C1 C1(C(=O)OC)CCN(S(=O)(=O)N2CCC(C)(C(=O)COC(C)=O)CC2)C1 c1(C(=O)NCC2CC(NC(CC3C(C)OCC3)=O)C2)ccc2oncc2c1 C(=O)(CCOC)NCCN(CC(=O)OCCCC)C(=O)CC1CCOC1 c1(C(=O)NC2(CNCc3cccc(N(C)C)c3)COC2)c(O)ccc(Br)c1O C1(CC(NOCCOCC#C)=O)CC(NC(=O)C=Cc2ccncc2)C1(C)C c1(OCC)ccccc1C(=O)NC(C)(C)CCCNC(=O)C(CC)OC c1(CCNC(CCCn2cc(C(N3CCCC3)(C)C)nn2)=O)ccc(F)c(Br)c1 c1(C(=O)NCCCCNC(c2cnncc2C(F)(F)F)=O)ccc(O)c(Cl)c1 C1(O)(CNC(=O)C=C2CCCC2)CC(CNC(c2ccnn2CC(F)F)=O)C1 N1(C(C2C(CC(C)(C)C)C2)=O)CCCCCC(NC(=O)CC2CCC(=O)O2)C1 C#CCC(CC#C)C(=O)NC1CN(C(C2(N3CCCC3)CCC2)=O)CC1OC C(C(COC)CC(=O)NC1CC(O)CN(C(=O)CCCc2cnccn2)C1)OC c1(C(=O)NC(CC)CN(C(=O)C(CCO)OC)CC)ccnc2c1cnn2C c1(CNC(c2cc3cc(Cl)ccc3o2)C)c(Cl)c[nH]c2nccc1-2 C(=O)(C1=C(Cl)CCOC1)NCC12N(C(CCOCCN(C)C)=O)C(CC1)CC2 N1(CC)CCC(NC(=O)CCCn2cc(C3CCCC3)nn2)C(C)C1 c1(C(N2CCN(C(CN(C(CC(C)F)=O)C)=O)CC2)=O)cc2[nH]ccc2s1 C(=O)(C(F)(F)CC1CC1)N(C1CCN(C(C2CCCCC2C)=O)CC1)CC C#CCCC(O)C(=O)NC(C)CNC(c1cc(CC)ccn1)=O C1(CC(=O)NCC2CCC(NC(C3CC(C)C3)=O)CC2)CCC(C)(C)CO1 c1(NC(=O)NCC2OCCC2CC2CC2)ccc(F)c(N2CCOCC2)c1 C1(NC(COCCC=C)=O)(CNC(=O)C(c2ccccc2F)C)CCCCC1C CC1CN(C(=O)C(C2CCCCCCC2)O)CC(C)N1C(c1cnsn1)=O S(=O)(=O)(c1cnc(NCCc2ccccc2F)c(Cl)c1)NCC1CCCC(C)O1 N1(C(C2C(C(C)C)C2)=O)CCOCC(CNC(=O)CCc2ccc(Cl)c(F)c2)C1 Cc1ccc(CS(=O)(=O)NC(c2cccc(N3CCCC3=O)c2)C)c(C)c1 C12(C(=O)NCC3C(CNC(c4cn(CCOC)nc4)=O)C3)CCC(SC)C1C2 c1(-n2cc(CN(CC(=O)OC)C(=O)CC3(CS(C)(=O)=O)CC3)nn2)cccnc1Br Cc1csc2c(C(=O)NCCCNC(=O)C(n3cc(Br)cn3)C)ncnc12 N1(C(CC(C)C2CCCO2)=O)CC(C)(C)OC2(C1)CN(C(c1cc[nH]c1)=O)C2 CC1(C)CC(NC(=O)Cc2ccco2)CCN(C(=O)Cc2ccc(Cl)c(Cl)c2)C1 C1(CC(=O)N(CC(O)C2CCC2)C)CCCN(C(C2(C)CCN(C)C2)=O)C1 c1(C(=O)NC(CN(C(C(CC)N(C)C)=O)CC)C)sc(C)nc1C(F)(F)F c1(C(N2CC(NC(=O)CC3CC4CCC3O4)C2)=O)cnn2c1OCC(O)C2 Cc1noc(C)c1-c1cn(CC2COCCN2C(C2(C)CCCCC2)=O)nn1 Cn1ncc(C(=O)NC2CCCN(C(c3cccn3Cc3cccs3)=O)C2)c1Cl c1(C(N2CCCC(NC(COCCCCOC)=O)C2C)=O)ccn2nccc2n1 C1(NC(Cc2c(C)ocn2)=O)C(C)(C)C(NC(=O)C(O)CC2CCCC2)C1(C)C c1(OCCCOC)ccc(C(=O)NC(C)CCNC(=O)CCC=CC(C)C)cn1 C(C1=CCN(C(=O)CCc2nc(C)c(C)o2)CC1)NC(c1c(SC)cccc1)=O C1(NC(C(CCC)O)=O)COC2C(NC(=O)C(C(C)C)n3cccc3)COC12 C(c1ccccc1C(F)(F)F)=CC(=O)NC(CSC)C(=O)N(C)CCO C1(C(N2C(C)CN(C(c3cccnc3)=O)CCC2)=O)CCc2nnc(O)n2C1 C(=O)(C1Cc2ccc(Cl)cc21)NC(C(C)NC(=O)CCCCc1cnn[nH]1)CO C#CC1(C(=O)NC2CCC(C3CC3)C2)CCN(C(c2cnc(N(C)C)nc2)=O)C1 Cc1cc(C(=O)NCC(CNC(c2cscc2Cl)=O)CO)nc(O)n1 C1(CNC(C=C(CC)C)=O)CN(C(=O)Cc2cc(F)cc(F)c2)CC12CC2 CC1(C)CCCC(CCNC(=O)NCC(N2CCCCC2)C2CCCCC2)C1 C1(NC(C(C)C2CC2)=O)Cc2ccccc2C1NC(c1cnsn1)=O C(=O)(CCC(C(=O)NC(C)(C)C)N1CCC(C(F)F)(OC(C)(C)C)C1)OC c1(C(=O)NC2CCC(CNC(=O)CCc3cnc(O)[nH]3)C2)cccc(C(F)F)c1 n1(C(C)C)cnc(C(=O)NC2CC(C(F)C(=O)NC(CN3CCCC3)CO)C2)n1 c1(OC)cc(-n2nnnc2C(CCC(F)(F)F)Nc2ccccc2C)ccc1F C1(CNC(=O)C(F)(F)c2cscc2Br)(CC2CC2)CCCCC1 C(=O)(CC1=NNC(=O)C1)NCC1CN(C(c2nc(CC)oc2)=O)C(C)CC1 C=CC1(CC(=O)NCC2CCN2C(c2cscn2)=O)CCC1 c1(C(=O)NC2C(CNC(c3ccc(C(N)=O)[nH]3)=O)CC2)[nH]cc2c1CCCC2 c1(C(C)(C)C)ccc2oc(C(CCN(C)C)NCC3CC34CCOC4)cc2c1 N1(C(C(CCC)NC(N)=O)=O)CCC=C(C(=O)NCC2CC(N(C)C)C2)C1 CC(C)(C)CC(O)CC(=O)NCCCN(C(=O)CC(F)(F)F)Cc1ccccc1 C1(C(=O)NC(C)CN(C(=O)CSC(F)(F)F)C)CN2CCCCC2CO1 C1(C(N(C2CC(C)C2)C)=O)C2CCC(C2)N1C(=O)CC(O)C1CCCC1 c1(C(=O)NC2C(NC(C(=Cc3cccs3)C)=O)C2)ccc(S(=O)CC#N)cc1 C(=O)(C(COCCOCCOC)CCC)NCCNC(COCC#C)=O C1(C(=O)NCC2(NC(CNC(=O)OCC)=O)CCOC2)CC2CCC(C1)N2C C12(NC(CSCC(C)C)=O)CCN(C(=O)Cc3ccccc3C#N)CC1C2 N1(C(c2c(OC)cccc2Cl)=O)CCC(C2CCN(C(=O)COCC(C)C)C2)C1 N(C1CCCc2cc(F)ccc21)C(c1ccc(Cl)cc1)CO CC(O)CCCC(=O)NC(C)CCNC(=O)C1=NNC(=O)C1 C(=O)(CC(=O)N(C1COCC1O)C)N(C(C)C(=O)OC)CC#C Cn1cc(C(C(=O)NC2CCSC2)NC(=O)CC2(C)CCN2C(N)=O)nn1 Cc1cc(N2CCC(C(C)NC(=O)CC(C)C(F)(F)F)C2)ccc1[N+](=O)[O-] c1(C(N2C(CNC(=O)Cc3ccc(Br)cn3)CC2)=O)nc2ccccc2s1 C1(NC(C2N(CC)CC2)=O)CC2CCC(C1)N2C(=O)Cn1ncc(C#N)c1N c1(CC)ncc(CC(=O)NC(C)=O)o1.C12CC(C1)NCC2 Cn1ncc2c(N3CC4(CC4)CC3CNC(C3(C(F)F)CC3)=O)ncnc12 c1(CCC(=O)NCC2N(C(C=CCCC)=O)CCC2C)cc(OC)cc(OC)c1 c1(C(=O)NCc2cccc(NC(C3C(C)COCC3)=O)c2)ccc(F)c(N)c1 c1(CCC(=O)NC2CN(C(c3cc(CC)c(Cl)cc3)=O)C2)nc2cnccc2[nH]1 N1(C(C(c2ccccc2Cl)C)=O)CCC(CN(C(=O)C=CC2CCC2)C2CC2)CC1 N1(C(CC2N(CC)CCOC2)=O)CC(O)(C2(CNC(=O)CNC(C)=O)CC2)C1 C1(NC(C(COC)COC)=O)CN(C(=O)COc2ccccc2)C(C)(COC)C1 N1(c2nc(C(N(C)C)=O)c3c(n2)n(C)cn3)CCS(=O)(=O)C2(CCCCC2)C1 O=C(C1CCOc2ccc(F)cc21)NCC1CCCCN(C(C2(CO)CC2)=O)C1 n1(C(CC)C)nc(C(N2CCC(CNC(=O)CC(C)(O)C3CC3)CC2)=O)cc1C CC1CN(C(C2CCC2C)=O)CCCN1C(c1ccc(-n2ccnc2)cc1)=O O=C(CC1=CCOCC1)NCC1CN(C(=O)CCc2ccncc2)CCO1 CC1CCCn2ncc(C(=O)NC3CCCCN(C(=O)CCc4ccco4)C3)c21 N1(C(CCc2c(C)cccc2)=O)CCC2(CC(C(=O)NC(C)CCO)=NO2)C1 C(=O)(C(C)(C)CNC(C1CC1C(C)C)=O)NCc1cnc(C(C)C)[nH]1 N1(C(Cc2ncn(C)c2)=O)CCCCC1CCNC(=O)CCC1CCCOC1 C(c1cccc(F)c1F)=CC(=O)NC(C1CN(C(C2(C)CCCN2C)=O)C1)C C1(CNC(C(CCCC)O)=O)CN(C(c2cnoc2C)=O)CC(C)(C)O1 c1(C(=O)OC)cccc(F)c1CNC1(CCCCSc2ccccc2)CCC1 N1(C(C(C)OCC=C)=O)CCC(N(C(c2cc(C(=O)OC)c(C)o2)=O)CC)CC1 C1(C(=O)NCc2c(C#N)cccc2)CC2OCCC2N(C(C2CNC(=O)C2)=O)C1 Cc1ccc(C(=O)NC(C)CCCNC(C2CC(c3ccccc3)C2)=O)c(N)c1 Cc1cc(CC(N2CC(F)CC2CNC(=O)C(C)CC2CC2)=O)cc(F)c1 C1(N(C(C(C)OCCC=C)=O)CC)CCCN(C(c2ccnn(C)c2=O)=O)CC1 N1(C(C2C(C)(NC(C(C=C)CC)=O)CCCC2)=O)CCc2nnnn2CC1 C(CC(=O)NC(C(=O)N(CC(O)COC)C)c1cccs1)OCC C(CC(F)F)(C(=O)N1CCC2(CCO2)C1)NC(C1CC(CC2CC2)C1)=O C1(C(=O)NCC(C)NC(=O)CC(=O)Nc2nccs2)CCCN1C c1(C(=O)NC(C(C)C)(C)CNC(=O)C(C)CSC(F)(F)F)cc2ccccc2o1 O(NC(=O)CS(=O)CC)CC(=O)NC1CN(CC)CC1(C)C c1(C(=O)NCCC2(NC(C3C(C)OCCO3)=O)CC2)ccn2cncc2c1 c1(C(=O)NC2CCN(C(CC3C(C)(C)CC3)=O)CC2O)cc(O)ccc1[N+](=O)[O-] n1(C(C)C(=O)NC(C)(CNC(=O)CC2(CO)CC2)C2CCC2)cnc(C#N)n1 C1(C#N)(CNC(C=CCN(C(c2ccc(CC)s2)=O)C)=O)CCOCC1 c1(NC(=O)CNC(C2CCC2(F)F)=O)cccn(C2CC2)c1=O N1(CC2CN(C(C)C)C2)CC2CC(N3CCCC(C)CC3)C1C2 c1(OC)ccc(C2CC(N(C)C(c3cc(Br)c(Br)o3)=O)C2)cn1 c1(C(N(C(CNC(CC(CC)(C)C)=O)C)C)=O)ccc(NCCOC)c(C#N)c1 CCCC(C)CC(=O)NCC1(F)CCN(C(c2cc(C3CC3)on2)=O)C1 C1(C(=O)NC2C(NC(=O)COCc3ccncc3)CCC2)Cc2cscc2C1 C1(NC(c2c(OC)scc2)=O)C2CCN(C(=O)C=Cc3nc(C)cs3)CC12 C1(C(=O)NCC(C)(O)CNC(C2COC2)=O)CCOC2(CCCC2)C1 c1(C(N2CC(C)(NC(C3CCC(CC)O3)=O)C2)=O)cccc(C#N)c1F c1(NC(Cc2ccc(OC)cc2C(F)(F)F)=O)cc([N+](=O)[O-])c(N(C)C)cc1F C1(C2CCC2)(C(=O)NC2CN(C(c3cn(C(C)C)nc3)=O)C(C)C2)CC1(F)F c1(C(=O)NC(C)CC2CN(C(c3c[nH]c(C(C)(C)C)n3)=O)C2)ccc(Cl)nn1 C1(NC(=O)C(c2cc(Br)c(Cl)s2)N2CC(O)CC2C(F)(F)F)CCC(F)(F)CC1 N1(C(CSCCCC)=O)CC(C(=O)N(CC2=CCCOC2)C)C(CC)C1 c1(NCC(N(C(c2c(C)scn2)=O)C)C2CC2)nc2c(cc1C#N)CCCC2 CC1CCN(C(=O)CNS(N)(=O)=O)C1CNC(=O)CCC=CBr Cc1nnc2n1CC(C(=O)NC(C1CCN(C(=O)C3=NNC(=O)CC3)C1)C)CC2 C1(C(N(CCC(N2CCC(C)(N(C)CC)C2)=O)C(C)C)=O)CC2(CCO1)CC2 Cc1ccc(C(=O)NCC2CCCC(NC(c3coc(C4CC4)n3)=O)C2)nc1 C1(C(=O)NC(CC)CN2CCCC2)CN(C(C2(CC)CCCCO2)=O)CC1(F)F C1(N(C(COCCC=C)=O)C)CN(C(c2cc(COC)ccn2)=O)C(C)(C)C1 C1(C(F)(F)F)CC(=O)N1.N1(OC(Cn2c(C(C)(C)C)nnn2)=O)CCC(O)CC1 C1(C(=O)NCC(CNC(c2cc(CC)[nH]n2)=O)C)(Cc2cnn[nH]2)CCOCC1 c1(C(C(=O)NC(C(=O)OC)Cc2ccc(Cl)s2)C2CC2)ccccc1F C(=O)(C(C)C1=CCCC1)N(C1CC(Oc2c(C(=O)OCC(F)F)c[nH]n2)C1)C(C)=O c1(C(N2CCC(C(=O)NCCCc3ccccc3Cl)C2)=O)n[nH]c2c1CCC2 C(CCC(=O)NCC1CC1CNC(=O)CCc1cnn[nH]1)SC c1(OC)cc(C=CC(=O)NCC#CCNC(c2cncc(SC)c2)=O)ccc1O c1(C(=O)NC2CC(CCNC(C3C(C)(C)C3)=O)C2)ncc(Br)cn1 N1(C(C(CC)(C)Cl)=O)CC2CCCC2(CNC(c2ccn(C)n2)=O)C1 CC1CCCCC1(CO)NC(C12CC(CN1C(=O)CSC(F)F)C2)=O Cc1nc2ncccn2c1C(=O)NC1CC(NC(c2ccc(Br)c(C#N)c2)=O)C1 n1(CC)ncc2c(C(=O)OCCCn3ccnn3)cc(C(F)(F)F)nc12 C1(CNC(c2cccc(C(N)=O)c2)=O)CN(Cc2ccc(F)cn2)CCCO1 c1(CC)cc(-c2nccn2C(C)C(=O)O)ccc1NC(c1nn(C)cc1CO)=O c1(C(=O)NCC(CN(C(c2cc(C)sc2)=O)C)C)ccc(CC2CCC2)cc1 C(=O)(CS(=O)(=O)C1CCCC1)N1C(CNC(C(CC)CC2CCCC2)=O)CC1 C(=O)(C1CCc2nccn21)N1CCC(N(CCC)C(C2CN(CC(C)C)C2)=O)C1 C#Cc1cccc(C(=O)NC2(CNC(c3ccsn3)=O)CCC(C)(C)CC2)c1F C(=O)(C(CCNC(=O)OC(C)(C)C)CC(C)C)NC(CC)CNC(=O)C(C)C c1(C(N2CC(C)(NC(=O)C=Cc3cc[nH]c3)C2)=O)cc2sccc2cn1 CC(F)(C(=O)NCCC1CCCCN1C(=O)CN1C(=O)CCCC1=O)C(F)(F)F N1(C(c2cc(OCC)no2)=O)CC(NC(C2CC2F)=O)C(CC)C1 C(=O)(C(C#N)C(C)(C)C)NCc1occ(C(N2CCC(SC)C2)=O)c1 Cc1cccc(C(=O)NC2CCCN(C(=O)COc3ccc(F)c(Cl)c3)C2)c1F C=CC1CN2CC1NC(=O)CCC(C)OCC2=O.C1(NC(=O)COC)CCCC1 C1(CC=C)(NC(C2CCC(CN(C)C)C2)=O)CCN(C(=O)Cc2ccnn2C)C1 N#CCCCC(=O)N1CCOCC1CNC(C1(c2ccncc2Cl)CC1)=O c1(C(=O)NC(CN2CCN(C(C(C)C3CC3)=O)CC2)C)nccn2nccc12 C#CC1CC(NC(=O)C(C)(C2CCC2)NC(=O)CSCC=C)C1 Cc1ccc(C#N)cc1C(=O)NCC(C)C(=O)NCCCC(=O)NC1CC1 C(=O)(CN=c1ccc(Cl)n[nH]1)N1C(CNC(c2n3c(nn2)SC(=C)C3)=O)CCC1 C1(NC(=O)CC2OCCO2)C2CCC(C2)C1C(=O)NCC12CCC(CO1)C2 CCC(CC)(CC)C(C(=O)N1CSCC1C(=O)OC)NC(=O)OC c1(CCCc2ccc(C(=O)NC(CN(CC)CC)C)[nH]2)cccc(C(F)(F)F)c1 N1(C(COC)=O)CCC(C(=O)Nc2cc(C)ccc2OC)C(C)(C)C1 N1(C(C(CCC=C)(C)C)=O)CCOC2(CCN(C(C34CCC3C4)=O)C2)C1 N1(C(CSCCC)=O)CCSCC1CCNC(C1CCCCC1C)=O Cc1ccc(-c2nc(C(=O)NC(C)(C)CCNC(=O)C(F)F)cs2)s1 CCCCCC(=O)NCC(C)N(C(=O)C(CCSC)NC(N)=O)CC C(=O)(C1CCCc2ccccc21)N1C(CC)CN(C(=O)CCC(F)F)CC1 c1(C(=O)OC)ncc[nH]c1=NC1CC(NC(=O)CC2C=CCCC2)C1 c1(CC(=O)N(C)CC2N(C(C(CC=C)C)=O)CCC2)c(F)cccc1Br C(=O)(CC(C(C)OC)NC(c1c[nH]c(C#N)c1)=O)N1CCN(C(CC)C)CC1 c1(C(N2CCC(C)(c3cn(C4CCNC(=O)C4)nn3)C2)=O)nccc2cc[nH]c12 CC1CC2(CCN(C(C3CCCN3C)=O)CC2)CN1C(c1coc(N(C)C)n1)=O CC1(C)CC(NC(C2CCC(=C(F)F)CC2)=O)CN(C(C2CCCC23CC3)=O)C1 N1(C(c2c(C)nsc2)=O)CCCCC1CNC(c1ccc(Cn2cccc2)cc1)=O c1(CC)ccc(-c2nc(COc3ccccc3)nn2Cc2ccccc2F)cc1 C1(C(=O)Nc2nccc(OC)c2C#N)CCOC2(CCSC2)C1 C1(C(=O)NC2(CF)CCN(C(C(C(C)C)F)=O)C2)CC2CCCC(C1)C2 C1(c2onc(CC(=O)Nc3c(C)c(O)ccc3)n2)CC2C=CC1CCC2 CC12CCC(=O)N1CCCN2C(=O)C(c1cccnc1)O C(C(C(=O)NC1CCN(CC2CC2)C1)C(C)(C)C)NC(c1cc(C)ncc1)=O c1(CN=C(NC(C=C)C)NC2CCC23CCC3)ccc(C#N)c(F)c1 C1(C(=O)NC2(CCC(=O)NCc3c(C)noc3)CCC2)CC(C)(C)CO1 N1(C(C2CC(=C)C2)=O)CC2CCCC2(CNC(c2cc(CC3CCC3)c[nH]2)=O)C1 C1(NC(c2c(C)cccc2C)=O)CN(C(c2cn(CCO)nn2)=O)CC(F)(F)C1 c1(C(N(CCNC(=O)COC2CCC2)CC)=O)c(O)nnc2c1CCCC2 Cc1cc([N+](=O)[O-])nn1CC(=O)NC1CN(C(C2CCC(C)(C)C2)=O)C1 c1(O)nn(C)cc1Br.N1(C(CN2CC(CCCCC)C2)=O)CCC(OCCF)C1 C#CCCCCCC(=O)N(C)CC1(C)CCCC1NC(c1ccccc1OC)=O C12CN(CCN1C(=O)CN(C)C)C(=O)C(c1ccccc1)OCC2.C(C)(=O)OC C(CNC(C1CC1C1(C)COC1)=O)(CC(=O)NOCC(C)(C)O)OC C1(CNC(c2cc(C)sc2)=O)CCCCC1NC(=O)Cc1ccc(C(N)=O)nc1 c1(C(=O)OC)ccccc1C(=O)N(C1CCN(C(=O)CC(F)(F)F)C1)C c1(N(C(C)CNC(C2(O)CCSC2)=O)C)cc(C(N)=O)nc(Cl)n1 c1(C(=O)OCC)cc(Br)ccc1I.N12CCOC(C1)CC(=O)NC1(CC1)CC2=O c1(CCCC)ccc(C(C)C(=O)N(CC(c2ccccc2)O)C)cc1 N1(C(COCCC#C)=O)CC(F)(F)CC1CCNC(c1ocnc1C(F)(F)F)=O CC(CCC(C)(C)C)NC(=NCC1CC1)NCc1c[nH]nc1C(F)F c1(CC(=O)NCCN(C(=O)CC2CCCCC2C)CCC)n[nH]c2c1CCCC2 C12(NC(CC3CC(OC)C3)=O)CCCC1N(C(C1CC3CCC1C31CC1)=O)CC2 N1(C(=O)Nc2cc(C)sc2)CCS(=O)(=O)CC1C1CCC1 CC(O)(CC(=O)NCC1(O)CN(C(C2CC3(CCC3)C2)=O)C1)C1CC1 CC1CC(CNc2ccc(CSc3ccccn3)cc2)CN1C(=O)OC(C)(C)C N1(C(c2cc(OCCN(C)C)ncc2)=O)CCC(NC(c2cscc2F)=O)C(O)C1 c1(C(N(CCC(=O)NCC2CCN(CC)C2)C(C)C)=O)ccc(C)cc1 c1(CC(N2CCCC(NC(CCCCC)=O)C2C)=O)cc2cccnc2nc1C C(C(CC(C)C)NC(=O)C(O)CC1CCOCC1)NC(CC1(C(=O)OC)CC1)=O c1(C(=O)NCC(C2CC2)NC(c2c(N)c(Cl)ncc2)=O)ccc2nn[nH]c2n1 N1(C(C(c2cccc(OC)c2)O)=O)CC(N(C)C(c2csc(C)c2)=O)C2(CC2)C1 C1(CC)CCCN(C(=O)CC(COC)NC(=O)Cc2cccnc2O)C1 N1(C(CN(CC)CC)=O)CC2C3CCC(C2C1)N(C(c1cccc(CO)c1)=O)C3 c1(CN2CC(CNC(c3ccc(C)s3)=O)OCC2)c[nH]c2cnccc12 c1(C(=O)NC(C(C)=O)C2CC2)ccn2ncc(Cl)c2n1 CCCCC(=O)C(=O)N(CC(C)(C)CNC(C1CCOC(CCC)C1)=O)C N1(C(c2cn(CC)nn2)=O)CCC2(CCCCN(C(=O)Cc3nnc(C)o3)C2)C1 C1(NC(C2(CC#C)CCCO2)=O)CN(c2nnc(CO)s2)C2(CCOCC2)C1 c1(OC)cc(-n2nc(C3CC=CCC3)nc2Cn2c(C)csc2=O)ccc1Cl Cc1cccc(F)c1C(N1CCC(=CCNC(c2cc(Br)c[nH]2)=O)CC1)=O c1(COC)nc(NCCc2cc(Br)ccc2C)cc(=NCCc2cnc(C)[nH]2)[nH]1 c1(C(=O)NCCC2(CNC(c3ccc(OC)cc3)=O)CC2)cccc(S(C)=O)c1 N1(C(C2(C)CC(=C)C2)=O)CCN(C)C(C(C)C)C1.c12ccc(nc1)s2 N1(C(C=C(CC)CC)=O)CC2CC(CNC(c3ccc4occc4c3)=O)CC1C2 c1(C(=O)NCC2(CNC(c3c(N)cnc(Cl)c3)=O)CC2)cn2ccc(F)cc2n1 S(=O)(=O)(c1cccc(C(=O)O)n1)NC1C(OC)C2(C1)CCC2 Cc1ccc2[nH]c(C(=O)NCC(C)CNC(C34COC(CCO3)C4)=O)cc2c1 c1(C(C(C)C)O)cn(CC2CCC(NC(=O)C(F)F)C2)nn1 N1(C(CC(=O)OC)=O)CC(C(=O)Nc2[nH]c(C)nc2C#N)C2(CC2)C1 C1(CCC(=O)NC(c2nccs2)CC)CCCN(C(c2cc(O)n(CC)n2)=O)C1 C12(C(=O)Nc3cc(C)c(NC(=O)C(O)C(C)C)cc3)CCC(CC1)C2(C)C CC(C)CC(=O)NC(C)CC(C)NC(c1csc(C(F)(F)F)c1)=O c1(C(C(=O)NC(C2CN(C(=O)CSC(F)F)CCO2)(C)C)(F)F)ccc(F)cc1 C1(CNC(C(COCC)C)=O)CC2(CO1)CN(C(=O)CCCCNC(N)=O)C2 N1(C(C2C(C)OCCO2)=O)CCCC12CCCN(C(C1(C)CCN(C)CC1)=O)C2 C1(C(=O)NCC2CC(OC)CN2C(=O)CCCCC2CC2)CC1C1CCCCC1 CC1COC2(C1)CN(C(=O)C(CCN(C)C)NC(=O)CN1CCCNC1=O)C2 n1(CC2CCN(C(C)=O)C2)nnn(-c2cccs2)c1=O.C1CS1 N1(C(CCNC(C(=CC2CCCC2)C)=O)=O)CCCC(C)C1C(N)=O C1(NC(C(C2CC2)OCC)=O)CN(C(=O)CN(S(C)(=O)=O)C)CCC1F C12(C(=O)NC(C(=O)OC)C3CC3)C(NC(=O)C(C)N3CCCC3)C3CC1C2C3 N1(C(C(=O)NCCCF)CC2CCC2)CCC(C2OCCO2)CC1C(F)(F)F C1(N(c2nnc(CC)o2)CCO)CCCN(C(=O)COC(C)(C)CC)C1 C1(C(N2CC(n3cc(-c4ccc(F)c(Br)c4)nn3)C2)=O)CCCC(C(F)F)CC1 N(C(=NCCOC)NC1Cc2ccccc21)C(c1ccc(COC)cc1)C C(CCCCC(=O)Nc1cccc(CO)c1)N(C(C(n1ncc(C)c1)C)=O)C c1(CC)nc(C(=O)NC(C)(CNC(=O)C(C)c2cncs2)C2CC2)co1 C12(C(N(CC(C)CO)C)=O)CC1CN(C(c1ccc(F)cc1)=O)C2 c1(-n2ccc(C(=O)NCCC(C)NC(c3cnnn3C)=O)n2)ccc(Cl)c(F)c1 Cc1cnc(Cl)c(NC(C2CSCCN2C(c2noc(C)c2C)=O)=O)c1 CC1C(NC(=O)CC2CCC(=O)NC2)CCCN1C(c1ccc(C(N)=O)cn1)=O c1(SC)ccc([N+](=O)[O-])cc1C(=O)NC1CCCC1NC(C1CC(F)(F)C1)=O C1(NC(CNC(C2C(C)C2)=O)=O)CCOCC1C(N1CCC(C(C)C)(CO)C1)=O C(=O)(C(C(C)C)NC(C)=O)NC(C(=O)NC1CC(OCC)C1)C1CCCC1 CCCC(O)CC(=O)N1CC(=C(F)CNC(c2nncn2C)=O)C1 c1(NC(C2CC(CCNC(C(C3CCCCC3)C)=O)C2)=O)cn(C)nc1C(N)=O C(=O)(CCCCCCC(=O)NC1CCCN(C(c2c(C)cncc2C)=O)C1)OC Nc1cc(C(N2CCC(NC(C3CC=CCO3)=O)C2)=O)ccc1-n1cnnc1 C1(C(N(C(CCO)C(F)F)C)=O)N(C(=O)C=CC(=O)N(C)C)CCCC1(C)C CCC(CC)C(O)CNC(C1(NC(=O)C(C)C(C)(C)C)CCOCC1)=O N1(C(C(C=C)O)=O)CC23CCCC2(C1)CN(C(=O)C=Cc1ccc(SC)cc1)C3 c1(OC)ncc(Cl)cc1C(N1CCC(NC(c2cn(C3CCOC3)cn2)=O)C1)=O Cc1cc(C(=O)NC(CNC(=O)C(C(C)O)N(C)C)C(C)C)c(O)c(C)n1 N1(C(C=CCCC)=O)CCC2(C=C(C(=O)NCC3CCCC34CCC4)C2)C1 Nc1ccc(-c2cn(CC3CCCCN3CCC3CCOC3)nn2)cc1[N+](=O)[O-] C1(NC(CNC(=O)OCC=C)=O)CC(O)CN(C(=O)CN2CCC(C)CC2)C1 S(=O)(=O)(c1ccccn1)N(c1nc(OC)c(Br)cn1)C1CCCNCC1 c1(NC(C23C(CN(C(c4ccc(Br)s4)=O)C2)C3)=O)cccc2cccnc12 c1(OC)ccc(Cl)c(CC(=O)NC2CC(F)CN2C(=O)CNCC(F)(F)F)c1F N1(C(c2c(OC)ccs2)=O)CCC2(CNC(C)=O)CC12 c1(C(C)NC(C=C(C)CNC(C2CC2C(C)C)=O)=O)ccc2ccccc2c1 C#CC1CCN(C(=O)C(CC2CC2)NC(=O)C=Cc2cncs2)C1 C(=O)(CCCC(F)(F)CO)N1CC(n2cc(CNC(C3C(C)OCCC3)=O)nn2)C1 C(=O)(CCCC(C)(F)F)N1CCN(C(c2cc(C(=O)OC)ncc2)=O)C2C1C2 C12(C(=O)OC)CC3CC(CC(C3)C1NC(c1cc(C)nc(C)c1O)=O)C2 N1(C(C(C)c2cccs2)=O)CC2CCC1CC2NC(=O)CCC(N)=O C1(CNC(C2C3CC4C(C3)C24)=O)C2CCCC1N(C(c1cn[nH]c1)=O)C2 S(=O)(=O)(c1ccc(Cl)cc1F)C(=O)NC1ON=C(C(=O)OCC2(SC)CCC2)C1 C12(NC(CCCN(C)C)=O)CN(C(C3CSCCS3)=O)CC1CS(=O)(=O)C2 c1(C(c2n(CC(F)F)nnn2)NCc2cscc2Br)cnc(C2CC2)nc1 CC1CN(C(C23CC(C#N)(C2)C3)=O)CC1(C)CNC(C1COCCO1)=O CN(S(=O)(=O)N1CCCCC(CO)C1)c1ccc(N(C)C)c(C(N)=O)c1 C(C1CCCc2nc[nH]c21)NC(=O)C(c1ccc(Cl)cc1F)O C(=O)(C1CCc2nccn21)N(CCC(=O)NC(C)(CO)C1CCC1)C1CC1 Cc1cccn(CC(N2CC3(CC3)CC2CNC(=O)CN2CC=CC2)=O)c1=O CS(=O)(=O)c1cc(C(=O)NCC2CCC2NC(=O)Cc2ccccc2)ccc1F C1(OC)CN(C(=O)Cn2cc(C(OC)OCC3CC3)nn2)C(C)(CSC)C1 N1(C(C(CC)OC)=O)CCC2(CC1)CCN(c1cc(-n3cncn3)ncn1)CC2 C12(CNC(c3nc(CC(C)C)sc3)=O)CC1CN(C(=O)CCCc1ccsc1)C2 C1(C(=O)OC)CCCN(C(=O)COC(c2cnccc2-n2cc(C)cn2)=O)C1 Cc1cccc(C(O)C(N2CCC(C(=O)O)C2)=O)n1 CCCCCCOC.C1(=O)C(C)(C)CC(=O)NCC2CC(C2)CN1C C(C(C(=O)N(CC(O)CN(C)C(c1ccc(Cl)cn1)=O)C)C(C)(C)C)OCC=C C1(C(N2C3CN(C(c4c(CC)non4)=O)C(CC3)C2)=O)COc2ccccc2C1 C1(C(=O)NCC(CO)NC(CCC)=O)(COC)CCCCCC1 CC(CN(C)N1CCOCC2(CCOCC2)C1)OCC(F)(F)F C1(C(=O)NCC(O)CNC(C2CCC(C(=O)OC)O2)=O)(COCC)CC=CC1 c1(C2(C(=O)NCC#CCNC(c3cn(C)nc3)=O)CC2)ccc(Cl)cc1Cl C(=O)(C(C)CC(F)(F)F)N(C1C(O)CCN(C(c2cn(CC=C)nn2)=O)C1)C N#Cc1ccc(N2CCCC(NC(c3ccn(-c4ccccc4)n3)=O)C2)nc1 C1(c2n(C)ncc2)CCCCC1NCc1ccc(O)nn1 C1(CC(=O)NC2CCCCC2CNCc2ccnc(F)c2)CCCC12CC2 N1(C(c2c(C)c(N)ccc2)=O)CCC2CC(NC(c3ccncc3)=O)CCC2C1 c1(C(=O)NCC(CN(C(C(C)CO)=O)C)O)ccc(F)c(Cl)c1F C(=O)(C1=C(Cl)CCC(C)C1)N(CCCNC(CCN1CCC(C)CC1)=O)CCO c1(C(N2C(C)(c3cn(CC(N)=O)nn3)COCC2)=O)cc2ccncc2cc1F N1(C(C=CCN(C)C)=O)CC(NC(=O)CC2CCC(C)(C)O2)C(C(F)F)C1 C1(C(CNC(C(C=C)C)=O)C)CCN(C(C2(C)CC2(Cl)Cl)=O)CC1 C1(NC(c2ccccc2)=O)CCC12CCN(C(=O)CCN1CCCCC1)CC2 c1(C(N2C(CCNC(c3cc(C4CC4)no3)=O)COCC2)=O)cc(F)ccc1O c1(C(N(C2CCN(C(c3cnccc3C#N)=O)C2)C)=O)ncc2cc(Cl)ccn12 C1(C(N2CC(NC(c3ccc(C)c(Cl)c3)=O)C(F)C2)=O)CCC2C(C1)C2(F)F N1(C(CC2CCCC(=O)N2)=O)CC(=O)NCC1C(=O)NCC=CC=C(Cl)Cl CCCC(C(O)C(=O)NCC1CN(CC)C(=O)O1)NC(=O)C=Cc1ccncc1 C1(O)(C(=O)NC(c2cc[nH]c2)C)CC2(CCNC2)C1 c1(C(=O)NCC(C)(C)NC(C(C)c2ncco2)=O)cc(Cl)cc2cccnc12 c1(C(N(CCNC(c2c(CC)scn2)=O)C2CC2)=O)ccc(C2CCOC2)cc1 C(=O)(CCC(=O)c1ccc(Br)cc1)NC(C1CCCCC1)(C)CO C1(C(N(CCC(C)NC(c2scc(OC)c2OC)=O)C)=O)CCCNS1(=O)=O C12CC(C1(C)C)NC(=O)N2.C(CS(=O)(=O)N1CCCC1)OC(C)C C(C(O)CC(F)(F)F)NC(CC1CCN(C(C2(C)CCN(C)C2)=O)C1)=O N1CC(NC(=O)Cn2ccc(=O)cc2)C2CCCC12.C=CCCC1(C=O)CC1 c1(N(CC(N2CC(N(C)C(c3ns[nH]c3=O)=O)C2)=O)C)ccc(Cl)cc1 N1(C(CC(CN(C)C)O)=O)CCC(NC(c2ccnc(C(C)C)n2)=O)C12CCC2 Cc1cc(F)ccc1NC(C12CC(CN1C(=O)CC1(O)CCOC1)C2)=O c1(C(N2CCC(C)(NC(C3CC4(F)CC3C4)=O)C2)=O)cccc2occc12 CC1CCc2ncc(C(=O)NC3CCC3NC(c3ccnn3CC(F)F)=O)n2C1 C(CC(C)C(=O)N1CCCC1C1(C(=O)NC2(C)CS(=O)(=O)C2)CC1)OC CCC(O)CC(=O)N1CC(O)CC1c1cn(-c2ccc(Br)nc2)nn1 N1(C(CCCC#C)=O)CC(=O)NCC1C(=O)NCC(C)(C)CC(C)C N1(C(C=C)=O)CCCC(CN(C(=O)C(CC)c2ccccc2)CC)C1 N1(C(C(c2cccs2)SC)=O)CCC(C2CC2)(NC(c2cc(C)cs2)=O)C1 C(CC(O)CC(=O)N(CC(C)CNC(C1CCC2(CC1)CC2)=O)C)SC c1(NCc2cc(C)nc(C)c2)[nH]c(=NCc2cscn2)nc2c1ncn2C(C)C c1(N(C(N=c2[nH]n(C)c(Cl)c2)=O)Cc2cccs2)ccc2ncccc2c1Cl c1(C(=O)NCCOC(CNC(C(C)C2CCCC2)=O)(C)C)cc([N+](=O)[O-])sn1 CCC(C(=O)N=c1ccn(-c2ccccc2Cl)[nH]1)=C1CCCCC1 c1(C(N(CCC)CCNC(C2(C(F)F)CC2)=O)=O)ccc(NC(C)=O)s1 C1(C(=O)NCc2ccnc(Cl)c2)CN(C(c2ccc(O)cn2)=O)CCC1O c1(CC(N2C(C)(CC)CC(NC(C3CC=CC3)=O)C2)=O)c[nH]c2c(C)cccc12 C=CC1(C(N2CCOC(C(=C)C)C2)=O)CCN(C(=O)C(O)CSC)CC1 C12(C(=O)NCCN(C(C34CCC(C3)C4)=O)C3CC3)CC3CC1C2C3 C1(S(C)(=O)=O)(C(=O)NC2CN(C(CC(C(C)C)C)=O)CC2F)CCCC1 C=C=CCCC(=O)NC(c1nocc1C(=O)N(C1CCOC1)CC)C C12(C(N3CCC(C)(NC(c4c[nH]cc(F)c4=O)=O)CC3)=O)CCCCC1C2(F)F C#CC1(N(C)C)CN(C(C2CCCC2CNC(c2ccc(OC)o2)=O)=O)C1 C1(C(=O)NCC2(CC)CCCCO2)CC(O)C(O)CC1CNC(=O)C(C)C1CC1 C1(C(N2CCCC(CCNC(CC(=C)C)=O)CC2)=O)CC2(CCC2)CCO1 c1(C(N2CCCCC(C(=O)NC)C2)C(=O)NCCCC)cc(C)nc(C)n1 Cc1ccc(C=CC(N2CCCC(CCNC(c3nn[nH]c3Cl)=O)C2)=O)cn1 c1(OC)ccc2c(n1)N(C)CCN2C(=O)CN1CCC(C(N)=O)CC1 S(=O)(=O)(c1cccnc1NC(CCO)C1CC1)NCc1n(CC)c(C)nc1 C=CCC(C(=O)NCC1(CNC(=O)C=Cc2cnn(C)c2)CC12CCC2)C(C)C C(=O)(C1CCCc2nncn21)NC(c1ccccc1)CNC(=O)C1=CC(O)CCC1 N1(C(C(C)NC(=O)NC)=O)CCC(ON(C(=O)CN(C)C(=O)C2CC2)C)CC1 N1(C(C2(CCC)CC2)=O)CC(CNC(c2cc(COC)cs2)=O)CC(C)(C)C1 CCCC(CNC(c1cc(CNC(c2cnn(C)n2)=O)ccn1)=O)CCO CCCCC(CC)C(=O)N1CCC(COC)(NC(C2CN3CCN2CC3C)=O)C1 N1(C(c2cn(C)nc2C(F)F)=O)CC(NC(c2ncn(C)n2)=O)CC2(CCC2)C1 c1(OC)ccc(Cl)c(Cl)c1C(N1CC2CCC1CN2C(C1CC1(C)C(F)F)=O)=O CCCCCCCC(=O)N1CC2CCN(C(c3cc(C(N)=O)co3)=O)CC12 N1(C(C(CNC(CC(CC)C2CCC2)=O)C(C)(C)C)=O)CC(C)(C)OC(C)(C)C1 n1(C(C)C)cc(C(=O)NC(C2CCCCC2)C(C)NC(c2nc(Cl)cs2)=O)cn1 C(=O)(C1=CCC2(COC2)OC1)N1CCC(=CCNC(c2cccc(O)n2)=O)CC1 N1(C(C2CCC(=O)OCC2)=O)CCC(CNC(C2CC3(CC3)CO2)=O)C(F)(F)C1 C1(C(=O)NC(C(C)NC(CCCN(CCC)CCC)=O)(C)C)CCCCN1N=O Cc1ccnc(C)c1C(=O)NC1CCOCC1C(=O)NCc1ncsc1C c1(C(C)C)ccc(C(=O)NCCCN(C)C(c2cscc2C2CC2)=O)nc1 C1(C(=O)NCC(C(C)C)NC(=O)COc2ccon2)Cc2c[nH]cc2S1(=O)=O Cc1nc(NC(c2nc(C(=O)NCCc3cccnc3)cs2)=O)nc(Cl)c1Br Cc1cc(C(F)(F)F)nn1CC(=O)NCCCNC(=O)C=C1CC1C(F)(F)F c1(OC)ccc(C(=O)NC(C2CCN2C(c2ccncc2Br)=O)=O)c(OC)c1 S(=O)(=O)(c1cccc(N2Cc3cnc(Cl)cc3C2)n1)N1C(C)C(O)CCC1 C(=O)(C1=CCC(C)(C)CC1)NCC1CC(NC(C2CN(C(=O)NC)C2)=O)C1 C#CC1CCC(COC(=O)COC2CC(NS(=O)(=O)CCCC)C2)CC1 c1(N2CC(CC(C)NC(c3cc(C)nn3C(C)(C)C)=O)C2)cc(Cl)nc(C)n1 C1(CC=C)(C(=O)NCC(F)C(C)(C)O)CCCN1C(=O)C(CN(C)C)CC CC1(C)CC(=O)NCC1C(=O)NC1CCN(C(c2ccsc2C#N)=O)CC1 Cc1ccc(C(=O)CN(CCSC2COC2)C)s1 CC(C)(C)CC(C)(C)C(=O)NCC1(C)CN(C(C2(F)CC=CCC2)=O)CCO1 c1(C(C(=O)N(C)CCn2cccn2)NC(CN(C(COC)=O)C)=O)ccccc1 C(C(CC(C)C)C(=O)NC1(CNC(c2nn(C)c(Br)c2C)=O)CCC1)OC C1(CNC(C(C2CC2)NC(CC2N(C)CC=CC2)=O)=O)CC12CCOCC2 C(=O)(CCC1=CCCCC1)N1C(C(N2C(C(=O)OC)CC2)=O)CN(C)CC1 Cc1nc(O)[nH]c1C(N1CC(F)(CNC(C2(C3CCCO3)CCOCC2)=O)C1)=O C(CCCC(=O)N1CCC(C)(CCC)C1)N(C(C(C)=CC=C)=O)C C#Cc1cccc(CC(=O)N(CCNC(c2ccc(COC)c(C)c2)=O)CC)c1 c1(C(N2CCC(C)(C(=O)NCCc3ccsc3)C2)=O)ccc2cc(O)ccc2n1 N1(C(C=C2C(C)(C)CCCC2)=O)CC2CC(NC(c3cncc(F)c3)=O)CC2C1 N1(C(c2c(C)con2)=O)CCC(CF)(CNC(C2(CF)CC2)=O)C1 C1(CNC(c2ccc(NC)cn2)=O)CCCCN(C(c2ncccc2Br)=O)C1 CC1=C(C(=O)NC2CN(C(c3snc(Cl)c3Cl)=O)CC2F)SCCO1 c1(NCC2CCC(=O)NC2)ncccc1S(=O)(=O)N1CCC2(C1)CC(F)(F)C2 c1(NC(c2n(CC=C)nnn2)C2(SC)CC2)ccc(-n2nccc2C)cc1 C1(OC)(OC)CCC1C(=O)NC(CNC(c1ccc(CO)o1)=O)CO C1(NC(=O)Cc2csnn2)CCC2CCN(C(c3cnn[nH]3)=O)C12 N1(C(c2cn(CCOCC)nc2)=O)CC(NC(=O)C(C)C(F)F)CCC1C CC(CNC(=O)C(C)(C)C)CC(=O)N1CC(OC(C2CC(n3cccn3)C2)=O)C1 C1(NC(c2cc(C)nn2C(C)(C)C)=O)CN(C(=O)Cn2cnnn2)CC2CC12 C1(C(=O)NCC(CNC(COC)=O)(C)OC)CC2C=CCC(C1)C2 N1(C(C2CC(N(C)C)C2)=O)CCCC2(C1)CN(C(=O)COC1(C)CCC1)C2 Cc1cccc(C(CNC(=O)CCC2CCOC2)NC(c2cc(C#N)c[nH]2)=O)c1 C1(OC)CC(CCNC(C2(OC)CCCC2)=O)N(C(C2CCSC(C)C2)=O)C1 CC1CCN(CCC(=O)NCC2(C(N)=O)CN(C(=O)CC(F)(F)F)C2)CC1 N1(C(c2c(O)ccc(SC)c2)=O)CC2CCN(C(=O)CCCN(C)C(C)C)CC12 Cc1nc(CNC(=O)C(C)CN(C)C(C2(O)CC2)=O)[nH]c1C CCCCCCCC(=O)N1CC2CCC2(CC(=O)Nc2c(O)cccc2F)C1 c1(CC(=O)NC2CCCCN(C(c3coc(Cl)n3)=O)C2)c[nH]c2cnccc12 N1(C(CCCOCCC)=O)CC(O)CCC1C(=O)Nc1cccc(OCF)c1 c1(C(=O)NCC(CO)NC(C(C)CC2CC2)=O)ccccc1OCC(N)=O c1(C(N2CC3C(CNC(c4cncc(C)c4)=O)C3C2)=O)ccc(F)c2c1OCC2 C(C(COC)CC(=O)NC1CC(O)CN(C(=O)CCOCCCOC)C1)OC N1(C(c2ccn(CC)n2)=O)CC(OC)CC(NC(c2ccc(I)c(C)c2)=O)C1 C#Cc1cc(C(=O)N(C)CC2CCN(C(=O)CC3(CC)CCC3)C2)ccc1C CC1CC(=O)NC1C(=O)NCc1cccc(NC(=O)CCC2CCCCC2)c1 C(C(C)(C)CC(=O)N1CCCC(CC2(CSc3ccccc3)CCCN2)C1)OC C=C(F)C1(CC(N2CC3(CCC3NC(=O)C3CC3)C2)=O)CCOCC1 Cc1ccnc(C(=O)NCC2(O)CCN(C(=O)CCCC3CC3)C2)n1 N1(C(C=C(CC)C)=O)CCC(N(C)C(c2cc(C3CC3)[nH]n2)=O)C1 C1(C(=O)NC2(C)CCCN(C(c3cc(Cl)ccc3O)=O)C2)CCCC2(CCC2)O1 c1(CCC(C)C)cccc(NC(=O)NCC2CC(n3ccnc3)C2)c1 C=C(C)CCCC(=O)NC1CC(O)(CNC(=O)CSc2cc(F)ccc2F)C1 C1(CC(C)Cn2cc(C)c3c2ccs3)CC2CCC(C1)N2C(=O)OC(C)(C)C Cc1cc(=NCC2CCOC2)[nH]cc1S(=O)(=O)N1CC2CS(=O)(=O)CC2(C)C1 n1(CC(=O)NCC(O)CNC(C2CC2(F)F)=O)nc2n(c1=O)CCCCC2 C(C(=O)NCc1ccsc1)(C1CCCC1)NC(C=CCOC)=O C(CN=c1[nH]c(=NC)[nH]c(=NC2CCC(OCC)CC2)[nH]1)NC1CCCN1CC Cc1nc2cc(C(=O)NCC3C(C)CCN3c3nccc(CO)n3)ccc2o1 c1(NC2(CNC(C3=CC(C)(CC)C3)=O)CCCC2)nc2c(C)c(C)ccc2s1 c1(OC(C)C)ccc(C(=O)N(CC(O)CNC(=O)CCc2cncnc2)C)nn1 Cc1c(C(=O)NC(C(=O)NCC(C)(F)F)C2CCCO2)ccn1C c1(C(=O)NCC(CNC(C(C)OCCOC)=O)OC)cnc(Cl)s1 c1(C(N(C2CCCN(C(C(CC)O)=O)C2)CCF)=O)cc2ccccc2nc1O N1(C(c2cn(CCCC)nc2C)=O)CCN(CC(C)O)CC1C C1(F)(CNC(CCC2C(C)(C)C2)=O)CN(C(=O)C(Cl)=CCl)C1 CCS(=O)CC(=O)N1CC(CO)(NC(=O)C=Cc2ccc(C3CC3C)o2)C1 C#CCC(CC(=O)NCC1CN(C(=O)CNS(N)(=O)=O)CC1OC)c1ccccc1 N1(C(Cn2c(C)c(Cl)cn2)=O)CC2CC(NC(=O)CC3CCCC3(F)F)C1C2 n1(CC)c(C(=O)NCC2(C)CC(NC(=O)C3=NOC(C)C3)C2)cc2ccccc12 C(=O)(C(C)P(C)(C)=O)NC1(C)CCN(C(C(CCC)c2cccc(Br)c2)=O)C1 Cc1cc(C(=O)NCCC2CCN(C(=O)C(C)C3CCC3)C2)c(Br)c(C)c1 C(=O)(C(CNC(=O)CCCOC)C(C)(C)C)N1CC(C(=O)NCC)C1 c1(C(=O)NCC(CNC(C(C2CC2)SC)=O)O)ccc(CS(N)(=O)=O)cc1 N1(C(C(C)C2CC2)C(=O)NCCC2CC2)CC(=O)N(C)C(C)C1 C(C)(CNC(=O)C=CC(C)(C)C)(CO)NC(C1C(C(=O)OC)CC1)=O c1(OC)cc(C(F)(F)F)ccc1CNC(C1(NC(C)=O)CC1)=O n1(CC(=O)NC2CCC(NC(C3CCO3)=O)CC2)cc(Br)ccc1=O C1(NC(C(C2CCOC2)NC(C)=O)=O)CCCCN(Cc2ccon2)C1 N1(C(c2c(CC)ncs2)=O)CCC2(C1)CN(C(c1cc(C(C)=O)on1)=O)CCO2 Cc1cc(OCCC(=O)N(C)CC2CCN(C(=O)C(C)CC(C)C)C2)cc(C)c1 C=CC(C)CC(=O)N1CC(C)(NC(CCC(O)C2CCCC2)=O)C1 c1(C(N2CC(C)C(CNC(C3SCCS3)=O)CC2)=O)ccc(F)c(S(N)(=O)=O)c1 C(=O)(C(C1=CCCCC1)N1CCCN(CCF)CC1)NCCSC Cc1cccc(CC(=O)NC2CCC2NC(=O)COCC2CCCOC2)c1Cl c1(NC(C2CC2C(=O)Nc2cccc(Br)c2[N+](=O)[O-])=O)cc(Br)ncc1[N+](=O)[O-] C(=O)(C(CCC=C)NC(c1nonc1C)=O)N1CCCC(CC=C)C1 S(=O)(=O)(c1cccc(Cn2cc(C34CC(CN3C(=O)C(C)O)C4)nn2)c1)NC c1(CC)c[nH]c2c(N3CCCC3CC3CCC3)nc(Cl)nc12 C1(C(=O)OCC(=O)NC)CC(C)CN1C(=O)CCCOCC(=O)NC(C)=O N1(C(C2(COC)CCCC2)=O)CCCCC(NC(=O)C(c2ccc(Cl)cc2)O)C1 C1(C)(NC(CN(C)Cc2ccccc2)=O)CCN(Cc2cc[nH]n2)C1 n1(CC(=O)OC)cc(-c2ccc(C(N3CCC(N(C)C)C3)=O)o2)nn1 N1(C(c2c(C)noc2C)=O)CCC(CNC(c2ccc(CC#N)cc2)=O)C(C)C1 c1(SC)nc(NC2C3CC2CN(C(=O)CC2CCCCO2)C3)cc(Cl)n1 c1(OC)ccc(C(N2CCC(NC(c3ccc(C(N)=O)[nH]3)=O)C2C)=O)c(OC)c1 c1(CC)cccc(C)c1C(N1CCC(CN(C(=O)COCCC(C)C)CC)C1)=O c1(CCC(=O)N(CC(C)NC(C2(C)ON=C(C)C2)=O)C)cccc([N+](=O)[O-])c1 N1(Cc2cc(C)c(OCC(=O)O)c(C)c2)CCC2(CC1)CNC(=O)O2 C1(O)(CN(C)C(C2CC(N(C)C)C2)=O)CCN(C(=O)Cc2cn[nH]c2)C1 n1(CC(=O)NCCC(C)N(C)C(C2C(F)(F)C23CC3)=O)nc(Cl)ccc1=O N1(C(CC(CC)C(F)F)=O)CCCC2(CCN(C(=O)C=CC3CCCC3)C2)C1 C1(F)(CNC(c2cncc(C)n2)=O)CCCN(C(=O)C2=CCCCC2)C1 C1(C(N2CC(NC(CCC(C)C)=O)C(F)C2)=O)CCOC2(CCCCC2)C1 C1(NC(c2cn(C)c(=O)cn2)=O)CC2CCC(C1)N2C(C1C2CCCCCC12)=O C1(CN(C(C(C2CC2)OCC)=O)C)CCCCN1C(=O)CCc1ccncn1 C(=O)(C(F)Cc1ccccc1)NC1CC(N(C(=O)CSC2CC2)C)C1 C(=O)(C1=COCCC1)NC(CC#C)C(=O)NC1CC(CN(C)C)C1 c1(OC)c[nH]nc1C(=O)NC(C1(O)CN(C(=O)CN(C(=O)C(C)C)C)C1)C C12(C(=O)NCc3nc(C)c(C)[nH]3)CCCC1N(C(c1nocc1Cl)=O)CC2 N1(C(c2cc(C)[nH]c2C)=O)CCC(CNC(C2(C)CCN(C)C2)=O)CC1C N1(C(CCN(CC(C(C)C)C)C)=O)CC(NC(c2nsnc2O)=O)C(N=[N+]=[N-])C1 C=CC(C)N=c1nc2c(ncn2CC)c(NCCCC2CCCCO2)[nH]1 C1(C(N2CC(CC)N(C(=O)CCc3nccn3C)CC2)=O)OCCOC12CCC2 n1(C2(C(=O)N(C3CC(NC(CC(C)(C)OC)=O)C3)C3CC3)CC2)cnc2ccccc12 C1(CNC(C2(OC)CC2)=O)CCN(C(=O)CC2CCCCC2(F)F)C12CC2 C(CN=C(NCc1cnc(-c2ccccc2)o1)NC1(CF)CC1)OCC=C c1(CC(N2CCC(NC(c3c(C)onc3Br)=O)C2)=O)noc2cc(F)ccc12 N1(C(C2CC(C)(F)C2)C(=O)NCCSC)CCC(C(c2ccccc2)=O)CC1 Cc1nccnc1C(=O)NC1CC(NC(c2ccnc(OC3CCOC3)c2)=O)C1 CC(CC(=O)NCCC1CC(NC(=O)Cn2cnc([N+](=O)[O-])n2)C1)C(F)F N1(C(c2ccc(OC)s2)=O)CCCC(C(=O)Nc2ccnc(Cl)c2)C1 c1(CC(N2CCC3CC2CN3C(c2ccsc2)=O)=O)ccc2nonc2c1 c1(C(=O)NC2(CO)CN(C(C(P(C)(C)=O)O)=O)C2)ccc2c(c1)CCCS2(=O)=O C1(NC(Cn2cc(-c3ccc(OC)nc3)nn2)=O)CCCC(C(C)(C)C)CC1 N1(CCNC(C23CC(CCC)(C2)C3)=O)CCN(C(c2cc(C3CC3)[nH]n2)=O)CC1 c1(C(N2CC(C)C(NC(=O)CSCC(N)=O)C2)=O)cnc2cccnc2c1 N1(C(c2cncc(N)c2)=O)CCCC(CCNC(=O)C(F)OC(F)(F)F)CC1 CC(CCCc1ccccc1)C(=O)NC1(c2nc[nH]n2)CCCC1 C1(C(N2C(C)(CC(=O)NCCCC#C)CC2)=O)(C(N)=O)CCCCC1 N1(C(c2c(OC)ccnc2)=O)CCOCC(NC(c2nccnc2Br)=O)C1 C(CC(C(C)(C)C)NC(c1ccc(C#N)o1)=O)N(C)C(c1cccc(F)c1Cl)=O N1(C(C(C(CC)O)C)=O)CCCC2(CCN(C(c3nc(=O)n(C)[nH]3)=O)C2)C1 N1(C(=O)CNCc2ccccc2)CCC(NC(=O)Nc2nccc(CO)n2)CC1 CC1COCCN(C(C23COC(C2)C(NC(C2CC2Cl)=O)C3)=O)C1 Cc1ccc(C(F)C(=O)NCCCN(C(=O)Cc2cnccn2)C(C)C)cc1 c1(C(N2C(C)CN(C(=O)Cc3c[nH]ccc3=O)CC2)=O)cc(F)c(Cl)cc1F N1(C(CCc2cn(C)nc2)=O)CC2CN(Cc3cc(C#N)ccc3F)CC2C1 CC(C(=O)NCC(C)(O)CNC(C1CCC(O)CC1)=O)C(C)(C)C C1(CC(N2CCCC(N(c3ncns3)C)C2)=O)COC(C)(C)CO1 c1(Cn2cc(CCCC)nn2)cccc(CNC2C3COCC23)c1OC Cc1cnc(C(=O)NC(C)(CO)C(=O)N(CCC(C)(C)O)C)c(F)c1 CCCCC(C)(F)C(=O)NCc1ccc(C(=O)NCC2CC23CC3(F)F)nc1 Cc1cc(Cl)cnc1-n1cc(CC(C)(C)C(=O)O)nn1.C(=O)(CN(CCO)CCO)N CCC(CO)(C(=O)NC1(CCCC(=O)NCC2CCCO2)CCC1)OC C1(C(N2CC(C(C)(C)O)(CNC(=O)Cc3ccsn3)C2)=O)CC(=O)C1(C)C c1(C(N(CCCNC(C(=Cc2ccccc2)CC)=O)CC)=O)cc2cscc2s1 CC1CN(C(c2nn[nH]c2Cl)=O)CC(C)N(C(c2cnc3cccnc3c2)=O)C1 N1(C(COCCCC)=O)CC23CCCCC2(C1)CN(C(c1cnc(OC)s1)=O)C3 C12(CC(=O)NOCCCC3CC3)CCCC1CN(C(c1ccccc1)=O)C2 CCC(C)CC(=O)N1CC(NC(c2ccc(C3CC3)s2)=O)C(CC)C1 Cc1cc(C(=O)NCC2COC(CNC(c3csc(C#N)c3)=O)C2)c(C)cn1 N1(C(C(C)SCC)=O)CC(NC(c2nc3cccnc3s2)=O)C2(CCC2)C1 C1(C(N2CC(OC)C(NC(C3(C(F)F)CCCC3)=O)C2)=O)CCCC2(CCC2)C1 C1(NC(c2cccc(CC)n2)=O)CN(C(C2C=CCS2)=O)C2CCCC12 N1(C(C2(C3N(C(c4cccc(CC)n4)=O)CCC3)CC2)=O)CCC(C)(CC)CC1 N1(C(=O)CSc2cccc(Cl)c2)CCN(C(=O)C2=CCOC2)C2CCC12 c1(CCC)ccc(C(N2CC3CC2C3NC(C2(C3CC3)CC2)=O)=O)cc1N C1(C(=O)NCCN(C(CC2CC(OC)C2)=O)CC2CC2)Cc2ccncc2C1 C1(CNC(c2c(C)ncnc2O)=O)C2CCCC1N(C(C1CC(C)OC1C)=O)C2 C(=O)(CC(CC)C(C)(C)C)N(C1(c2ccccc2)CC(O)(C(=O)NC)C1)CC C1(C(N2CCN(C(=O)CCc3cc[nH]n3)C(C(F)F)C2)=O)CCCC(F)(F)CC1 C1(C)(C(N2CCN(CC3CN(C(CCC#CC)=O)C3)CC2)=O)COC(=O)OC1 C1(F)(C(=O)NC2CC(C)(NC(=O)CCN3CCOC3=O)C2)C2CCCCC12 c1(C(N2CC3C(NC(C(CCCC)C)=O)(C3)C2)=O)cc(O)cc([N+](=O)[O-])c1 c1(NC(CCN(C)CCC2CCN(C(=O)CC(F)F)C2)=O)ccccc1 c12ccc(cc1)CN(C)C2=O.c1(C(=O)NCC2C(C)C2)cccc(C2CC2)c1 C1(C2CC2)(CNC(c2cc(CC(C)C)on2)=O)CCN(C(C2CNC(=O)C2)=O)C1 c1(C(=O)O)cc(NC2CCCCC2n2cc(CN3CC4CC4C3)nn2)cc(F)c1 Cc1cc(Cl)cc(Cl)c1OCC(N1CCN2CCCC2C1)=O C1(N(C)C)(CC)CCN(C(C2C3CC2N(C(=O)C(C)=C2CCCC2)C3)=O)C1 CC1(C)CCCC(O)(C(=O)NC2CCC2NC(c2cccc3nccn23)=O)CC1 c12ccnc(c1)C(=O)N2.c1(OC)cc(CO)sn1.C1(C)(C)CCNCC(=O)N1 c1(C(N2CCC(CNC(C3(OC)CCC3)=O)C23CC3)=O)cc2occc2n1C c1(C(=O)NC2CC(CCNC(C(C)(C)SC)=O)C2)n[nH]c(C)c1Br C1(NC(c2c(C)csc2)=O)CCN(C(c2cc(Cl)ns2)=O)CCC1CO C(C(=O)NCC1C=CCN1C(c1cc(C(N)=O)c[nH]1)=O)(C(C)(C)C)SC c1(OC)ccc2c(c1)CC(C(=O)NC(C1CCCCC1)C(C)NC(=O)C(F)F)O2 c1(C(=O)NCC(=C)CCNC(c2ccoc2C)=O)coc2ccc(C(C)C)cc12 c1(C2CCN(C(c3c(N)non3)=O)C2)ccc(F)cc1.c1(C(NC(C)C)=O)cccnc1 Cc1noc(C)c1CCNC(=O)CCN(C)C(C)C.C12CN(C1)C(=O)O2 N1(C(Cc2ncc(C)s2)=O)CC2C3CCC(C2C1)N(CC1CCOC(C)C1)C3 Cc1ccc(C(=O)NCCNC(=O)CC(=O)OC(C)(C)C)c2cccnc12 c1(C(=O)NCC2(OC)CN(C(C3(OC)CCC3)=O)C2)cn(C2CC2)nc1C Nc1ccc(C(N2CC3CC2C3NC(c2cnn(CCF)c2)=O)=O)c(Cl)c1 N1(c2nc(=NC)nc(N(CC#CC)C)[nH]2)CCC(C2CCN(C)C2)CC1 C1(CC(=O)NC(C#C)C2CCC2)CCN(C(=O)C(O)C=CCCC)CC1 C12(CNC(c3ncn(C(C)(C)C)c3)=O)CC(NC(C3C=CCC3)=O)(CO1)C2 Cc1cc(=O)ccn1CC(=O)N(C)CC1(O)CCN(C(=O)Cn2ccnn2)C1 c1(N2CCC(CNC(C(C)CCN(C)C)=O)C23CC3)ncnc2c1nnn2C C1(C#N)(C(=O)NCC(C)(C)OCCNC(=O)C=CC2CC2)C(C#N)C1(C)C N1(C(c2cc(CCNC(=O)CCc3cccs3)on2)=O)CCN2C(=O)OCC2C1 C(C(C)(C)CC(=O)NCc1cc(C(C)C)n[nH]1)NC(C1C(C)OCCO1)=O C1(C(N2C(C)CCC2)=O)CN(C(=O)CN2CCSCC2)CCC1(C)C NC(=O)C(O)CCCNC1CCCCC1OCc1ccccc1 N1(C(c2cc(C)[nH]n2)=O)CC(C)(C)CC1CC(=O)NOC(c1ccccc1)C c1(C(=O)NCCNC(C(C)NSS(C)(=O)=O)=O)ccc(C2(C(F)(F)F)N=N2)cc1 N1(C(c2c(CC)nn[nH]2)=O)CC(NC(=O)C(c2ccccc2)C)C(SC)C1 c1(CN2CC3CC3(C(=O)NC3CC(C(=O)O)C3)C2)c[nH]c2ccc(Br)cc12 N1(C(CC(C)N(C(=O)C(Cl)=CCl)CC)=O)CCN(C(=O)Cn2cnnc2O)CC1 Cc1ccnc(N(CC(C)C)C(c2ccc(C(F)C(F)F)cc2)=O)c1 c1(CC)ccc(CNC(=O)C(C2(O)CN(C(=O)CCOCC(C)(C)C)C2)F)o1 c1(C2(C(=O)NC(c3cn(C4COCC4=O)nn3)(C)C)CC2)cccc(Cl)c1 C[S+](C)CCC(O)C(=O)NCC1(C)CCN(C(=O)CC23CCCC2C3)CC1 C1(C(=O)NC2CC(F)(CNC(c3cc(C4CC4)no3)=O)C2)CCC2C1C2(F)F n1(CC)cc(CC(=O)NCC2CC(NC(c3cnoc3C3CC3)=O)C2)cn1 C=CC1OCCC1NC(c1nc(C)cs1)=O CC(C)CC(O)C(=O)NCCCCC1CN(C(=O)C(C(C)C)c2cccnc2)C1 c1(C(=O)NC2C(C(N(C(CC)C)C)=O)OCC2)ncccc1Cl CCCC(C#N)C(=O)N1CC(CNC(c2cnc(C3CC3)nc2)=O)C(O)C1 CCC(CC)C(C)C(=O)N(C(C)C(=O)N(C)CC1CCCCC1O)C CC1(C)CCCOC1C(N1CC(CNC(c2cc(=O)cc[nH]2)=O)CC1(C)C)=O CC1(C#N)CCCN(C(=O)C(C)(C2CCC2)NC(c2nsnc2O)=O)C1 c1(C(=O)NCC(C(=O)OCC)CC)cc2cc(C)cc(C)c2[nH]1 CC1CC=C(C(=O)NCC(O)CCNC(=O)C=CC(F)(F)F)CC1 C1(C2CCC2)(CNC(CN2C(C)CC2)=O)CCN(C(c2cn[nH]c2)=O)CC1 N1(C(CCC)=O)CCCC(C(N2CCC(N(C)C(c3cc(Cl)n(C)n3)=O)C2)=O)C1 CC(C)C(CNC(c1csc(O)n1)=O)NC(=O)C=CCn1cncn1 N1(C(c2ccc(C(F)(F)C(F)F)cn2)=O)CC2CC1CN2Cc1ccccc1 c1(CNC2C(C(N(C(C)C)CCO)=O)C2)cc2ccccc2nc1O N1(C(CC(C)NC(C(C)c2ccsc2)=O)=O)CC(C)C(C)C1C Cc1cc2c(C(=O)N(C(C)CNC(C3CCC4(CCC4)C3)=O)C)cccc2o1 c1(C(=O)NCCC(C)NC(=O)C(C)Cc2ccco2)ccc(F)c2cnccc12 c1(C(=O)NC(CC2CN(C(c3c(C)onc3)=O)C2)C)cccnc1C(F)(F)F c1(OCC(N2C(C(C)NC(=O)C3=NNC(=O)C3)CCC2)=O)cccc([N+](=O)[O-])c1 C1(F)(CNC(c2cccc(F)c2F)=O)CCCN(C(=O)C(C2CCOCC2)O)C1 C(=O)(CC(C(C)(C)C)NC(C1CC2(CC2)C1)=O)N1CCC(C(C)C)C1 C12(NC(CC3(C)CC3(Cl)Cl)=O)CCC(C1)N(C(c1ccc(O)cc1)=O)C2 c1(C(CC)(C)C)ccc(C(C)NC23CC4CC2C3C4)cc1 C1(NC(C2CCC(C(=O)O)C2)=O)CCC(NC(C2CC(n3ccnn3)C2)=O)CC1 c1(C(N2CC(O)CCC(N(C)C(C3CCOC3)=O)C2)=O)cn2cccc(Cl)c2n1 C1(NC(C2CCSC2)=O)CN(C(C2CS(=O)(=O)C2)=O)CC2(CC2)C1 C1(C)(C(=O)NC(CCC)CCCNC(c2ccc(C)o2)=O)CCS(=O)(=O)CC1 C1(NC(CN(CCCCCC)C)=O)CC2(C1)CN(C(C1CCOC1C)=O)C2 c1(C(N2CC3CCC(C2)N3C(=O)CC2CCOC2)=O)ccc2c(c1)OC(F)(F)O2 CCC(CCNC(=O)CCCn1cc(C2CC2COC)nn1)C1CCC1 C1(C(=O)NC2C(NC(Cn3nnc(C)n3)=O)C2)CCc2ccccc2O1 N1(C(C(CC)N(C)Cc2ncnn2C)=O)CC(NC(=O)C2CC2)CC(C)C1 c1(C(=O)NC2CN(C(C=CS(C)=O)=O)CC2O)cc(F)c(Br)cc1F c1(C(c2nnnn2CCCF)NC(C(=C)C)C2CC2)c(C)ccnc1C C(=O)(C1CCCc2n[nH]cc21)NCC1C(C)CCN1C(=O)CCc1cnoc1 c1(C(=O)NCC2(CNC(=O)C=CC3CCOCC3)CC2)cc2cc(O)ccc2[nH]1 c1(C(=O)NC(CNC(C2CCC(=O)N2C2CC2)=O)C2CC2)cc2cnccc2o1 CC1(C#CC(=O)N2CCOC3(C2)CN(C(=O)C#CC2(C)CC2)C3)CCCO1 CC1CC2CCC(C(=O)NC(C)CCCCNC(=O)CC3(O)CCOC3)CN2C1 c1(C(N2C(CC(=O)NCC(O)CO)CCC2)=O)ccc(O)nc1 c1(CN2CC(CC(N3C4CCC3COC4)=O)C2)c(Br)ccc(F)c1F c1(N(C(CCOC)=O)C(=O)CN(C)CCCCN=[N+]=[N-])ncnc2[nH]cnc12 N1(C(c2c(C)onc2)=O)C2CCC1C(CNC(=O)Cc1csc(Cl)c1)C2 Nc1cc(C(=O)NC(=O)C(O)Cc2ccccc2)cnc1Cl.C12CC1CNC2 CCCCCCC(C)C(=O)NC1COCC1CNC(=O)CC1(SC)CCC1 c1(C(=O)NCCC(Cc2ccccc2)NC(COC)=O)cn2cccc(C)c2n1 c1(-c2cnn(-c3c(OC)cccc3)n2)ncc(F)cc1N c1(C(N2C(CNC(=O)CC3CC3C3CC3)C=CC2)=O)ccccc1C(F)F CC1CCC(CNC(=O)CCc2ccc(Cl)cc2)N(C(=O)COCC(C)(C)C)C1 C1(CCCC)CN(C(C2NC(=O)C3CC23)=O)CCN1C(=O)C1=CCCC1 CCCC(CC)CC(=O)N1CCC(OC2CN(C(c3cnn(C)c3N)=O)C2)CC1 c1(C(C)O)ccccc1C(=O)NC1(C)CCN(C(=O)CC2(C(F)(F)F)CCC2)C1 c1(C(=O)OCC)cc(C(N2CC(C(=O)NCCCCC3CC3)C2)=O)no1 c1(C(=O)NC(c2c(C)ccc(C(=O)OC)c2)C)ncc(F)c2ccccc12 C1(NC(COc2ccn(C)n2)=O)CCCCC1C(=O)NCC(F)(F)CO Cc1cnccc1C(C)C(=O)NC1CCCCC1N(C)C(c1cccs1)=O C1(C(N2CCN(c3ncc(C)c(C)n3)C(C(C)C)C2)=O)CCOC2(CCCC2)C1 c1(CC)cc(NC(c2ccc(Oc3ccc(C)nn3)cc2)=O)cnc1C n1(CCC(N2C(CNC(C(C)OCC)=O)CC(O)C2)=O)cnc(C)cc1=O C(=O)(CCCC(F)(F)C(F)(F)F)N1CC(NC(=O)CC(C)(C)CN(C)C)CC(C)C1 c1(C(=O)NCC2C(C)CCN(C(COCC)=O)C2)cccc([N+](=O)[O-])c1OC C12(C(=O)NC(C(=O)OCC)CCc3ccccc3)CCC(CC)(C1)OC2 Cc1cc(C#N)nc(NC23CCCC2CN(C(c2cn(C4CCC4)nn2)=O)C3)n1 c1(C(=O)NCc2nnc(C)o2)ccc(S(=O)(=O)N2CCCCC2)o1.C12CCC1C2 c1(CC(OCC)OCC)cn(CCNC(=O)CCn2ccnn2)nn1 c1(C(=O)NCCC2CCC2)cncc(-n2cc(C3CC3)nn2)c1 c1(C(=O)OC)ccc(N2CC(CCCCNC(c3cnc[nH]3)=O)C2)nc1 c1(OC)ccc2c(c1)C(CCNC(c1cccc(C)c1)C1CCCO1)=CC2 N1(C(Cc2c(CC)con2)=O)CCC(O)(CNC(=O)C(C)(CO)NC(C)=O)C1 CCCN=C(NCC1CC1Cl)N1CCC(F)(c2cc(OC)cc(C(N)=O)c2)CC1 c1(NC(c2n(C(CC)C)nnn2)c2ccc(C(F)F)o2)ccc2nncn2c1 C#CCC(O)C(=O)NC1CC(NC(=O)C(F)(F)c2ccsc2Cl)C1 N1(C(C(C)OCC#C)=O)CCOCCC1C(=O)NC(CC=C)C(=O)OCC C(=O)(C#CC1CCC1)NC1C(CNC(c2c(COC)cccc2)=O)CCCC1 C1(C(N2CC3C(NC(C=C(COC)C)=O)(C3)C2)=O)CC2(CC(C)=NO2)C1 N1(C(c2cnc(CC)nc2)=O)CC2CCC1CN(C(=O)CCc1cn[nH]c1)C2 O=C(C(C1=CCCSC1)N1CCSCC1C1CCC1)NCCSc1ccccc1Br N1(CC(=O)N(CC(C)NC(=O)CSC(F)F)CC)C(=O)c2ccccc2S1(=O)=O c1(OC)c(C(N2CC=CC(NC(=O)CSC(F)(F)F)C2)=O)[nH]c2ccccc12 [N-]=[N+]=NC1CN(C(C2(CO)COC2)=O)CC1NC(C1CN2CCCC2CO1)=O c1(C(=O)NCCN(C(CN(C)C(=O)OC(C)(C)C)=O)C)cc2ccsc2s1 c1(C(=O)NC2CC3CN(C(C(C)O)=O)CC2C3)cc(Br)c2c(c1)[nH]c(=N)n2C c1(OC)ccc(CN2CCNCC2C(=O)NCc2ccc(Br)cc2)c(Br)n1 N1(C(CC=CCC)=O)CC2CCC(C1)N2C(=O)Cc1nnc(S)n1C c1(COC)c(C(N2CC(CC(C)NC(C)=O)C2)=O)oc2ccccc12 N1(C(C2(C(=O)OCC)CC2)=O)CCCN(C(=O)CC2CC(C)N(C(C)=O)C2)CC1 N(C(=NCCCF)NCC1CC(C)C1)Cc1ccc(CC)c(F)c1 C12(CNC(CC(=O)OCC)=O)CCC(C1)N(C(=O)C(C)OC1CCCCCC1)C2 C1(NC(C2CC(N(C)C)C2)=O)C2CC(O)C1N(C(=O)C=CCN1CCOCC1)C2 c1(OCCCC(=O)NCCN(C(C2C(CCOC)C2)=O)CC)cccc(C)c1C c1(NC(c2ccnc(C)n2)=O)ccc(NC(c2scnc2C)=O)c(F)c1 c1(SC)cc(NC(c2cc(-c3ccn(C(C)C)n3)[nH]n2)=O)ccn1 C(CC(C(C)(C)C)NC(=O)C1=C(Cl)CC1)N(C(CCCN(C(C)C)C)=O)C C1(NC(COC(CC)(C)C)=O)CN(C(=O)C2=CC(C)(C)C2)CCC1C(F)(F)F C1(C(C)(F)F)(C(N(CCN(C)C(C2CCCS2)=O)C)=O)CCOCC1 C12(C)CCN(C1)C(=O)C2.C1(CN(C(C)=O)CC23CCC(C2)C3)CCCCC1F N1(C(C=CC=CC)=O)CCCCC1C1CCN(C(=O)C(C)n2cnnn2)CC1 N1(C(C2C(COC)C2)=O)CCN(C(=O)C=CSCc2ccco2)CC(C)(F)C1 C#CC1(CNC(=O)C(CC(C)C)NC(=O)C=CC=CC)CCOCC1 c1(C(=O)NCC2(C(=O)O)C(C)(C)C2)cc2occc2[nH]1 C1(C(=O)NCC2CN(C(C(C)OCOC)=O)C2)CN(C(=O)C(C)(C)C)CCO1 C1(CNC(=O)CN2CCOCC2)CCCCC1NC(=O)COC(F)(F)C(F)(F)F Cc1cc(C(N2CC3(NC(c4cc(C(C)C)[nH]n4)=O)CCC2C3)=O)cc(C)c1N C1(CNC(c2c(C(C)C)ccs2)=O)CCC2(CN(C(c3[nH]ncc3C#N)=O)C2)O1 C1(NC(C=CC(=O)N(C)C)=O)(CF)CCN(C(C2COC(=O)O2)=O)C1 CN1CC(O)CCC1C(=O)NCCn1cc(C(N2CCOCC2)CSCCO)nn1 N1(C(C(C)OC)=O)CCCCCC1CNC(c1ccc(Br)nc1O)=O N1(C(Cn2ncc(C)c2)=O)CCC(F)C(NC(c2nc(C)oc2C)=O)C1 c1(C(CNC(=O)C(C)(O)C2CCC2)NC(C2(C)CC2(F)F)=O)ccccc1F c1(C(=O)NC(CC(=O)NCC(=O)NCC)C)nnn(C)c1N Cc1ccc(C(=O)NCCCC2CCCN2C(C23COCC2C3(F)F)=O)nc1C C(=O)(CCCN(C(=O)CC1CC1CNC(=O)Cc1cscn1)C)OC C(=O)(C1=CC2CC(C1)CC2O)NCC1C2CN(C(CSCC=C)=O)CC1CC2 C=CCCC(C(=O)NC(C)(C)C)N1CCC(CO)C(C)C1 CCC(S(=O)(=O)NC(C1CCC(N)CC1)=O)c1ccccc1 C1(C(=O)NC(COC)C)CN(C(C2CCCCC2C(C)(C)C)=O)CC1(F)F C(=O)(C1=C(C)CCCC1)N(C1CCN(C(c2cc(C(N)=O)[nH]n2)=O)C1)CC C1(OC)C(NC(=O)CCc2nnc(CN)s2)CC1(C)C N1(C(c2n(CC)ccn2)=O)C2CCCC1CC(N=c1[nH]c(Cl)ncc1C(C)C)C2 N1(C(C=Cc2cn(C)nc2)=O)CC2CCCN(C(C34COC(CCO3)C4)=O)C2C1 N1(Cc2ncc(C3CC3)s2)CCOC2(CCCNC2)C1 c12ccc(O)c(c1)C(=O)NCC(=O)OC2.N1(C(C)=O)CCOC(CNC(C)=O)C1 c1(CNC2(CC(=O)Nc3n(CCOC)ncc3)CCC2)cc(C)cc(F)c1 c1(C(=O)NCCC2CCN(C(C3CCNC3=O)=O)C2)cccc2c(O)nncc12 C1(NC(c2c(OC)n[nH]c2)=O)CN(C(=O)C(C)(F)F)CCC1C N1(C(CCC(=O)NCCC)=O)CC2CC(N=c3[nH]c(Cl)ncc3F)C2C1 CC(CC(=O)NC1(CNC(c2ccccc2C2CC2)=O)CC1)C(F)F C1(CN(C)C(=O)C2CC2)CCN(C(C2CC(N(C)C)C2)=O)CC1 N1(C(CC(CC)O)=O)CCCC2(CCCN(c3ncnc4[nH]cc(I)c34)C2)C1 N1(c2nc(COC)nc(C)c2)CC2CCC1C1CN(C(C3CC3(C)Br)=O)CC21 C1(C)(CNC(C2CCN(C)CC2)=O)CCCN(C(=O)CCCNC(=O)C(C)(C)C)C1 N1(C(c2c(C)oc(Cl)n2)=O)CCC(C)(C)C(CNC(C2CCCN2C)=O)C1 C1(NC(c2c(CCC)nco2)=O)CCN(C(=O)CC2CCCC(C)(C)O2)CC1O CC(C)(CC#N)C(=O)NC1CC1NC(=O)CCC1CCC(Cc2ccccc2)O1 C12(NC(C(CCSC)O)=O)CCCC(NC(=O)CCc3ccc(N)cn3)(C1)C2 c1(C(N2C(C)CC(CNC(CN(C)CC)=O)C2)=O)cc(Br)cc2c1OCO2 C(=O)(C1=CCCCC1C)N(CCOC)CCNC(=O)Cc1ccc(OC)cc1 C(CCCl)(CCCl)(N(C1CCSCC1)C)C1CC1c1ccccc1 N1(C(COCC=C)=O)CCC(C)C(CNC(=O)Cn2cccn2)C1 CC(C)CC(c1ccccc1)NC(=O)OCC(C1CCCO1)C1CCC1 C(=O)(C(CC1CCCC1)NC(C1CC(CF)C1)=O)NCC(=O)NC1CCCCC1 CC1(C)C(=O)CC1(P(C)(C)=O)CNC1CCC2CNCCN12 C(=O)(C#CC1CCOC1)N(CC)CC1CCCCN1C(c1ccsc1)=O c1(OC(C)C)ccc(=NC(=O)CC2CCCN2Cc2cccc(Br)n2)[nH]n1 N1(C(c2ccc(CN3CCN(C(=O)CO)CC3)o2)=O)CCOC2COCC12 c1(C(=O)NC2C(OC)CN(C(C3N(CC)C(=O)CC3)=O)C2)cnc2[nH]ccc2n1 C=C(C)CC(C)C(=O)NCC(C)N(C(=O)CCc1ccc(OC)c(Br)c1)C CCS(=O)(=O)CC(=O)NNC(=O)C(C)(C)CCCCNC(C1CCCCO1)=O N1(C(Cc2nc(NC=O)sc2)=O)CCN(C(=O)Cn2nnc(=O)[nH]2)C2CC12 c1(C(N(C)CC2CCN(C(C3(CO)CCC3)=O)C2)=O)csc2ccncc12 c1(C(N2C3C(NC(CCc4ncn(C)c4)=O)C(C3)C2)=O)ccc2ncccc2c1 Cc1cc(=NC(=O)C(C)NC(c2cc[nH]c2C2CC2)=O)[nH]n1C C(=O)(C(C)CCCCCC)NCCC(C(=O)C(CCCC)N(C)C)C=C N1(C(CC(CC)CN(C)C)=O)CCC(NC(c2cc(CO)[nH]n2)=O)CC(C)(C)C1 S(=O)(=O)(c1ccc(NC(C2CCOCC2)C)cc1Br)NCc1nnc(COC)s1 C1(N(C(C2C(=C)C2)=O)CC)CCCN(C(c2cc(OC)cc(Cl)c2)=O)CC1 CC(C)(CCN=c1ncc2ccccc2[nH]1)NC(C1(c2ccc(F)cc2)CC1)=O CCC1=C(C(=O)NCCOC(C)(C)CNC(c2c(C)noc2CC)=O)CCCO1 N1(C(CCCC(=O)NCC)=O)C2CCC1CN(C(=O)C(C)C(O)CC)C2 C1(C(=O)NC(c2ncc(C)o2)C)C(C)OCCN1C(=O)C(C)N=[N+]=[N-] N1(CC)OCC(NC(=O)CC2(C)CCN(C(C3SCC=C3C)=O)C2)C1=O CC1COCC(C(=O)NC(C(=O)NCCC2CC=CC2)C(C)O)O1 N1(C(CC(=O)NCC#C)=O)CCC(C)C(NC(=O)CCN(S(C)(=O)=O)C)C1 c1(C(=O)NC(CN(C(CN(CCC)C)=O)C)(C)C)cccc(C2CNC(=O)C2)c1 c1(C(N(C2CN(C(C(C)OCC#C)=O)CC2(C)C)C)=O)cccc2nn(C)nc12 N1(CC(NOC(CC(C)C)C(=O)O)=O)CCC23CCC(CC12)C3(C)C c1(C(=O)NC2C3CN(C(CC=CC=C)=O)C2CC3)ccc2cnc(C)n2c1 c1(CC)onc(C(N2CCCC2C=CC(N2CCCCC2C2CCC2)=O)=O)c1C C1(NC(CC(CCC)C)=O)CN(C(=O)CCc2cc(C)[nH]n2)Cc2ccnn2C1 C(=O)(C(C)(C)CC(=O)NC(C)(C)CNC(=O)CCN1CCC(F)C1)OC N1(C(CN(C(=O)OC)C)=O)CCC(NC(=O)C(C)CC(F)(F)F)C12CCC2 C=CC(C)CC(=O)N(C)CC1CN(C(c2coc(C(C)(C)C)n2)=O)CCO1 S(=O)(=O)(c1cnc(Cl)nc1)N1C(C(N2CC3CCC2C3)=O)CC2CC21 C1(CNC(c2ccc(F)c(CO)c2)=O)CCCN(C(C2CC2C(F)F)=O)CC1 c1(C(=O)NCC(C)(C)OCCN(C)C)cncc2c1CCC2.N12CC(C1)C2=O c1(C(N2CC(CNC(c3cc(CCC)nn3C)=O)(OC)C2)=O)cc(C)c(O)nn1 C1(O)(CNC(CCNC(C2CCCCC2)=O)=O)CCCN(C(C2CCCO2)=O)C1 c1(C(=O)NCCOCCNC(c2c(C)cnnc2)=O)ccc2cc(F)ccc2n1 C1(CNC(N2C(C#C)CCCCC2)=O)CCCCC1C1CC1 Cc1ccc2c(c1)CCC(C(=O)OCc1cn(C(c3ccccc3)(C)C)nn1)O2 N1(C(c2ccc(C#C)c(Cl)c2)=O)CCOC2(C1)CN(C(c1cc(O)n(C)n1)=O)C2 N1(C(C23CC(OC)C2C3)=O)CCC(NC(=O)C(c2cccn2C)=O)CC1 CCC(C)CC(=O)NCC1(c2ccccc2)CC(NC(=O)CNC=O)C1 C(=O)(C1Cc2ccccc21)NCC1CN(C(c2ccnc(C)n2)=O)CC1O c1(C(=O)NCCCC(C)NC(c2ccncc2)=O)cccc(C2(F)CC2(F)F)c1 c1(OC)cc(CC(N2CCC(O)C(NC(=O)CC3CCCOC3)C2)=O)ccc1C Nc1cc(F)ccc1C(N1CCN(c2ccccc2Br)CC1)=O C1(NC(c2ccc(Br)cc2)=O)CN(C(=O)Cc2cnccn2)CCC12CCC2 N1(C(CC(=C)Br)=O)CC(CNC(c2ccc(OC)nn2)=O)CC12CCC2 C(CN=c1nc(N2CC(CO)C3(CC3)C2)c2c([nH]1)CSC2)c1ccc(C)c(F)c1 C1(CC(C)NC(c2cccnc2)=O)CCN(c2ccnc(C3CCC3)n2)CC1 C1(CNC(C2(SC)CCC2)=O)CCN(C(=O)CC2CCOC2C)CC1 C(=O)(C1SCc2cccnc21)N1CC(C(=O)NCC2(CO)CCC2)C1 c1(OC)cc(C(=O)NC(C(C)NC(C2CC3CC2C3)=O)C(C)C)ccc1Cl N1(CCC)CCCCC1C(N1CCC(F)(CNC(c2coc(C)n2)=O)C1)=O C(=O)(CCC(=O)NC1CCCN(C(=O)CN2CCCC2=O)C1)N(CC)CC c1(C(C(=O)NCCS(CC)(=O)=O)NC(=O)Cc2cc[nH]n2)c(C)cccc1Br C12(C(N(CC(CC)(O)CC)C)=O)COCC1CN(C(C1CCCC(C#N)C1)=O)C2 C(=O)(C(C(C)CC)NC(C12CCCC1CCC2)=O)NC N1(C(CC2C(C)OCC2)=O)CCN(C)C(CNC(c2ccccc2C(F)F)=O)C1 C1(CCNC(C(CC)OC)=O)CCN(C(=O)C(C)(C)COc2ccccc2)CC1 Cc1cc(Cl)ccc1C(=O)Nc1cc(-c2ccccc2NS(C)(=O)=O)ccn1 c1(C(=O)NCC(C)(C2CC2)NC(=O)Cn2nccn2)cc(F)ccc1Cl C(=O)(C(F)C(C)(C)O)N(C1CCN(C(CC(=C)Br)=O)CC1)CC C1(C(C)(C)C)(CNC(C2(CC#C)CC2)=O)CCN(C(c2ccc(F)cn2)=O)C1 c1(NC(C2CCC(C(C)C)N2C(=O)C=CCF)=O)cc(F)c(O)cc1C n1(CC(=O)NC2C(NC(CC3(C)CCCCC3)=O)C2)ccc(O)nc1=O Fc1ccc2c(c1)C(c1nc(-c3cncnc3)nn1C13CC(C(F)F)(C1)C3)CO2 n1(C2(C(N(CCCNC(C3CC(O)C3)=O)CCO)=O)CC2)cc(Br)cn1 c1(NC(CC)CNC(c2ccsn2)=O)nccc(-c2ccccc2)n1 C(=O)(C(C(C)(C)C)NC(N)=O)NCC(C)NC(C(C)CC1CCCC1)=O C(=O)(C1CCCc2cncn21)N1CCCC2(CN(C(C3C(=C)C3)=O)C2)C1 N1(C(C2(C=C)CCN(C(C3OCCCC3(C)C)=O)C2)=O)CC(OC)C(C2CC2)C1 c1(C(N2CCCN(C(C3CCCN3C3CC3)=O)CCC2)=O)ncc2ccccn12 O=C1CCN(CCC2OCCO2)C(=O)N1CC1CC1c1ccco1 c1(OC)ccc(NC(=O)C(C2CCN(Cc3cccs3)CC2)C)c(C)c1 c1(C(=O)NC2C(NC(c3cc(C)c(O)cc3)=O)CC2)cc(P(C)(C)=O)cs1 C1(CNC(CCOCCNC(C(CC)=CC)=O)=O)CCCCC(O)C1 c1(C(=O)OCC(c2n(CC)cnn2)=O)ccccc1N(S(C)(=O)=O)C c1(OC)ccccc1OCC(=O)NC1C=CCN(C(C2C=C2C)=O)C1 O=C(CS(=O)(=O)CC1CCCO1)NCCC1(CNC(=O)C2=CCCCO2)CC1 N1(C(C2CSCCN2C(C2CC2C(F)F)=O)=O)CCCC2(CC(O)C2)C1 c1(N(C)Cc2ccoc2)nc(NCc2cc(Cl)ccc2CO)c2ccsc2n1 Cc1cccc2c(C3CCN3C(C3Cc4ccccc4S3(=O)=O)=O)c[nH]c12 c1(C(=O)NCCN(C(c2ccc(F)cn2)=O)CC)cccc(C)c1[N+](=O)[O-] c1(CN(C(=O)CNC(=O)CC2CC2)CC)cccnc1 C1(NC(C(C)N(C(C2(OC)CCCC2)=O)C)=O)CCN2CCC1C2 Cc1c[nH]c2ncc(C(N3CC(NC(C4NC(=O)CC4C)=O)CC3C)=O)cc12 C1(c2ncn(C)n2)CCN(C(c2csc(C3CCCCC3)n2)=O)CC1 Cc1ccc(OCCC(=O)NC2CCC2NC(=O)C(O)c2ccco2)c(C)c1 CC1(C)CC2(CC(C(N3CCC(OCCNC(=O)C(F)(F)C(F)(F)F)C3)=O)C2)C1 C1(CCO)CCC(N=c2nc(N3CCC4(CCNC4=O)CC3)c3sccc3[nH]2)C1 C1(NC(COC(C)=O)=O)CCC(N(C)C(c2sc(Cl)cc2Cl)=O)CC1 c1(OC)cc(CN2CC3C(C2)N3C(c2cccc(F)c2Br)=O)c(Cl)cn1 Cc1cccc2c(C(=O)NC3CC(C)(NC(=O)CNc4ccccn4)C3)coc12 Cc1ccc(Cl)c(C(=O)NC(C2(O)CCN(C(=O)C(C)C3CCOC3)C2)C)c1 c1(C(=O)NC)cc([N+](=O)[O-])ccc1N1CC2(CN(C(=O)CC(C)SC)C2)C1 C1(CNC(CNC(C)=O)=O)CC(CNC(c2ccc(CNC(C)=O)o2)=O)CO1 N1(C(CCC#C)=O)CCC(NC(=O)CCSCc2ccccc2)CC1C1CC1 N1(C(c2ccnc(N3CCCCC3)n2)=O)CCc2c(I)n[nH]c2C1 C1(NC(CNC(CNC(C2CC(C(N)=O)C2)=O)=O)=O)C2CCC(C2)C1CO C1(CC#C)(C(N2CC(OCCNC(=O)CCc3cccnc3)C2)=O)CCCCO1 c1(N(C(=O)NCCN2CCCCC2)CCc2ccccn2)nsc2ccccc12 C(=O)(C#CC1CCOC1)N1CCC(C)(NC(c2c(C)ccc(CC)c2)=O)CC1 c1(CCCC(=O)N(CC(C)(C)NC(C(C)C(C)(C)C)=O)C)nc2ccccc2[nH]1 C1(O)(CCNC(=O)Cn2cnnc2O)CCN(C(=O)COC2CCOCC2)C1 CCCC(CC(=O)NC(C)C(N)=O)NC(C1C=CCC1)=O N1(C(c2cc(C)[nH]n2)=O)CCC(C)(C)C1CC(N1CC(OCC(N)=O)C1)=O Cc1cc(Br)ccc1CC(=O)Nc1c[nH]nc1C(=O)NCc1ccc[nH]1 CC1=CC(C)CN(C(=O)NCc2cccnc2N(C)C)C1 c1(C(N2CCN(Cc3cc(I)c(C)c(I)c3)CC2)=O)cccc([N+](=O)[O-])c1 Cc1cccc2c1OCC2C(=O)NC(C)C(C)(C)NC(=O)C(F)=C1CCCC1 N1(C(c2nc(N(C(C)=O)C)sc2)=O)CCN(C2CCCNC2=O)CC(O)C1 C(=O)(C(C)(C)C(=C)C)N1C(C(CN(CC=C)CC2CCCC(O)C2)C(=O)O)CCC1 C1(C(=O)NC2(CC(=O)OC)CC2)CCC(C)CN1C(=O)CC(C)F N1(C(CC=C)=O)C2CCC1CN(C(=O)C(O)C1CC1)C2 C1(CNC(C(C)(C)NC(=O)OC)=O)CC(C)N(C(c2ccc(C(N)=O)[nH]2)=O)C1 CC1CCCCC1(C)C(N1CCC(C(=O)Nc2ccccc2)C(C)C1)=O C1(C(=O)NC(CNC(Cc2cn(C)nc2)=O)(C)C2CC2)Cc2cc(Cl)ccc2O1 c1(C(N(C)CC2CN(C(C3CN4CCN3CC4)=O)C2)=O)ccc2c(c1)ncn2C C(=O)(CCC1=CCCCC1)N(CCC(N1CCC(N(C)C)C1C)=O)CC c1(CC)nc(N(C)CCN(C)C(c2ccc(Cl)c(C(F)F)c2)=O)cc(C)n1 C12(NC(C3C(NC(c4cccc(C)c4F)=O)CCOC3)=O)CC3CC(CC1C3)C2 C1(C(N2CC(C(N)=O)(CNC(CCC3CC(C)C3)=O)C2)=O)CC(=O)CCO1 C(=O)(N=c1cnn(C2CCOCC2)[nH]1)N(C(C#N)C(N)=O)CC C(=O)(C(O)CC[S+](C)C)NCC(CC1CN(C(CC(C(C)C)O)=O)C1)(C)C c1(CNC(C2C(CNC(C3C(C(=O)OCC)C3)=O)CCC2)=O)ccc(O)c(C)c1 C1(N(CC(CC)C)C)CCN(C2CCN(C(C3CCCC3C)=O)CC2)CC1 Cc1nccc(C(=O)NCC2CCC(NC(c3ccnnc3Cl)=O)C2)n1 N1(C(c2cccnc2)=O)CC2CCC(C1)C2CNC(C12COCC1C2)=O C(CCCCC(=O)NCc1cccc(O)c1)N(C(=O)CC1CCC(=O)C1)C c1(C(=O)NC(C)C(C)(C)NC(=O)CC2C=CS(=O)(=O)C2)ccc2nn[nH]c2c1 c1(C(=O)NCC(C2CCCCC2)NC(CC(C(C)C)O)=O)cc(F)cc(Cl)c1N CC(C)CC(C(=O)OCc1cc(C(F)(F)F)co1)C(C)C C1(C(N2CC(NC(=O)CC(=O)N(C)C)CC(C)(C)C2)=O)CC2OC(C)(C)OC2C1 c1(C(c2n(C(C)C)nnn2)NCCCn2ccnn2)cnc(N(C)C)cn1 C1(NC(CC2CC(C)N(C(C3CC4(CC4)CO3)=O)C2)=O)CCOC2(CCC2)C1 N1(C(COC)=O)CCC(=C(c2ccccc2)NC(c2cccnc2SC)=O)CC1 Cc1c(C(=O)N(CC(C)(C)CNC(=O)CC2NC(=O)NC2=O)C)ccn1C c1(C(N(CCCNC(C(C)C(F)F)=O)C2CC2)=O)n[nH]c2c1CC(F)(F)CC2 N1(C(COCCCCC)=O)CC2CC(NC(c3cccc(OC)n3)=O)C1C2 c1(C(=O)NC2(C)CC(NC(c3c(C)cc(C(F)(F)F)s3)=O)C2)ccc([N+](=O)[O-])[nH]1 N1(C(c2c(C)occ2)=O)CCCN(C(C2CCN(CCO)C(=O)C2)=O)CC1CO C1(C(=O)NCC(CC)NC(=O)CCCCOC)CCCN1S(=N)(=O)N(C)C c1(OCC)cncc(C(=O)NCC23CC2CN(C(C2CN(CC)C2)=O)C3)c1 C1(NC(C(CO)OC)=O)CN(C(=O)C(c2ccccc2F)C)C2CCCC12 CCC(CNC(c1cccc(F)n1)c1nnnn1CCOC)(CC)C(F)(F)F Cc1ccc(C)c(CC(=O)NCCNC(=O)C(c2cccc(Br)c2)C)c1 C12(C(=O)NCC3C(NC(c4c(CC)occ4C)=O)C3)CCC(CC1)C(C)(C)O2 C1(C)(CNC(C2N(CCC)C(=O)CC2)=O)CCN(C(C2(CCO)CC2)=O)CC1 C(=O)(C1=C(CC)OCCS1)NCC(CC)(CC)NC(=O)CC(C)(F)F N1(C(c2cc(C(C)C)on2)=O)CC2CCC(C(N3CCC(F)(C(N)=O)C3)=O)(C2)C1 n1(CC)nc(C)c(C(=O)NC2CC(CC(N3CCCC(C)CC3)=O)C2)c1C C(=O)(CCCCCNC(=O)C(C)(C)C)N1CCC(C(C)O)C1 C12(C(N3CCC(C)(NC(C4CCCCC4)=O)C3)=O)CCC(CC1(F)F)C2 c1(CNC(C2(NC(CCc3ncn(C)c3)=O)CCCC2)=O)cc(F)ccc1O CCCC(C(=O)NCCCOCCCNC(c1ccoc1Cl)=O)c1ccccc1 CC1Oc2ccccc2N(CCC(=O)Nc2cn(C)nc2Cl)C1=O C=C(C)c1cncc(C(N2CCOC(COC)CC2)C(=O)NCc2ccco2)c1 N1(C(CCc2cncc(C)c2)=O)CCCCC12CCCN(C(=O)C(C)NC=O)C2 c1(C(=O)NCC2CC2NC(C2CCC(F)(F)CO2)=O)ccn2ccccc12 N1(C(C2(OC)CCSC2)=O)CC2(CCCC(CNC(=O)CCCOC(C)C)O2)C1 N1(C(c2scc(OC)c2)=O)CC(C)(C)CC1CNC(c1cc(C)sc1C)=O c1(C(N2CCCN(C(C(CCC)C(C)C)=O)CCC2)=O)cccc2c1C(=O)CC2 N1(C(C2CC(NC(C3C(C(=C)C)OCC3)=O)C(O)C2)=O)CCN(C)C(C)(C)C1 CC1(C)CC(=O)NC1NC(=O)Cc1nnn(C2CCCC(=O)N2)n1 CC(C)CC(O)C(C)C(=O)NCCOCCN(C)C(c1ccc2cnnn2c1)=O C1(CCNC(CCC=CC)=O)CC(F)(F)CN1C(=O)C(c1ccc(F)cc1F)=O N1(C(CC(C)C)=O)CCN(C(C2CCC(C(C)C)CC2)=O)CC(C)(C)C1 C(=O)(C#CC1CCOCC1)N(CCC(C)(C)NC(c1cccc(CO)n1)=O)C c1(C(N2C(C(=O)NC3CCCN(C)CC3)CC3CC32)=O)ncc2ccccn12 C1(CCCC)CCC(C(=O)NC2(CNC(=O)COC(F)(F)F)CCCCC2)CC1 c1(-n2cc(CCC)nn2)cccc(C(C(=O)NCCN(C2CC2)CC)OC)c1 N1(C(c2cc(C)c(C)nc2O)=O)CCC2CCC(C1)N2C(C12CC(C)(CO1)C2)=O N1(C(c2ccc(OC)c(F)c2)C)CCNC1=NCCC(C)F C1(NC(c2n(CC)ncc2)=O)CC2CCC(C1C)N2C(=O)CC(C)n1ccnc1 c1(C(=O)NC2CCN(C(C3C(C)CC3)=O)CC2)ccc(F)cc1O C(C=O)(C(C)O)NCC(=O)O.c1(CC(=O)NC(CC)(C)C)csc(-c2ccoc2)n1 c1(CNC(C(C)NC(=O)Cc2ccccc2)=O)cnn2c1CNCC2 C(=O)(C1CCCc2nn[nH]c21)N(C1(CNC(=O)CN2CC3CC3C2)CCCC1)C Cc1scc(CNC(=O)COC2CN(C(C3(C#N)CC=CC3)=O)C2)c1C C1(OC)CN(C(=O)C(=Cc2cn[nH]c2)C)CC1C(=O)NC1CCC(=O)NC1 C12CC(CCO1)NC(=O)NC2.C1(C2CCC2)(C(=O)NCC2CC2)CC1.c1cccnc1 C(=O)(CS(=O)(=O)CC(=O)N(C)CC1CCN(C(c2ocnc2C(F)F)=O)C1)OC CC(C)CCCC(C)C(=O)N1CCCC(C)C1CNC(=O)CCC1(C)CC1 C1(C(C)NC(c2nc(C(F)(F)F)cs2)=O)CN(C(c2cnoc2)=O)CCO1 C1(C)(NC(c2c(C)occ2)=O)CCCN(C(=O)CC2CCCOC2)C1 C1CN=C2C=CC=C(S(=O)(=O)N1CCC)N2.n1(CCNCCCCO)ccnn1 Cc1nc(C(N2CCCC(CN3CCOCC3)C2)C(=O)N(C)C)nn1C CC(CNC(=O)CC1CCn2cncc2C1)CN=c1[nH]cc([N+](=O)[O-])cc1C#N C(=O)(CC(O)C(Cl)(Cl)Cl)NCCN1CCCN(C(CC)=O)CC1 N1(C(COCCCC#C)=O)CCCC(CCCCNC(C2CCN(C)C2)=O)C1 CCCCC(CC)CCC(=O)NCCC(C)(C)NC(C1CC(=O)NC(=O)N1)=O N1(NC(CCc2cn(CC)nn2)=O)CC(C(F)(F)F)CC1CO.c12ccsc1C2 c1(C(=O)NC2CN(C(=O)CC3(O)CCCC3)CC2F)cc([N+](=O)[O-])ccc1Cl C(N=c1[nH]cnc(Cl)c1F)C12CCC(CNC(=O)C=Cc3cocn3)(CC1)OC2 C1(C(N(CCOC)CCNC(=O)CCn2ccc(C)n2)=O)CC(F)(F)C1(C)C C1(CCNC(CC2(C)CCN2C(c2cc(Cl)c[nH]2)=O)=O)CCCC2CC12 C1(C(N(CCN(C)C(c2ncc(F)cc2F)=O)C)=O)CC(C)(C)CCO1 N1(C(C2(F)CCCN(C(CCC=C(C)C)=O)C2)=O)CCn2cnnc2C1 Cc1cn2ccc(C(=O)NC3COCC3NC(=O)C(C#N)C(C)C)cc2n1 C(=O)(CCCCc1ccccc1O)N1CCC(N2C(=O)CCC2)C1 c1(C(=O)Nc2ncc(-c3c(OCCC)ccc(F)c3)s2)nc2ccc(C)cc2s1 Cc1nccc(C(=O)NCC(C)(C(C)C)NC(c2cccc(OCF)c2)=O)c1C C1(C(C(C)NC(=O)CC2CCCC2)NC(COCC)=O)CCCCC1 C(C(=O)NCC(C)CNC(c1ncn(C)n1)=O)(C(C)C)NC(=O)OCC C1(C(=O)NCC(C)NC(c2c(C(F)(F)F)cnn2C)=O)CC12CC(C)(C)C2 C=CCC(CC)C(=O)NCC1(CO)CCN(C(=O)C(c2ccc(F)cc2)F)CC1 C=CC(C)(CC)C(=O)N1CC2CC(NC(=O)Cc3ccccc3C(F)(F)F)C2C1 C(=O)(C(F)CC(C)(C)NC(=O)CCn1cnc(=N)[nH]1)NC(c1ccncn1)C C1(NC(C(C)Cc2ccco2)=O)COCCN(C(c2cscn2)=O)C1 CN1C(=O)CCCC1C(N1CCCC(N(C(=O)CCC(=O)NS(C)(=O)=O)C)C1)=O N1(C(c2c(C)n[nH]c2)=O)C(C)CC2CN(C(c3ccc4ccnn4c3)=O)CC12 C=CCC(CNC(=O)CN1CC2CCC1C2)C(=O)NCCCOCC(C)C c1(C(N(CC(=O)NCCCCSc2nc[nH]n2)C2CC2)=O)cscc1F c1(OC)cccc(CCC(=O)NCC2(CNC(=O)COC3CCOCC3)CC2)n1 c1(NC(Cc2cccc(NC(Cc3ccc(C)nc3)=O)c2)=O)cnc(Cl)c(C)c1 N1(C(CSC(C)C)=O)CCOC2(CCN(C(C3CC3c3ccccc3)=O)C2)C1 Cc1cc(CC(=O)NCC(C2CC2)N(C(=O)CCc2cc[nH]n2)C)c(C)s1 C1(NC(C(CCF)NC(c2cn(CC)nc2C)=O)=O)CCC(=O)N(C)C1=O CC1(C)CN(C(c2cc(C(N)=O)no2)=O)CC1NC(=O)Cn1cnccc1=O c1(C(=O)NC2C(NC(C(c3c(C)noc3C)C)=O)CCCC2)cc2n(c1)CCC2 N1(C(c2c(C)onc2)=O)CC(NC(=O)Cn2cc3ncccc3n2)CC2(CC2)C1 C(=O)(CC(C(F)(F)F)c1ccon1)N(CCNC(C(C(C)C)SC)=O)C1CC1 N1(C(c2ccc(C)o2)=O)CC2C3CCC(C2C1)N(CCC1CCCO1)C3 c1(CC(N2CCC(C)(CNC(c3c(SC)nn(C)c3)=O)C2)=O)cc(Cl)ccc1Cl C=CC(CC)CC(=O)NC(C)(CNC(c1cc([N+](=O)[O-])c[nH]1)=O)C1C(CC)C1 Cc1nc(NCC2COCC2(C)C)cc(NC2CCN(C3CC3)CC2)n1 C1(NC(CCN(C)CC)=O)CN(C(c2cc(Cl)cnn2)=O)C2(CCCOC2)C1 C1(CC(=O)OC(C)(C)C)CCN(C(C2CC(C)(C)CO2)=O)C2(CC2)C1.CN1CC1 c1(C(=O)NCC(CCNC(C=C(C)C)=O)O)cc(Cl)ccc1OC(F)(F)F c1(SC)cc(C)c(C(=O)NC(C2CCN(C(=O)Cc3cn[nH]c3)C2)C)o1 c1(C(=O)NCC2(CCNC(C(C)SCCCC)=O)CC2)ncc(F)cc1C N1(C(C(F)=C(C)C)=O)CC(F)(F)CC1CCNC(c1ncoc1C1CC1)=O Cc1ccc(OCC(O)CSc2ccn(C(C)C)c2)c(F)c1 C1(O)(CNC(C2(NC(N)=O)CC2)=O)CCCN(C(c2ccon2)=O)C1 Cc1nc(C(=O)NC2CC(F)CN(C(C3CCC(O)CC3)=O)C2)c2n1CCCC2 C(=O)(C(C)(C)CS(C)(=O)=O)N1CC(OC)C(NC(c2cc(Cl)n(C)n2)=O)C1 c1(OC)ccc(F)c(C(C(=O)NC2COC2)N(C)Cc2nccs2)n1 c1(NC(=O)CC2CCC(NC(c3c(O)cccc3O)=O)CC2)cc(Cl)c(Br)cc1Cl N1(C(c2ccc(C(F)(F)F)cc2Cl)=O)CCC2(CCN(C(C3CCSC3)=O)C2)C1 C#CC1(NC(C2(CNC(=O)C(O)CCSC)CC3(CC3)C2)=O)CCC(C)CC1 N1(C(CN(C)C)=O)CCOCC1CC(=O)N(C)Cc1cccc(F)c1 c1(C(=O)NCCN(c2nnc(CO)s2)CC)c(C)oc(C)c1C C1(NC(CCN(C)CC)=O)CC2CC(NC(=O)C(C)Cc3ccccc3F)CC12 c1(C(N(C(CN(C(CC(=C)C)=O)C)C)C)=O)nc(C(F)(F)F)oc1Br c1(C(=O)NCC(C(C)C)NC(=O)CCc2ccc[nH]2)cccc2occ(Br)c12 C1(CCC(=O)NC2CC(C)(NC(=O)CC#N)C2)NC(=O)NC1=O C1(CC(=O)NCC(CN(C)C(c2cocc2C(N)=O)=O)O)CCCCC1O N1(C(C(c2c(C)noc2C)C)=O)CC2CC(NC(c3cn[nH]c3)=O)C1C2 Cc1ccccc1C=CC(=O)NC1C=CC(CC(=O)Nc2cncnc2O)C1 CC1CC(CNC(C2(S(N)(=O)=O)CC2)=O)CN1C(=O)CCNc1ccc(F)cc1 n1(CCC(=O)NCC(CNC(=O)C(O)CSC)OC)ncn(C)c1=O C1(C)(C(N(CC(CN(C(=O)CNc2ccccn2)C)O)C)=O)CC1(F)F C1(CNC(C2(OC)CCSC2)=O)COC(C)(C)CN1C(=O)COCC1(F)CC1 c1(OC)nccnc1C(=O)NCC(C1CC1)NC(c1cccc(OC(C)C)n1)=O Cc1ncc(C=CC(=O)NCCC2(C)CCN(C(C3CC(N(C)C)C3)=O)C2)s1 N1(C(C(=O)NCCCSCC)C2CCCC2)CCCCC1c1cccc(O)c1 CC(C)CS(=O)(=O)N(C1CCC(CN)C1)C C1(CC(N2CCC(C(C)(C)NC(=O)Cc3cnco3)C2)=O)CCCC(F)(F)C1 Cn1cnc(C=CC(=O)NC2CC23CC(NC(C2(C(=O)O)CCOCC2)=O)C3)c1 Cn1nc(CNC(=O)Cc2cncs2)cc1C(N1CCC(C)(C)C1)=O C=C(C)CC(C(=O)NC1CC2CC(NC(c3ccc(=O)n(C)c3)=O)C2C1)NC(C)=O N1(c2n(CCC#C)c(C3CC3c3ccccc3Br)nn2)CC2(C1)CC(C)(O)C2 C1(C(N2CCC(C(=O)N(C)C)C2)C(=O)NCCC)CCC2COCCC2C1 C1(CC(C)C)COCCN1C(=O)NC(C)CCc1cn(C)nn1 C(CNC(c1ccc(C(F)F)c(Cl)c1)=O)(CCS(C)(=O)=O)OC CC1CN(C(c2ccnc(C(C)(F)F)c2)=O)CCC1N(C(=O)CCOC1CC1)C C1(OC)CC2(C1)CC(C(=O)NC(C)CCNC(=O)CC(CC)OC)C2 C1(F)(CNC(C(c2cccs2)SC)=O)CC(NC(c2cnccn2)=O)C1 C1(C(C)C)CN(C(C2CCCCS2)=O)CCN1C(=O)CC1CCC(C)CC1 c1(CC(=O)NCC(=O)NCC(CO)NC(c2csnc2Cl)=O)ccc(Cl)cc1 C1(Nc2cc(OCC)ncn2)CC2(CCN(C(c3cc(Cl)ccc3C)=O)C2)C1 c1(CC(=O)NC23CC2CN(C(=O)C=Cc2cnccn2)C3)ccccc1C1CC1 c1(C(=O)NC2C(NC(c3c[nH]c(=N)o3)=O)CCC2)nc(Cl)sc1Cl C=C(Cl)C(C)(C)C(=O)NCC(CCOC)NC(=O)COC(c1nccn1C)C C1(O)(C(=O)NC2CCN(C(C34CC(CC)(OC3)C4)=O)C(C)C2)CCC(C)(C)CC1 CN1CCCC(C(N2CCCC2CCC(=O)NC(C2CCCO2)(C)C)=O)C1 C1(NC(C2CC3(CC3)C2)=O)CN(C(=O)C=CCO)CC1c1ccccc1 c1(SCC)ccc(C(N2CC(OC)CC2CNC(C2CCC(C)O2)=O)=O)cn1 c1(C(C)C)n[nH]cc1C(=O)NC(C1CCCC1)CNC(C1(C)CC(F)C1)=O C1(C(=O)NCC(C)(C)NC(=O)C(F)=C2CCC2)CCCN1C=O c1(OC)ncc(C(=O)NCCC2CC(OC)CN2C(=O)CC2CCCCO2)cn1 C1(N(C(C(C)N2CCCC2)=O)C2CC2(F)F)CCCC2CN(C(C(C3CC3F)=O)=O)CC12 C1(C)(C(C)C)C=CCN1Cc1ccnn1CCF c1(C(=O)NCC(CNC(COCCC(C)C)=O)O)n[nH]c2ccc(Cl)cc12 C(=O)(C(CC(F)F)NC(C1CC(C)(C)C1)=O)NC1(C)CS(=O)(=O)C1 Cc1cn(C)nc1C(=O)NC1CN(C(=O)CSC(C)C)CC1C(F)(F)F C1(CCNC(N2CC(NC(COC)=O)C2)=O)CC2CCC1O2 C1(N(C(=O)C=C2CC2)CC)CCCN(C(=O)C(C)OC)C1 C1(C(N2CCC(=C)CC2)=O)CN(C(=O)C(C)NC=O)CC(C)(C)C1 N1(C(CC(=C)Br)=O)CC(CNC(=O)COC2CCOC2)C2(CCC2)C1 c1(C(=O)OC)cnccc1N1CC2C(CNC(c3nccnc3C)=O)C2C1 N1(C(=O)CCOCC(F)F)CC2CC1CN2C(c1nccc(Br)c1O)=O N1(Cc2c3cccc(C)c3ccc2)CCCC2NC(=O)C(C)(C)C12 c1(CC(=O)NC2CC(C(C)NC(=O)CCc3cnn(C)c3)C2)ccc(Cl)nc1 N1(C(C(C(C)C)(C)O)=O)CC2C3CCC(C2C1)N(C(c1sccc1CC#N)=O)C3 C1(CCNC(C2C(C)C2C)=O)CN(C(c2n[nH]cc2Cl)=O)CCS1(=O)=O C(c1ccc(C(N)=O)o1)=CC(=O)NC(CNC(C(C)CN(C)C)=O)(C)CO C1(CNC(CSCCOC)=O)CC(F)CN1C(c1cc(CO)c(C)o1)=O CCC(C)(C)CC(=O)NC(C)C(C)NC(c1ncoc1-c1cnn(C)c1)=O C1(C(=O)NCc2n(CC)ncn2)CCCCN(C(c2ccc(CO)cc2F)=O)C1 N1(C(c2ccc(C(C)=O)o2)=O)CCCC(C(=O)NC(C)C(F)F)CC1 c1(C(=O)NCC2(C)CCCN2C(=O)CC2CC3CC3C2)cc2c(cn1)CCCC2 N1(C(CSCC=C)=O)CCOCC1CC(=O)NC1(CCO)CCCCC1 C1(NC(CN(CC)CC)=O)CCCN(C(=O)CCCOC(C)(C)C)C1C N1(C(C(C)=C(CC)C)=O)CC(NC(=O)Cn2nnc(-c3cccs3)n2)CC(O)C1 N1(C(CC(=C)Br)=O)CCC2(CCN(C(=O)C(C)C(F)F)CC2)C1 C#CC1CCN(C(=O)C(=O)N(c2nc(C)c(C(C)OC(C)=O)s2)C)C1 N1(C(c2c(C)nco2)=O)CC2(C1)SCCC2NC(=O)C(c1c(C)noc1C)C Cc1ccc(O)c(CN2CCCCC2c2n[nH]cc2N)n1 c1(C(=O)NC(C2CCN(C(C(C)=C3CC3)=O)C2)(C)C)ccc(C(C)=O)cn1 Cc1oc2ccccc2c1CNC(=O)C(n1cc(C2(S(=O)(=O)NC)CC2)nn1)C N1(C(C2CC=C(C)CC2)=O)CCC(C2CC2)(CNC(=O)CCS(C)=O)C1 c1(N(C2CCN(Cc3cc4ccc(Br)cc4[nH]3)C2)C)ncc2cccc(O)c2n1 C1(C(=O)NC2CC(CNC(=O)C3=CCCOC3)C2)CCn2c(O)nnc2C1 N1(C(C2(C)N(C(c3nc(C)sc3C)=O)CC=C2)=O)CCC2(CC(CO)C2)C1 c1(OC)ccc(-c2cnc(CNC(c3ccn(C(C)(C)C)n3)=O)nc2)c(C)n1 N1(C(C2C(C)(C(F)F)C2)=O)CC(CNC(c2cnoc2C2CC2)=O)C2(CCC2)C1 O=S(=O)(c1cc2sc(=NCCC3CCCO3)[nH]c2cc1Cl)NCCc1nccs1 N1(C(c2c(CC)ccs2)C(=O)NC2CCC2)CCC(C2(O)CCC2)CC1 c1(C(N2C(CNC(C(C3CCCC3)OC)=O)CC2)=O)cc(N)cnc1Br C1(NC(C(C=C=C)C)=O)CCN(C(c2ccsc2C)=O)CCC1(F)F c1(NCCOCCN(C)C(C2CCN2S(C)(=O)=O)=O)c(F)cccc1[N+](=O)[O-] C1(C(N(C2CCN(C(CC(=C)Br)=O)C2)C)=O)CC2OC(=O)OC2C1 CCCCCC(=O)NC(C)(C)C(C)NC(=O)C(C)(CC1CCC1)OC c1(N2C3CC(=C)CC2CC3)nc(=NCSC2(OCC)CC2)[nH]c2c(F)cccc12 CC1COC(C)(C)CN1C(CC1(C#N)CC1)C(=O)Nc1ccccc1 Cn1ccc(C(N2CC(NC(c3cn(C4CC4)cn3)=O)CC3(CC3)C2)=O)c(O)c1=O c1(C(C)NC(C2(CC)CN(C(=O)C(O)C(F)(F)F)C2)=O)ccc(F)c(Cl)c1 Cc1[nH][nH]c(=NC(=O)C2CN(C(c3ccc4n[nH]cc4c3)=O)C2)c1Br C1(CNC(c2cccc(SC)c2)=O)C(C)CCCN1C(=O)CCC1CCC1 N1(CCN)CCC(NC(C23CC(C(N(C)CCO)=O)(C2)C3)=O)CC1.C1CO1.OC C1(C(NOCCC(C)C)=O)CN(C(=O)CCc2cccnc2)CCC1(C)C C1(CCOC)(C(=O)NCC2CC2Cl)CCN(C(C2CCCCN2C)=O)CC1 S(=O)(=O)(c1ccc(NC2CC(CF)C2)cc1Br)NC(CC#CC)C C1(NC(C(C(C)O)(F)F)=O)CC2(CCCCN2C(c2cnncc2O)=O)C1 c1(OC)ncccc1CC(=O)Nc1cccc(CNC(=O)CC2CS(=O)(=O)C2)c1 c1(NCCCN(C(C2OCCC2c2cnn(C)c2)=O)CC)ccccc1Cl c1(CNC(c2ncc(C(C)C)s2)c2nnnn2CC(F)F)ccc(S(C)=O)cc1 Cc1nccc(C(=O)NCC23CC(NC(c4cc(CO)oc4C)=O)(C2)C3)c1C N1(C(C2N(C(C)=O)CSC2)=O)CCCCC1CNC(=O)CC1C=CCC1 C1(COC)CN(C(c2cccc(SC)c2)=O)CCN1C(=O)C(C)C(F)F c1(O)cccc(OC(=O)C(CC)SCCCCCC)c1 c1(C(=O)NC(c2c(C)noc2C)C)ccc(S(=O)(=O)Nc2ccc(Cl)cc2)cc1 C(=O)(CCOCCN(C(=O)COC)C)C(CS)N.C(C(C)N)OCC N1(C(C(n2c(C)ncc2)C)=O)CCN(C(=O)CC2(C)CC2(Cl)Cl)CC2(CC2)C1 C(=O)(C1=CCCNCCC1)NC(c1ccc(Cl)cc1)C(N)=O C(C)(C)(CCCCC(=O)N1CC2CC(NC(C34CC3COC4(C)C)=O)C1C2)OC c1(C(=O)NC2CC(C)N(c3cc(C4CC4)ncn3)CC2)occ2c1CCOC2 N1(C(C2CCCC(=O)N2)=O)CC2(CCC2NC(=O)C(=C2CCCCC2)F)C1 N1(C(CC(CC)(F)F)=O)CCOCC12COCCN(C(=O)CCC(C)O)C2 C1(NC(C(=Cc2ccco2)C)=O)CCN(C(C2CN(C)CCO2)=O)CCC1(F)F c1(C(=O)NCC2(O)CC(CNC(c3ccc(C)s3)=O)C2)ccc2c(c1)C(=O)NC2 CN1C(=O)CCC1(C)CNC(C1CN(C(c2ncncc2N)=O)CC12CC2)=O N1(C(C(C)NS(CC)(=O)=O)=O)CCC2(CC1)CC2CNC(=O)CSC(F)F O=C(C1=CC2(CCN(C(=O)CC3OCCO3)C2)C1)N1CCC(F)(F)CC1 N1(C(C(C)N(C(=O)C(N2CCOC2=O)C)C)=O)CCC(C(=O)NO)C1C(C)(C)C Cc1ncc(Cl)cc1CC(N1CCC(NC(=O)CC2CNC(=O)C2)C(O)C1)=O c1(NC(C(CN(C)C)NC(c2n(CC)c(O)nc2)=O)=O)c(C)cc(C)cc1C c1(CC(N2CC(CCNC(=O)C=Cc3cn[nH]c3)OCC2)=O)cc(F)ccc1O c1(C(=O)NCC(CNC(CCCOC(C)C)=O)O)cnc2c(Br)c[nH]c2c1 Cc1cc(C(=O)NCCC2(NC(=O)CCC3CCC(=O)N3)CCC2)c(C)cc1Cl c1(C(=O)NC2C(CNC(C(C)n3ccnc3)=O)COC2)ccc(P(C)(C)=O)o1 C1(CC(N2CC(NC(C(C)COc3ccccc3)=O)C2)=O)CCCS1(=O)=O CC1(C(=O)NCC2(CCNC(c3cncnc3)=O)CC2)CCC(=O)NC1 C1(C(=O)NC2CCCC2NC(=O)CCS(C)=O)(NC(C)=O)CCCCC1 C(=O)(C1=CCCOCC1)N1CCC(CC)C1CNC(c1c[nH]c2nccc-2c1)=O N12CCCN(CC1)C(=O)c1cc2ncn1.C1(OC)CC(c2ccccc2)CO1 CC1CC(N=c2ccnc(NCC3(F)CC3)[nH]2)c2ncnn21 c1(NC(C2CC3CCC2N3C(=O)C(O)O)=O)ccc(S(=O)(=O)c2ccccc2)cc1 Cc1ccc2c(c1CO)CCCN2CC(c1cccc(C#N)c1)O c1(N2CCC(NC(C3C(C(=O)OC)C3)=O)C23CCC3)nc2ccc(N)cc2s1 c1(C(=O)NCCCNC(c2cc(-c3cccnc3)on2)=O)sccc1Br C1(C(=O)NC(CN(CC)CC)C)CC2CC1CC2NC(c1ncnc(C)c1C)=O c1(CC)nccnc1C(=O)NCCC1(NC(=O)CC2C=CCC2)CCCC1 c1(C(=O)NCCN(C(=O)CS(C)(=O)=O)CCC)ccc(Cc2nc[nH]n2)cc1 N1(C(CC(C)N2CCCC2=O)=O)CCN(C(=O)CSCC(F)(F)F)CC12CC2 c1(C(=O)NCC(C2CCC2)NC(C2CCS(=O)(=O)C2)=O)ccc2nn[nH]c2c1 c1(SCc2nc(-c3nccc(SC)c3)nn2Cc2cccs2)cnc(Cl)c(F)c1 N1(C(c2c(NC)cc(Cl)cc2)=O)CCC2(CC1)CC(C)N(C(=O)C(C)CO)C2 C1(N(C)CC)CCC(n2cc(-c3sccc3C)nn2)CC1 c1(OC2CN(C(c3cnc(C(C)C)o3)=O)C2)ccc(F)nc1.C(=O)(CO)NCCC N1(C(C=CCC)=O)CC2CC(NC(c3cc(Br)n(C)c3)=O)C(C2)C1 O=S(=O)(c1ccccc1-c1cnn(C2CC2)c1)NC(=O)C(O)C(O)c1ccccc1 CC1CCCCCC1NC(C1(O)CC(CNC(=O)OC(C)(C)C)C1)=O C1(COC)CN(C(c2cc(O)nc(C)n2)=O)CCN1C(C1CCCC1C1CC1)=O c1(C(=O)OCC)n[nH]c(=NCC2CCCC(NC(C3CCC(=O)N3C)=O)C2)s1 C1(CNC(c2cc(C(F)(F)F)ccn2)c2n(CC)nnn2)CC=CCC1C C1(CC(=O)NCC(C)CNC(=O)C=Cc2ccc[nH]2)COC2CC1C2 c1(C(N(CC(CNC(CC(CC)SC)=O)(C)C)C)=O)cc(C)ccc1N N1(C(C2C(C3C(C)C3)C2)=O)CC2CN(C(=O)C(C)CC(F)(F)F)CC2C1 N1(C(c2c(C)cncc2F)=O)CCC(C)C(C)(C)C1 N1(C(CNS(CC)(=O)=O)=O)CCN(C(c2cscc2C)=O)C(C)CC1C C(=O)(C1=NOC2(CCC2)C1)N(CCCCNC(=O)Cc1cc(F)ccc1F)C C1(c2n(CCCF)nnn2)(NCc2ccc3c(Br)c[nH]c3c2)CCN2CCC1C2 Cc1cc(=O)ccn1CC(=O)NCCC1CN(C(=O)CC2(O)CCC2)CCO1 O=C(C#CC1CCCCO1)NCC1CCCCN1C(c1cnc(O)o1)=O c1(C(=O)NC(C2CN(C(=O)Cc3cc(Cl)ccc3Cl)C2)C)csc2nnsc12 C1(CC(=O)NCC2C(NC(C3(CC)CC(C)(C)C3)=O)CCC2)CCCCC1(F)F C1(C(c2n(CC(F)F)nnn2)Nc2ccc(F)c(Br)c2)CC12CCC(F)(F)CC2 CCCC(C(=O)NCC1CC1(C)C)NC(=O)C(C)OC(C)=O C(C1=CCN(C(=O)C(C2CCCN(C)C2)(C)C)CC1)NC(Cc1c(C)noc1Cl)=O c1(C(=O)NC2(C)CC(NC(C3COCCC3(F)F)=O)C2)ccc(=N)[nH]c1Cl N#Cc1ccc(C(=O)NCC#CCNC(c2cc3c(s2)CCC3)=O)c(F)c1 C(=O)(CCS(C)(=O)=O)N1C(C2(C(=O)NC(CCC)(C)CC)CC2)CCC1 C1(N(C(=O)Nc2cccnc2-c2cnn(C)c2)Cc2ccccn2)CCCC(F)C1 C1(CCNC(C23CC(C)C2C3)=O)CCN(C(=O)C(C)(C)CN(C)C)CC1 N1(C(C(CO)NC(C2C(C)N(C)CC2)=O)=O)CC(CO)C(C2CC2)C1 N1(C(C2C(CCC)C2)=O)CC2(C)CC1(C(=O)N(C(CC)CC)C1CC1)C2 Cc1oc(CO)cc1C(=O)NC1(CC(=O)NC2CCN(CCCO)C2)CC1 N1(C(C=C(C)Cl)=O)CCCCC(NC(c2cc(Cl)c(Cl)cc2O)=O)CC1 C1(CNC(N2C(C)CC(C(=O)OC)C2)=O)CCCCCC1C1CC1 c1(Cn2cc(C(CCC)NC(=O)CCc3cc[nH]n3)nn2)cc(Cl)ccc1C c1(CN2C(C(N3CCn4ncnc4C3)=O)CNCC2)ccc2ccccc2c1Br N1(C(C(CCSC)O)=O)C2CCC1C(CNC(c1oc(CC(C)C)nc1C)=O)C2 c1(OC)cncc(C(=O)NC2COCC2NC(=O)CSc2c(C)n[nH]c2C)c1C C1(CC(N2CCC(O)C(O)C2)=O)C2CCCC2N1C(C1CCC(=O)N1)=O C1(NC(C2CN(C(=O)NCC)C2)=O)CC2CC(NC(C3(C)CC(F)C3)=O)CC12 c1(C(=O)NCC2C3CN(C(C4CC(C)OC4)=O)CC32)c(Cl)nc2ccccn12 CCC(C(=O)NC1CCCC(NC(=O)Cc2ccc(F)c(F)c2)C1)C(C)(C)CC C1(C2CCCN(C(c3ccno3)=O)C2)(NC(c2cc(C)nnc2O)=O)CC1 Cc1cc(NC(c2nn(C)c(C)c2Cl)=O)ccc1NC(c1[nH]nnc1C)=O C1(CNC(c2c(SC)snn2)=O)CC12CCN(C(=O)C=CCCC(C)C)CC2 N1(C(c2ccc(OC)c(Cl)n2)=O)CCC2(C1)CN(C(c1ocnc1C)=O)C2 n1(CC(=O)NC(CNC(CC(COC)(C)O)=O)C2CC2)ccc2ccc(F)cc12 C1(NC(C(C)NC(=O)C(N2CCOCC2)C)=O)C2CCCC1COC2 C(CC(C)CC(C)(C)C)NC(Cn1cc(CNC(c2ccc(C)c(C)c2)=O)nn1)=O c1(CC)nc(C)c(CC(N2CCCN(C(c3cncs3)=O)CC2CO)=O)c(C)n1 c1(C(=O)NC2CN(C(c3n(C)ncc3)=O)CC2F)nccn2ccnc12 N1(C(C2CC(CCC)C2)=O)CCCC2(C1)CN(C(=O)Cc1ccsc1)CCO2 C=C(C)C(C)(C)C(=O)NC1C2CC(NC(C3CCC(F)C3)=O)CC12 CCC(C(=O)NC12CC(NC(c3ccnn3C(C)CC)=O)(C1)C2)C(C)(F)F c1(C(N(C)CC2CN(C(c3ccc(-c4cnco4)cc3)=O)C2)=O)cc(Br)cnc1O N1(C(C(SC)SC)=O)Cc2occ(C(N3CCC(C(C)(C)C)C3)=O)c2C1 c1(C(=O)NC(CN(C(CNC(=O)NC)=O)CC)C)cncc2ccccc12 CC(C)CC(C)C(=O)N(CC(C)(C)C(=O)N(C(C)C(C)C)C1CC1)C N1(C(C)=O)CCN(C(c2cncc(C)n2)=O)C(C(N2CCOCC2)=O)C1 c1(CNC(C2(CNC(=O)CCn3ccc(C)n3)CC(=C)C2)=O)c(C)cnn1C c1(OC)cc(C(=O)NCC2CC2NC(C23CC2COC3(C)C)=O)cc(C)n1 c1(N(CC(C)NC(C2CS(=O)(=O)CC(=O)N2)=O)C)ncc([N+](=O)[O-])cc1Cl C1(NCCn2c(NC(=O)NC3CCCC3)nnn2)CCCN(CCO)C1 c1(C(=O)NC2(C(=O)NCC3(O)CCC(C)C3)CCOCC2)cc(N)cc(F)c1 Cc1cc(F)cc(C(=O)NCC2CCCC2NC(=O)CC2CC3(CCC3)C2)c1O C1(F)(C(=O)NCC=CC(=O)NC(C2CCCO2)CO)CCCCC1 CC(F)(F)CCCNC(=O)NCC1CC1(C)Br C(CCC(C)C(=O)NCC=CC(N1CC(=O)NCC1C)=O)OC c1(CNC(CCCC)=O)ccc(CNC(=O)CC2CCC(=O)N2)c(F)c1 CCC(CC)C(C(=O)NC1CC(O)(CNC(=O)CC2C(C)(C)C2(C)C)C1)OC CC1=C(C(=O)NC2CCN(C(=O)C=CC3CCCO3)C2(C)C)CCC1 c1(C(C)C(=O)NCCC2CCN(C(C3CN(C)C3)=O)CC2)noc2ccccc12 Cc1cn(CC(=O)NC2CC2CNC(c2nnsc2C(F)F)=O)c2ccccc12 C1(NC(c2ccc(CC)o2)=O)(CO)CCCN(C(=O)Cn2ccc(C(=O)OC)n2)C1 c1(CC)oc(C)cc1C(=O)N(C(CNC(c1cnc(O)n1C)=O)C1CC1)C CC1SCCN(C(c2cc(-c3ccccc3)n(C)n2)C(=O)NCCCSC)C1C C1(NC(C(CC)C)=O)CC1C1CCN(C(c2cc(NC(C)=O)ccc2F)=O)CC1 C(=O)(C(C)(C)CSC)NCC(C(C)C)NC(C1CC(SC)C1)=O Cc1nccc(C(N2CCN(C(=O)C3=COCCO3)C3CC23)=O)c1O O=C(CCCCO)NC1CCCC1CNC(c1ccnc(C2CCCC2)n1)=O C1(C)(C(=O)Nc2cc(C(C)C)on2)CCN(C(=O)NC2CCOCC2)C1 C(=O)(C(C)CC(C)CC)NCC(CC)NC(c1cccc(NS(C)(=O)=O)c1)=O C(CC(C)C)(C(=O)NCc1ncccc1C(=O)N(C)CC1(O)CCC1)OC C=CCC(CNC(=O)CC1COCCO1)C(=O)N(C)CCC c1(C(c2nn[nH]n2)NC(c2cccc(OC(CC)C)c2)=O)ccc2cc[nH]c2c1 C(C(=O)Nc1cccc([N+](=O)[O-])c1)(C(C)C(C)(C)C)N1CC(C#C)OCC1 N1(C(Cc2c(C)n[nH]c2C)=O)CC(N=[N+]=[N-])CC1C(=O)NC(C1CCCC1)CO c1(C(=O)OC)ccc(COC(C2(c3ccc(C)cc3Br)CC2(F)F)=O)cc1O c1(C(C)NCC(=O)N(C2CC2)Cc2ccc(OC)cc2)ccc(OC)c(Cl)c1Cl C1(CNC(=O)C=Cc2nccs2)CN(C(c2ccn(CCF)n2)=O)CCCO1 c1(C(N2CCN(C(C(CC(C)C)F)=O)CC2)=O)ccc2c(c1)N(C)CCO2 CC(C)CC(C(=O)NC1CCCCC1NC(c1ncccc1N)=O)n1ccnc1 N1(C(C(CCC)=CCC)=O)CCN(C(=O)CC(O)CC(C)C)CC(O)C1 c1(CNC(c2nc(C(=O)NC(CC)C)sc2)=O)ccc2ccc(O)nc2c1 Cc1cccc(Cl)c1C(=O)NCCOCCN(C)C(c1nscc1N)=O Cc1[nH]nc(C(=O)NCc2cn(C3CN(C(C4CCCC(=O)O4)=O)C3)nn2)c1C N1(C(C2(COC)CCCO2)=O)CCCC(N(C(=O)C=CC=C(Cl)Cl)C)C1 c1(C(=O)NCC2CN(C(c3cc(SC)c(C)o3)=O)C(C)C2)cnn2c1N(C)CC2 C(CN=c1[nH]nc(CO)s1)C1C(C)CCCN1C(c1ccnc(N(C)C)c1)=O C1(C(=O)OC)CN(C(=O)CNC(=O)CC(C)C)CC1C N1(C(c2n(CC=C)ccc2)=O)CCCN(C(c2cc(OC)nc(F)c2)=O)CC1C C1(CNC(C=C(C)C2CC2)=O)CCN(C(=O)CC2CCOC2)CCC1(F)F C1(CC(=O)NCC(CNC(c2ccn(C3CC3)n2)=O)OC)CCC(C)(C)C1 CC1c2c[nH]nc2CCC1C(N1CC(CNC(c2ccc(C#N)nc2O)=O)C1)=O Cc1cccc2nc(C(=O)N(C)CCN(C(=O)CCn3ccccc3=O)C)cn12 Cc1noc(C(=O)NCCCCCNC(=O)C(F)(F)c2csc(C)c2)n1 C(=O)(C#CC1(CC)COC1)NC(C1(C(=O)NC(CCC)C2CCC2)CC1)C C=CCC(CNC(C1CC(C)N(C)C1)=O)C(=O)N1CCC(C)(CO)C1 C1(OC)CC(C(=O)NC(C)(CNC(=O)Cc2c(C)cnn2C)C(C)C)CC1OC C1(C(N2ON=C(C(=O)NCCSCCCC)C2)=O)CCC(N=[N+]=[N-])C1 C1(NC(c2ccn(COC)n2)=O)CN(C(c2ccc[nH]2)=O)CC1n1ccnn1 C(C(C)(O)CSC)NC(=O)OC(C)(C)C.CCC1CN1 CC1CCN(C(CCS(C)(=N)=O)=O)C1c1cn(C)nn1.c1(C(=O)N)nc(C(=O)O)cs1 c1(CC(=O)NCC(=O)NCC(COC)C)ccn(C)c1 C1(F)(CNC(C2CCCO2)=O)CCN(C(c2cccc(-c3ccoc3)c2)=O)C1 C1(CN(C(=O)CCS(C)=O)C)CCCCN1C(c1ccc(CO)cc1)=O C1(C(N(CCOCC)CC)=O)CCN(C(=O)CC2CCCC(=O)N2)CCO1 CC1=NNC(=O)C1CN1CCOC(CN)(CO)C1.c12ccc(cc1)C(=O)N(C)C2 Cc1cc(Cl)c(C(N2CCS(=O)(=O)C(CCNC(=O)CC=CCCO)C2)=O)cc1C CN1CCC(C)(C(=O)NCCCOCCCNC(c2cnn(C)c(=O)c2)=O)CC1 C(=O)(CC(C)CC(=O)NCC1CC1CNC(c1cc(C(F)(F)F)no1)=O)OC c1(C(N2CC3(CN(C(CC(C)OC)=O)C3)C2)=O)cc(Br)cc2c1CCN2 CC(C)CCCCCC(=O)N1CC2CCC(C1)N2C(=O)Cn1ncc(C#N)c1N N1(C(C=CCOCC)=O)CCCC1(C)CNC(=O)COCC(c1ccccc1)C c1(-c2nnc(CC(C)NCCS(=O)(=O)N(CC)CC)o2)ccccc1Br C1(NC(c2ccc(CC)nc2)=O)CCC2(C1)CN(C(C1(C)CCCC1)=O)C2 c1(COC)cccc(C(c2nnnn2CC(F)F)NC2CC(C(F)(F)F)C2)c1F c1(CNC(CCNCC2N(S(C)(=O)=O)CCC2)=O)ccnc(F)c1F C=CCC(F)(F)C(=O)N1CC(C(C)(C)O)(CNC(C2(CC)CCC2)=O)C1 C(=O)(C(C)(F)C(C)(C)F)N1CCN(CC(=O)N(C(CC(C)C)C)C)CC1 N1(C(c2scc(C)c2)=O)CC2CCOC2(CNC(=O)C(O)c2cnc[nH]2)C1 S(=O)(=O)(c1ccc(NCC2CCC2N(C)C)c(Cl)c1)NCc1c(C)scc1 CCC(CC(=O)NCC=CCNC(c1ccsc1C(=O)OC)=O)C(C)C CC1CN(C(C2(C)CC2(Cl)Cl)=O)CCCN1C(=O)Cc1cnn(C(C)(C)C)c1 C1CCCOC12CC2.C(C)(C)(CN1CCCC1)NC(=O)NC1C(OC)C1 C1(N(C(c2c(C)cno2)=O)C)CC2CCC(C1)N2C(=O)CCS(C)=O Cc1[nH]c2ccc(C(N3CC(NC(c4ccc[nH]4)=O)C4CC4C3)=O)cc2c1C C1(CC(=O)N(C2CCN(C)C2)CC)CCCC12CN(C(=O)CC(O)C1=CCCC1)C2 C1(c2ccc(OC)cn2)NC(=S)N(CC(C)C)C2=C1C(=O)NC(C)(C)C2 C(=O)(C1=Cc2ccccc2C1)N(CC(N1CC2(C=CCO2)C1)=O)CC1CC1 c1(OC)ccc(OCc2cn(C(C)(C)CC(=O)N(CC(=O)O)C)nn2)cc1 C(=O)(CCCCSC)N1CC(C(=O)NCC2(C(N)=O)CCCC2)(CC)C1 N1(C(C2(C(C)C)CCN(C(C=C(C)C(C)C)=O)C2)=O)CC2CC(O)CC1C2 c1(C(N2CCN(C(c3cc(C4CC4)on3)=O)CC2)=O)c[nH]c(=O)c2ccnn12 c1(C(=O)NCC2(CNC(C(COC)C)=O)CC2)cn(C)c(=O)cn1 Nc1ccc(F)c(C(N2CCN(C(=O)CN3CCS(=O)(=O)CC3)C3CC23)=O)c1 C(=O)(CCCN(C(=O)C(n1ccnc1C)C)C)NCC(=CCCC)C C1(C)(CNC(CCCCC=C)=O)CN(C(C2CSCCS2)=O)C(C)(C)C1 c1(OC)cc(NS(C)(=O)=O)ccc1C(=O)NC(CSC)CO Cc1cc(C(=O)NCCCN(C(=O)CCc2csc(Br)c2)C)nc(O)c1 c1(OC)cc(OC)nc(C(=O)NCC2(C)CCN(C(C3NC(=O)CC3C)=O)C2)n1 Cc1ccc(Cl)c(OC(C)C(N2CCC(CNC(c3cc(C#N)cs3)=O)C2)=O)c1 c1(C(=O)NCCC2(O)CCCN(C(=O)CC(F)(F)F)C2)cnnc2ccccc12 c1(C(=O)NCC2N(C(c3c(C)nc(Br)o3)=O)CC2)ccc2c(c1)C=CCC2 c1(C(=O)NCC2CCN(C(c3scnc3Cl)=O)C2)cc(Cl)cc(Cl)c1O c1(OC)ncc(Cl)c(C(=O)NCC2C3CN(C(C4CC5(C4)CC5F)=O)CC23)c1Cl N1(C(=O)C(F)F)CCOC2(CCCN(c3ncc4c(Br)cccc4n3)C2)C1 c1(C(=O)NC(C(=O)NC2CCC(=O)NC2=O)CO)ccn2ccnc2c1 C1(CNC(C=CCCC(C)C)=O)CN(C(C2(F)CCC2)=O)CCC1C(F)(F)F CC1(C)CC(Nc2cc(F)ncn2)CN(C(C2CC(=O)N(CC(F)(F)F)C2)=O)C1 C(=O)(C(CC)CCc1ccccc1)NCCC1(NC(CS(=O)(=O)NC)=O)CCC1 N1(C(C(C)Sc2ccc(F)cc2)=O)CC(NC(c2c[nH]c(=N)s2)=O)C(C)C1 N1(C(C(C)SCC)=O)CC(C(N2CCCC(F)(F)C2)=O)C2(CC2)C1 C(CC(=O)N1C(C(=O)OC)CC1C)(CC(C)C)NC(C1(OC)CCOCC1)=O C(c1cccc2ccccc12)=CC(=O)NC(CCCC)CNC(C1(CO)COC1)=O N1(Cc2cn(C3C(NC(C4(C5CC5)CC4)=O)CCC3)nn2)CCNC(=O)C1 c1(CCC(=O)NC2CC(NC(=O)CCOCC(F)(F)F)C2)ccc(Cl)cc1Cl O=C1CCC(C(=O)NCC(C(F)(F)F)N2CCN(C(=O)C#CC3CC3)CC2)CN1 N1(C(CCCC(=O)OC)=O)CCC2(CCN(C(C3CC3F)=O)CC2)C1 c1(C(N2C(C(N3CCC(C(=O)OCC)C3)=O)COCC2)=O)cc(Cl)cnc1F O=C1NC2(C(=O)NC3CC(NC(C4(n5ccnn5)CC4)=O)C3)CC3CC1C2C3 C(=O)(C1(C)CCOc2ccccc21)NC(C)CNC(=O)CC1CC2C=CC1CC2 c1(CC)nn(C)c(CC)c1C(=O)NCC(C)(C)CN(C(=O)CCCC#N)C C(=O)(CCCCNC(C1(F)CCCCC1)=O)NCCC1C(C(=O)OC)C1 CCC(CC(=O)N1CCC(NC(=O)CN(C(=O)C(C)C)C)C(C)(C)C1)C(F)F C12(C(N(CC(C)(C)CO)C)=O)CC(C)(CN1C(C1CCC(=O)C1)=O)C2 c1(C(C(=O)NC(C2CCC(C)CC2)C#N)N(CCCSC)C)ccnc(Cl)c1Cl Cc1ccc2c(-c3nc(C(=O)Nc4ccc(I)nc4)cs3)c[nH]c2c1 C(=O)(C(COC)CC(C)C)N(C(C(=O)N(C(=O)CCC)C)C(C)O)C.CN N1(C(C2CC(O)(CC#C)C2)=O)CCC(NC(=O)CC2CCC(=O)O2)C(C)(C)C1 C1(C(=O)NC2CN(C(C(C(CC)O)C)=O)CC2O)(CF)CCC(F)(F)CC1 C(CC(C(=O)NCC1CCN(C(=O)C(C)N(C)C)C1)NC(C)=O)SC N1(C(C(CSC)C)=O)CC(N(C)C(c2cncc(C#N)c2)=O)C2(CC2)C1 c1(C(N(C(CN(C(C(CC(C)C)O)=O)C)C)C)=O)cc2ccsc2n1C Cc1cc(C(N2CCC(CNC(c3csc(Br)c3Cl)=O)C2)=O)[nH]c1C N1(C(=O)C=CC=C(Cl)Cl)CC2OCCN(C(=O)CC3CC4C=CC3CC4)C2C1 CC(CCO)CCN=c1nc(N(C)Cc2ccncc2Cl)c2cc(Cl)ccc2[nH]1 C(=O)(C(O)C(C)(C)SCC)NCCN(C(C(C)(C)NC(=O)OCCC)=O)CC CC1CCCN(C(N2CCCC(COc3cc(N)n(-c4ccccc4)n3)C2)=O)C1 Cc1cc(F)c(C(=O)NC2CCN(C(c3cccc(F)c3Br)=O)CC2O)cc1F c1(C(=O)NCCN(C(C2CC2Cl)=O)CC2CC2)cc(-c2ccccc2)ccc1Cl C1(C(C)C)CCC(C(=O)NC2CCCC2NC(C2(c3ccno3)CCC2)=O)CC1 N1(C(C(CC)(C)CC)=O)CCC2(C1)CN(C(c1sc(C)c(C)c1C)=O)CC(C)O2 C(=O)(C(CCCCO)NC(C1CC(F)CN1C)=O)NCC1CC(CN(C)C)C1 c1(C(N(CCNC(c2nc(CC)oc2)=O)CCOC)=O)ccc(OCC)nc1Cl c1(C(=O)NCC(CNC(=O)Cc2c(O)ncnc2O)CO)c(F)ccc(O)c1F c1(C(C(=O)NC(C)C)N(C)Cc2cc(-c3ccco3)on2)cnn(CCO)c1 C(CC(=O)N1CCN(C)C2(CC2)C1)(C(C)(C)C)NC(C(C)=C1CC1)=O N1(C(c2nc(C)c(Br)cc2)=O)C2CCCC1CC(n1cc(C#CC(=O)O)nn1)C2 c1(C(C)=O)ccccc1C(=O)NCCC(O)CNC(=O)C=CC1CCCC1 N1(C(CC2ON=C(C)C2)=O)C(C(=O)NC(C)Cn2cc(C)cn2)CCC1C1CC1 C#CCCCCS(C)(=O)=NC(=O)C(c1ccc([N+](=O)[O-])cc1F)N1CCOCC1 c1(C(=O)NC2CC2C(=O)Nc2ncccc2C(F)(F)F)cnc(O)nc1O C1(NC(c2scc(C)c2)=O)C2CCN(C(=O)CCn3cnnn3)CCC12 c1(C(=O)NC(CC)(CC)CCNC(C2CC2Cl)=O)ccc2ccccc2c1 C1(NC(=O)NCC(c2c(OC)ccc(Cl)c2)O)CCC12CCCCC2 c1(C(=O)NCCNC(C23CCCCC2C3Br)=O)sc([N+](=O)[O-])cc1Cl C(N=c1[nH]c2cccc(OC3CC3)c2s1)c1ccc(NC(C(OC)OC)=O)cc1 c1(C(N2CC(NC(c3cc(C)sc3C)=O)C2)=O)ccnc2ccc(F)nc12 C12(C(=O)OC)C3C4C1C1C2C3C41NC(=O)NC(C1CCCCN1)=O C(=O)(C(Cc1cn(-c2ccncc2)nn1)NC(C1CCN1S(C)(=O)=O)=O)OC C1(C(N2CCCC(CCC)(NC(c3csnn3)=O)C2)=O)Cc2cc(F)ccc2O1 c1(C(N(CC(CC)NC(=O)CC2CCC(=O)O2)C)=O)cc([N+](=O)[O-])ccc1C NS(=O)(=O)c1ccc([N+](=O)[O-])c(NCCc2ncc[nH]2)c1 N#Cc1cnc(NCC2CCCCC2NC(=O)CCCCc2cnn[nH]2)c(F)c1 C1(NC(C(CSC)O)=O)(CO)CCCN(C(c2cccc(C)n2)=O)C1 CCCCC(C)C(C(=O)NC1CC1)N1CCc2cc(C(C)(C)C)ccc21 N1(C(c2nc(-c3cccc(OC)c3)oc2C)=O)CCN(C2CC2)C2(CCOC2)C1 C1(CCNC(CN(CC)CC)=O)CCCN(C(c2c(C)oc(C)c2C)=O)CC1 c1(OCC)ccc(CNC2CC(NC(=O)CCc3ccc(C)c(F)c3)C2)cc1Br N1(Cc2nc(N(c3ncc(C#N)cc3Br)C(C)=O)sc2)CCc2sc(Br)cc2C1 Cc1ccc(C(C)C(=O)NCCOC2CN(C(=O)CC(C)C3CCCCC3)C2)s1 C12(CNC(=O)C(Cc3ccccc3)n3cnnn3)CCC(C1)N(C(=O)C1CC1)C2 N1(C(C2(OCC)CCC2)=O)CCC2(CC1)CCN(C(=O)C(C#N)CC)C2 C1(NC(c2cccs2)=O)CC2CC1N(C(c1cc(Br)c[nH]1)=O)C2 N1(C(CC=CCC)=O)CCC(OCC(=O)OCC)C1 Cc1cc(C)c(C(N2CCC(N(C)C(C3CC(C(F)F)C3)=O)C2)=O)cc1C CCC(CC)C(F)C(=O)NC1CN(C(c2c(F)cccc2F)=O)CC1F N1(CC(=O)NCC(n2cc(-c3cnc(CC)o3)nn2)C)CCOCC1=O C1(C(=O)NC(C(C)C)(C)CO)CN(C(c2cncc(F)c2)=O)CC1(F)F C1(C(=O)Nc2nc(C)c(C)s2)C2CCC(C2)C1NC(c1cnnc(Cl)c1)=O CCCC(C(=O)N(C(C)CN(C(=O)CCc1cc(Cl)no1)C)C)c1ccccc1 c1(SCC(=O)NCC(C)(CC)NC(CCC=C=C)=O)cc(=O)n2ccsc2n1 C1(C(N(CCSC)C)=O)CC(F)CN1C(=O)CC1CCCC1O C(C)(C(=O)NCC1(O)CN(C(=O)CSC(F)(F)F)C1)(C1CCOCC1)OC C(=O)(C(O)CC(F)(F)F)OC1CN(c2ccc(C(=O)OC(C)(C)C)cn2)C1 N1(C(c2nc(C(=O)OC)sc2)=O)CCN(C)CC1CNC(=O)C(C)(CC)OC c1(C(C(=O)CNC2(CNC(C3CCC4CC34)=O)CC2)(F)F)ccc(Cl)cc1 Cc1cccc(O)c1C(N1CC2CN(Cc3cccnc3)C2C1)=O CCCCCC(c1nnnn1CCCF)NCC(O)CC(C)C c1(C(=O)NC(C)(C)CCNC(C2CC23CC3(F)F)=O)nccc2cccnc12 C(=O)(CC(C)C(=O)NC(C)(C(=O)NC1CC(C)OC1=O)C1CCC1)OC N1(C(C(C)(C)NC(=O)OC)=O)C2CCC1C(F)C(NC(=O)CC(F)(F)C(F)F)C2 c1(CN(C(c2cc(C(C)C)on2)C(=O)NC2COC2)CCC)ccccc1F N1(C2C(NC(CC)Cn3ccnc3)CCC2)CCN(C)CC1 CS(=O)(=O)c1ccnc(NC2CN(Cc3ccc(C#N)cc3)CC23CC3)n1 Cn1cc(C(N2CCC(NC(=O)C=CSc3nc[nH]n3)C2)=O)cn1 c1(OC)cc(C#N)ccc1C(=O)NCC1CCCCN(C(c2scnc2Cl)=O)C1 C1(CCNC(C(CNC(C(CSC)O)=O)N(C)C)=O)OCCC1(C)C C1(C)(CNC(C(CCC)N(C)C)=O)CCCN(C(=O)Cc2cc(C)cs2)C1 CC(C)CCCC(=O)N1CCCCC1C1(NC(=O)COCCF)CC1 C1(C(N2CCC(CS(C)(=O)=O)C2)C(=O)NCC)CCC(C(C)C)CC1 C1(CC(=O)NC2C(NC(C(=O)NCCNC(C)=O)=O)CC2)OCCOC1(C)C c1(C(N2CC(C)(C(=O)NC(CCC)c3ccco3)C2)=O)[nH]cc(C)c1C Cc1cc(C=CC(=O)NC2CC3OC2C2CC32)ccc1Br c1(C(=O)NCC2CCN(Cc3n(C)ncc3Br)CC2)cc2ccccc2cn1 NS(=O)(=O)CCCC(=O)N1CC(O)C(O)C1CNC(C1CC2CC2C1)=O c1(CN(C)C(C2CC2c2cc(Br)cc(Br)c2)=O)noc2c1CCCCC2 C1(NC(C2(COC)CC2)=O)(CNC(=O)C(c2nc(C)cs2)C)CCOCC1 c1(C(=O)NC2CC(NC(C3(C)COCCO3)=O)C2)ccc(S(N)(=O)=O)nc1 N1(C(C23CCC(OC)C2C3)=O)CCC2(CC1)CC2CNC(=O)C1=COCCC1 C1(C(=O)NCCC(C)NC(c2ccc(CC)o2)=O)COC(C)(C)O1 c1(CNC(=O)Nc2cccc(CN3CCOCC3)c2)cnc(S)nc1.C(=O)(C1CC1)N C1(CNC(C(C)SCC)=O)(OC)CCCN(C(=O)CCSCC(C)C)C1 C1(C(=O)NCC2(C#N)CCC2)(COC)CN(C(c2ccc(C)o2)=O)C1 CCC(C)(C)CCCC(=O)NC(C)(C)CNC(c1cc([N+](=O)[O-])ccc1OC)=O c1(OCC)nc(C)ccc1C(=O)NC1CCC1NC(=O)C=Cc1cscn1 Cc1ccc2scc(C(N3CCC(C)C(NC(=O)Cc4cscn4)C3C)=O)c2c1 c1(CCC(N2CCC(CN(C(=O)CSCCC#N)C)C2)=O)ccc(Cl)c(Cl)c1 Cc1cc(F)cc(C)c1C(=O)NCC(C)(O)CNC(C1CC(C(F)F)C1)=O C1(CNC(C(c2cc(C)sc2)(F)F)=O)CC2CCC(C1)N2C(=O)C(F)(F)C1CC1 C#CC1CN(C(=O)CC2C(=O)N(C)N=C2C)CCN1C(=O)COc1cc(C)on1 CC1CCCC=C1C(=O)NCCCCCNC(=O)Cn1ccc([N+](=O)[O-])n1 Cc1ccc(C#N)cc1S(=O)(=O)N1CCC2C(CCN2C(c2cc(C)[nH]n2)=O)C1 C12(C(=O)NC3CCC(NC(C(CC)CC(F)F)=O)C3)CC3CC(C1)CC(O)(C3)C2 c1(COC)nnc2ccc(=NCC3CCC(C(F)(F)F)O3)[nH]n12 C1(CNC(C2OCCN(C(C(C#C)(C)C)=O)C2)=O)CCC2(CCC2)O1 C#CC1(O)CC(C(N2CC(NC(c3nccn3CC)=O)C(CCC)C2)=O)C1 CCCCC(C)(F)C(=O)NCCOC1CCN(C(c2cncc(F)c2Cl)=O)C1 C1(C(N2C(C3(NC(C(C4CCC(=O)N4)C)=O)CC3)CCCC2)=O)CN2CCN1CC2 S(=O)(=O)(c1ccc2[nH]c(=NCC(CO)OC)sc2c1)N(CCCC(=O)NC)C N1(C(c2ccc(OC)o2)=O)CCOC(C(=O)NOC2CC2C)CC1 C1(C(N2C(CCC)CN(C(C3CCN(C)C3)=O)CC2)=O)CCc2ccnn2C1 c1(C(=O)NC2C(NC(CC3(OC)CCC3)=O)COC2)ccc(C2CC2)c(F)c1 CCC(CCC(=O)N1CCC(NC(c2ccc(Cl)cc2OC)=O)C1(C)C)OC CCC(C)C(C(=O)N1CC(COC)(NC(=O)C=CC(C)(C)C)C1)OC C#CC1(NC(C2C=CCN(C(=O)CCCOC(C)=O)C2)=O)CCC(C)(C)C1 c1(C(N2C(C(NOCCOC)=O)C=CC2)=O)ccc(O)cn1 C1(NC(C2(CCCC)CC2)=O)CC2CC1N(C(c1csc(CC)n1)=O)C2 c1(CC)noc(CN(C)CC2CC2)n1.C1(C(=O)N)CCN(c2ccccc2)C1 C1(NC(C(c2ccc(Cl)s2)C)=O)COCCN(C(C2(S(C)(=O)=O)CC2)=O)C1 n1(C(C(=O)NCC2(F)CC(NC(C3(C#C)CC3)=O)C2)C)nc(C)c([N+](=O)[O-])c1C N1(CCC(N2CCN(c3ccc(Cl)cc3)CC2)=O)CCC(F)C(O)C1 C1(NC(=O)COCC2CCOCC2)C2CC1N(C(=O)CC(O)C1CC1)C2 Cc1ncc(C(=O)N(CCCNC(=O)Cc2ccc(C(F)(F)F)nc2)CCO)n1C c1(NC(c2c(Cl)n[nH]c2C)c2n(CC)nnn2)ccc2c(c1)CN(C)C2 CC(CCN=c1[nH]c2c(c(=NC(CC3CC3)CC3CC3)[nH]1)COCC2)N(C)C Cc1ncccc1NC(C1CCC1NC(=O)CC1COCC1O)=O c1(C(=O)NCC2(CCNC(C34CCC(C3)C4)=O)CC2)coc2cc(F)ccc12 c1(C(=O)NCC(C)NC(C(c2cccc(C)c2F)O)=O)cc2n(c1)CCOC2 c1(SC)cc(C(=O)N(C(C)CNC(=O)C=Cc2ccc(C)s2)C)cc(Cl)c1 n1(CCC(=O)NCC2(OC)CN(C(c3cc(C)c(C)o3)=O)C2)cc[nH]c(=O)c1=O c1(OC)cc(CO)ccc1C(=O)NC1CCN(C(=O)Cc2cccnc2)C(C)C1 N1(C(c2nc(C)sc2)=O)C2CCCC1CN(C(c1nc(C3CC3)ncc1Cl)=O)C2 C(=O)(CCCCCC(C)O)NCCCN(C(C(CC)c1cccnc1)=O)CC c1(NC(C(=O)NCc2n(CCC)ccn2)=O)ncc(C)cc1F C(=O)(CC(C)C(C)(C)C)NC1C(CC(=O)NC(C)CN2CCCC2)C(O)C1 C(=O)(C1=C(C)CCCC1(C)C)NCC(CC=C)NC(C1CNC(=O)C1)=O c1(CSC)cc(C(N2CC3(C2)CN(C(C2(C)CCC2)=O)C3)=O)ccc1F N1(C(c2c(C)nn3c2CCCC3)=O)CCc2cc(Br)cc(F)c21 c1(NC(C2C(c3cccc(OC)c3)C2)=O)cc2[nH]ccc2cc1C CCCC(C(=O)N1CCCC1C1(O)CN(C(c2ncn(C)c2C)=O)C1)OCC N1(C(CC(C(C)C)C)=O)C(CNC(c2nc3ccccc3[nH]2)=O)CC2COCC12 Cc1cnc(C(N2CC(CNC(=O)CCn3cc(C)cn3)C2)=O)c(F)c1 N1(C(C(C(=O)OCC)CC)=O)CC2(C=C(C(=O)NCC3CC4(CC4)CO3)CO2)C1 N1(C(C=C(C)C)=O)Cc2occ(C(=O)Nc3cnn(CCF)c3)c2C1 C(=O)(C(C)(C)C(N)=O)NCCCOCCOCCNC(CC(C)F)=O C=CCC(CNC(C1CC1c1ccccc1)=O)NC(=O)C(C)=C(C)CC O=C(CS(=O)(=O)CCO)NCC1CCCCN1C(=O)C=CC(c1ccccc1)=O N1(C(C(CSC)O)=O)CC(C2CC2C(N2CC(S(C)(=N)=O)C2)=O)C1 c1(C(=O)NC(C2CC2CC(N2CC(F)CC2CO)=O)C)ccccc1C(N)=O N1(C(c2c(C)snn2)=O)CCCC(CCNC(=O)C(N2CCN(C)CC2)C)C1 c1(C(=O)NC2(C)CCN(C(c3c(C)cnn3C)=O)CC2)cnc2c(c1)NCC2 C12(CN(C(C)C)CC1C)c1n(nnn1)CCC(=O)N2C.C(C(=O)N(C)C)SCC.CO C(C(=O)NCC12CCCC1OCC2)(C(C)(C)C)NC(c1n(CC)nc(C)c1)=O C1(O)(C(N(C(C)CO)CC)=O)CCN(CC2(NC)CCCC2)CC1 C1(C(=O)NCC(=O)N(CC)CC)CC2CCC1N(C(C1(C(=O)NC)CCC1)=O)C2 CC(C)CCCC(C)C(=O)NC(C1(O)CCN(C(C2CCCC2(C)C)=O)CC1)C Cc1nc2ccc(NC(=O)NCCc3cncn3C)cc2nc1C N1(C(C)=O)CCOCC1NC(Cc1ccccc1)CCNC(=O)C(C)NC(N)=O c1(C(=O)NC2C(CNC(CCC=C)=O)C2)ccc2nccc(Br)c2c1 S(=O)(=O)(c1cccc(=NC(C)CCCO)[nH]1)NCC1(SC)CCC1 C1(C(=O)NCC(C)(C)NC(=O)CSc2nc[nH]n2)CCCCC1C1CC1 C(=O)(CCCS(N)(=O)=O)N1CCC(N(CCC)C(c2cc(F)cc(F)c2)=O)CC1 C12(NC(C(COC)N(C)C)=O)CC(CO)(C1)C2(F)F N12CC3C4CCC(C3C1)N(C4)C2=O.c1(OC)cc(CO)c(Cl)cc1C(=O)C(C)C N1(C(C(c2ccc(C)s2)C)=O)CCOC(CN(C(=O)C(c2cncn2C)O)C)C1 N1(C(c2c(CC)nnc(C)c2)=O)CC2CCC1C(CO)C2 C12(NC(C(C)C3CCC3)=O)CC(C1)N(C(=O)COCc1cccnc1)C2 Cc1cc(F)cc(C)c1C(N1CCC(O)(C(=O)N(C2CCOCC2)C(C)C)C1)=O C(CC1=CCN(C(=O)CC2CCC2OC)CC1)NC(CC1(OC)CCOCC1)=O N1(C(CC2CC(=C)C2)=O)CC(C2CN(C(c3cncc(F)c3)=O)C2)C1 C1(F)(C(=O)NCC(C)N(C)C)CCN(C(C2CCC(C)(C)C2)=O)CC1 C(=O)(C(C)CCOC(CC)(C)CNC(c1cccnc1)=O)Nc1ccccc1 C1(C(=O)NC2(CC=C)CN(C(=O)Cc3cncn3C3CC3)C2)OCC2CCCC12 C(=O)(C(=O)CC(C)C)NCC(C1CCCC1)NC(c1cc(C)no1)=O N1(C(c2cc(SC)nn2C)=O)C(CNC(c2sc(C)nc2C)=O)CC2CCCC12 C(c1ccc(C(=O)NC)cc1)=CC(=O)NCC1C(NC(c2nc(C)sc2)=O)CC1 N1(C(C(CCC)F)=O)CCC(C)C(CC(=O)Nc2cn(C)nc2C2CC2)C1 N1(C(C2CN(C)C(=O)N2)=O)CC2CCC1C(NC(c1c[nH]nc1C(C)(C)C)=O)C2 c1(OC)cc(-n2nc(CC3CCCCC3)nc2C2C=CCC2)cc(F)c1 n1(CC)cnc(C(=O)N(C(C(=O)NCC2(CO)CC2(C)C)C2CC2)C)n1 C#CCC(C)(C(=O)NC(C)C(O)C(F)F)NC(c1cnsc1)=O C(C(CC(C)C)C(=O)N1CC(C)C(C)(CNC(=O)C(C)(C)OC)C1)OC Cc1cc(C(=O)NC2CC(CNC(=O)C(C)C3CC3)C2)c(Br)cc1F C1(NC(=O)C2=CCCC2)CS(=O)(=O)CC1NC(c1ccc(OC(F)(F)Cl)cc1)=O Cc1cccc2[nH]c(C(N3CCN(C(c4ccc(F)cc4N)=O)C4CC34)=O)cc12 CC(O)(CNC(c1csc(C2CCCO2)n1)=O)CNC(=O)C=CSc1nc[nH]n1 C1(C(=O)NC2CN(C(C(CCC#C)O)=O)CC2(C)C)CCC2CC1C2(C)C c1(CNC(C2C(C(N3CC(=O)NCC3)=O)CCCC2)=O)cnc2n1CCOC2 C1(C(=O)NCC(C(C)C)NC(C2(C)COC2)=O)CCc2cnnn2C1 c1(C(=O)NC2CC(NC(c3ccc4c(n3)CCC4)=O)C2)ccc(F)c2occc12 c1(C(C(=O)N(CC(C)NC(c2c(CC)scc2)=O)C)(F)F)nc2ccccc2s1 c1(C(CCC(=O)N(C(CCNC(C(C(C)C)O)=O)C)C)=O)ccc2c(c1)CCC2 C1(NC(=O)C2=COCCO2)CN(C(c2occ3c2CCCC3)=O)CC(F)(F)C1 N1(C(=O)Cc2cccs2)CC2CN(C(c3cc4scnc4[nH]3)=O)CCC2(CO)C1 CC1(C)CCCN(c2nnc(C(F)F)o2)C1CNC(=O)CCc1nc[nH]n1 Cc1[nH]c(=NC2CCN(C(c3ncc(Cl)nc3Cl)=O)C2)ccc1C#N C1(C(=O)NCC2(Nc3cc(OC)ncn3)CCOCC2)CCN(C)C(=O)C1 Cc1ccc(CC(C(=O)O)NC(=O)Cc2conc2C)cc1F c1(OC)nc(N(C(C2CCNCC2O)=O)CC2CCCCN2C)ncc1C c1(C(=O)Nc2cc(C(=O)OC)sc2)ccc2ncc(-c3cc(O)ccc3F)n2c1 C1(C(=O)NC2(C)CCN(C(c3cc(OC)n(C)n3)=O)C2)CCC2(CC1)CC(O)C2 c1(C(=O)NCCn2cc(CCC(=O)O)nn2)cc(F)c(F)cc1Cl N1(C(Cn2c(C)cc(C)n2)=O)CC(C)CCC1CNC(C1(CO)CCOCC1)=O c1(C(N(C)CCN(C)C(c2ccc(C(C)(C)C)s2)=O)=O)cc(N)cc(O)c1 N1(C(CCC=CC)=O)CC(C)(C)OCC1CNC(C1CCC(=O)N(C(C)C)C1)=O N1(C(C=CC(CC)C)=O)CCOC2(C1)CN(C(c1cc3ncccc3s1)=O)C2 c1(CNC(COCC=C)=O)cc(C(=O)NCC(C)C(C)C)on1 c1(C(=O)NCC2C3CN(C(C(CC)O)=O)C(C3)C2)nc2ccccc2o1 CN=c1[nH]c(C(=O)NC2CCCN(C(c3cccc(Cl)c3)=O)C2)cs1 N1(C(C(=O)N(CC)CC)=O)CCC(C2(NCCS(=O)(=O)C(C)C)CC2)C1 C(CCN=c1nc(N2CCC(CC3CC3)CC2)c2sccc2[nH]1)c1cc(C)no1 CC1OC(C)CC1CC(=O)NCCOCCN(C)C(C1(CO)CC(F)(F)C1)=O N(C1CCCc2occc21)C(C(C1CC1)NC(C1CC(Cc2ccco2)C1)=O)=O CCC(CCCC(=O)NC1CCN(C)CC1C)NC(C1(n2cccn2)CC1)=O C(CNC(=O)CCc1cscn1)(C(C)(C)C)NC(CCOCCCOC)=O c1(C(=O)NC2(C)CCN(C(CC(C=C)C)=O)C2)cc(OC(F)F)cc(Br)c1 C1(NC(c2ccn(CC(F)F)n2)=O)CCC2CN(C(C3OCCCO3)=O)CC2C1 C(=O)(C1=CS(=O)CCC1)N1CCC(=CCNC(C2ON=C(C)C2)=O)CC1 N1(C(CNC(=N)N)=O)CCOC2(C1)CN(C(c1ccc(SC3CC3)cc1)=O)C2 c1(C(N2CC(NC(C(CCC)c3ccccc3)=O)C2)=O)cc(C)c(F)cc1N C(CC(=O)N1CCC(CC2CC2)C1)(C(F)(F)F)NC(C(CC)(C)NC(C)=O)=O C1(C(=O)NCc2nnc(CC)s2)CCN(C(c2ccc(O)nn2)=O)CC1O C(=O)(CC(C)(C)C(=O)N1CC(CCCCNC(=O)C(C)CSC)C1)OCC CCCCC(C(=O)NCCC(O)C(C)C)NC(=O)CN1CCCCC1C c1(C(N2C(C(C)NC(c3c(C)cno3)=O)CCC2)=O)ccc(Cl)cc1F N1(C(CC(=O)OCC)=O)CC2CCCN(C(C3CC(F)(F)C3(F)F)=O)C2C1 c1(CNC(C2(C)CC(C)OCC2)=O)nc2c(s1)CN(C(=O)C(C)(F)F)CC2 n12cc(nn1)CN1CC(C1)CC2.n1(NC(CC)=O)nccc1C(=O)O CC(C)(F)CCC(=O)NC12CCOC(CNC(C3CS(=O)(=O)C3)=O)(C1)C2 CC(C)(C(=O)NC1CCC(CNC(C2(n3cccn3)CCC2)=O)C1)n1cccn1 CC1=C(C(=O)Nc2nccc3c(Br)ncn23)C(C)(C)CCC1 Cc1nn(C)c2ccc(C(=O)NC3CC(NC(C4CCC(F)(F)C4)=O)C3)cc12 C1(C(N(C(CC)CSC)C)=O)C(C)OCCN1C(=O)C(C)NC(C)=O N1(C(c2ccc(SC(C)C)cc2)=O)CC(NC(C2CCC(=O)C2)=O)CC12CCC2 C1(NC(C2(C)N(C)CC(OC)C2)=O)CCN(C(=O)CC2(C#N)CC2)CCC1CO C1(C(=O)NCC=CCNC(C2(OC(C)C)CCOC2)=O)CCC(C)(C)O1 C1(C(N2C(C#C)CC2)=O)(NC(c2nc(C)c(C)s2)=O)CCN(C)C1 c1(C(N2CC(NCC3CC3)CC(C)C2)=O)c2c(nn1-c1ccccc1)CCCC2 n1(CC(=O)NC(CC)(C)CNC(=O)C2=C(Cl)CC2)cc([N+](=O)[O-])cn1 C1(C(N2CCC(O)(Cn3cc(CN)nn3)C2)=O)CC12CCOC(C)C2 N1(C(C(CC)C(C)C)=O)CCCC2(C1)CN(C(c1ccc(C)c(F)c1F)=O)C2 C(=O)(CCCCC(C)=O)NCC1C(C(=O)NCc2c(CC)cncc2)CCO1 C1(NC(CCSCCCC)=O)CCCC12CN(C(c1cc[nH]c3nccc1-3)=O)C2 C(CN=c1nc2ncn(C)c2c(NCCCc2ccsc2)[nH]1)NC(=O)NCC C[Si]1(C)CCC(CNC(=O)CCCC2(NC(c3csc(F)c3)=O)CCC2)C1 Cc1ccc(C(=O)NCC2CC(NC(C3(C)C=CCC3)=O)C2)cc1F N1(C(C)=O)CCC(C(N2CCCCC2)=O)CC1.N1(NC(C2CC2C)=O)CCCCC1 c1(CC)cc(C(=O)NC2CC(NC(C3CC34CCCC4)=O)C2)nn1C c1(C(=O)NC(CN(C(CCC)=O)CC)C)ccc(Oc2ccccc2)cn1 C(=O)(CC(CC1CC1)NC(=O)CNC(N)=O)N(CCCCO)C C12(C(=O)NCC3(NC(c4cn(C)[nH]c4=N)=O)CCOC3)CCN(CC1)CC2 C(C)(CCC(=O)N1CC(C)CC1C(N1CCC=CC1CC)=O)OCC c1(NC(=O)CCC2CCOC2)cc(C(=O)NCc2cnsc2)no1 N1(C(c2c(C)cccc2)=O)CCCN(C(c2coc(Br)c2)=O)C(CO)C1 CCCC(CNC(C1(N(C)C)CCCSC1)=O)C(=O)N1CC(OCC(F)F)C1 C12(C(C)NC(C(C)(N(C(C3C(C)CCO3)=O)C)C3CC3)=O)CCC(CO1)C2 C1(CNC(CN(C2CC2)CC)=O)CN(C(c2cc(CC3CCC3)c[nH]2)=O)CCO1 C1(CC(C)C)CCN(C(=O)CNC(=O)CNC(c2ccc[nH]2)=O)C1 Cc1c(C(=O)NCC(O)CN(C)C(c2sc(F)cc2Cl)=O)ccn1CCO CC(C)C(CCNC(C1CC1Cl)=O)NC(C12CC3CC1C2C3)=O C1(NC(C(CC)n2nccc2C)=O)CCC2CCN(C(=O)CC3CCCCC3)C12 C1(CC)(NC(=O)CC2COC(C)(C)C2)CCS(=O)(=O)CC1 C1(C(=O)NC(C(C)C)C(C)(C)O)CN(C(=O)CCc2ccccn2)CC(C)(C)C1 Cn1cc(C(N2C3CCC2C(CNC(C2CC4CC4C2)=O)C3)=O)ncc1=O CC(C)C(C)C(C)CC(=O)NCCCCN(C(=O)C(C)(C)c1ccnn1C)C c1(C(=O)NCC2(CNC(C(C)(C)OC)=O)CCOCC2)cc2n(n1)CCCC2=O c1(CNC(=O)NC2CC(CNC(=O)OC(C)(C)C)C2)cc(F)cc(Br)c1 C1(C)(C(=O)NCc2c(C(N(CC=C)CCC)=O)c[nH]n2)COC(=O)N1 N1(C(C2(O)CCC2)=O)CCCC(F)(C(N2C3CSCC2C3)=O)C1 C(=O)(CCCc1nc(C2CC2)no1)N(C(C)CNC(=O)COC)CC C1(C(=O)NC(C)C)CCC(C)N(C(=O)C(F)(F)CCn2cc(CN)nn2)C1C Cc1nc(=NC(=O)C2CCC(c3ccc(F)c(F)c3)CC2)o[nH]1.N1CCOCC1 CC1=C(C(=O)Nc2ccc(NC(=O)CSC3CC3)cc2C)CCS1(=O)=O c1(C(=O)NC(CC(C)Nc2cc(SC)nc(SC)n2)C)nccc2ccccc12 C12(NC(c3ncc(OC)cn3)=O)CCC(C1)N(C(C1(n3cccn3)CC1)=O)C2 c1(C(N2C3CC(CN(C(C4=C(CC)OCCC4)=O)C3)C2)=O)ccc2oc(O)nc2c1 N1(C(C2CC(=O)CC23CCC3)=O)CCSC2COCCC12 c1(C(=O)NC2(CC=C)CN(C(c3snc(C)c3N)=O)C2)cc(F)c(F)c(Cl)c1F N1(C(c2c(CCC)nns2)=O)CCCN(C(=O)CNS(N)(=O)=O)C(CO)C1 N1(C(c2cn(CCC)nn2)=O)C(C(N2CCNC(=O)C2C)=O)CCC12CC2 C12(CNC(C(CCC)NC(N)=O)=O)CN(C(=O)CC3CCC(O)C3)CC(F)(C1)C2 N1(CC(=O)NCC2N(C(C(CCC#C)O)=O)CCC2)C(=O)c2cccnc2C1=O C1(NC(C2C(CCC)C2)=O)COC2(CCN(C(c3cccs3)=O)CC2)C1 c1(CCCC)ocnc1C(=O)NCC1(F)CC(NC(=O)C(C)OCCC(C)C)C1 c1(OC)ncc(Cl)c(=NC2CC3CC(C2)N(C(c2cccc4cc[nH]c24)=O)C3)[nH]1 N1(C(c2cn(C)nc2)=O)CCC=C(C(=O)Nc2cc(F)c(F)c(F)c2)C1 N1(C(C2C3CN(C(Cn4ccc(C)n4)=O)CC2CC3)=O)CCC2(CCCOC2)C1 CCC(CCCC(=O)NC1CCC(C)CC1)NC(c1cc(C)n(C)c1)=O C(=O)(C(C#N)(CC)CC)N1CC2(CN(C(c3c(C(C)=O)cc(Cl)s3)=O)C2)C1 C1(NC(=O)CCc2ncc[nH]2)CN(C(c2ccon2)=O)CCC1C(F)(F)F C1(C(=O)NCC(C=C)O)(CC=C)CN(C(C2CCCO2)=O)C1 N1(C(C(COC)C)=O)CC(C)(C)CC1CC(=O)NCC(F)Cl C1(CC(=O)OCC)CN(c2ncccc2C(F)(F)F)CC(C)O1 c1(C(=O)NCCC(C)NC(c2nnc(O)nc2O)=O)ccc(C(F)F)c(F)c1 C1(CN(C)C(c2cocn2)=O)CCCC(NC(c2ccc(C(F)(F)F)cn2)=O)C1 CCC(CC)C(=O)NC1CCCCC1CNC(c1ccccc1Br)=O C12(CC)CN(C(c3cnc(CO)nc3)=O)C(CNC(=O)CC(C)NC(N)=O)(C1)C2 CC(C)C(CO)C(=O)NCCCN(C(C1(C)CCCN(C)C1)=O)C1CC1 CCCC(O)CC(=O)NC(CO)C(C)NC(=O)CCCc1nc(C)no1 C1(CC(=O)NC2C(NC(=O)CC3CC(=O)NC3=O)C2)C2CC3CC(C2)CC1C3 C(=O)(C1CCCc2n[nH]cc21)N1CCN(C(C(C(C)C)(C)O)=O)CC(C)(F)C1 c1(C2(C(NOCCCCn3cc(CC(=O)OC)nn3)=O)CC2(C)C)cccc(F)c1 C=C1CCC(C(N2CC(OC)CC2CNC(=O)CNC(=O)CC)=O)CC1 c1(C(N2CCC(CCNC(C=CC(C)=O)=O)C2)=O)ccc2nc(O)n(C)c2c1 c1(CC)ccc(NC(=O)CCC(C)NC(C2CCN(OC)CC2)=O)cc1C c1(C(=O)NC(C)CN(C(=O)C=CCN(C)C)C)cn(CCO)nn1 C=CC1CC(N=c2ccc(Br)c(S(=O)(=O)NCC(N3CCOCC3)C)[nH]2)CCO1 C1(C(N2CCCC(NC(CCCC#CC)=O)(CC)C2)=O)CCC2(CC1)CC2(F)F C1(CC(=O)NC(C2CN(C(=O)CCCC3CC3)CCO2)(C)C)CCCCC1(C)C C1(C2CCN(C(=O)CC(c3cccs3)N(C)C)C2)(NC(CCC(=C)C)=O)CC1 C=CC(C)(C)CC(=O)NC(C)(C)C=CC(=O)NC1CCN(C)CC1C N1(C(c2ncc[nH]2)=O)CCC2CCC(C1)N2C(C1CCCCCCN1)=O C1(CC(=O)OCC)CN(C(c2cn(CC3CC3)nn2)=O)CC1CO.C12(CC1)C(=O)N2 N1(C(CN(CCOC)C)=O)CC(C)(C(N2CC3CC2CN3C(C)C)=O)CC1(C)C Cc1cccc(C(CNC(C2CC2(C)C)=O)NC(c2ccc(C3CCC3)[nH]2)=O)c1 C(=O)(CCCCC(F)(F)F)NC1(C)CCCN(C(CC2CCC(C)(C)CO2)=O)C1 Cc1cccc2c1CC(C(=O)NC(CNC(=O)C(C)N(C)C)C(C)C)O2 C(=O)(C(F)(CNC(C1CC(=O)NC1(C)C)=O)C(C)C)NC(C(=O)NCC)CC c1(CC)ccc(C=CC(=O)NC2CN(C(=O)CCn3ccccc3=O)C3CC23)o1 C1(NC(C(N2CCSCC2)C)=O)CC2CC1N(C(=O)C=Cc1cn(C)nn1)C2 C1(N(C(CCC2(CCC#C)N=N2)=O)CC2CC2)CCN(C(=O)C(C)C2CCCC2)C1 N1(C(c2nc(C)c(F)cc2)=O)CCC2(CCCN2S(=O)(=O)c2ccncc2)CC1 CC(C)C(C)CN(C(=O)C(=O)Nc1cnn(-c2ccccc2)c1)C N1(C(CCC2CC(OC)C2)=O)CC(NC(c2conc2C)=O)C2CCCC2C1 N1(C(C(C)O)=O)CC2CC1CCN2C(=O)CCc1cc(Cl)no1 C(CC(=O)NCC1(C)CCOCC1)(C(F)(F)F)NC(Cc1c(C)cnn1C)=O c1(NC(C2N(C(c3cn(C)nc3)=O)CCCC2)=O)cc(F)c(Cl)cc1Cl N1(C(C(Cc2ccco2)NC(c2cc(CC)[nH]n2)=O)=O)C2CCCC1COC2 c1(C(N2CCN(C(CN3CC(C(=O)OC)C3)=O)CC2)=O)c[nH]nc1[N+](=O)[O-] c1(N(CCc2c(OC)cccc2)C)nccc(=NCc2noc3c2CCCC3)[nH]1 Cc1cc(O)c(Cl)cc1C(=O)NCC1CCN1C(C12CC1COC2(C)C)=O C1(C(=O)OC)CCC(C2CCCCC2)CN1C(C1CC1c1ccco1)=O C1(CC(=O)NC(CN(CCCC)C)C)CN(C(=O)Cc2cnns2)C(C)(C)C1 N1(C(CNC=O)=O)CC2CCN(C3C(C(=O)NCCN(CC)CC)C3)CC2C1 N1(C(C2(CC#C)CCOC2)=O)CCC2(CCN(C(=O)CCC3CCCN3C)C2)C1 N1(C(c2scc(C(=O)OC)c2)=O)CC(C2CN(C(=O)C(C)CC(N)=O)C2)C1 C#Cc1ccc(CCCC(=O)Nc2cnn(CCN3CCNC3=O)c2)cc1 C#CC1(C(=O)NC(C)CCSC)CN(C(=O)C(CC)=CCCC)C1 Clc1cc(Cn2cc(C3CCOCC3)nn2)on1 C(=O)(C(O)CCC(C)C)N1C(CNC(Cc2nc(CC)sc2)=O)CCCCC1 C1(NC(c2c(C)nco2)=O)CCCC12CCN(C(=O)C=C1CCSCC1)C2 C(=O)(CCS(N)(=O)=O)N1CC(SC)C(NC(=O)C(c2cnn(C)c2)N(C)C)C1 c1(C(=O)NCC(C)N(C(c2cnnc(O)c2)=O)CC)cc2cccnc2cc1F n1(CC)nc(C(=O)NCCC(C)NC(=O)C(C)CN2CCCCC2)ccc1=O CCCC(C(=O)N(C)CCC1CCN(C(=O)C(C)(O)C(C)C)CC1)S(N)(=O)=O C(CCN=c1[nH]c(=NCCC(OC)OC)[nH]c2c1COC2)N.C=CCSCC Cc1ccc(NC(=O)CC2COCCN2C(c2cc(F)ccc2I)=O)c(CO)c1 c1(CC)cc(C(N2CCCC2CC(N2C(CO)CCC2CO)=O)=O)c(C)o1 c1(C(=O)NCC2N(C(=O)CN3CCCC3)CC2)ccc(SC2CCOC2=O)cc1 CN1CCN(C(=O)CCCNC(C23CCCN2CCC3)=O)CC1(C)C C(C1CCc2ccccc21)OC(Cc1c(CC)cccc1CC)=O Cc1cccc(CCC(=O)N(C(C)CCNC(C2CCC2)=O)C)c1Cl c1(CC)nnc2n1CCCC2C(=O)NCC(C)CNC(c1ccc(OC)s1)=O C1(CN(C(C(CC)O)=O)C)CN(C(=O)CCn2ccnn2)CC12CC2 N1(C(CC(C)(C)SC)=O)CCC2(CC(NC(=O)C(C)(C)c3cc[nH]n3)CO2)C1 C=CC1(C(=O)NC2CN(C(c3cc(N)ccc3F)=O)CCC2CO)CCCCC1 C1(NC(=O)CC2CCCOC2)CC2CN(C(c3ccc4cncn4c3)=O)CC2C1 N1(C(C2(c3c(OC)cccc3)CCC2)=O)CCC(O)C(C(=O)NC2CCCC2)C1 C#CC1(O)CC(C(=O)N(CCNC(c2cc(Cl)cnn2)=O)Cc2ccccc2)C1 N1(C(C2ON=C(CC)C2)=O)CCN(C(=O)CCCCCC(C)O)C2CCCC12 C(C(C)NC(c1ccc(CO)cc1)=O)(C(C)C)NC(C(=Cc1cccs1)C)=O CCC(C)CCC(=O)N1CCN(C(C2COCCOC2)=O)C(C(C)C)C1 N#Cc1ccc(C(=O)NC2C3CN(C(c4coc(Cl)n4)=O)CC23)c(O)n1 Cc1cc(O)n2ncc(C(N3CCCC3CN(C(=O)Cc3cnsc3)C)=O)c2n1 c1(C(N2C3C(N(C)C(c4cccc(=O)o4)=O)CC(C3)C2)=O)cc2cn[nH]c2cn1 C1(C(=O)NC2(CNC(CCC3CCC(C)O3)=O)CCCCC2)COCCN1C=O N1(C(C2N(C)C(=O)NC2)=O)CCC(C2CCN(C(=O)C(C)(C)CCC#N)CC2)C1 c1(C(=O)NC2(C3CN(C(Cc4ncc(C)s4)=O)C3)CC2)noc2c(F)cccc12 C1(NC(Cc2ccc(C)cc2Cl)=O)CN(C(=O)CN(C)C)C2(CCC2)C1 c1(C(=O)NC2CCC(C)(CNC(c3nnn(CC)c3C)=O)C2)ccc(C)cc1N c1(C(=O)NCCCN(C(CCOC)=O)CCO)ccc2n[nH]c(C)c2c1 C=CCC(F)(F)C(=O)N1CCSCC1c1cccc(OC(F)(F)F)c1 CCCCCS(=O)(=O)CC(=O)N1CCCN(C(C2CCCCCC2)=O)CC1CO c1(SC)ccc(Cl)c(C(N2CCC(CNC(C3C4CCCOC34)=O)C2)=O)c1 C1(CC(=O)NCC2(C)CCC(=O)N2)C2CCCC2N1C(=O)C(=O)NCC(F)F Cc1onc(Cl)c1C(=O)NC(C)CCCNC(=O)CCCOc1ccc(F)cc1 C(CCC(=O)N(CC)CC1CCCC1NC(=O)Cc1cnns1)OCCC C1(C(=O)NCC(N(C(CCc2onc(CC)n2)=O)C)C2CC2)CCCCC1(F)F C12(C(N3C(C)(CNC(C(C(=O)OC)OC)=O)CCC3)=O)CCCC(C1)OC2 C=C1CON(C(=O)C2CCC(C)N2C(=O)Cc2ccc(O)cc2)C1 C1(C(=O)NCC2CN(C(Cn3ncn(C)c3=O)=O)C2)CCCN2CCCC12 C=C(CNC(C1CCCS1)=O)CCNC(c1cn(CCCF)nn1)=O c1(OC)ccc(C(C)NC(C2CC2NC(C2CCC2)=O)=O)c(C)c1 c1(OC)ccc(C(=O)C(=O)OC(c2ccc[nH]2)C)cc1F c1(C(=O)NCC2CC(NC(CC3(OC)CCC3)=O)C2)cc2sccc2s1 C1(CC)C(C(=O)N(CC(O)CN(C)C(c2cc(Br)ccn2)=O)C)CCN1C C(=O)(CC1OCc2cc(Cl)ccc21)NC1CN(C(CN(C)CC)=O)C(CO)C1 c1(C(=O)NCC2(F)CC(NC(C(C)O)=O)C2)c(Cl)cc(Cl)nc1N C(N=c1[nH]c2ccc(Cl)cc2s1)C1C(NC(C2CCCC(C(N)=O)C2)=O)CCC1 c1(C(=O)NC(CNC(C(CC)OC)=O)CO)ccc(OCC(N)=O)cc1 C1(CC(=O)N(CCC#C)CC)C2CCCC2N1C(C1CC(CCO)C1)=O N1(C(C(C)(C)CC#N)=O)CCC2CC(NC(=O)CCS(N)(=O)=O)CCC2C1 C(CC1=CCN(C(=O)C(O)C(F)F)CC1)NC(C(n1cc(Br)cn1)C)=O c1(C(C)(C)C)nc(=NCCCc2ccccc2Br)s[nH]1 Cc1cccc(C)c1C(=O)NCC(F)CNC(c1cc(Br)cn1C(C)C)=O C1(CO)(COCC)CCCN(C(C2(NC(COCCC)=O)CCC2)=O)C1 c1(NCC)ccc(C(N2CCC(C)(CNC(=O)CCCOC)C2)=O)cc1[N+](=O)[O-] C1(CNC(C(C)CO)=O)CCCC2CN(C(=O)CC3(N(C)C)CCC3)CC12 CCCCCC(C(=O)N(C)CC1CN(C(=O)CCCOCCOC)CCO1)C(C)C C12(CNC(C(CC#C)C)=O)CCC1CN(C(c1ccc(Br)cc1O)=O)C2 C1(C(=O)NC2C(NC(c3cccc(C(C)=O)c3)=O)CC2)C2CCC1(C)C2(C)C c1(C(C)(C)C)nnc2ccc(N3CCCC3)nn12.N12CC(C(C(F)F)C1)NC2=O c1(CNC(C(CCC)NC(=O)CC2CCCC23CC3)=O)cc(F)ccc1C C1(NC(=O)NCc2cc(C(=O)OC)cc(F)c2)CCC2=NN=NN(C2)C1 C1(CNC(=O)C=CCO)CCC2(CO1)CC(NC(c1csc(Cl)c1Cl)=O)C2 c1(NCC(O)CN2CCN(CC(c3ccccc3)O)CC2)ccc(O)cc1 C1(c2nnnn2C(C)(C)C)(NC(c2cncc(NC)c2)=O)CCN(C)C(C)C1 N1(C(c2c(C(C)C)nns2)=O)CCCCC(CNC(c2cc3n(n2)CCO3)=O)C1 CCC1C(=O)Nc2ccc(C(=O)N(CCCOCCNC(C3CCC3)=O)C)cc21 C(C(C(C)C(C)C)NC(=O)CC(=O)NCC(F)(F)F)NC(CCCNSC)=O c1(C(=O)NC2CCC(NC(=O)COCCF)C2)sc(N2CCOCC2)nc1Cl N1(C(C=C(C)c2ccsc2)=O)CCC(CNC(c2cc(Cl)n(C)n2)=O)C12CC2 C1(NC(C2N(C(c3c(C)n(C)nn3)=O)CC2)=O)CCC(C)(C)CC1C Cc1ccc(O)c(CC(=O)NC2CCOCC2NC(C2(C)CCCS2)=O)c1 Cc1cc(C(=O)N(C(C)CNC(=O)COCc2cc(C)no2)C)nc(O)n1 c1(OC)ccc(C(=O)NC(C2CCCCN2C(=O)CN2CCCC2)C)nc1 C12(C(NOCCOC)=O)CC(CO1)N(C(=O)CCCCCOC)C2 c1(NC2CC(CNC(c3c(C)nc(CCC)o3)=O)C2)cc2c(cn1)C(=O)CCC2 c1(CN2CC(C(N3CCC(C(=O)OC)CC3)=O)C(O)CC2)ccccc1[N+](=O)[O-] C1(C(N2CCOCC2(C2CC2)CO)=O)CSC(c2ccccc2O)=N1 C1(C(=O)NC2(COC)CN(C(C3CC4CCC4C3)=O)C2)COCC(C)O1 C(=O)(CC(F)(F)Br)N(C)CC1N(C(c2cc(C)ns2)=O)CCC1 c1(CNC(C2N(CC)CCOC2)=O)ccc(CNC(C2(F)CC2C)=O)c(F)c1 CC1CN(C(C2CNC(=O)CN2C(C2CCC3(CCC3)C2)=O)=O)CC(C)(C)O1 C1(C(N2CCN(C(c3ccc(O)cc3)C)CC2)=O)C2C3CC4C1C2C34C(=O)OC C(=O)(C(C)C(O)CC(C)C)N1CCC(COC)(NC(=O)COC2CC=CC2)CC1 CC(C)CC(C)CC(=O)N1CC2CCCC2(NC(C2CCS(=O)(=O)CC2)=O)C1 c1(C(=O)NCC(C)N(C)CC2CCC3CC3C2)ccc2sccc2c1 N1(C(C#CCNC(Cn2c(C)nnn2)=O)=O)CC(C#N)(N(C)C)C1 C(=O)(CCCC(CC)NC(C1Cc2nccn2C1)=O)Nc1ccc(CC)nc1 C(CCN=c1nc2scnc2c(N2CCC(C3CC3)C2)[nH]1)c1n(C)ncn1 N1(C(C(C(C)NC(c2c(C)non2)=O)C)=O)CC2OC(=O)N(C)C2C1 N1(C(C(C2CC2)NC(CC(CC)C(C)C)=O)=O)CC2CCOC(=O)C2C1 c1(C(N2C(C(=O)NCC(O)C(F)(F)F)CC2)=O)ccc(F)c(C(F)(F)F)c1F Cn1ncc(C2CCC2)c1C(N1CCC(C)(NC(=O)CC2(C)CCOCC2)C1)=O C1(NC(c2n(CC=C)nnn2)c2occc2Br)CCOC(c2cccc(Cl)c2)C1 CC1(C)OC(C)(C)C1(O)C(=O)NCCOCC1CCOC1 C(=O)(C1=NOC2(CCC2)C1)N1C(C)C(NC(=O)C(=O)NCC(F)F)CC1 C1(CCn2cc(CN(C(c3cc(OC)ns3)=O)C)nn2)CCCCCC1 CCCC(C)(O)CC(=O)N(CC(=O)NCC(N1CCCC1)=O)CC(C)C C(=O)(C(C)(C)CCC(=O)NCC1CCCC2(CN(C(=O)C(C)(C)F)C2)O1)OC N1(C(c2cn(CC(C)C)nc2)=O)CCN(C(=O)C(C)C2(O)CCC2)CC1C(C)C C(=O)(C(C(C)(C)C)c1cc[nH]n1)N1CC(OC)C(NC(=O)C(=O)C(C)(C)C)C1 N1(C(C2(C)CCNC2=O)=O)CC2(C1)CN(C(C1C3CC4C(C3=O)C14)=O)C2 C(N=c1[nH]cnc(Cl)c1C(OC(F)(F)F)C)C1(NC(=O)OCCO)CC1 c1(C(N(C2CCCN(C(=O)C(C)CO)C2)CC)=O)cc(C(F)(F)F)cc(F)c1 N1(C(c2onc(CC)n2)C)CCC2C(CCCN2C(C2C3CCCC23)=O)C1 N1(C(C2C(CNC(C3CC(C(C)C)C3)=O)OCC2)=O)C2CCCC1CC2 C(=O)(CC(C)C(=O)OC)NC1CCN(CCNC(C=COCC)=O)CC1 c1(C(N(CCN(C(C2CCC(CCC)CC2)=O)C)C)=O)ccc2nn[nH]c2c1O N1(C(C)=O)CC(NC(=O)NC2CCCC2CN=[N+]=[N-])C2(COC2)C1 c1(C(=O)NC(C2CCCC2)CNC(C2(C)C(C)C2)=O)cc2n(n1)CCCO2 N1(C(c2cc(C)cc(F)c2)=O)CCC2(CC1)CC(C(=O)Nc1cncc(F)c1)C2 c1(-n2c(C(C3(CCl)CCC3)NC(CCC=C)(C)C)nnn2)ccc2c(c1)CCC2 CN1C(=O)NCC1C(=O)NC1CC(CNC(=O)C(F)OC(F)(F)F)C1 C1(C(CN(C(c2ccccc2)CSC)C)C)CCOCC1 N1(C(c2occ(C)c2)=O)CC2CC(C1)CN(C(c1cc3ccnn3cn1)=O)C2 N1(C(C23C(C)OC(C)(C2)C3)=O)CCC(C2CC2)(CNC(c2ccc[nH]2)=O)C1 N1(C(c2ccc(SC)cc2)=O)CCC2(CCN(C(=O)Cn3cncc3C)C2)C1 N1(C(C(CC)CC)=O)CC2C3CCC(C2C1)N(C(C1CCC2(CCOC2)O1)=O)C3 C1(NC(C(n2ncc(C)c2)C)=O)CC12CC(NC(C1(N=[N+]=[N-])CC1)=O)C2 S(=O)(=O)(c1ccc(Br)c(F)c1)N1CCC2(C(C(=O)Nc3ccc(Cl)nc3)C2)CC1 N1(C(CC=CCC)=O)CCOC(CCNC(C2(C#N)CCOC2)=O)C1 C12(C(=O)NC3CCC(N(C(=O)CS(=O)(=O)NCC4CC4)C)CC3)COCC(C1)OC2 CCCC(C(O)C(=O)NCCOCCCF)NC(=O)C1=CCOCC1 c1(C(=O)NCC(C)NC(=O)C(c2ncc(Cl)n2C)(F)F)cc2cc(Cl)ccc2o1 N1(C(=O)NCC2C(NC(=O)OC(C)(C)C)CCC2)CCCC(N=[N+]=[N-])C1 c1(C(N(CC(CC)NC(=O)CN2CCOCC2)CC)=O)cc2n(n1)CC(O)CO2 C1(N(CC(F)(F)F)C(c2occc2Cc2ccccc2)=O)CCS(=O)(=O)C1 c1(OC)cc(N2CCC(NC(C3CCC3)=O)CC2)nc(COc2cnccn2)n1 c1(C(N(CCCNC(CC(C)OC)=O)C(C)C)=O)cc(C2CC2)cc(F)c1 C12(CNC(c3c(C)nc(O)[nH]3)=O)CCCC1N(C(=O)CCC1(O)CCC1)CCC2 C1(C(=O)NCCCCNC(CC)=O)CCC(=O)N(CC)C1 c1(CNC(CSC)=O)n[nH]cc1C(=O)NCCCC1(C)N=N1 CCCC(C)CC(=O)N(CC(CO)(CO)NC(c1cc(C2CCC2)no1)=O)C N1(C(c2cnc(N(C)C)nc2)C(=O)NC)Cc2ncsc2C1 N1(C(C(CCC)C(C)C)=O)CCCC2CN(C(C3CCCCC3(C)C)=O)CC12 c1(CNC(=O)CC2C=CCCC2)ccc(CNC(C2CC23CCOC3)=O)cc1 C=CCCCC(C(=O)NC(c1ccn(C)c1)C)NC(c1ccc(C#N)cc1)=O N1(C(C(COC)O)=O)CC2CN(C(c3ccnc(OCCO)c3)=O)CC2C1 C1(F)(C(N2CC3C(CNC(c4ccn(C)n4)=O)C3C2)=O)C(C)(C)C1(C)C C1(NC(CCC2CC(OC)C2)=O)CN(C(C2(C#N)CC3(CC3)C2)=O)CCC1CO c1(Cc2n(CC)c(N(C)CC=Cc3ccccc3)nn2)c(F)cccc1F c1(C(=O)NC2C(C(C)C)CN(C(c3ccc[nH]3)=O)CC2)noc2cc(F)ccc12 C1(CNC(CCC(=O)OC)=O)(NC(=O)CCC2NC(=O)NC2=O)CCCCC1C N1(C2CCCN(C(C3C(C)(C)CCC3)=O)C2)CCN(CC=CCO)CC1=O Cc1cc(C(C)C)nc(N2CC(NC(c3cnc(C(F)F)nc3)=O)C(C)C2)n1 c1(NC(C=C)=O)ccc(-c2ccc(NC(=O)CCOC3CCNC3)c(F)c2)cc1F c1(C(=O)NC(C(C)C)C(C)NC(c2cn(C)ccc2=O)=O)ccc(O)c(F)c1 C1(NC(c2c(C(C)=O)ccs2)=O)CCOCC1NC(c1ccc(C(F)F)cn1)=O c1(OC)ncc(C)cc1C(N1CC2CC1C2NC(C1CC1[N+](=O)[O-])=O)=O CC1OC(C)C(C)N(C(=O)NC(c2nccn2C)C)C1C c1(C(=O)NCC2CC(C)N(C(C3CCCCO3)=O)C2)cnc2[nH]nnc2c1 c1(C(N2CCC(CCCNC(CC3C(C)C3)=O)CC2)=O)ccnc(Cl)c1N c1(C(=O)NCC2COCCN2C(c2cccnc2)=O)c(O)nnc2c1CCCC2 c1(OC)ccnc(O)c1C(N1CC=CC(NC(c2cncn2C)=O)C1)=O C1(N(C(=O)Cn2[nH]cnc2=N)C)CCCN(C(=O)CCOc2cccnc2)C1 N1(C(c2c(C)nns2)=O)CCC(C)(CCNC(c2cn(CCCC#N)nn2)=O)C1 c1(C(N2CC(C(C)NC(=O)C(C3CCOCC3)=O)C2)=O)ccc(CN(C)C)nc1 c1(C(=O)NC(CC(C)NC(C2CC2c2cccs2)=O)C)cc2occc2[nH]1 N1(C(C2CCCC23CC3)=O)CC2CCCC(C1)N2C(c1c(F)ccc(F)c1O)=O C1(CNC(C2C(CC)CCC2)=O)CCCC12CCN(C(C1C=C1C)=O)CC2 c1(C(=O)OC)nccnc1C(=O)NC(C)CC(C)NC(=O)C(c1cnn(C)c1)=O c1(N(C)Cc2ccc(F)cc2)ccc2c(c1)CN(Cc1ccc(N)cc1Br)CC2 Cc1nnc2n1CC(C(=O)NCC1CCCN1C(=O)Cc1ccc(CO)cc1)C2 N1(C(C(C)N2CCC2)=O)CCN(C(C2CC(F)(F)C2)=O)C(CC2CC2)C1 C1(C(C)C(=O)NCC=CBr)CCN(C(=O)CCc2cccn2C)C1 c1(C(c2nnnn2CCCF)NC(c2ccc(C)o2)CC)ccc(OC)nc1 c1(C(=O)NC2(CO)CCN(C(CSCCCC)=O)C2)cc2ccc(OC)nc2[nH]1 c1(CNC(CCN(C)CC)=O)c[nH]nc1C(N1CCCC1C(=O)NC)=O C1(=CCNC(C(CC)O)=O)CCN(C(=O)Cc2ccc(-n3cccc3)cc2)CC1 c1(CC)cc(C(N2CCCCC2c2cn(-c3ccc(CC)cc3)nn2)=O)c(C)o1 CC1COC2(C1)CN(C(=O)C#CCNC(c1csnc1Cl)=O)C2 C1(CC(=O)NC2C(NC(c3c(COC)ncs3)=O)C2)Cc2ccc(Cl)cc2C1=O CC1(CNC(=O)CCOC2CCC2)CCN(C(=O)CC2CC3CC(=O)C2C3)CC1 NS(=O)(=O)C1CCC(C(=O)NCCNC(c2ccc([N+](=O)[O-])cc2O)=O)CC1 CCCCC(C(=O)N(CCCN(C)C)CC)NC(c1cc(C)c(C)[nH]1)=O N1(C(c2n(C(C)C)ncc2)=O)CC2ON=C(CNC(c3ccsc3)=O)C2C1 c1(CC)cc(C(N2CC(CC(C)NC(=O)C=CBr)C2)=O)ccc1F c1(COC)cc(C(=O)NC2COCC2NC(=O)Cc2csc(C)c2)no1 c1(C(=O)NCC(C(C)C)NC(C(CNC(C)=O)(C)C)=O)nc2ccccc2[nH]1 C1(CN(C(=O)CC2CC2C)CC)CCN(C(=O)CC2CC3CCC2O3)CC1 C(=O)(C(C)CCCC(C)C)NC1CC2CN(C(c3ncc(C)nc3)=O)C(C1)C2 CC1CN(C(c2c(O)cccc2F)=O)CCC1CNC(C1(CF)COC1)=O N1(C(c2c(OC)c(C)cs2)=O)CC(N(C(=O)C(C)=C2CC2)C)C(C)(C)C1 C(=O)(C1=CCCCO1)NC1CCC(CCNC(=O)Cc2nc[nH]n2)C1 C1(CC(=O)NCC(N(OC)C)=O)CCN(C(=O)C(C)CC#N)C1(C)C c1(C(=O)NC2C(NC(c3nc(C)oc3)=O)CCC2)ccc2nncn2c1 c1(C(=O)NCCN(C(CC)C)C)n[nH]c2c1CN(C(=O)C1=CCCCCC1)C2 Cc1cc([N+](=O)[O-])cc(Cl)c1NC(C1(O)CCN(Cc2cc(F)ccc2Cl)C1)=O Cc1cncc(C)c1C(=O)NC(CC1CC1)C(=O)NCC1CC12CC2(F)F C1(CC(N2CC(C)(OCC(=O)N(CCCOC)CCO)C2)=O)CCCC(C)O1 C1(C(=O)NCC(C)C#N)(CNC(c2c(C)noc2)=O)CC12CCC2 c1(OC)cccc(C(C)C(=O)NCCC(C)NC(=O)CSC)c1 C(=O)(C1CCCc2nn[nH]c21)N(CCOCCCNC(C1C(C)C1C)=O)C N1(C(c2c(CC)cc(Cl)cc2)=O)CC2(CC(NC(=O)C(C)(O)CC)CO2)C1 N(C(=NCCc1ccc(CO)cc1)NC1CCCC1)CC1CCCC(C)O1 C1(C(N2CCC(C)(NC(c3ccc(Cl)cn3)=O)CC2)=O)CCCCC1P(C)(C)=O C(CCCCC(=O)N1CC(O)CC1(C)C)N(C(C1C(CC)CCO1)=O)C c1(OC)ccc(C(C)C(=O)NC2(C)CCN(Cc3cnc(C)o3)C2)c(C)c1 C(=O)(C(C)(C)C(=O)N1CCCC(C)(NC(=O)Cc2ccc(C(F)F)cc2)C1)OC N1(C(COCCCCC)=O)CC(O)C(O)C1CNC(=O)CC1OC(C)(C)OC1=O c1(C(N2CCC(CNC(C3(C4CC4)CC3)=O)C2)=O)cc(Cl)ccc1[N+](=O)[O-] S(=O)(=O)(c1ccccc1S(=O)(=O)N1CCOCC1)NCC(N(C)O)=O C(CCF)(C(=O)Nc1ccc(CO)nc1)NC(C1CC=CC(O)C1)=O C1(C(N(CC(C)NC(COC)=O)C)=O)(NS(CC)(=O)=O)CCSCC1 C1(C(=O)OC)Cc2ccsc2CN1C(=O)CNC(C)=O.c12ccc(C)cc1S2 C1(NC(CSCCC)=O)CCN(C(=O)CC23CCCC2C3)C12CCC2 c1(C(=O)NC(CNC(COCCOCC)=O)CO)c(F)cc(F)cc1Cl c1(CCC(=O)N(CCN(C)CC2CCN(CC)C2)C)ccc(O)nc1 N1(C(CCCNC(C(C(C)(C)O)F)=O)=O)CCC(C2CCC2)C1 N1(C(C(C=C)OC)=O)CC(C(=O)NC2(COC)CCC2)C(C2CC2)C1 N1(C(C(C(C)C)N(C)C)=O)CCCOC(CNC(C2CCC3(CC3)C2)=O)C1 CC1CCCC=C1C(=O)N1CCOC(CNC(=O)Cc2c(F)cc(F)cc2F)C1 CCC(C)C(C(=O)N(CCCCCNC(c1ccc(F)cc1)=O)C)N(C)C N1(C(C(CC=C)C)=O)CC2CCCC(C1)N2C(C1CCN(CC(F)(F)F)CC1)=O C1(CCC)C(=O)NCCN1C(C1CCN(C(c2n[nH]cc2[N+](=O)[O-])=O)CC1)=O N1(C(C(CC)=CC)=O)CC(CNC(c2cc(-c3ccccc3)ns2)=O)CC1C C=CCC(C)C(=O)NC(C)C(C1CCCCC1)NC(=O)CCCNC(=O)C1CC1 N1(C(C#CC)=O)CCC2(C1)CN(C(c1ccc(-c3cccc(OC)n3)cc1)=O)C2 N1(C(CN(CC(=O)NC(C)C)C)=O)CCN(C(C2(C)C=CCC2)=O)CC(C)(F)C1 CC#CCC(CO)NC(C1CCCC1CNC(C1(C(C)(C)OC)CC1)=O)=O C1(NC(c2ccc(CC)nc2)=O)CCC12CN(C(=O)C=CC(=O)NC1CC1)C2 c1(OC(COC)C(=O)OC)cccc(NC(=O)CC2(NC(C)=O)CC2)c1 c1(C(=O)NC2CC(NC(=O)COCc3nc[nH]n3)C2)cc(C2CC2)cc(F)c1 c1(CCNc2cc(N(C)Cc3cnccn3)ncn2)cccc(Cl)c1Cl C(CCCC(C)NC(=O)C(C)COc1ccccc1)NC(CC(=O)NCC)=O C1(C(N2CCCN(CC(N3CCOCC3)=O)CC2)=O)CC2(CCC2)CCO1 O=C(N=c1c(Br)c[nH]cc1I)C1CCN(S(=O)(=O)C2CCCCC2)C1 c1(C(=O)NC2CCC3CC2CN3C(C2CC(Cl)(Cl)C2)=O)coc2ccc(F)cc12 C1(NC(C2(C)CC2)=O)CN(C(=O)C(c2cccc(Br)n2)(F)F)C(C)(C)C1 c1(CNCCCCCC(C)(C)C)cccc(S(=O)(=O)NC2CC2)c1 C12(CNC(CN(C3CC3)CC)=O)CC1CN(C(=O)COCc1nc(C)no1)C2 N1(C(C(C)(C)SCCC)=O)CC2CN(C(=O)CCCOC(C)=O)CC2C1.C1CO1 Cc1nc(C(C)C)sc1C(C)N(C)C(=O)NCC1CCCC1C Cc1ccc(F)c(C(=O)NOC(CC(C)C)C(=O)N(C2CCN(C3CC3)C2)C)c1 CC1=C(C(=O)N2CCOCC(F)(CNC(=O)CN3CCNC(=O)C3)C2)CCCO1 S(=O)(=O)(c1c(C)cc(C)cc1C)NCCC(=O)NC(CC#C)C(N)=O c1(C(=O)NCC(CNC(CCC#C)=O)F)cc(F)ccc1-n1ccnc1 c1(C(N(CC(CNC(C(CC)(C)F)=O)C)C)=O)ccc(C)c(N)c1 CC1(C)CCCCC1NC(=O)CC1C2CC1N(C(C1CN3CCC1CC3)=O)C2 C(CCCC(=O)N1CCC(F)(CNC(C2(Cl)CC2(C)C)=O)C1)N(C(C)=O)C N1(C(CC(=O)OCC)=O)CC2(CC(CC(=O)NC3(CO)CCOC3)C2)C1 CC1(C)CC(=O)NCC1C(=O)NCC=C1CCN(C(=O)CCP(C)(C)=O)CC1 CC(O)C(F)(F)C(=O)NC1CCC(CNC(C2COC(C)(C)C2)=O)CC1 N1(C(C2CC(C)C2)=O)CCC(C)(CC(=O)NCC(C)CN2CCCC2)C1 C1(NC(C)=O)CCCN(Cc2cnn(C)c2CCO)C1 c1(C(N2CC(NC(C3CCCC3)=O)CC(C)(C)C2)=O)cc(F)c(C#N)c(F)c1 C1(C(=O)OC)N(C(C2CCCOC2)C(=O)NCc2cccs2)CCOC1(C)C C#Cc1cc(C(=O)NC2CCCCC2NC(C2CCC(C)(C)C2)=O)ccc1C Cc1ccc(C(N2CCC(C(F)(F)F)C2C)=O)cc1S(=O)(=O)N(C)C C12(C(=O)NCc3c(C)non3)CC(C)(CN1C(c1sccc1C#N)=O)C2 c1(OC)cc(C2CC2)ccc1NC(C1NC(=O)N(C(C)(C)C)C1=O)=O.c12nnnn1C2 N1(CC)CCC(NC(=O)OC(C(=O)OC(C)(C)C)Cc2cc[nH]n2)CC1 CC(C)C(C(=O)NC1CCN(C(C2(C)CCC2)=O)CC1F)C(C)C C(=O)(C1COc2ccccc21)N1CCCC2(CN(C(=O)Cc3ccc(Cl)s3)C2)C1 C1(CNC(CC(C=C)CC)=O)CN(C(C2CC(CC(F)F)C2)=O)CCC12CCC2 N1(CC)CCCC(C(=O)NC2CC(O)(CNC(c3csc(C(F)(F)F)n3)=O)C2)C1 C(=O)(C1CCc2c(Cl)cccc21)NC1CN(C(C(C)CCc2cccc(F)c2)=O)C1 c1(C(N(CC)CC2CCCN2C(=O)CSCC(F)F)=O)cc(=O)cc(Cl)[nH]1 CS(=O)(=NC(=O)CCC1CS(=O)(=O)C1)c1cc(F)ccc1F CC1CC(N(C)C(=O)NCc2ccnc(-c3ccccc3)c2)CC(C)O1 c1(NC(c2ccc(Cl)nc2NCc2ccc(I)c(F)c2)=O)ccc(O)cc1Cl CC1COCCN1C(=O)CCC1CCN(C(C2(C)CCCC2O)=O)CC1 C1(C(C)(C)C)CCN(C(C2CCCOCC2)=O)C(CNC(c2cc[nH]n2)=O)C1 N1(C(C(CCO)N(C)C)=O)CC2CS(=O)(=O)CC2(CNC(c2csnn2)=O)C1 Nc1ncc(C(=O)NCCOC2CCN(C(=O)C=Cc3cnc[nH]3)C2)cc1Br c1(OCC)cnccc1CCNC(N1CC(N2CCOCC2)C1)=O CC(Cc1cnn(C)c1)C(=O)NC1CN(C(=O)COc2ccsn2)C1 N1(C(CNC(C(C)(C)OC(C)C)=O)=O)CCC(O)C(C)(C)C1 C1(O)(C(=O)NC2CC3(CC(NC(c4scc(C)c4C)=O)C3)C2)CCCC(C)(C)C1 N1(C(N2CC(SCC(C)CNC(=O)C(C)Cn3ccnc3)C2)=O)CCCS1(=O)=O C1(CCNC(c2cc(C(C)=O)[nH]c2)=O)C(C)CCCN1C(=O)C1=COCCC1 c12ccccc1NC(=O)C1(CCC1)C(=O)N2.C1(Sc2ccccn2)CCOCC1 c1(C(=O)NC2C3CN(C(C4C(C(C)(F)F)C4)=O)C2C3)cnc2c(c1)COC2 c1(C(N2CCCC3(C2)CN(C(C2CC=CC2)=O)C3)=O)ccc2cc[nH]c2c1F c1(N2CCN(CC(C)(C)NC(=O)C(F)C3CC3)CC2)nc(Cl)nc2c1CCOC2 C1(NC(C(CC=C)CC=C)=O)CN(C(c2nc(=N)cc[nH]2)=O)CCC12CCC2 N(C1CCc2c(Br)cccc21)C(=O)NC1C(c2c(C)cccc2)(C)C1 CC1(C)CN(C(c2ccncc2Cl)=O)CC1C(=O)NC1CC2(C1)CC(O)C2 C1(CN(C(CCCOCC=C)=O)CCN(C)C)COCC(C)O1 Cc1cc(CC(=O)NC(C)CNC(=O)C(F)CC2CCCCC2)on1 C1(CNC(c2ccc(OCC)cc2)=O)CCCN(C(=O)CC(C)CF)CC1 O(N=C1CCCCCC1)CC(N1CC(OC)(CNC(=O)C(O)CN(C)C)C1)=O C1(C(N2C(C(N(C)Cc3cnc[nH]3)=O)CC(O)C2)=O)CCCC2(CC2)C1 C1(C(=O)OC)CN(C(=O)C(=O)NCc2c(Cl)cnn2C)CCN1C N1(C(CSC)=O)CCc2[nH]nc(CNC(=O)C(C)Oc3cccc(CO)c3)c2C1 N1(C(c2c(C)c[nH]n2)=O)CC(NC(=O)Cn2nnc(=N)[nH]2)C2(CCC2)C1 N1(C(C=Cc2ncn(C)c2)=O)CC2CC(C1)N2C(=O)CC1CC(C)(C)CO1 N1(C(C2CCC(C)O2)=O)CCCCC1CN(c1ncncc1I)C C(=O)(C(=O)C(F)(F)F)N(C1CCCC(NC(=O)Cn2ccc(C(F)F)n2)C1)C c1(NC(C2(NC(C(C)CCN(C)C)=O)CC(F)C2)=O)cnc2[nH]ncc2c1 C12(NC(C(c3ccc(CC)s3)=O)=O)CC1CN(C(C1CCC(C)CC1)=O)C2 C1(SC)CN(C(=O)CC2(C)CC2)CC1NC(C1CN(C2CCOC2)C1)=O Cc1nc2ccc(C(=O)NC3CC4CC3N(C(=O)CC35CCCC3C5)C4)cc2o1 c1(NCc2ccc(CC)[nH]2)nc(OCC(F)(F)F)ccc1Cl N1(C(C(C(CC)C)c2ccccc2)=O)CCC(C#N)(C(C)C)CC1 N1(C(c2c(CN)noc2)=O)CC(=O)N2CCCCC2C1 c1(C(N(C(CN(C(C(C)SCC)=O)C)C)C)=O)cc2c(cn1)OCCO2 Cc1c(C(=O)CNC(=O)C(c2ccc(Cl)cc2)C2CC2)sc2ccccc12 N1(C(C2N(C(C)C)CCC2)=O)CCN(C)C(C(NC[Si](C)(C)C)=O)C1 c1(NC(N2CCC(N(c3ccccc3)C)C2)=O)ncnc2c1ncn2C c1(C(=O)NC(CCOC)CNC(=O)CC(F)(F)Cl)ccc(N=[N+]=[N-])cn1 CC(CS(=O)(=O)N1CCC(O)C(N2CCCC2)C1)C(C)(F)F Cc1ccc(C(=O)NCC2(C(=O)NCC3NC(=O)NC3=O)CCCC2)nc1 Cc1nncc(C(=O)NCC23CC(C2)C(NC(=O)C(O)C2CC2)CO3)c1C N1(C(C(=O)NCCSc2ccccc2)=O)CCn2c(cc3c(Cl)cccc23)C1 c1(C(=O)NCC(c2cccc(C)c2)NC(C(CC)F)=O)cccc2nn[nH]c12 C1(C(N2CC(OCC)(CNC(=O)CC3CC(OC)C3)C2)=O)CC12CCCC2 c1(CC)cccc(NC(c2cn(C3CN(C(C4CCC(C#N)C4)=O)C3)nn2)=O)c1 Cc1nc(C(=O)N(C)C)ccc1C(N1CCCC1CNC(C1C2CNC(=O)C12)=O)=O c1(C(C(=O)NCCC(=C)CNC(C2CC(n3ccnc3)C2)=O)(F)F)ccc(C)cc1 N1(C(=O)NC(c2cc[nH]n2)C2CC2)CCS(=O)(=O)CC1C1CC1 C1(C(N2CCCC(NC(CSCC#C)=O)C2)=O)CCCC2(C1)CC2(F)F c1(OC)cccc(NCCC(C(C)C)NC(C2CC3(C2)CC3F)=O)c1[N+](=O)[O-] N1(C(C(C)(C)C#N)=O)CC2CC1CC2CNC(=O)CCC1CC(C)(C)CO1 c1(C(=O)NC(CC=C)CNC(c2cc(OC)n[nH]2)=O)cc(O)ccc1OC(F)F C(C(F)(F)C(C)(C)O)NC(C1(CNC(C=C(C)C(C)(C)C)=O)CC12CCC2)=O c1(C(=O)NC2(C)CCN(C(c3ccn(C)c3)=O)C2)cccc(F)c1Br C1(CC(=O)NC2CCN(C(=O)Cc3ccno3)CC2O)CCCCC12CC2 N1(C(c2sccc2Cl)=O)CC(CO)C2(C1)CN(C(c1sccc1C1CC1)=O)C2 C(=O)(C(CCC)C(C)C)NCC1(F)CCN(C(COCC(=C)C)=O)C1 Cc1ccccc1NC(N1CCN(C(=O)NC23CCC(CO2)C3)CC1)=O CC1CN(C(c2cnc(Cl)c(Cl)c2)=O)CCC1NC(c1cc(O)no1)=O Cc1csc2ncc(C(=O)NCCC3CCCN3C(=O)Cc3cccc(N)c3)n12 C12(C(=O)NC3(C(CC)O)CC3)COCC1CN(C(=O)CCCC1CC1)C2 c1(C(C(=O)N(CC(C)O)CCNC(CC(=O)OC)=O)C)cc2ccccc2o1 N1(C2CC2)CC(CNC(c2cn(CCC)nn2)=O)CC1C.C12(CC1)C(=O)NC2=O c1(C(N2CCCN(C(C(C)C3CC3)=O)C(C)C2)=O)cc2c(n1C)CCOC2 C1(CC(=O)NCC2CC(NC(=O)CCn3cccn3)C2)CCCCCO1 C(=O)(C1=C(C#N)CCC1)NC(C(=O)N(C)Cc1ccoc1)CCF N1(C(C2(CC)CCCC2)=O)C2CCC1CN(C(=O)C(C)SC)C2 N#CC1(C(N2CCC(F)(CNC(c3cncn3C3CC3)=O)C2)=O)CC2(CC2)C1 Cc1cc(NC(=O)CCC2CCN(C(C3(Cl)CCC3)=O)C2)cc(C)c1C Nc1ccnc(C(N2C3CCC2C(NC(=O)Cn2cc([N+](=O)[O-])cn2)C3)=O)c1Cl Cc1nc2c(C(=O)NC3CC3CNC(c3ccc(C)c(C#N)c3)=O)ccnc2[nH]1 CC1=NOC(=O)C1CC(N1CCOC(CNC(c2cn(C)cn2)=O)C1)=O c1(CNC(C=C(C)CNC(=O)CC(C)N(C)C)=O)nocc1C N1(C(C(CO)N(C)C)=O)CC23CCCCC2(C1)CN(C(c1ccc(Cl)o1)=O)C3 CC(C)C(O)C(=O)NCC12CC1CN(C(c1ccc(CO)cn1)=O)C2 C1(C(=O)NCC2CCCN(C(=O)Cn3cncn3)CC2)Cc2cccc(F)c2O1 C1(CCNC(CC=CCC)=O)CC(F)(F)CN1C(C1CC2OC1C1CC21)=O CC(C(O)C(F)F)NC(C1(NC(=O)C#CC2CC2)CC(F)C1)=O N1(C(CN(C2CCC2)C)=O)CCCCCCC1C(N1CC=CC1CF)=O c1(C(N2CC(NC(C(CC)(C)CO)=O)C(O)CC2)=O)c[nH]c2cc(F)c(F)cc12 C12(CNC(CN(C(C(n3ncc(C)c3)C)=O)CC3CC3)=O)CCCC(CO1)C2 Cc1ccn(CC(=O)NC2(CCCCNC(C3C(N)CCO3)=O)CC2)n1.C(C)C CCC(CC(=O)NCCCC(=O)NC1CCCN(CC2CC2)C1)C(C)(C)C c1(C(=O)NCC(CC)NC(C(C2CCC2)OCC)=O)oc(Br)cc1C CC1(C(=O)N(CCCO)CCO)CCCN(C(C23C(=O)C4CC2C3C4)=O)C1 C1(O)(C(=O)NCC2(C)CCN(C(CC3(C(=C)F)CCC3)=O)C2)CN2CCC1CC2 c1(NC(=O)CNC(c2cc(C3(O)COC3)on2)=O)cccc(Br)c1 c1(OCC(=O)N(CCCNC(C2CCC(CC)C2)=O)CC)ccc(F)nc1 C(C)(C)(CC(=O)NCC(C)(O)CN(C)C)NC(C(CC)SC)=O C1(NC(c2ncc(CC)s2)=O)CCC(C)N(C(=O)CN2CCCS2(=O)=O)C1 C1(NC(C2C(OC(C)(C)C)C2)=O)CC2(CCC2)CCO1.N12CCC1(C)CC2=O C1(CNC(C(Cc2cc[nH]n2)NC(=O)C=CC(F)(F)F)=O)C2CCCCC12 c1(N2CCC(NCC(C(C)C)NC(=O)C3=CCOC3)C2)ncccc1C(F)(F)F N1(C(COCCCOC)=O)CCCC12CCCN(C(c1cc(C)oc1C)=O)C2 c1(NC2CCCCCN(C(C3N(C)CCCC3)=O)C2)nc(Cl)nc2[nH]c(O)nc12 N1(C(C2(COCC)CC(=C)C2)=O)CCCCC1c1nn[nH]n1 c1(C(=O)NCCOC2CCN(C(CC=CCC)=O)C2)cc2ncccc2o1 N1(C(C(C)NC(=O)OC)=O)CCN(C(C2CCN(C)C(=O)C2)=O)CC1C(C)C Cn1cc(C(C(=O)NC2CC(C)(C)C2)NC(=O)C=Cc2nccs2)cn1 C#CCC(CC#C)C(=O)NC1CN(C(=O)C(n2ccc(C)n2)C)CC1C1CC1 C1(C(=O)NCC(C)NC(c2c(C)noc2C(C)C)=O)CC(c2ccncc2)=NO1 c1(C(=O)NCC(CNC(C(C=CCCC)O)=O)(C)F)c[nH]c(C#N)c1 C1(CCCC)CN(C(=O)CN2CCP(C)(=O)CC2)CCN1C(=O)CC(F)(F)F Cc1cc(N)c(C(N2CCCCC2CNC(=O)Cc2ccsc2C)=O)c(F)c1 C1(NC(c2ccc(SC)o2)=O)CC(F)CN(C(=O)CC2CC2(Cl)Cl)C1 C1(CSCC(=O)NC2C(CNC(CCC#C)=O)CC2)CC(=O)N(C)C1=O C(CC1CCC1)(C(=O)NC1CCC2CC12)NC(C(C)=C1CCC1)=O n1(CC)ccnc1C(=O)N(CCC(=O)NCC(Cl)C(C)O)C(C)C C1(C(=O)NC2CN(C(C(F)=CCC)=O)CC2(C)C)Cc2ccccc2C1(C)C C1(NC(c2c(C)cc(F)c(Cl)c2)=O)CC1C1CCN(C(=O)Cc2cnc[nH]2)CC1 C(=O)(C#CC1CCCOC1)NC1(CO)CCN(C(C2CCN(C)CC2)=O)CC1 N1(C(C2CC(OC)C2)=O)CCN(C(=O)C(C)C(=O)N2CCCC2)C(C)C1 N1(C(c2c[nH]nc2F)=O)CC2CCN(C(C3COC4(CCC4)C3)=O)C2C1 C1(C(=O)NCC(CC)O)C2CCCC2CN1C(C1CCC1C)=O CC(C)C(C)(O)C(=O)NC(C)C(CO)NC(C1(F)CCCC1)=O C1(CC(=O)N(CCC)CCNC(c2ccc(CN(C)C)o2)=O)CCOCC1 C1(C(N2C(CC#C)CCCC2)=O)CN(C(=O)CC2CCOC2(C)C)CCC1(C)C N1(C(c2oc(C)c(CO)c2)=O)CCN(C(C2OCCC2C(F)(F)F)=O)CC1C CCC(CC(=O)N1CC(C2CN(C(c3c(CC)nc(C)n3C)=O)C2)C1)C(C)C c1(C(N(CCCCNC(Cn2c(C)cc(C(F)F)n2)=O)C)=O)ccc(Cl)cc1N Cc1cc(C2CC2)nc(=NCCC2CCN(C(=O)C3=NOCC3)CC2)[nH]1 c1(OC)ccccc1OCC(=O)NC(C1CCN(C(c2ccnnc2Cl)=O)C1)C c1(C2N(C(c3ccc(C(F)(F)F)cc3)=O)CCC2)nc2cnccc2[nH]1 N1(C(C(=O)N(C)CC2(CNC(CCOC(C)=O)=O)CC2)C)CCCC(O)C1 C1(CNC(c2ccc(CNC(C3C(C)=CCS3)=O)s2)=O)CC12CCOCC2 Cn1cc(CNC(c2cc(CCNC(=O)CC3CC(F)(F)C3)on2)=O)cn1 N1(C(=O)CCc2ccccn2)CCOC2(CCN(C(C3CC3F)=O)C2)C1 C1(NC(c2c(CC)nc(=N)[nH]c2)=O)COC2(C1)CN(C(=O)C1=C(Cl)CCCC1)C2 CCCC(C)C(=O)NC1(C)CN(C(C23CCC2C3)=O)C1 N1(C(CSC(C)(C)C)=O)CCC=CC1C(N1CC(C#N)(CCF)C1)=O N1(C(CCOC(C)=O)=O)CCC2CN(C(C3(c4ccno4)CC3)=O)CCC12 Cc1cccnc1C(=O)NCCC(C(C)C)NC(c1ncnn1C)=O CC1CC(C)N(C(c2cnc(O)n(C)c2=O)=O)CCN1C(c1c[nH]c(=O)cn1)=O C(CC(C)C)(C(=O)N(C)OC1CCCC1)ONC(C(C)=Cc1cccnc1)=O CCCCCCC(F)C(=O)NC1CN(C(c2ccncc2)=O)CC1C(F)F c1(OC)ccc(C(N2CC(N(C(=O)CCC3CCCO3)C)C2)=O)c(F)c1 N1(C(C=CC(CC)C)=O)CC2(NC(C3CC(C(F)(F)F)C3)=O)CCC1CC2 c1(C(N2CCOC(c3nc(C(=O)OC)cs3)C2)C(=O)NCC)cccc(CC)c1 c1(C(N2CCC(N(C(C(CCCCC)O)=O)C)C2)=O)cnc2ccccc2c1 N1(C(c2ccccc2C(F)F)=O)CC(CO)C2(C1)CN(C(C1CC13CCC3)=O)C2 C1(CC)CCN(C(c2ccc(Cl)s2)=O)C(C(=O)NCCOCCN=[N+]=[N-])C1 Cc1cnn(CC(=O)N(C)CC2CN(C(c3cnc(C(F)(F)F)s3)=O)C2)c1 c1(C(N2C(CN(C(=O)Cc3ccoc3)C)CCC2)=O)cnccc1Br C1(CCC(=O)NCC2(C)C(C)(C)C2)CCCCN(C(c2cccs2)=O)C1 N1(C(C=NOC)=O)CCC(C)(C)C(NC(=O)C(C)Oc2ccc(Br)cc2)C1 N1(C(c2cc(OC)no2)=O)CCC(C2CCCN(C(c3sccc3C#N)=O)C2)C1 C1(NC(CC(C)(C)SC)=O)CCN(C(=O)CCOC2CC2)CC1c1ccccc1 c1(CC(=O)NCC2(F)CCCN(C(c3c(C)c[nH]n3)=O)C2)ccc2ncsc2c1 n1(CC(=O)NCC(N(C(=O)CC2CC2)C)C2CC2)ncnn1 CN1N=C(CC(=O)N2CCCC(NC(C3(n4cncn4)CC3)=O)C(F)C2)CC1=O C1(CC(=O)NC(C(=O)OC)C2CCC2)CN(C(=O)CC2CCCN2C)CCO1 c1(OC)ccc(CN=C(NCC2(C)COC(=O)N2)NC2CC(C)(CC)C2)cc1 N1(C(CC2CCN(C(CC(C)O)=O)C2)=O)CCC2(CCCNC2=O)CC1 C(CN=C(NCc1ccc(C)n1C)NC1CCCC(F)(F)C1)SC Cc1nn(-c2ccccc2)cc1CNC1CCOC1C c1(CCC(=O)NCC2C(NC(C3(CCOC)CC3)=O)CC2)ccc(O)nn1 c1(C(=O)NC2C(C)CCN(C(=O)C(C)(C)C)C2)cc(F)cc2cnccc12 N1(C(Cc2c(C)ocn2)=O)CCC(C2CCN(C(=O)CC3=NNC(=O)C3)CC2)C1 CCC(CC)C(F)C(=O)NCC1CC(COC)CN1C(=O)Cc1cccnc1O C(CC1=CCN(C(C)(C)C)CC1)NC(=O)NCC(CC(=C)Br)(C)C CC1C(NC(c2cn(CC(F)F)cn2)=O)CCN1C(C1CCOCC1)=O N1(C(C=C(CC)CC)=O)CCC2(CC1)CN(C(C1CCCC(C(N)=O)CC1)=O)C2 c1(C(N(C(CC(=O)NCCOCCC=C)CC)C)=O)c[nH]c2cnccc12 S(=O)(=O)(c1ccc(N)cn1)NC(c1ccnn1C)CC C1(O)(CC(N2CC=CC2CN(C(=O)C(F)(F)Sc2cnn(C)c2)C)=O)CCCC1 Nc1c(C(N2CCOC3CN(C(=O)C4=CCOCC4)CC23)=O)sc2nccnc12 C1(C(N(C(CC)C(=O)N(C)Cc2c(C)cnn2C)C)=O)CC(C)CC(=O)N1 C1(NC(CC(C)N(C(c2cc(C)nn2C)=O)C)=O)CCCCCC1(C)C c1(C(=O)NC(C(=O)NC2CC(OC)C2)Cc2ccccc2)cc(F)ccc1O N1(C(C(C)CNC(c2cn(C3CC3)nn2)=O)=O)CCn2ncnc2C1 c1(C(=O)OC)cc(C(c2nnnn2C2CCCC2)NCC(c2nncn2C)C)cs1 O=C1CCC(C(=O)NCC2(O)CCN(C(=O)CSCc3ccccc3)C2)CN1 N1(c2nnc(-c3c(C)cco3)s2)CC2CCCC(NC(=O)C(CC)NC(N)=O)C2C1 c1(CC)cccc(C(N(c2nccc(CO)n2)CC(C)(C)C)=O)n1 C1(NC(=O)CCSC(F)(F)F)CC12CC(NC(c1c[nH]nc1F)=O)C2 N1(C(c2ccn(C)n2)=O)CC2C3CCC(C2C1)N(C(c1ccc(S)cc1)=O)C3 C1(C(=O)NC2CC2CNC(C(OCC)OCC)=O)(CSC)CC(F)(F)C1 [N-]=[N+]=Nc1cc(NC(c2cc(Br)nn2C2CCCCO2)=O)ccn1 N1(C(COCCOCC#C)=O)CCN(C(=O)C(c2cnn(C)c2)=O)C(C(C)C)C1 C1(CC(=O)NCC(C)(C)NC(=O)CCc2nc(=N)[nH][nH]2)CCCCC1F c1(C(N2CCCC(C)(NC(c3cc(C)ncc3)=O)C2)=O)ccc2ccccc2c1 C(=O)(CCCS(C)(=O)=O)NCC(C)(CNC(C1CCCCS1)=O)OC O=C1CCc2cc(C(N3CCCC(NC(C4C=CCC4)=O)CC3)=O)ccc2N1 C(C(C)C(=O)NCC1CCCCS1)N(C(C1(CC(=O)OC)CC1)=O)C C=CCCC(CC(C)C)C(=O)NC1(CN(C)C(C2CCN(CC(C)C)C2)=O)CC1 C12(C(=O)NCCCN(CCOC=C)C3CC3)CCCC1NCC2 C(=O)(C1CNC(=O)c2ccnn21)N1CC2(CN(C(CCC(=C)Cl)=O)C2)C(CO)C1 Cc1ncc(Cl)cc1C(=O)NCC#CCNC(c1cnn(-c2ccncc2)c1)=O N1(CCNC(C(n2ccc(C)n2)C)=O)CCN(C(C2(n3nccn3)CC2)=O)CC1 c1(C(N2CC(O)(CCNC(C(CC)(C)O)=O)C2)=O)cnc2c(c1)c(C)nn2C C1(c2nc(C)on2)CC2CCC(C1)N2C(c1cc(I)ccc1O)=O c1(OC)cccc(SCC(N2CCOCC2CN(C)C(C2CCCOC2)=O)=O)c1 c1(C(=O)NC2(COC)CCN(C(=O)CCOC3CCC3)C2)cccc([N+](=O)[O-])c1 c1(C(=O)NC2(C)CCN(C(CC=CC=C)=O)C2)cc2c(Br)c(F)ccc2[nH]1 c1(C(c2nnnn2Cc2cccc(Cl)c2)NCc2n(CC)ccc2)cccc(I)c1 c1(OC(C(=O)N(CCN(C(C=CC(CC)=CC)=O)C)C)C)ccc(Cl)c(C)c1 CCC(CC)(CC)C(=O)NC1CCC(F)(CNC(c2ccc(C)cc2N)=O)C1 N1(C(C2CC3(C2)CS(=O)(=O)C3)=O)CC(NC(C2CS(=O)(=O)C2)=O)C2CCCCC12 CC1=C(C(=O)NC2CC2NC(C2(CC3CC3)CCCC2)=O)C(C)(C)CCC1 C1(CC(N2CCC(N(C(=O)Cc3nnc(C)o3)CC)C2)=O)OCCOC1(C)C CCCC(C)CC(=O)N1CC2CC2C1CNC(=O)CN(C)CCc1ccccc1 c1(C(=O)NC(CCCC)CNC(=O)C#CC2CC2)cnc(OCC(F)F)c(Cl)c1 c1(CC(C)(C)CO)nc(C2=NOC(C(C)(C)C)C2)n(Cc2ccc(F)cc2)n1 N1(C(C)=O)CCc2cc(O)ccc2C1C.c1(C2COC2=O)ccccc1 Nc1[nH]c(=NCCC2CCCN2)ccc1[N+](=O)[O-] C1(C(=O)NCC2CCC3(CCC3)OC2)CC2(CO1)CC(F)(F)C2 C1(C(N2C(C(N3CC(C(=O)OC)C(F)C3)=O)CC2)=O)CC2CC(=O)C1C2 C(CN=c1nc(C)c([N+](=O)[O-])c[nH]1)NC(C1(C)C(CC)CCC1)=O c1(C(N2CCCCC(CO)C2)=O)cn2ccccc2n1 c1(C(=O)NCCCCNC(CC(C)F)=O)cncc(-c2ccc(F)cc2)c1 c1(OC)cc(C(=O)NCC(CO)NC(C2(C)CCCNC2=O)=O)cc(Cl)c1 CN1CCN(C(c2cccnc2N)=O)CC1CNC(=O)C#CC1(C)CC1 CCCC(C)(C)C(=O)N1CCCCC(CNC(=O)CC2CCCN2C)C1 c1(N2CCC(NC(CS(CC)=O)=O)C(C)C2)nc(Cl)nc2nc(Cl)n(C)c12 CCCC(CCCO)C(=O)N1CCC2(CNC(=O)C(F)(F)C3CC3)CCCCC12 n1(CC(=O)NCCN(CC(C)O)C(=O)C=CC2CC2)ncnn1 c1(CC(=O)NCC(C)(CC)NC(CN(CCC#C)C)=O)c[nH]c2c(F)cccc12 c1(NC(CN(C2CCCN(C(=O)C(C)(C)C)C2)C)=O)ccc(N(C)S(N)(=O)=O)cc1 N1(C(c2cnc(Cl)s2)=O)CC2CC(C1)N2C(c1cnn2ccsc12)=O c1(C(=O)NCCC2CCC(NC(C(CSC)(C)C)=O)C2)n[nH]c2c(C)cccc12 C1(C(N(C2CCSC2)C)=O)CC(C)(C)CCN1C(=O)C=CCO N1(C(C2CN(C)C(=O)N2)=O)CCC2(CCCN(C(C3CC(Cl)(Cl)C3)=O)C2)CC1 C1(C(N2CC(NC(CSCCC(C)C)=O)C(C(F)F)C2)=O)CCCCN(C)C1=O CN1CCC(C)(C(N2CC(CCCCNC(=O)C(F)CC3CC3)C2)=O)C1=O N1(C(C2CC(C)(NC(C3CC4C=CC3O4)=O)C2)=O)CCCN2CCCC2C1 C(CCc1ccc(Br)cc1)(C(=O)NCC)N(C)Cc1ccc(CC)s1 Cc1ccc(S(=O)(=O)NC(C)(C)C(c2ccc(O)cc2)=O)cc1C Cc1[nH]c(C#N)cc1C(=O)NC(C(=O)NC1C=CCCCC1)C(C)(C)O CCC(C)CC(=O)NCCCCN(C)C(C1CC(C)C(C(=O)OC)O1)=O N1(C(C=CC(CC)C)=O)CCCC(O)(CNC(c2ccsc2)=O)CC1 c1(C(N2CCC(F)(CNC(c3c(C)cco3)=O)CC2)=O)cc(Cl)c(F)c(Cl)c1 C(=O)(CCS(=O)(=O)c1ccccc1)NC1(CNC(C2(C)CC(C#N)C2)=O)CCC1 C=C(C)C1OCCCC1C(=O)NCC1CN(C(C2(O)COC2)=O)CCC1(C)C Cc1oncc1C(=O)NCC(=O)NC1CC1CNC(C1CCNC1=O)=O c1(C(C)C(=O)NC(C)C=CC(=O)NC(C)(C)Cn2cccn2)ccn(C)c1 C1(CC(=O)NCCOC)CCCN1C(c1ccsc1Cl)=O c1(C(N2CCC(CC)(CO)C2)C(=O)NC(CC)C)cc(Cl)ncc1Cl c1(CN(C(=O)CCn2cc(-c3cc[nH]n3)nn2)C)cccnc1Cl Cc1cc(Br)cc2cc(C(N3CCC(N(C)C(c4ccco4)=O)C3)=O)oc12 CCN=c1[nH]cc(C(=O)N(C)CC2CCN(C(C3CC3F)=O)C2)s1 Cc1coc(C)c1C(N1CCN(C(N2CCN(C(=O)C(C)N(C)C)CC2)=O)CC1)=O C(C(C)(O)CNC(c1csnc1C(F)F)=O)NC(C(c1ccccc1)C)=O CCC(F)(F)CC(=O)NCCCNC(C1COCC1C(F)(F)F)=O C1(C(N(CCn2cc(CN3CCOC3=O)nn2)CC)=O)CCC2(CCC2)C1 N1(C(CC2N(C(=O)CCC3CCCC3)C3C2CCC3)=O)CCC(F)(F)CC1 Cc1cc(Cl)c(C(N2CC(NC(c3coc(C(C)(C)C)n3)=O)CC2C)=O)cn1 N1(C(C2(COC)CC2)=O)CCC2C(COC2CC(N2CCOC(O)C2)=O)C1 c1(C(=O)NCC2(C)CCCN2C(c2cc(N)cc(N)c2)=O)ccc2nsnc2c1 C1(CNC(c2n[nH]c(C)c2O)=O)CC2(C1)CN(C(=O)CCCN1CCCC1)C2 C1(CNC(CCC(=O)NCC)=O)CC2(CO1)CN(C(C13CCC(C)(C1)OC3)=O)C2 c1(CNC(=O)CONC(=O)c2ccsc2)nccc2[nH]ccc12 OCCC(N=c1ccnc(N2CC3CSCC(C3)C2)[nH]1)c1ccccc1 c1(OC)ccc(C(N2CCC(C)C(NC(C3(C)CCC(F)(F)C3)=O)C2)=O)c(Cl)n1 Cc1nnccc1C(=O)NCC(C(=O)NC1COC(C)(C)C1)N(C)C C1(NC(c2c(C(C)=O)ccc(F)c2)=O)CC2CC1CN(C(=O)C(C)(C)F)C2 C#CCC(C)(C(=O)N1CCC(CC(C)O)CC1)NC(c1cc(CC)[nH]n1)=O N1(C(c2c(C)ocn2)=O)CC2CCC2(NC(=O)Cc2ccc(OCC#N)cc2)C1 CC1NC(=O)CCC1CNC(=O)C(N1CCC(Cc2nccs2)C1)=O c1(N(CCCNC(c2cc(CCC)c(C)s2)=O)C)ncnc2cc(Br)sc12 c1(CC(N2CCC(C)(NC(C(C)=C3CCCC3)=O)C2)=O)cccc2cnccc12 N1(C(c2c(S(C)(=O)=O)csc2)=O)CCC2(CCN(C(=O)Cc3ccco3)CC2)C1 C1(C(=O)NCCC(C)NC(=O)Cc2csc(CCn3cnnn3)n2)CC=CCO1 C(CCCCCNC(=O)C=CCCC(C)C)NC(Cc1c(C)ocn1)=O CC1COCC(C(=O)NC(c2ccnn2C)C(=O)NCc2cnccc2Cl)O1 c1(C(N2C(C(=O)NC(CCC)C)CSCC2)=O)cc(Cl)nc(Cl)c1 c1(C(C(=O)NCCC(C)N(C(c2ccc(C)s2)=O)C)C)c(C)noc1C Cc1n[nH]c2cc(C(=O)NCC3CN(C(=O)CCN4CCCC4)C4CC34)ncc12 N1(C(c2n(C(C)C)ccc2)=O)CCC(C)(NC(c2cc(-c3cccs3)on2)=O)C1 c1(C(=O)NCC2(OC)CN(C(C34CC(C#N)(C3)C4)=O)C2)ccc(F)c(O)c1 C1(N(C)C(=O)NC2CCC(=O)N2)CC2CC1N(C(=O)OC(C)(C)C)C2 N1(C(c2cnc(CNC(C=C(C)C(C)C)=O)nc2)=O)CCn2ncc(C)c2C1 C1(CC)CCCCC1C(N1CCCC1CC1CCOC1)C(=O)NCC1CC1 c1(C(=O)OC)ccc(Cn2cc(CN3CCCCCC3)nn2)cc1 C1(CC(=O)NCc2ncc(C)[nH]2)CN(C(c2cc(C3CC3)[nH]n2)=O)CC12CC2 C1(NC(C2(CC)CCCC2)=O)CN(C(=O)CCCCC#N)C2CCCCC12 N1(C(c2cccc(-n3cccn3)n2)=O)CC2CCC1CN2C(C1CSC1)=O CC1OC2(COC)CC1(C(=O)NC(C)(C)CNC(=O)C=C1CCN(C)CC1)C2 C(=O)(C(C(C)C)C(C)C)N1CCC(C(C)NC(CCc2cc(C)nn2C)=O)CC1 N1(C(c2cc(OC)n[nH]2)=O)CCCC(NC(=O)CCC(=O)NC2CCCC2)C1C c1(C(=O)NC2C(CN(C)C(C3(F)CCCOC3)=O)CCC2)cccnc1O c1(C(=O)NCC(COCC)O)cc(Br)c(C)cc1Nc1ccccc1OC C1(NC(C(C)NS(CCC)(=O)=O)=O)CN(C(C2(C#N)CC2)=O)CC(F)(F)C1 C1(CNC(C(C)OCC)=O)CCCC2(CN(C(=O)CCc3cncs3)C2)O1 C1(CNC(=O)C(O)C(F)F)CN(C(=O)C=C(Cl)Cl)CCC12CCOCC2 C1(C(=O)OC)CN(CC2CC3CCC2N(C(=O)OC(C)(C)C)C3)CCC1(F)F C=C1CC(C(=O)NCc2cscn2)(CNC(c2cnn(C(C)C)c2)=O)C1 c1(C(=O)NCC(CN(C(C(C)N(C(C)=O)C)=O)C)C)cnn(CC(F)F)c1C S(=O)(=O)(c1cc(C(=O)NCC2CCN2C(C2(C)CC=CC2)=O)ccc1OC)NC Cc1cnc2c(C(N3CCN(C(c4cc(Cl)on4)=O)CC(C)(F)C3)=O)cnn2c1 Cc1nc2cc(C(N3CCN(C(=O)CC(C)(F)F)C(CC(F)F)C3)=O)cnc2[nH]1 CC1(C)C2CCC1(C(=O)O)C(NC(c1c[nH]nc1Cl)=O)C2 c1(C(c2nc(C(C)(CN=[N+]=[N-])OCCN3CCN3)on2)C)ccc2ccccc2c1 CC1CCOC(C(=O)NCC=CC(=O)NC2(c3nc[nH]n3)CC2)C1 C1(NC(Cc2ccc(C)c(F)c2)=O)CC12CCN(C(C1CC=CC(O)C1)=O)CC2 CC(C(=O)NCCC1CN(C(c2cccc(CS(C)(=O)=O)c2)=O)C1)C(C)O c1(CN(C(C(COCC)n2cc(C3(C)CCCCC3)nn2)=O)C)ccc(F)cc1 Cc1ncccc1CC(=O)N(C)CC1CCCN1C(=O)C(C)c1cccs1 C1(NC(=O)C(F)F)CN(C(=O)CCc2ccc(Br)cc2)C2(CCOC2)C1 C=CC1(CC(=O)NCC(C)(CC)OC)CN(C(=O)CC2CCCO2)C1 O=C(C1=NOC2(CCN(Cc3cccc(I)c3O)C2)C1)N1CCC(C2CC2)C1 n1(CC)nnc(C)c1CNC(=O)C(c1ccoc1)NC(=O)CCc1nc[nH]n1 Cc1noc(C)c1S(=O)(=O)NC1CC2CN(Cc3cc(F)cc(Cl)c3)CC2C1 C(=O)(C#CC1(CC)COC1)N1CCC(NC(c2c(Cl)cn(CCC)n2)=O)C1 c1(C(N2CC(NC(C=CC(=O)OCC)=O)C3C(C2)C3)=O)csc(S(N)(=O)=O)c1 Cc1csc(C(N2CCC(OCCNC(=O)C(=O)N(C)C)CC2)=O)c1Cl Fc1c(Br)cc(OCCCn2cc(-c3cc(F)c(F)c(F)c3)nn2)cc1I N1(C(C(F)OC)=O)CC2(C1)CN(C(c1c[nH]nc1Br)=O)CC2CO Cc1ccc(CCC(=O)NC2CCC2NC(=O)CSC2CC2)o1 C1(N(C2CCOCC2)C(C(=O)Nc2ccccc2F)=O)COC2(CCNCC2)C1 c1(C(=O)NCCCNC(CSc2n(C)cnn2)=O)cccc(CSCC#N)c1 N1(C(c2c(OCC)ccc(C)n2)=O)CCC2CC2(NC(=O)Cn2cccn2)CC1 C1(CNC(c2ncn(C(C)C)c2)=O)CCN(C(C2(C)CNC(=O)C2)=O)CC1C C1(CC)(NC(=O)C(C)S(N)(=O)=O)CCN(C(=O)CCc2nc(C)cs2)CC1 c1(OC)ccc(CCC(N2CCOC(C(C)NC(=O)COCCCF)C2)=O)cc1 c1(C(=O)NCCC(C(=O)N(CC(O)CO)C)OC)ccc(O)c(F)c1 C(C(C)C)(C(C(=O)Nc1cccc(Cl)c1C)N1CCC(COC)CC1)OC c1(-c2scc(C(C)NC(=O)NC3CCC(C4CCNCC4)N3)n2)ccc(Cl)cc1 CCCCC(C(=O)N1CCC1C(C)O)NC(c1cccc(F)c1O)=O C(=O)(C(C)(O)CCC)N(C1CCN(C(C(C(=O)OCC)F)=O)CC1)C Cc1c(C(N2CCC(C)(NC(=O)CC(O)C(C)C)CC2)=O)sc2cncn12 C(C1CCOCC1)=CC(=O)NCCC(=O)NOCCCF c1(C(F)(F)CNC(=NCC2CCCO2)NCc2ccc(Cl)o2)cccc(F)c1 CN1CCN(C(=O)CCC2CC3CCC2C3)C(CNC(=O)CC(C)(C)C#N)C1 C(=O)(C(O)C(C)CC)NC(C1CCN(C(c2c(OCC)nccc2)=O)CC1)(C)C Cn1cncc1CC(=O)N(CCCNC(=O)Cc1nc[nH]n1)CC1CCCC1 c1(OCC)cnccc1CNC(C(CO)C(C)C)=O.c1(C)ccccc1 CC1(CNC(C2SC3C=CC2CC3)=O)CCN(C(C2CCOCC2)=O)CC1 Nc1c(F)ccc(Cl)c1C(N1CCC(CNC(=O)Cc2cnccc2Cl)CC1)=O CCCC(C(=O)NCC1(Cn2cc(-c3ccc(C)s3)nn2)CC12CCC2)N(C)C c1(CC)cccnc1C(N1CCCC1C(C)NC(C1(N2CCOCC2)CC1)=O)=O C1(C(=O)NCC(CC)(C)CC)CN(C(c2ccc(C)c(C)c2)=O)C(C)(C)C1 N1(C(c2c(C)cccc2Br)=O)CCN(C(C2CC(C)C2)=O)C2(CCC2)C1 C1(CC)(NC(c2ncccc2N)=O)CCN(C(c2cnsc2C)=O)CC1 c1(C(=O)NC2(C)CCN(C(=O)COCC3CCCO3)CC2)ccc([N+](=O)[O-])cn1 CC1CC(NC(=O)C=Cc2ccsc2)CN1C(c1cnn(C(C)(C)C)c1N)=O c1(N(N2CC3CC3C2C#N)C)cc2ncc(-c3cnn(CS(C)(=O)=O)c3)cc2[nH]1 C1(NC(Cc2n(C)ccc2)=O)CCC2(CCN(C(C3(C)C=CCCC3)=O)C2)C1 c1(OC)nc(Cl)ccc1S(=O)(=O)Nc1cnc2ccnn2c1 c1(-c2ccc(C(N(CCCN(C(C)=O)C)C)=O)s2)ccc(Br)c(C)c1 C=CC1(C(N2CCC2(C)C(=O)NC2CCC(C)(C)CC2)=O)CCOCC1 C(=O)(C(C)(C)N(C)C)NCC1(NC(CSCC=C)=O)CC1 C(=O)(C(C)CC(N)=O)N1C(C(C)NC(c2c(C)oc(-c3cccs3)n2)=O)CCC1 CC1CCOC1C(=O)NCC1CC(C(N2CC(O)(c3nn[nH]n3)C2)=O)C1 c1(-c2cccc(OC)c2C)cccc2c(C(=O)NCc3noc(CO)n3)n[nH]c12 C(=O)(C1=CS(=O)(=O)CCC1)N1CCN(C(CSC(C)C)=O)C(CO)C1 C#Cc1cccc(CC(=O)N(C(CC)CC(=O)NC(C)C(=O)NC(C)C)C)c1 c1(OCC#C)c(Cl)cc(CNS(=O)(=O)CCC(C)(C)C)cc1Cl c1(C(C)C)ccc(C(=O)NC(CNC(c2n[nH]cc2C2CC2)=O)C2CC2)c(F)c1 c1(C(N2CCC(N(C(CN(CCC#C)C)=O)CC)C2)=O)cccc2c1CCC2 N1(C(Cc2n(C)nnc2)=O)CCC(C)(C)CC1C(N1CC(CC(N)=O)C1)=O CC(C)(O)C(F)C(=O)NC1CC2CN(C(=O)CCOc3ccc(F)c(F)c3)CC12 C(=O)(C(C)CC#N)N(C(C)C(N1CCCC1CN=[N+]=[N-])=O)CC C#Cc1cc(C(=O)NC(C)(CNC(c2cc(CCOC)on2)=O)CC)cc(F)c1 C1(NC(Cc2ccc(CC)cc2)=O)CCCCN(C(C2CCCN(CC)C2)=O)C1 N1(C(C(CCOC)OC)=O)CCC2(CC1)COC(CNC(=O)CP(C)(C)=O)C2 Cc1nc(C2CCCC2)sc1C(=O)NC(C)CNC(=O)CCCN1CCCCC1 c1(C(N2CC(CCCNC(C=CC)=O)OCC2)=O)ccc2oc(C)nc2c1 c1(C(=O)NC(c2ccncc2Cl)C)ncccc1N1CCOCC1 C1(N(C(CCCOCCC)=O)CC)CCCN(C(=O)CC2CCCC2C)CC1 C1(NC(c2c(C)snc2)=O)CCC2(CC1)CN(C(c1ccc(CO)cc1)=O)C2 N1(C(c2cccc(I)c2)C(=O)NCCOCC)CC(C)(C)OCC1CC CC(C)CC(C)CNC1(CO)CCCOC1 C[Si](C)(C)c1ccc(-c2cnc(Nc3cccc(N4CC4)c3)s2)cc1 C1(C(C)NC(c2cc(CN(CCC)C)on2)=O)CN(C(=O)C=C(C)C)CCO1 C1(O)(C(C)NC(c2c(CC)ocn2)=O)CCN(C(=O)C=Cc2cncs2)CC1 C(C(C)(C(=O)NC1C=CCN(C(=O)Cn2cc(Br)c(C)n2)C1)OC)OC C(CNC(C1CC(=O)N(C)C1)=O)(CC(F)(F)F)NC(c1cc(OC)ncn1)=O c1(C(=O)NCC2(F)CCN(C(=O)Cn3cc(CO)nn3)C2)cc2ccccn2c1 c1(OCC)oc(C)nc1C(=O)NCC(C)(CC)NC(c1ccon1)=O c1(OC)cc(C)c(C(c2nnnn2C(C)(C)C)NCc2conc2C2CC2)cn1 N1(C(CC2C(C)C2)C(=O)NCc2ccco2)CC2(C3CC3)CC1CCO2 C(=O)(C1CCOc2ccccc21)NCC1(F)CC(NC(c2cc(C)c(C)s2)=O)C1 c1(OC)cncn(CC(C)NC(c2cccc(Br)c2)=O)c1=O C(=O)(CC(O)(C(F)(F)F)c1ccccc1)OC.C1(C(=O)OC)SCC(C(F)(F)F)N1CC Cc1ccc2c(C(=O)NCC=CCNC(=O)C(C3CCOCC3)O)n[nH]c2c1 N(C1c2ccccc2CCC1C)C(=O)Nc1c(C)n(C(C)C(C)(C)O)nc1 C1(C)(NC(c2nccc(C)n2)=O)CCCN(C(=O)C2=CSCCO2)C1 Cn1nc2ccccc2c1Cn1cc(-c2ccc(Cl)c(N)c2)nn1 CCC(C)(C)C(C(=O)N1CCCC(CNC(=O)Cc2ccc(F)c(C)c2)C1)OC C(CC(=O)NCCC(=O)NCCC1(C(=O)NC)CC1)SCCC c1(CC(=O)N(CC(C)NC(C2COCCC2C(F)F)=O)C)c(F)cncc1Cl C1(C)(C(c2n(CCCCCC)nnn2)NCCCn2cnnn2)CC=CCO1 CCC(CC(=O)N1CC(C)(C)CC1CNC(C1(C)CC1)=O)C(C)(C)C C1(C(=O)OC)CCC(C)(C)N(C(=O)CCc2cn(C(C)CO)nn2)C1 O=C(C1=CCCN(C(C2CC3CC(=O)C2O3)=O)C1)NCCN1CC2CC2C1 N1(C(CC(CCC)O)=O)CC(NC(c2c(Cl)nn(C)c2Cl)=O)CC2(CC2)C1 Cc1ncc(C(=O)NC23CC(CNC(=O)CC4CC4C)(C2)C3)cn1 c1(CNC(=O)C(=O)NCc2ccon2)ccc(C2CCOCC2)cc1 CN1CCC(CN(C(=O)C(CC2CCOCC2)NC(=O)CCC2CCOC2)C)C1 c1(C(=O)NC(COC)CC(=O)NCc2cnnn2C)ccc(F)nc1F C(=O)(C1=NN(c2ccc(C)cc2C)C(=O)C1)NCC1C2CN(C(CC)=O)C1C2 c1(C(c2nnnn2C)NCc2occ(C)c2)cccc(C(C)C)c1 N1(CCC)CCN(C(=O)CCC2CCCN(C(C3CCCS3)=O)C2)CC1 c1(C(=O)NC(CN(C(C(C)=CC)=O)CC)C)c[nH]c2cc([N+](=O)[O-])ccc12 c12ccc3c(c1)CN(C3)C2=O.C1(N(C(C)(C)C)C)CCN(Cc2cccnc2)C1 C1(=O)C(CCC2CCCC2)N1C1C=CCC1.C(C)(C)(C)OCCSC.C(=O)O c1(COC(C)C)cn(C(C)C(=O)NC2CC(CCl)C2)nn1 c1(CN2CCCC(O)(CCO)C2)ncnc2c1ncn2-c1ccc(F)cc1F N12CC(C(C)(C)C1)C2=O.c1(CC)ccc(C(=O)N(CC(C)C)C)cn1 C1(N(C(CCCCC)=O)C)CCN(C(=O)C(c2ccc(C)o2)C)CC12CC2 N1(C(c2cnc(O)c(F)c2)=O)CC(NC(C2CC(F)C2)=O)CC2(CC2)C1 C(=O)(CS(=O)CCC(F)(F)F)NC1(C2CCN(C(c3ccn(CC)n3)=O)C2)CC1 N1(C(c2c(SC)nn(C)c2)=O)C(CNC(C2CC2[N+](=O)[O-])=O)CC2CCCC12 N1(C(C(CSC)C)=O)CC(=O)CC1C(=O)NCC1(C)CCOCC1 C#CCCCCCC(=O)N1CCCCC1C(C)NC(c1c(C)ncn(C)c1=O)=O C(=O)(C(F)(F)C(O)C(C)C)NC1C=CCN(C(c2ccc(S(=O)(=O)NC)o2)=O)C1 Cc1c[nH]nc1C(=O)NCC1CCC1C(=O)NC1(CO)CCSC1 CCC(CC1CCCC1)C(=O)NC(C)CCN(C)C(C1CSCN1C(=O)NC)=O c1(CCN=C(NC2C(C)(C)SC2)NCCF)ccc2occc2c1 c1(OC)cccc(C(C)(C)C(=O)N2CCC(NC(c3csc(CSC)n3)=O)C2)c1 c1(C(=O)OC)ccc(C(=O)OC)c(NC(N2CCOC3(CCSC3)C2)=O)c1Cl CC1(O)CCCCC1NC(C1CC(=O)CN1C(C1(Cl)CC1)=O)=O c1(C(N2C(C)CN(C(=O)CN3CCC(C)(O)C3)CC2)=O)cnc2c(c1)CCCO2 C1(NC(CSCC=C)=O)CC1C1CCN(C(=O)C(c2cc(F)cc(F)c2)C)CC1 N1(C(CCc2c(C)noc2)=O)CCCCC(CCC(=O)NCCCCN=[N+]=[N-])C1 Cn1ncc2nc(Cl)nc(NC(CNC(c3ccc4nc[nH]c4c3F)=O)CO)c12 N1(C(C2(CC=C)CC2)=O)CCCCC(C(N2CCCC(OCC)C2)=O)C1 C(=O)(C1=COCCC1)N1C(CN(C(=O)C=Cc2ccccn2)C)COCC1 C(=O)(C(C(C)NC(=O)Cn1cc(CN2CC3CCC2C3)nn1)C(C)C)OC N1(C(C2CCCC(NC(c3cccc(CO)c3)=O)C2)=O)CCn2ccnc21 c1(C(=O)O)ccc(C(N2CC(C(=O)O)CCC2C(=O)O)=O)c(Cl)c1 C1(NC(C2C(C)CCC2)=O)CCCOC12CCN(c1cnc(C#N)cn1)CC2 N1(C(C(C)OCCC=C)=O)C(C(=O)NOCCn2cc(CO)nn2)CC1C c1(C(=O)NCC(C)N(C)C(C2CCC(C(N)=O)O2)=O)cccc(S(=O)(=O)CF)c1 c1(C(=O)NC(CC)CNC(=O)CCc2ccc(OC)cc2)ncc2n1CCCC2 CC1(Cn2cc(CS(=O)(=O)CCNC(=O)C(F)(F)F)nn2)COC(=O)OC1 N1(C(CC(C=C)(C)C)=O)CCOC2(CCCN(C(=O)C3=C(CC)OCCC3)C2)C1 C=C1CC2(C1)CC(C(N1CC(N(C)C(c3cc(Cl)cc(Cl)c3)=O)C3(CC3)C1)=O)C2 C#Cc1cc(C(=O)NC(C)(C)C(C)NC(=O)Cc2ccc(Cl)cc2C)cc(F)c1 C1(CNC(C2CCOCC2)=O)CN(C(C2CC(=O)N(O)C2)=O)CC1(F)F C1(C)(C(N2CCCC(N(C(COCCCC#C)=O)CC)C2)=O)CCCCC1(F)F c1(CC(N2C(CNC(=O)CCC3CCOC3)C=CC2)=O)ccc2c[nH]nc2c1 C1(C(N(c2cccnc2)C(c2cn(C3CC3)nn2)=O)=O)CCCCO1 N1(C(C(C(CNC(CCC(C)(C)OC)=O)C)F)=O)CCOC2(CCC2)CC1 N1(C(C2CC2c2ccc3ccccc3c2)=O)CCCc2c(F)ccc(Br)c21 Cc1ccc(C(=O)NC2CC(CNC(=O)C(C)C3CCC3)C2)c([N+](=O)[O-])c1 c1(NC(C2N(C)C(NC(=O)OC(C)(C)C)CC2)=O)cc2oc(O)nc2cc1F C(N=c1[nH]c2c(c(=NC3CC(C(N)=O)C3)[nH]1)SCC2)c1nc(CC)[nH]n1 N1(C(CCNC(C(C2CCC(=O)N2)C)=O)=O)CCC12CCCC2 c1(C(C)=O)cnc2n1CCN(C(c1ccn(CC3CC3)c1C)=O)C2 N1(C(C(C)OC(=O)OCC)=O)CCC2(CC2NC(c2cccnc2C2CC2)=O)C1 c1(C(N2CC(C)C(CNC(c3ccncc3F)=O)CC2)=O)ncc([N+](=O)[O-])n1C Cc1cc(C(N2CCC(C(c3ccccc3F)F)CC2)=O)c(N)s1 c1(C(=O)NC(CN(C(c2cc(C)c(C(=O)OC)o2)=O)CC)C)cc(Cl)c(C)cn1 N1(C(C(C)(C2CCC2)NC(c2ccc(CC)nc2)=O)=O)CCOC2(CCC2)C1 c1(C(=O)NC2C(NC(CC(C(=O)OC)(C)C)=O)CC2)nccc2ncccc12 N1(C(c2ccc(CC)[nH]2)=O)CCC(O)(C(C)NC(=O)Cn2ccnn2)C1 c1(CC(C)C(=O)NCC(F)CNC(=O)C2=CCSC2)ccccc1Br c1(C(=O)NCC2N(C(c3cc(SC)oc3)=O)CC2)c(C)cc(=O)oc1C c1(C(=O)NCC(CC)NC(c2c(CC)nns2)=O)ccc2nc(O)cn2c1 C1(CNC(c2n[nH]c(CC)c2Cl)=O)CCN(C(C2CCCC2(C)C)=O)C12CC2 Cc1coc(C)c1C=CC(=O)NC1CC1NC(=O)Cn1cnc([N+](=O)[O-])c1 C12CCC3(CCN(C3)CC(=O)O1)C2.c1(COCCOCCN(C(C)C)C)ccccc1 N1(C(Cn2c(C)cc(CO)n2)=O)CCCC2(C1)CN(c1cncc(Cl)n1)CCO2 Cc1coc(C(N2CCCC2CCNC(=O)CCc2c(C)noc2Cl)=O)c1C c1(C(N2CCC3(C(C(=O)NC(C)CO)C3)C2)=O)cc2cc(F)ccc2s1 N1(C(C(=O)N(CC)CC)=O)CC(NC(=O)C(F)(F)CCn2cccn2)C(C)(C)C1 C(=O)(CS(=O)(=O)CC(C)C)NCC1N(C(C2C(OCC)C2C)=O)CCC1C N1(C(C2C(C)C2)=O)CC2CC(C1)N(C(c1ccc(C3CCCC(=O)N3)cc1)=O)C2 CN=c1nc(C(=O)NC2CC(CNC(=O)C(C)(C)CCF)C23CCC3)cc(C)[nH]1 N1(C(C(Cc2ccco2)NC(c2c(C)c(O)ccc2)=O)=O)CCC(F)(F)C(O)C1 c1(CCC(=O)O)ccc(CNC2CCCCC2n2ccnc2)nc1 C1(CNC(C2CCCC2O)=O)CC2CCC(C1)N2C(c1cc(CF)on1)=O c1(C(=O)NC(CNC(Cn2cc(C(=O)NC)nn2)=O)(C)C)cc(C)c(C)s1 c1(C(C(=O)NC2CC(N(C)C(c3cc4occc4s3)=O)C2)=O)ccc(F)c(F)c1F N1(C(CCCOCCOC)=O)CC(C(N2CC3CCC3(C)C2)=O)CC(C)C1 N1(C(CC(C)n2cccc2)=O)CC(=O)NCC1C(=O)NOCC(O)C(C)(C)C C1(C(=O)NCC(=C)CCNC(c2ccc(SC(F)F)cc2)=O)CCC(C)(C)CC1 C(CC1=CCN(C(C2CCN(C)C(=O)C2)=O)CC1)NC(C1(CC)CCNC1=O)=O N1(C(CN(CCC)C)=O)CCC(F)(CNC(c2ncccc2OC)=O)CC1 c1(C(N2CC(CN(C(c3c(C)c[nH]n3)=O)C)OCC2)=O)cc(C)c(C#N)c(C)c1 C(C)(CCC(C)C)NC(C1(NC(C=CC(CC)C)=O)CC1)=O C1(CN(C(c2c(C)onc2)=O)C)CCCN(C(c2cccnc2C(F)F)=O)C1 C1(CNC(C(C=CCCC)O)=O)CCCN(C(=O)C=Cc2cncn2C)C1 N1(C(C(=O)NC2COC2)CCc2ccccc2F)CCC2(CCCOC2)C1 N1(C(Cc2cccc(C)n2)=O)CCC2(CC1)CCN2C(C1C=CCN1)=O Cc1cnn(C)c1C(=O)NC(C)(C)CCCNC(C1CCN(C2CC2)CC1)=O C1(NC(c2c(C)cc(C(F)(F)F)nc2)=O)CCc2n[nH]cc2C1C N1(C(C2C=C(C)CS2)=O)CC2OCC(NC(c3cccc(F)c3)=O)C2C1 CC1C(C(=O)N2CCC3(CCCN3C(=O)C#CC3(C)CC3)C2)=Cc2ccccc21 N1(C(C(C)Cn2ccnc2)=O)CCCC2(CCCN2C(=O)CC2CCSCC2)C1 CC(=O)CC(C)(C)CC(=O)NCC1CC(NC(c2cnoc2)=O)C1 c1(C(N(C2CCCC2)CCNC(C=CCC)=O)=O)oc2ccc(Cl)cc2c1C N1(C(=O)OC(C)(C)C)CC2CC(C1)N2C(=O)CC.C12CCCCC1C(CO)N2 O=C(CC(F)(F)C(F)F)NC1CCCCCN(C(=O)CC2CCOCC2)C1 c1(C(=O)NCC(O)C(=O)N2CCC2CC2CCCC2)ncn2c1CCC2 CC(C)(CCC#N)C(=O)NC1CC1NC(c1ccc(C2CCCC2)cc1)=O c1(C(=O)NC(CC)CN(C)C(C2(OC)CCC2)=O)cnc(OC)c(Cl)c1 CON(C)C1CN(C(c2nc(CNC(=O)Cc3ccccn3)oc2C)=O)C1 c1(C(N2CCC(CNC(c3cnoc3-c3ccco3)=O)C2)=O)csc2cncn12 C1(CNC(C=CCC)=O)CCN(C(=O)CCc2cncn2C)C12CC2 C1(NC(c2sccc2C2CC2)=O)CN(C(=O)CN2CCOCC2)C2CCCCC12 c1(C(=O)NCC2C(CNC(c3cn(C(C)C)nn3)=O)C2)ccc(O)c(C(N)=O)c1 N1(C(CC(C)(C)NC(C2CC3CC2CC3O)=O)=O)CCC2(CCCCO2)C1 CC(C)CC(C)CC(=O)NC1(C(=O)NC2CC3CCCC3C2)CCCC1 CC1(C)CNCCCN1C(=O)NC1CCN(Cc2ccsc2)CC1 C1(CC)CCN(C(=O)CC2CC(CN(C)C(C3(C)CC3)=O)C2)C1(C)C C1(CCC)CN(C(=O)CCN2CCC2)CC1C(=O)Nc1csc(Cl)c1 CCCC(C(=O)NCc1c[nH]nc1C(=O)NC1CNC(=O)C1)OCC C1(CN(C(C(C)NC(C)(C)C)=O)C)CCN(C(=O)CCN2C(=O)CCC2=O)CC1 N1(C(C(C)(C)OC)=O)CCCCC2(CCN(C(=O)CNC(=O)CCCCO)C2)C1 C#CCCCCCC(=O)NCC(COC)NC(C1CCN(C(=O)OC)C1)=O C1(NC(=O)Cc2ccccc2O)CN(C(c2[nH]ccc2C2CC2)=O)C2(CCC2)C1 n1(CC)nnc(-c2nc(-c3ccc(OC)cn3)nn2-c2cnnn2C)c1C Cc1cc(C(N2CCC(C)(C)C2CC(=O)NCC(C)(C)O)=O)cc(C)c1 c1(OC)ccn2cc(C(=O)NCCCN(C(c3csc(C)c3)=O)C(C)C)nc2c1 c1(C(=O)NC2CN(C(c3c(COC)cco3)=O)C2)ccc(C(C)(C)OC)cc1 CC1(C#N)CCCN(C(=O)C(=O)NCc2ccc3c(c2)OCC3)C1 c1(N(C(=O)CCC(=O)N2CCOCC2)Cc2nccc(OC)n2)cc(C)ccc1Br N1(C(CC2CCCC(C)O2)=O)CC2(CCN(C(=O)CN(S(C)(=O)=O)C)CC2)C1 C(=O)(C(C(C)C)NC(c1ncc(F)cn1)=O)NC(C(=O)NCC)C C=CCC(C)(CC=C)NC(=O)C1=CCC(NC(=O)CCn2cccc2)C1 CC(C)C(CCN(C)C(c1cn(C)nc1Cl)=O)NC(=O)C(C)n1cccn1 N1(C(C(CC)N(C)CC)=O)CCOC(NCC=CCl)C1 c1(C(N2CCC(OCCNC(C3CC3[N+](=O)[O-])=O)CC2)=O)cnn2c1NCCC2 c1(C(=O)NCC(CNC(C(C=C=C)C)=O)(C)O)ccc(OC)cc1Cl C=CCCCC(=O)N1CCC1(C)CC(=O)NOC(C)(C)C C1(C(N(CC#CC)CC#C)=O)CCCCCCN1C(=O)C(C)OCC=C N1(C(c2scc(C)c2)=O)CCCCC(C(=O)NCC2OC(=O)CC2(C)C)C1 c1(C(N(CC(C)NC(=O)C(O)C2CC2)C)=O)ccc(N2CCCCCC2)cc1 C(=O)(C(C(=O)Nc1cccc(NC(C2(C)CCN(C)CC2)=O)c1)C(C)C)OCC C(CCC(C(=O)NC1CCCC1C(=O)OC)NC(=O)C(C)CC#N)OC c1(C(N2C(c3cn(CC(C)O)nn3)CCCC2)=O)ccn(CC(F)F)c(=O)c1 c1(C(=O)NCC=CCNC(Cn2c(C)cnc2)=O)cnc2c(cnn2C)c1 c1(C2C(C)CCS2)nc(-c2cccc(F)c2)nn1-c1ccnc(O)c1 CCCCCC(=O)NCCOC1CCN(C(=O)CCC2CCCN(C)C2)C1 c1(C(N(CC(C)(C)NC(=O)CCc2nccn2C)C)=O)c(F)ccc2c1OCC2 C#CCC(C)(CC)C(=O)NC1CN(C(=O)Cc2nc(C3CC3)nn2C)CC1SC n1(CC(=O)NC2C(NC(CCCCC#C)=O)CC2)c(=O)c(=O)[nH]c2ccccc12 c1(NC(C2CCN(C(C3=NOC(C)C3)=O)C2C2CC2)=O)ccc2ccncc2c1 c1(C(N2CCC(C(N)=O)C2)C(=O)NCCC(=O)OCC)cc(Cl)sc1C N1(C(c2cccc(N(C)C)n2)=O)CCCC(B2OC(C)(C)C(C)(C)O2)C1 CC1=C(C)C(NCCCN2CCC(C(F)(F)F)CC2)CCC1 c1(SC)cc(NC(=O)COC2CCN(C(=O)OC(C)(C)C)C2)cc(Cl)c1 C1(N(C(=O)CCn2cnnn2)C)CCC(NC(c2cnc(S)[nH]2)=O)C1 C(C)(C(=O)N1CC(O)CO1)N(C(C(COC)OC)=O)C1CC1 N1(C(C)=O)CCCC(NC(=O)CC(c2cccs2)NC(=O)C=Cc2cc[nH]n2)C1 c1(CC(=O)NC(C2N(C(c3nc(SC)sc3)=O)CCC2)(C)C)cncc(C)c1 N1(CC)C(=O)CCC1C(N1CC(c2c(C(=O)OCC)nco2)(NC(=O)NC)C1)=O O=C(C(Cn1cccn1)NC(=O)C1CC1)NC(c1ccncc1)CO N1(C(C2(C(C)NC(C3CCCC3)=O)CC2)=O)CC2CCC1C(O)C2O Cc1nc2ccc3nc(NC(C4CC5C=CC4CC5)=O)sc3c2s1 c1(OCC(N2CCC(N(CC)CC)C2)=O)cc(F)ccc1C(N)=O c1(NC(C2(CC#C)CCCO2)=O)cccn(-c2ccccc2)c1=O Cc1nc(C(=O)NCC2CC2CNC(c2nc(=N)cc[nH]2)=O)c(C)o1 c1(C(=O)NC(C2CCN(C(=O)C(Cl)=CCl)C2)(C)C)cnc2ncccc2c1 CCCCC(C(=O)N1CCC(NC(c2ccc(C(C)=O)cc2)=O)C1)N(C)C N(C1=NCc2ccc(cc2)C(=O)N1)C1C(C)(C)C1.c1(NC2CC2)ccncc1 C1(CNC(C2CCN(CCCC)C2)=O)(CNC(=O)C(C)(C)SCC)CC12CCC2 c1(C(N(CCCN(C(C(C(C)C)O)=O)C)C)=O)cc(C(F)(F)F)cnc1N Cn1cc(C(N2CC3CC3(C3CC3)C2)=O)c(C(F)F)n1.C1(C(=O)NC)CCCO1 N#CC1(C(=O)NC2CC(NC(=O)CC3CC=CC3)C23CCC3)CC2CCC1CC2 c1(N(C)C)ccc(CNC(c2ccccc2C(N2CC(N)C2)=O)=O)c(F)c1 N1(C(c2c(C)cccc2)=O)CC(NC(c2ocnc2C)=O)C2CCCC12 c1(C(=O)NC2CC(C)CN(C(=O)COC(F)F)C2)cc(Br)cn2ccnc12 C(=O)(CCCC(=O)C(C)OC(c1ccc(CC(F)F)cc1)=O)OC c1(SCC)ccc(C(=O)NC(C)C(C)NC(c2cn(CC3CCOC3)nn2)=O)cc1 c1(CC)nc(C)c(CC(N2CCCC(C)C2CNC(C2(CC)CC2)=O)=O)c(C)n1 c1(C(N2CCCC(O)C2O)=O)cc(F)ccc1OC(F)(F)F CC1(C)CCCC(CN2CC(c3nc(C(F)(F)F)no3)C2)CC1 C1(C(=O)NCC2CCN(C(=O)Cn3cnc(Br)c3)C2)CCCS(=O)(=O)C1 c1(C(=O)NCC2(NC(C=CCC)=O)CC2)cccn2ncnc12 c1(SCC)ccccc1CCNC(=O)Cn1cc(CC2CCCC(CO)C2)nn1 c1(C(=O)NCC2(NC(c3nc(CCC)sc3)=O)CCC2)nc(OC)ccc1Cl C#Cc1ccc(F)c(C(=O)NCC2CC2NC(C2(Cl)CC2(C)C)=O)c1 c1(C(N2CC(CNC(c3c(C)noc3C)=O)N(C)CC2)=O)cc(F)c(F)cc1O C1(CNC(c2ccn(CC)n2)=O)CC2COCC2N1C(=O)CSc1nncs1 C1(COC)CCOCCN1C(C1CCCN(CCOc2ccc(Cl)cc2)C1)=O C1(NC(C2(CCC=C)CC2)=O)CC(C(N2CC=CC(O)C2)=O)C12CCC2 CC1C(NC(=O)Cc2cc(Cl)ccc2Cl)CCCN1C(=O)Cn1cccnc1=O Cc1ccc2c(c1)CCC2Nc1conc1C1CCNCC1 C1(CNC(C(C(COC)C)C)=O)C(C2CC2)CCN1C(=O)C(CCOC)OC C(=O)(N=S(C)(=O)C1CCNCC1)C1(NCc2ccccc2)C(C)(C)NC1 C1(C(=O)NC2C(CCOC)C2)CCN(C(=O)Cn2cncn2)C1C C(C(=O)NC1CC(CCNC(=O)C=Cc2ccccc2)C1)(C(C)C)OCC CCS(=O)(=O)C=CC(=O)N1CCC(C)C(NC(c2ccon2)=O)C1 c1(-n2ncc(C(N(C3CCC(NC(C)=O)C3)C)=O)n2)ccc(F)cc1 N1(C(C23OCC(C)(C2)C3)=O)CCCC(CCNC(=O)CCCCCN(C)C)CC1 c1(OC)cc(C(C(=O)NCCC2CC2)N(CCC(=O)NC(C)C)C)ccc1C c1(C(N2CCCC2CCC(N2CCCC2CO)=O)=O)ccoc1-c1ccccc1 CC(=NO)C1CC(C(=O)NCC2(NC(=O)CCCCO)CCC2)C1(C)C S(=O)(=O)(c1ccnc(NC(c2ccc3c(c2)CN(C(C)=O)C3)=O)c1)NC N1(C(C=CC(C)C)=O)CC2C(C(=O)NCCn3cc(-c4ccccc4)nn3)C2C1 C1(NC(c2cc(C)ncn2)=O)CCSC12CN(C(c1cccnc1C1CC1)=O)C2 C1(CCC)(NC(C)=O)CCCN(C(c2cnn(C3CCOCC3)c2)=O)C1 N1(C(CC2CCN(C(c3cc(=N)[nH][nH]3)=O)CC2)=O)CCC(O)C12CCCC2 C(C(C)C(=O)N1CCC2CC12)NC(COCC#C)=O N1(C(C2CC(C)(O)C2)=O)CCN(C(=O)Cn2cccc(N)c2=O)C2CCCCC12 N1(C(C=CC(=O)OCC)=O)CCC(C)(CNC(C2CC(CN(C)C)C2)=O)C1 c1(CC)nc(C)c(C(=O)N)s1.C1(C(N2CC(C(N)=O)(C)C2)=O)C2CC3C(C2)C13 c1(C(=O)NC2CC(NC(C3(Cl)C(C)(C)C3)=O)C2)cc([N+](=O)[O-])cc(Cl)c1Cl c1(CNC(C2(C)CN(Cc3cccnc3-n3cncn3)C2)=O)cccnc1Cl N1(C(C2CCN(C)CC2)=O)CCCCC2(CCN(C(C3CC4CC34)=O)C2)C1 c1(-n2c(C(CCCc3ncoc3CN)=O)cnn2)c(Cl)cccc1Cl.N C(=O)(CCN=c1ccc(C)c[nH]1)N1CCN(C(C(CC)(C)CO)=O)CC1 CCC(C)CC(=O)NC(CC)C(=O)N(C1CCNC1=O)C c1(SC)ccc(C=CC(=O)N(CCCNC(C2C(C)C2(F)F)=O)C(C)C)cc1 C(C1CCCCC1)=CC(=O)NC1(C(=O)NCC(COC)OC)CC(CO)C1 N1(C(c2cncc(OC)c2)=O)CC2CC(NC(c3c(C)nn(C)c3Cl)=O)CC1C2 C1(CCOC)(NC(=O)CC(C)O)CCN(C(=O)CCSc2ccccc2)CC1 C=CC(C)CC(=O)NC(C(=O)NCCC(C)(C)F)C1(O)CCC1 c1(C(=O)NCC(C)NC(Cc2cc(OC)ncc2)=O)cc(C)c(Br)cn1 N1(C(COC(C)C)=O)CCN(CCCCCNC(c2scnc2C2CC2)=O)CC1 N1(C(c2c(C)c(Br)no2)=O)CC(C)(C)CC1CNC(=O)C(C)CO c1(C(=O)NC2C(CNC(=O)CSc3ccc(Cl)s3)C2)csc2cnccc12 CC1(C(=O)NC2CC(NC(=O)CCC3(c4ccccc4)CC3)C2)CCCO1 N1(C(C(OC)OC)=O)CCC2(CCC2CNC(c2ccc(C(C)C)cn2)=O)CC1 C1(NC(C2(COC)CC=CC2)=O)COC2C(NC(=O)C(C)(C)OC(C)=O)COC12 c1(C(C)C)ccsc1C(N1CCC(c2cn(CCNS(C)(=O)=O)nn2)C1)=O C12(CNCCOc3c(OC)cccc3)CC3CC(CC(C3)C1N)C2 C12(NC(C3CN(C)C(=O)C3)=O)CCC(C(=O)NOCc3cccnc3)(CC1)C2 N1(CC)CCN(C(=O)C(C)N(C(c2cn3c(n2)CCC3)=O)CC)CC1C N1(C(C2C(OC)CCC2)=O)CCOC2(CCCN(C(=O)CNS(N)(=O)=O)C2)C1 c1(N2C(C)CC(NC(=O)CCCn3ccccc3=O)C2)ncnc2sccc12 c1(OCc2c(OC)ccc(C#N)c2)cccc2c1S(=O)(=O)CC2 N1(C(c2cc(C(=O)OC)oc2)=O)CCC2(CC1)CN(C(=O)C=CCO)CC(C)O2 Cc1cccnc1CNC(=O)CN(C(c1c[nH]c(C)c1)=O)CC1CC1 CC(CC(F)(F)F)C(=O)NCC(C)N(C)C(C1CC2(CCCC2)C1)=O CC1CCCC=C1C(=O)N(CCCNC(=O)CCc1ncc(F)cn1)CCO CS(=O)(=O)c1cncc(-c2ccc(C(=O)N(CC(F)(F)F)CCN)nc2C)c1 c1(OC)ccc(C)c(C(=O)NCCC23CCC(C2)N(C(C2(OC)CCC2)=O)C3)c1 c1(C(N(CCC(C)NC(C(C(C)C)SCC)=O)C)=O)cc2cc(C)ccc2o1 C1(C(=O)NCC(F)Br)CC(O)CCN1C(C1CCC2CC1CO2)=O Nc1ccc(CC(C(=O)O)NC(=O)Cn2cc(C3CCCCC3O)nn2)cc1 C1(N(C(=O)Cc2cnsc2)C)CC2CC1N(C(=O)C(c1ccccc1F)(C)F)C2 CC(C)(C(=O)NC1CCC(CNC(c2cc(-c3cnccn3)[nH]n2)=O)C1)C1CC1 N1(C(CC2(C#N)CCC2)=O)CCOC2(CCN(C(=O)CC3CC3(Cl)Cl)CC2)C1 c1(C(N2C(CCNC(C(C(C)C)O)=O)CC(F)(F)C2)=O)cccc2ccoc12 N1(CCNC(c2c(C)nco2)=O)CCCN(C(c2ccc([N+](=O)[O-])o2)=O)CC1 N1(C(=O)NCC(C)NC(C2CC=CCC2)=O)CCC(CO)CC1 c1(OC(C(=O)NC(CCCNC(C(COC)(C)C)=O)C)C)cc(C)ccc1Cl C1(C(=O)NC2CC(C)(NC(c3nc(CC)oc3C)=O)C2)CCN(CCO)C(=O)C1 N1(CCC(=O)NCC(F)(F)Cn2cc(-c3csc(C4CC4)n3)nn2)CCCCC1 N1(C(c2c(Cl)ccc(OC)n2)=O)CCCCCC(NC(=O)C(C)(C)CF)C1 C1(CN(C(CCNC(C2C(C)C2)=O)=O)C)CCCCN1C(=O)C(C1CC1)C1CC1 C1(NC(c2cc(C(C)C)[nH]n2)=O)CCC(F)(CNC(C2CC2C(F)F)=O)C1 c1(OC)cccc2c(N3CC(CC(C)NC(=O)Cc4cc(C)cs4)C3)ncnc12 N1(C(Cc2n(C)cnn2)=O)CCCCC(NC(=O)CCn2ncn(C)c2=O)C1 C(=O)(C1=CNC2=NCCC2=C1)N1C(C)C(NC(=O)CC2CC2(Cl)Cl)CCC1 CC(N=c1[nH]c(=NCc2nncs2)c2c(F)cccc2[nH]1)c1cc(Br)ccc1F N1(C(c2c(CC)ncs2)=O)Cc2n[nH]cc2C1C(=O)N1CCC(CCN(C)C)C1 C(C(C)(C)C(=O)NCCC(C)N(C(=O)Cn1cnnn1)C)OCC CC1(C)CN(C(c2cnc[nH]2)=O)CCN(C(c2ncoc2Br)=O)C1 c1(C(N2C(CNC(CC(C)F)=O)CC(O)C2)=O)ccc2cccnc2n1 c1(C(N2CC(COC)(NC(=O)C(C3CCC(=O)N3)C)C2)=O)ccc(F)cc1O c1(C(=O)NCCC(C)N(C)C(C2CCCC2(F)F)=O)ccc(-c2ncc[nH]2)nc1 C(CCN=C(NCC1=NOC2CCCCC12)N1CCCC(CSC)C1)OC N1(C(C2C3CC2N(C(c2cn(C4CC4)nn2)=O)C3)=O)CCc2ncccc2C1 C1(NC(c2c(C(C)(C)C)noc2)=O)CCCCN(C(=O)CC2COC(C)(C)C2)C1 Cn1cc(C(=O)NCC(C2CCN(C(C3C=CCCC3)=O)CC2)F)c(O)n1 N1(C(C(=O)N(C(CCC)C)C2CC2)C)CC2C(C1)C2(F)F C1(NC(c2scc(CC)c2)=O)CCN(C(c2cn(CCOC)nc2C)=O)C1(C)C c1(COC)cccc(C(N2CC=CC2C(N2CC[Si](C)(C)C2)=O)=O)c1 c1(CCC(=O)NCCC(C)N(C(=O)C2=NNC(=O)CC2)C)ccc(C#N)cc1F CC1CCC(Cl)=C(C(=O)NCC(O)CCNC(=O)COc2cccc(F)c2)C1 CCC(C(=O)OC)C(=O)NCC1CCCCN1C(c1cc(Cl)ccc1F)=O CC1C(NC(C2CCCN2C=O)=O)CC2CCC1N2C(c1ccnc(C#N)c1)=O N12CC3C(CS(=O)(=O)C3C1)C2=O.CC1CC(C)(CNC(C)(C)C)C1 c1(C(C)NC(C(=O)N(C)Cc2nnc(C(=O)OCC)s2)=O)ccc(C)cc1F c1(CC(=O)NCC(C)CNC(C2(C3CC3)CCOCC2)=O)cccc2sccc12 Cc1noc(C)c1C(C(=O)NC1COC1)N(c1ccccc1)C1CC1 Cc1ccsc1CNCC1(c2ncccn2)CCOC1 C#Cc1ccc(C(=O)NCC2CN(C(=O)Cc3ccnc(Br)c3)C2)cc1Cl c1(CN(CC)CC)ccc(-c2ccc(Nc3cccc(O)c3)nc2)cc1 c1(C(=O)NCC(CC)NC(=O)CC2CC(C)=NO2)c(C)nn(C)c1N C1(CNC(C(C)(F)F)=O)COC(C(F)(F)F)CN1C(C1CCCC1)=O c1(C(N(CCC)CCNC(C2CCN2C(C)=O)=O)=O)ccc2c(c1)CC(C)O2 N1(c2nnc(Cc3n(C)ccn3)n2CC2CCOC2)CCOC2(CCCC2)C1 c1(CN(C(C2C(C(=O)OCC)CNC2)=O)C2CC2)nc(C)cc(O)n1 c1(C(=O)NC2C(NC(C3CN(C)C(=O)N3)=O)CC2)cc(Cl)ccc1F C(CCN=C(NC1CC(C)(C)C1)NC1CCCCC1C)OC(C)C N1(C(C2(SC)CCC2)=O)CC2(CC(CNC(C3(CF)CCOCC3)=O)C2)C1 Cn1c(C(N2CCCC2CNC(C2CCCCC(=O)C2)=O)=O)cccc1=O C1(NC(C2C(C)CC(=O)N2)=O)CCC2CN(Cc3ccncc3Cl)CC2C1 C1(C(N2CCCC(CNC(CCCOC(C)=O)=O)C2)=O)Cc2nn(C)cc2C(=O)N1 Cc1cccn2ncc(C(N3CCC4C(CCN4C(=O)COC4CCC4)C3)=O)c12 c1(C(=O)OC(C2(O)CN(C(=O)OC(C)(C)C)C2)C)cc(C(C)(F)F)ccc1C C(=O)(C(COCc1ccccc1)OC)N(CCCC)CCNC(C)=O C1(c2ccccc2)(C(=O)NC(CN(C(COCC)=O)CC)C)CCOC1 C(=O)(CCCCCNC(C1(C(=O)N(C)C)CC1)=O)N1CCC(CCC)C1 N1(C(c2cn(CC)nc2C)=O)CC2CC1CN2C(=O)CCC1CCOC1 C(=O)(C(C)(C)C(F)F)N(CC(CNC(c1cc(OC)no1)=O)O)C C(CCCN=c1ccnc(N2CCOC(c3ccc(Cl)cc3)C2)[nH]1)OC C1(CNC(=O)CC2(CO)CCC2)CCCCN(C(C2C=CC=CC=C2)=O)C1 c1(C(N(C2CC2)CC2CCCN(C(C=CSC)=O)C2)=O)cc(C)ccc1O CC1=CC(C)=NS(=O)(=O)N1CC(=O)NC1CCC2(CC1)CC(NC(=O)C=C(Cl)Cl)C2 C1(CCOC)(C(=O)NC2CCC2N(C)C)CCN(C(=O)CCc2csnn2)CC1 C1(CCC)CCCC1C(=O)NCCC1(CNC(=O)Cc2csc(=N)[nH]2)CC1 c1(OC)cc(OC)nc(C(N2CCC(C(C)NC(=O)CCCC3CC3)CC2)=O)n1 c1(NC(c2c(C)nnn2C)CC)csc2c1CCCC2 c1(OC)cc(CC(=O)OCC(=O)C2(C(F)(F)F)CC2)ccc1C C1(C(=O)NCCNc2c(C)ccnc2)CCC(C)C(C)C1 C12(C(=O)NCC(CC)(C)C)CCC(CC1)N(C(=O)C(C)C1CCC1)C2 C1(NC(CC2CCCN(C)C2)=O)CCS(=O)(=O)C12CN(C(C1(CO)CC1)=O)C2 Cc1nn(C)c(Cl)c1NC(C(C1C(C(=O)O)CCCC1)N(C)C(C1(C)CC1)C)=O c1(OC)cc(C(N2C(C)CN(C(=O)C(O)CSC)CC2C)=O)c2occc2c1 C12(CNC(C3CCS3(=O)=O)=O)CCCC1N(C(=O)CSCCC(F)(F)F)CCC2 c1(C(=O)OC)nccc(C)c1NC(C1(C)CC2CC2C1)=O C1(CN(C(=O)C(C#N)C2CC2)C)C2CN(C(c3ncncc3Br)=O)CC12 Cc1cc(N2CC(CO)C(CC(C)(C)C)C2)nc(=NCCc2ncccc2F)[nH]1 N1(C(c2cnoc2C2CC2)=O)CCN(C(=O)CCc2ccc[nH]2)C(C2CC2)C1 N1(C(c2cc(OC)no2)=O)CCN(C(C2CCN2C)=O)CCC1C c1(C(C)OC)ccc(-c2nc(-c3nccs3)nn2C(C)CO)cc1 c1(C(=O)NCC(C(=O)NC2(CC=C)CC=CC2)CC2CC2)cc2n(n1)CCO2 c1(C(N2CC(CNC(CCCOC)=O)C(C(F)(F)F)C2)=O)c(F)ccc(F)c1F C(=O)(CC(C)C(C)(C)NC(c1ncoc1CC)=O)NC(C=C)C1CCC1 c1(CCCC)nc(CN2CC(F)CC2CN2CC(NS(C)(=O)=O)C2)c(Cl)[nH]1 Cc1nc2cncc(C(=O)NCC(C(C)C)NC(=O)C(F)OC(F)(F)F)c2[nH]1 c1(C(N2CCC(CN(C(C(C)S(C)(=O)=O)=O)C)C2)=O)c2ccccc2nn1C c1(C(=O)NC2(CC=C)CN(C(=O)CSCC3CCCCO3)C2)cc(C)sc1C O=C1CCC(C(=O)N(c2ncnc3occc23)C2CC3CCC(C2)N3)=NN1 C12(C(N3CC(NC(C45CCCCC4C5(F)F)=O)C3)=O)CCCN(CCC1)C2 C1(NC(Cc2c(CC)con2)=O)CC(C(N2CC3(CC(O)C3)C2)=O)C12CCC2 C(CCCCC(=O)N1CCCC1C(C)(C)CNC(=O)COC1CCC1)OC c1(C(=O)NCC2C3CN(C(CC4(N(C)C)COC4)=O)C2C3)cc(O)ccc1Cl c1(C(C(=O)NCC=C)N(C(C)C(=O)OC)CC(C)C)nn(CC)cc1Br Cn1nccc1C(F)=CC(N1CCC(C)(CNC(C2CC3CCC2O3)=O)CC1)=O N1(C(c2cc(C)ncn2)=O)CCC(NC(=O)CC2CCC(C3CC3)O2)C12CCCC2 C=C1CCC(C(=O)NCC2(C(=O)N(CCC(N)=O)C)CCCO2)CC1 C1(CNC(COc2c(OC)cccc2)=O)CN(CC(=O)N(C)C)CC12CCC2 C(=O)(CCCC(C)(C)C)NC1CN(C(C2(CC)CC(C)(C)C2)=O)C1 Cn1ncc(C(=O)NC2CC3C(NC(C4CCC(CC#N)CC4)=O)C3C2)c1Cl C1(NC(Cn2ncc(C)c2)=O)CCCC(Nc2ncnc(=N)[nH]2)C1 C(c1ccc(Cl)cc1)=CC(=O)NCC(C1CC1)NC(CCNC(C1C(C)C1)=O)=O C12(CCNC(=O)NC(c3ccc(NS(C)(=O)=O)cc3)C)COC(C)(C1)C2 C1(C(=O)NC(CNC(=O)C=Cc2ncc[nH]2)C2CCC2)CCc2nnnn2C1 C1(CC(=O)N(CC(CC)NC(c2cc(OCC)n[nH]2)=O)C)CCCNC1=O C(=O)(C(O)CNC(c1ccccc1)C1CC1)OCC(=O)N(c1ccccc1)CC N1(C(C2(CC#C)CC2)=O)CC2CC(C1)N(C(=O)C(C)CC(C)(C)C)C2 C(C(=O)NCCC(F)Cn1cc(CCCC(C)=O)nn1)(C(C)C)OC C1(CN(C(CNS(CC)(=O)=O)=O)C)CCCN(C(c2cnn(C3CC3)c2Cl)=O)C1 N1(C(COC(CC)(C)C)=O)CCN(C(c2cc(N)c(OC)cc2F)=O)CCC1C C1(C(=O)NC2CCN(C(c3ccc(SCC)cc3)=O)CC2)CCN(OC)CC1 CCC(CC)C(C)C(=O)NCC1(C2CC2)CCN(C(C2CCOC2)=O)C1 c1(NC(=O)Nc2cc(SCc3ccccc3)ncn2)nc2cnc(Cl)cc2s1 C(C(C)(C)C#CC(=O)N1CCC(CO)C(O)C1)NC(COC(CC)(C)C)=O C(=O)(C1=CCCCCC1)N1CCCC(NC(=O)CCn2cnnn2)C1 c1(CC)nc2c(C(=O)Nc3cc4c(cc3Br)CCC4)ccnc2[nH]1 C1(CC)C(NC(c2ccc(CO)s2)=O)CCCN1C(=O)C=CC1CCOC1 C(=O)(CCCCCCCCCO)NC1CC(F)(CNC(=O)C=CC2CCCC2)C1 C1(C(N2CC(O)(c3cnn[nH]3)C2)=O)(CC)CCCN1C(=O)C=C1CCOCC1 N1(C(C(C2CCC2)OCC)=O)CC2(C1)CN(C(C1(CO)CCOCC1)=O)CCO2 N1(C(c2cnc(CCC)s2)=O)CC2(C1)CN(C(=O)C(C1CC(F)(F)C1)OC)C2 c1(CC(=O)NCC2N(C(C(C)SC)=O)CC2)ccnn1C C1(C2CC2)(CNC(c2ccnc(CO)c2)=O)CCN(C(=O)C(=O)C(F)(F)F)C1 N1(C(=O)Nc2cc(C)c(Oc3ncccn3)cc2)CCOC(C)(C#N)C1 c1(OC)cccc(O)c1NC(C1CC1C(C)NC(=O)C(O)CC(C)C)=O C(=O)(CCC(=O)NCC(C1CCOC1)NC(=O)C(C)(C)N(C)C)NCC C#CCC(C)(C)C(=O)N(CCN(C(C1C2CCC1CC2)=O)CC)CC CC1(NC(=O)C2CC2)CCN(C(C23CCC(CO2)C3)=O)CC1 C(=O)(C(Cc1ccnnc1)NC(=O)COCC(F)(F)F)OCC c1(C(N2CCC(COCCO)C2)C(=O)NCC=C)nc(Cl)cc(Cl)c1C c1(C(N2CCC(O)(C(C)CNC(=O)COCCF)C2)=O)cccc2scnc12 C1(CCN(C2CCCC2)C(CN(C)CC2CCCCN2)=O)CCS(=O)(=O)C1 CCC(O)(CC)CCNC(C1CC(NC(c2sccc2C#N)=O)C12CCC2)=O C1(C2CCOCC2)(C(=O)NCC=CCNC(C(F)=CCC)=O)CC1(F)F c1(C(N(CCCCNC(C2(O)CCSCC2)=O)C)=O)c(F)ccc2cnn(C)c12 CCC(CNC(=O)CC=CCNC(c1cc(C(C)C)n(C)n1)=O)(CC)OC C(C(C(C)(C)C)NC(c1cnn(-c2ccc(Cl)cc2)n1)=O)NC(CC(C)OC)=O C1(NC(c2nnnn2CCCC2CC2)C2(SC)CCC2)C2CCCOC12 C1(NC(C2CCC(=C)CC2)=O)CN(C(c2ccsc2C#N)=O)CC1N=[N+]=[N-] C(=O)(CCC(F)(F)C(=O)N1CCC(NC(=O)CCc2ccccc2Cl)C1C)OC n1(CC(=O)NC(c2cc(C(=O)NCC(C)Cc3cn[nH]c3)no2)C)cnc(=N)[nH]1 c1(C(N2CC3(CN(C(C=C(C)C(F)F)=O)C3)C2)=O)cc(C)c(C)c2ncccc12 C1(C(C)C)(CO)CCCN(N2CC(NC(=O)OC(C)(C)C)C3(CC3)C2)C1 N1(C(C(COC)NC(c2cc(C)sc2C)=O)=O)CCC(COC)C(C)(C)C1 C#CC1(C(=O)NCC(C)CN2CCCC2)CN(C(c2cncnc2)=O)C1 C#CC1(O)CC(C(=O)NC(C)C(C)(C)NC(=O)C(C)OCc2ccncc2)C1 c1(C(=O)NC(C(C(C)C)NC(COCCC)=O)C)ccn2ncnc2c1 c1(C(N(CC(CNC(COC)=O)C)C)=O)c(C(F)(F)Cl)n[nH]c1C C1(NC(C(C2CC2)SC)=O)C2CC1N(C(=O)CCCc1nc(C)no1)C2C c1(C(=O)NCC2C3CN(C(C(C)(F)F)=O)CC32)cc(Br)c2cccnn12 C1(CN(C(CCOCCOCCCC#C)=O)C)CCN(C(C2(CO)COC2)=O)C1 C1(CNC(c2cnoc2)=O)CC2(CCOCC2)CN1C(c1cc(F)ccc1Cl)=O C12(CNC(C(C3CCN(C(c4cn(CC)nc4)=O)CC3)C)=O)CCCC1CCO2 n1(CC)cc(CC(=O)NCc2ocnc2C(=O)NCC(F)Cl)nn1 Cn1cc(C=CC(=O)NC(Cn2cncn2)C(=O)NCCc2nccn2C)nn1 C1(CNC(c2c(C)scn2)=O)(NC(=O)C(F)=CC2CC2)CC2CCC1CC2 c1(C(N(CCOC)CC)=O)cnc(CNC(=O)C(C)(C)Cl)nc1 CC1NC(=O)CCC1NC(=O)CC1(C)CCN1C(=O)Cn1cncn1 C(=O)(CC(C)(C)C(C)=O)N1CCC(C(N(CC(CC)C)C)=O)C(C)C1 N1(C(C(C)N(C(C)=O)C)=O)CC2(C1)CN(C(=O)CC1CCN(C)C1)CC(C)(C)O2 C1(NC(c2cc(COC)sc2)=O)CC(NC(c2cccn2C)=O)C12CCOCC2 C1(=CCNC(C(c2cccnc2)C)=O)CCN(C(C23CC(C#N)(C2)C3)=O)CC1 C1(C(=O)N(C)CCN(CCCc2ccccc2)C(C)C)(OC)CCSC1 C1(C(N2C(C)(CNC(=O)CCc3cnn[nH]3)CCC2)=O)CCC2(CCOCC2)C1 C1(NC(C2(C=C)CCC2)=O)CN(C(c2ccnc(SCC)c2)=O)CCC1CO Cc1ccc(NC(=O)CCC2CCCN2C(c2ccc(O)cn2)=O)c(O)c1 C(CCCCCNC(C1SCCS1)=O)N(C(c1c(C(C)C)scn1)=O)C N1(C(C(CC)N(C)C)=O)CC2(CNC(=O)C=Cc3scnc3C)CCC1CC2 N1(C(c2cnc3sc(Br)cn23)C(=O)NC(CC)C)CCc2c(C)cc(Br)cc2C1 C(CC(C)(C)C(=O)NC1CCCN(C(c2ccc(F)c(O)c2)=O)CC1)OC C1(COC)CC(C)N1CCCC1(Cc2ccccc2)CC1 Cc1cc(CC(=O)N(CCC(=O)NC2CCOCC2C)CC2CC2)n(C)n1 N1(C(C(CC)SC)=O)CCOC(CCNC(=O)CC2(O)CC2)C1 N1(CCC(C)C)CCCC1C(=O)NCC1(CNC(c2ccon2)=O)CC1(F)F C12(CNC(C3CC(=C)C3)=O)CCCCC1N(C(=O)C(C)CCOC)CCC2 C(C)(N=c1[nH]c(Cl)ncc1C(F)(F)F)C1CCN(C(C2C(CC)CCC2)=O)C1 C1(C)(C(=O)NC(C2CN(C(c3nnc(O)cc3O)=O)CCO2)C)C(C)(C)C1(C)C CC#CC1CN(C(=O)C(C)N(C(=O)C=CC(=O)N(C)C)C2CC2)C1 C(c1cccc(Cl)c1Cl)=CC(=O)NCCCNC(C1CC2C=CC1O2)=O N1(C(C(CC=C)N(C)C)=O)CCC2(CCN(C(c3cccc4nc[nH]c34)=O)C2)C1 C12(NC(C3C4CCCCCCC34)=O)CCCC1N(c1ccc3cc[nH]c3n1)CC2 Cc1cnc(N2CCC3(CCCO3)CC2)c(S(=O)(=O)NC2CCC(C)(C)CC2)c1 c1(C(N(CC(O)CNC(C23CC(C)(C2)C3)=O)C)=O)cccc(C(N)=O)n1 c1(C(N2CC3CC(NC(=O)Cn4ncnn4)CC3C2)=O)cc2ccc(Cl)cc2o1 Cc1cccc2oc(=NCC3(O)CCN(C(=O)CCC(C)(C)F)C3)[nH]c12 C(CC1CC1)(CC(=O)N1CCC(CF)C1)NC(CSCCC)=O C(=O)(C(C)(C)C(F)(F)F)NC(CNC(c1cn(CC(CC)O)nn1)=O)CO C1(NC(CNC(=O)OCC=C)=O)C=CC(CNC(c2csc(C(C)C)n2)=O)C1 C1(NC(C(C)c2ccco2)=O)CCC(O)CN(C(c2cn3cnnc3cn2)=O)C1 N1(C(CC2(C)CCCC2)=O)CC(NC(C2CCCC(O)C2)=O)CC2(CC2)C1 c1(CCC(N2C(C)(CNC(CN(C3CC3)CC)=O)CCC2)=O)c(F)cccc1Cl c1(C(=O)NCC2C(NC(C3CCC(=C)CC3)=O)C2)ccc(F)cc1C(F)(F)F N1(C(CN(CC(C)C)C(=O)CC2CC3CC3C2)=O)CCCC(CCF)C1 c1(C(N2CCC(NC(C3CCCC3)=O)C2)=O)cc(C(F)(F)F)ccn1 c1(N2C(CCCNC(c3cnn(CC4CCCC4)c3)=O)CCC2)ncc(I)cn1 N#Cc1cc(C(=O)NCC23CCCC(CN2C(=O)C=CCN=O)C3)cc(O)c1.C(CO)O CC(C)(C#N)CC(=O)NCC1CCCC(NC(=O)C(C)(C)N2CCOCC2)C1 N1(CC)CCC2=C(C1=O)C(c1ccncc1)NC(=S)N2c1ccc(Cl)c(OC)c1 Cc1nn(C2CCCC2)c(Cl)c1C(N1CCC(CO)(NC(=O)COC(C)C)C1)=O C(C1=CCN(C(=O)CC2CCC3CC23)CC1)NC(C1NC(=O)OC1)=O C#Cc1cccc(C(N2CCN(CC(=O)N(CC)CC3CCC3)CC2)=O)c1 N1(C(C(C)OCC)=O)CCn2nc(C)c(CNC(c3cc(COC)[nH]n3)=O)c2C1 C12(CNC(CSCCOC)=O)CCC(NC(=O)C(C)OCCC(C)C)(CC1)CO2 N1(C(c2ncc(Cl)s2)C(=O)NCCCSCC)CCC2CCC(C2)C1 CC(C)CC(C(=O)N(CCCNC(=O)Cc1cccs1)CCO)C(N)=O Cc1nc(N(CCCCN2CCCCC2)C)cc(=NCc2cc(F)ccc2C)[nH]1 N1(C(C2CCCC2C)C(=O)NC(CC)(C)C)CC2(CCC2)c2ccccc21 CC1CN(C(=O)C(O)C(C)c2ccccc2F)CCN1C(c1cc(CF)on1)=O Cc1cc(O)ncc1C(=O)NC1CCN(C(=O)Cn2cnnn2)CC1 C1(NC(c2cnc(C)[nH]2)=O)CN(C(=O)CCc2cn(C)nn2)CCC1(C)C c1(C(=O)OC)cc2[nH]c(C(=O)NCCCCN(CCCNC(=O)CO)C)cc2s1 C1(NC(C(=O)NCC2CC2)=O)CCN(C(c2occ3c2CCC3)=O)CC1CO N1(C(CC2CC(CC)OCC2)=O)CC2CC(C1)N2C(=O)C(C)(C)CN(C)C Cc1cc(C(c2ccccc2)NC2CN(C)C3(CCC3)C2)c2ccccc2n1 N1(C(COCCOCC#C)=O)CCC(CNC(C23COCC2C3)=O)C12CCC2 C=C1CC(C)(C(=O)NCCN(C(=O)CCCC2CCCCC2)CC(C)O)C1 C1(C2CCN(C(=O)CCc3cnc[nH]3)C2)(NC(=O)CCCc2cnn[nH]2)CC1 c1(OC)ccc(C(N2CCC(CS(N3CCNCC3)(=O)=O)CC2)=O)c(Br)c1 C1(C)(CNC(C(C2CC2)OC)=O)CCCC1NC(=O)C=Cc1ccn(C)c1 Cc1scnc1C(=O)NCCc1n[nH]cc1C(N1CCCC1C(C)(C)C)=O c1(C(N(CCCCCNC(C(C)OCCC#C)=O)C)=O)cc2nnn(C)c2s1 C1(CNC(c2nc(CC)oc2)=O)CC(O)C(O)CC1C(=O)NCCCC(N)=O C(CC(C(=O)NC(C)CNC(=O)CCSc1cccc(Cl)c1)NC=O)SC C1(c2cccc(OC)c2)CN(C(=O)C(F)C2CCC2)CCN1C(=O)CC(C)(F)F C1(C(N(C(CCNC(CN(C(C)C)C)=O)C)C)=O)CCc2cc(F)ccc2O1 N1(c2n(CC)nnn2)CCn2c(C)nnc2C1.C(=O)CC(Cc1ccccc1)C(F)F O=C1CC(C(=O)NC2COCC2NC(C2CCC(=O)O2)=O)c2cc(F)ccc2N1 C(C(CC(F)(F)F)NC(=O)C(F)F)NC(C1CN(C(CC)CC)C(=O)C1)=O O=C1NC(=O)C2(CCN(Cc3ccc(N(O)C)cc3)CC2)N1.C12CCN1C2=O CCCC(C(=O)N1CCCC(C(=O)Nc2ccccc2F)C1)NC(N)=O CC1CN(C(C2C3CN(C(=O)CCc4cccc(O)c4)CC23)=O)CCC1=O N12CCC3(CC1)C(OC)CC3C2=O.c1(CC(=O)NC2(CC)CC2)ncn(C)c1C Clc1ccccc1-c1ccc(-c2ccc(OCC3CC3)s2)cn1 Cc1ccc2occ(CC(=O)N(C)CC3CN(C(=O)CSC(F)(F)F)C3)c2c1 C(CN=c1nc(C#N)[nH]cc1Cl)=CCNC(C(CC)C(C)O)=O c1(C(=O)NC(C2CN(C(C3CCCC3O)=O)CCO2)C)ccn2cccc2c1 c1(N2CC(COC)N(c3ncc(C(F)(F)F)cn3)CC2)ncnc2n[nH]c(Br)c12 N1(C(c2ccc(NC)cc2)=O)CCC(CNC(=O)CC2CCCS2(=O)=O)C12CC2 N#Cc1ccccc1C(N1CCC2(C(=O)NC34CC(C3)C4)C(C1)C2)=O c1(C(C)NC(c2n(CC)ccc2)=O)cccc(-c2cccc(F)c2)c1 C1(C(N(C2CC(O)C2(C)C)C)=O)CCC2(CC1)CC2.c12ncccc1C(=O)NC2 CN1C(=O)CC2CN(C(C3CCCN(CCCCCF)C3)=O)CCC12 CCCCC(O)C(=O)N1CC(NC(=O)C=CSC)C(CC(C)(C)C)C1 C#CCC(C)(C(=O)N1CCC(CC)CC1)NC(C1CCCO1)=O C1(C#N)(Nc2nccc(Br)n2)CCN(Cc2c(SC)cccc2)C1 N1(C(C2C(CC)CN(C(=O)CC3(O)CCCC3)C2)=O)CCC(C2CCCC2)C1 Cc1ccc2cc(CNC(=O)C=C3CCN(C(=O)C(C)NC=O)CC3)ccc2n1 c1(NC(C(=O)NC2CCC(SCC)CC2)=O)ccc2ncsc2c1 C(=O)(CCCC(=O)NC(C1(NC(C2CCOC2CC)=O)CC1)C)NCC Cc1cc(C(C)NC(=O)C=CC(C)(C)NC(c2ccn(C3CC3)n2)=O)no1 Cc1cc2[nH]c(C(N3CCC(n4cc(-c5cc[nH]n5)nn4)C3)=O)cc2o1 c1(C(=O)NCCNC(CC(C)C2CCCO2)=O)cc(Cl)cc(Br)c1 C1(CCC)CCCC1CNC(=O)COCCNC(=O)CN1CC(C)(OC)C1 c1(C(N(C(c2cn(CCN3CCOCC3)nn2)C)C)=O)cnn2c1OCCCC2 C1(CNC(C(C)(C)OC)=O)CCCC(CNC(c2nocc2C2CC2)=O)C1 CCCC(C)(CCC)C(=O)N(CCCNC(=O)C(C)(O)C(F)(F)F)C C=C(C)CCCC(=O)NC1CC(C(=O)NCC(CC(C)C)OC)CC1O N1(C(C(N2C(C)CC(N)CC2)=O)=O)CCC2(CC1)C(=O)NCc1ccccc12 CCC(C)C(C)CNC(C1(C)CN(C(C2(n3cccn3)CC2)=O)C1)=O C1(O)(CNC(CC2CCCN(C(C=NOC)=O)C2)=O)CCCC1(C)C N1(C(c2c(C)nc(C)s2)=O)CC(=O)NCC1C(N1CC=CC(O)C1)=O C12(CNC(C=C(C)Cl)=O)CCC(CN(C(=O)CCN(C)C(=O)OC(C)(C)C)C1)C2 N1(C(c2cccc(SC)c2)=O)CCC(NC(C2(C(F)(F)F)CC(F)C2)=O)CC1C N1(C(C2C=CC(NC(=O)C(=O)C3CCCC3)C2)=O)CCn2c(O)nnc2C1 C(=O)(C(F)C(C)CNC(c1sccc1F)=O)NCc1cc(OC)ncn1 N1(C(COCC#C)=O)CC(NC(=O)C(F)C(F)(F)F)CC12CCC2 CN1CCCCCC1C(=O)NC1(CC(=O)NC2C(O)C3CCOC23)CCC1 C1(NC(CCNC(=O)NC)=O)CCN(C(=O)COC)C12CC2 c1(-c2n(CC)c(N3CCC(F)(c4cccc(Cl)c4)C3)nn2)ncc(C)cc1Br c1(C(=O)NCC2CN(C(C3(COC)CCOCC3)=O)C2)cc(N)c(F)cc1F N1C(=O)NC2(CCC2)C1=O.C(C1CNc2ccccc21)OC(C(CC#N)c1nc[nH]n1)=O CC1CCOC1C(N1CCCC1CN(C(=O)CCc1nc[nH]n1)C)=O c1(CC(=O)NC2CC(NC(C(Br)=C(C)C)=O)C(O)C2)cccc(C)c1C C1(CC#C)CCCCN1C(C1CCCCC1NC(c1ccoc1C)=O)=O C1(N(C(=O)C=C(Cl)Cl)CCF)CCCN(C(c2ccc(-c3cnco3)cc2)=O)C1 C(=O)(C(C)(C)C(O)C(C)C)NC(CCCC(=O)NCCSCC#C)CC N1(C(C(CC)N(C(=O)C(C)CC2CCC2)C)=O)CC(C2=NOC(C)C2)C1 c1(C(=O)NCC2CCC(NC(c3cccc(=O)o3)=O)C2)cc(F)cc(F)c1 C1(CN(C(C=COCC)=O)C)CCCN(C(=O)C(=CC2CCCC2)C)C1 N1(CC)CC(C(=O)NCc2cc(C(N3CC(CCO)C3)=O)n[nH]2)CC1=O c1(CC)ncc(CNC(C2CC(C)N2C(=O)CCN2CCCC2)=O)[nH]1 CC1CCC(C(=O)NCCc2noc(=O)n2C)CN1C(c1ccc([N+](=O)[O-])o1)=O N1(C(C(C)(C)N2CCCC2)=O)CCOC(CC(=O)NC2CCCC(O)C2)C1 C(N=c1[nH]cnc2c(OC(C)=O)cccc12)C1CCCN(C(C(COC)(C)C)=O)C1 N1(C(C2CC(C#C)(O)C2)=O)CCCCC(CCC(=O)N(CC(C2CC2)OC)C)C1 C12(C(=O)NC3CN(C(=O)CCCn4cccn4)CC3O)CCCCC1CCCC2 C1(C(N(CCCNC(=O)CCCn2cccn2)C)=O)CC12CCC(=O)CC2 C1(C)(COC)CC(NC(c2cn[nH]c2)=O)CN1C(C1CC(F)(CF)C1)=O N1(C(CCOCCOCCCC#C)=O)CCN(C)C(NC(=O)C(O)CC(N)=O)C1 C1(C(=O)NC(CC#C)C(=O)NC)CCN(C(C2SCCS2)=O)CC1(C)C C12(NC(c3csc(-c4ccccc4)c3)=O)CC1CN(C(C1CC1C(F)F)=O)C2 C1(C(C)C)(C(=O)N(C)CC=CC(=O)N(N2CCCC2)C2CC2)COC1 c1(C(=O)NCCOC2CN(C(c3cc(C)no3)=O)C2)ccc(C)c(F)n1 C(CCCC(=O)NCC=Cc1cccnc1)N(C)C(c1ccnnc1O)=O c1(C(=O)NCC(CC=C)NC(=O)CCC(F)F)ccccc1C(=O)NCCCC C1(C(N2C(C)(C(=O)OC)CC2)=O)C2CCCC2CN1C(=O)CC1C=CCCC1 C1(C(N2C(C(=O)NC)CCC2)=O)(N(C(=O)C2=C(Cl)CC2)C2CC2)CCCCC1 Cn1c(NCC2(C)CCCN(C(=O)CC3CCC(=O)N3)C2)cc(O)nc1=O c1(C(=O)NCC(CN(C(=O)C(C)(C)n2cncn2)C)O)n[nH]cc1C1CC1 N1(C(C2C(CC(C)C)C2)=O)CCC(C)(C(=O)NCC2(C)CSC2)CC1 C(=O)(C1=CCOCC1)NCCC1CCC(NC(C=C2CCN(C)CC2)=O)C1 C1(C(N2C(C)(C(=O)NCCC3C(C)CCO3)C=CC2)=O)CCCC1C1CC1 C1(C(=O)NCC2CN(C(=O)CCCc3nccs3)C2)CCS(=O)(=O)N1 C(N=c1[nH]c(NCC(c2ccccc2)C)nc2c1CCCC2)c1ncc(C)cn1 N1(c2ncc(C(=O)OC)cc2Cl)CC2CC1CCC2NC(=O)C1=CCSC1 N1(C(c2c(OC)ccc(C)n2)=O)CC2CCCN(C(C3CC3C)=O)C2C1 CC1CCC(CC(N2CCCC2Cc2cn(Cc3cccc(O)c3)nn2)=O)CC1 C(C(C(=O)NC1CN(C(C2C3CCC(F)(F)C23)=O)C1)C(C)(C)C)OCC=C CN=c1[nH]cc(C(=O)N(C(C)CNC(C2CC2(c2ccccc2)C)=O)CC)o1 C1(NC(=O)NCC2N(CC(=O)N(CC)CC)CCC2)CN(C)CCO1 C1(C(=O)Nc2cnc(Cl)c(Cl)c2)CCc2nc(-c3cccc(O)n3)sc2C1 C12(C(=O)NCC(CC(C)C)(C)NC(c3ccc(Cl)o3)=O)CCCC1CC(=O)C2 N1(C(C(CC2CC2)NC(CCC#C)=O)=O)Cc2cccc(F)c2C1 C(C)(C)(CC(C)(C)C)NC(C(C)Cc1cn(C2CCCC2O)nn1)=O c1(C(=O)NCCC2CN(C(C3(CC)CC3)=O)CC2C)cc(=O)c2ccncc2o1 c1(C(C)=O)cccc(C)c1NC(c1cc(C)nc(C2CCC2)n1)=O C1(NC(C2OCCC(C)C2)=O)CN(C(c2cc(C3CC3)on2)=O)CCC1C C(CC1=CCN(C(C2CC2C)=O)CC1)NC(C1N(C(C)=O)CCCC1)=O C(C(O)C(=O)NCCN1CCCC1)SC.C(=O)(C(COC)NC(C)=O)NC(C)C C(CC(CC)C(=O)NC(C)C(CO)NC(c1ccccc1SCC)=O)=CC C1(C(=O)Nc2nc(O)cc(C(=O)OC)n2)CCCC2CCCCC12 C(=O)(CCCC(=O)NC1CS(=O)(=O)CC1NC(=O)C(F)(F)c1cnccn1)OC C1(C(=O)NCc2cn(CCC3(CO)CCCC3)nn2)CCc2nn[nH]c2C1 CC1CCN(C(=O)CCc2cccc(Cl)c2)C1CNC(=O)Cc1cc(Cl)n(C)n1 O=C(C#CC1CCC1)NCC12CC1CN(C(=O)CCC1CCC(C(F)(F)F)O1)C2 N1(C(c2c(C)ncs2)=O)CC2(CNC(=O)C(c3ccccc3Cl)(C)C)CC1CO2 c1(C(NOC(C=C)C)=O)occc1CN(C(=O)C(OC)OC)C1CCC1 C(=O)(C(N=[N+]=[N-])C(C)C)NC12C(CN(C(C(COC)N(C)C)=O)C1)C2 C1(OCC)CC2(C1)CC2C(=O)NCC1CC(O)CN1C(=O)C(C1CCCCC1)C C12(NC(C=CC)=O)CCN(C1)C(=O)CS(=O)(=O)N(CC)C2.OC.C(C)SC N1(C(C(C)(O)C2CC2)=O)CCC2(CCCCN(C(C3(C(F)F)CCCO3)=O)C2)C1 N1(C(C2C(=C)C2)=O)CCC2CCC(C1)N2C(=O)C(=O)N=S(C)(C)=O C1(CNC(C=COCC)=O)CCCC(CNC(c2cnn(C3CCC3)c2)=O)C1 CC1(NC(C2CC3CC3C2)=O)CC(NC(c2ccsc2-n2cnnn2)=O)C1 Cc1nc2c(C)cc(C(N3CCOC(CN(C(=O)C(C)CO)C)C3)=O)cn2n1 N1(C(=O)OC(C)(C)C)CCC(C2CC2)C1NCCN1CCC(C)(O)C1 CC(C)S(=O)(=O)CC(=O)N(C)CC1(CNC(C2CCC(=O)O2)=O)CC1 CCCC(CCC)C(=O)NC1(C)CC(NC(=O)CC2CCS(=O)(=O)C2)C1 C(=O)(CC(C)C(F)F)NCC(CC)(CC)NC(=O)C(F)(F)C(O)c1ccccc1 Cc1ccc(C(=O)NC(C2CC2C(=O)NCCC(=O)N(C2CC2)C(C)C)C)c(C)c1 c1(C(N(CCNC(C(CC=C)Cc2ccccc2)=O)CC)=O)ccc(N)c(Cl)c1O N1(C(C=Cc2ncn(C)c2)=O)CCN(C(c2n[nH]cc2Br)=O)C2CC12 C1(C)(C(=O)NCC(C2CCN(C(C3(O)CCC3)=O)CC2)C)CC=CCC1 c1(C(C)C)ccc(C(N2CC3C(C2)N3C(c2cc[nH]n2)=O)=O)c2ccccc12 C(=O)(C1=C(C)CCC1)N(C(C(=O)NCC1(CCOC)CCC1)C)C1CC1 CCC(=O)NNC(=O)C(C)OC(c1cnn(C)c1C(C)(F)F)=O C1(CC(=O)NC2CC(CNC(c3csnc3Cl)=O)C2)CCCOC1 c1(C(=O)NC2CCC(N(C(CS(=O)(=O)NC)=O)C)C2)ccn2c1CCCC2 Cc1nnn(CC(=O)N(CCC(C)NC(C2(CO)COC2)=O)C)n1 c1(CC(=O)NCC(C)N(C(c2cc(C3CC3)nn2C)=O)CC)sc(O)nc1O C1(CC(=O)NCC(CNC(=O)CC(F)(F)F)CO)NC(=O)CNC1=O c1(OC(C)C(N2CC3CCN(C(=O)COC4CCC4)C3C2)=O)c(F)cccc1F N1(C(CCOCCOCC)=O)CC(C(=O)NC2(CC)CC2)C(C)C1 S(=O)(=O)(c1ccc2oc(=O)ccc2c1)N(C)CC1(F)CCOC1 C1(C(CNC(CNC(=O)OC)=O)(C)C)CCN(C(c2cscc2C(N)=O)=O)CC1 C1(NC(c2nc(C)sc2C)=O)CCC2(CC1)CN(C(=O)Cc1cnc[nH]1)CCO2 C1(NC(N2CCC(C(C)C)C2)=O)CCC(C)(C)CC1c1ccccc1 Cc1cc(C)n2nc(C(=O)N(c3ccc(F)cc3Br)C3CCN(C)CC3)cc2n1 C1(C(N(C(CC)CO)C2CC2)=O)CC2CN(C(=O)C(C)N3CCCC3)CC2C1 n1(CCC)nc(-c2ccccc2Br)nc1C1CCCc2scnc21 N1(C(C(n2ccc(C)n2)C)=O)CCCC(NC(C2Cc3nccn3C2)=O)CCC1 N1(CC#C)CCN(C(=O)C(O)CNC(c2sccc2C)=O)CC1=O c1(C(N2CCCC(N(C(=O)CN(C)C(C)=O)CC)CC2)=O)cc2ccncc2s1 c1(OC)ncc(C(=O)NCC2CN(C(=O)CN3CC(C)(C)C3)C3CC23)cn1 N1(C(c2ccc(Nc3ccncn3)cc2)=O)CCC(N2CC(F)(F)C2)CC1 C=C(C)c1cn(CC(C2CN(C(=O)CCNC(=O)NC3CC3)C2)F)nn1 CCCS(=O)(=O)C1CCCC1CNc1nnn(C2CCC3(CC2)CNC(=O)C3)n1 N1(c2nc(=N)nc(N3C(CO)CC(OC)C3)[nH]2)CCC2(CCCOC2)C1 c1(C(N2CC3C(NC(c4c(CC)ccs4)=O)C3C2)=O)cc(C)cc(C)c1 C1(NC(COCCC=C)=O)(CNC(=O)CC2CCCOC2)CCC(F)(F)CC1 CCC(F)(F)CC(=O)NC1(CNC(=O)Cc2cc(F)cc(F)c2)CC2CCC1C2 C(CCF)(C(=O)NC(C)CCO)NC(c1c(COC)cc[nH]1)=O N1(C(C(CSC)OC)=O)CC2COCC2(C(=O)NCc2cccc(F)n2)C1 c1(CC)c(N2CC3C(NC(=O)Cc4cccc(OC)c4)C3C2)nc(C)nc1Cl c1(OC)cc(C(N2CCC(NC(=O)C3=CCOCC3)C(O)C2)=O)c(Cl)cn1 N1(C(c2ccc(NC)cc2)C(=O)Nc2ccccc2)CC2(CC3CC3)CCC1C2 CC(CCN(C)C(C1CN(C)C1)=O)NC(=O)COCC1CC1 CC1(C)CN(C(C2CCC2)=O)CC(CNC(C23CCCCC2C3)=O)O1 C(C(CC1CCCC1)C(=O)N1CCCC(CCO)C1)NC(C1CCCCC1)=O N1(CCCOC)CCC(C(=O)NCC=CCNC(C2CCCC2C(F)F)=O)CC1 n1(CC(=O)NCC(C2CC2)NC(C2(SC)CC2)=O)cnc(Br)n1 c1(C(N2C(c3cc(OC)c(C)cc3)CCC2)=O)cc(Cl)cc(Br)c1F C(=O)(C1(C)CCn2c(C)nnc21)NC1C2CN(C(CS(CC)=O)=O)CC1C2 C(C(CC(=O)N(CC(C)(C)C)CC1CC1)C1CCC1)NC(COCCSC)=O c1(C(=O)NCCN(CCOCCO)C(C23CCCCC2C3)=O)nccn2ccnc12 c1(C(=O)NCC(CN(C(=O)CC2COCCO2)CC)O)csc(CC(F)(F)F)n1 c1(OCC)n[nH]c(=NC(C)(C)CCCO)o1 CCCC(C(O)C(=O)N(CCOCCO)CC)NC(C1CC(CC(F)F)C1)=O N1(c2nccc(C#N)n2)C2CCCC1CN(C(c1ccc(O)nn1)=O)C2 N1(C(c2c(OC)ccc(C)c2)=O)CC(C2CCCN(C(C3CCC(=O)N3)=O)C2)C1 C1(OC)CN(C(c2ccnc(CN(C)C)c2)=O)CC1NC(=O)Cc1cccs1 N1(CCC)CCC(C(=O)NC2(CNC(=O)C(=C3CCCCC3)F)CCOC2)CC1 CC1(C)CCC(C(=O)NCC(O)CNC(C2(CO)CC2)=O)CO1 N1(C(C2(CO)CCN(C(C(C)NC(CC)=O)=O)C2)=O)CCN(C)CC1CO c1(OC)ncc(F)cc1C(=O)NCC1CC1NC(=O)CCCc1ccc(C)cc1 N1(C(C(C2CCC2)OCC)=O)CCC(C)(CNC(c2c[nH]nc2C(F)(F)F)=O)C1 N1(C(CCCC(CC)CC)=O)CC23CCCC2(C1)CN(C(c1cccs1)=O)C3 N1(CCC)CCCC(C(N2CCC(O)(CNC(c3ccoc3CCC)=O)C2)=O)C1 N1(C(CCc2onc(C)n2)=O)CC(C)CCC1CNC(=O)C(C)(C)F C1(C2CC2)(C(NOCC(C)O)=O)CN(C(C2CN(C(=O)OC(C)(C)C)C2)=O)C1 C12(C(=O)NCC(CC)NC(C3CC(S(C)(=O)=O)C3)=O)CCC(C)(CC1)OC2(C)C Cc1[nH]nc(C(=O)NCC(C2CCC2)NC(C2CCCCC2C(C)(C)C)=O)c1C CCC(CC(=O)N(CC(O)CNC(=O)CCn1cccn1)C)SC C(CCC(C)C)(C(=O)NCC1CCOC1(C)C)NC(CC1(C(=C)F)CCC1)=O N1(C(CCC=CC)=O)CCC2(CC1)OCCC2NC(=O)C(C)NC(C1CCC1)=O CC1(C)CCCC1C(=O)NC1CCCC1NC(c1ccon1)=O C1(OCC)CCCN(C(=O)C(CCF)NC(=O)CC2CCSCC2)C1 Cc1ncc(C(=O)NC2CN(C(c3cn(C)nn3)=O)CC2C)n1-c1ccccc1 C1(C(N(CC(C)(C)NC(C=C(C)C(C)C)=O)C)=O)CCCCN1NC(N)=O C1(C(=O)NCC2CCC(NC(c3ncn(C(C)(C)C)n3)=O)C2)CC(S(N)(=O)=O)C1 N1(C(C(C=C=C)C)=O)CC2(CC2)CC1CC(=O)NCC(c1cccs1)C Cn1c(C(N2C(CC(=O)NCC3C=CCC3)C3CCCC23)=O)cccc1=O N1(C(C(C)OCCC=C)=O)CCC(C2CC2)(CNC(=O)COc2ccn(C)n2)C1 c1(C(=O)OC)sc(C(=O)NC(C)CCNC(c2nocc2C)=O)cc1C C(=O)(CCCC(=O)C(C)(C)C)N1C(CNC(C(C)CCCc2ccccc2)=O)CC1 C(C(C)(O)CC(=O)N1CCC(n2cc(-c3ccc(Cl)cc3)nn2)C1)OCC C1(C)(CNC(CC=CC=C)=O)CCCC1NC(=O)Cc1cccnc1F C=CCCCCC(C(=O)NC1COC1)N(C1COCCC1O)C CC1=CCC(C(=O)NCC2(C)CCCN2C(=O)C=Cc2cc(C)no2)CC1 c1(CC)nc(NCC(C2CC2)N(C(=O)Cc2cc(C)on2)C)c(C#N)cc1C N1(C(C(NOC)=O)=O)CCC2(CC(C(N3CCCC(F)(F)CC3)=O)C2)C1 c1(C(N(C(C(N2CCCC2C2CCCC2)=O)C2CC2)C)=O)nnc(O)nc1O C1(C(N(C(CNC(=O)C(C2CCCCC2)O)C2CC2)C)=O)CC(O)(C(F)(F)F)C1 C#Cc1ccnc(C(N2CCC(C=C)(C(=O)NC3CCCC3)C2)=O)c1 N1(C(c2nc(CC)oc2)=O)CC=C(CCNC(c2cc(Cl)ncc2OC)=O)CC1 N1(C(C2CCC(C)CC2)C(=O)NCCOCC)CCC(C(F)(F)F)C2(CCC2)C1 C(C)(C)(CC(C)(N=c1ccn(CCOC(C)C)[nH]1)c1nnnn1C)SC C1(NC(CN2CCC(C)CC2)=O)(CNC(=O)CN(C)C)CCCCC1C C#CCC(C)(CC)C(=O)NCCC1CCCN1C(=O)CCc1cc[nH]n1 C=CC(CC)CC(=O)NCC=C1CCN(C(=O)CC2CC(C)(C)CO2)CC1 CN(C)S(=N)(=O)N1CCCC1C(=O)NC1CN(C(=O)C=Cc2cnc[nH]2)CC1O c1(C(N2C(C)CC(NC(c3ccnnc3O)=O)CC2)=O)cc(O)c2sccc2c1 Cc1ccc(Cl)c(C(=O)NCC(C2CC2)N(C)C(C2CC2(F)F)=O)c1O C1(C(N2CCC(N(C(=O)CN(C)C(C)=O)CC#C)CC2)=O)OCCN(C)C1=O C1(C(=O)NC2(CC)CCCN(C(C3CC(C#C)(O)C3)=O)C2)CCC([N+](=O)[O-])CC1 C1(C)(CCC)CCCN(C(=O)CC2CCCCN2C(C2C=CCCC2)=O)C1 N1(Cc2ccc(C(C)C)cc2)CCNCC12CCC2 CC(C(=O)NCC1(CC(=O)NCCCSC(F)F)CC1)n1cncn1 CC(CC(=O)N1C(C(=O)NCCN(C)C)CCC1C1CC1)C(C)(C)C C1(C(N(CC(C)NC(=O)C2=COCCO2)C)=O)CCCCC(=O)C1 N1(C(C(CC)(F)F)=O)CCN(C(=O)CN2C(=O)CCC2=O)CC12CC2 c1(CCC(=O)NC2CCCC2NC(c2ccc(C(F)F)o2)=O)nnc(O)nc1O c1(C(=O)NC(C(=O)NCC2CC(=C)C2)C2CCC2)ccn(C)c1 c1(C(C(=O)N(CCCNC(=O)C(C)Cc2ccncc2)CC)C)ccc(C)cc1 C1(CNC(c2ccnc(C)n2)=O)CC2CCC(C1)N2C(=O)CC1CCS(=O)(=O)C1 Cc1ncc(CC(=O)NCCC2CN(C(c3ccns3)=O)CCO2)c(O)n1 C(C(O)CC(=O)N1CC(O)(CO)C1)NC(=O)Cc1ccsc1 C#Cc1cccc(C(=O)NCC2(C(=O)N(C)CC3CCCC4CC34)CC2)c1C CC1(C)C(=O)CC1C(=O)NC(C)(C)C=CC(=O)NCC1(C)CCCS1 C1(CC(=O)NCC(C2CCC(F)(F)CC2)C)C(=O)Nc2ccccc2S1(=O)=O CC(CN(C)C)CCC(=O)N1CCC2C(NC(=O)COCCCN(C)C)C2C1 C1(NC(c2c(CC)non2)=O)CCOC(C(=O)N(CC)Cc2cn(C)nn2)C1 Cc1[nH]c(C)c(C(N2CC(CNC(C3CCCOC3c3cn[nH]c3)=O)C2)=O)c1C CN=S(C)(=O)c1cccc(C(=O)NCCN(C(=O)CC2OCCCC2(C)C)C)c1 c1(OC)ccc(CC(=O)NC2CCC2NC(c2cn(C)nc2C(C)C)=O)c(Cl)c1 N1(C(C2N=C(C)SC2)=O)CCCC(NC(C2(S(N)(=O)=O)CC2)=O)C1C C#Cc1cccc(C(=O)NCC2CC(C(=O)N(C3(CO)CC3)C)CO2)c1C CCCC(C)(CCC)C(=O)NC1(CNC(c2nccn2CC)=O)CCCCC1C C1(C(=O)NC(C2CCOCC2)C)CC=CCN1C(c1cccnc1)=O C1(CC=CC)CCCN(C(=O)C(C2CCN(C(=O)C(C)c3ccsc3)CC2)C)C1 c1(NC(C(C)N(C(=O)CCC2CCCCO2)CC)=O)cc(C)cc(C)c1O C1(CNC(C2(C(C)C)COC2)=O)CN(C(c2nc(=O)cc(N)[nH]2)=O)CCC1(F)F C1(C(=O)NC(C(=O)NC)CC2CCC2)CCC2(CC2)N1C(=O)C(C)CSC N#Cc1ncc(C(N2CCOC(CCNC(=O)CCNC(N)=O)C2)=O)s1 c1(CCC)cc(C(=O)NC(CN(C(c2nnn(C)c2C)=O)CC)CC)c(C)o1 C(=O)(C(O)C1=CCCCC1)NC1CCC(C)(N(C(=O)C2=CCOCC2)C)CC1 c1(NC(CNC(C2COCCO2)=O)C2CC2)ccn2ccnc2n1 c1(C(C)NCCNC2CNCC(C)(C)O2)cc2ccc(Cl)cc2o1 C1(C(N(CCCNC(=O)C(c2ccccc2)C2CC2)CC)=O)COCC(C)(C)O1 C(C(C)(C)CC(=O)NCC(C1CC1)N(C)C(c1c[nH]nc1C(F)F)=O)OC c1(C(N(CC)CC)=O)ccc(SC)cc1.C1(CO)C(C)NCCC(=O)N1 c12nc(C)c(s1)OC(=O)C21CCC1.c1(C(=O)OC)ccc(OC(F)(F)F)cc1 C(C)(C1CCCCC1)=CC(=O)NCC(c1ccccc1)N(C(C1C(C=C)C1)=O)C Cc1nc(NC(C(C)NC(C2CC3CCCCN3C2)=O)C(C)C)cc2nncn12 C1(C2CCCCC2)(C(=O)NC2CC(NC(C3(C)C=CCC3)=O)CC2O)CC1 C1(OC)CN(C(=O)Cn2ncn(C)c2=O)CC1NC(c1ccc(Cl)o1)=O c1(C2C(NCc3ccn(C(C(=O)OC)C)n3)C2)ccc(C#N)cc1 c1(CC)onc(C)c1C(N1CCCC1c1cccc(I)c1)C(=O)NC1CCCC1 C(C)(CCCCCO)NC(C1CCC(CNC(C(CC2CCC2)OC)=O)C1)=O c1(SCC(=O)NCCC(CNC(=O)CC2CCOC2C)OC)ccc(C)cc1C C12(CC)CN(C(=O)NCc3ccc(C)c(O)c3)CC(CO)(C1)C2 c1(C(=O)NC(CCNC(CC(C)C)=O)C)cncc(-n2cccn2)n1 C(C)(C)(C(=O)N1CC(c2ocnc2NC(C2CC2C)=O)C1)CNC(=O)OC N1(C(c2c(C)cco2)=O)CCN(C(=O)C2CC2)C(c2cn[nH]c2)C1 C1(C(=O)NCc2n(CC)ccn2)CCC2CCC1N2C(=O)CC1CC(C)=NO1 c1(C(=O)NCC(CNC(C(C)OCC#C)=O)(C)C)cnc(S)n1C C1(C)(C(=O)NC(=O)C(C)(C)C)CCCN(C(=O)CSCC)C1.C1CS1 C(C)(CN=c1[nH]cnc(Cl)c1Br)N(C(C(C)CCN(C)C)=O)C N1(C(C2C(CC)OCCC2)=O)CCN(C(=O)COc2cn[nH]c2)CC12CCC2 N1(C(C2(OC)CCC2)=O)CCC(CCNC(=O)C(F)=CC2CC2)C1 C1(C(N(CCCNC(=O)Cn2cnc(Br)c2)C)=O)CCCC(N(C)C)C1 c1(OC)cccc(CC(=O)NC2CC(N(C(=O)C(C)NC(C)=O)C)C2)c1OC c1(C(N2CCC3(NC(c4conc4C4CC4)=O)C(C2)C3)=O)cnc2ccccn12 S(=O)(=O)(C1CCN(C(c2cccc(C(C)N(C)C)c2)=O)C1)NC.n12cc(nn1)C2 C(C(CC(=O)N(CC(C)(C)O)C)NC(c1csc(F)c1)=O)OC c1(N(C)CC2(C)CCC2)nc(N(CCCOC(C)(C)C)C)c2ccccc2n1 Cc1sc(O)nc1C(=O)NCCC(C)(C)CNC(c1csnn1)=O N1(C(C2CC3CN(C(CCCSC)=O)CC3C2)=O)CCC2(CCCCO2)C1 C(=O)(C1SCCc2ccccc21)N(CC(C)N(C(c1nccc(OC)c1)=O)C)C c1(OC)cc(F)ccc1N1CCN(C(=O)NCC(c2cccnc2)N2CCCC2)CC1 c1(OC)nccc(C(=O)NCC(C)NC(=O)CCn2cnccc2=O)n1 c1(C(=O)NCC(CC)NC(c2conc2C2CC2)=O)cnc2c(cnn2CC)c1 N1(C(COc2cccc(C)c2)=O)CCC(NC(C2(C)CCCS2)=O)CC(O)C1 C12(C(N3CC(C)(NC(C4(C)CCCN4C)=O)C3)=O)CCC(CF)(C1)OC2 C1(C)(CNC(C2CN(C(C)C)C2)=O)CCN(C(c2c[nH]nc2-n2cnnn2)=O)C1 Cc1ccc(-c2ncn(C)c2CN(CCN2CCCC2)C(C)C)c(F)n1 Cn1cc([N+](=O)[O-])cc1C(=O)NC1CN(C(c2ccc3nccn3c2)=O)C2CC12 C1(C(=O)NCC2(C)CN(C(c3ccc(F)s3)=O)CCO2)CN2CCCN1CC2 C(CC1=CCCCCC1)NC(C1CCC(C(C)C)N1C(C1CCC(F)(F)C1)=O)=O C12(CNC(COCc3ccc(C)cc3)=O)CN(C(=O)C(C)(Cl)Cl)CC(F)(C1)C2 C(=O)(C(O)CC(F)(F)F)N1CC(SC)C(NC(C23CC(CO)(C2)C3)=O)C1 c1(C(N(C(CNC(=O)CCC2CC(F)(F)C2)C2CC2)C)=O)ccc(O)c(F)c1F c1(C(N2C(CNC(C3(F)CCOCC3)=O)CC(OC)C2)=O)ccc2c(c1)CCN2 Cc1ncc(NC(C2(C)CCN2Cc2ccnc(F)c2Cl)=O)cc1Br Cc1ccc(=N)[nH]c1C(N1CCC(C)(CNC(C2(C)CC=CCC2)=O)C1)=O c1(CN(N2CCCCC2)C(N(CC(C)(C)O)CC(C)(C)O)=O)ccc(F)cc1F C=C(C)C(CC(=O)NC1CCC(N(C)C(C2CCC(F)(F)CC2)=O)CC1)OCC N1(C(CCCC(=C)C)=O)CCC2CN(C(=O)CSCc3ccncc3)CCC2C1 CC(C)(C)C(CNC(c1cn[nH]c1)=O)C(=O)NCCC1CCCC12CC2 C1(C(N2CC(N(C(C3CC(OCC)C3)=O)C)C2)=O)COCCO1 C1(c2cn(C)nc2)CN(C(c2ccc(Cl)cn2)=O)CCN1C(=O)C=CS(C)=O C1(C(N2CCC(CCNC(=O)Cn3cccnc3=O)CC2)=O)(OC)CCCOC1 Cn1c(CN2CCC(CO)C(O)C2)nc2cc(Br)ccc12 N1(Cc2c(C)cccc2)CCC2(CN(C(c3cc(Cl)ccc3F)=O)CC(C)O2)C1 c1(C(=O)NCC2(C)CCN(C(C3CCCC4CC34)=O)C2)c(Cl)oc2ccccc12 CC1(NC(=O)CCc2nnc(C(F)F)o2)CCCN(C(C2CC2F)=O)C1 C1(OCC)CC(NC(=NCCCOC)NCC(F)=C(C)C)C12CCCCC2 N1(C(C2CCC(C)N2C(=O)CCC2CCCO2)=O)CC2CCCC2C1 N1(C(c2cccc(OC)c2F)=O)CCn2c(C(=O)Nc3cnns3)cnc2C1C N1(C(c2c(SC)ccc(N)c2)=O)CC2CC(NC(c3c[nH]nc3C)=O)CC1C2 NS(=O)(=O)c1n[nH]cc1C(N1CC(C(N)=O)(CNC(C2(F)CCCCC2)=O)C1)=O C=CC(CCC)CC(=O)NCC1(CNC(C2Cc3ccccc3O2)=O)CC1 c1(CC)conc1C(c1nnnn1C)NCC(C)COC N1(C(C2C(CC)CCC2)=O)CCN(C(C23CC=CCN2CCC3)=O)CCC1C C1(O)(CNC(C2(C)CC2(F)F)=O)CCCN(C(c2cncn2C2CC2)=O)CC1 N1(C(C2N(C)CC2)=O)CCCC1C(N1CCC(c2ncc[nH]2)C1)=O C(=O)(C(=O)N=S(C)(C)=O)N(CC(C)NC(C1CCCN1C1CC1)=O)C C(C)(CC(=O)N1CCC1CNC(c1cnc(S)n1C)=O)(C(F)F)NC(C)=O C1(OC)CC2(C1)CC(C(N1CCOCC(CNC(c3ccc(F)o3)=O)C1)=O)C2 C1(C2CCCCC2)(C(N(CCN2CCN(c3nccc(OC)n3)CC2)C)=O)CC1 c1(C(=O)NCC2C(OCC)CN(C(c3n[nH]cc3CC)=O)C2)cc(C#N)cn1C c1(CCC(=O)N(CC(C)NC(C2CCC(C)(F)CC2)=O)C)ccc(F)cc1F c1(OC)ccc2[nH]cc(C(=O)NC3CN(C(c4coc(SC)c4)=O)C4CC34)c2c1 c1(OC)ccc(Br)cc1CCC(=O)NC1(CN(C(=O)C2=CC(C)(C)C2)C)CC1 c1(NC(C2CC2C(N2CCOC(O)C2)=O)=O)ccc(Br)nc1[N+](=O)[O-] N1(C(C(C(C)C)N)=O)CCCCC2(C1)CN(C(c1cocc1C)=O)C2.C(C)(=O)OCC S(=O)(=O)(c1nccs1)NCC1CCC(C(=O)NCCc2ccc(Br)s2)CC1 N1(C(C(C)=CC=C)=O)C(C(=O)NC2(CO)CCC2)CCC1C(C)C c1(C(=O)OC)ccc(NCC2CCC(OC)CC2)c(C#N)c1 CN1CC(NC(C2CCN(C(c3ccc(F)c(F)c3)=O)C2C2CC2)=O)C2(CC2)C1=O c1(C(=O)NC2CC3C(NC(c4ccccc4)=O)C3C2)ccc(F)c(F)c1 C(=O)(C(=O)C(C)(C)CC)N1CCCC(C(N(C2CC(N=[N+]=[N-])C2)CC)=O)C1 N1(CCOCC)C(=O)NC(NC(=O)CC2CCCC(C)C2)C1=O N1(C(CC)=O)CC(C2CCCN(C(=O)C=CCN(C)C)C2)C1 N(C(=NCCCF)NCCC=CBr)C(c1cccc(Cl)c1)C c1(C(C)NC(=O)NCC2(c3ccccc3Cl)CC2)ccc2c(c1)CC(C)O2 C1(C(N(CC(=O)OCC)C)=O)CCN(C(=O)CCOCC(F)F)C(C)(C)C1 c1(C2CCN(c3nnn(Cc4ccc(OCC)nc4)n3)CC2)ccc(F)cc1Cl Cc1nccc(N2CC3CC2C3C(N2CCC2c2ccccc2)=O)n1 CC1(NC(=O)CCSc2ccccc2)CCCN(C(C23CC(CF)(CO2)C3)=O)C1 C1(NC(=O)CCOC2CC2)C2COCC1CN(C(C1CC3CC(=O)C1C3)=O)C2 N1(C(Cc2nc(C)oc2)=O)CC2(CCN(C(C3CCCCC3C(F)(F)F)=O)C2)C1 c1(OC)ccc2ccc(NC(C3CC(C4CC4)=NO3)=O)cc2n1 C1(NC(c2cc(CC)c(C)o2)=O)CC2(CCC(C)(C)CC2)C1 C(=O)(C1CNC(=O)c2ccccc21)NCC1CC(NC(=O)CCC2CCCC2)C1 CCC(CNC(=O)C(C(C)C)NC(=O)Cn1ccnn1)C(C)(F)F c1(OC)ccc(Cl)c(C)c1C(=O)NC1CC(C)(NC(=O)CN(C)C2CC2)C1 c1(C(=O)NCC2C(C)CN(C(c3cscn3)=O)CC2)ccc(C#CC2CC2)cc1 C1(NC(CC(=O)Nc2nccs2)=O)CCOC12CCN(C(=O)C(O)C1CC1)CC2 c1(C(=O)NC2CCC(C)(NC(C(CC)O)=O)CC2)cn2cccc(F)c2n1 C1(NC(C(CC)(F)F)=O)CCN(C(c2cc(C(=O)OC(C)(C)C)n[nH]2)=O)C12CC2 C1(C(N2CCC(O)(COC)C2)=O)CC1C1CCCCC1 N12CCCCC3(C1)CN(C3)C(=O)CC2=O.CC(C(C)C(=O)N1CCC1)S(C)(=O)=O C1(NC(CC(=O)NCC)=O)CCCN(C(=O)CCc2nc(CC)no2)C1C c1(NC(N2C(CN(C)C3CC3)C(C)(C)C2)=O)ccnc2c1ncn2C C1(C(=O)NCCc2c(C)[nH]nc2O)CCCCCN1C(C1CCS(=O)CC1)=O C1(NC(=O)COCC(F)(F)F)CCC2(CC1)CCN(C(C1CC=CC1)=O)C2 C(=O)(C1=CCC(C(F)(F)F)OC1)NCCN(C(c1n(CC#C)ccc1)=O)C1CC1 C(CCC(=O)N(CCNC(=O)CCc1cnn(C)n1)CC1CC1)OCCC c1(C(=O)NC(CNC(C2CCCC(CC)C2)=O)(CC)CC)cncc2c1CCC2 Cc1c(C(=O)NC2CCN(C(c3cnn(C)c3Cl)=O)C(C3CC3)C2)cncc1Cl C1(CNC(CC=C)=O)CC2(CO1)CN(C(=O)CCCC(OC)c1ccccc1)C2 c1(CCC(=O)NC2CN(CC3CC(n4cc(Cl)cn4)C3)C2)ncccn1 c1(COC(C)C(=O)NC2(NC(=O)C=CSc3ccccc3)CC2)cccc(Cl)c1 Cc1cc(C(C(=O)O)NCc2ccc(-c3cn[nH]c3)cc2)cc(C)c1 C(CCCCCNC(C1C2CCCCC12)=O)NC(C1C(C)C1C)=O C1(C(=O)NC2(CNC(C3CC(C)(O)C3)=O)CC(OC)C2)CC2CCC1C2 C1(C(N(c2ccc(F)c(F)c2)C(C)C)=O)CCC2CCCCN12 CC(C)C(C(C)NC(C1CC(N(C)C)C1)=O)NC(c1cncc(O)c1)=O c1(C(=O)NCCN(C(=O)C(C)(F)C(=O)OC)CCC)c(F)ccc(C)c1Cl C#CC1CN(C(C2CCCN2C=O)=O)CCN1C(=O)C=CCOCCOC c1(C(N2CCN(C(C=C3CCC(C)(C)CC3)=O)CC2)=O)noc2c1CCCCC2 c1(C(=O)NCC2(O)CCN(C(C(CC)(F)F)=O)C2)cnc(CC2CCC2)nc1O C(=O)(C(CO)C(C)(C)C)NCC1C(NC(CC(=C=C)C)=O)CCC1 C1(CCCC)CCCC1N=c1[nH]c(=NCc2c(Cl)cccc2Br)[nH]c2c1CCC2 c1(C(=O)NCC(C)CNC(=O)C(C)CC(N)=O)cc2ccccc2o1 N1(C(CC2(C=C)CC2)=O)CCC(C2CN(C(c3ccccc3-n3nccn3)=O)C2)C1 C(CC(C(C)(C)C)NC(=O)C(C)=C(C)C)N(C(C(C1(O)CCCCC1)CC)=O)C c1(C(N2CC(F)(CNC(c3ccc(F)s3)=O)C2)=O)coc2c(F)cc(Cl)cc12 c1(OC)cccc(-c2cc(C(=O)NCCN(C)C(C3CCCSC3)=O)no2)c1 C12(NC(C(CC)OC3CCCCC3)=O)CC(CNC(C3CC3(F)F)=O)(C1)OC2C Cc1nc(S(=O)(=O)N2CCCC(NC(=O)Nc3cc(F)cc(F)c3)C2)cn1C S(=O)(=O)(c1cn[nH]c1)N1CC2(C(C(=O)NCCC(F)(F)F)C2)C1 c1(C(=O)NC(C2(C(=O)NCCCCN3OOC3)CC2)=O)ccccn1 c1(CN(C(C)C)C(=O)Nc2nc(Cl)ccc2Cl)ccc(Cl)c(Cl)c1 N1(C(=O)OCC)CCN(Cc2ccc(-c3onc(-c4scc(C)c4)n3)cc2)C2CC12 C1(C(=O)NCC2C(C)(C)NC(=O)O2)CCCN1NC(=O)C(=O)NC1CC1 N1(C(C2(CC#C)CCCO2)=O)CC=C(C(=O)NC2CCCC(C3CC3)C2)CC1 N1(CC)CCCC1C(=O)NC(C)C(C)(C)NC(C1(OCc2ccccc2)CC1)=O c1(C(=O)NC(C)CCCNC(=O)C(O)CC(F)(F)F)ccc2ccccc2c1 c1(C(=O)NCCCCCN(C(=O)CC(C)(C)C(F)F)C)ccc2c(n1)CCO2 c1(NC(C)=O)ccc(C(=O)NC2CCCC2Cn2cc(CCO)nn2)s1 Cc1c(CO)cc([N+](=O)[O-])c(NC2(C)CC2)c1[N+](=O)[O-].C12CCC(C1)N(C(C)C)C2 c1(C(=O)Nc2c(C)ccc(O)c2)ccc2c(c1)COC(=O)N2 CCC(CNC(=O)C(O)Cn1cncn1)(CC)C(=O)N(C)Cc1nccn1CC N1(C(C(n2ccc(C)n2)C)=O)CCC(NC(=O)CSCc2cccnc2)C1C CC1CN(C)C(C)CN1C(C1CC2CC2N1Cc1ccc(F)c(F)c1Cl)=O c1(C(N2CCC(C)(NC(C(CCSC)OC)=O)C2)=O)ccc(C)c2c1NCCC2 C1(CCOCC#C)(NC(=O)Cc2n[nH]c(C)n2)CCCCC1.C12CCCN1C2=O N1(C(c2cn(CC)nn2)C(=O)NCCCC)CC(C2(O)CCC2)C12CCC2 CC1(C(N2CC(F)(C(=O)NCC(CO)C3CCC3)C2)=O)CCCS1 c1(OC)cnc(C(=O)NC2CN(C(=O)CCCn3cccc3)CCC2O)c(F)c1 N1(CC)CC(C(=O)NC2(CCNC(=O)CC3CCC(=O)N3)CCC2)CC1=O c1(N(C)CC2CC=C(C)CC2)ncc(C)cc1S(=O)(=O)N1CCC1 c1(C(=O)NC2CCN(C(CCCNC(=O)OC)=O)C23CC3)cnc2nccn2c1 c1(OC)ncnc(Cl)c1NC(C1C2CC1N(C(=O)CNC=O)C2)=O C1(CNC(CCC(=C)C)=O)(NC(=O)C(C)CC(C)C)CCC(F)(F)CC1 C1(CNC(C2C(C)CCC2)=O)CN(C(=O)CCCC#N)CCC12CCC2 n1(CCC)ncnc1CNC(=O)C=CC(C)NC(C1CC2CC2C1)=O c1(C(=O)NC(CC(C)NC(c2c(N)ccc(C)c2)=O)C)ccc2c(c1)CCCO2 CCCCCCC(C)C(=O)N1CCC2CCC(C1)N2C(=O)C(C)(C)CCCF C1(CCNC(C=CC=CCC)=O)CCCN1C(c1cc(C)[nH]n1)=O CC1CCSCCN1C(=O)C(CNC(=O)C(F)(F)C(F)F)N(C)C N1(C(C2(CF)CCN(C(CCCCCC)=O)C2)=O)CCC2(COC(=O)N2)C1 C(=O)(C#CC(C)(C)C)N1CCC(c2c(CNC(C3(CCC)CC3)=O)c[nH]n2)C1 C1(NC(c2cc(C)c(C)s2)=O)CCN(C(C2CCCN(C)C2)=O)C12CCCC2 CCC(C)CC(CO)NC(C1(NC(c2ccccn2)=O)CCOCC1)=O C1(NC(C2CN(C)C(=O)N2)=O)CN(C(=O)CCOc2ccccc2Cl)CC12CC2 c1(CONC(C2CC(CNC(CC(CC)C3CC3)=O)OC2)=O)ccc(F)cc1F c1(N(CCCC)C)ccc(C(=O)N(CCC(C)NC(=O)C(C)(C)COC)C)cc1 N1(C(c2occ(C)c2)=O)CCC(F)(CNC(C2CCCCN2C(N)=O)=O)CC1 C(=O)(C(O)C(C)(C)C)N(CCNC(C(CC)C#N)=O)CC1CC1 c1(-c2n(CC3CCN(C)C3)ccn2)ccc(-c2cnn(C)c2C(F)(F)F)cc1F C(c1ccc2c(c1)CCO2)=CC(=O)NC1CC(F)(F)CC1C(=O)O N1(C(C23CC(NC(CCC=C=C)=O)(C2)C3)=O)CCC(O)C(F)(F)C1 C12(C(=O)NC3CC(CNC(=O)CC4=CCCC4)C3)C3CCC(CC13)C2(F)F C(=O)(CCC(CC)OC)NCCN(C(=O)C(C(C)C)c1cccc(Cl)c1)CC CC1(C)CCC=C(C(=O)N2CCN(C(C3C(F)(F)C34CC4)=O)CC23CCC3)C1 c1(C(=O)NC(CNC(CC2C(C)CCC2)=O)C)c(F)c(F)cc(F)c1F c1(C(N(CC(C)(C)NC(=O)C2=CCCS2)C)=O)cnc2ccnn2c1 C(c1cc(F)c(F)c(F)c1)=Cc1onc(OCCOc2ccc(OCC)cc2)n1 c1(CN(C(=O)CSCC(N)=O)N(C(C(F)OC)=O)CCCSC)cccnc1 C#CCCC(O)C(=O)NCCCN(C1CCCC1)C(C1CCCC(F)(F)C1)=O C#CC1(C(N2CCC(C=O)CC2)=O)CCCC1.c1(CCN(CC)C)cn(C)nc1C C(=O)(C(C)CC(C)C)N(C(C(NOCCOCC#C)=O)C)CC=C c1(CNC(C2CC(=O)NC2)=O)cccc(CNC(c2ncc(Cl)s2)=O)c1 c1(N2CCC(C(C)NC(CCCOCCOC)=O)C2)ncc2c(ncn2C)n1 N1(C(C(C(C)(C)C)O)=O)C2CCC1CN(C(=O)CC1OCCCO1)CC2 C1(CNC(C(C2CCOC2)OCC)=O)CC2(CCC2)CN1C(C1COC(=O)C1)=O c1(C(N2CC3(CCN(C(C(CC)F)=O)C3)C2)=O)cc2c(cc1OC)CCC2 Cc1cnn(CCC(=O)NC2CC(NC(C3CC34CCC4)=O)C2)c1 N1(C(CC(C)(F)F)=O)CCC2CCN(C(c3cc4c(cn3)OCCC4)=O)CC12 C12(NC(CCC(=O)NCC)=O)CC(CNC(C3(C)CC3(Cl)Cl)=O)(C1)OC2C c1(C(N2CCC(CCNC(C(C)n3ccnc3)=O)CC2)=O)cc2n(n1)CCCN2 Cn1ncc2ncnc(N3CC(F)CC3C(=O)Nc3ccc(F)cc3[N+](=O)[O-])c12 CCCC(CCNC(=O)C(C)(CNC(=O)CC1CCC(C)CO1)CC)CCC C1(CCCC(=O)NC(C)CC2CN(C(=O)C(F)OC(F)(F)F)C2)CCCC(=O)N1 C1(O)(NC(N(C2(C#C)CC2)C)=O)CCCC1.C1(=O)C=CC(C)N1 n1(CCC(=O)NC(CC)CN(C)C(C2COC2)=O)sc2ccccc2c1=O C1(N(C(=O)CC2CC2C2CC2)CC)CCN(C(=O)C=CC(=O)OC(C)(C)C)CC1 c1(C(C)OC)nc(-c2cncc(-n3cnnn3)c2)n(-c2cccnc2)n1 N1(C(c2cc(C)sc2C)=O)CCCCCC1CNC(=O)CCc1cn(C)nc1C c1(CC)cccc2sc(NC(=O)NCCc3ncc(-c4ccc(F)cc4)[nH]3)nc12 C1(NC(C(CSC)O)=O)CCN(C(c2cc(C)n(C(C)C)c2)=O)CC(O)C1 CC(C(F)(F)C(F)(F)F)=CC(=O)NC(C)CNC(=O)COCCN(C)C C1(C(=O)NC2C(NC(CCOC)=O)C2)CCS(=O)(=O)N1C N1(C(C=CCC(C)(C)NC(C(C2CC2)OCC)=O)=O)CCN(C)CC1C(N)=O N#CC1(NC(=O)Cc2cnc[nH]2)CCN(Cc2cc(F)cc(Cl)c2)C1 N1(C(=O)COCC2CC2)CCC2CCC(C1)N2C(=O)CCCOC1CCCOC1 C1(CNC(c2cc(C(=O)OC)[nH]c2)=O)CC(C)N(C(c2cc(C(N)=O)on2)=O)C1 Cc1nc(NC2CC2)sc1C(=O)NCC1CC2CC2N1C(=O)CC1CC12CC2 Cc1ccc(N)c(C(N2CCC(C(=O)N(C)C)C2c2ccccc2)=O)c1 c1(C(=O)NC2C(NC(CCC(N)=O)=O)CCOC2)cncc2cccnc12 N1(C(C2N(C)CC(O)CC2)=O)CC2CCC(C1)C(NC(c1ccc(F)o1)=O)C2 c1(NC(C2CCN(C(c3cnco3)=O)CC2)=O)ccc(C(F)(F)F)c(Cl)c1 c1(CC(=O)NCCCN(C(c2c(C)cnnc2O)=O)C)ccc2cnccc2c1 c1(C(=O)NCCCCNC(COc2ccc(C)cc2)=O)nn(C)c2c1CCC2 C=CC1(C(=O)NCC2CC(NC(=O)C(CC(C)C)OC)C2)CCCCC1 c1(CC)nc(C)[nH]c1C(N1CCC(C)(CNc2nccc(OC(C)C)n2)C1)=O C=C(C)C1CN(N(C)Cc2ccn(-c3ccc(F)cc3)n2)CCO1 c1(OC)ncc(Cl)cc1C(=O)NCC1CCCN(C(=O)CC2(O)CCCCC2)C1 N1(C(C(c2nc(C)sc2)=O)=O)CCOCC(CNC(C2(C)CC3CC3C2)=O)C1 C1(C(=O)NCC(C)(CO)NC(=O)Cc2n[nH]c(C)n2)(CC)CNC(=O)C1 c1(OCC)cc(C(N2CC3CC3(CNC(C3CC=CC3)=O)C2)=O)oc(=O)c1 c1(C(N2CC(C)C(CNC(C3COC(=O)O3)=O)CC2)=O)n[nH]c2c1CCSC2 CCC(C(=O)OC)C(=O)NCCCN1CCN(C(C2CNC(=O)O2)=O)CC1 N1(C(CC=CC=C)=O)CCCN(C(=O)C(C)=C2CCC2)C(C)C1 N1(C(C2CCN(CC)C2)=O)CCOC2CN(C(C3(C#N)CCCCCC3)=O)CC12 Cn1cnc2[nH]c(C(N3C4CCC3CC(NC(=O)CCC(F)(F)F)C4)=O)cc12 C(=O)(CC(C)C(F)F)NCCN(CC(C)O)C(c1nc(C2CC2)ncc1Cl)=O S(=O)(=O)(c1ccc2nc(N3CCC(C#N)CC3)ccc2c1)N1CCSC(C)C1C C(CCC(C)(C)NC(c1cnc(OC)s1)=O)NC(CC=C)=O c1(C2C(C(=O)NCC(CNC(c3scnc3Cl)=O)CO)C2)ccccc1OC(F)F C1(C(=O)NCC(n2cc(C3CC=CCC3)nn2)C)CC2CCC(C1)O2 C1(C(=O)OC)C2CN(C(c3cnn(-c4ccc(F)cn4)c3)=O)CC12 Cc1cc(N(CC(C)NC(c2ccc(F)cn2)=O)C)nc(C2CCC2)n1 c1(C(N2C(CNC(c3ccc(C)cc3)=O)C3CC3C2)=O)cc2sccc2n1C c1(C(=O)NCC2CC(NC(C(C)=C(CC)C)=O)C(O)C2)ccc([N+](=O)[O-])[nH]1 c1(CC)ccc(C)nc1O.c12c[nH]nc1C(=O)NC(C)(CO)CNC2=O c1(NC(C2(C)CCN2C(=O)CCCCCBr)=O)cccc2c1CC(=O)N2 C1(NC(c2c(CC)n(CC)nc2)=O)CCN(C(=O)CSC2CCOC2=O)C(C)C1 N1(Cc2cn(CC(C)O)nn2)CCCC(NC(C2(C)CC2(Cl)Cl)=O)C1 CC1(C)CCC(CNC(c2cccnn2)=O)N(C(c2cnns2)=O)C1 c1(C(=O)NC(C2(O)CCN(C(C(C=C)C)=O)C2)C)ccc2cc[nH]c2n1 Cc1ccc(C(N2CCC(N(C(=O)C#CC(C)(C)C)CCO)C2)=O)c(=O)n1C C1(CNC(C2(C)CC2(Br)Br)=O)CC(NC(=O)CNC=O)CC1O C1(C(=O)NCC2(OC)CC2)CC(O)CN1C(=O)CC(C)OC C1(C)(C(=O)NCC(CCOC)NC(=O)Cc2ccc(C)cc2C)CC2CCC1O2 c1(COC)ncc2c(n1)CC1CCC2N1S(=O)(=O)C1CCN(CCF)C1 Cc1ccc(C(=O)NC2CC3CC(NC(C4OCCN(C)C4=O)=O)C2C3)c(O)n1 Cc1nc(O)[nH]c1C(=O)NC1(C2CCCCN2C(=O)CC2C(C)(C)C2(C)C)CC1 Cc1cnc(C(=O)NC2(C(N3CCC(CC(C)C)CC3)=O)CCCC2C)cc1C C(=O)(C1=CCC2(COC2)OC1)N1CCC(C)(CNC(Cc2cccc(C)c2)=O)C1 CC1CCCCC1CNC(C1CCN(C(c2cncc(N(C)C)c2)=O)CC1)=O N1(C(c2c(C)n[nH]c2)=O)CC(NC(c2cccc(C(F)(F)F)c2C)=O)C(C)(C)C1 c1(C(=O)NCC(CNC(C2CCSC2)=O)C(F)(F)F)cnnc2ccccc12 c1(C(Cn2cc(CC3CCN(C(C4(C=C)COC4)=O)C3)nn2)O)ccc(F)cc1 N1(C(c2cn(C)nc2)=O)CCN(Cc2conc2C(F)(F)F)CC1 c1(CC2C(C)CCO2)cccc(NCC(C)(C)C2CCOC2)c1 c1(C(=O)NCCCNC(c2cnc(Cl)[nH]2)=O)cnnc(-c2ccccc2)c1 c1(C(=O)Nc2c(C(C(=O)OC)NC(C)=O)cccc2)ccc(SC)c([N+](=O)[O-])c1 C1(CC)(NC(=O)Cc2occc2C)CCN(C(C2(C(F)F)CCOCC2)=O)CC1 C=C(C)CCCOC1CCN(C(N2C(C(=O)OC(C)(C)C)CCC2)=O)C1 N1(C(C2(OCC)CC2)=O)CCCC(C2CCN(c3c(C#N)cccc3[N+](=O)[O-])C2)C1 c1(CCN2CCC(COC)C2)cccc(CN2CC3C(NC(CCOC)=O)C3C2)c1 C1(NC(c2c(C)ccn2C)=O)CN(C(=O)C2=COCCO2)CC1N=[N+]=[N-] c1(C(CNC(C(C)C)=O)NC(c2cc(-c3cccs3)[nH]n2)=O)cccc(Cl)c1 N1(C(CC2(C)CCOC2)=O)CC2CC(C(=O)NCCCCCCC3CC3)C(C2)C1 c1(C(=O)NC(c2cn(Cc3cc(C)on3)nn2)C)onc(Br)c1C N1(C(C(C)(C)C(F)(F)F)=O)CCCC(C2CC2NC(=O)C2=CCCCO2)C1 c1(C(=O)NCC2N(C(C=CC(CC)=CC)=O)CC2)nc2sc(C)cn2c1C Cc1cncc(C(=O)NC(c2cn(C)nn2)C(=O)NCC2CC2Cl)c1 c1(NC(C2N(Cc3cccc(C)n3)CC2)=O)ccc2c(Br)nn(C)c2c1 Cc1ccc(N)c(C(=O)N(CCCCNC(c2cnn3ncccc23)=O)C)c1F N(C(=NCC1CC(C)(C)CO1)NC1CC1)CC1CN(CC)C(=O)C1 c1(C(N2CC3C(Nc4nccc(C(=O)OC)n4)C3C2)=O)ccc2ccnn2c1 C=C1CC2CC1CN2C(=O)CN(C(=O)C=C(C)C1CC1)C C12(CNC(C3C(C)C3)=O)CC(NC(C3CN4CCC3CC4)=O)(C1)C(C)O2 c1(C(c2nnnn2CCCCCC)NCCC(CCC)O)c(F)ccc(Br)c1C Cc1ccc(C(CNC(=O)C(C)O)NC(=O)C(C)(C)c2ccno2)cc1 CCC(C)C(CC(=O)NCc1ccnc(O)c1)NC(=O)CC1CC(=O)C1 c1(NCC(=O)NC(C(=O)NCC)C)ccc(Br)c(OC)c1 c1(C(=O)NC2(CO)CCN(C(CC(CC)C)=O)C2)ncc(C#N)cc1Cl C1(C(=O)NC(CC)C)C=CCN(C(c2cc(Cl)cn2C)=O)C1 Cc1ccc2c(c1)CCC(C(=O)NC(C)CNC(C13CC(F)(C1)C3)=O)O2 N1(C(C(C)(O)C2CC2)=O)CCN(C(=O)Cc2cccc(F)c2F)CC1CF C(C(CC(C)C)C(=O)N1CC(C(O)C(=O)NC2CCC3CCCC2O3)C1)OC N1(C(Cc2nc(C)sc2Cl)=O)CCCCC12CN(C(C1CCSCC1)=O)C2 C(C)(C(C)(C)C(=O)NCCC1(OC(C)=O)CCC1)NC(CC1CC(SC)C1)=O C1(C(=O)NCCC2CN(C(c3cncc(C)n3)=O)C2)Cc2nccn2C1 C(CCCC(C)(C)NC(=O)C(C)O)NC(c1ncc(CC)cn1)=O CC1(C(=O)NC2C3CN(C(=O)COC4CCCCCC4)CC23)CS(=O)(=O)C1 c1(C(CNC(C(CC)NC(C)=O)=O)Nc2nocc2Cl)ccccc1F.C1CO1 C(=O)(C1=CC2CCCCCC12)N1CCC(CCNC(c2cccnn2)=O)CC1 C1(O)(C(=O)NC2CCC(NC(C3(CO)CC3)=O)CC2)CCCCCC1 CN1CCC(C(=O)NCC(c2ccccc2)NC(c2cc(CCCO)on2)=O)C1 Cc1ncc(CC(=O)NCC2C(C)CCN2C(=O)CC2(C)CC(F)(F)C2)c(O)n1 C1(C#N)(C(=O)NCC2C(CC(=O)NCC(C)(C)F)C2)CCCOC1 CC1CN(C(C2CCN(C)CC2)=O)CC1CNC(c1ccc(-c2cccs2)o1)=O N1(C(c2c(C)[nH]nc2C(C)C)=O)CCC2(C1)CN(C(c1nnsc1N)=O)C2 N1(C(CCC(=C)Cl)=O)CCC2(CCC2NC(=O)CC2=CCCCC2)CC1 S(=O)(=O)(c1ccc(NCCC2CCC3CC23)c(C#N)c1)N1CC(C)OC1 c1(CC(=O)NC(C2CCN(C(c3cncc(CC)c3)=O)C2)C)cc(C)ccc1C c1(C(=O)NC2CC(CNC(C3(C)CCCC3(F)F)=O)C2)ccc2c(c1)CNC2=O S(=O)(=O)(c1ccccn1)N1CC(CNC(c2cc(OC)c(O)cc2)=O)OCC1 Cc1cc(C)c(OCC(=O)Nc2ccc3nnnn3n2)c(C)c1 CCC(C)(C)OCC(=O)C(=O)CN1CCC1C.C(CCSC)N c1(C(=O)NCC(C)NC(C)=O)c(Cl)ccc(Cl)c1O C1(O)(CNC(C2CCN(CC)C2)=O)CCN(C(=O)C(F)=C2CCCC2)C1 c1(CS(C)(=O)=O)ccc(NC(C2CC3CC3N2C(c2cn[nH]c2)=O)=O)cc1 c1(CC)cn2c(n1)CCC(C(=O)NC1(C3CN(C(c4ccncn4)=O)C3)CC1)C2 C1(CC(=O)NCC2CCN(C(=O)Cc3ncc[nH]3)C23CC3)CCCC2(CCC2)O1 c1(NCCCNC(C2CC(OC)(OC)C2)=O)ccccc1SCC(=O)OC C1CN(C)CCN(C)C1.C(CCF)(C(=O)N)NC(c1c(CC)ncs1)=O CC#CCC(C(=O)NCC1CC[Si](C)(C)C1)NC(=O)C(O)C=CC C1(C(=O)NCCC(C)CO)C2CC3C(C2NC(C24CCN(CC2)C4)=O)C13 C1(CC(N2CC(C)(CCC(=O)NCC(C(C)C)O)C2)=O)CCCOCC1 Cc1cc(Cl)c(C(=O)NCC(C)(C)CNC(C2(C(O)C(F)(F)F)CC2)=O)cc1F Cn1nc(C(=O)NCC2(F)CCC(NC(=O)C=CS(C)=O)C2)cc1Cl N=c1nc(O)cc(NC(=O)NC(COC(F)F)C2CC2)[nH]1 N1(C(c2occ(C)c2C)=O)C(CNC(c2coc(Cl)n2)=O)CC2CCCC12 N1(C(Cn2nc(C)oc2=O)=O)CC23CCCCC2(C1)CN(C(C1CC1(Cl)Cl)=O)C3 N#Cc1cccc(CNCC(c2ccccc2Cl)O)n1 c1(OC(CC)C)ccccc1C=CC(N1CC=CC(NC(C2CC2F)=O)C1)=O C1(C(=O)NCC2N(C(CC3CCC(OC)CC3)=O)CC2)Cc2cscc2C1 C1(NC(C(C)OCCC#C)=O)CC(C)(CNC(c2ccccn2)=O)C1 C1(CC)CN(C(=O)CC2CC(CC)C2)CCC1NC(=O)C(C(C)C)SC CS(=O)(=O)c1cncc(NCC23CCC(CN)(CC2)CO3)n1 C=CCCC(C(=O)N1CCN(C(C)=O)CC1)NC(C1(CC=C)CCCC1)=O C1(NC(=O)CN2CCC(F)(F)C2)COC2(C1)CN(C(=O)CC1CC3CC3C1)C2 C1(CC)CN(C(=O)CCC2(C)CC2)CCN1C(=O)Cc1nnc(C)o1 CC(C(=O)NC(C1(C(N2CC(O)(CC3CC3)C2)=O)CCC1)=O)C(F)(F)C(F)F Cc1nn(C)c(Cl)c1C=CC(=O)NCC1CCN(C(c2ccccn2)=O)C1(C)C c1(C(N(C2CN(C(C(C)OCCC=C)=O)CC2(C)C)C)=O)ccnc2[nH]nnc12 N1(C(C2CCCCN2C(=O)C=Cc2cscn2)=O)CCOC2(CC2)C1 N1(C(CCN(C(C)(C)C)CC2CCOCC2)C)CCCC(C(=O)OC)CC1 c1(NC(C2N(Cc3ccc(C(=O)OC)cc3F)CCC2)=O)cnc2cccnn12 N1(C(CCCC#C)=O)CCCC2(CCCCN2C(C23CC(C(F)(F)F)(C2)C3)=O)C1 C1(C(=O)OC)CCCCN1CCN(C)C(=O)OC(C)(C)C.C1(C)(C)C(=O)N1 N1(C(COCCNC(C(CCC)OC)=O)=O)CCC(C)(COC)CC1 Cc1cccc(C)c1-n1cc(C2(F)CN(C(c3cccc(I)c3Cl)=O)C2)nn1 C12CCCC(C1)OC(=O)OC=CC(=O)N1CC(C1)N(C)C(=O)N2.C(C)(C)(C)OCC c1(C(=O)OC)cc(CN2CCN(C(CC(=O)NC(C)(C)C)C)CC2)nn1C C1(C(=O)OC)CC(F)(F)CC1C(=O)NC1CCCN(C(C2(CO)CCCC2)=O)C1 CC(CN(C)C(c1coc(C(C)NC(c2ccnnc2)=O)n1)=O)C(C)(C)C C=Cn1ncc(C(N2C(C(N3CC4CC3(C(N)=O)C4)=O)CCC23CC3)=O)c1N Cc1ccc(C(=O)NC2CC2NC(=O)C(C(C)C)N2CCCC2=O)c(C)c1 c1(C(=O)NC(C)C)cc(-c2csc(NCC3CCSCC3)c2)ccc1F C1(S(C)(=O)=O)(C(=O)NC(CCCNC(CC(C)C)=O)C)CCCCC1 C12(C(=O)NC(CC)C(C)C)CC(CN1C(=O)Cn1cnc(C#N)n1)C2 C1(O)(C(C)NC(=O)CSc2n[nH]c(O)n2)CCN(C(=O)CC2CNC(=O)C2)C1 C1(CC(=O)NCCCn2cc(-c3c(C(=O)O)scn3)nn2)CCCC(F)(F)C1 C1(CC)CCN(C(=O)CCOC2CC2)C(C(N2CCC=C(C)C2)=O)C1 c1(OC)ccc(C(N2CC(C(C)NC(=O)CC3(C)CC3)C2)=O)c(F)c1Cl N1(C(C(COC)(F)F)=O)CCC(CO)(CNC(=O)CCc2nncs2)CC1 c1(-n2c(C(F)C(F)(F)F)nc(CCC(C)(C)C)n2)ccc(S(N)(=O)=O)cc1 c1(CC)cc(CC)nc(NC2(CNC(=O)C(CC)OC)CCCCC2)n1 N(C1CN(C(C2(C)CCCOC2)=O)Cc2ccccc21)c1snc(CCOC)n1 C1(OC)CN(C(c2cncs2)=O)C(C)(CNC(=O)CC#N)C1 CN1CCC2(CN(C(c3cnn(CC(F)(F)F)c3)C(=O)NC3COC3)CCO2)C1 C1(O)(C(C)C)CCC(NC(c2cnn(C3CC3)c2Cl)=O)C1 C(C(=O)N1CCCC(CNC(=O)Cn2ccccc2=O)C1)(C(C)C)OC C1(NC(C(C2CCCN(C(C3CC(N=[N+]=[N-])C3)=O)C2)C)=O)CN2CCC1(C)CC2 C1(CC)CN(C(=O)Cc2c(Cl)cnn2C)CCN1C(=O)C(C)c1cncs1 N1(C(c2cc(COC)no2)=O)CCC(O)(CNC(=O)CC2CCCC2)C1 C(C)(CNC(C1CC(N2CCCC2)C1)=O)(CC(C)C)NC(c1c(C)ocn1)=O C(C)(C(=O)NCCCOCCCNC(C1CC1C(C)(C)C)=O)OC C1(NC(C2CCN(CC#C)CC2)=O)CC(O)CN(C(=O)C(COC)NC(C)=O)C1 C1(C(N2C(CCNC(c3cscc3Cl)=O)CC(OC)C2)=O)CN2CCN1CC2C CCC(CC)C(F)C(=O)N1CCC(C(F)C(N2CC(CO)CC(C)(C)C2)=O)C1 c1(CCC(=O)NCCCCCCNC(C(C)C2CCC2)=O)ccc2[nH]ccc2c1 C=CC1COCCN1C(C1CCCC1NC(C1CCCCS1)=O)=O CCC(C)C(O)C(=O)NCc1ccc(C(=O)N(C)CC2CCCN2C)o1 Cc1cc(C(N2CC(CNC(c3cncnc3)=O)C2)=O)c(Br)cc1F c1(OCCCC(=O)NC2C(CNC(CC3(C)CC3)=O)CCC2)ccccc1F Cc1cnc(C=CC(=O)NC2CCCC2NC(=O)COC2CCC2)[nH]1 N1(C(c2c(C)cns2)=O)CC(C(F)(F)F)C(CNC(C2CCCCC2)=O)C1 C1(NC(CCCOCC)=O)CC2CN(C(=O)CC(CC)C3CCC3)CCN2C1=O C(CCC(O)C(=O)NCc1cnn(C)c1O)NC(c1ccc(SC)o1)=O CCC(CC(=O)NC(C12CCC(CC1)C2)CNC(=O)CN(C)C)NC(=O)CSC N1(C(c2cc(CC)no2)=O)CC(CNC(=O)CCc2cnc(O)[nH]2)C(C)C1 C(CNC(=O)CCC1CCCCCC1)(CC(F)(F)F)NC(COCC#C)=O CC(CCNC(=O)CC1(C)CCCO1)CCNC(c1coc(Br)n1)=O C1(C(N2CC(C(=O)NC(C(=O)OCC)CC)C2)=O)CCC2(CCC2)O1 N1(C(CSc2n(C)cnn2)=O)CCC(NC(c2ccon2)=O)C(F)C1 N1(C(C2CC(OCC)C2)=O)CCC(N(C(=O)CCN2CCC2)CCO)CC1 CCC(C)N=c1[nH]c2c(c(=NCCOC(F)(F)C(F)(F)F)[nH]1)CC(C)CC2 c1(OCC)cc(C(=O)NC2CCC(CNC(c3cnc(COC)s3)=O)C2)on1 C1(NC(CN2CCC(C)CC2)=O)CCCN(C(c2cc[nH]c2C2CC2)=O)CC1F C1(NC(C(=O)NC(C)CCC2CCCO2)=O)(CO)CCOCC1 c1(C(N2CCC(C)(NC(C(C(C)(C)C)SC)=O)CC2)=O)cnn2c1OCC(F)C2 c1(C(N(CCNC(C2OCCC(C)C2)=O)C)=O)nn(C)c(Cl)c1Cl C1(NC(CC(C)N(C)C)=O)CCCCC1NC(=O)Cc1cnco1 C=C(Cl)CC(C(=O)NCC(C)(O)C1CCCC1)NC(=O)C(C)CO N1(C(CC(=C)C)=O)C2CCCC1CN(C(c1cccnc1NC(C)C)=O)C2 C1(N(C)C(c2cccnc2O)=O)CCCN(C(c2cnc(Cl)s2)=O)CC1 N=C1NC(=O)C(CC(=O)NC2(CNC(C3(O)CCOCC3)=O)CCCC2)S1 C1(NC(C2CC(=O)NC2)=O)CCCCN(C(C23CCCN2CCC3)=O)C1 c1(C(=O)NCC=C2CCN(C(c3c(C)nc[nH]3)=O)CC2)nc2ccccc2[nH]1 N1(C(c2ccncn2)=O)CC2(CC(C(N3CCC4CC34)=O)CO2)C1 C1(C(=O)NC(C2CCN(C(C(CC=C)(F)F)=O)C2)(C)C)CCc2ncncc2C1 N1(C(C2C(CCOC)C2)=O)CCC2C(C(=O)N(C3CC3C)C)C2C1 C1(OC)CCn2cc(C(=O)NC(CNC(=O)C=Cc3nccs3)C(C)C)nc2C1 CC1CCCC(C)N1C(C1CCCN(C(c2cscc2Br)=O)C1)=O N1(C(c2c(CC)n(C)cc2)=O)CC2CC(C1)N2C(C1(C(C)C)CCC1)=O c1(CCC(=O)NC2(CN(C(=O)CC3CC(CF)C3)C)CC2)nnc(N)[nH]1 C(CCCCNC(=O)Cc1cnc[nH]1)N(C(=O)CSCc1ccccc1)C O=C(C1=CCOC1)NCC(O)COc1ccccc1.C12CCC13CC23 C1(NC(C2CC(OC)C2)=O)CCC(NC(=O)CC(O)CC2CNC(C(C)C)C2)CC1 N1(C(c2c(CC)ncs2)=O)C2CCC1C(CNC(c1cc(C)c(Cl)s1)=O)C2 Cc1nn2ccccc2c1C(=O)NCCCNC(=O)C=CC1CCCO1 c1(OC)ccc2c(n1)NC(C(N1CCC(C(C)NC(c3nocc3C)=O)C1)=O)C2 C(CN=C(NCc1nc(C(N)=O)cs1)NC(C)C1CC1)(C1CC1)OC C(CC(C)(C)CC(=O)NCC1CC1CC(N1CCCC1C)=O)OC C1(C(N2CC(OC)(CNC(=O)CCCC3CC3)C2)=O)CCCCN1S(N)(=O)=O C(C(C)(C)CC(=O)NC(CO)CCO)NC(C(COC)OC)=O C#Cc1ccc(C(N2CC(O)(C(C)NC(c3cnn(C(C)C)c3)=O)C2)=O)cc1F C1(C(=O)Nc2ccc(C)c(O)c2)(CC)CCCN(C(=O)C(C)C(C)(C)C)C1 C1(NC(c2cccc(Cl)c2)=O)CC2CCC1N(C(=O)CCN1CCCC1)C2 c1(CC)ccc(CC(=O)N(CC(O)CN(C(=O)C(C(C)OC)N(C)C)C)C)cc1 C1(C(=O)NC2(C)CC(NC(c3ccncc3Cl)=O)C2)CCc2nc[nH]c2C1 C(=O)(CCCC(C)(C)C)NC12CN(C(Cc3c(C)nc(S)s3)=O)C(C1)CO2 N1(C(C(CCC)C)=O)CCC2(CCOCC2)C(NC(=O)C(CC(C)C)OC)C1 N(C(=NCCC(=O)N(C)C)N1CCC(CS(C)(=O)=O)C1)CC(C)C c1(CN2C3CN(C(c4n(C)nnc4)=O)CC2CC3)cc([N+](=O)[O-])c(Cl)cc1F C(=O)(C1=NOC(CNC(c2cccc[n+]2[O-])=O)C1)N(CC(C)(C)O)CC N1(C(C(C=C)OC)=O)CCC12CN(C(=O)CC1CCCN1C)C2 CCCS(=O)(=O)CC(=O)N1CC2CCOC2(CNC(C2CC2(C)C)=O)C1 n1(C(CC)C)cc(CNC(=O)Nc2cc(-c3ccncc3)[nH]n2)nn1 N1(C(c2cncc(OC)c2)=O)CC(C2CN(C(=O)CC3CC34CC4)C2)C1 C[Si]1(C)CCN(C(C2C3CCC2(c2ncco2)C3)=O)C1 c1(CC(=O)N(CC)CC2CCCN2C(=O)COC(C)C)ccc(F)c(Cl)c1F c1(C(=O)Nc2c(OCCOC)ccc(F)c2)cc2ccc(O)nc2s1 O=C(C1=CCCCCC1)N1CC2C(C1)N2C(C1CC12C(=O)Nc1ccccc12)=O c1(C(N(CCCNC(=O)CCc2ccoc2)C)=O)cc(F)cc([N+](=O)[O-])c1 c1(C(N2CCC(C)C2CNC(C2C3(CC3)C23CC3)=O)=O)nc2cc(O)ccc2[nH]1 c1(C(N(CCC(C)NC(c2cn(CC)nn2)=O)C)=O)cccc(N)n1 C1(NC(c2ccc(CC)cc2)=O)CCN(C(c2csc(CC)n2)=O)CC1O CCC(CO)NC(CCC1CCCC1)C1CC1 c1(NCC(CC)(C)c2cnccn2)ccc(F)c(OCCN2CCCCC2)c1.OCC C(C1=CCCN(C(=O)C(=Cc2ccccc2)C)C1)NC(CN(C(C)=O)C)=O C1(CN(C(C(CC)OCC)=O)C)CN(C(=O)CC2(C)CCCO2)CCO1 c1(C(N2CCN(CCO)CC2)=O)cnc(OCC(F)(F)F)cn1 Cc1cnccc1CN(C)C(c1ccc(CNC(=O)CC2CC2C2CC2)nc1)=O C1(C(N2CC(N(C(c3c(C)nn(C)c3C)=O)C)C2)=O)COc2ccc(F)cc2C1 c1(C(N2CC3C(CNC(C(CC)CO)=O)(CC3)C2)=O)ccnc2ccccc12 C1(C(C)C)CCC(C)N(C(C23CC(CO)(C2)OC3C)=O)C1 C1(C(=O)NC(C=C)(C)C)CN(C(C2CC23CCOCC3)=O)CC12CCC2 c1(OC)ccc2cc(CN3CC4C(C3)N4C(=O)CCCCCl)ccc2c1 C=CC(C)(O)C(=O)NC1CCCC(NC(=O)C(F)(F)C2CC2)C1 C(c1cccc(O)c1)=CC(=O)NC1(CCCNC(=O)CC2(O)CCCOC2)CC1 c1(C(=O)NC2CN(C(c3c(C)nc(CO)o3)=O)C(C)C2)cnc2ncnn2c1C C(=O)(C#CC1CCCO1)N1CCC(F)(CNC(=O)C=Cc2cnc[nH]2)C1 c1(C(=O)NC2CN(C(C(CNC(C)=O)(C)C)=O)CC2(C)C)ccc2cncn2c1 c1(C(N(CCOC)CCNC(C2CC(C)(C)CO2)=O)=O)noc2ccccc12 c1(C(N(C2CCCC2)CCNC(C=CCCC)=O)=O)cc(CSC)on1 N#CC1=C(C(=O)NCC2CCC(NC(c3cnc(C4CC4)nc3)=O)C2)CCC1 C1(OCC)CN(C(=O)CNC=O)CC1C(=O)NCC1(O)CC1 c1(C(=O)NCC2CC(C)N(C(=O)CC(C)(O)C3CC3)C2)ccc2cccnc2c1 C1(CC#C)(C(=O)N(C)CCN(C)C(C2CN(C3CCC3)C2)=O)CCOC1 N12CC3C(C3C1)NCC2=O.C1(NC(CNC(=O)NC)=O)CC(C(C)(C)C)C1 CCC(CC(=O)N1CC=CC1(C)C(=O)NCC1(O)CC(C)(C)C1)C(C)C n1(CCOC)nc(-c2ccc(F)cc2)nc1-c1ccc(CC(C)C)s1 C1(NC(c2c(OC)ccs2)=O)CC(NC(C23CC(C2)C3)=O)CC1O N1(C(CCCC)=O)CC(CNC(=O)C(C)(O)CC)OC2(CCC2)C1 CCCN=C(NCc1cc(F)ccc1CS(C)(=O)=O)NCc1nnnn1CC N1(C(C23CN(C(CCC(C)SC)=O)C(C2)CO3)=O)CC2(CCC(O)CC2)C1 Cc1cc(C(=O)N(C)CC2CN(C(C3CCCCS3)=O)CCO2)c(C)nc1C c1(C(=O)NCCC(C)N(C(=O)C(C)CC(F)F)C)cnc2sccn12 CCCCCCCC(=O)N1CC(O)CCC1C(=O)NCc1nnc(O)n1CC c1(CCC)cc(C(=O)NCCC(C)N(C(=O)CC(F)(F)F)C)nn1C C=CCCCC(=O)NCCC1CCCN1C(c1cc(Cc2ccccc2)c[nH]1)=O N1(C(C(C)NC(=O)OC)=O)CCOCC(C)(CNC(=O)CCc2cc(C)[nH]n2)C1 N1(C(C2C(=C)C2)=O)CCCC(CNC(c2ccc(CC(C)C)cc2)=O)C1 C1(CNC(=O)CONC(=O)C2CC(OC(F)F)C2)CC2CCCC2C1 N1(C(CCCC#C)=O)CCN(C(c2cc(C(C)=O)c[nH]2)=O)C(COC)C1 C(=O)(C1CCCc2ncnn21)N1CCC(NC(C2CCOC2)=O)C(O)C1 C1(C(C)C)(C(=O)NC(CCO)C(C)C)CCCN1C(c1csnn1)=O N1(C(C2C(=C)C2)=O)CC=C(CNC(=O)C(CN(C)C)c2ccccc2)CC1 c1(CNC(=O)NC(c2nc(CC)on2)C)ccc([N+](=O)[O-])c(F)c1 C1(NC(c2cn(C(F)F)cn2)=O)CC2(CCN(C(=O)C=C3CCSCC3)CC2)C1 CC(C)(CC1CCC1)C(=O)NCCC1(O)CCN(C(=O)C=Cc2cc[nH]n2)C1 C1(F)(c2ccc(OC)cc2)CCN(N2CCn3c(nc(OC)c3Br)C2)C1 C1(C(=O)OCC)(COC)CN(C(=O)OC(c2ccccc2)C2CC2(C)C)C1 c1(NCc2ccc(CNC(c3cc(CC)n(C)n3)=O)cc2)ncnc2scnc12 N1(C(c2c(C)c3c(cc2)C(=O)CC3)=O)CCc2ccccc2C1C C(C)(C(=O)NCC1(NC(=O)CCc2ncccc2C)CCCCC1)(C(C)C)OC Cc1nn(C)c(Cl)c1CN(C)C(C1CC1(c1ccc(Br)cc1)F)=O CC1CCC(S(C)(=O)=O)CN1C(c1ccc(=O)n(-c2ccc(F)cc2)c1)=O N1(C(CCC(=O)NC)=O)CC2(CNC(=O)Cn3c(C)cc(O)cc3=O)CC(F)(C1)C2 C(c1cccc(Br)c1)=CC(=O)NCC(C)=CC(=O)NCC1CCC(C)N1 Cc1cc(C)c(C(=O)NC2(C(=O)NC(CO)CC(C)(C)C)CC(F)C2)cn1 c1(C(C2CC2)NC(C2N(C(C(CC)C)=O)CSC2)=O)ccccc1COC c1(C(=O)NCCN(C)C(c2cc[nH]c2)=O)n[nH]c(C2CC2)c1Cl Cc1ccc(CN2CCC(n3cc(COC(C)CC4CC4)nn3)C2)cc1 c1(CNC(Cn2c(C)cc(C)n2)=O)cc(O)nc(CNC(=O)C(C)NC(N)=O)n1 C1(CCCOCC2(CO)C(C)(C)C2)CS(=O)(=O)CCO1 CC(C)CC(O)C(C)C(=O)NC1C(C(N2CCC(O)C(C)(O)C2)=O)C1(C)C c1(C(=O)NCCC(C)N(C(CC2CCC(CC)CC2)=O)C)cnc(CO)nc1C N1(C(C(CC)CCOC)=O)CC(C)CN(C(c2ccc3nc[nH]c3n2)=O)CC1C N1(C(C)=O)CC2CC2(C(N2CC3CC3(NC(=O)CCc3cc(C)on3)C2)=O)C1 c1(C(N2CCN(C(C(CC)=CC)=O)CC2COC)=O)cnc(O)c2ccccc12 CC1CN(CCO)CC1(c1nnnn1C1CC1)Nc1c(Cl)nsc1Cl c1(C(=O)NCC=CCNC(C(CC)n2nccc2C)=O)cc(SC)ccc1C C(=O)(C(O)CCCC)N1C(C(N2C(CCC)COCC2)=O)CSCC1 c1(C(=O)NC2CC3(C(C(N(C4CCCCC4)CCC)=O)C3)C2)ccc(C)nc1C C1(NC(c2ccc(SC)cc2)=O)CC2CC1CN(C(=O)CNc1cccnc1)C2 N1(C(c2cnc(C(C)C)o2)=O)CCCCCCC1C(=O)NCCCOCCCO c1(OC)cc(CCOC(c2ccc(CCS(C)(=N)=O)cc2)=O)cc(OC)c1OC C(=O)(C1=CCC2CCC1N2C(c1ccnn1C)=O)N1CCC(SC)CC1 c1(CNC(c2cc(CC)oc2C)=O)ccc(CNC(C2(C)CC(C)C2)=O)c(F)c1 CC#CCC(C)N=c1nc(N2CCC3(CC2)CC3(F)F)c2c([nH]1)CCC(C)C2 C12(CNC(C3(CC#C)CCOCC3)=O)CCC(C1)N(C(C1CCCCS1)=O)C2 C(C)(CNC(=O)Cc1csc(C)c1)(CC(C)C)NC(C(CC)OCC)=O C1(CNC(=O)Cn2cccn2)CC2CCC1N(C(c1ccc(CO)o1)=O)C2 N1(C(c2cc(C(=O)OC)ncc2)=O)CCCC(CO)(NC(=O)CC(C)N(C)C)C1 C1(CC(=O)NC2(C)C(NC(Cn3nc(C)oc3=O)=O)CCC2)CCC(C)(C)CO1 C1(NC(C2CC2C2CC2)=O)CN(C(c2cc(I)ccc2F)=O)CCC1(F)F c1(NCC2(NC(C3CC4CCC3C4)=O)C(C)CCCC2)ncnc(Cl)c1[N+](=O)[O-] n1(C(CC)CC)nccc1C(=O)NCC(C)(O)CNC(=O)CC(C)OC C(=O)(C(C)C(=O)N1CCCC(NC(c2n[nH]cc2OC)=O)C1)OC C1(NC(c2c(CNC(=O)CCn3cnnn3)cc[nH]2)=O)CC2CC3C(C2)C13 C1(CC)CN(C(C2(C)CCCS2(=O)=O)=O)CC(C)N1 C1(C#N)(CC(=O)NC(CN(C(c2ccnc(C(C)C)n2)=O)C)C)CCOCC1 O=C1CCC(c2ccn(NC(=O)CC(F)(F)F)n2)CN1.C12CCCC1C(=O)N2 C(Cc1cn[nH]c1)(C(=O)N1CCCC1CC(N)=O)NC(CC1(C)CC1)=O CC1CC(NC(=O)C=Cc2cn(C)nn2)CN(C(c2ccc(N)c(F)n2)=O)C1 Cc1ccc(O)c(C(N2C3CCC2C(C(=O)NC2(C)CCC(C)C2)C3)=O)c1 N1(C(C2CCC(C3CC3)CC2)=O)CCC2OCCN(C(=O)COCC3CC3)C2C1 n1(CC)ncc(C(=O)NCC(C)CN(C)C(c2oc(C3CCC3)nc2C)=O)c1C N1(C(C)=O)CCCC(NC(=O)C(CC2CC2)NC(=O)Cc2cnn(C(C)C)c2)C1 N1(C(c2cc(OCC)n[nH]2)=O)CC(CO)C2(C1)CN(C(=O)C(F)CCC(C)C)C2 CCCCC(CC(=O)N1CCC(C)(CC)CC1)NC(c1coc(C)n1)=O C(CC(C)(C)CC(=O)N1CCN(C(=O)C(C)C)C(C)C1)OC C1(NC(=O)CC2(O)CCC2)CCN(C(=O)CCc2nc(CC3CC3)no2)CC1O N1(C(C2CN(CCC)C(=O)C2)=O)CC(CO)C2(C1)CN(C(=O)Cn1ccnn1)C2 C=CC1(CC(=O)N(C)Cc2nnc(CC)o2)CN(C(=O)CCCC2CCCO2)C1 C(=O)(C(C)CC(=O)OC)NC(CC(=O)NC(CCOC)C)CC1CC1 C#CCCCC(C)C(=O)N(C)CCNC(c1cc(O)cc(F)c1F)=O N1(C(C(C)S(N)(=O)=O)=O)CCC(CNC(=O)CCC(F)F)C(F)(F)CC1 Cc1cc(CC(=O)NC2CS(=O)(=O)CC2NC(c2cnc(S)n2C)=O)cc(F)c1 c1(C(=O)NCC=CCNC(C2C(CC)C2)=O)ccc([N+](=O)[O-])cc1C(F)(F)F c1(CC(=O)Nc2cccc(-c3ccco3)n2)cn2cc(-c3nccs3)ccc2n1 C1(NC(CC(COC)C)=O)CC(N=c2[nH]nc(CO)s2)C12CCOCC2 N1(C(C(CC)CC)=O)CCN(C(=O)Cn2[nH]cnc2=N)CC2CCCCC12 CC(c1ccccc1)=CC(=O)NC(C)CCCNC(c1cocn1)=O c1(C(CNC(C(C)N(C)C)=O)NC(=O)CCc2cn[nH]c2)ccc(F)cc1F Cn1ncc2cc(C(N3CCC(NC(C4CSCC(=O)N4)=O)C(F)C3)=O)cnc12 N1(CCC(=O)NC2C3CN(C(C(C(C)C)SC)=O)C2C3)Cc2ccccc2C1=O c1(C(C)NC(CC(C)C)c2ccccn2)ccc(OC(C)(C)C)cc1 N1(C(CCCOCC)=O)CCN(C(C2ON=C(C)C2C)=O)CC1c1cnn(C)c1 C1(C2CCN(C)CC2)(C(=O)NCCCN(C(=O)CCCC(C)(C)C)C)CC1 N1(C(C(CC=C)CC)=O)CCC(C)(C)C(C(N2CCC(OC)C2C2CC2)=O)C1 c1(CC)cc(C(=O)N(CC(C)NC(C2CCC=CO2)=O)C)c2c(c1)CCO2 C(CCC(C)C)(C(=O)N1CC2(CCC2)C1C1CC1)NC(c1c(OC)noc1C)=O N1(C(c2cn(C3C(OCC)COC3)nn2)=O)CCN(CCC(Cl)Cl)CC1 CCC(CC(=O)NCC1(C)CCN(C(C2(C)CS(=O)(=O)C2)=O)C1)OC C(=O)(CC(=O)NC(C(=O)NCC(F)C1CCC1)c1cccs1)OC c1(C(N2CCN(C(c3c(CC)ncs3)=O)CC2)=O)ccc(CO)c(Cl)c1 C(CCC(=O)N1CCC(CCNC(=O)Cn2cc(Cl)cn2)C1)=C(C)C C1(C#CC(=O)NCC(C)(C(C)C)NC(c2cc(C#N)ccc2F)=O)(CC)COC1 c1(OC)ccnc(C(N2CC(NC(=O)CCCC(C)C)CC2CO)=O)c1O c1(C(C(N2CCCC(c3cn(CC(=O)OC)nn3)C2)=O)C)ccc(F)c(OC)c1 c1(C(=O)NCC(C)NC(C2C(C)C2)=O)cc(C(N)=O)c[nH]1 c1(C(=O)NCC2CC(CNC(CCSC)=O)OC2)cccc2c1C(=O)NC2 Cn1nc(CC(=O)NC2(C)CC(NC(c3csc(C#N)c3)=O)C2)cc1Cl N1(C(C2CC3(CC(=C)C3)C2)=O)CCN(C(C2CCC=CO2)=O)CC12CCC2 C(=O)(C(CC(C)CC)NC(C1C=CCC1)=O)N1CC(C=C)(O)C1 C1(NC(c2scnc2Cl)=O)CC(F)CN(C(=O)CCc2cnc[nH]2)C1 C1(C(=O)NC(c2cccs2)C)CC(C)(C)CCN1C(c1cnn[nH]1)=O c1(OC)cc(F)c(CC(N2CC(NC(C3CCCCC3)=O)C(O)C2)=O)c(F)c1 CC1C(NC2CCN(C(=O)CN(C(c3cncn3C)=O)C(C)C)C2)CCCC1C C(=O)(C1=CC(C)CC1)NC(CNC(C(c1ccccc1O)OC)=O)(C)C c1(C(N(C)CC2CN(C(CCc3cnc(C)o3)=O)C2)=O)cncnc1C1CC1 CC1(C)CN(C(=O)CC2C=CCC2)CC1CNC(C1C=CCS1)=O CC1CC(C(=O)NCc2nncn2C)CN(C(=O)C(C)C#N)C1 CC(C(=O)NC1(CCC(=O)N(CC(Cl)Cl)C)CCC1)NC(=O)C1CC1 C1(NC(c2c(C)cns2)=O)CCN(C(C2CCSCC2)=O)CCC1CO N1(C(CS(CC)=O)=O)CCN(C(c2ccc(Cl)c(C)c2)=O)C(COC)C1 c1(C(=O)NC2CC(NC(C3CC(C)C3)=O)C2)c[nH]c2ccc(Br)cc12 N1(C(c2cncc(OC)n2)=O)CC2(C1)CN(C(C1CC1c1ccc(Cl)s1)=O)C2 CCCC(C(=O)NC1C=CC(CNC(c2nccnc2C(F)(F)F)=O)C1)OC N1(C(C(C)N2CCC2)=O)C2CCCC1CN(C(C1CC1C(C)(C)C)=O)C2 C1(NC(C(CC=C)OC)=O)CC12CCN(C(c1ccc(C)nc1NC)=O)C2 C1(C2CC2)(CNC(c2cc(OC)nn2C)=O)CCN(C(=O)CC(C)C2CC2)C1 c1(C(N2CCC(C)(NC(C(CC)OC)=O)C2)=O)cc(C)c2c(O)nc(O)nc2n1 C1(CCNC(=O)CC2CCOC2)CCCN(C(=O)C=Cc2ncc[nH]2)CC1 C1(NC(c2cc(C(C)C)on2)=O)CCCCC1NC(=O)CCc1ccccc1Cl C(=O)(CCC(=O)NCC(C)(O)CNC(=O)CCc1nnc(S)n1C)NC N1(C(c2c(C(C)C)cco2)=O)CCN(C(=O)CC2CC3(CC3)CO2)CC(O)C1 Oc1ncccc1CNC(=NCC1CC1)NC1CCOC(c2cccc(F)c2)C1 C1(NC(c2ncc(C)nc2)=O)CCCN(Cc2nc(C)c(C)o2)CC1 N1(C(C2(CC#C)CCCCC2)=O)CCCC2(NC(c3cncc(C)c3)=O)CC2C1 c1(C(=O)NC(C)CN(C(=O)CCc2ccccc2O)C)c2c(nn1C)CCCC2 Cc1cc(C(=O)N(CC(=O)NCCOCC(N)=O)C(C)C)nn1C CC1CCC(C(=O)O)N(C(C2CCN(c3ccc(C#N)cn3)CC2)=O)C1 Cc1ccc(CC(=O)N(C)CC2CCN(C(c3nscc3C)=O)CC2)c(F)c1 O=C1CC(CC(=O)NCC2CC3CCC2N3c2ncc(Br)c(O)n2)CCCN1 NC(=O)CCC(=O)N1CCC(NC(=O)C=CCOC2CCOCC2)C1 c1(C(N(C2CCCC(NC(c3ccc(CC)[nH]3)=O)C2)C)=O)cc(N)nc(Br)c1 C(=O)(CCCCCC(=O)NC1C=CC(CNC(=O)C(C(C)(C)C)OC)C1)OCC C(C1CCOCC1)=CC(=O)N(CC(C(=O)N(CCCF)CC)C)C CC1CC(CNC(=O)Cc2ccc(CO)cc2)CN1C(c1cccc(Cl)n1)=O S(=O)(=O)(c1c[nH]ccc1=NC1CCc2ccccc2C1C)NCCSCCCC c1(OC)cc(Cl)c(C(N2C(C(N3CC4CCC3CC4)=O)CCC2C)=O)cc1OC N1(C(CC2CC(C)(C)C2)=O)CC(NC(=O)CC2CC(=O)NC(=O)C2)CC12CCC2 C1(C)(C(=O)NC2CCC(CNC(C(C)OC3CCCC3)=O)C2)CC(F)(F)C1 Cc1ncnc(C)c1CC(=O)NCC(=O)NCC1C=CCOC1 C1(O)(COC)CCN(C(c2n[nH]c(C)n2)C(=O)NCC2CCCO2)C1 c1(OC)ccc(OCC(=O)NC2(C3CCCN3C(=O)C(C)CN(C)C)CC2)cc1 CC1(CNC(C2(C)CC2Br)=O)CCCN(C(C2CC(=O)N2)=O)C1 c1(NC(=O)Nc2cc(C)cc(Cl)c2)c[nH]c2nccc-2c1.C12CC(C1)C(=O)CC2 C1(NC(CCCCC)=O)CN(C(C2OCCC2C(=O)OC)=O)CC(C)(C)C1 N1(CC)CC(NC(c2conc2CNC(=O)CC2CCCC(=O)C2)=O)CCC1=O c1(OC)ccc([N+](=O)[O-])cc1C(C)NC(=O)C(c1ccccc1F)(F)F CC(O)CCCCCC(=O)N1CC2(CC(NC(c3ccncc3N)=O)C2)C1 c1(C(=O)NC(CNC(c2c(CC)cco2)=O)(C)CC)ccc2c(c1)CCCO2 C1(C(=O)NC2C(CC)C2)CCC(NC(c2ccnn2C2CC2)=O)CC1 Cc1sc(Cl)nc1C(N1CC2CC2(NC(c2cc(Cl)ccn2)=O)C1)=O c1(C(N2CCC(NC(=O)CC3(CSC)CC3)C2)=O)ccc(C(F)F)nc1 C(C(C)(C)CNC(c1cnn(-c2ccccn2)c1)=O)NC(C(C)n1cccc1)=O N1(C(C2Cc3c(C)[nH]nc3CC2)=O)CCc2ccccc2C(O)C1 N1(C(CCCCN(C)C)=O)CCC2CN(C(c3cc4c(s3)CCOC4)=O)CC12 c1(CC)[nH]c(Cl)nc(=NC(C)CNC(C2(C)CCOC(C)C2)=O)c1C#N C1(N(C(CS(=O)(=O)NCC)=O)C)CN(C(=O)C=Cc2cc[nH]c2)CCC1O c1(C(=O)NCC(C)N(C(=O)COCCF)C)cn(C)c(C(F)F)n1 N1(C(c2c(COC)scc2)=O)CCOCC(NC(=O)Cc2ccns2)C1 CCC(CC)CC(F)C(=O)NC(C1CCN(C(=O)CCCCOCC)CC1)CO CC(CC(=O)N1CCN(C(=O)Cn2cccn2)C2COCC12)CC(F)(F)F c1(OCC)c(NC(=O)NCC(=O)Nc2cc(C)cc(C)c2)cccc1F c1(C(=O)Nc2ccc(NC(C(CN(C)C)(C)C)=O)cn2)cc2cnccc2[nH]1 N1(C(c2c(C)nsc2)=O)CCN(C(C2CS(=O)(=O)C2)=O)CC1C(F)F C1(N(CCC)CC)CCN(C(c2csc(CNC(C(C)=CC)=O)n2)=O)CC1C C(N=c1nc(N2CC3CC2CS3(=O)=O)c2ccccc2[nH]1)c1n(C)cnn1 N1(C(=O)NC2C(C)CCCC2)CCN(C(=O)C(C)(C)NS(C)(=O)=O)CCC1C N1(C(C=C(C)c2ccccc2)=O)CC2CCC(N(C(=O)CCF)C)C2C1 C1(NC(C(CC)F)=O)CC2(C1)CN(C(C1CCCN(C(C)=O)C1)=O)C2 CC(CNC(c1cccnc1-c1ccccn1)=O)(C(F)(F)F)C1CCCCC1 N#Cc1cn[nH]c1C(N1CC(OCCNC(=O)C(C2CCCCC2)F)C1)=O N1(C(C2(c3cc(F)ccc3F)CC2)=O)CC(NC(c2cnc(C)[nH]2)=O)CC(F)C1 N(C(=NCCCC1CC1)NCC1CCOC1=O)C(C)C1CC1 Cc1nc(-c2nc[nH]n2)sc1C(=O)N(CCCCNC(C1CC12CCCC2)=O)C C1(CNC(C=C(CCC)C)=O)(NC(=O)CCSC(F)(F)F)CCCCC1C N1(C(CNC(c2cc[nH]c2)=O)=O)CC2CC2C2CC12 C#Cc1cncc(C(N2CC3(CC(CNC(c4cnc(O)s4)=O)C3)C2)=O)c1 N1(C(CCOCCC)=O)CCC(N(C(=O)CCc2cscn2)C)C2(CC2)C1 O(NC(=O)CCCCOC)c1c(OC)nsc1 c1(-c2cnc(CNCc3ccc(F)c(Br)c3)nc2)cc(F)c(Cl)c(F)c1 CCC(C)C(C(=O)NCc1cccc(CO)c1)N(C(=O)CC1(O)CCCOC1)C C(=O)(C(CC(F)F)N(C(=O)C1=COCCC1)C)NCP(OCC)(C)=O N1(C(C2CC(OC)CN2C(=O)CC(C)(C)OC)=O)CCC2(CCCCO2)C1 N1(C(C(CC)F)=O)CCN(C(c2cn(C)cn2)=O)CC1c1cccnc1 N1(C(c2nn(CC)nc2C)=O)CC(C(N2CCC2(C)CCO)=O)CC12CCC2 N1(C(c2ccc(SC)s2)=O)CCN(C(C2CCOC2(C)C)=O)C(CCO)C1 CN1CCN(C(c2cc(CCNC(=O)CCc3cnco3)on2)=O)CCC1=O CC1CCCc2cc(C(N3CCC(CC(C)NC(=O)C4CC4)CC3)=O)nn21 C1(=O)CC(C)CC(=O)OC(CC)CN1.C(=O)(C(C)(C)CO)Nc1ccccc1 c1(OC)cc(NC(c2cccc(NCc3ccc(F)cn3)c2)=O)ccc1Br CCC(O)C(C)(C)C(=O)N1CCC1C(=O)NCCC(=O)OC(C)C c1(C(N2C(C(N3CCCC(C#N)C3)=O)CC3CC32)=O)cc2ncccc2[nH]1 Cc1cc(Cl)c(C(=O)NC2CC3CC2N(C(=O)CCc2cn[nH]c2)C3)cc1F Cc1cc(C(=O)NC2CCCCC2CNC(c2cc(C)c(C)[nH]2)=O)ccc1F C1(NC(C2CC2F)=O)(CO)CCCN(C(=O)CCC2CCCCO2)C1 c1(C(N2CC(C(C)(C)O)(CNC(c3nc(C)c(C)s3)=O)C2)=O)ccc(Cl)nc1N N1(C(C2CCN(C)C(=O)C2)=O)C2CCCC1CC(NC(C1C=CCC1)=O)C2 c1(C(=O)NC2C(CCC)CN(C(C3C=CCC3)=O)C2)cnc(C)cc1C C12(CNC(=O)Cc3cnc[nH]3)CCC(C1)N(C(c1ccc(F)cc1Cl)=O)C2 C1(C)(C(=O)NC(CCCNC(c2c(CCC)n[nH]c2)=O)C)CCC(C)=C(C)C1 CC1CC(C(=O)NCC2CC2CNC(c2ocnc2C2CC2)=O)CO1 C1(CNC(C2CC(C)(C(=O)OC)C2)=O)CN(C(=O)C(O)C(C)C)CC12CC2 Cc1cc(OCC(=O)NCCCOCCNC(=O)Cc2csc(C)c2)no1 CC(C(CO)NC(c1cn(CC2CC2)nn1)=O)NC(=O)CC1(CC(=O)OC)CC1 c1(C(=O)NC2CCC(NC(C3(COC)CCCO3)=O)CC2)cc(=O)c(O)c[nH]1 c1(OC)cc(NC(C2CCCC2NC(c2cnn(C(C)(C)C)c2)=O)=O)c(F)cn1 Cc1oc2ccccc2c1C(=O)NC1(CNC(=O)CCc2cc[nH]n2)CC1 N1(C(CCCCC)=O)CCC(C2CCN(C(=O)C(c3cnn(C)c3)O)C2)CC1 Cc1cc2ncc(C(N3CCC4(CCCN4C(=O)Cc4cnc[nH]4)C3)=O)cn2n1 C1(CNC(C(COc2ccc(CC)cc2)C)=O)CCCCN(C(=O)C(=O)NC)C1 c1(OC)ccc2[nH]cc(C(N3CC(N4CCN(C(=O)COC5CC5)CC4)C3)=O)c2c1 c1(C(=O)NC)ccc(CNC(=O)NC(C)(CO)C2CCC2)o1 C=CC(CCC)CC(=O)N1C(CNC(c2ccc(Cl)cc2)=O)CC2CC12 C(C(=O)N1CCCC1CN(C(=O)CCc1cc(C)no1)C)(C(C)C)SCC C1(C)(CNC(c2n[nH]c(C)c2C)=O)CN(C(=O)CCCCCF)CCO1 C(=O)(CCS(C)=O)NCC1(CCNC(Cn2cc(C(C)O)nn2)=O)CC1 c1(NC23CCC(CNC(=O)CNC(=O)CO)(OC2)C3)cccc2nc[nH]c12 CCCC(C(=O)NCCCc1cc(C)no1)NC(c1ccc(C#N)o1)=O c1(C(=O)NC(C2CCN(C(=O)Cc3cnn(C)c3)C2)C)c(F)cc(C#N)cc1F C1(NC(c2c(C)cn(C)c2)=O)CC2CCC(C1C)N2C(c1ccoc1)=O n1(CC(=O)NCC(C)NC(=O)C=CCOC2CCCCC2)nnc(C2CC2)n1 c1(C(=O)NCCC(C)N(C(=O)CC2CCCO2)C)cnc2c(N)cccc2c1 C1(C)(NC(C(C)c2cc[nH]n2)=O)CN(C(c2scnc2C2CC2)=O)C1 N1(c2nnc(C(C)C)o2)CCN(C2CCCN(C(C3CC=CCC3)=O)C2)C(=O)C1 C(CCC(C)C)(C(=O)NCc1ccn(C2CC2)n1)NC(c1c(C)nn[nH]1)=O c1(CC(N2CCC(NC(CN(S(=O)(=O)C3CC3)C)=O)CC2)=O)ccccc1S(C)=O CC1CN(C(C2CSC2)=O)CCC1NC(=O)C1=CSCS1 CC1(C(=O)NC2CC3C=CC2C3)CCCN1C(=O)CN1CCCC1=O CC1CN(C(c2ccc(Cl)[nH]2)=O)CC(C)N(C(=O)COc2ccc(Cl)cc2)C1 N1(C(c2cnc(OCC)c(Cl)c2)=O)C2CCC1CN(C(c1cccs1)=O)CC2 N1(C(C(COCC)C)=O)CC(C(N2CC3CCC3(CO)C2)=O)C(F)(F)C1 C1(NC(CCCC(C)O)=O)CCCOC12CCN(C(=O)COc1ccon1)CC2 CC1(C)CCC(NC(=O)CCc2cnco2)C(CNC(=O)C(C)(C)F)C1 C1(C)(C(=O)NCC2OCCN(C(CCc3n(C)c(S)nn3)=O)C2)COC(=O)OC1 c1(C2(NC(c3n(CC=C)nnn3)c3ocnc3C)CC2)ccc(OC)cc1 C1(CCNC(CCNC(C)=O)=O)COCCN1C(=O)C(C)Sc1ccc(Cl)cc1 C(=O)(C(CC)C(=O)N1CCC(C)(C(=O)NCC(O)C(F)F)CC1)OCC C1(C2CC2)(C(=O)NCC(CC)NC(c2cnn(C)c2F)=O)CC=CC1 C1(CNC(CN(CCC)C)=O)CC2(CCN(c3cc(C)ccc3[N+](=O)[O-])C2)CO1 N1(C(COCC)=O)CCN(C(C2CCC(NC(=O)C(C)C)CC2)=O)C2(CCC2)C1 N1(C(c2cnc(C)[nH]2)=O)CC2CC(NC(=O)CCCc3ccc(C)s3)C2C1 c1(C2C(C(N(C3CCN(C(c4sncc4Br)=O)C3)CC)=O)C2)ccccc1 C=CCC(C)(C)CC(=O)N1CCOC(C(N2CCC(F)(F)C(O)C2)=O)CC1 N1(C(CC(CC=C)NC(=O)CCCN(C)C)=O)CCC(O)CC12CC2 N1(C(CNC(CCC)=O)=O)CC(C)N(C(=O)CCc2ncccc2OC)CC1C C1(C(N2C(CC)CC2)=O)C2CC(O)C(C2)N1C(C1(OC)CCCCC1)=O N1(C(C=C(CC)CC)=O)CCCCC1CNC(=O)CC1CC(C)OC1C C1(CCNC(C2CN(C(N)=O)C2)=O)CCC(NC(c2ccoc2Br)=O)C1 C1(CNC(c2nc(CCC)oc2)=O)CC(F)(F)CN1C(C1CCCC(CF)C1)=O Cn1nc(C(N2CCC(O)(CNC(C3CCC(CCO)CC3)=O)C2)=O)cc1C#N O=C(C1=CC2(CN(C(c3ccnc(O)c3)=O)C2)OC1)NC1(CF)CCCC1 C1(CNC(COCCCC)=O)CC12CCN(C(c1cc[nH]c3nccc1-3)=O)CC2 CC(O)CC(C(=O)O)NC(c1ccc(CN2CCCC2)cc1)=O Cc1cc(C(=O)NC(C)CCNC(=O)CC2COCC2(C)C)c(O)c(C)n1 c1(N2C(CNC(C(c3cccc(C)c3)O)=O)CCC2)ccc2nccnc2n1 CC(O)C(F)(F)C(=O)N1CCOC(CN(C)C(c2cncs2)=O)C1 c1(C(N2CCN(C(C#CC(C)(C)O)=O)C(CN(C)C)C2)=O)ccn2cccc2c1 N1(C(c2n[nH]c(O)n2)=O)CCCC(CNC(=O)C(c2ccc(F)cc2)(F)F)C1 c1(C(=O)NCC2(CO)CCCNC2)cnn2c1NCCC2C(F)(F)F N1(C(C2OCCN(C(C(CC)N(C)C)=O)CC2)=O)CCN(CC)C(C)(C)C1 N(C(=NCCCC(F)F)NCc1cc(C)ccc1Br)CCOCC Cc1nc(Br)sc1C(N1CCC(C)(CO)C1)C(=O)NCCC1(C)CC1 C(=O)(C1=CCCC1)N(C1CCN(C(=O)CC2CC2)C1)CC#C C1(NC(CCSCCCC)=O)CC(CNC(=O)CCCc2cncs2)C12CCC2 c1(CNC(=O)CC2CCCC2O)cccnc1CNC(c1ncccn1)=O C#Cc1cc(F)c(C(N2CCC3(C2)CN(C(=O)C(C)(CC)CC=C)C3)=O)cc1F Cc1oc(CO)cc1C(N1CSCC1C(N1CCSCC1C)=O)=O c1(CC(=O)N(CC(C)NC(=O)CC2CCOC2=O)C)ccc2nc[nH]c2c1 C(=O)(C1CCCc2nncn21)NCC(CC(C)C)NC(CN1CC(C)C1)=O C(C(C)(C(=O)N1CC(c2nncn2C)C1)OC(C)(C)C)ONC(=O)OC c1(C(=O)NC(CNC(c2cc(C)c(C)nc2)=O)(C)C)cc(F)cc2c1NCCC2 N1(C(C(C)c2ccsc2)=O)CCN(C(=O)C=CSc2ccccc2)CC1C(F)F N1(C(C=CC)=O)CCN(C(=O)C(CC(=O)OC)N2CCCCC2)CCC1C N1(C(C(C)(C)CCNC(c2ccoc2Cl)=O)=O)C2CCC1CC(F)C2 c1(NC(C)=O)ccc(C(N2CC(N3CCCC3)C(O)C2)=O)c(Cl)c1 N1(C(CC2CC(=C)C2)=O)CC2(CC2)CC1C(=O)NCC1(CO)CCN(C)C1 C=CCCC(C)(C)C(=O)N1CCC=C(C(=O)N(C)Cc2cnc(C)cn2)C1 C1(CCC(N2C(C(N)=O)CC2)=O)CCN(C(C2CCC(F)(F)C2)=O)CC1 N1(C(CCNC(C(C)(C)C)=O)=O)CCCc2cccc(OC(F)F)c2C1 N1(C(C2COC(=O)O2)=O)CCC2(C1)CN(C(c1cc3cn[nH]c3cn1)=O)CCO2 Brc1cc2ncnc(NCc3scnc3-c3ccc(C4(CBr)N=N4)cc3)c2s1 c1(C(=O)NCC2CN(C(c3ccc(OC)s3)=O)C(C)C2)c(F)ccc(O)c1F N1(CC2(NC(c3c(C)onc3)=O)CC2)CCN(C(C2CCC(F)C2)=O)CC1 N1(C(=O)NCC)CCC(C(=O)NCC(C)NC(C2OCCC2C(F)(F)F)=O)CC1 c1(NCC(CC)CC)ncccc1S(=O)(=O)NC(C)C(C)COC CN1CC=C(CC(=O)N2CC3CCCC(C2)N3C(=O)Cc2ccc(O)nc2)CC1 c1(OC)cccc(Br)c1C(N1CC(O)(CNC(c2cc(C)nc(C)c2)=O)C1)=O CC(C)(CNC(=O)C(O)C1CC1)CNC(C1CCN(S(C)(=O)=O)C1)=O c1(OC)cc(C(=O)NC(C2CCCN2C(=O)CCC2CC2(C)C)C)n(C)n1 C1(C(=O)NC(C2CCOCC2)C)CC=CCC1NC(c1[nH]nnc1C1CC1)=O C(CC)(CC)(CCNC(=O)CSc1ccc(O)cc1)NC(CC=CC)=O C1(O)(C(CC)C(=O)NC2CCC2CNC(C2(C(=O)NC)CC2)=O)CCCCC1 c1(C(=O)NC(C(C)C)CCN(C)C(c2cccnc2Cl)=O)cccc2c[nH]nc12 CC(=NO)C1CC(C(=O)NCC2CCCCN2C(=O)C(C)C2CC2)C1(C)C c1(C(=O)NCC2CN(C(=O)CCc3ccccc3)CCO2)nccc2nn[nH]c12 C1(F)(CNC(C=C(C)C(C)C)=O)CCCN(C(c2cnc3[nH]nnc3c2)=O)CC1 C1(C(=O)NC2CC3CC(NC(C4CC(O)(CC)C4)=O)CC32)CCOC2(CCC2)C1 C(=O)(C(C)(C)C(F)F)N1CCC(C(CNC(C(C=C)OC)=O)O)CC1 C(=O)(CC(C)(C)C(F)F)NC1C(OC)CN(C(Cc2cc(OC)c(O)cc2)=O)C1 C1(CNC(c2ncc(NC)nc2)=O)CN(C(=O)C=CC(N)=O)CCCO1 C(=O)(CC(F)(F)C(F)(F)F)NCCCN(C(CC(=O)NCC1CC1)=O)C1CC1 c1(C(N2C3CC(N(C(CCC#CC)=O)C)CC2CC3)=O)ccc(F)c2occc12 N1(C(C2CCN(C(CNC(=O)NC)=O)C(C)C2)=O)CC(C)CC(C)(C)C1 C#CC1CC2(CC(C(N3CCCCC(NC(=O)CC(C)(C)C4CC4)C3)=O)C2)C1 Cn1nc(Br)nc1C(c1nnnn1CC(F)F)NCCc1cc(Br)no1 C1(O)(CNC(C2CC(C3CCC3)C2)=O)CCN(C(=O)C(F)CC2CCOC2)CC1 c1(C(N2C(C(N(C)Cc3c(C)occ3)=O)CCCC2)=O)ccc2cc[nH]c2n1 c1(NC(c2cncc(NCc3c(N)cccc3F)c2)=O)ccc2c(c1)OCCO2 c1(OCC)ccc(C)cc1C(N1CCC(C)(NC(c2cccnc2OC)=O)C1)=O N1(C(C(CC)CC2CCCC2)=O)CCN(C(=O)C(C)(F)F)C(C(C)C)C1 c1(NC(CCCN(C(=O)COCCC(C#N)C2CC2)CCO)=O)ccnc(O)c1 N1(C(COCCCOC)=O)CC2C(NC(=O)COCc3ccncc3)C2C1 c1(CC(=O)NC(c2ccccc2)C(C)NC(=O)CC(C)C)cc(Cl)n(C)n1 CC#CCC(C(=O)N(C1CC(C)CC(C)C1)C)NC(C1CCCCC(=O)C1)=O CCCCC(CC)CC(C(=O)NCC)N1CCOC(CC)(CC)C1 Cc1ccc(NCC(=O)N(C(C)CCNC(=O)CC2CC(C(F)F)C2)C)cc1 Cc1cc(C)c(CC(=O)NCC(C)N(C)C(c2cnc3nccn3c2)=O)c(O)n1 C(C)(CCCCNC(=O)CCC(C)c1ccccc1)NC(CN1CC(CC)C1)=O N1(C(CCNC(C)=O)=O)CC2CCOC2(CNC(=O)C(C)(C)CC(F)F)C1 N1(C(c2ccc(CC)nc2C)=O)CC2CCCC1C2CNC(C1CS(=O)(=O)C1)=O c1(OC)cccc(C(=O)NC(C)C(C)(C)NC(=O)CC2CC(F)(F)C2)n1 c1(C(N2CC(O)(CN(C)C(C3CC3(F)Cl)=O)C2)=O)ccccc1-c1cncnc1 N1(C(c2c(C)snc2)=O)CC(C)C(NC(c2cc(O)cs2)=O)C(C)C1 c1(C(=O)NC2CCC(NC(CC(C)(C)SC)=O)C2)cccn2c(O)nnc12 Cc1cc(C(=O)N(C(C)C(=O)OC(C)(C)C)CC(=O)N(C)C)nn1C1CNC1 CC1(C)CN(C(c2cc(Cl)c(F)c(Cl)c2)=O)CC(C)(C)C1NC(=O)C1=CCCS1 Cc1cc(C(=O)NCCCN(c2ncc(Br)c(O)n2)C)cc(O)n1 C=CCC(CNC(c1cscc1C(C)C)=O)NC(C1CC1C)=O Cc1nc(O)[nH]c1C(=O)N(C(CNC(c1cc(O)nn1C)=O)C1CC1)C c1(C(=O)NC2C(NC(CCn3ccc(C)n3)=O)CC2)ccc2c(c1)C(=O)CCC2 C1(NCc2n(C=C)nnc2)CCN(Cc2ccccc2)CC1C c1(C(N2C(C(=O)NC(C=C)COC)CC2)=O)cc(NCC)no1 CCCCC(C(=O)N(CCOC)CC)NC(=O)C(C)N(C(=O)COC)C C(C(C)(O)CNC(=O)C(Cc1cn[nH]c1)NC(=O)CCCNC(N)=O)OC C1(C(=O)NC2CN(C(CCCCSC)=O)C2)CC(C)(C)CCO1 C#Cc1ccc(C(=O)NC2CCC2C(=O)N(C(CO)CO)CC)cc1C c1(C(=O)NCC(C)CN(C)C)cccc(C2(CO)CC2)n1.N1(CC)CCCC1CO N1(C(C2(C=C)CC2)=O)CCCC(C2CCN(C(=O)C3=CCC3)C2)C1 C1(NC(=O)NCc2n(CC)cnc2)CCc2nc(NC(C)(C)C)ncc2C1 N1(CC(=O)NCCC(C)NC(=O)C(C(C)(C)C)N(C)C)CC(=O)N(C)C1=O N1(C(c2c(OC)cccc2C)=O)CC2CCCC2(CNC(C2CC(SC)C2)=O)C1 C(C1=CCN(C(=O)CC2CCCC(C(C)C)O2)CC1)NC(c1cnn(CC)n1)=O CON=CC(=O)NC(CNC(C1CC1(F)F)=O)C1CCC1 Cn1ncc(C(=O)NC2CCCCC2NC(C2CCC(=O)O2)=O)c1C(F)F c1(C(=O)NC2(CNC(=O)C(F)(F)c3ncc[nH]3)CCOC2)cccc(OCF)c1 C(CCN=C(NC1CCOCC1)N1CCC(F)(c2ccccc2Cl)C1)=CC=C Cc1ccoc1S(=O)(=O)NCCC1CNCCCO1 C(=O)(C(C)(O)CNC(=O)C(O)CNC(C1CCSC1)=O)OC C(=O)(C(CC(F)(F)F)c1ccccc1)N1CC2C(COC(C)(C)C)C2C1 c1(CC(=O)NC(CC)(C)CNC(c2nc(Cl)sc2C)=O)c(C)cc(C)cc1C C1(CNC(N2CC(C(=O)OC)C2)=O)CCC(=O)N(C)C1=O c1(OC)cc(C(=O)NC2CCCCN(C(c3ccsc3)=O)C2)c([N+](=O)[O-])cc1F CON=C(C(=O)N1CCOCC(NC(=O)C(c2ccccn2)C)C1)c1ccco1 C1(C2CC2)(NC(c2nc(C)sc2)=O)CCN(C(=O)CC(C)(C)C(F)F)C1 N1(CC(=O)NCC(F)(F)Cn2cc(-c3c[nH]c(C(=O)O)c3)nn2)CC=C(CO)CC1 c1(N2C(c3c(OC)cccc3)CCC2)ncnc2[nH]cnc12 c1(C(=O)NCCC(=O)NC2CC3CCCC3C2)ccc2ccccc2c1 C12(C(N3C(C4(NC(CCC#C)=O)CC4)CCC3)=O)CCC(N(C)C)(CC1)CC2 C1(CC(=O)NCCNC(c2ccc(C(C)(C)C)cc2)=O)Cn2ccnc2NC1=O c1(CC(N2C(CCCNC(C3CC=CCO3)=O)CCC2)=O)ccc(O)c(F)c1 c1(C(=O)NCCCN(C(CC(CC)CN(C)C)=O)CCO)cc2scc(C)c2[nH]1 C1(NC(c2c(C(C)C)n[nH]c2)=O)CC(C)CN(C(c2cn(C)nc2Br)=O)C1 c1(C(=O)NCCC2CC(C(=O)NCCn3cncn3)C2)c[nH]c2ccccc12 c1(CC(N2CC(OC(C)C)C2)=O)nc([N+](=O)[O-])n[nH]1 C(=O)(CC1=CCOCC1)NC(CCCC)C(=O)NCCc1n[nH]c(C)n1 C1(NC(C=CC(C)(C)SC)=O)CC(C)CN(C(=O)Cc2[nH]cnc2C)C1 c1(C(=O)NC2CC(CNC(C(C=C=C)C)=O)OCC2)ccc(Cl)cc1C N1(C(c2cc(C)[nH]n2)=O)CCC(C(=O)NCC(C2CCCC2)C)(C(C)C)C1 c1(OC)cc(F)ccc1C(N1C2CCC1(CNC(c1ccc(CO)o1)=O)CC2)=O C1(C)(CC)CC(NC(c2cc(-c3ccoc3)on2)=O)CN1C(c1cccn1C)=O C1(NC(CN2CCC(OC)C2)=O)CN(C(=O)CCCN=[N+]=[N-])C2(CCCC2)C1 C1(C(F)(F)F)(C(N(CC(CNC(C#CC(C)C)=O)C)C)=O)CC2CCC1CC2 C1(CC)(NC(=O)CCCCCCN)CCCN(C(c2nnc(C3CC3)o2)=O)C1 C1(CC)CCC(NC(=O)CCOCCN(C)C(c2cnc(Cl)s2)=O)CC1 c1(CN(CC)CC)ccc(C(=O)NC(C)CN(C(C2(F)CCOC2)=O)CC)o1 C1(NC(c2ccc(COC)o2)=O)CC2(CCCN(C(=O)COC3CCOC3)C2)C1 N1(C(CC(CC)C(F)F)=O)CC2(NC(c3sc(F)cc3C)=O)CCCC2(F)C1 CC(CC(=O)NC12CC(CNC(=O)C(O)Cc3ccccc3)(C1)C2)C(C)(C)C C(=O)(C(F)CC(C)(C)C)NCC1CC(CNC(c2c(CCC)cccc2)=O)C1 c1(C(=O)NCC(F)(F)C(F)(F)F)ccc(F)c(Br)c1F C1(C(=O)NC(C)CNC(=O)CCCCc2ccccc2)Cc2cccc(F)c2O1 c1(CC)nc(Cl)cc(=NCC2(C)CCN(C(c3cc(C)nc4ncnn34)=O)C2)[nH]1 c1(OC)nc(C(=O)NCC2CCCN2C(C2CCCC(F)C2)=O)sc1C c1(CNC(C2CN(C)CCO2)CC)c[nH]c2cc(C(=O)O)ccc12 c1(C(=O)NCCCC2(NC(C3ON=C(C)C3)=O)CC2)cccc(C)c1F C1(CNC(C(CC)C)=O)CC2CCC(C1)N2C(C1CCS1(=O)=O)=O C1(C)(C(=O)NCCC2CC(C(=O)NC(C)C3CC3)C2)CC=CC1 c1(C(N(CCN(C(c2ncoc2C)=O)CC)CC)=O)cnc2sccc2c1 CN1CC(C(=O)NCCCC2(NC(C34CC5CC3C4C5)=O)CC2)CC1=O C(c1nc(C)c(C)[nH]1)=CC(=O)NCC1C(NC(Cc2nc(C)oc2)=O)CCC1 Cc1noc2cc(NN3CC(CC(C(=O)C(F)(F)CN4CCCC4)=O)C3)ccc12 C(=O)(C(O)CC(F)F)N1CCC(N2CCN(C(C3(C(=O)NC)CC3)=O)CC2)CC1 C1(CNC(COC(CC)C)=O)CN(C(C2CCN(C(C)=O)C2)=O)CC1N(C)C C=CC(C)(O)CC(=O)NC(CN=[N+]=[N-])C(=O)NCC1(CC(N)=O)CC1 N1(C(c2cnc(C(C)C)nc2)=O)CC2(C1)CN(C(C1CC1OC(C)(C)C)=O)C2 Nc1cc(C(=O)NCCC2CCN(C(=O)CN(c3ccncc3)C)C2)ccc1F CC(C)(C)C(CC(=O)N1CCC(NC(=O)COC(F)F)C2(CCC2)C1)C(F)F CCC(C)(C)C(=O)C(=O)NC(CC(N)=O)c1cn(-c2ccccc2C)nn1 c1(-c2n(CC(=C)C)nc(C(C)O)n2)cn2cc(C)nc2s1 c1(C(CCC)NC(=O)C(C)NC(N)=O)ccc(Cl)cc1 CCC(O)C(C)C(=O)NCC1CC1CNC(c1n[nH]cc1Br)=O N1(C(c2c(C(C)C)occ2)=O)CCC(F)C(NC(=O)C=C2CCCCC2)C1 CC(CC(F)F)C(=O)NCC1CC(F)CN1C(c1coc(CO)c1)=O c1(C(N2CCC(NC(CCOCCC)=O)C2(C)C)=O)cc(Cl)cc2c1CCC2 N1(C(CCNC(=O)OCC)=O)CCCC(N(C(=O)C(C)(COC)OC)C)C1 C1(NC(CCC=CCC=C)=O)(CF)CCN(C(c2snnc2C2CC2)=O)C1 C1(CC(=O)NC2CCN(C(C3(C)C(C)C3)=O)C2)CC2CCC1C2 N1(C(COCCOC)=O)CCC(CCNC(c2ccc(OC)cc2Cl)=O)CC1C CCC(CC(=O)N(CCC(=O)NCCC1CC=CCC1)C1CC1)SC C(C(C)(C)CC(F)F)OCc1ccc(OCc2ccc(OC)cc2)cc1 C1(NC(c2c(C)nc(Br)o2)=O)CN(C(C2CC3(CC3)CO2)=O)C2(CCC2)C1 c1(C(N2CCCN(C(c3c(C)n(C)nc3)=O)CC2)=O)csc2ccccc12 Cc1[nH]c(CNCCN(c2ccc(Br)cc2C(=O)NC)C)c(C)c1-c1nn[nH]n1 c1(C(N2CC(NC(C3C(C(=C)C)OCC3)=O)C(OC)C2)=O)cnn2ccncc12 C12(C(=O)NCCCC3(NC(C(CO)N(C)C)=O)CC3)CCCN1CCC2 N1(C(CCN(CC)CC)=O)CC(N(C)C(c2ccc(C)cn2)=O)C(O)C1 c1(C(=O)NC(C2CCOC2)CNC(C2CCN(C)CC2)=O)c(O)ccc(Cl)c1F c1(OC)ccc(C(=O)NC(C)(C)CC(=O)NCC=CCl)cn1 c1(NCCC(C)SC)ncc(S(=O)(=O)NCC=CBr)cc1Cl c1(C(=O)NC(CC(C)NC(c2n(CCC)ncc2)=O)C)cc(F)cc(F)c1 N1(C(C2(OC)CC(C)C2)=O)CCC(C2(O)CNC2)CC1 N1(C(c2c(C)coc2)=O)CCC(C(=O)NC2CCCSCC2)CC1 C1(C(C)C)CCN1C(C(=O)NC1COC1)c1cccs1 N1(C(C=C(C)C(F)F)=O)CC(C2CCCN(C(=O)CCn3cc(Cl)cn3)C2)C1 CC1(C)CN(C(c2ccnc3ncsc23)=O)CCC1NC(c1cccc(Cl)c1)=O c1(C(N2CCC(C(C(=O)N(C3CCCC(CF)C3)C)F)C2)=O)cc2occc2[nH]1 C#CCCC(C(=O)OC)NC(=O)CNC(=O)CNC(C1C2CC(=O)CC12)=O C=CC1(CC(=O)NC2CCC(O)C2)CN(C(=O)Cc2ccc(C)nc2)C1 c1(C(=O)NC2C(OC)CN(C(=O)COC(F)(F)F)C2)nc(Cl)ccc1N c1(ON(CCCC(=O)O)C2(c3csc(C4CC4)n3)CC2)cccc(OC(F)F)c1 c1(C(=O)NC2CCCC(NC(=O)C3=CSCS3)C2)cc2n(c1)CCCC2 CN1CC(C)(C)CC1C(N1CCCC(O)(CNC(=O)CC2(N(C)C)CCC2)C1)=O C1(NC(C2C(CNC(C(c3ccn(C)n3)C)=O)C2)=O)CC(C)(C)C12CCC2 c1(C(=O)NCC(CN(C(=O)CCC2CCC(=O)N2)CC)(C)C)cc(O)nc(Cl)c1 C1(C(=O)NCCN(C(C(C)(C2CC2)OC)=O)C)CCC(CCC(C)C)CC1 N1(CC)CCC(CC(=O)NCC=C)CC1.C12CC1C(=O)NC2.C1(=O)CC2CC2N1 C1(CNC(CSCCN(CC)CC)=O)C(C)CCN1C(=O)CCC(=O)NC C1(C(C(=O)NCCSC)N2CCC2CC2CC2)CCC(C(C)C)CC1 CC1C(NC(=O)CC2CCCCCCC2)CCCN1Cc1ccsc1 c1(C(c2nnnn2CCCC2CC2)NC(c2cn(C)nn2)C)scnc1C N(C(=NCC1CCCN1CC)NCC1(C2CCC2)CC1)Cc1n(CC)cnn1 C1(OCc2cc(C)no2)CCCCC1n1cc(CNn2c(C)nnc2S)nn1 N1(C(c2c(Cl)ncc(OC)c2)=O)CCN(C(=O)CC2CC3(CC3)CO2)CC(O)C1 c1(C(N(C2CC(NC(C(C)C#N)=O)C2)C)=O)ccnc(SCC(F)(F)F)c1 C1(CNC(CCNC(=O)OC)=O)CC2CCC1N(C(=O)CC1CCOC(C)(C)C1)C2 C1(NC(C(N2CCCCC2)C)=O)COCC1C(=O)NCCn1cnnc1 C1(CNC(C(C=C)OC)=O)CN(C(=O)Cc2cnn(C)c2)CC1(F)CO CCCC(C(=O)NCC1CCCCN1C(c1oc(C)nc1CC)=O)OCC C1(CNC(c2c(CC)nn[nH]2)=O)CCC(C)(C)CN1C(=O)C(C)C(C)C c1(C(C(N2CCCC(c3cc[nH]c(=N)n3)C2)C)=O)cc(I)cc(I)c1 c1(N2CCC(NC(c3ccn(CC)n3)=O)C23CCC3)nc2ccc(OC)nc2s1 CC(CO)CCN=c1nc(N2CC(C)OCC(C)(C)C2)c2[nH]ccc2[nH]1 C=Cn1nccc1C(N1CCOCC1CC(=O)NCC(CC)CO)=O C(=O)(CCCCC(=O)NCC1CCC2(CN(C(c3c(C)n[nH]c3C)=O)C2)O1)NC c1(C(=O)NC2CCN(C(c3ccncc3Br)=O)CC2O)ccn2ccnc2c1 N1(C(CCCNC(C)=O)=O)CC(NC(c2nccnc2N)=O)CC(C)C1 N1(CC(=O)N(C(CNC(C(C(C)C)O)=O)C2CC2)C)CCP(C)(=O)CC1 C1(C)(NC(C2CC(CNC(C3C(C)=CCS3)=O)C2)=O)CCCCCC1 CC1(C)CN(C(c2ccnc(N(C)C)n2)C(=O)NCCOCC2CC2)CC(C)(C)O1 c1(C(=O)NC2C(NC(c3n[nH]c(C)c3C)=O)CC2)ccc2nsnc2c1 c1(C(=O)NCCCN(C(=O)Cc2cncnc2)C)nccc2ccn(C)c12 C1(NC(CC2C(CC)C2(F)F)=O)CCCN(C(=O)CSc2n[nH]c(O)n2)CC1 c1(C(N2CC(C(N3CCC(CCCO)CC3)=O)C2)=O)ncc(Cl)cc1Cl c1(COCC)nc(C(=O)NCC(C)(C)NC(C2CCN(CC(F)(F)F)C2)=O)co1 C1(CC(=O)Nc2c(C)nsc2)CCCN(C(=O)CC(C)C)C1 c1(C(=O)NC2CC(C)(NC(C3=C(C)CCCC3)=O)C2)ccc2c(c1)C(=O)N(C)C2 c1(C(N(CC)Cc2cc(C)on2)=O)cn2c(n1)CCN(CC1(CO)COC1)CC2 C(=O)(CS(=O)CCC(F)(F)F)NCC1CN(C(C2C(OC)(OC)CC2)=O)C1 N1(C(c2c(CC)ocn2)=O)CCCC2CN(c3cnc(C#N)c(C#N)n3)CCC12 C1(NC(C2C(CCC)CCC2)=O)CCCC12CN(C(=O)C(C1CCCC1)OC)C2 c1(C(=O)NC(COC)C)cc(SC)ccc1Cl.C12CN(C1)C2=O c1(C(=O)NCC2C(NC(c3coc(Cl)c3)=O)C2)cc2ccc(Cl)cc2s1 c1(CC(=O)NC(c2cn(C3C=CCCC3)nn2)C)c(OC(F)(F)F)cccc1F Cc1occc1C(=O)NCC1CCCC1C(=O)NCC1CC1Cl C1(NC(C2(CN(C)C)CC2)=O)CN(C(=O)CCn2cccc2)CC2(CCC2)C1 c1(C(=O)NCC(C2CC2)NC(c2cc(SC)oc2)=O)cncc(Cl)c1Cl N1(C(c2c(OC)c[nH]n2)=O)CC2COCCC2(NC(c2cc(N)ccc2Cl)=O)C1 C1(CC(=O)NCC(CCOC)NC(C2(CO)CCCO2)=O)CCN(OC)CC1 Cc1ccc2nonc2c1C(=O)NC1(CO)CCN(C(C2CCOC2)=O)C1 C1(C(C)C)CN(C(=O)Cc2c(Cl)cccc2Cl)CCC1NC(=O)Cn1ccnn1 c1(C(=O)NC(COC)C(=O)NCc2nn[nH]n2)ccc(=O)n(C)c1 N1(C(c2c(C(C)C)ncs2)=O)CCC(C(F)(F)F)C(CNC(C2(F)CC2)=O)C1 Cc1cccc(-n2nnc(CNC(=O)COc3cccc(I)c3)c2C)c1 N1(C(c2ccc(SC)cc2)=O)CC2CC(C1)N(C(=O)CSCc1ccccc1)C2 CC1CCCCN1CCC(=O)NC1CCC1CNC(=O)Cc1ccsc1Cl c1(C(=O)OC)ccc(Br)cc1S(=O)(=O)N1CC(c2cccc(F)c2)C1 c1(CC(=O)NC2C(CNC(C(C(CC)O)C)=O)CCCC2)noc2ccccc12 CCCC(CCCNC(C1(N2CCOCC2)CCCC1)=O)NC(C1C2CCC12)=O C(CC(C(=O)NCC(=C1CCCCC1)F)NC(C1COCCN1C)=O)SC N1(C(c2nn(C)c(F)c2)=O)CC(C2CN(C(C3CC3c3ccnn3C)=O)C2)C1 c1(N(C(C2N(C(C#C)=O)CCC2)=O)Cc2ccccc2)ccc(OC)cc1F c1(C(C)C)c(C(=O)NC2CN(C(=O)Cc3ccns3)CC2F)cnn1C N1(C(C(CCC)F)=O)CCC(CNC(=O)C2=C(C)CC2)C12CC2 C1(CC(=O)NCCCC(C)O)CCN(C(C2CC2C2(C)COC2)=O)C1(C)C c1(CCCNC(CCN(CC#C)C(C2CCC(F)C2)=O)=O)nc(C)no1 c1(OC)ccc(F)cc1C1CCCN1CCCNS(C)(=O)=O c1(OC)cccnc1C(N1CCOCC1c1cn(CCNC(C)=O)nn1)=O C(C(C(=O)NCC(O)CN(C)C)C(C)(C)C)NC(C(OC)OC)=O Cc1sc(Br)nc1C(N1CC(CNC(=O)C(F)CC2CC2)C(O)C1)=O N1(C(C(=O)NC(c2ccc(Cl)s2)CN(C)C)=O)CCC(NC(=O)CO)CC1 c1(C(N(C2CN(C(CC(COC)C)=O)CC23CC3)C)=O)ccc([N+](=O)[O-])n1C N1(C(C(N2CCCC(SC)C2)=O)=O)CCOCC(C2CCC2)C1 C(=O)(C#CC1CCOCC1)N(CCCCC(=O)NCC1(O)CCCOC1)C c1(CNC(C23CC(C)C2C3)=O)cnn2c1CN(C(=O)CSc1n[nH]c(O)n1)CC2 C1(N(C(c2cnc(CC)o2)=O)C)CN(C(C2CCN2C)=O)CC1(C)C c1(C(N2C(CCNC(CC3CC(C)(C)C3)=O)CCC2)=O)ccc2c(c1)COC2 CC(C)CCC(F)C(=O)N1CC(NC(c2ccncn2)=O)C(F)C1 c1(C(=O)NCCCC(C)NC(C=C(C)c2ccsc2)=O)cccc2nsnc12 N1(C(CCCCC#C)=O)CCN(C(c2csc(=NC3CC3)[nH]2)=O)CC(O)C1 c1(C(N2CC(CC(N3CCOCC3C3CC3)=O)C2)=O)cc2c(F)cc(F)cc2[nH]1 C1(NC(c2ccc(Cl)nn2)=O)CCN(C(C2CC23CC(O)C3)=O)C12CCCC2 n1(CC(N2CC(N(C(c3c(COC)noc3)=O)C)C2)=O)cnc2ccc(C)cc12 N1(CCCN(CCOC)CCO)CCN(Cc2ccccc2C)CC1 c1(CC)ccc(NC(C2CCC(CNC(=O)CC3CCCC4CC34)C2)=O)c(F)c1 C#CCC(C)(CC)C(=O)NC1CC1NC(=O)CCCC#CC C1(C(=O)NCCCC#C)C2CC(CC2F)N1C(c1ccc(C(F)(F)F)cc1I)=O C=CCCCCC(=O)NCCc1n[nH]cc1C(=O)NCC1(O)CCSC1 c1(N(CC(C)CO)C)nc(N(C)C(c2c(F)cccc2F)C2CC2)c2c(n1)CCC2 C(CCN=C(NCCOCCOC)NCc1cncc(O)c1)OC.c1ccccc1 C1(NC(CC2(CC)CCC2)=O)C(C)CCN(C(=O)C(CC)n2ccnc2)C1C C1(C(C(=O)OCC)(C)C)CCCN(C(=O)NC2CCC3(NC(=O)C4CC4)CC23)C1 Cc1ccnnc1C(=O)NCCC(O)C(=O)N(C)Cc1ccon1 C1(C(=O)Nc2cnccc2Cl)CCN(C(c2cccc(F)c2O)=O)CC1F N1(C(Cc2c(C)noc2C)=O)CCOCC(C(=O)NC(C)CCO)C1 C1C(CCCC)C(C)(C)CC(=O)N1C(CC)C N1(C(C=CC(C)=O)=O)CCC(C2CCCN(C(C3CCC4CC4CC3)=O)C2)CC1 c1(NC(c2csc(NC(c3ccc(Br)nc3)=O)n2)=O)cccc2ncsc12 c1(C(=O)NCC(CC(=O)N(C)CCN(C)CCO)OC)ccc(=O)n(C)n1 c1(CC)ccccc1C(N1CCC1CNC(=O)C(C)(F)c1ccccc1)=O C1(NC(C2(C(C)C)CC2)=O)CCN(C(=O)CC#N)CC1F C(=O)(C(CNC(=O)CC(C)C)CC1CCCC1)NC1(CC=C)CC1 C(=O)(CCCCO)N.C(C(C)(C)CNC(=O)C(C)NC(C1CCC1)=O)N(CC)CC c1(C(N2CCC3(CCCN(C(C4CCC4)=O)C3)C2)=O)ccnc2cc(F)cnc12 N1(C(CCc2c(C)nn(C)c2C)=O)CC2CCOC2(CNC(=O)C=CBr)C1 C1(C(N2C3CN(C(C4(O)CCCCC4)=O)C(CC3)C2)=O)COc2ccccc2O1 CCS(=O)(=O)CC(=O)NC1CCN(C(c2ccc(Br)c(C)n2)=O)CC1C C1(C(=O)NC(CC)C2CCC2)CC1C1CN(C(C2(C#N)CCOCC2)=O)C1 C(=O)(CC1=Cc2ccccc2C1)N(C(C)CCNC(C1(C(F)F)CCCC1)=O)C C1(OC)CCC(NC(C2(NC(c3nccn3C)=O)CCSC2)=O)CC1 C1(CC(=O)N(C2(CC3CC3)CCC2)C)CCCN(C(c2ccc([N+](=O)[O-])[nH]2)=O)CC1 c1(C(=O)OC)ccc2c(c1)CN(C(C1(C#N)CCC1)=O)CC2 C1(C2CN(C(C3Cc4cscc4C3)=O)C2)(NC(c2cc(C3CC3)ns2)=O)CC1 c1(C(=O)NCCSC)c(CNC(C2(C#N)CCCO2)=O)nnn1C c1(NC(=O)CCCCN2CCOCC2)cccc2c1CCC2 c1(C(=O)NCC(CNC(C2(CC#C)CCOC2)=O)F)cnc2cccnn12 C(=O)(C1CSc2ccccc21)NCCC1(O)CCN(C(C#CC(C)(C)C)=O)CC1 n1(C(C)C)nc(C(N2CC3C(C(=O)NC4(C)CCC(F)C4)C3C2)=O)cc1C(=O)O N1(C(C2(COC)CC=CC2)=O)CC2(CC(C(=O)Nc3cncc(F)c3)CO2)C1 C1(CNC(c2c(C)nc(N(C)C)s2)=O)CCC(C)N(C(c2ccn(CF)n2)=O)C1 C1(C(=O)NCCOCCCN(C(C(COC)OC)=O)C)CCC2(CCC2)O1 c1(CNC(NCC(=O)NCC#C)=NCCCCl)noc2c1CC(C)CC2 c1(CCCNC(C(C)N(C(=O)CCc2nc[nH]n2)C2CC2)=O)ccccc1 C(=O)(CC(F)(F)F)NCc1cccc(CN(C)Cc2nnn(C)n2)c1 C(=O)(C(C)C(C)NC(=O)CC1CCCCC1)NCc1cn(C(C)C)nc1 C(CCCCC(=O)NC(CC1CCCC1)C(=O)Nc1cnc(O)c(F)c1)OC C1(CC=C)(NC(C2CC(n3ccnn3)C2)=O)CCN(C(=O)C(C)SCCCC)CC1 N1(C(C23N(C(c4n(CCC)ncc4)=O)CCC2C3)=O)CC2(CCNC(=O)O2)C1 C1(NC(C(c2cnn(C)c2)NC(C(C)C2CC2)=O)=O)CCCC(O)C1O C=CC(C(=O)N(C)CCOCCNC(c1n[nH]cc1F)=O)c1ccccc1 c1(C(=O)NC(C(=O)NC(CC#C)C(N)=O)CCSC)ccc(C=C)cc1 C1(NC(CC=CC=C)=O)CN(C(=O)CC(C)F)C2(CCCCCC2)C1 N1(C(c2c(C)cco2)=O)CCC2CCN(C(=O)CCCc3cccnc3)CC2C1 OC1c2ccccc2CC1n1cc(CSc2ncnc(C(F)(F)F)c2Br)nn1 C12(CNC(c3c(C)n[nH]c3)=O)CN(C(c3occ4c3CCOC4)=O)CC1CCO2 c1(CC)cc(OCC(=O)NC2(C)CCN(C(=O)CC=C(C)C)C2)ccc1Cl CC1C(=O)CCC1CC(N1CCC(C(C)NC(=O)CC2CCCCCC2)CC1)=O Cc1ccc(-n2cncc2C(=O)NCC2CCN(C(c3cc[nH]n3)=O)CC2)cc1 Cc1nc(C)c(CC(=O)NCC2C=CC(NC(=O)Cc3cncc(F)c3)C2)s1 c1(C(N2CC(C)C(NC(c3cc(C4CCC4)on3)=O)C2)=O)cc2sccc2cn1 C(=O)(N1CC2COCC2O1)C1N(C(C(C(C)C)O)=O)CCCC1(C)C Cn1cc(NC(=O)CC2CNC(C)(C)C2)c(O)nc1=O C(=O)(N=c1ncn(Cc2cccc(F)c2)[nH]1)c1ccc(OCC)cc1 c1(C(N2C(CC)CN(Cc3ccn(CC)n3)CC2)=O)ccc([Si](C)(C)C)cc1 C(=O)(CN=c1ccc(Cl)n[nH]1)NC(C(=O)OC(C)(C)C)Cc1ccccc1 N1(C(CC(C)N(C(c2nc(CC)sc2)=O)C)=O)CC2CC(C1)C2(C)C c1(CNC(N2CC(N3CCCCC3=O)C2)=O)ncc(C2CCCCC2)cn1 C1(C(=O)NC2(CF)CCN(C(c3cccc(Cl)c3F)=O)C2)C2CCC(F)(F)C12 c1(C(=O)NC2(C)CCN(C(=O)CN3CCCCCC3)C2)ccnc2c1CC(=O)N2 c1(C(N2CCC3CCN(C(c4ccco4)=O)CC32)=O)cc2ncccc2cc1Cl N1(C(c2c(OC)noc2C)=O)C(C)C2CC1C2NC(c1c[nH]c(=N)s1)=O C1(C(N2CC(CC)C2)=O)CC(C)N1C(C1(C)CC(=O)C1)=O C1(C(=O)NCCOCC(N2C(C)(COC)CCC2)=O)CC2CC1CC2O N1(C(CCC=CC)=O)CCC(CCO)(CO)C1 C(C(CNC(C1(C(F)F)CCCO1)=O)S(C)(=O)=O)NC(c1ccn(C)c1)=O C(CN=c1[nH]c(=NC2COC(C3CC3)C2)[nH]c2cccnc12)N1C(=O)COCC1 C1(CNC(C(CC)(C)C)=O)CCC2(CCC2)C1NC(c1ccc2occc2n1)=O C1(CNC(C2(C#N)CCCO2)=O)CC2CCC1N2C(=O)Cc1ccc(Cl)cc1 C1(CC(C(=O)NCCCC)N(CC(C)C(=O)OC)CCC#N)CCCCN1CC c1(C(=O)NC2CN(C(c3cnn4ccsc34)=O)CCC2O)nc2cnccc2s1 c1(C(=O)NC2CC(C(C(=O)NC(c3ncc[nH]3)C)F)C2)cc(C(N)=O)co1 C1(NC(C(C)(C)C2CCC2)=O)CCCC(NC(C2(c3ncccc3F)CC2)=O)C1 C1(NC(C2CC2(Cl)Cl)=O)CC2CC1N(C(c1ccn(CCF)n1)=O)C2 c1(CC)c(C(=O)NC(CNC(c2cocn2)=O)CO)cccc1C C(=O)(CC(C(CC)CC)NC(C)=O)NCC(CC)NC(CCOCCOCC)=O C1(CNC(CCC#CC)=O)CCCCCN1C(=O)CNc1ccccc1OCC C1(CC(=O)NCC(CC)N(C)C)CC(C)(C)CN1C(=O)CC1CNC(=O)O1 C1(C(=O)NCC(CN(C(CCOCC#C)=O)C)C)CCCCC1n1cccc1 C1(COC)CN(C(=O)C(OC)OC)CCN1C(c1nc(=N)cc[nH]1)=O C1(C(=O)NCc2cn(C3CN(C(c4ccns4)=O)C3)nn2)CC2CCC1O2 CC1(C)COCC1CC(=O)NCCCCCNC(c1snc(O)c1Cl)=O C1(CNC(c2c(CC)nns2)=O)CC2CC(C1)N(C(c1c[nH]nc1C)=O)C2 c1(C(N)=O)cc(C(=O)NCC(CO)NC(c2cc(-c3ccco3)c[nH]2)=O)co1 N1(C(c2c(C)ccc(I)c2)=O)CCc2cc(C(N3CC4CC4C3)=O)ccc2C1 c1(CC)csc(CNC(=O)CCC2CCCN2C(=O)C(CSC)OC)n1 N1(C(c2cc(C)[nH]n2)=O)CCN(C(=O)COCP(C)(C)=O)CC1CC(F)F c1(OC)ccc(-n2nnnc2C(c2occc2Br)NC(C)CC2CCC2)c(C)c1 N1(C(c2c(=N)[nH][nH]c2)=O)CCC2(CCC2)C(NC(C2CCCC(F)(F)C2)=O)C1 c1(C(=O)NCC2=CCN(C(c3c(C)nc(N)cn3)=O)CC2)cccc2nn[nH]c12 N1(C(CC=C=C)=O)CCCC2CN(C(C3(OCC)CCSCC3)=O)CCC12 Cc1cnnc(O)c1C(N1CC2(NC(C3CCCN3C3CC3)=O)CC1C2)=O C1(COC)C=CCCN1C(C1(NC(=O)CCCNC(=O)NC)CCCC1C)=O S(=O)(=O)(c1cc(C(=O)N=c2ccn(C3CC3(F)F)[nH]2)ccc1Cl)NC(=O)C1CC1 CC(C(=O)NC(C)(C)CCCNC(c1ccon1)=O)C(F)(F)F c1(CC)ccc(C(=O)NC2CC(C)N(C(=O)CCC(C)CN(C)C)C2)c(C)c1 NC(=O)CCCCC(=O)NC(Cc1cn[nH]c1)C(=O)NCC(O)CNC(N)=O CCC(C(=O)NCCCOCCC(=O)N(CCOCCO)CC)C(C)(C)CC CC(C)(C(=O)NCC(CNC(C1CC2C=CC1O2)=O)C(F)(F)F)C1=CCSCC1 N1(C(C)=O)CC(CO)CC1(C)C.C1(=O)C(O)(C(F)(F)F)c2cn(nn2)CCN1C C1(O)(C(C)C)CCCN(C(=O)CC2COCCN2C(c2ccncc2O)=O)C1 CCC(CC(=O)NCCC(O)C(C)C)N(C(=O)C(c1ccn(C)c1)C)C c1(NC(=O)OCC)ccc(C(=O)N(C(C)CNC(=O)CSCCCCCC)C)s1 C(CC1c2ccccc2CCN1C(C1CCCCC1)=O)NC(=O)CO C1(NC(Cc2c(C)ncs2)=O)CCCC(N(C)C(c2ccc(C(F)F)cc2)=O)C1 CC1(C)CCc2onc(C(=O)NCCC3CN(C(=O)C=Cc4ccsc4)C3)c2C1 Cc1sc(C(N2CCC(C)(NC(c3cc4occc4[nH]3)=O)C2)=O)c(C)c1C CN1CCCC1CC(=O)N(C(c1cccnc1)C(=O)NCC1CC1[N+](=O)[O-])C1CC1 C1(N(C(=O)CSCC(=O)Nc2cccnc2)C)CCCN(C(C2CCCS2)=O)C1 C1(CC=C)(C(=O)NCCCc2ccco2)CCCN1C(c1cn(C)c(C)n1)=O C(C)(C)(CC(F)C(=O)N1CCN(C(C)(C)C)CC1)NC(C(C(COC)C)C)=O C1(CNC(C2(C3N(C(c4c(C)nns4)=O)CCC3)CC2)=O)CCCNC1=O N1(C(C(C(C)(C)C)O)=O)CCC(C2CN(C(=O)CCCNC(=O)C3CC3)C2)CC1 N1(C(c2cccc(C#C)c2)=O)CC2CC(C1)CN(C(c1cnn3ccsc13)=O)C2 N1(C(c2ccn(C)c2)=O)CC2CCN(C(c3cc(F)cc(Cl)c3)=O)CC2C1 n1(CC(=O)NCCC2(O)CCN(C(C(C)SCC)=O)C2)cnc2ccccc12 Cc1ccc(C(N2CC=CC2CNC(C2(C)CCC(=O)N(C)C2)=O)=O)c(N)c1C N1(C(C2CCC(C)(C)C2)=O)CCOC(C)(CNC(=O)Cc2csnn2)C1 C1(C2CN(C(=O)CCF)C2)(NC(=O)CC2CCCCC2F)CC1 c1(CC(=O)NC2CC(CCNC(C3(OC)CCSC3)=O)C2)ccc(Cl)cn1 N1(C(c2c(C)cn(C)c2)=O)CC2CCN(C(c3cnc4[nH]ccc4n3)=O)CC12 C1(C(=O)NC(CC(=O)NCc2c(C)cncc2)C2CC2)CCOC(=O)CC1 CCC(C)(COC)C(=O)N(CC(C)(C)NC(c1nccn1C)=O)C Cc1cccc(C)c1C1C(NC(C(C2CCOC2)N(CCC#N)C)=O)C1 N1(C(CCC=C)=O)CC(C)CCC1C(=O)Nc1cccc(C(C)=O)c1 c1(C(C(=O)NCC(=C)C)N(C2CCC2)C(C)C)cnn2c1CCC2 c1(C(C)=O)ccc(CC(=O)NC2CCN(C(c3ccnnc3)=O)C2(C)C)cc1F c1(C(N(CCOCCO)CC)=O)occc1CNC(=O)C(C)C1CCC1 Cc1cc(C(=O)NC2CC(O)CN(C(c3ccnc(C4CC4)n3)=O)C2)cc(C)n1 Cc1cc(C(=O)NC2CCN(C(C3CCC(=O)N3)=O)CC2CO)c(N)c(Cl)n1 N1(C(c2nc(COC)oc2)=O)CCC(C(=O)NC2(C(=O)OC)CC2)C1(C)C C(N=c1cc(NCc2nc(-c3ccc(Cl)cc3)no2)nc[nH]1)c1n(CC)cnc1 c1(C(N2CC(NC(C3(C(F)(F)F)CC(=C)C3)=O)C(OC)C2)=O)ccc(F)c(C)c1 C1(C(=O)NCC2CC(NC(C3CCCSC3)=O)C2)CCn2cncc2C1 CC1=C(C(=O)N2CC(O)(CCNC(=O)C=Cc3ccc(C)o3)C2)CCCC1 O=C1Cc2cc(C(O)CN3CCC(Oc4ccccc4)CC3)ccc2N1 C12(CNC(CN(C)C)=O)CCC(CC1)N2C(c1cn(CC2CCOC2)nn1)=O CC1=C(C)CC(C)(C(N2C3CCC2CC(NC(c2cnc(C)cn2)=O)C3)=O)CC1 C1(NC(C(C)OCC(C)C)=O)(CO)CCCN(C(c2ncsc2C(F)(F)F)=O)C1 Cc1nn(C)c(N)c1C(=O)NC1C=CC(C(N2CCCC(C(N)=O)C2)=O)C1 C(=O)(CS(=O)(=O)CC(C)C)NCC1C(NC(COCC(=C)C)=O)CCC(C)(C)C1 N1(C(Cc2n[nH]c(=N)s2)=O)CCCCC(CNC(=O)C(c2ccccc2)F)C1 c1(CCC(C)C)noc(C(C)NC(=O)N(C2CC2)Cc2csc(Br)n2)n1 Cc1c(C(N2CC(O)(C(F)C(=O)N3CCC3CC3CC3)C2)=O)cccc1F C(=O)(C(O)C(C)(C)C)N(CCC(=O)NCCN1CCCOCC1)C N1(C(CC)=O)CC2CS(=O)(=O)CC2(CNC(C2(OC)CC2)=O)C1 c1(C(N2CC(NC(=O)C(O)c3ccco3)C3(C2)CC3)=O)cccc2nc(O)[nH]c12 C1(C(=O)NCCCNC(c2ccnc(N3CCCC3)c2)=O)CCN(C2CC2)C1=O C1(O)(CNC(C2C(CC(C)(C)C)C2)=O)CN(C(C2CC3CC3C2)=O)C1 C1(CNC(Cc2c(C)ocn2)=O)C(O)C(O)CN1C(c1cncc(Br)c1)=O n1(CC(=O)NCC2CCCC2NC(C23CC(CO2)C3)=O)cc(Cl)cn1 c1(C(=O)NC23CN(C(C(C)c4ccco4)=O)C(CC2)C3)cccc2[nH]ccc12 C(=O)(C1=CCC(C)(C)CC1)NC1(CF)CCN(C(CCCCCOCC)=O)C1 c1(C(=O)NCC(C2CCCCC2)C)cc(C2CC2)nn1-c1ccc(Br)cc1 Cc1c[nH]c2cc(C(=O)NC3CCN(Cc4c(F)cccc4I)CC3F)ccc12 C1(C(N(C2CCCN(C(C(F)=C(C)C)=O)C2)CCO)=O)CCc2c[nH]nc2C1 C1(O)(CN(C(CN2CC(C)C2)=O)C)CCN(C(C2C3COCC23)=O)C1 c1(C(N2C(C)C(NC(c3ccc(CCF)cc3)=O)CC2)=O)c[nH]nc1S(N)(=O)=O CCCCCCCCCC(=O)NC12CC1CN(C(C1CN=C3N=CNN3C1)=O)C2 C12(CNC(C(CC)n3ccnc3)=O)CC(CO1)N(C(c1c[nH]c(=NC)o1)=O)C2 CC1CCC=C1C(=O)NCCCOCCOCCNC(c1cc(Cl)cnc1O)=O C1(C(=O)NCc2c(C)coc2C)CN(C(c2cnsc2)=O)C2(CCC2)C1 CC(C)(C(=O)N1CC2CC2(CNC(c2c[nH]c(C(F)(F)F)c2)=O)C1)C(N)=O C1(C)(NC(CN(C)CCc2ccccc2)=O)CCN(C(C2CC2F)=O)C1 C=CC(CCC)CC(=O)NC(CNC(c1ccc(CC)[nH]1)=O)CC(C)C c1(C(N2CCCC(NC(C(CCC)O)=O)C2)=O)ccc2sc3ccccc3c2c1 c1(C(CNC(N2CCC(c3ccc(C)cc3)(C)C2)=O)O)cccc(Cl)c1C c1(NCC(CC)(C)COC)ncnc(N2CCN(C3CN(C)C3)CC2)c1C C1(CCC(=O)NC(C(=O)NC(C)C)C)CCC(NC(=O)C(C)N(C)C)C1 c1(C(=O)NCC2(CCNC(C3C(C)OCC3)=O)CC2)ncn2ccccc12 c1(OCC)ccc(C(=O)NC2CSCCN2C(=O)C(O)CC)cc1[N+](=O)[O-] Nc1c(C(N2CCNC(C(F)(F)F)C2)=O)ccc(F)c1Br Cc1ccc(C(=O)NCC2C3CN(C(c4nc(Cl)cs4)=O)CC23)c(F)c1F Cc1ccc(N2CCCC2COC(=O)C(c2ccc(C)cc2)N(C)C)cc1 N1(C(c2cc(CC)on2)=O)CCCN(C(=O)CN2CCCC2CO)CCC1 C(=O)(CCC(C(N)=O)NC(N1CCN(CCS(C)(=O)=O)CC1)=O)OC(C)(C)C C1(C(N2CC(NC(c3cc(CCC)oc3C)=O)C(C)C2)=O)C2CCC(C2)C1(C)C c1(NC(c2c(C3CC3)ccc(OC)c2)=O)cccc(S(C)=O)c1 C1(O)(C(=O)NC2C(NC(C3(C)CC4CCC3O4)=O)CCC2)CC2(CCOCC2)C1 C1(C(=O)NC2(CC=C)CCN(C(c3ccc(CO)cn3)=O)C2)CCCCC(=O)N1 c1(C(=O)NCCN(C(C(CC(N)=O)O)=O)CC2CC2)cnc2c(c1)NC(=O)CN2 C(=O)(CCCCCC(C)C)NC(CC#C)(C)C(=O)N(C)CC1CCN(C)C1 n1(CC(=O)NCCC2CCC(NC(C3(CC)CC3)=O)C2)ccc2cc(F)ccc12 C1(C(N(CC(CC)NC(c2cnn(CC)c2C)=O)C)=O)C=CC=CC=C1 C1(C)(C(N2CC(C)N(C(=O)C(F)=CCCF)CC2)=O)Cc2ccccc2C1 C1(NC(c2c(CCC)[nH]cc2)=O)(CO)CCN(C(=O)CN2C(=O)CNC2=O)CC1 C(=O)(CC1=CCCCC1)N1C(C2(NC(C(c3cccc(C)c3)C)=O)CC2)CCC1 c1(C(=O)NCC(CC)NC(=O)CN2CCOCC2=O)ccc(NC(C)=O)cc1Cl C12(CNC(c3c(COC)cccn3)=O)CCC(CN1C(=O)CCn1cnnn1)C2 O=C1CCc2cc(C(N3CC4CC3CN4C(C3CC3(Cl)Cl)=O)=O)ccc21 c1(C(=O)NC23COC(CNC(C4CC4(Cl)Cl)=O)(C2)C3)c(F)cc(F)cc1F Cc1ccc2c(CN3CC4(CCN4C(c4ccncc4)=O)C3)c[nH]c2c1 C1(NC(c2ccc(CSCC)cc2)=O)CCCN(C(c2conc2C)=O)CC1F N1(C(c2c(CC)occ2)=O)CC2CCN(C(c3ccc(C(F)F)cc3F)=O)CC12 CCCCCC(O)CC(=O)NC(C1(C(=O)OCC)CCCC1)C c1(OC)ccc(F)cc1-c1nc(C(=O)Nc2cc(C3CCCCC3)no2)cs1 C(=O)(CC(F)(F)CC(=O)OC)N1CCN(C(c2ccn(CC)n2)=O)CC1CF C1(C)(NC(C(C(C)C)SC)=O)CCN(C(=O)CCNc2ccccc2O)CC1 C(N=c1[nH]c(Cl)ncc1Cl)C1CCN(C(c2cnc(C)o2)=O)CC1C c1(NC(C(CC#C)N(C(C)C(=O)N(C)C)C)=O)cccc2ccoc12.OC Cc1ccc2c(c1C(=O)NCC(O)CN(C(=O)C1=CCCCC1C)C)CCCN2 C1(NC(=O)CCn2cc(CNC3CCC3)nn2)CC(O)C(O)CO1 c1(C(=O)NC2CCC2)cccnc1CNC(C1CCCCC1F)=O CCC(C)(C(=O)NC1CN(C(=O)COCC2CCCC2)C1)OC C1(CNC(C2(NC(C)C)CC2)=O)CC(NC(=O)C=CBr)C1(C)C c1(CC(=O)NC2CC(NC(c3cccc4nncn34)=O)C2)ccc2c(c1)COC2 c1(C(=O)NCC(C(C)(C)C)NC(C2=CC(C)(C)C2)=O)cc([N+](=O)[O-])c(F)cc1N c1(CNc2ccc(-c3c(C#N)nccc3)nc2)c(Cl)ccc(F)c1F C1(CNC(C(C)=CC2CC2)=O)CC2(CCC2)CN1C(c1ccc(F)c(N)c1F)=O C=C(C)C1OCCC1C(N1CCC(CO)(NC(c2cncc(CC)c2)=O)C1)=O CC1=CC(C)=NS(=O)(=O)N1CC(N1CC(NC(=O)C(C#N)C(C)(C)C)C(C)C1)=O c1(CC)cn2c(n1)CC(C(=O)NCCNC(c1cccc(COC)c1)=O)CC2 n1(CCC(=O)NC2CCN(C(c3c(C)nns3)=O)C23CC3)ccc2ccccc12 c1(C(=O)NCC2CC(NC(COCC)=O)C2)ccc(F)cc1OC N1(C(c2c(C)cns2)=O)CCC(NC(=O)Cc2ccc(Cl)nc2)CC1C N1(C(C=C2CCN(C)C2)=O)CCOC2(C1)CN(C(=O)CCn1cnnn1)C2 N#Cc1c(N2CCC(C3(NC(C4CCCC4O)=O)CC3)C2)cccc1F N1(C(CNC(CCC)=O)=O)CCCC1CN(C)C(C1(N2CCC2)CCC1)=O Cc1ccnc(C)c1C(=O)NCC1CCCC(NC(C2CC2c2cn[nH]c2)=O)C1 C(C(O)CC(F)(F)F)NC(CC1CCCC(NC(c2cn(C(C)C)nn2)=O)C1)=O N1(C(CC(CC)C)=O)CCCC2C1CCN2C(=O)CCCCCl C(=O)(N=c1[nH]n(C)cc1P(C)(C)=O)NC1C(CC)CN(S(=O)(=O)C(C)C)CC1 Cc1csc2c(C(=O)NC(C)CC(C)NC(C3(C#N)CCSCC3)=O)ncnc12 N1(C(C=CC(C)C)=O)CCOC2(CCN(C(C3CCOC(=O)N3)=O)CC2)C1 c1(C(=O)NCCC(CNC(c2csc(Cl)n2)=O)O)c[nH]c(=O)c2ccnn12 C1(CC)CN(C(=O)C(C)CC(C)C)CCC1CNC(c1cn(CC)nn1)=O C1(NC(C(C)c2cc[nH]n2)=O)CC2(C1)CC(C(=O)N(C1CC1)CC1CC1)C2 S(=O)(=O)(c1ccc(C)cc1)NCC(=O)NCCOCC1CCCC(C(=O)OC)C1 C(c1cc(F)cc2c1OCOC2)=CC(NOCCCC)=O c1(OC)cnnc(C(N2CCC(CCC(=O)N(CCN=[N+]=[N-])C)CC2)=O)c1 C#CC1CN(C(C2(C#C)CN(C(c3cnncc3O)=O)C2)=O)CCO1 C(=O)(CCCC(=O)N1CCCC(n2ccnn2)CC1)N(c1c(C)cccc1)C C1(CNC(c2c(OC)csc2)=O)CC(NC(=O)C=C(C)Cl)C1(C)C Cc1ccc(C)c(C(N2CC(CNC(=O)Cc3csc(Cl)n3)CCC2C)=O)n1 c1(C(=O)NC2C(NC(C3(C)COC3)=O)CCCC2)ccc(Br)c(Cl)c1 C1(NC(CC(C)SC)=O)CC2(C1)CC(NC(=O)Cc1c(Cl)cccc1Cl)C2 c1(C(=O)NC2CC(C(=O)NC(CC#C)CC#C)CC2O)ccc([N+](=O)[O-])[nH]1 c1(C(=O)NC2CCN(C(CSCC)=O)C(C)C2)ccc(C)c(Cl)c1Cl N1(C(c2ccc(C(C)=O)cc2)=O)CCC2C(NC(c3ncn(C)n3)=O)C2CC1 c1(N(C(CC=O)=O)C)cc(Cl)c(Cl)n1C.CC(CCO)N(CCCN(C)C=O)C N1(C(CN(C(CCC)=O)Cc2ncc(Br)s2)=O)CCCC1C(C)(C)CN1CCC1 N1(C(C)=O)CC(O)CC1C(N1CC2(NC(=O)CSc3ccccc3)CC1C2)=O C1(C(=O)NC2(CC)CC2)CNC(=O)CN1C(=O)CC1CC2CC2C1 Cc1nn(C)c(NC(=O)NC2(O)CC(CO)C2)c1-c1ccccc1 N1(C(c2cc(OC)c(Br)s2)=O)CCC(C)(CCc2cn(C3CCOC3)nn2)CC1 c1(CNC(C2CCOCC2)=O)cn(CCNC(C2(C(F)F)CC(O)C2)=O)nn1 CC(Cc1ccccn1)C(=O)N1CCCC1CNCC(=O)OCC12CNCC1C2 N1(C(C(N2CCCCCC2)C)=O)C2CCC1CN(C(C1CC1C(C)(F)F)=O)C2 C(CNC(c1cnn(C2CCC2)n1)=O)(C(C)(C)C)NC(CCC1C(C)C1)=O C1(C(=O)NC2C(OC)CN(C(c3cc[nH]n3)=O)C2)CC(=O)NC(=O)N1 C(=O)(C1CCc2c(Cl)cccc21)N1CC(O)(CNC(C(C(C)(C)F)(C)F)=O)C1 c1(CCC(=O)NCC2CCC(NC(=O)CNC(=O)C3CC3)C2)cccnc1Cl C1(F)(C(=O)NC2CCN(C(Cn3c(C)c(Cl)cn3)=O)C2)CCC2(CCC2)C1 C1(CNC(CC(C)SC)=O)CC(C)(C)CN1C(c1coc(N(C)C)n1)=O C1(C(=O)NCCN(C(CC2C(C)(C)C2)=O)C2CC2)CC2(CCOCC2)C1 C(C(=O)N1CC=CC(NC(=O)C(C)NC2(CO)CCCC2)C1)(C(C)(C)C)OC c1(CNC(=NCC(=C)C)NC2(C)CCCOC2)cc(OC)c(OC)cc1C N1(C(C)=O)CCC2CN(C(C3CCC=CCC3)=O)CCC2C1 N1(C(c2cc(C)c(C)o2)=O)CCCOC(CNC(=O)Cc2cc(F)cc(Cl)c2)C1 C1(C2N(C(CCOC(C)=O)=O)CCC2)CCCN(C(c2ccn(C)n2)=O)C1 C(=O)(C1CCc2snnc21)N1C(CNC(=O)C2=CCCOCC2)COCC1 c1(C(=O)NC(CNC(COC(C)C)=O)(C)C)coc(C(N)=O)c1 C(=O)(C1=CC2CC=CCC12)NCCC1(NC(c2c(CCC)nco2)=O)CC1 c1(OC)cc(C(=O)NCC2(F)CN(C(C3(OC)CCOC3)=O)C2)c(Cl)cn1 CC1CN(C(c2cc[nH]c2C2CC2)=O)CCC1N(C)C(c1ccnc(CO)c1)=O N#CCCCCCC(=O)N1CC(F)CC1CNC(=O)C=Cc1cccc(Cl)c1 c1(C(=O)NC2N(CCC)C(=O)CC2)ccccc1[N+](=O)[O-].C12(CC1)CN2 C1(C(N2CC(CCC#C)C2)=O)COC(CNC(=O)C(C)CN(C)C)C1 C(=O)(CC(C(F)F)N1CCOCC1)N1CCC(NC(=O)C2=CCOC2)C1 Cc1ccc(C(=O)NC2CCN(C(c3cccc(Cl)c3O)=O)C2C)cc1C N1(c2snc(CC)n2)CCOCC12COCCN(C(c1cc[nH]n1)=O)C2 CC(C)C(C#N)C(=O)N1CCC(CNC(=O)Cc2nn(C)cc2Cl)CC1C c1(C(=O)NC(CN(C(c2cc(C(C)C)ccc2F)=O)CC)C)cnc(N)c(N)c1 C=CC(CC)CC(=O)NC1CCN(C(c2ncsc2C)=O)CC1CC N1(C(C(F)OC)=O)CCC(O)(CNC(=O)C(C)(C)C(N)=O)CC1 CC1COCCC1N(C(=O)CC1CCCC1NC(=O)CC1(O)CCC1)C C(=O)(C(C(=O)NCC1CN(C(c2ccc(C(F)F)s2)=O)CC1O)OC)OC N1(C(CCCn2c(C)ncc2)=O)CCN(C(=O)CC2(C(F)(F)F)CC2)C(C)C1C S(=O)(=O)(c1cccnc1NCC1(CO)CC1)N(CCCC=C)C CC(C(=O)NC(CCF)C(=O)NC(CCO)C1CCCC1)C(F)(F)F N1(C(C(=O)NCCOC)=O)CC2(CC1CNC(c1occ(C)c1C)=O)CC2(F)F C1(N(C(C2CC3(CC3)C2)=O)CCF)CCCN(C(c2csc(C(F)F)c2)=O)C1 N1(C(C2(CC)CCCC2)=O)CC2(CNC(=O)CCc3cncc(F)c3)CC1CO2 CC#CCCC(=O)N(c1ccccc1)CCN(C(=O)Cc1cc(C)sc1C)CC N1(C(COc2cn(C)nc2)=O)CC2CC(NC(C3CC4COCC4C3)=O)C1C2 Cc1nn(C)cc1C1=NOC(C(=O)NC2CCN(C(=O)Cn3cccc3)CC2)C1 c1(C(C)C)ccc(O)cc1C(=O)NC1CC(NC(=O)CC2CCC(C3CC3)O2)C1 Cc1oc(C(C)C)nc1OC(N1CCC(SC(C)(C)C)C1)=O C=CC1CN(C(=O)CN(C)C(C)C)CC1NC(c1ccc(-n2cccc2)nc1)=O C1(CC=C)(NC(=O)CNC(N)=O)CN(C(=O)C(CC)n2cncn2)C1 C1(CNC(C2CC2(Cl)Cl)=O)CCN(C(c2csc3nnsc23)=O)C12CC2 CCC(C(=O)N1CC(NC(C2(OC)CCCC2)=O)C1)n1nccc1C C(CC(F)F)(C(=O)NC(CCC)CCO)N(C(CC(C=C)C)=O)C C12(CNC(CCCC(N)=O)=O)CN(C(c3ccc4cnoc4c3)=O)CC1CCO2 C1(NC(CC(n2ccc(C)n2)C)=O)CCN(c2snc(C)c2C#N)CC(C)(C)C1 C1(NC(CCCCN(C)C)=O)CCN(C(=O)Cn2cc(C3CC3)nn2)CC1F C1(NC(C(C)CN(C)C)=O)CC2CC1CN(C(=O)CCCC1CC1)C2 c1(CCCC(=O)NC(CN(C)C(C2CC3CCC3C2)=O)(C)C)ccc(Cl)cc1 C1(NC(C2CCN(C(=O)NCC(F)(F)F)C2)=O)C2CCN1CC2 C(C(C(C)C)NC(=O)C(Cc1ccco1)NC(=O)COC(C)(C)C)OC c1(NC)ccc(C(=O)NCC(C)(CNC(C2CC(n3cccn3)C2)=O)OC)nc1 CCCCCCCC(=O)N1CCCCC(NC(=O)CN2CCOCC2)CC1 c1(OCC)ccccc1OCC(=O)NCC1CCN(C(c2nn(C)cc2Cl)=O)C1 C1(NC(c2c(C)csn2)=O)CCCC(NC(C2(C)CCNC2=O)=O)C1 c1(C(=O)NC2CCN(C(c3cc(C)ncc3)=O)C(C)C2)c[nH]nc1S(N)(=O)=O c1(C(=O)NCC(C)(C2CC2)NC(C2N(CC)CCC2)=O)cc(N)c(F)cn1 N12CCN(C)CC1C(=O)OCC(O)C2.C(CN(C)C)OCC C(=O)(CC(C(F)(F)F)NC(=O)CC=C(C)C)N1CCC(CC#C)CC1 c1(C(=O)NCC(CNC(C2N(C(C(C)C)=O)CCC2)=O)C)cnn2ncccc12 C(=O)(CS(=O)(=O)C(C)(C)C)NC1CCCN(C(C(C(C)C)OCC)=O)CC1 C1(O)(c2cn(CCC(C)C)nn2)CCN(C(C2COC(C)(C)C2)=O)CC1 c1(C(=O)NCC2CN(C(C(C)SC)=O)CC(C)(C)C2)ccc(S(C)(=O)=O)cc1Cl C1(NC(c2cc(OC)ncc2F)=O)COC2(C1)CN(C(c1ccc[nH]1)=O)C2 N1(C(C(CCC#C)O)=O)CC2CCC(C1)N2C(=O)C(CCC)NC(N)=O c1(CCC(=O)N(CCCNC(c2c(C)onc2)=O)C)c(C)nc2ccnn2c1C C(=O)(CCC(C)(C)C(=O)N1CCC(C)C(CNC(C2(C(F)F)CCC2)=O)C1)OC Cc1ccc(CNC(C2CC23CN(C(=O)CCC(=O)OC(C)(C)C)C3)=O)nc1 c1(OC)cccc(NC(=O)C(c2ccc(Cl)nc2)N(C2(C)CC2)C)c1 C1(c2nc(-c3cc(-c4ccncc4)[nH]n3)no2)(OCC)CCOCC1 CCC(CNC(=O)C(C)CNC(C1OCCOC1C)=O)(CC)OC CC1CC(CCNC(c2cc(O)cc(Cl)c2)=O)CCN1C(=O)Cn1cnnn1 N1(Cc2onc(C)n2)CCC(NC(C2(C)CCCC2C)=O)C(C)(C)C1 N1(C(C(CC)C(C)C)=O)CCN(C(c2csc(O)n2)=O)CC(O)C1 O=C1COc2cc(C(=O)NC3CCN(C(c4ccc(Cl)nc4O)=O)C3)ncc2N1 C=CCCC(C(=O)NCC(Cl)=CCl)NC(C1CC=C(C)CC1)=O C1(CN(C(C2CCCOCC2)=O)CC)CCN(C(=O)C#CC(=O)N(C)C)CC1 C1(NC(c2nc(COC)oc2)=O)CC2CC1CC2C(N1CCCC(C#N)C1)=O C1(C(c2n(CCOC)nnn2)NC(c2c(C)noc2C)C(C)C)CCOC(C)(C)C1 Cc1nn2c(c1C(=O)N(CCCNC(c1[nH]ccc1C1CC1)=O)C)CCCC2C N1(C(C2OCCN(C)C2)=O)CCN(C(=O)COc2ccccc2O)C2COCC12 C(=O)(C(c1cccs1)NC(=O)C(=O)NC(C)C)N(CC=C)CC=C C12(CC)CN(C(=O)C(O)COc3ccc(OC)cc3)C(CNC(=O)C(C)O)(C1)C2 N1(C(C(C)=C2CCC2)=O)CCCC1(C)CNC(c1ccnc(C(N)=O)c1)=O C(C(C)(C)CC(=O)NC1C=CCCC1C(=O)NC1CN(C)CC12CC2)OC N1(C(CCC#CC)=O)CC2CCCC2(NC(c2cc(OC)ns2)=O)C1 C1(NC(c2c(C)ccs2)=O)CC(O)CN(C(=O)CC2CCC2)C1 C(C1=CCCOC1)NC(C1C(CNC(C(C)(C)C2CC2)=O)OCC1)=O c1(CC)ccoc1C(=O)NCC(C)(CC)NC(c1cnc(C(F)F)s1)=O c1(CC)cc(C(=O)NC(C(=O)NCCc2nccc(C)n2)C2(O)CCC2)c(C)o1 c1(CSCCNC(C=CCNC(C2CC2)=O)=O)ccc[nH]1.CC N1(C(CCC)=O)CC(CNC(=O)C(C)Sc2ccccc2)CC(C)(C)C1 CC1C(C)N(C(=O)CN(C)S(=O)(=O)N(C)C)CCN1C(C1CC(O)C1)=O CCC(C)(C)C(=O)C(=O)NCC(C(=O)NCCN1CCNC1=O)N(C)C c1(C(=O)NC(CCCNC(c2cn(C)nc2Cl)=O)(C)C)coc2cc(O)ccc12 CC1CCCC(OCC(=O)NC2(NC(=O)CN3CCC(O)CC3)CCCCC2)C1 N1(C(C=CC=CCC)=O)CCC2(CCCN2c2ncc([N+](=O)[O-])cc2F)C1 c1(OC)ccc(C(=O)O)c(C(F)(F)F)c1.c12ccc(cc1)CC(=O)N1CCC2C1 N1(C(C(C2CCC2)OCC)=O)CCC(C(C)(C)NC(=O)C(C)n2ccnc2)CC1 c1(OC(C)C)cc(C(N2CCC(CNC(C3CCC(C)S3)=O)CC2)=O)ccn1 CC(C)(C(F)(F)F)NC(C1CCN1C(=O)CC1CCCNC1=O)=O c1(C(=O)NC2C3(CCN(C(C4C(=C)C4)=O)C2)CCC3)ccccc1C#CC1CC1 CC(C)CC(CC(C)C)C(=O)NC1C2CCN(C(=O)C(C)N3CCC3)CC12 N1(C(CC2(OCC)CC2)=O)CCCCCC1C(=O)Nc1cc(C)cc(Cl)c1 Cc1cc(C(=O)NCC2CCN2C(=O)C=CCOc2ccccc2)cnc1O C1(CNC(C2(CC(C)C)COC2)=O)(NC(C2CCCCO2)=O)CCCCCC1 c1(C(N2CC=CC(NC(C3C(C=C(C)C)C3(C)C)=O)C2)=O)ccccc1N=[N+]=[N-] c1(C(N2C3CC(NC(c4c(C)oc(C)c4C)=O)C2CC3)=O)cn2ccnc2cn1 c1(CC)cncc(C(=O)NC(CNC(c2cnn(C)c2)=O)(CC)CC)c1 Cc1ncc(NC(=O)CSCCNC(=O)COCc2cnn(C)c2)n1C Cc1cccc(C)c1CNC(C1CN(C)CCN1C(C1CC(C)(O)C1)=O)=O C1(NC2C(NC(C3(c4ccc(O)cc4)CC3)=O)CC2)CCN(C2CC2)CC1 C=CC(C(F)(F)F)NC(C1CC(O)CN1C(=O)CCC1CC1(F)F)=O N1(C(C=CC(CC)=CC)=O)CCN(C(c2cc(C)n(C)n2)=O)CC1CC(F)F c1(OC)cc(C)cc(C(=O)NCCC(C)NC(=O)CCCC(=O)NC(C)C)c1N Cc1cc(O)ccc1CNC(=O)CC1CCN1C(=O)C=CCN1CCC1 c1(C(N2CC(CNC(C(C(=O)OC)C)=O)C2)=O)csc2ccc(F)cc12 c1(NC(C23C(CN(C(c4c(C)ncnc4)=O)C2)C3)=O)nn(C)c2ncc(I)cc12 c1(C(=O)NCC(CNC(C2(OC)CCCC2)=O)(C)C)sc2cccc(F)c2c1Cl c1(C(N2CC(C)CC(NC(c3c(OC)csc3)=O)C2)=O)ccc2c[nH]nc2c1 c1(Oc2c(Cl)ccc(C)c2)ccc(C#N)cc1Cl C(CCOC(C)C)(C(C)C)(c1n(CCCCCC)nnn1)NCCCOC Cc1ccn(C)c1C(N1CCC(NC(c2ccc(OC3CCOC3)cc2)=O)C1)=O CC#CCC(C(=O)N1CCCC(C(=O)OC)C1)NC(=O)C(C(=O)OC)OC N1(C(c2c(CC)n(C)nc2)=O)CCCC(N(C)C(c2occc2C)=O)CC1 C(=O)(CCN=c1ccc(C)c[nH]1)NCC(CC)NC(c1cccc(Cl)c1C)=O N1(C(c2cc(C)cc(C)c2N)=O)CCN(C(=O)CC(=O)NC2CC2)CC2(CC2)C1 C1(NC(C(CSCC)NC(C2C(OCC)CC2)=O)=O)CC2C=CC1C2 C1(NC(COC(CC)C)=O)CCCCCC1NC(c1nc[nH]c1C(C)(C)C)=O c1(C(N2CCC(CCNC(C=C(C)Cl)=O)C2)=O)cn2c(n1)C(C)CCC2 c1(NC2CCC(OC)CC2)ncc(C)cc1S(=O)(=O)NCC1CCOC(C)(C)C1 N1(C(c2ccc(C)s2)=O)CCC(C(N2CC(c3ccccc3C)(O)C2)=O)CC1 C1(C(=O)NC(C2CCN(C(c3n(C=C)nnc3)=O)C2)(C)C)CCn2cnnc2C1 C(C(=O)NCCOC1CN(C(=O)C(c2ccccc2)O)C1)(C(C)C)NC(=O)OC CC1CN(C(C2CCC(C(=O)NC(c3ccc(O)c(F)c3)=O)O2)=O)CC1(C)CO N1(C(CCN(C)CCO)=O)CCC2(CC1)CC2CNC(=O)C=CCO C(C(=O)N=c1cc(OC)n(C)[nH]1)CCC.C1(N2C(=O)CS2)CCN(C(C)C)C1 c1(NC(C(=O)NC2CN(C(C(=C)Cl)=O)CC2C)=O)ccc(C)c(C)c1 C#Cc1cn(C)nc1C(=O)N(CCCCCNC(c1cn(C)nn1)=O)C(C)C CC1(O)CCN(CC(N2CC=CC(NC(=O)CCN3CCCS3(=O)=O)C2)=O)C1 N1(C(C(C)Oc2ccccc2)=O)CC(CNCC(=O)Nc2cn[nH]c2)C(F)(F)C1 CCN(Cc1ccc2ccccc2c1)N1CC2CC2(NC(=O)OC(C)(C)C)C1 C1(CNC(C(C)(C)OCC)=O)CCC2CN(C(c3cc(C)ns3)=O)CC12 c1(C(N(C(CCNC(c2ccc(OC)cc2F)=O)C)C)=O)ccn2ccccc12 C1(CNC(C(CCCC)C)=O)CCN(C(=O)CCSCC(N)=O)CCC1(F)F C1(C(=O)NC(C2(O)CCN(C(=O)CN3CCOC3=O)C2)C)CC2(C1)CC2F c1(C(N2CCOCC2c2ccc(Cl)cc2)C(=O)NCC(=C)C)cc(C)ccc1F CC(C)C(CO)ONC(=O)C=CCF.C1(C(=O)N)C=CCS1 c1(CSC)c(C(=O)NCC(c2ccc(F)cc2)N)oc2ccccc12 C1(C(C)(C)F)CCN(C(c2cc(Br)sc2Cl)=O)CC1 N1(C(CCN(C(C)C)C(c2ncccc2N)=O)=O)CCN(C)CC1C C1(C(N(C(C)CNC(c2cn(C)c(C(F)F)n2)=O)C)=O)CC(C(C)(C)C)=NO1 CC1CN(C(C2CCSCC2)=O)CCC1CNC(c1ccccc1C(F)(F)F)=O Cc1cc(CNC(=O)CC2CCSCC2)oc1C S(=O)(=O)(CC(=O)NCCN(C(=O)C=CS(C)=O)CC(C)O)NC C1(C(=O)NCC2CC(NC(C=CC(C)C)=O)CC2O)Cc2ccc(F)cc2O1 Cc1nc(CC(=O)NCC#CCNC(=O)CSC(F)F)c(C)s1 N1(C(CC(C)C)=O)CCCC2CN(NC3COc4ccccc4O3)CC12 C(CC(=O)N1CC2(CC(N(C)C)C2)C1)(C(F)F)NC(C(CC#C)O)=O C1(CS(C)(=O)=O)(n2cnnn2)CC(F)(F)C1.n12cc(nn1)C1CN(C1)C(=O)C2 C1(C(=O)NC2CN(C(c3nc(Cl)c(Cl)s3)=O)CC2O)CC2COCC2C1 c1(C(N2CCCC(C3(C)COC(=O)N3)C2)C(=O)NCCOC)cccc(CO)n1 Cn1nnc(=NS(=O)(=O)c2ccc(Cl)c(NC(c3cc(F)c(F)c(F)c3F)=O)c2)[nH]1 Cc1ncc(Cl)cc1NC(=O)N(C1CCCCC1(C)C)C C1(C(N(CCC(C)C)CCC(C)C)=O)C2CC1N(C(c1cc[nH]c1)=O)C2 C1(C(=O)NC2CCCC2c2ccc(C(F)(F)F)cc2)CCC(C=CCO)C1 C1(N(C(=O)CC2CC(=O)C2)CC)CCN(C(C2(SC)CC2)=O)C1 C1(NC(C)CCCCNC(=O)OC(C)(C)C)CCNC(=O)CC1 C1(C(=O)NCC(c2ccccc2)N(C(=O)CN2CC=CC2)C)CCCNC(=O)C1 c1(CNC(COCCCn2cc(C(C)O)nn2)=O)cnc2scnc2c1 C1(OC)(CNC(C2CNC(=O)C2)=O)CCN(C(=O)Cn2cnnc2)C1 C1(NC(Cc2c(C)noc2)=O)CCCN(C(=O)Cn2cnnc2)CC1 C#Cc1ccccc1CNC(=O)NC1CN(C(=O)OC(C)(C)C)C1 C1(NC(CCCC#C)=O)CN(C(C2CCCC(C)(C)O2)=O)CC2(CCOCC2)C1 CC(C)C(C(C)NC(c1coc(Cl)n1)=O)NC(c1cn(CCC2CC2)nn1)=O C1(C(=O)NCC)CCCC12CCN(C(=O)NCC13CCCC1(OC)OCC3)CC2 Cc1nc(C#N)ccc1C(N1CCC(C)C(NC(c2cnc3n2CCS3)=O)C1)=O c1(C(=O)NCC(CNC(CC(COC)C)=O)(C)C)cccc(N)c1O N1(C(CCSCC)=O)CCCC(O)(CNC(C2CC2C)=O)C1 CCCC(C(=O)NC(COC(C)=O)CO)NC(c1nc(O)sc1C)=O N1(C(c2n(CC)nc(C)c2)=O)CC(NC(c2ncnc(O)c2Cl)=O)CC(C)(C)C1 c1(C(=O)NC2CC(NC(C3(F)CC3)=O)C2)nsc2cc(Br)ccc12 c1(OCCC)ccc(Cl)cc1C(=O)Nc1ccc(-c2cc(F)ncc2O)cn1 C#Cc1cc(F)c(C(N2CCC(NC(c3ccsc3Cl)=O)C(C)C2)=O)cc1F c12cccc(c1)O2.c1(CCNCCF)ccsc1C(F)(F)F C12(NC(CC=C(C)C)=O)COCCC1CN(C(c1cn(C)nn1)=O)C2 N1(C(C(=O)NCCOC)=O)CCC(C)(CCNC(=O)C2=COCC2)C1 c1(OC)ncnc(N2CCCC(CO)(NC(C3COC(C)(C)C3)=O)C2)c1OC N1(C(C2C(C=C(C)C)C2(C)C)=O)CCN(C(c2ccsc2C)=O)C2(CCC2)C1 N(C(=NCC1CN(C2CC2)CCO1)NC1CC1)C1CCS(=O)(=O)C1 C1(NC(=O)CCc2cnc(O)[nH]2)CCC2CC1CN2C(C12CCC(CC1)OC2)=O c1(C(=O)NC(CNC(=O)C(O)Cc2cnc[nH]2)CO)nnn2c1CSCC2 C#Cc1ccc(Cl)c(C(=O)NCCN(C(=O)C(O)CC(C)(C)C)CCOC)c1 c1(C(=O)NCCNC(C2C(c3nc(C)[nH]n3)C2(C)C)=O)n[nH]c(C)c1F Cc1ncnc2c1CC(C(N1CCN(C(=O)CP(C)(C)=O)C(C(C)C)C1)=O)CC2 N1(Cc2c(OC)cco2)CCc2c(C(=O)Nc3ccc(C)s3)n[nH]c2C1 CN1CCC(C(=O)NCC2CNC(=O)C2)(NC(=O)CS(C)(=O)=O)C1 Cc1ccc(-c2n[nH]cc2C(=O)NCCOCCCNC(=O)CC(C)(C)F)cc1 c1(CN2C(CC(=O)Nc3cc(C)c(Br)cc3F)COCC2)ccc(O)c(C#N)c1 c1(C(=O)NC(CCC)CCCNC(=O)CS(N)(=O)=O)cc(F)c(C)cc1F C1(CNC(CC(CNC(c2nn(C)c(Cl)c2)=O)O)=O)CCCOC1(C)C CCCC(CCCNC(c1c[nH]nc1CC)=O)NC(C1ON=C(C)C1C)=O Cc1cccc(-c2cn(C(C)C)nn2)c1NC(C1(N(C)C)CCOC1)=O Cc1cc(F)ncc1C(=O)NCC1CCCN(C(=O)CSS(C)(=O)=O)CC1 N1(C(C2N(C(C)C)C(=O)CC2)=O)CC2CCN(C(c3cc(Br)n[nH]3)=O)C2C1 CCCC(CC)C(=O)NC(C)(CNC(C1(CF)CC1)=O)CC(C)C N1(C(CSCCOC)=O)CCCN(C(=O)CCSc2ccc(C)cc2)CC1CO N1(C(CC)=O)CCCC(C2CN(C(=O)CNc3ccc(C)cc3)C2)C1 C1(CCNC(C(C2CN(C(=O)CCc3nccn3C)C2)OC)=O)OCCC1(C)C c1(C(=O)NC2C3CN(C(CCC4CCC(=O)NC4)=O)CC32)ccc2ncsc2c1 c1(C(=O)NCC(C2CCOC2)NC(c2n(CC#C)ccc2)=O)csc(C)c1C c1(C(=O)NCC2(CNC(C3CCCSC3)=O)CC2)cc2cccc(F)c2s1 c1(C(=O)NC(C(=O)N2C(C)(CCC)CC2)(C)CO)cncc2[nH]ccc12 c1(C(=O)NCC2CC(NC(COCCOCC#C)=O)C2)ccc([N+](=O)[O-])c(O)c1 c1(C(N2CC3CC3(CNC(C34CCCC3OCC4)=O)C2)=O)n[nH]c2c1COCC2 C1(C(=O)NCC(C)CNC(=O)Cc2ccc(O)cc2)Cc2nn(C)cc2C(=O)N1 N1(C(c2c(C)n(C)cc2)=O)CCOC2(C1)CN(C(c1cccc3c1OCC3)=O)C2 CCCCC(CN=c1[nH]cc([N+](=O)[O-])cc1CO)NC(c1nc(C)c(C)s1)=O N1(C(C(CSC)O)=O)CCC2CN(C(c3cncs3)=O)CC2C1 C(=O)(NNc1cc(C(=O)NC)ccc1Br)C1N(C(=O)OC(C)(C)C)CCC1 C(C(O)CN=c1nc(C2CCCCC2)[nH]s1)NC(c1cccc(CN=[N+]=[N-])c1)=O CC(C)(C)CC(F)C(=O)N1CCC(C(=O)NCCCOCC(F)F)C(O)C1 c1(CCC(N(C(CN(C(=O)CC(C)(C)C)C)=O)C)=O)ccccc1OC(F)F C1(C(N2CCC(C(C)NC(C3CC3F)=O)C2)=O)CCC(=O)N1C1CC1 N(C(=NCc1ccnc(OCc2ccco2)c1)NC1CCC(=O)NC1)C(CC)C C1(C(=O)NCCC(C)NC(=O)CSc2n[nH]c(=N)s2)CCCCCCC1 C1(NC(CNC(C)=O)=O)CN(C(=O)CC2CC3(COC3)C2)CC1S(C)(=O)=O N1(C(C2=NOC(C)(C)C2)=O)CC(NC(c2cn(C3CC3)nn2)=O)CC12CCCC2 CC(C)(C)C1=NOC(C)(C(=O)NC2CC3CCC2(NC(=O)COC2CCC2)C3)C1 N1(C(c2c(F)ccc(C)c2)=O)CCOCC(C)(CNC(C2C3(CC3)C23CC3)=O)C1 CCC(CC(=O)NCC(CCNC(c1cnc(C2CC2)[nH]1)=O)OC)C(C)C n1(CC(=O)NCC(CN(C(C(CN(CC)CC)F)=O)C)C)ncc(Cl)c1C c1(C(=O)NCC2(CCNC(c3c(C)ccnc3)=O)CC2)ccc2c[nH]nc2n1 C1(NC(CCC#C)=O)CCN(C(c2ccc(OC)cc2OC)=O)C12CCC2 CN1CC(C)(C)CC1C(N1CC(O)CC1CNC(C1(CC2CC2)CC1)=O)=O N1(C(c2c(OC)noc2C2CC2)=O)CCc2sc(CNC(=O)COC)nc2C1 C1(NC(c2ccn(CCOC)n2)=O)CCC2CN(C(=O)C(C)C)CCC2C1 CC(C)CS(=O)(=O)CC(=O)N(C1CCN(C(c2c[nH]c3cc(F)ccc23)=O)C1)C c1(C(=O)NCCC2(NC(C3C(OC)C3)=O)CCCC2)[nH]c2ccc(F)cc2c1C n1(C(C)C)ncc(C(N2CCCC2C(C)NC(C2(C(F)(F)F)CCC2)=O)=O)c1N c1(CC(=O)NC23CC(NC(=O)CC4CCC5(CCC5)O4)(C2)C3)cc(F)cc(Cl)c1 c1(C(=O)NC2C(NC(C3(C)COC(=O)C3)=O)CCC2)cc2ncccn2n1 c1(C(N(C2CCN(C(=O)CCn3ccnn3)C2)CC#C)=O)csc(CO)n1 C12(NC(CCOCCC)=O)CCN(C(c3cncc(N(C)C)c3)=O)CC1C2 c1(C(=O)NC(C(C)NC(c2ccc(F)cn2)=O)CO)cc(N)nc(Br)c1 C1(CNC(C=CCCC)=O)CN(C(C2CC(C(F)F)C2)=O)CC1(F)F c1cnc(C2CCCO2)c(-c2noc(C3C4CCC34)n2)c1 C(=O)(CCS(N)(=O)=O)N(C)CC1(CNC(C2N(C(C)=O)CC(F)C2)=O)CC1 Cc1[nH]c(=N)[nH]c(=NCCC2CC(C)(C)NC2=O)c1C C(CC(=O)NC1CCC1C1CC1)(C(F)(F)F)OC C(=O)(C1=CCCOC1)NC1CCN(C(c2c(C(C)C)ncnc2)=O)C1 C1(C(=O)NCC=CCNC(c2cccc(CC)n2)=O)CCC=CCCC1 c1(C(N2CC(NC(=O)C#CC3CC3)CC(C)C2)=O)ncnc2sccc12 CC(C)CC(CNC(c1cn(CC(F)(F)F)nn1)=O)NC(=O)C(F)C(C)C c1(OCC(=O)NC2CCN(C(CC)=O)CC2O)cc(F)c(F)cc1F C#Cc1cc(C(=O)NC2CCCCC2NC(c2cn(C)nc2C)=O)cc(Cl)c1 N#CCCCCCC(=O)N1Cc2occ(C(N3CC(C4=NOCC4)C3)=O)c2C1 c1(C(=O)NC2CN(C(C3(c4cccs4)CC3)=O)CCC2O)ccc2ccsc2c1 c1(C(N2CC(C(C)NC(C3C(C=C)C3)=O)C2)=O)cc(OC)cc(Br)c1N CC1CCN(C(=O)C=CC2CC2)C1CNC(c1cn(Cc2ccccn2)nn1)=O CC1(C)OCC2CC12C(N1CCOCC1CNC(c1ccnc(S)c1)=O)=O CC(C)CC(C)C(=O)N1CCCC(CCNC(=O)Cc2ccn(C)n2)C1 c1(C(N2CCC(CC(=O)NC3(C(N)=O)CCOCC3)C2)=O)ccnc2ccnn12 C(=O)(CC1=CCN(C)CC1)N1C(C)CCN(C(=O)CC2(C)CCOC2)CC1 c1(OC)cc(C(=O)N(C)CCNC(C2CSCN2C(=O)C(C)(C)C)=O)ccc1F C1(C(=O)NC(C#C)CC2CC2)CN(C(=O)Cc2c(C)cccc2C)C2(CCC2)C1 C(=O)(C(O)CC(N)=O)NCC1(O)CC(CNC(c2cnn(C)c2C(F)(F)F)=O)C1 C(=O)(C1CCc2cccc(F)c21)N1CCN(C(C(CCSC)OC)=O)C2(C1)CC2 c1(C(C)(C)C)nccc(C(=O)NCC2(C)CCN(C(C3(F)CCOC3)=O)C2)n1 N1(S(CCNC(=O)CCc2ccc(F)cc2)(=O)=O)CCN(C(C)C)C(C)C1 N1(C(c2n(CC=C)ccc2)=O)CCC2(CCN(C(C3CCCN3C)=O)C2)C1 c1(NC(C(C2CCN(Cc3ccncc3Cl)CC2)C)=O)c(Br)cc(Br)c(Cl)c1Cl C(C(C)(C)CC(=O)OCc1c[nH]c(C)c1CCC(=O)OC)OC c1(C(=O)NCC2C(NC(CN(CC)CC)=O)C2)ccc(F)c(CC)c1F C1(CNC(C2(COCC)CCC2)=O)COC(CNC(=O)CCc2cn(C)cn2)C1 C1(C(=O)NCC2C(NC(c3csc(-c4ccco4)n3)=O)C2)CCC2CC2CC1 C1(O)(CNC(=O)CC2CCC2)CC(C(=O)NC2CC(N(C)C)C2)C1 c1(C(=O)NC(C)C=CC(=O)NCC2(N(C)C)CCC2)ncccc1CO N1(C(C2N(C)C(=O)OC2)=O)CCOCC(C(=O)NCC2CCCS2)C1 c1([SH](CC(=O)O)(C)=O)ccc(C(N2CCN(c3cccc(O)n3)CC2)=O)c(Cl)c1 c1(CC(=O)Nc2c(C)nn(CCOC)c2C)ccc2c(cnn2C)c1 CCC(C)C(C)C(=O)NC1(C)CC(NC(=O)CCc2nc(-c3cccs3)no2)C1 c1(NC(=O)OC(C)(C)C)cnccc1C(=O)Nc1ccno1.C12CC3CC3N1C2=O Cc1cc(C)c(C(N2CC(NC(=O)CC3CCC(F)(F)C3)C(C)C2)=O)c(=O)o1 Cc1nnc2n1C(C(=O)NCCC1CCN(C(C3CCS(=O)(=O)N3)=O)CC1)CC2 c1(C(C(=O)NCCCCNC(c2cncn2C(F)(F)F)=O)OC)cccc(Cl)c1 C(C1CCN(C(C2CC3CC3C2)=O)CC1)=CC(=O)N(C1(C)CC1)C c1(SC(C)C)ccc(C=CC(=O)Nc2cc(C(F)(F)F)ccc2C)cc1 n1(CCCSC)nnnc1C(C1CCOCC1)NC(C1(n2cc(Br)cn2)CC1)C C1(CC=C)(NC(=O)C2=C(Cl)CCOC2)CC2CCC(C1)N2c1nc(C2CC2)ns1 N1(C(CCc2cncc(C)c2)=O)CCC2CN(C(C3CC34CCC4)=O)CC12 c1(CC(CNC(=O)CCSC2CCCC2)NC(=O)CC2C=CCC2)ccccc1 CCC(C)C(C(=O)NCc1cncc(OC)n1)NC(=O)CCC(C)(C)F Cc1cc(F)cnc1C(N1CCCCC1CCC(C)(C)NC(=O)C(C)O)=O C1(n2cc(C3(OC)CCOC3)nn2)(C(=O)OC)CN(C(=O)C(C)C#N)C1.c1ccccc1 C1(NC(C2CC(SC)C2)=O)CC(NC(C2(C(C)(F)F)CCC2)=O)CC1O CN1C(=O)C(=O)N(CC(=O)NCC2C=CC(NC(c3ccc[nH]3)=O)C2)C1=O C(=O)(CCCCC(N)=O)N1CC(C(N2CCC(O)(CN(C)C)C2)=O)(CC)C1 c1(C(=O)NC2(c3cn(C4C(C)(O)CCC4)nn3)CCC2)cc(F)c(Cl)cc1F C1(NCC2(OC)CCCC2)CCCCC2(CC2)C1 Cc1nc2ccccn2c1CC(=O)NCC1C2CN(C(=O)CN(C)C(N)=O)CC12 CC1C(NC(c2ccnc(Cl)c2)=O)CC2CCC1N2C(c1nc(F)ccc1Cl)=O C1(CC)CC(C(=O)NC2CC(CC(=O)Nc3ccc(SC)nc3)C2)CCO1 C(C(O)CNC1C2CCCC12)(OCC)OCC.OCC N1(C(c2cc(-c3ccco3)no2)=O)CCC2CCN(C(=O)C3=CCCCO3)C2C1 C1(C(=O)NC(C(N2CCCC(CCF)C2)=O)C2(O)CCC2)CC2CC1CC2O c1(C(N2CCC(C)=C(C)C2)C(=O)NCc2cccc(OC)c2)ccn2nccc2c1 C1(C(N(CCNC(c2cc(CC(C)C)[nH]n2)=O)CC)=O)COC(C)(C)C1 c1(CSCC(=O)N(CCC(C)NC(c2ccccc2)=O)C)csc(=N)[nH]1 C(=O)(CC(C)CC(C)C)NC1(CNC(C2CCCN(C(CC)=O)C2)=O)CCCC1 c1(C(=O)NC(CNC(c2ccc[n+]([O-])c2)=O)C2CC2)cccc2c1COCC2 C(CCS(C)(=O)=O)(C(=O)NCC1CCCCN1C(C1(SC)CCC1)=O)OC C=CCCCC(C(=O)NCC12CC(CN1C)C2)NC(=O)Cn1ccc(C)n1 C1(CNC(c2cc(Br)c[nH]2)=O)CCC2CN(C(c3ccoc3)=O)CCC2C1 CC1CCN(CCC(=O)NC2CC2NC(=O)CC2CC(=O)NC2=O)CC1 C1(NC(C(F)OC)=O)CCN(C(c2cnc(C)nc2C)=O)C12CCCC2 C(C(=O)Nc1nc(Cl)ccc1Br)(C1=NOCC1)N1CCCC(N(C)C)C1 N1(c2c(C)cncn2)CC(NC(=O)C(C)CO)CC2(CCC2)C1 N1(C(C2OCCN(C)C2)=O)CC2(CC2)CC1CNC(=O)C(F)(F)c1cnccn1 N1(C(C(CC)(F)F)=O)C(CC(=O)NCCS(C)(=O)=O)C2CCCC12 C1(O)(C(=O)NC(C2CN(C(C3CCc4nc[nH]c4C3)=O)C2)C)CCCC(C)(C)C1 O=S(=O)(c1cncc(Br)c1)NC1CN(CC23CC4CC(CC(C4)C2)C3)CCC1(F)F c1(C(=O)NCC(CC)(C)NC(=O)CC(C)N2CCCC2=O)cccc2sccc12 C1(NC(CSCC(=O)OC)=O)CCC(NC(=O)CC2CCC(C)CC2)CC1 c1(COC)cccnc1C(=O)NCC1(CNC(c2nocc2C)=O)CC1(F)F C1(CC(=O)NCCN(C(C2(C)C(C(=O)OC)CC2)=O)C)CCC2(CCC2)O1 N#Cc1cc(C(N2CC(NC(=O)COCC(F)(F)F)C(F)C2)=O)ccc1O N1(C(C(CC#C)C)=O)CCC2(CCCN2C(=O)CC2(COC)CC2)C1 C1(NC(c2ccc(OCCC#C)cc2)=O)CCN(C(C2(CC)COC2)=O)CC1O N1(C(C2C(C)C2)=O)CCC2(CC(NC(c3cncc(-n4cccn4)n3)=O)CO2)C1 c1(C(=O)OC)ccc(O)c(NC(C2CN(C(C3CCCO3)=O)CCC2O)=O)c1 CC1CCCC(CS(N2CCC(NS(C)(=O)=O)C2)(=O)=O)O1 CC(C)CC(C(=O)NCc1cn(C)nn1)NC(c1nnc(O)nc1O)=O C(=O)(C(C)(C)C(C)(F)F)NC1CC(NC(c2nc(C(C)C)sc2)=O)C12CCC2 C1(COC)(NC(=O)CCC2(C)CC2)CCN(C(=O)C#CC2(C)CC2)CC1 N1(S(CC)(=O)=O)CCC(Oc2ccc(NC3CCCC3C3CC3)cc2)CC1 c1(C(=O)NC(C)CCCNC(c2ccc(F)cc2)=O)ccc(OC(F)F)c(Cl)c1 N#Cc1ccc(C(=O)NCC2OCCC2C(=O)N(CC(O)CO)CCO)o1 C(=O)(CCCCBr)N1CCC(CN(C)C(C2CC2(C)C)=O)CC1 C1(NC(C(CC)CC)=O)CC(CNC(=O)CC=CCc2ccccc2)C12CCC2 CC1CC(C(=O)N(CCCn2cc(COCC(N)=O)nn2)C)CO1 c1(C(=O)NCC2(CCNC(C(CSC)C)=O)CC2)ccc2n[nH]cc2n1 c1(C(=O)NC(C)(C)CCNC(C2CCCCO2)=O)ccnc(-c2ccccc2)n1 C(CC(=O)N1CC2CC1CN2c1nc(C2CC2)nc(=N)[nH]1)(C(F)(F)F)OC N1(C(C2(C#C)CCCC2)=O)CC(NC(=O)C(C)n2cccc2)CC(F)C1 C1(C(N2CC(NC(c3c(Br)cn(C)n3)=O)C(O)C2)=O)SC2C=CC1CC2 C(CC(C(C)(C)C)NC(=O)CP(C)(C)=O)N(C(=O)C=CCN1CCCCC1)C c1(OC)cc(C(N2CCC(C)C2CNC(c2csnn2)=O)=O)ccc1F c1(CC)c(C(=O)NC2CCOCC2NC(c2[nH]cnc2C)=O)sc2ccccc12 C1(C(N2CC(N(C(CN(CC)CC)=O)C)C2)=O)CCOC1(C)C c1(CC(=O)NCC2C3CN(C(C(C=C)O)=O)C2C3)ccc(C)c(OC)c1 C1(CSCC)CCN(c2cc(N3CCCC(c4ncccn4)C3)ncn2)CC1 n1(CC)ccnc1C(=O)NC12CC(C(=O)Nc3cnsc3)(C1)C2 C1(C(=O)NC(CN(C(C(C)=CC)=O)C)C)CCC2(CC2)N1C(=O)OC(C)(C)C N(C(=NCC1(OCc2ccc(Cl)cc2)CCCC1)N1CCC(C(N)=O)CC1)C(C)C NS(=O)(=O)CCC(=O)N1CCCC1CNC(=O)CC1CC(O)C12CCC2 CCC(C)CC(C(=O)NC1(CF)CCC1)NC(=O)C(=O)C1CCCC1 C1(C2CCN(C(C3CSCCS3)=O)C2)(NC(c2onc3ccccc23)=O)CC1 c1(CC)cnccc1C(=O)NC(CCF)C(=O)NC1(C(O)COC)CC1 C(=O)(C#CC(=O)NC1CCCC(NC(=O)CN2CC(C)(C)C2)C1)N(C)C C1(C(C)C)CCC(C)CC1C(=O)NC1CC12CC(NC(C1(F)CCCCC1)=O)C2 c1(C(c2nnnn2C(C)(C)C)NC(CC)(C)C)nc2ccc(Br)cc2o1 N1(C(c2c(CC)n[nH]c2)=O)CCCC(C(=O)NC2CC(CC(C)(C)C)C2)C1 n1(CC)nc(C(=O)NC(CCOCCO)C(=O)N2CCC(SC)C2)c(C)n1 C1(NC(CC(CNC(C2(C)CCCCC2)=O)OC)=O)CN(C)C(=O)C12CC2 CCCC#CC(C)(C)NC(C1CCN(C(=O)C(F)C2CCOC2)CC1O)=O C1(NC(c2cccc(Br)c2F)c2n(CCCCCC)nnn2)CCCCC12CC2 C(=O)(C1=NNC(C(F)(F)F)C1)N1CCC(N(C(=O)CSc2cccs2)CCC)C1 C1(C)(CNC(C(C)=C(C)C)=O)COCCN(C(c2cccc3ccsc23)=O)C1 n1(CC)ncc(C(=O)N(C2CCCCC2)CCNC(C2CCCC2C(N)=O)=O)n1 C(=O)(C1Cc2ccccc21)N1CC(CNC(=O)CC2CC=CCN2C)CC(C)C1 CCCC(C(O)C(=O)N(C(C)CC(=O)OC)C)NC(=O)CC#N Cc1cc(C(=O)NC(CNC(C2CC2(C)C(F)(F)F)=O)C(C)C)cc(C)c1F O=C(C#CC1CCOC1)N1CCCC(N(C(=O)Cc2ccc(Cl)cc2Cl)CCF)C1 CC(C)CS(=O)(=O)CC(=O)NC12CCOCC1CN(C(=O)C#CC(C)(C)C)C2 C(=O)(CCCCc1ccccc1)NCC(C)(C)CNC(C1(C)CC1(F)F)=O C1(NC(c2c(Cl)cnc(C)n2)=O)CN(C(=O)C=CCCC(C)C)C2(CCOC2)C1 C1(NC(C2CCCC(=O)N2)=O)CCN(C(C23CCC(CC2)CC3)=O)CC1F c1(C(=O)NCC2(F)CCC(NC(C(CCC)(C)C)=O)C2)cnn2ccnc(N)c12 c1(C(=O)NCCCCC(=O)NC2C=CCN(C(N)=O)C2)ccnc2cc[nH]c12 C1(C(N(CCN(C(C)C)C(C2CCS(=O)(=O)C2)=O)C)=O)(C(F)F)CCCSC1 C1(C(N(C(CC(C)C)C)C)=O)CCN(C(c2ocnc2C2CC2)=O)C12CCC2 c1(NCC2CC2)ccc(SC)cc1.C(=O)(CN)N(CC=CC#C)C(C1CC1)C C(=O)(NN1CCCC1C(=O)NC(CO)C1(C)CC1)c1cc(C)on1 C1(NC(=O)COCF)CCC2(CC1)CCN(C(=O)C(F)(F)c1ccncc1)CC2 C(CCCCC(=O)N1CC(NC(=O)CP(C)(C)=O)C1)=CCCC C1(C(C(N2CC(C)(O)C2)=O)F)CCN(C(=O)CC2CC3CCC2C3)C1(C)C C(=O)(CCS(=O)(=O)N(C)C)N1CCC(N2CCN(C(C(N3CCSCC3)C)=O)CC2)C1 c1(CN2CC(C(=O)Nc3ccc(NS(C)(=O)=O)cc3)C(O)C2)cc(Cl)ccc1Cl N1(C(C(C)=CC)=O)CCCC(N(CCO)C(c2cc(COC)oc2C)=O)C1 N1(C(CCOCC#C)=O)CCOC(C(=O)N(CC(=O)NCC)C2CCC2)C1 CCCC(C)(O)CC(=O)N1CCCC(C)(CNC(C2CN(C)CC(C)O2)=O)C1 C(C(=O)NCC(C)NC(=O)CCc1cn[nH]c1)(C(C)C)NC(C)=O c1(C(c2cn(C)nn2)(c2ccccc2)NC(=O)CO)nc2cnccc2s1 Cc1nc(CO)oc1C(N1CCOC(CNC(=O)CC2CCCN2C(C)C)C1)=O CC(C)C1(C)CNC(=O)N(C)CC(=O)N1.c1(CO)ccccc1.C(=O)(C=CCF)N C1(NC(C2C(c3c(C)cccc3)C2)=O)CCN(C(=O)Cc2nccs2)CC1O c1(C(=O)NC(C2CC(NC(C(C(CC)C)C)=O)C2)C)cccn2ccnc12 N1(C(C2(C)CC2)=O)CCC2CCN(C(=O)CCC(=O)NC3CC3)CC2C1 C(CC(C)(C)C)(c1ccccc1)NC(c1n(CCC)nnn1)c1ccno1 c1(OCC)ncc(F)c(=NCc2ccc(C(N3CCC(CC(C)C)C3)=O)[nH]2)[nH]1 Cc1cc(NC(=O)C(C)(C)C)sc1C(=O)NC1CC1CNC(=O)CC1CCCO1 Cc1ccnc2sc(C(=O)N(C)CC3(CNC(=O)C4=COCC4)CC3)c(C)c12 N1(C(C2C(CC)OCC2)=O)C2CCCC1CC(NC(c1cnn(C(F)F)c1)=O)C2 CCC(C)C(C(=O)NCC(C1CC(C)(C)C1)O)N(C)C(c1n[nH]c2c1COC2)=O c1(SC)c(C(=O)NC2CCOC(c3cccs3)C2)cccc1Cl c1(C(N2CC(O)(CNC(C(CCOC)C)=O)C2)=O)cc(OC)cc(C(F)F)c1 Cc1ccncc1C=CC(N1CCC(F)(CNC(=O)CC2NC(=O)NC2=O)C1)=O C1(CC)(CC)CC(C(N2CCCC2C(C)NC(c2ccn(CC(F)F)n2)=O)=O)C1 C(=O)(C(CN(C)C)C(C)C)N1C(CC=C)(C(=O)NCc2cc(C)sc2C)CCC1 C(C(C)(O)C(=O)NCC=CCNC(=O)C(c1ccccc1)n1cccn1)OC N1(C(C(C(C)C)F)=O)CC2CC1CC2CNC(=O)Cc1c(Cl)cnn1C c1(CNC(C2(C)CN(C(C3OCC(C)C3)=O)C2)=O)ccc(F)cc1O CC(CC(=O)NC(C1CCCCCC1)CNC(c1nocc1C1CC1)=O)C(F)F C1(C(N2CC(N(C(c3cn(C(C)C)nn3)=O)C)C2)=O)C(C)(C)CCCC1(C)C N#Cc1cc(F)c(F)cc1NC(C1CC(F)CN1C(c1sc(Br)cc1Br)=O)=O CC(C)CC(CNC(=O)CN1CC(C)(C)C1)NC(=O)C(C)n1cncn1 Cc1cc(C(=O)NC2(C)CC(NC(=O)Cc3cccnc3O)C2)cc2c[nH]nc12 N1(ON(CC)C(c2cc(C=O)cc(Br)n2)=O)CC(C)CCC1c1ccccc1 c1(C2(C(=O)OCC)CCC2)ccc(NC(=O)OC(C)(C)C)cc1.C1C(F)C1.C(=O)(N)N C1(C2CC2)(NC(c2cn(CCC)nc2)=O)CCN(C(=O)C2=COCC2)C1 C1(COC)(CNC(c2ccno2)=O)CCCN1C(=O)CCC1CCC(=O)C1 n1(CC(=O)NC23C(CN(C(C)=O)C2)C3)nc(C)c(Br)c1C c1(N2CCCC(CCO)C2)nc(N2CCOC(CCO)C2)nc2c1COC2 c1(C(=O)NCC(CC)C(=O)OC)ccc2c(c1)CCCS2 c1(CN(C)CC2N(C(CCc3c(C)ncs3)=O)CCOC2)cc2ccccc2[nH]1 c1(C(=O)NCCCN(C(C(CCC#C)O)=O)C)cccc2c1CCCN2 n1(C(CC)CC)nc(C(=O)NCC2CCN2C(c2c(OC)noc2C)=O)cc1C c1(C(N2C(C(=O)Nc3c(C(C)=O)scc3)CCCC2)=O)ccc([Si](C)(C)C)cc1 C1(C(=O)NCCC2(C)CCN(C(CCCOC)=O)C2)CC2OC(=O)OC2C1 C(=O)(C(C)(C(C)C)OC)NCC(CC=C)NC(c1ccnn1C1CCC1)=O C12(C(=O)NCCCCN(C(C3N(CC)CCC3)=O)C)CCC(OC)C1CC2 c1(C(N2CC(NC(CC=C)=O)C(O)C2)=O)cc2cn[nH]c2cn1 c1(C(N2CCC(F)(C(=O)Nc3nccc(I)n3)C2)=O)cc(Cl)c2cn[nH]c2c1 c1(N2CC(CCNC(=O)CC(C)(C)OC)(OC)C2)cnc(C(C)=O)c(C)n1 CCCN=C(NCc1cc(Cl)ccc1OC)NCC1CCCC(C(F)(F)F)O1 C1(CC(=O)NC(CCCC=C)C2CC2)CCN(C(=O)C(F)C2CCC2)C1(C)C C1(CNC(C2CC(=C)C2)=O)CC2(CCN(C(c3cncc(C(F)F)c3)=O)CC2)C1 c1(N(C2CC3(CNC3)C2)C(C2(C3CC3)CC2)=O)ncnc2c(Br)c[nH]c12 n1(CC(=O)Nc2ccccc2C2CC2)c(=O)ccn(CC2CCCC2)c1=O C1(C(N(CCNC(=O)CNC(=O)C2CC2)CC)=O)CC2C=CC1C2 N1(C(C(C)(C)OC(CC)=O)=O)CCN(C(c2cc(OCC)n(C)n2)=O)CC2(CC2)C1 C1(C(N(CC(=O)OCC)C)=O)CN(C(=O)C(O)CCSC)CC(C)(C)C1 c1(OC)ccc(CC(=O)NC2CN(Cc3nccnc3Cl)CC2O)cn1 Cc1nn(C)c2c(NCC3CCCN3C)nc(N3CCc4[nH][nH]c(=N)c4C3)nc12 N1(C(c2ccc(SC)cc2)=O)CC(NCc2ccc(N3CCCC3)o2)C(C)(C)C1 c1(C(C)(C)C)ccc(NNC(=O)C2CC(=O)N(Cc3ccccc3)C2)cc1 C12(NC(C(C3CCN(C(C)=O)CC3)C)=O)CCC(C1)OC2C c1(C(N(C2CN(C(=O)CCn3ccnc3)CC23CC3)C)=O)cc2ncccc2[nH]1 S(=O)(=O)(c1cc(C)cnc1N(C(CO)C1CC1)C)N(C)Cc1ccc(OC)cc1 N1(C(C2CCC(=O)O2)=O)CCCCC1CC=O.C1(N(CO)CCO)CCC(F)(F)C1 C1(C(=O)NCCC2CCN2C(C)(C)C)CCCCC1.CC1C(=O)N1C1CC1 CC(CC(=O)N1CCC(N(C(=O)COCCF)CCO)C1)P(C)(C)=O C(c1ccc(Cl)cc1Cl)=CC(=O)NC(C1CN(c2nnnn2C2CC2)C1)C C=C1CC(C(F)(F)F)(C(=O)NCC2CCN2C(=O)CSc2cnn(C)c2)C1 CC1=C(C(=O)NC2(CN(C)C(c3nc(C)nn3C)=O)CC2)CCC(C)(C)C1 C1(CCCNC(C(C)NC(CC)=O)=O)CCCCN1C(=O)CCc1ccc(C)s1 Cc1nc2ncc(C(=O)NC3CC3CNC(=O)Cc3nn(C)cc3Cl)c(=O)n2[nH]1 CC(C)(C#N)CCC(=O)NCC1CN(C(C2Cc3cccnc3C2)=O)C1 C1(C(=O)N(CCCOC)C)(CC)CN(C(=O)C(C)=C(C)CC)C1 CCC(C)(C)CC(=O)NCCCN(C(c1oc(CO)nc1C)=O)C(C)C N1(C(c2c(C#C)c[nH]n2)=O)CCN(C(c2cnc(C3CC3)nc2)=O)CC1C(F)F c1(C(N2C(CCNC(Cc3c(C)nccc3)=O)COCC2)=O)ccc(=O)n(C)n1 C1(CC(=O)NCC2N(C(C3CC(C(C)(C)C)C3)=O)CC2)CCC2(CC1)CCC2O N1(C(=O)Cc2csc3ccccc23)CCN(C(C2CC=CCC2)=O)C2CCCC12 C1(C(=O)NC(CC)(C)CC)C2CCCC2CN1C(=O)OC(C)(C)C Cc1cnc(C(=O)NCC2CCCN(C(C3(C)CCCC3)=O)C2)cc1Br N1(C(c2[nH]cc(CC(C)C)c2)=O)CC2CN(C(=O)C(N3CCOCC3)C)CC2C1 C1(C(=O)NC2(CNC(C3CCCS3)=O)CCCC2)CCc2ncc(Br)n2C1 c1(COC)ccnc(C(=O)NCC23CC2CN(C(=O)C=CC2CCC2)C3)c1 C1(OC)CCCC(CC(N2CCCC2(CNC(=O)CCC(C)C)CO)=O)C1 c1(C(=O)NC2CC(CNC(C3CC3CF)=O)C2)nccn2nccc12 c1(C(=O)NCCC(CNC(C=CC=CCC)=O)(C)C)ccc(S(N)(=O)=O)s1 c1(C(=O)NC2CC(NC(C34CCCN3CCC4)=O)C2)ccc2sncc2c1 CCCCS(=O)(=O)CC(=O)NCC1CCN1C(=O)CCCCC#N c1(C(N2CC(C)C(NC(=O)C(C)Cn3cccn3)CC2)=O)ccc(C#N)cc1O N1(C(C(c2cccc(Cl)c2)OCC)=O)CCC(NC(c2nc(C)n(C)n2)=O)C1C c1(C(N2CCC(C)(CNC(CC(CC)C3CCC3)=O)C2)=O)cnc(OC)c(C)n1 N1(C(c2c(CC)ccnc2)=O)CCCCC(CNC(c2cc(CC)ncn2)=O)C1 N1(C(CC2(C)OCCO2)=O)CCCC(C)(NC(=O)C(F)CC2CC2)C1 c1(C(N2OCC(n3cc(CC=C)nn3)C2)=O)cc(S(N)(=O)=O)cc(Cl)c1Cl N1(C(c2ccc(CC)cn2)=O)C2CCC1C(NC(=O)Cn1cc(C)cn1)C2 c1(OC)cccc(Br)c1NC(=O)CC1CCN(Cc2cccc(C3CC3)c2)CC1 c1(C(=O)NCCCN(C(=O)C(c2cccnc2)O)C)cc(=O)c(Br)c[nH]1 C(C)(CCC(=O)N(CCCCCNC(c1ccnc(S)c1)=O)C)OC C12(NC(CC3CCCC(OC)C3)=O)CCCC1N(C(C1CCN(C)CC1)=O)CC2 C1(CC(=O)NCCNS(CC)(=O)=O)CCN(C(C2CN(C(C)C)C2)=O)C1(C)C CC1(C(=O)NC2CCC(NC(c3ccc(F)cc3)=O)C2)OCCc2ccccc21 N1(C(C(C)CO)=O)CC2CCC1CN2C(c1ccc([N+](=O)[O-])[nH]1)=O C(CC1CCCCC1)(C(=O)NC(C)CCCNC(C1(CO)COC1)=O)OC N1(C(C2(C=C)CC2)=O)CCC(C2CCN(C(=O)C(C)SC(F)(F)F)CC2)C1 c1(C(=O)NCC2(C(=O)Nc3cncc(Br)n3)CC2)cccc2c(Br)n[nH]c12 C1(CC=C)(NC(c2csc(S)n2)=O)CCN(C(C2CCCC23CC3)=O)C1 CC1CCC(NC(c2cc(CCO)on2)=O)CN1C(C12CC(F)(C1)C2)=O N1(C(c2cn(CC)nn2)=O)CC2CC(NC(=O)C=C(C)C(F)F)C2C1 c1(C2(C(N(CCCNC(=O)C3CC3)CC)=O)CCC2)cccc(C#N)c1 c1(CNC(=O)CC2OCCCO2)cccc(NC(c2ccc(F)o2)=O)c1 C1(NC(C2(OC)CC(C)C2)=O)CC12CCN(C(=O)CC1CC(N(C)C)C1)CC2 CC1(C)COCCC1CNC(=O)CC(C(F)F)NC(=O)CC1CCCCCC1 c1(C(N(CCC(C)NC(COC(C)C)=O)C)=O)cnc2c(c1)c(O)nc(=O)n2C Cc1ccc(C(=O)NC2CC(C(=O)Nc3ccc(Cl)c(Cl)c3Cl)C2)c(I)c1C C1(NC(c2ccc[n+]([O-])c2)=O)CCCCC1C(=O)NCc1cccnc1O Cc1cc(F)cnc1C(=O)NC1(CCCC(=O)N2CC(CC(N)=O)C2)CCC1 C(=O)(C1CCc2cc(F)ccc21)NCC(C)N(C(COCCC=C)=O)C c1(C(=O)NC2CCCN(C(c3nnc(CC)s3)=O)CC2)c(O)nnc(C)c1C C1(NC(C(CC)OC)=O)CC2C1CCN2C(=O)CCCc1ccc(Cl)cc1 S(=O)(=O)(c1ccc(Cl)cc1)NC(CC)C(=O)NCC1(C(F)(F)F)CC1C(=O)O Cc1cc2c(C(=O)NCCC3CN(C(=O)CCc4cnn(C)c4)C3)nccn2n1 CCC(CC(=O)NC(C1(O)CCN(C(c2c(Cl)csc2Cl)=O)CC1)C)C(C)(C)C C#Cc1ccc(C(N2CCCC2C2(NC(=O)C(O)C=C)CC2)=O)cc1Cl N1(C(C)C(=O)NC(N)=O)CC2CC1CN2C(C1CC12CCCC2)=O C(=O)(C(CO)NC(=O)C1CC1)N(CC(CC)NC(=O)C(CC)C1CCOCC1)C N(C1c2ccccc2CC12CCCC2)c1cc(N2CC(CCF)OCC2)ncn1 c1(C(N(C2CN(C(=O)CCc3cc(Cl)cs3)CC2F)C)=O)ccc(F)cn1 C1(C(=O)NC(c2nc(C(=O)NC(C3CCC3)C)cs2)=O)C=CC(=O)N=N1 C1(NC(CCCNC(C)=O)=O)COC2C(NC(c3nc(C)c(C)s3)=O)COC12 N1(C(C2CC(C)(C)C2)=O)CCN(CC(=O)Nc2cc(C3N(C)CCC3)[nH]n2)CC1 Cc1nonc1CC(=O)NC(C)(C)CCNC(=O)CC(C)NC(N)=O Cc1c(C(=O)N(CC(O)CN(C)C(c2cccc(N(C)C)c2)=O)C)cccc1F c1(C(N2CC(O)CC(NC(c3c(C)nn[nH]3)=O)C2)=O)c(O)cc(Cl)cc1F N1(C(C(C(C)CNC(=O)C(=C2CCCCC2)F)F)=O)CC2C3CCC(C3)C2C1 n1(CC(=O)NC(C(C)NC(=O)CC23CCC(CC2)C3)(C)C)ncc(C#N)c1N N1(C(CC=C)=O)CC2(CCC(C(N3CCCCC3CCO)=O)O2)C1 c1(OC)cccc(C(C)=CC(=O)NCC2CN(C(c3cc[nH]n3)=O)CC2C)c1 C(=O)(CCCCCC#N)N(CCNC(C1(OC)CC(C)CC(C)C1)=O)C1CC1 CC1CN(C(C2COCCOC2)=O)CC1(C)CNC(=O)CN(C)S(N)(=O)=O c1(COC(C2CCc3n[nH]cc3C2)=O)cnn2cc(Br)ccc12 c1(CCN(C)Cc2cccc(Br)c2)ccc(CO)c(F)c1 C=CC1(CC(=O)NC(C)CC(C)O)CN(C(=O)C(C)N(C)C)C1 CN1CCC(CCC(=O)NCC(C)(CO)NC(c2ccc(F)s2)=O)C1 c1(CC)cc(CC)[nH]c(=NCC2CCCCN2C(c2ccc(Cl)c(Cl)c2)=O)n1 C1(C(=O)NC2C(CNC(=O)Cn3cccn3)CC2)CCCC1C1CC1 C(=O)(CCCC(F)(F)F)NC1(CF)CCN(C(C(C)C=Cc2ccccc2)=O)C1 CC1CCC(=CC(=O)NC(C)(C)CN(C(=O)C(C)NC(=O)CC(F)(F)F)C)CC1 C(CC(C)(C)CC(=O)NCC12CN(C(c3ccc(F)cc3)=O)CC1CCO2)OC c1(C(N)=O)ccc(C=CC(=O)NCC2(N(C(C3(Br)CC3)=O)C3CC3)CC2)cc1 C1(SC)CN(C(C2CC=CC(Cn3cc(-c4cncc(C)n4)nn3)C2)=O)CCO1 c1(C(C)NC(=O)COCC2CCOCC2)n[nH]c(C(C)(C)C)n1 c1(C(=O)Nc2cnc(F)cc2C(=O)NCC(O)C(F)(F)F)ccc(O)c([N+](=O)[O-])c1 Cc1coc(C)c1C=CC(=O)NCCC1(C)CCN(C(=O)C(C)C2CC2)C1 c1(C(=O)NC(C(=O)NC(c2ncc[nH]2)C)Cc2ccoc2)ccc(Cl)cn1 Cc1cc(CC(=O)NCCN(C(C2CCC(C(N)=O)C2)=O)C(C)C)sn1 c1(C(N2CC(C)(NC(C(n3ncc(C)c3)C)=O)C2)=O)ccc(C(=O)O)nc1O O=S(=O)(c1ccnc(C(F)(F)F)c1)NCCOc1ncccc1Br C#CC1(NC(=O)CC2(C)CCN2C(=O)CN(C2CC2)CC)CC2CCCC12 C#CCCCCC(=O)NCCN(CCOC)C(C1CCCCC1O)=O C12(CNC3CCN(C(=O)COc4ccccc4)C3)COC(CCF)(C1)C2 c1(C(N2C(C(C)NC(Cc3c(C)noc3C)=O)CCC2)=O)cc(F)ccc1O N1(C(c2cc(C)cc(Cl)n2)=O)CCC2(CC1)CCN(C(C1C(C)(C)C1(C)C)=O)C2 c1(C(=O)NCC(C2CCOC2)NC(c2c(C#N)ccs2)=O)ncnc2sccc12 Cn1cc(CCC(=O)NCC(C)(CNC(C2(CCO)CC2)=O)OC)cn1 C(=O)(C(CNC(=O)C=C(C)C)C(C)C)N(CCCC)CC(C)C C1(C(N(C)CC2CCN(C(c3c(OC)csc3)=O)C2)=O)Cc2c(C)cccc2O1 C(C(C)(C(=O)NC(c1nc(C)no1)CO)NC(=O)CCCc1ccco1)SC Cc1cc(F)ncc1NC(C1(CNC(=O)C(O)Cn2cncn2)CC12CCC2)=O N1(C(C(COC)OC)=O)CCC2CCN(C(c3cnc(OC)c(C)c3)=O)CC12 N1(C(C(N2CCSCC2)C)=O)CCN(C(=O)CCCc2cncs2)C(C2CC2)C1 S(=O)(=O)(CCCN=[N+]=[N-])NCC1C(OC)CCCN1C(=O)OC(C)(C)C c1(C(N2CC3C(NC(C(C)OCC=C)=O)(C3)C2)=O)cnn2c1CC(F)(F)C2 c1(C(=O)NC2C3(NC(C(C)OC)=O)CCC(C2)C3)nc2ccccc2cc1Cl N1(C(C(CC)C)=O)CCC2(CC1)CC2C(=O)Nc1ccnc(C(=O)OC)c1 N1(C(c2c(=N)cc[nH]c2)=O)CC=C(CNC(c2ccnc(C3CC3)c2)=O)CC1 CCCC(C#N)C(=O)NCC(CC(=O)NC1C2CCC(F)(F)C12)C1CCC1 C1(C(=O)NC2(CN(C)C)CCC2)CCCC(NC(=O)CC23CCCC2C3)C1 c1(CNC2CCCC(C)C2)cn(C)c(=O)c2cnccc12 CC1CC(CNC(C2CCN(C)C2)=O)CCN1C(c1ccc(O)cn1)=O c1(CNC(c2cc3c[nH]cnc-3n2)=O)cccc2c1CCN(c1ncns1)C2 C(C(C)CC(=O)NOC(C)CC)NC(C1C(CC)CCO1)=O C1(CNC(CCCC(=C)C)=O)CN(C(=O)Cc2ccn(CC)n2)CCC12CCC2 N1(C(C2(Oc3ccc(F)cc3)CCC2)=O)CCC2(CC1)NCNC2=O c1(C(N(CCCN(C(C(C)OCCC#C)=O)C)C)=O)cc(C(C)(F)F)ccn1 c1(C(=O)NC2CCN(C(c3c(C)con3)=O)C(C)C2)scc2c1OCCO2 C1(NC(=O)CN2CCCC2)CC(CNC(=O)C(=O)Nc2ccc(Cl)s2)C(O)C1 C1(C(N2CCC(NC(CC3(OC)CCCC3)=O)C2C)=O)CCC2(CCC2)CC1 C1(CCC)(NC(=O)CC2(N(C(=O)CCc3cccnc3)C)CC2)CCNC1=O CC1(C)CCC2(CCN2C(C2(O)CC2)=O)CC1 CC(CSc1ccccc1)C(=O)NC1CC(C)(CNC(=O)C(C)(F)F)C1 C12(C(=O)NCCOCCCNC(c3n[nH]c4c3CCC4)=O)OCCCC1C2(F)F C1(C)(C(=O)NCCCn2c(C)nnc2)C=CCN1C(=O)CCC1CCCO1 c1(C(=O)NCCCC2(NC(C3C(C=C)C3)=O)CC2)cc(O)nc(C2CC2)n1 C1(C(=O)NC(C(=O)NCC)C(C)C)CCC2CCC1N2C(c1ccn(C)n1)=O c1(C(=O)OC(CC)C(N)=O)ccc(Nc2cncc(C(=O)O)c2)cc1 c1(Cn2cc(C(CC)O)nn2)nn2c(c1C(=O)N(C(C)C(C)C)C)CCC2 CC1(C)CCCC(C(=O)NCCC2CSCCN2C(c2cc[nH]c(=N)c2)=O)CC1 c1(OCC(N2CC3C(CNC(C4(O)CCOC4)=O)C3C2)=O)ccc(Cl)c(F)c1 c1(C(=O)NCC2C(NC(CCS(C)(=O)=O)=O)CCC2)ccc(N)c2ccncc12 N1(C(C(C)(C)OC(C)C)=O)CCCC2(C1)CN(C(=O)CCn1ccnc1)CCO2 c1(CC(=O)NCC(C)NC(=O)C(C)NC(=O)N(c2ccco2)C2CC2)cncnc1 CCC(CC)(CC)C(=O)N1CC2CC1C2NC(C1OCCC1C)=O CCC(CC(=O)NCC1(C(=O)NC2CC(OC)(OC)C2)CCCCC1)C1CC1 N1(C(C(C=C)C)=O)CCC2(NC(=O)C3=CCN(C)C3)CC2C1 N1(C(C2(CC)CCCO2)=O)CC(CCNC(c2cnc(O)n2C)=O)C(C)C1 c1(C(N2CC(C(=O)NC3CCN(CC)C3)OCC2)=O)cc(S(=O)(=O)N(C)C)c[nH]1 C(CF)(C(=O)C1(CNC)CC1)OC.c1(O)ccncc1.C12(CCC1)C(=O)NC2 c1(C(N2C(C(N(CCCO)C(C)C)=O)C=CC2)=O)c[nH]c2cc(Cl)ccc12 C1(C(=O)NCC2(n3ccnn3)CC2)CCC2CCC12 N1(C(C=CCN(C)C)=O)CCCC2(NC(c3nncn3C3CC3)=O)CC2C1 C1(NC(C(=C)Cc2ccccc2)=O)COCCN(C(=O)CSC)C1 C1(C(C)NC(c2cscc2C(F)F)=O)CN(C(=O)CC2(N3CCCC3)CC2)CCO1 c1(N(C(=O)NCc2cccn2C2CC2)Cc2ccccc2)cn2ccnc2s1 c1(CC(=O)OC)cccc2c1CN(C(c1ccncc1C)C(=O)NC(C)C)CC2 c1(C(N(CC(C)N(C(C(CCC)C)=O)C)C)=O)ccc2cc(C)ccc2n1 c1(C(C(=O)OC)OC(=O)Cc2csc(-c3ccco3)n2)ccc(F)c(Br)c1 NC1CCOCC1C(=O)N(CC(F)(F)C(F)F)Cc1ccccc1 c1(CN2CC(CNC(C3(CC)CCOCC3)=O)OCC2)csc([N+](=O)[O-])c1 C(=O)(C(C)CC(F)F)NC1(CCO)CN(C(C2CCC(CCC)CC2)=O)C1 Cc1ccc(C(=O)NC(C2CCCN(C(c3cc(O)cc(F)c3)=O)C2)C)c(F)c1 C1(C(=O)NC2(CNC(c3nc(C4CC4)cs3)=O)CC2)CC2C=CC1C2 N1(C(Cn2c(C)cc(C(=O)OC)n2)=O)CCN(C(=O)C2=CCOCC2)CC1C c1(OC)cccc(C2=NOC(C(=O)OCc3cnsc3)C2)c1 C1(NC(c2cnc(C#N)s2)=O)CN(C(=O)CSc2ccccn2)CC2(CCC2)C1 N1(C(C2CCN(C)C2)=O)CC2(CNC(c3cccc4nncn34)=O)CCC1CC2 N1(C(=O)CC2CCCCO2)CCC2CCN(C(c3nccc4occc34)=O)C2C1 N1(C(c2ccc(C)s2)=O)CCOC2(CCN(C(C3CCCC(=O)N3)=O)C2)C1 N1(C(CCCCC=C)=O)CC(C(N2CCOC(C(C)(C)C)C2)=O)C2(CCC2)C1 C12(C(N3CCC(NC(Cc4c(C)occ4)=O)C(CO)C3)=O)CC(C)(C1)OC2(C)C C1(C)(CC)CC(NC(c2c(F)cnn2C(C)C)=O)CN1C(=O)Cc1ccco1 C(=O)(C(O)C(F)(F)F)N1CC(OCCOCCNC(c2c(OC)n[nH]c2)=O)C1 c1(CC(=O)NC(c2cnn(C)c2)C(=O)N(C(C=C)C2CC2)C)csnc1C C[Si](C)(C)CNC(=O)CCOCCNC(C1CC1c1ccco1)=O c1(CNC(C(N2CCCCCC2)C)=O)ccccc1CNC(C1CCCS1)=O c1(C(c2nnnn2C)NC(c2cnc(C)s2)C)c(F)ccc(C)c1Br N1(C(C(C)=C2CC2)=O)CCC2(CC2)CC1C(N1CCC1C(C)C)=O c12cnc(F)cc1C(=O)N1CC(C1)NC(=O)CCO2.c1(OC)ccc(CO)cn1 N1(C(c2cccc(COC)n2)=O)CCC(NC(C2CC(OC)C2)=O)C12CCC2 NC1C=CCCC1C(N1CC2CCCC12)=O.n12cc(cn1)C2 c1(C(N2CCN(C(C(N3CCC(C)C3)=O)=O)C(C)C2)=O)coc2cc(O)ccc12 C1(CC(=O)NCC(=C)CC)CC(C)(C)CN1C(=O)CC(C)(C)O CON(CCC(=O)NOCC=CCl)C(=O)Nc1ccc(Cl)cn1 c1(-n2cc(C(C)(C)C(=O)CC3CC4CCC3(CO)C4)nn2)ccc(C#N)c(Cl)c1 N1(C(c2c(C)nsc2N)=O)CCC=C(CNC(=O)Cn2ncn(C)c2=O)C1 N1(C(C2CC2OC(=O)NC)=O)CCCC1CN.CCCCCN(CCCC)C N1(C(CC2(C)CCCC2)=O)CCC(O)(CNC(c2coc(C3CCC3)n2)=O)C1 N(C1CC(C)(C)Oc2ccc(F)cc21)C(c1c(OC)cncn1)=O CC(C)CCCCC(=O)N(C1CCC2CN(C(=O)CC3CCOC3C)CC12)C N1(C(C(C)C2CC2)=O)CC=C(C(=O)NCC2CCC(C)(C)CO2)CC1 C1(C(N(C2C(C)C2)CCO)=O)CCCC(NC(=O)CCCN(C)C)C1 N1(C(C2CC(C)(C)C2C(F)(F)F)=O)CCC(CO)(NC(=O)Cc2cc[nH]n2)CC1 C(C)(CO)(CN=c1[nH]c(=NC(C)CN2CCCCCC2)[nH]c2cccnc12)OC N1(C(c2cc(O)ncc2Br)=O)CCn2c(C3CCCCN3)nnc2C1 C(N=c1[nH]c(N2CCSC(C)C2)nc2c1CCC2)C1(CC)CCCC(=O)N1 N1(C(c2cc(OC)n(C)n2)=O)CCC(C)C(NC(c2cccnc2)=O)C1C C(=O)(CC(C)CC(C)(C)C)NCC(CC=C)C(=O)N1CCN(CC)CC1 c1(C(N2C(C(=O)NC(c3ncnn3C)C)CC3CC32)=O)c[nH]c2nccc-2c1 C(N=c1[nH]c2ncnc-2c(C(F)(F)F)[nH]1)C1N(C(C(C)SC)=O)CCCC1 c1(C(c2n(CCOCC)nnn2)NC(c2scnc2C)C)cnc(Cl)n1C C1(NC(c2cc(C)no2)=O)CCN(C(=O)Cn2ccc(=O)n(C)c2=O)CC1(C)C c1(C(N(C(C)CCNC(C2CCC(F)(F)C2)=O)C)=O)cccn(C2CCC2)c1=O CC1C(C(=O)NC2(C)CSC2)CCN1C(=O)C(=O)N(C)C N1(C(C2N(CCC)CCC2)=O)CCCC(CC)C1C(=O)NCCCSC(F)F c1(-c2ccn(C)c(=O)c2)nc(C(=O)Nc2cccc(C#N)c2Cl)n2ccccc12 N1(C(C=Cc2n(C)ncc2)=O)CCN(C(=O)CCc2cncs2)C(CO)C1 N1(C(CC2C(C)=NNC2=O)=O)CC2(C(=O)NCC3(C)CNC(=O)O3)CC1CCO2 CCC(CCCO)N=c1[nH]c(N2CCOCC2)nc(=NCc2cnn[nH]2)[nH]1 C1(NC(C2(CC)CCCCO2)=O)CC=C(C(=O)N2CCC(COC)CC2)C1 N1(C(C(=O)Nc2cccc(C3(N)CC3)c2)=O)CCC(O)C(F)(F)CC1 C(=O)(C1=NOC(C)C1C)NC1C(CC)CN(C(=O)CN2CC(=O)NC2=O)C1 c1(N(C(C(C(C)C)NC(C)=O)=O)CCNc2ccccc2F)ncccc1C#N n1(CC(=O)NC(COC)CNC(=O)CC2(CO)CCC2)cc(Cl)c(C)n1 c1(Nc2cc(C(N3CCCC(C(=O)OCC)C3)=O)no2)cc(Cl)ccc1[N+](=O)[O-] c1(CC(=O)NC2CN(C(C(c3ccc(C)cc3)=O)=O)C(C)C2)cc(O)nc(O)n1 C(CC(C(=O)N(CCCC(=O)OCC)C)NC(=O)CC1CC1CC)=CC C(C(O)CC(F)(F)F)C1CN(C(C(c2ccccc2)NC(CCN=[N+]=[N-])=O)=O)C1 Cc1cccc2c1OCC(NC(c1occc1CSCC(=O)O)=O)C2 C#CCC(C(=O)NCCCCCC)NC(N1CC(NC(=O)C(C)(C)C)SCC1)=O N#Cc1ccc(O)c(NC(=O)C(C2CCOC2)NC(c2cc[nH]c2)=O)c1 c1(OC)ccc2[nH]cc(C(=O)NC3CCOCC3NC(C3CSC3)=O)c2c1 C1(C)(CC)CCC(CNC(=O)C(C)=CCNC(c2ccc[nH]2)=O)O1 c1(C(N(CCOC)CCNC(c2cc(C)sc2C)=O)=O)cncn(C)c1=O N=c1nc(Cl)cc(C(N2CCCC(CNC(=O)CCN3CCCCC3)CC2)=O)[nH]1 Cc1nn(C)c2sc(C(=O)NC34CCCC3CN(C(=O)C=C3CCC3)C4)cc12 CCC(CC)CC(=O)NCCOCCNC(=O)CCCOC(C)(C)C Cc1c(NC(=O)C(=O)N(C)CCc2cccc(Cl)c2)cccc1Cl C(=O)(C1=CCCO1)N1C(C(=O)ON(CC(N2CCOCC2)=O)CC2CC2)CCC1 CC1CCC2(CC1)CCN2C(c1ccc(F)c(Cl)c1F)C(=O)NCCCF C1(C2CCC2)(c2onc(Cc3c(CC)c(C)ccc3)n2)CCNC1 N1(C(C=CC(C)(C)SC)=O)CCCCC1C1CCN(C(c2ccc(Cl)s2)=O)C1 C1(OC)CN(C(c2ncc(F)cn2)=O)CC1NC(=O)C(c1ccc(Cl)s1)=O c1(OC)cccc(CCC(=O)NC(C(C)NC(=O)Cn2ccnn2)C(C)C)c1F N1(C(C(C)Cn2cccn2)=O)CC2(COC(CNC(c3ccccc3F)=O)C2)C1 Clc1cscc1CNC(c1ccnn1CC(F)F)c1nnnn1C1CC1 c1(C(=O)OC)ccc(O)c(C(=O)NC2CC2CNC(c2csc(Br)c2)=O)c1 Cc1cc(C(N2CC(C3(NC(=O)Cc4nccn4C)CC3)C2)=O)c(C)n1C(C)C Cc1cc(=NC(=O)CN(C(C)(C)CO)C(c2cccc(F)c2C)=O)[nH]o1 c1(CC(=O)NC2CC3CN(C(c4cc[nH]c4C4CC4)=O)CC23)c(F)cccc1F N1(C(COCCC(C)C)=O)CCC2(NC(=O)CCCn3c(O)nnc3O)CC2C1 C(=O)(C(C)(C)CC(F)F)N(C)CCOCCC(=O)NC1CCCCC1C(N)=O c1(C(=O)NCC2(C)OCCN(C(C=NOC)=O)C2)cccc2c1CCS2(=O)=O C1(CCNC(=O)CCc2ccc(C)o2)(OC)CN(C(c2ccoc2)=O)C1 CCS(=O)(=O)CC(=O)N1CCC(n2cc(-c3ccccc3O)nn2)C1 C1(CCNC(C2C=CCC2)=O)CCCN(C(=O)Cc2cc(C3CC3)no2)C1 C1(NC(C(c2ccoc2)NC(C(C)CO)=O)=O)CCCC(C2CC2)C1 c1(C(N2C(CCNC(c3c(C)cnnc3)=O)COCC2)=O)ccc(Br)c(F)c1 C1(C(=O)NC2(CC=C)CN(C(=O)Cc3[nH]cnc3C)C2)COCCN1C c1(NC(C2C3CN(C(C(CCC)CCC)=O)C2C3)=O)ccc2c(c1)OCCO2 c1(C(=O)NC2C(CNC(C(=O)NCC3CC3)=O)CC2)c[nH]ccc1=O N#Cc1cc(C(N2CCCC(CS(=O)Cc3ccccc3)C2)=O)sc1Br C1(NC(C2(NC(CCOC)=O)CCC2)=O)CCNC(=O)C1 c1(C(C(C)NC(=O)NCc2c(I)ccnc2F)OC)cc(Cl)cc(Cl)c1 C1(C(N2C(CN(C(=O)CC(C)(C)O)C)CCC2)=O)COC2CCCCC12 CCC(CC)CC(F)C(=O)NC(C)CC(=O)N(C)CC1CCCN(C)C1 c1(NC(C=C)C(=O)OC)ccc(C(N2CC(OC(C)C)C2)=O)cn1 c1(C(N(CC(C)NC(=O)CN2CCNC(=O)C2)CC)=O)cc([N+](=O)[O-])c(C)s1 C1(CC)(NC(=O)CN2CCCOC2=O)CCCN(C(c2cc(Cl)nnc2O)=O)C1 CC(CF)C(=O)NCC(C)(C1CC1)NC(=O)CSS(C)(=O)=O C1(NC(c2ccc(Cl)s2)=O)CN(C(=O)Cc2ccc(Br)cn2)CC2CC12 c1(N(C)Cc2cc(F)cc(Cl)c2)nc2ccc(Cl)cc2c(=NCC2CC23CC3)[nH]1 C1(C(F)(F)F)(NC(C2CCN(C(CNC=O)=O)C2)=O)CCCCC1 N1(CC2=CCC(NC(=O)C3=NOCC3)C2)CCC(CO)=C(F)C1 c1(C(=O)NC2(CNC(C3CC4CC3C3CC43)=O)CCCC2)scc2c1OCCO2 C1(NC(C(C2(O)CN(C(C3(C)CCNC3=O)=O)C2)F)=O)C2CCC3C(C2)CC13 C#CCC(C)(C)C(=O)NC1CC2C(NC(=O)C(C)(C)CC#N)C2C1 N1(C(C2CN(C(C(COC)N(C)C)=O)C(C)(C)C2)=O)C2CCCC1CN(C)C2 c1(C(N2CC(NC(C3CCN(C(C)=O)C3)=O)C2)=O)cc(Br)nn1C CCC(CC)CCCNC(=O)C(C1CCN(C(=O)CCS(C)(=O)=O)CC1)C CC1CCCC=C1C(=O)N1CCC2CN(C(c3ccc(F)cc3Cl)=O)C2C1 N1(C(C23C(NC(c4c(C)cccc4)=O)C4CC2C3C4)=O)CCOC2(CCC2)CC1 N1(C(C2C(C)C2)=O)CCC(C(F)(F)F)C(NC(C2(C)CCCOC2)=O)C1 C1(C(=O)NC(CCNC(CCS(=O)(=O)NC)=O)C)Cc2ccncc2N1 C(=O)(C1=C(C#N)CCC1)N(C)CC1CCCC(NC(c2ccc(C)s2)=O)C1 CC(C)(CCNC(=O)CC1CCSC1)C(=O)NC1CCN2CCC1C2 C(=O)(CC(C)C(C)C)N1CCC(C)(C(NOC(CC)CC)=O)C1 C1(C(N2CCCC(NC(CC(CC)CN(C)C)=O)C2=O)=O)CNC(=O)CC1(C)C C(=O)(C1CCc2nccn21)NCC1(C)CC(C(NOCCCC#C)=O)C1 Cc1nn(C)c(-n2cncn2)c1NC(N1CCC(c2cc(Cl)ccc2O)CC1)=O c1(C(=O)NCCC(C)N(C)C(C23CCCN2CCC3)=O)ccc(Cl)c(F)c1 c1(C(=O)NCC(CNC(CCC(CC)OC)=O)OC)cc2nccnc2cc1F CC1(C)C2CCC(C2)C1C(=O)N(CCNC(C1CCCSC1)=O)CC1CC1 C1(C(N2CC3CCC2C3)=O)CCCCN1C(=O)Cc1ccc(Cl)cc1 C1(C(=O)NCC2(C)CC(NC(=O)CSC3CC3)C2)CC2C(C1)C2(F)F c1(NC(N2CC(C(CC)C)C2)=O)ccn2nccc2n1 CC(C)C(F)(F)CC(=O)N1CCC1NC(=O)CNS(=O)(=O)C1CC1 N1(C(=O)NC2CN(C(C)=O)C3C2C3)CCCc2ccccc2C1 C(C(=O)NCc1ccc(Cl)c(Cl)c1)(C(C(C)C)C(C)C)N(CC(=O)OC)C(C)C c1(NC(C(CC)N(C)CC)=O)ncccc1C(N1CCCCC1C(=O)OC)=O C(=O)(C(C)(C)C(C)(C)C)NCC(CC(F)(F)F)NC(Cc1cc(C)c(F)cc1)=O C(=O)(C1COc2ccccc21)NC1CCC(NC(C(CSC)(C)C)=O)CC1 CCC(CC)(CCC(=O)NC1CC(C)N(C(c2nocc2C(C)C)=O)C1)[N+](=O)[O-] C(=O)(C(CNC(=O)C(C1CC1)OC)CC1CCCC1)N(CCCN(C)C)CCC C(c1ccccc1)=C(OC)C(=O)NCC(C)NC(=O)CCc1cncn1C C1(OCC(=O)NCCC(=C)CNC(=O)C(F)=CCCF)CCCCCC1 c1(C(N2CC(CNC(CC(CC)O)=O)N(C)CC2)=O)ccc2c(C)[nH]nc2c1 C1(C(=O)NC(C2CN(C(CCc3onc(C(C)C)n3)=O)C2)C)CC12CCOC2 c1(NC(C2CNCCN2Cc2cc(Br)ccc2F)=O)ccnc(Cl)c1I N1(C(CCc2cnc(C)s2)=O)CCOCC1CN(C)C(C1C2COCC12)=O Cc1occc1C(N1CCCC1C1CCN(C(=O)CNC(=O)C(F)(F)F)C1)=O c1(C(=O)NC2(CF)CCN(C(C(C)OCC=C)=O)C2)cc(=O)c(Br)c[nH]1 c1(C(N2CCC(CNC(c3c(OC)scc3)=O)C2(C)C)=O)nc2ccccc2[nH]1 c1(N2CCC(CC)(CN(C)C)C2)nc2cccnc2c(=NC2CC2)[nH]1 N1(C(=O)CONC(C23CCC(C2)C3)=O)CC(OC)C2(CC2)C1 C1(NC(COC2CCN(C)C2)=O)C2CC1N(C(C1(C)CC(C)(C)C1)=O)C2 N1(C(c2ccc(C)cn2)=O)CCN(C(=O)CC2=CCCC2)C2CCCCC12 c1(C(=O)NCC2CCN(C(C3N(CC)CC3)=O)C2(C)C)scc2c1OCCO2 C#CCCC(C(=O)N1CCC(CN=[N+]=[N-])C1)NC(c1cnc(C)nc1C)=O C(=O)(C1=NOC(C2(O)COC2)C1)NCC(CC)NC(c1cnnc(Cl)c1)=O C(=O)(CCC(C)(C)C#N)N1CCC(C(C)NC(c2ccnc(OC(C)C)c2F)=O)C1 CC1CN(C(=O)Cc2ccc(F)c(Cl)c2)CCN1c1ccc(F)cn1 C=CC1(C(=O)N(CC(C)(C)C(=O)Nc2c(C)cccc2C)C)CCOCC1 S(=O)(=O)(c1cnn2ccc(=NCCc3ncccc3F)[nH]c12)NCCCC(C)C c1(CC)conc1CC(=O)NCC(CC)NC(=O)C(F)(F)C1CCOCC1 N1(C(Cc2cnc(C)s2)=O)CCC2CN(C(c3cccc(Br)c3F)=O)CC12 C1(NC(c2nc(CC)oc2)=O)CN(C(c2c(Br)cncc2Br)=O)CC12CC2 CC(C)C(O)C(=O)N1CCC(C)(CNC(=O)CN2CCN(C)CC2)C1 C(=O)(N=c1cnc(I)c[nH]1)c1nc(N(C(C2C(C)=CCC=C2)=O)C(C)C)sc1 Cc1cc(Cl)ccc1OCC(=O)N(CC(C)N(C)C(C1CCC(C)(C)C1)=O)C C(CCC)(C(=O)NC1(C(=O)NCC2CC(SC)C2)CC1(C)C)=CCC Cc1c(C(=O)NC2CCCC(N(C(=O)CCS(=O)(=O)N(C)C)C)C2)cccc1F C1(NC(=O)CC2C3CN(C(c4coc(C5CC5)n4)=O)CC23)CCN2CCC1C2 N1(C(C2(CC#C)CCCO2)=O)CCC2(CCCN(C(=O)Cc3nccn3C)C2)C1 N1(C(c2cc(C)nc(Cl)c2N)=O)CC2CC(O)C1C2NC(c1c(OC)csc1)=O c1(C2(COC)CC2)ccc(C(=O)NCC(C)CNC(=O)CC2CSCCS2)cc1 c1(C(=O)NCC2CC(C)N(C(=O)CC34CNC(=O)C(C3)C4)C2)ccc(F)c(O)c1 N1(C(c2c(NCC)cccc2)=O)CCCC(C)(CNC(C2CCC(F)C2)=O)C1 N1(C(C2CCC(C)(CC)O2)=O)CCC(CNC(c2cccc(N)c2F)=O)C1(C)C c1(C(=O)NCC(CNC(c2ccc(C(N)=O)o2)=O)O)cccc2ncnc(O)c12 N1(C(C2CCCN(CC)C2)=O)CCC2(CCCN2C(=O)C=Cc2csnc2C)C1 C12(C(=O)OCC)CCC(NC(c3cc(Cl)cnc3F)=O)(CC1)C2 c1(C(C(=O)NC(CCNC(c2c(C)cno2)=O)C)O)ccc(F)c(Cl)c1 C1(CNC(CCC=C(C)C)=O)CCN(C(C23CC(C2)C3)=O)CC1 O=S(=O)(c1cnc(NCC2C3CCCC23)c(Cl)c1)N1CCOCC(O)C1 C1(NC(c2c(C)nc(O)[nH]2)=O)CCN(C(c2cc(Cl)ccn2)=O)C1(C)C C12(CCCCC1)c1ccc(cc1)N(C(=O)CC(C)(C)C1CCCCC1)C2.CCN CN1CCC(CNCCC(=O)Nc2ccncc2)C1c1ccc(F)cc1 C1(c2ccccc2Cl)(C(=O)NCC2C(NC(COCCC=C)=O)C2)CCCCC1 C(c1nc2ccccc2s1)=CC(=O)NCCN(C)C(C1CCC=CCC1)=O C1(NC(C(C)N(C(C=CC(C)C)=O)C2CC2)=O)C2CCCCCC12 C#Cc1cnn(C)c1C(=O)NC(CC(C)C)C(=O)NCC12CCC(CO1)C2 c1(C(=O)OC)ccc(NC2CCNC2c2ccccc2)c(F)c1 c1(C(=O)NCC23CC(CNC(C=CC)=O)(OC2)C3)cn2cccc(C)c2n1 c1(NC(CC)(CNC(=O)CC2CC=CC2)CC)ncc2ccnc-2[nH]1 C1(NC(CCCOC(C)C)=O)COCCN(C(=O)C(c2ccccc2)C2CC2)C1 C(=O)(C1CSc2ccccc21)NCCCCCCCC c1(OC)ccc(C(=O)NC(C2CCCCN2C(=O)C=C2CC2)C)cc1C1CC1 C12(C(=O)NC(C(N3CC(C=C)OCC3)=O)CCC)CCC(OC)(CC1)CC2 CCC(C)CC(=O)N1CCCCC1CCNC(=O)Cn1cnc(C(N)=O)n1 CCCCC(C)(C)NC(=O)C(CN(C)C)NC(=O)C(C)(C1(C)CC1)OC Cc1cc(C(=O)N(CCCN(C(=O)C(C)NC(=O)CC(C)(C)C)C)C)nn1C C1(C(N2CC(CC(C)NC(Cn3ccc(C)n3)=O)C2)=O)CCC2(CCOCC2)C1 c1(C(=O)NC2(C)CN(C(=O)C(F)(F)CC3CCCO3)C2)cc2ccccc2o1 CN1CCN(C(C2CC3(CC3)CO2)=O)CC1C(N1CC(C#N)C1)=O N1(CC(c2cccc(C#N)c2)(C)C)CCc2sc(-c3c[nH]nc3C3CC3)cc2C1 c1(OC)cnc(Cl)cc1C(N1CCC(CN(C)C(c2ncccn2)=O)C1)=O c1(CN2C(C(N3CCC(O)C(F)C3)=O)CC(F)C2)c(Br)cccc1[N+](=O)[O-] C1(CNC(C(C2CCCCC2)C)=O)CN(C(c2cnc(O)n2C)=O)CC1O C1(CC(=O)NCCN(C)CCF)CCN(C(C2CC3(CC3)C2)=O)C(C)(C)C1 C1(NC(C2CCN(C(=O)NC)C2)=O)CCN(C(=O)C=Cc2ccco2)C1C c1(OC)ccc(Cl)cc1C(=O)NCC(C)(C)CN(C)C(C1CCOC1C)=O C(CC(=O)NC(CO)C(C)(C)C)(C(C)C)NC(C1(COC)C=CCC1)=O Cc1scc(C(=O)NCC(CO)NC(=O)CN2CCN(S(C)(=O)=O)CC2)c1N C(CC(C)(C)C(=O)NCC(C)O)NC(c1c(C)cccn1)=O N1(C(C(C)OCCC=C)=O)CCC(CNC(c2coc(Br)n2)=O)(OC)C1 c1(C(=O)NC2CCC(N(C(c3cc(C)sn3)=O)C)C2)c(Cl)ccc(C)c1N C(=O)(C(O)C1=CCCCC1)NCCC(C(=O)NCC(CC)(CC)CO)(C)C c1(OCC(N2CCC(C(N(CC)CC3CC3C)=O)CC2)=O)ccc(C)cc1C CS(=O)(=O)c1ccc(C(=O)OCc2ncccc2C(F)F)o1 CCN=c1cc(C(=O)NC2CC(NC(=O)C3=C(Cl)CCCC3)C23CCC3)cc[nH]1 c1(C(C)OC(C(C)Sc2ccc(OC(C)=O)cc2)=O)cc(=O)n2c(C)cccc2n1 C1(C2CCN(C(c3sc(Cl)cc3Br)C(=O)NCC3CCCO3)C2)COCCC1(C)O C1(CCNC(C2C(C)(C)COCC2)=O)CCN(C(C2(O)COC2)=O)CCC1(F)F C(CCN=C(NCC(c1ccccc1)O)NC1C(C)(C)C1(C)C)SC N1(C(C2C(C=C)C2)=O)CCOC2(CCN(C(C3(COC)CCCCC3)=O)C2)C1 O=C1c2ccc(F)cc2CC12CCC(=O)N2CN1CCCCC1c1ncc[nH]1 c1(CC(=O)NC2C3CN(C(C(C(C)(C)C)SC)=O)CC32)ccccc1S(N)(=O)=O N1(C(C(C(C)C)N(C)C)=O)CC2OCC(NC(=O)CCc3cccc(F)c3)C2C1 Cc1ncnc(C)c1CC(N1CCC(OCCNC(=O)C=CC2CCCC2)C1)=O C1(C(N(C(CC)C)CC(=O)Nc2ccccc2F)=O)CCCC12CCOCC2 c1(CC(=O)NC(CC(C)C)Cn2cc(-c3nccs3)nn2)cccc([N+](=O)[O-])c1 N1(C(C2(OC)CCOCC2)c2nnnn2C2CCCC2)CCCC(OC)C1 c1(C(=O)NCC(C)NC(C2(CCC)CCNC2=O)=O)ccnc(O)c1F Cc1cc(C(=O)NCC(C)NC(=O)CC2NC(=O)NC2=O)n(-c2ccccn2)n1 C(=O)(CC1=CCN(C(=O)C(C)(C)CC(C)=O)CC1)NC(CCOC)C(C)C CC(C)C(CCCC(=O)O)NC(c1ccc(-n2cc(C(C)(C)O)nn2)cc1)=O CC1=C(CNC(C2(NC(=O)CC3COCCO3)CC2)=O)CCC1 C1(CNC(=O)CCC2CC2)CC2(CCOCC2)CN1C(=O)CCCC1CC1 c1(C(N2C(C(=O)Nc3c(I)ccc(C)n3)CSCC2)=O)ccc([N+](=O)[O-])cc1C Cc1ccc(C(N2CCC(C)C(NC(=O)CCSC(F)(F)F)C2)=O)cc1C#N Nc1cccc2c1ccn2CC(=O)OCCCCC1CCCC1 n1(CC)ccnc1-c1cn(C(C)C(=O)NC2CC(CC(=O)OC)C2)nn1 c1(CCC(=O)NCC(C)NC(c2nc(COC)sc2)=O)nnc(C)n1C c1(C(=O)NC(CCC(=O)NC(CC)CC(=O)OC)(C)C)ccc(F)c(O)c1 c1(CC(=O)NCCOC(CNC(C2C(CC)OCC2)=O)(C)C)ccc(O)c(F)c1 c1(C(=O)NCC2C(OC)CCC2)cccc(CC#N)c1 N1(C(C2C(C(C)C)C2)=O)CCC(NC(c2cn3c(n2)CCCC3)=O)C12CCC2 C1(CC(=O)NC2C(C(N(C(CC(=O)OC)C)C3CC3)=O)OCC2)CCCCC1O N1(C(c2ccc(C(C)=O)[nH]2)=O)CC2CN(C(c3ccc(I)cc3)=O)CC12 Cc1cc(F)cc(C(=O)NC2CN(C(c3c(O)cccc3F)=O)CC23CC3)c1C Cc1nc2cc(C(=O)NC(C3CN(C(=O)Cc4cnco4)C3)C)ccc2o1 CS(=O)CCC(=O)NCC1CCC(CNC(c2csc(S)n2)=O)CC1 CC1(NC(c2cc(F)ccc2F)=O)CCN(C(C2CCCCN2N=O)=O)CC1 C1(CC(=O)NCCOC2CN(C(Cc3cnn(C)n3)=O)C2)CC2(CCC2)CO1 C1(CN(C(=O)Cc2ccccn2)C)COCCN1C(c1ncc[nH]1)=O N1(C(c2c(CC(C)C)n(C)nc2)=O)CCC(NC(C2(C)CCC2)=O)C(CO)CC1 N1(C(c2cc(CC)n[nH]2)=O)CC2(C1)CN(C(c1cccc3scnc13)=O)CCO2 Cc1cc(C)c(C(N2CC(CNC(C3(F)CC3)=O)C3(CCC3)C2)=O)c(C)n1 N1(C(C(C)=C2CC2)=O)CC(CNC(=O)COCC2CCOCC2)CC12CCC2 C1(OC)(CNC(c2conc2C(C)(C)C)=O)CCN(C(c2cnsn2)=O)CC1 C(=O)(C(F)C(F)(F)C(F)(F)F)NCC(CO)NC(C(C(C)(F)F)(C)C)=O C1(CC(=O)NC2CCN(C(C3SC4C=CC3C4)=O)CC2)CCC2(CC1)CC2 C(=O)(C(C)C(=O)OC)NC1CC(C(=O)NC(CCC=C)C)C1 C1(O)(C(=O)NCC2CC(COC)CN2C(=O)CCSC)CC2CCC1C2 CC1(C)CC=C(C(=O)N2CCCC(CO)(NC(C3CCS3(=O)=O)=O)C2)CC1 Cc1ccc(CC(=O)NCCOCCNC(c2occc2C)=O)c(Br)c1 C(=O)(CCN=c1[nH]c2ccccc2s1)N1C(CNC(CCC(N)=O)=O)COCC1 C1(OC)CC(C)CN(C(C2(C)CCN(C(=O)Cc3nocc3C)C2)=O)C1 c1(C(=O)NCC2(NC(C(C)n3cncn3)=O)CCOC2)csc2nccn12 CCCCC(CC(=O)Nc1ccc(C)nc1C)NC(c1cnsc1)=O C1(C(N2CCC(C)N(C(=O)Cc3cnn(C)c3)CC2)=O)CCC2(CC1)OCCO2 N1(C(CCC)=O)CCCN(C(=O)NC2(n3cc(Br)cn3)CC2)CC1 C1(NC(CCC(=O)NCCC)=O)CCN(C(=O)C(OC)OC)CCC1CO C=C(Cl)CC(C(=O)N1CC(C2CCCO2)C1)NC(=O)CN1CCCC1 C1(C)(C(=O)NC2C3(CC(NC(C4OCCN(C)C4)=O)C3)C2)Cc2ccccc2C1 c1(CNC(C2CC2F)=O)cc(O)nc(CNC(C2(C3CC3)CCC2)=O)n1 CC1(C)COC(C)(C(=O)NC2CCCN(C(=O)Cn3cnnc3)C2)CO1 c1(C(=O)NC2(CF)CCN(C(=O)CN3CCCCCC3)C2)cc2c(s1)CCCC2 C1(CCNC(C(CC)(C)CO)=O)CC2CCC(C1)N2C(=O)C(C(C)OC)N(C)C c1(C(N2CC3C(C(=O)OC)(C3)C2)=O)cc2cc(O)ccc2cc1O N1(C(CCc2cc(C)n(C)n2)=O)CCN(C(C2(CO)CCC2)=O)CC1C1CCC1 CCCC(CC)C(=O)NC1CCC(C)N(C(=O)Cn2ncccc2=O)C1 c1(C(N2CCN(C3CCN(C(=O)CCF)CC3)CC2)=O)cccc2sccc12 C1(F)(CNC(c2ccn(CCC)n2)=O)CCC(CNC(C2CC2[N+](=O)[O-])=O)C1 c1(CC)c(C(=O)NCc2cncc(C(=O)NCCOC(C)CO)c2)ccn1C Cc1ccc(C)c(OCCC(=O)NC(CNC(=O)CP(C)(C)=O)C(C)C(C)C)c1 N1(C(Cc2ccc(OC)nc2)=O)CC2(CNC(c3cscc3Cl)=O)CCC1CC2 c1(C(=O)NC2C(NC(CSCCC)=O)CCOC2)ccc2nncn2c1 CCCCCC(O)CC(=O)N(C(C)CCNC(=O)CC1CCCN1C(C)=O)C Cc1cc(C(=O)NCC2(C(C)NC(=O)Cn3cnccc3=O)CC2)ncc1F c1(NC(c2ccco2)COC)nc(N(C)CCCCC(C)(C)C)nc2sccc12 N1(C(=O)COc2ccccc2)CCC(OC2CCC2(F)F)CC1 c1(NC(c2scc(C(=O)Nc3c(I)ccc(C)c3)n2)=O)cc(F)cc([N+](=O)[O-])c1 N(C(=NCCC1=CCCCC1)NC(c1ccco1)C)Cc1nc(COCC)on1 CCC(CC(=O)N1CC(C(N2CC(O)CC2(C)CO)=O)C(C)(C)C1)C(F)F C1(C(=O)NCC2C(C(=O)NCCc3c(C)ncs3)CCO2)CC12CCOCC2 c1(CNC(C23N(C(c4c(C)nc(CC)o4)=O)CCC2C3)=O)ccc(O)cc1C c1(C(=O)NC(C)CCN(C)C(C2(CF)CCC2)=O)ccc(Br)nc1O C(=O)(C1=CCC(NC(c2sc(F)cc2C)=O)C1)NC(C#C)(C)C1CC1 c1(CNC(C(CCC)NC(=O)CN2CCCCC2C)=O)c(C)cccc1F c1(CNC2(CCCOCC3CCC(F)C3)CCC2)cc(O)ccc1Cl c1(C(N(C2CN(C(=O)COC(F)F)CC2F)C)=O)cc(F)cc2nn[nH]c12 C1(CNC(C=C(COC)C)=O)CCC(C)N(C(c2csnc2OC)=O)C1 N1(C(CCC2(NC(C3OCCN(CC)C3)=O)CCCC2)=O)CC2CCCCC2C1C c1(CCC(=O)NC(CNC(C2C(C=C)CC2)=O)(C)CO)ccnc(Cl)c1 N1(C(CCC=C(C)C)=O)CCCC(NC(=O)Cc2cc(C)no2)CC1 c1(C(=O)NC2CC3(CN(C(C(CC)C(C)C)=O)C3)C2)cc(C)c(C)c2ncsc12 Cc1c(OC(C2CCCN(C(=O)CN3C(=O)CNC3=O)C2)C)ncn1C.C(CSC)O N1(C(c2cn(CC)nc2C)=O)CC2(CC2)CC1C(=O)NC(C)(C)CC1CCC1 C1(C)(C(=O)NCCCN(C(C2CC2(C)C(F)(F)F)=O)CC)CC=CC1 N1(C(CCOCC#C)=O)CC2CC(NC(=O)CCc3ccsc3)C1C2 N1(C(C(C(C)(C)C)NC(C)=O)=O)CCC(C)N(C(=O)CC2CCC(=O)N2)CC1 Cc1cc([N+](=O)[O-])c(Cl)cc1S(=O)(=O)N1CC(C)N(C)CC1C C1(C(=O)NC(C)(C)CCNC(c2ccnn2C2CC2)=O)Cc2ccncc2C1 C(CCC(O)C(=O)NC1(CC2CC2)CC1)NC(CC1C(C)OCC1)=O C12(CNC(C(C=C)(C)CC)=O)CCCC1N(C(=O)COCCF)CCC2 c1(C(=O)NC(C)CN(C)C(C2CC2(Cl)Cl)=O)ncccc1OCC(F)(F)F Cc1oc(C(N2CC3(COC(CNC(=O)C=CC(C)C)C3)C2)=O)cc1S(C)(=O)=O c1(OCC(=O)NCC(CN(C(Cc2nnc(C)o2)=O)C)O)ccc(C2CC2)cc1 n1(CC)nnnc1CNC(=O)CCN(CCCO)C(=O)CC1CC1(C)C C1(CNC(c2snnc2C2CC2)=O)CN(C(=O)C2=COCC2)CC1C(F)(F)F O=C(CCCc1cnn[nH]1)NCc1cc(C(=O)N(C2CCOC2=O)C2CC2)no1 C(=O)(C(CC(F)F)N(C(=O)C=Cc1cc[nH]c1)C)N(CCC(N)=O)CC N1(C(C=CCC)=O)CCC(NC(=O)C(N2CCCCCC2)C)C(CO)C1 C1(NCCOCCOCCC)CN(C(=O)NC(C)(C)C)CCC12COC2 CC#CC1CCN(C(=O)C(C2CCC2)NC(C2COCC2(C)C)=O)CC1 c1(C(N(C2CCN(C(C3CC(C)OC3)=O)CC2)CCO)=O)cnc2[nH]ncc2c1 CCC(CC)(CN=c1[nH]nc(C)o1)NC(C1=CC(F)(C(F)F)C=C1)=O Cc1ccc(C(=O)NC2CCCCN(C(c3ccn(CC#N)n3)=O)C2)cc1F c1(C(N(C(C)CNC(c2cnc(OC)s2)=O)CC)=O)cc(Cl)ccc1[N+](=O)[O-] c1(C(=O)NCC2CN(C(C(=O)NCC)=O)CC23CC3)cc(F)c(C)cc1Cl N1(C2CC2)CCC(OCCN(C(=O)C(=O)NC)C(C)C)C1.C(C=O)OC c1(COCC)nc(-c2ccnnc2)n(C2CCCCC2C)n1 C(CCCCC(=O)NC(c1nn(C)cc1O)C)NC(C1CC(C)SCC1)=O N1(C(CS(=O)(=O)NC)=O)CCN(C(=O)C(C)C(C)(F)F)CC1c1ccccc1Cl C1(F)(CNC(C(CO)OC)=O)CCN(C(C2CC(F)(F)C2)=O)CC1 c1(CCN(C)C(=O)NC(C2CCCO2)(C)C)ccccc1[N+](=O)[O-] c1(C(=O)NCCOC2CCN(C(C3(CC)CCC3)=O)C2)cc2c([nH]1)CCC(C)C2 c1(C(=O)NCC2(OC)CN(C(CCN(C)CC)=O)C2)cc(OC)c2c(c1)OCO2 C(=O)(C1CCc2nccn21)N1CCC(C(C)(C)NC(=O)Cc2cnoc2)C1 N1(C(CC(c2cccs2)NC(C)=O)=O)CCN(C(c2cscc2C)=O)CCC1C C1(N(C(Cn2c(C)ccn2)=O)C)CCCN(C(C2(C)CC3CCC2O3)=O)CC1 CCC(C)(C)CCCC(=O)NCCC1(C)CCN(C(C2CCOC(=O)N2)=O)C1 c1(C(=O)NC2CC(NC(c3ccc(CC)[nH]3)=O)C2)cc(OC)cc(Br)c1C CCC(CC(=O)NC(CC(=O)NCc1cc[nH]n1)CC(C)C)C(C)(C)C O=C1Cc2ccc(C(=O)NC3(CNC(c4cc5ncccc5s4)=O)CC3)cc2N1 CC(CNC(=O)C(=O)NCC1CC1)CN(C)C(C1(C(F)F)CCC1)=O C1(NC(C2CCCO2)=O)CN(C(c2cnc(-c3ccccn3)s2)=O)CC1C(F)F C1(C(N(CC(C)NC(c2cc(CSCC)on2)=O)C)=O)CN2CCN1CC2C c1(CC(C)N(C(=O)C(=O)N(C)Cc2cncs2)C)ccc(F)c(F)c1 C1(F)(CNC(C=C(C)C(F)F)=O)CCN(C(c2cc(C(N)=O)cn2C)=O)CC1 N1(C(C=C(C)C)=O)CC(NC(C2(C(F)F)CCOCC2)=O)C(c2ccnn2C)C1 CC1CN(C(c2ccc(=O)n(C)n2)=O)CC1(C)CNC(c1ccc(Cl)cc1F)=O N1(C(C2CC2CC2CN(CC(F)F)CCO2)=O)CCOCC1C1CC1 C1(SC)CC(C(=O)NC(C2(C(=O)N(CC(C)C#N)C)CC2)C)C1 N1(C(C=C(C)CNC(C2COC(=O)N2)=O)=O)CCCC(C)(CO)C1 Cc1ncnc(C)c1CC(=O)NCC1CCC1CNC(c1ccc(Cl)s1)=O N1(C(C(C)(Cl)Cl)=O)CC2CS(=O)(=O)CC2(NC(=O)C=CC2CCC2)C1 c1(CNC(C(CC)NC(=O)CSC)=O)n[nH]c2c1CCC2 Cc1nc(CO)sc1C(=O)N(CC(O)CN(C(=O)C(O)Cc1cn(C)cn1)C)C N1(C(CCSCCC)=O)CCCC1(C)CNC(C1(F)CC(C(=O)OCC)C1)=O CC1CCN(C(C23CC2CCC3(F)F)=O)CCN1C(=O)CCc1cn[nH]c1 c1(OC)nn(C)cc1C(=O)N(C)CCN(C(=O)C(O)C(C)c1ccc(C)cc1)C C1(OC2CN(C(c3cnc(C)s3)=O)C2)CCN(C(C2(C)CCSCC2)=O)CC1 C(Cc1ccccc1)(C(=O)NCCC(N1CCOCC1)C)OC C1(COC(c2ccc(CC)[nH]2)=O)CC=C(C(C)C)CC1.C1(CC(C)C)CN1 C1(NC(=O)COCCNC(=O)CC(Cl)Cl)CCN2CCCCC12 c1(NC2CC(NC(C(CC)C(C)O)=O)C2(C)C)cc2nnc(C)n2cn1 C(=O)(CC(F)(F)CC)N(C(C(=O)NC(CN(CCCC)C)C)C)C N1(C(C(CC)=O)=O)CC(F)CC1C(=O)Nc1ncc(Br)nn1 CCC(C(=O)N1CCCC1CNC(=O)CCOCC(F)(F)C(F)F)C(C)(F)F N1(C(C2N(CC)CCC2)=O)CC(CNC(c2cncnc2C(C)C)=O)CC1(C)C N1(C(CCCN(C(C)=O)C)=O)CC2(C1)CN(C(C1CC(Cl)(Cl)C1)=O)C2 n1(CC)cnc2[nH]c(=NCC(C)C(F)F)nc(N3CCC(CC)(CO)C3)c12 c1(SC)ccc(C(=O)NC(C)CCCCNC(=O)C=Cc2sccc2C)c(Cl)c1 CC(N=c1cc[nH]cc1)C(=O)N1CCCC12CCN(C(=O)CC(C)(C)O)C2 C1(CC)(NC(C2C3CC2N(C(=O)CNC(=O)NC)C3)=O)CC(F)(F)C1 Cc1nnc(Cn2cc(SCCNC(=O)Cc3n[nH]c(C(=O)OC(C)C)n3)nn2)o1 c1(C(N2C(CC)C(NC(=O)CC(C)(C)C#N)CCC2)=O)ccc2c(c1C)CCC2 c1(C(C(=O)NCCCNC(C(C2CCCC2)OC)=O)(C)O)ccc(Cl)cc1 N1(C(C(C)=C2CC2)=O)CCC(C2CCN(C(C3CC(=C4CC4)C3)=O)C2)C1 C(=O)(CC(C)(C)C(C)(F)F)N1CCC(C)C(NC(=O)C(=O)NCC(F)(F)F)C1 C1(NC(C2CCN(C(N)=O)CC2)=O)COC2(C1)CN(C(=O)C(O)C1CCCC1)C2 C(=O)(C#CC1(C)COC1)N(C1CN(C(c2c(C(C)C)occ2)=O)CC1(C)C)C C1(CC)CN(C(=O)CC(C)(C)N(C)C(c2cccc(F)c2N)=O)CC(CC)O1 c1(CC)cc(C(N2CCCCC(NC(C3(COC)CCOC3)=O)C2)=O)c(C)nn1 c1(NCCC(=O)NC(CC)(C)CNC(C2CCOC2)=O)ccc(C)cc1 C(=O)(C(C)(C)CS(C)(=O)=O)NCCCNC(C(C)N(C(C)=O)C)=O Cc1cccc(NC(C2(F)CCN(Cc3cc(C(=O)O)ccc3O)C2)=O)c1Cl C1(C(=O)NC2CCCN(C(C(C=CC)O)=O)C2C)CCOCC12CCCCC2 c1(C(CNC(CCSC)=O)N(C(=O)C(C)OCc2ccccc2)C)ccccc1 c1(C(=O)NC2(C)CN(C(C3CC4(CCOC4)C3)=O)C2)nccc2ccsc12 Cc1cc(C2(C(=O)NCCC3CCCN(C(C4CC4(Cl)Cl)=O)C3)CC2)cc(C)c1 c1(OC)ncc(C(=O)NC2CCCC2C(N2CC3CC(C2)O3)=O)cc1Br c1(OC)ccc(CCC(=O)NCC23CC2CN(C(c2nnn(C)c2N)=O)C3)cn1 CC(C)CCC(F)C(=O)NCC(C)(C)OCCNC(=O)COc1cn[nH]c1 CCC(C(C)O)NC(C1(CCNC(c2cn(C3CC3)cn2)=O)CCCC1)=O N1(C(c2n[nH]c(C)c2F)=O)CCC(CNC(=O)CN2CCC(C)CC2)C12CCC2 C(CC)(CCCO)NC(c1c(CNC(CC(=O)NCC)=O)cc[nH]1)=O C(=O)(CCC1CC1(C)C)C(C1(C(=O)OCC)CC1)=O.C(=O)(C=CCC)OCC.NCC c1(C(N2CCCC(C)(CNC(C3(C#C)CCCC3)=O)C2)=O)nc2ccccc2[nH]1 C1(O)(C(N(c2ccccc2)C(C)C)=O)CCN(CC=CCN2CCCC2)CC1 C(C1CN(C(C23CCC(OC)C2C3)=O)CC1C(=O)NC(C1CCCCC1)C)=CC C1(NC(C(C)(C)C2CC2)=O)CCC(N(C2CC2)C(=O)CC2CCOC2)CC1 CCCC(C(=O)N1CCC(C(=O)N(C)C(c2cc(C)on2)C)(CO)C1)NC(N)=O C#CCC(C(=O)OC)NC(=O)C(c1ccoc1)NC(C1CC1(C)C)=O C1(NC(C2(C(C)C)COC2)=O)CCCN(C(C2CC(O)CN2C)=O)C1 C1(NC(C(C)OCCC(C)C)=O)CC(NC(c2c[nH]nc2C2CC2)=O)CC1O C1(C(=O)NC(C2CCCN(C(c3ccc(N)c(Cl)n3)=O)C2)C)CN2CCN1CC2 c1(NCC(C)N(C(c2c(OC)ccnc2)=O)C)ncnc2sc(C)nc12 c1(CC(CNC(C2(C(F)(F)F)COC2)=O)CO)ccc(-c2nn[nH]n2)cc1 C(C(N=c1[nH]ccn2c(NC3CCN(CC)C3)nnc12)C(C)C)OCC N1(S(CCCC)(=O)=O)CCOCC1(C)C(=O)Nc1cccc(C(=O)OC)c1F c1(C(=O)NCC(CNC(C(CC)C)=O)(C)C)coc2ccc(O)cc12 c1(CC)n[nH]cc1C(N1CCC1C(=O)NCCCOCC1CC1)=O Cc1cc(=O)n(CCC(=O)N(c2cccc(C#N)n2)C(C)C)cn1 C1(NC(C(C2CCN(C(c3cnc(O)o3)=O)C2)C)=O)CCC2CC1C2(C)C C(=O)(C=C1SCC(=O)N1C)N1C(C2(NC(C=CC=CC)=O)CC2)CCCC1 c1(NC(=O)C2=CSCS2)ccc(C(=O)O)cc1.C12C=CC(C1)NC(=O)C(=O)NC2 C1(C(C(N2C(CNC(C3CCN(CCF)CC3)=O)CC2)=O)O)CCCCCCC1 N1(C(C(C)Oc2cccnc2)=O)CCC2(CN(Cc3ccncc3Cl)C2)C1 N1(C(c2c(CC)noc2)=O)CCCC(CNC(C2(CO)CCCC2)=O)CC1 N1(C(c2cc(C)[nH]c2C)=O)CC2CCOC2(CNC(C2CCN(C)S2(=O)=O)=O)C1 C12CC3CN(CC13)C(=O)c1noc(c1C)N2.C1(C2C(=C)C2)CC12CCOCC2 C(=O)(C(CC)CC(C)C)N(C1CCN(C(c2cc(Cl)cc(C)c2O)=O)C1)CCC CC1CN(C(c2cnc(S)nc2)=O)CC(C)N(C(c2ccc(Cl)c(F)c2N)=O)C1 N1(C(CSC(C)C)=O)CCOCC1CNC(=O)C=Cc1ccc(C(N)=O)o1 c1(NC(=O)CC2CN(C(c3cccnc3Cl)=O)C2)cc(Cl)ncc1Br CC(CC(=O)NC1(CC(N2CCC(CC(F)F)C2)=O)CCCCC1)C(F)F C1(NC(c2c(C)ccn2C)=O)COC2C(NC(C3CC4(CC4)CO3)=O)COC12 Cc1ccc(CNC(=O)C(C2CCOC2)NC(=O)CN2CC3CC3C2)c(O)c1 N1(CCNC(c2c(C)nc(O)[nH]2)=O)CCCN(C(c2cnnc(O)c2)=O)CC1 c1(C(=O)NCC2CC(NC(c3c(C(C)=O)ccs3)=O)C2)ccnc(F)c1Cl c1(CN2CC(N(C)C3CC3)C2)cn2cccc(Br)c2n1 Cc1cnc2n1CCN(C(=O)Oc1ccccc1F)CC2 C1(C(=O)NC23CC(CNC(c4n(CCC)ccc4)=O)(C2)C3)CCC(C)(F)CC1 CC1(C)CC(C(=O)NCCN2CCOCC2)CN(C(=O)CC(C)(C)C(F)F)C1 c1(C(N2CC3C(CNC(C(C)CF)=O)(C3)C2)=O)cc(P(C)(C)=O)cs1 N1(C(CC2N(C(C)C)CCC2)=O)CCCC(C(N2CCCCC2)=O)C1 C1(CN(C(=O)CC2CC2)C)COCCN1C(C1C2CCC1(c1ccccn1)C2)=O C(=O)(C1=NNC(=O)C1)NCCN(C(c1nc(C)c(C)s1)=O)CC C1(NC(c2ccc(C)o2)=O)CN(C(c2cnc(Cl)s2)=O)CCC1CO Fc1ccc(-c2noc(C34CCCCC3C4)n2)c(OC2CC2)c1 c1(C(=O)NCC2C3CC2N(C(c2cc(C(F)F)no2)=O)C3)cc2n(n1)CCCC2 N1(C(C2CCCC(C)(C)C2)=O)CCC2CCC(NC(c3ncc(F)cc3N)=O)C12 CC(CCN=c1[nH]c(=N)[nH]c(=NCc2ncc(Br)c(O)n2)[nH]1)N1CCC1 c1(OC)cc(C(=O)NC(C2CCN(C(=O)C(C)(C)c3cc[nH]n3)C2)C)ccc1O c1(CC(=O)N(C(CNC(c2cnc[nH]c2=N)=O)C2CC2)C)ccc2c(c1)OCO2 C1(C(CNC(CC(C)F)=O)C)CCN(C(C2(n3ccnc3)CCCC2)=O)CC1 C(=O)(CC(C)C(F)(F)F)NC1CC(CC(=O)NC(COC)(C)C)C1(C)C C=CCC(C)(CC)C(=O)NC1CCCC(N(C)C(c2cnc(OC)c(Cl)c2)=O)C1 N1(CC)CCc2cc(-c3cccc(CC(C(=O)OCC)NC(=O)CSC)c3)ccc21 c1(OC)ncccc1CC(=O)NCC1(F)CC(NC(=O)C=CC(=O)N(C)C)C1 C1(COC)(CNC(=O)CSC)CN(C(c2cc(C(C)=O)c[nH]2)=O)C1 N1(C(CCSCCCC)=O)CC(C(=O)NC(=O)C(CCC)N(C)C)CC1(C)C N1(C(CC2N(CC)CCC2)=O)CCC2CC1CN2C(=O)CCCN(C)C(C)=O S(=O)(=O)(c1csc(C2CC2(F)F)n1)N(CC(CC)O)Cc1ccccc1 c1(CNC(C23CC(NC(C4C(OC)CCC4)=O)(C2)C3)=O)c(C)ncnc1C N1(C(C=CC(CC)=CC)=O)CC(CCNC(c2ncnc(O)c2Cl)=O)OC(C)C1 N1(C(C(CC#CC)NC(C2CCC(C)(C)CC2)=O)=O)CC2(CCC(=O)N2)C1 c1(C(CNc2n(CCOC)ncc2)O)ccc(OCC)c(OC)c1 c1(C(N2CC(CCC)N(C(C3CC3F)=O)CC2)=O)csc2c1CCCC2 C1(NC(C2(NC(c3cc(Cl)cn3C)=O)C(C)C2)=O)CCCN2CCCC12 C1(OC)CCCCC1C(=O)NCCCCCNC(=O)C(C)(C)c1cscn1 CN1CCCC1(C)C(N1CC(CNC(c2ncnn2C2CCOCC2)=O)C1)=O C1(C(=O)NCC2(C(N)=O)CN(C(=O)CCC3CCCC(=O)N3)C2)CC(F)C(=O)N1 C=CC(C(F)(F)F)NC(C1C(NC(=O)C(C)NC(=O)C2CC2)C1(C)C)=O c1(N2C(C)CC(NC(c3cnc(Cl)s3)=O)C2)ncc(C#N)cc1Br C1(CNC(C(COCC)(C)C)=O)CC2CC(C1)N(C(c1c[nH]cc(Cl)c1=O)=O)C2 C(=O)(C1COc2ccc(Cl)cc21)NC1C(CNC(c2c(CC)cno2)=O)CC1 n1(CCCC)nnnc1C(CC)(C1CC1)NCC1CCOC1.OC C12(CNC(=O)CC3CC(F)(F)C3)CCC1CN(C(=O)C(F)CC1CCCC1)C2 CC12COC(C(N3CCC(N4CCN(C(C5(F)CCOC5)=O)CC4)C3)=O)(C1)C2 C12(C(=O)NCC3N(C(C4CCC(=O)C4)=O)CCCCC3)CCCC(CCC1)C2 N1(C(c2cccc(CC)c2)=O)C(C)CC2CN(C(C3OCC4CCCC34)=O)CC12 Cn1c(O)nc2cccc(C(N3CC(CCNC(C4CCCC(O)C4)=O)C3)=O)c12 C(=O)(C1=CCCCC1)N1CC(C=C)(CC(=O)NCCN2CC(OC)C2)C1 N1(C(CC2CCN(C(c3c(C(C)C)onc3)=O)C2)=O)CCC(F)(CO)C1 CC1(C(N2CCCC(CNC(=O)Cc3ccc(F)cc3)CC2)=O)CCNC(=O)C1 Cc1cc(N)ccc1C(=O)NCC12CCC1CCN2C(=O)CCCNC(N)=O C1(NC(c2ccc(C)s2)=O)CC12CCN(c1ncc3c(n1)CCC3)CC2 C(=O)(C#CC1CCCCC1)NC(CN(C(C=C(C)C)=O)C)(CO)CO Cc1c(N(CC(C)(C)O)Cc2c(F)ccc(Br)c2Cl)ccc(Cl)c1Cl N1(C(CCC#C)=O)CCCCC1CCC(=O)NCC(C)(C)C(=O)NC CCCCC(O)C(C)C(=O)NCCC(C)(CC)NC(=O)C(O)CCC(C)C N1(CC(=O)NC2C(CNC(c3c(COC)nn[nH]3)=O)CCC2)CCNC(=O)C1 c1(C(C)C)ccc(C(=O)CN2CC(NC3(c4ccc(O)nc4)CCC3)C2)cc1 C1(OC)CC(NC(c2ccc(C(C)C)o2)=O)CN(C(C2CC2Br)=O)C1 c1(N2CC(C)(C)C(NC(C3CC4CC4C3)=O)C2)c(Cl)cncc1[N+](=O)[O-] n1(C(C)C)cnnc1C1CC1C(N1CC(C(c2cc(C(C)(C)C)n[nH]2)=O)C1)=O n1(CCC)cc(C(=O)N(CC(C)NC(C2CCCC2O)=O)CC)nn1 N1(C(c2n(CC)ccc2)=O)CCN(C(c2cscc2C(F)F)=O)C(C)C1 Cc1nc(C(N2CCC(C(=O)NC3CCCC3N(C)C)C2)=O)co1 C(CC1=CCC2CC1C2(C)C)NC(c1c(C(C)C)n(-c2cccc(Cl)c2)nn1)=O Cc1nc(Cl)ccc1C(N1CCCC(n2cc(CN3CCOCC3)nn2)CC1)=O C1(C2CN(C(C3(n4ccnc4)CCCC3)=O)C2)(NC(C=CC(=O)OCC)=O)CC1 c1(C(=O)NCC(CNC(=O)CCc2ccoc2)CO)c[nH]c2cc(F)ccc12 c1(C(N2CCC(O)(CNC(=O)CCn3cccn3)C2)=O)cnc2ncccc2c1 C(=O)(C(CO)C(C)(C)C)NC1CN(C(C(C(C)O)NC(C)=O)=O)C1 N1(C(c2c(C)n(C(C)C)cc2)=O)CC(NC(C2CC23CCC3)=O)C2(CC2)C1 C1(NC(c2c(CCC)nns2)=O)(CNC(=O)CCc2ccncn2)CCOCC1 c1(C(N(CC(C)(C)NC(C2C(CC)OCC2)=O)C)=O)nc(C)n(C)c1C N1(C(CC)=O)CCC2(C1)CN(C(=O)C(C)NCS(=O)(=O)Cc1ccccc1)C2 N1(C(C23CCC(NC(CC4C(C)(C)C4)=O)(CC2)C3)=O)CCN2CC(O)CC2C1 c1(C(c2n(C)nnn2)NC2CC2(C)C)cn(C)nc1C(F)F C12(C(=O)NCCc3c(CNC(COCC)=O)cccc3)CCCC1C2(F)F C(c1ccc(C)s1)=CC(=O)NC1C(CNC(C2(CC#C)CCCO2)=O)COC1 CC(F)CC(=O)N1CCC(NC(=O)N(C)C)C1 c1(NCCC(C)C)[nH]c(=NC2CSCC2C)nc2scnc12 C(=O)(CC(O)CNC(=O)CCC1CCOC1)N(CCC(=O)NC)CC c1(CC)ncc(C(=O)NCC2CC(NC(c3nnsc3C)=O)C(O)C2)cn1 Cc1nc([N+](=O)[O-])cn1CC(N1CCOC(CCNC(=O)C(C)CC(F)F)C1)=O C#Cc1ccc(C(N2CCC(NC(C3CC(OC)C3)=O)CC2C)=O)cc1 C1(NC(c2c(C)c[nH]c2)=O)CC2CCC(C1)N2C(C1(C(F)(F)F)CCCCC1)=O N1(C(C(C)OCCOC2CCCC2)=O)CC2CC1C2C(=O)NC1CCOC1C C(=O)(C1c2ccccc2Oc2ccccc21)NC1C(NC(=O)CCF)C1 C1(CNC(=O)CCOCc2ccco2)(CSC)CC(F)(F)C1 C12(CNC(CC3(C)CC3(F)Cl)=O)CC(CO1)N(C(C13CCC(CC1)C3)=O)C2 CC1(C)CCC(C(=O)NCC2(O)CC(O)C2)(NC(C23C(=O)C4CC2C3C4)=O)C1 c1(C(=O)NCC(CNC(C2C(COC)C2)=O)OC)cc(C)nn1C1CCOCC1 C1(CCCC)CCC(C)N(Cc2ccc(C(=O)Nc3cn(C)nc3C#N)cc2)C1 Cc1cccn(CC(=O)NCC2CC(C)CCN2C(C2CCCC23CC3)=O)c1=O CC1CN(C(C2CCOC2)=O)CC(C(=O)NCC2=CCCCC2)O1 C1(CCNC(CC2(OC)CN(C(C3CCS(=O)CC3)=O)C2)=O)CCC(C)(C)C1 C(=O)(CCCC(CC)CC)NCC(CCC)C(=O)N1CCC1C1CCCCC1 c1(OC)ccc(C2CC2)c(C(=O)NCCC(O)CNC(=O)C2=CCCC2C)c1 c1(C(N(C2CC(NC(C3(OC(C)=O)CC3)=O)C2)C)=O)cc2c(C)c(Cl)ccc2[nH]1 Cc1ccc2oc(N3CCC(C(C4C5Cc6ccccc6C45)=O)CC3)nc2c1 N1(C(c2c(C)cc(C(C)C)cc2)=O)CC2CCC1CC2NC(C1SCCCS1)=O c1(C(=O)NCC(CC)NC(=O)CCC=C(C)C)cnc(C)[nH]c1=N C1(C(=O)NCC(COC)OC)N(C(=O)C(C)NC(=O)NC)CCC1(C)C C1(C(N2CCC(NC(c3ccc(=O)oc3)=O)(CF)C2)=O)Cc2cc(F)ccc2O1 CCCC(C(=O)NCC(O)CC(=O)NC(CC)CCOC)OC C1(C(N2CCC(O)(CNC(C3(c4cccs4)CC3)=O)C2)=O)CC2(C1)CC1(CC1)C2 C1(CC(=O)NCC2N(C(CSc3n[nH]c(=N)s3)=O)CCC2)CCCC(C(N)=O)C1 C1(CCC#C)CC(CO)CN(c2nnc(CC(O)C=C)n2C)C1 c1(OC)ccc(OC)c(C(N2CCCC(CCNC(=O)C=CC(C)C)C2)=O)c1 c1(NC(C)=O)ccc(C(N2CCC(C(C)NC(c3c(C)ncn3C)=O)C2)=O)cc1 N1(C(C(CC)n2cncn2)=O)CCC(C(=O)NCc2ccc(Cl)cc2)C(C)(C)C1 N1(C(C(C)Cn2ccnc2)=O)CCN(C(c2cncc(O)c2)=O)CC(C)(F)C1 c1(C(=O)NC2CC(OC)C2)c[nH]nc1C1CCOCC1 C1(NC(CCn2c(C)nc(C)n2)=O)CC2CC(C1)N(C(c1c(O)noc1C)=O)C2 c1(C(=O)NC(CN(C(=O)C(=O)N(c2ccccc2)C)CC)C)nn(CC)nc1C C1(CC)CN(C(C23CC(CCO2)C3)=O)CCN1C(=O)C(n1nc(C)cc1C)C C=CCC(CNC(=O)C(C)(C)C)NC(C1CCN(Cc2ccccn2)C1)=O CC(C)C(F)C(=O)N1CCC(c2cccc(F)c2)(NC(=O)CCc2ccon2)C1 C1(CC)CN(C(=O)CC2CCCC(NC(C3CCC4(CC4)C3)=O)C2)CCN1C N#CC1CCCC(C(N2CCCN(C(c3ccc(C4CC4)s3)=O)CC2)=O)C1 C1(CN(C(=O)CN2CCCCCC2)CC)CCCCN1C(c1cc(CO)[nH]n1)=O c1(C(N2C(CN(C(=O)C3=C(Cl)CC3)C)CCCC2)=O)ccc2c(O)n[nH]c2c1 N1(C(CC(CC)C)=O)CCCC(NC(C2CCC(=O)N2)=O)C1C c1(CC(=O)NC2C(CNC(c3ncn(C)n3)=O)C2)ccc2ncccc2c1 C12(C(=O)NCCCOCCOC)COCC1CN(C(c1cnc(C)o1)=O)C2 CC1(CNC(=O)CC(C)n2ccnc2)CC(NC(c2ccc(C(N)=O)s2)=O)C1 c1(C(N2C3C(NC(CC(C=C)CC)=O)C(C3)C2)=O)cc(C)cc2c1NCCC2C N1(c2nc(COC)nc(O)c2)CC2(C)CN(C(c3cc(OC)ns3)=O)CC2(C)C1 c1(C(C)C)nn(C)c(Cl)c1C(=O)NCC1(NC(=O)CN2CC=CC2)CCOC1 c1(CC)cccc(CC(N2CCN(C(=O)CN(CC)CC)CC2)=O)c1 C1(CNC(CCc2cc(C)no2)=O)CC(C)CN(C(C2CC(N(C)C)C2)=O)C1 S(=O)(=O)(c1ccc(NC(CC2CCCCC2)CO)cc1Cl)NCC(C(C)C)(C)C Cc1cc(C(=O)NC(CNC(=O)C(F)(F)c2cncs2)C(C)C)co1 Cc1cc(C(=O)N(CCC(C)NC(=O)CN(C2CCCC2)C)C)on1 c1(C(=O)NCC2(NC(c3[nH]c(=NC)sc3)=O)CCC2)c(C)nc2cccnn12 C=C1CCC(C(=O)NCc2nocc2C(=O)NC(C)(CO)CCF)CC1 N1(C(C)=O)CCCC(O)(NC(CN(C)C(c2cnc(C(C)C)nc2C)=O)=O)C1 N1(C(COCCCC)=O)CCCC(NC(c2cccc(C3(C)CC3)c2)=O)C1C C12(CNC(CSSCC)=O)CC1CN(C(=O)CN(c1ccncc1)C)C2 C(CCC(C)C(=O)N1CCCC(NC(c2nonc2N)=O)C1)OC C1(COC)(NC(C2CCCCC2O)=O)CCN(C(=O)C(C)(C)O)CC1 c1(C(N2CCC(C)(CNC(CC3(C)CCC3)=O)C2)=O)ccc2c(=O)ccoc2c1 c1(OC)noc(-c2nc(C3CCCC3)nn2-c2nc[nH]n2)c1Br C1(C(=O)Nc2c(OCC)cccc2)CC2CCC1N2C(=O)C(CC)NC(C)=O C1(C(=O)NC2CC(NC(=O)CCCn3cccn3)C2)(OC)CCOC1 c1(C(=O)NCC(c2cccc(F)c2)NC(c2ccc[nH]2)=O)cccc2nonc12 N1(C(CC=CC=C)=O)CCCC1(CO)CO.C12(CCCC1)C(=O)NC(C)(C)C2 N1(C(C2=CCCN(C(c3[nH]cc(C)c3)=O)C2)=O)CCCC12CCNC2=O C1(C(N2CC(C)C(NC(c3cnn(CC(F)F)n3)=O)C2)=O)CCCCC1(F)F c1(C(N(CC(CC)NC(=O)C(c2cnn(C)c2)OC)C)=O)[nH]c(C)nc1C N1(Cc2c(C)nc(-c3ccc(OC)cc3)s2)C(=O)CCN(CC2C3CCC23)C1=O c1(C(=O)NC(Cn2cccn2)C(=O)O)ccc(CO)c(Cl)c1 C1(C(N2CC(CN(CC(C)C)CC)C2)=O)C2CC(O)C(C2)N1C(=O)CSC c1(C(=O)NC(CN(C(c2ccc(O)nc2Cl)=O)CC)C)cc(O)ccc1Cl c1(C(N2CC3CC(CNC(C4(C)CCCCO4)=O)C3C2)=O)ccc2cncn2c1 C(=O)(CC(C(F)F)C(=O)OC(C)(C)C)NCCCC(C)NC(C1(C)CC(=C)C1)=O C1(C(=O)NC2CCN(C(C=CC)=O)C2Cc2ccccc2)CCCC2(CC2)C1 C1(CNC(Cc2cn(C(C)C)nc2)=O)CCCCN(C(c2ncccn2)=O)C1 C1(C(=O)NC(c2cccc(C)c2)C)CN(C(C2CC3(CSC3)C2)=O)CC1(F)F c1(C(N(CCC=C)CC=C)=O)n[nH]c2ccc(-c3cnn(CCCOC)c3)cc12 C(=O)(CC(O)CC(C)(C)C)N1CCCCC(N(C(C(=O)NCC)=O)C)C1 N1(C(c2c(F)ccc(C)c2)=O)CCC2CCN(C(C3CCCN3C=O)=O)C2C1 c1(C(N(CCN(C(C2CC(=O)N(O)C2)=O)CC)CC)=O)cc(CC(C)C)nc(O)c1 c1(CN(CCOC(C2CCCN(C(=O)C(O)C(C)C)C2)=O)CC)ccc(C#N)cc1 c1(CNC(c2ccc(C)nc2)=O)nc2c(s1)CN(C(c1csc(C#N)c1)=O)CC2 C#CCC(C)(C)C(=O)NCC(CC=C)C(=O)N1CCC(N2CCC2)C1 CC1Cc2n[nH]cc2CN(C(c2cc(Br)c(F)cn2)C(=O)NCC2CCCO2)C1 c1(C(=O)NC(CCCNC(c2c(CC)occ2)=O)C)ccc2ccccc2n1 N1(C(C2CCN(C)C2)=O)CCCC2CN(C(=O)Cc3ccc(F)c(Cl)c3)CC12 C1(C(=O)NC2(CC=C)CCC2)CCN(C(=O)C(=O)NCC)C12CCC2 CC(C)CC(C(=O)NCC1CNC(=O)CO1)NC(c1cccc(=O)o1)=O c1(OCC)ccc(C(=O)Nc2nccc(C#N)c2OC)c2ccccc12 c1(CNC(C(CN(C(C(CC)(F)F)=O)C)C)=O)cccc(F)c1C CN1CCC(c2ncc(C(=O)NCCOC3CN(C(=O)C=CCF)C3)[nH]2)CC1 C(=O)(CCC(=O)NC(CO)C(=O)NC(C1CCCC1O)C)NCCC Cc1cc(C(=O)N(CC(C)C(=O)NC(C)(C)C(N)=O)C)cnn1 N1(C(C2(C)CCC(F)(F)C2)=O)CC2(CCCN(C(c3nocc3Cl)=O)C2)C1 C1(NC(=O)C(c2ccc(Cl)c(F)c2)O)CC12CCN(C(C1OCCCO1)=O)CC2 C1(NC(CCC#C)=O)CCN(C(=O)C(COC)OC)C2CC12 C1(NC(C(CC)N(C)C)=O)CC(F)CN(C(=O)Cn2nc(C)cc2C)C1 C(=O)(C1=CCCSC1)NC1C(NC(=O)Cc2cccc(OC(F)(F)F)c2)C1 C(=O)(C1=NOC(NCCCCNC(=O)C(F)(F)CC=C)C1)NCCCOCC#C c1(CNCC23C(CN(C(c4cc(C)on4)=O)C2)C3)cc(F)c(Cl)cc1Cl C1(S(C)(=O)=O)(C(=O)NCCN(C(=O)CC2CCCS2(=O)=O)C)CCC1 c1(OC)cc(N)c(Cl)cc1C(=O)NCC(C)(CC(C)C)NC(=O)C=CS(C)=O CC(C)C(C(=O)NC12CC1CN(C(=O)CCCCC1CC1)C2)c1ccccc1 C1(C(=O)NCC2(CNC(CC)=O)CCCC2)CCCCC1C1CC1 c1(C(=O)NC2(C)CN(C(CC3(CSC)CC3)=O)C2)ccnc(-n2cncn2)c1.CN CC1CN(C(C23CC(F)(C2)C3)=O)CC(CCNC(c2cc(Cl)cn2C)=O)O1 CC1(C)CC(NC(=O)CC2CCC(=O)NC2)CN(c2nnc(C(F)F)o2)C1 Cc1cnc(C(=O)NCc2ccc(C(=O)NC(C3CCOCC3)C)s2)cn1 N1(C(CCC#C)=O)CC(C(F)(F)F)OCC1CNC(=O)CCC(C)(C)C C1(C(N2CCC(SC)C2)=O)CN(C(C2CC3(CCC3=O)C2)=O)CC1(F)F C(=O)(C1CCCc2nncn21)NCCC(C)NC(C(C)NC(C1CCCC1)=O)=O N1(C(c2c(F)cc(C#C)c(F)c2)=O)CC2CCCC(C1)N2C(=O)CC1(C)CCC1 [N-]=[N+]=NC1(C(=O)NC23CCN(CC2)CC3)CCN(C(c2c[nH]c(=O)cn2)=O)C1 N1(C(=O)CC2COCCN2C(c2cccnc2)=O)CCc2ccsc2C1 N1(C(CNC(C(CC)(F)F)=O)=O)CC(C)OC(C)C1 C1(C(=O)NC(CC=C)C2CC2)CCCC(NC(C2CC(C)=NO2)=O)CC1 N1(C(C(C)NC(CC)=O)=O)CCCC(C(=O)NCC(=O)NCC(C)C)C1 N1(C(c2snc(C)c2N)=O)CC(F)(F)CC1C(C)(C)O.C1CCN1 c1(C(=O)NCCN(C(c2c(C)snn2)=O)C)ccnnc1NC1CC1 c1(-c2nc(C3C(C)CCC3)on2)ncnc2ncncc12 c1(CC(=O)NCC2N(C(c3cccc(OCC)c3)=O)CC2)ccc(C)c(F)c1 CCC1(C)CC(=O)N1.C1(NC(=O)OC)CC(=O)N(C)C1=O CC(c1ccsc1)=CC(=O)NCCN(C(=O)C=CCF)Cc1cccnc1 N1(C(=O)Nc2cn(-c3cccc(C)c3)nc2)CCCc2c(N(C)C)cccc21 C1(C=O)CCN(C(=O)C2=CCCC2)C12CCCC2.c1(CC=O)cnccn1 c1(CNC(=O)NC2C(OC(C)(C)C)CCCC2)cccc([N+](=O)[O-])c1 C1(C2CCN(C(c3nncs3)=O)CC2)(NC(=O)COCCF)CCC1 C(=O)(CC(C(F)(F)F)NC(c1cc(Cl)n(C)n1)=O)NCC1(CC)CC1 C1(OC)CCC2CN(C(=O)CCCCN(C(=O)CCCC3CCC3)C)CC12 c1(C(=O)NC(CNC(c2ncn(C(C)C)n2)=O)C)ccccc1F c1(CN(C)C(=O)OC(C)(C)C)ccc(C(=O)Nc2ccccc2C2CC2)cc1 C1(C(=O)NC(CNC(C2(CCN(C)C)CC2)=O)C(C)C)(CC)CCCO1 c1(C(=O)NC2CCCC(CNC(C3(CF)CCC3)=O)C2)cc(Cl)cnc1O Cc1c(C(=O)NC2COCC2NC(=O)C(C)(O)C2CCC2)ccn1C(C)C C(=O)(C(O)CCS(C)=O)NCC(=C)CCNC(c1cnn(C2COC2)c1)=O C(=O)(CC(C)CNC(c1cc[n+]([O-])cc1)=O)NCc1ccc(C)o1 C1(OC)CC(NC2(C)CCN(C(=O)OC(C)(C)C)C2)C12CCCO2 C1(CC)(CNC(C2CCN2C2CCCC2)=O)CCN(C(C2CC3CC3C2)=O)CC1 C1(CNC(c2cnc(C(=O)OC)s2)=O)CN(C(=O)C2=NOC(C)C2)CC12CCC2 c1(C(c2nnnn2C2CC2)(OC)NCC2(C)CCCS2)cc(C(F)(F)F)ncc1F Nc1ccc(CC(=O)NCC2(NC(C3CC3CC3CC3)=O)CC2)cc1 C1(CCNC(Cn2cc(C(C)O)nn2)=O)CSCCN1C(=O)CC1CCCOC1 CCC(C)(CC)C(=O)NCC12CC(CO1)N(C(c1cc(F)cnc1Cl)=O)C2 C=CCC(CC)C(=O)NCCOCCN(C(=O)Cc1cc(C)cc(C)c1)C C1(NCc2nccc(C)n2)CC(=O)N(c2cccc(C(C)C)c2)C1=O c1(SC)cccc(CNC(c2nnnn2C2CC2)c2ccno2)c1 CC(C(=O)NCCCNC(C1(CO)CCOC1)=O)C(=O)N1CCOCC1 C(CN(C)C)(CC(C)C)N(CC)CC.C123COC(C1)(C2)CNC(=O)C3 N1(C(C2(C)CCN(C)C2)=O)CC2(CC(CNC(c3ccc(Cl)cc3CO)=O)C2)C1 N1(C(c2c(C)cccc2)=O)CCC(O)(C2CCN(C(=O)C3=CCCC3)CC2)CC1 c1(C(N2CCC(O)(C(C)NC(C(C)N(CC)CC)=O)C2)=O)ccn2nccc2c1 N1(C(C(CC)N(C)C)=O)CCCC2(C1)CN(C(c1cccc3nnn(C)c13)=O)C2 c1(OC)ncnc(C(N2CCC(NC(C3(C#N)CCCC3)=O)C(C)C2)=O)c1F C1(NC(COCCOC)=O)CC12CCN(C(c1cnc(Br)o1)=O)CC2 C(=O)(C(F)CC(C)(C)C)N1CCC(C(N2C(COCC#C)CCC2)=O)(CC#C)C1 C(=O)(C(C)(C)C1=CCN(C(c2ccsn2)=O)C1)NCC(C)Cc1cn[nH]c1 c1(C(F)F)ccc(CCNCc2sc(-c3ccccc3)cc2Br)cc1 Cc1n[nH]c(=NCC(CNC(c2ccc(F)nc2)=O)C(F)(F)F)o1 N#Cc1ccc(C(=O)NCCC(O)CNC(=O)CCOCC2CC2)s1 C1(CNC(c2sc(CC)c(C)c2)=O)CC(C)(C)CN1C(C1CCCC(C)(C)C1)=O Cc1cc(NC(C2CC(F)CN(C(=O)Cc3cnc(C)s3)C2)=O)cc(Br)c1 CC(CC(=O)N(C)CC1CCCN(C(=O)C(CO)C(F)(F)F)C1)C(C)(C)C C1(CNC(C2CCCC2)=O)CCC(C2CC2)N1C(=O)CN1CCSCC1 c1(C(=O)NCC(C)N(C)C(C2CC(C)(C)CN2C)=O)nc[nH]c2ncnc1-2 C1(NC(=O)Nc2cccc(O)c2)CCCN(C(c2cnccn2)=O)C1 N1(C(c2n(CC)nc(C)c2)=O)CCOCC(CNC(=O)CN2CCC(C)CC2)C1 Cc1cnc(C(=O)NC2C3CC2CN(C(=O)CCc2nc(=N)[nH][nH]2)C3)cc1C c1(C(=O)NCCCNC(c2ccnc3cc[nH]c23)=O)csc2c(F)cc(F)cc12 Cc1nc(F)ccc1-c1cc(C(=O)Nc2nccnc2C)ccn1 c1(CC)cc(NC(=O)C(C)(C)CCNC(=O)CN2CCCC2C)cc(O)c1 N1(C(CCC#C)=O)CCC2(CC2C(=O)NC(CN(C)C)C(C)(C)C)C1 C(=O)(C(O)C1=CCCCC1)NC(C(NOCC(=O)OC)=O)C1CCC1 O=S1(=O)C=Cc2ccc(NS(=O)(=O)c3cnn(C4CCOC4)c3)cc21 C1(C(C)(C)C)CCCCN1C(C1(NC(=O)CC2(O)CCCCC2)CCC1)=O C=CCC(C(=O)NCc1cc[nH]c1C(=O)NCC(C)CCC)C(C)C C1(NC(C=C(C)C(F)F)=O)C2CC3CN(C(C4CN(C(C)C)CCO4)=O)C1C3C2 n1(C(CC)CC)ccc(C(=O)NCCC2CCN(C(c3cn(C)cn3)=O)C2)n1 N1(C(C(C(C)(C)C)CNC(C2(Cl)CC2(F)F)=O)=O)CCN2C(=O)OCC2C1 c1(N(C(C2(C)CCCN(C(C=CC(C)=O)=O)C2)=O)CC#N)ccc2oc(C)nc2c1 N1(C(C2(F)C(C)C2)=O)CCOCC(CNC(c2ncc(C(N)=O)cc2Cl)=O)C1 CC1(C)CN(C(=O)C2=COCC2)CC1CNC(=O)C=Cc1cnccn1 S(=O)(=O)(c1ccc(NCCOC)c2cnccc12)NC1C(CC)OCCC1 CC1CCC(CN)N(Cc2cccc(C(=O)NC(=O)OC(C)C)c2)C1 c1(C(N2CCC(NC(c3nc(C)oc3)=O)C2)=O)cnc2ccoc2c1 Cc1ccc(C(=O)NC(CO)C(C)NC(=O)Cn2cc(C3CCC3)nn2)cc1 C(=O)(C(C)(CCC)CCC)N1CCC(OCC(=O)NC(CC#C)CO)C1 N1(C(c2cccc(C(=O)NC)c2)=O)CC2CN(C(C3(C(N)=O)CCC3)=O)CC2C1 Cc1cnc(N2CC(NC(C3CCc4nncn4C3)=O)C(C)C2)nc1S(C)(=O)=O Cn1ccc(C=CC(N2C(C(=O)NCCC(=O)NC3CC3)CCC2C2CC2)=O)c1 c1(C(N(CC(CC)NC(=O)CC2CCCOC2)C)=O)ccc2cnccc2c1 C1(C(=O)NCCCCCN(C(c2cc(OC)no2)=O)C)CNC(=O)C(C)(C)C1 c1(OCC)ncc(C(=O)NC2CN(C(=O)C=C3CCC3)CC2C)cn1 C1(NC(=O)Cc2csc(C(F)(F)F)n2)COCCN(C(=O)C(F)(F)C2CC2)C1 c1(CSCC(=O)NC(Cc2ccccc2)C2CC2)nc(-c2nc[nH]n2)no1 C(CCC(=O)NC1(CCNC(=O)C(C)NC(C)=O)CCCC1)OCC C1(NC(COCCCC#C)=O)CCC(NC(c2cc(COC)cs2)=O)C1 C1(C2(O)CN(C(=O)C(CO)C(C)C)C2)(CNC(c2c(C)ccc(N)c2)=O)CC1 c12ccc(cc1)COC2=O.c1(CC(=O)NCC)ccc(OCCO)cc1 C1(C(=O)NC2C(NC(C3(C=C)CCC3)=O)CCOC2)CCc2nc(C)[nH]c2C1 c1(C(=O)NC(CNC(C(C=C)O)=O)C2CCC2)cccc(C(F)(F)F)c1 C(=O)(C(O)CCC(C)C)NCC(Cn1cc(C(c2cccnc2)O)nn1)OC C1(CNC(CNC(C)=O)=O)CC2(CCN(C(=O)C=C(C)c3cnn(C)c3)C2)CO1 Cc1noc2nc(C(F)(F)F)cc(C(=O)NCC(C)NC(C3C4CCCC34)=O)c12 c1(COCc2sccn2)nc(CC2CCOCC2)n(-c2ccnc(O)c2)n1 c1(C(=O)NC2(C)CC(NC(CCNC(=O)NC)=O)C2)cnc2c(cnn2C)c1 c1(OC)ccc2cc(C(=O)NC3CN(C(C4(CO)CCC4)=O)CCC3O)[nH]c2c1 c1(NC)cc(C(=O)N(CCCNC(=O)C(C)C(F)F)CCO)cc(Cl)n1 c1(C(N)=O)nccnc1C(=O)NCCOCCCNC(=O)CC1CSCCS1 C(=O)(C(C)(C)CC#N)N1CCC(N2CCN(C(C3(CCC=C)CC3)=O)CC2)CC1 c1(C(N(CC(C)N(C(=O)C(O)C(F)(F)F)C)C)=O)cc(O)nc2cc(F)ccc12 Cc1ccc(-n2cc(CCCNC(c3cc(CC(C)C)on3)=O)nn2)nc1 c1(CC)cc(C(=O)NC2CC3CC2N(C(C24COC(COC)(C2)C4)=O)C3)cc(O)n1 C1(C2CCN(C(c3ccn(CCF)n3)=O)CC2)(NC(C2CC(OC)C2)=O)CCC1 N#CCCCCC(=O)NCCNC(=O)CCC(=O)NCCNCc1ccccc1 C1(NC(C2(C)CC=CCC2)=O)CCN(C(c2ccc(O)c(N)n2)=O)CC1F C1(C(N2CC(CN(C)CCO)C2)=O)CCCC(F)(F)C1.C12(CC1)C(=O)N2 CCCC(C)(CCC)C(=O)NC(CC1CC1)C(=O)N(C)Cc1cccc(O)c1 N1(C(c2c(OCC=C)cccn2)=O)CCCCC(NC(=O)CCCC(=O)OC)C1 N1(C(C=Cc2cn(C)nn2)=O)CCC(C2CCCN(C(c3ccoc3)=O)C2)CC1 C1(C(C)C)CC(C(=O)N(C)Cc2cn(-c3ccccc3Cl)nn2)CCO1 c1(C(=O)NCCN(C(=O)CC2(COC)CC2)CC)ccc(C(C)C)nc1C N1(c2nc(C)cc(OC)n2)CC(NC(=O)CN2CCCCCC2)C2CCCCC12 C(=O)(CCOC1CN(C(=O)Cc2ccsc2)C1)NCC(C)NC1CC1 C1(C)(CC)C=C(C(=O)N2CCC(CC(=O)NCC(F)(F)C(F)F)CC2)C1 c1(NC(CNC(C=Cc2n(CC)ncc2)=O)C)c(F)cc(C#N)cc1[N+](=O)[O-] c1(C(N(C)CCN2CCN(C(C3CC3CF)=O)CC2)=O)c(F)cccc1Br N1(C(Cc2cccc(C)c2)=O)CCCC2(CCN(C(C3CC4(CCC4)C3)=O)C2)C1 N1(C(C2CCC3(CC3)N2C(C2CC(O)C(F)C2)=O)=O)CC=CC12CCOCC2 C12OCCC1CNC2=O.C1(CNC(C2(C(=O)OCC)CC2)=O)CCC1CC C1(NC(c2c(CC)oc(C)c2)=O)CCN(C(=O)CC2CSCCO2)CC1(C)C C1(CC)CCN(C(=O)CC2CC(C)=NO2)C1CNC(=O)Cc1cnc(C)s1 c1(OCC=C)cccc(CN2CC(NC(c3ccc(CO)o3)=O)C(F)C2)c1 c12ncc(s1)COC(=O)C1(CC=CC1)NC2=O.C(C)(C)(C)O.CC n1(Cc2cc(C)on2)nnc(NC(=O)CCC2CCC(C(N)=O)O2)c1C c1(C(N2C(C(=O)O)CSC2c2ccncc2)=O)sc2sccc2c1Cl N1(c2cnc(CSCC)c(Cl)c2)CCn2nc(C(F)OCCOCCOC)cc2C1 Cc1nc(CC(C)C)oc1C(=O)N(C(C)CCNC(=O)CNC(N)=O)C N1(C(C2ON=C(C)C2)=O)CC2CC1CN(C(c1c(C)ccc(F)c1O)=O)C2 C(=O)(CN=c1ccc(Cl)n[nH]1)N1C2CN(C(C3CCCC4(CCC4)O3)=O)CC1CC2 N1(C(CNC(C2C(C)C2)=O)=O)CC(NC(=O)C2=NOCC2)C(N=[N+]=[N-])C1 C1(NC(Cc2cc(OC)ncc2)=O)CCCCCN(C(c2cc(C)nn2C)=O)C1 C1(C(N(c2cccc(C)c2)C)=O)CN(C(C2C3CCCCC23)=O)CC(C)O1 C1(C#N)(C(N(CCCN(C(=O)C(C)(C)c2cnco2)C)C)=O)CC2CCC1CC2 c1(SC)cccc(CC(N2CCCC(Cc3cnc(C(C)C)nc3)C2)=O)c1 c1(OC)ccc(C)cc1C=CC(=O)N(C(C)CCNC(C1CCC(=O)NC1)=O)C C12(C(=O)NCC3CN(C(CC4CC(C)C4)=O)CC3O)CCC(C)(CC1)OC2(C)C CCCCC(O)CC(=O)NCCN1CCCN(C(c2cc3scnc3[nH]2)=O)CC1 CC1CCC(S(=O)(=O)NC(c2cccc(F)c2)c2nccn2C)C1 c1(OC)cc(C(N2CCCC(NC(C3CC(C)CO3)=O)C2C)=O)ccc1C CN1CCC(C#N)(C(N2CCC(CCNC(=O)C=C3CCOCC3)C2)=O)CC1 C1(C(=O)NCc2cccc(C(N(C3CCCC3)CC#C)=O)n2)CC2CC1CC2=O c1(CC(C)C)c[nH]c(C(=O)NC2COCC2n2cc(C3(C(=O)O)CC3)nn2)c1 c1(CCC)cc(NCC)ccc1O.C1(CC(F)F)CCC1 CCC(C)(C)C(O)C(=O)NCC1(CNC(c2cc(CO)[nH]n2)=O)CC(F)(F)C1 CC(CC(=O)NC(CNC(=O)COc1c(F)cccc1F)C1CC1)CC(F)(F)F Cc1ccc(SCC(=O)NC2CCC(N(C)C(c3c[nH]c(Br)c3)=O)C2)cc1 C(=O)(C#CC1CCOC1)N1CCN(C(COCC)=O)CC1COC N1(C(CC)=O)Cc2ccccc2C(CNC(c2cnc(O)n2C)=O)C1 N1(C(CCC(C)NC(C(CCC)C#N)=O)=O)CCCC12CCOCC2 C1(CCNC(c2cnc(C(C)C)[nH]2)=O)CN(C(c2cc(CO)[nH]n2)=O)CC(C)O1 N1(C(C(N=S(C)(C)=O)=O)=O)CCC(C2CCN(C(=O)C3=CCCCC3)C2)C1 C1(C(=O)Nc2ccc(C#C)cc2)CCCCCCN1C(=O)CN1CSCC1=O N1(C(c2c(C(C)=O)cccc2)=O)CCOC(C)(CNC(=O)CCn2cnnn2)C1 C=CCCC(F)(F)C(=O)NC(CCC)CCCNC(c1[nH]nnc1C1CC1)=O c1(C(=O)NC(CNC(c2[nH]nc(OC)c2Cl)=O)C)ccc(C)c(F)c1Br c1(C(=O)Nc2cccc(NC(C3(SC)CCC3)=O)c2)nccc2c(C)cccc12 N1(S(CC)(=O)=O)CC(C(=O)NCc2ccccc2F)Oc2ccccc21 c1(C(=O)NC(C)CN(C)C(C2C3(CC3)C23CC3)=O)cc([N+](=O)[O-])cc(Cl)c1Cl N1(C(CCCOC)=O)CCN(C(=O)CCOCC2CCC2)C(CC(F)F)C1 c1(OCC(=O)N(CC(C)NC(CSCC#C)=O)CC)ccc(F)nc1 C1(CC(=O)NC2CCN(C(C3CC(Cl)(Cl)C3)=O)C2)COC(C(F)(F)F)C1 C1(CNC(C(CC)OC2CCCCC2)=O)CC2CCCCC2N1C(=O)CCOC C12(CC(=O)N(C3CCCN(C(=O)CS(=O)(=O)N(C)C)C3)C)CC3CC(CC(C3)C1)C2 Cn1cc(CCC(=O)NCC2(O)CN(C(C3CCC(=O)O3)=O)C2)cn1 c1(C(N2C(CCNC(C3COC4COCC34)=O)CCCC2)=O)cc2c(s1)CCC2 CCC(C)(CCNC(=O)C(C1CCCCC1)F)NC(=O)C1CC1 N1(C(c2cn(C)nc2O)=O)CCN(C(=O)CCc2cccnc2)CC1C1CCC1 c1(C(=O)NCCOC2CN(C(C3(C)CCOCC3)=O)C2)cnn2c1OCC(F)C2 c1(-c2nc(C(C)OCC)nn2CC)cc(C(F)F)ccc1F C1(C(=O)NC(C2(O)CCN(C(c3cnc(N)cn3)=O)C2)C)Cc2ccccc2O1 C1(C(C(=O)N(CCCCN(C(C(c2cnccn2)C)=O)C)C)F)CCCCC1 CCCC(CNC(c1c(C)ccn1C)=O)C(=O)NC(C)CC(C)(C)OC c1(C(=O)NCC2CC(C)N(c3ccccc3)C2)cnc(N)c(N)c1 O=C(CC1CCc2ccccc21)NC1(CNC(C2CC2C2CCCC2)=O)CC1 c1(CC(=O)NC2(CNC(C3CC(F)C(=O)N3)=O)CC2)c(F)cncc1Cl C1(C(=O)NCC(CCNC(=O)Cc2cc[nH]n2)O)CC(c2ccccc2)=NO1 N1(C(C(=O)NCC(F)(F)F)=O)CC2CN(C(C3CCC(F)CC3)=O)CC2C1 N1(C(CC(CC)C2CC2)=O)CCN(C(c2csc(C(C)(C)C)n2)=O)CC1C(F)F C(=O)(CCC(C)(C)F)NCC(C)NC(=O)C(c1ccccc1)N(C)C c1(C(N2CC(CNC(c3n(OC)cnc3C)=O)OCC2)=O)cnc2[nH]cnc2c1 Cc1cn(CC(N2CCN(C(c3cccc(C4CC4)c3)=O)CC2)=O)c(=O)nc1O C(=O)(C1=CCSC1)N(C)CCNC(=O)CNC(N1CCCCC1)=O C1(N(C(=O)CCc2cnco2)CC)CCCN(C(=O)C(c2cccnc2)O)C1 Cc1nn(C)c(C(=O)NC2COC3C(NC(C4CSCCS4)=O)COC23)c1Cl CC1CN(C(=O)CCc2nccs2)CC(C)N(C(c2ccc(C3CC3)nc2)=O)C1 C(=O)(C(C)(C)CC(=O)N1CCC(CN(C)C(c2nccc(F)c2Cl)=O)C1)OC c1(C(N(C)CCNC(=O)C(=Cc2ccccc2)C#N)=O)nnc(O)cc1O c1(OC)cccc(CC(N2CCCC2CN(C)C(c2cc(N)ccn2)=O)=O)c1 C(C(=O)N1CCC(C(N2CC3CC3(CO)C2)=O)(CO)C1)(C(C)C)SCC c1(C(=O)NCC(CNC(COC)=O)F)cnc(NC(=O)OC(C)(C)C)cn1 N1(C(C=C(C)C2CC2)=O)CCOC(CCNC(C2CCN(C)C2)=O)C1 N1(C(C2CC(Cl)(Cl)C2)=O)CCc2ccc3ccccc3c2C1 N12CCOCC1CC2=O.C1(CNC(=O)CC2CSC2)C=CCOC1 C=CCC(CN)C(=O)N(c1ccc(-c2cncnc2)cc1)C C(=O)(C(F)C(C)C(F)(F)F)N(CCNC(c1cncc(Br)c1)=O)CC c1(C(=O)NCCCOCCNC(=O)CC2C=CCC2)csc(N2CCCC2=O)n1 C12(C(=O)NC(Cc3ccc(OC)c(O)c3)C)CCCCC1(C(=O)O)CC2 CCC(C)CCCC(=O)N1CCOCC1CNC(=O)CCCC(N)=O CCCC(CC(C)C)C(=O)NC1CCCCC1NC(c1ccncc1C1CC1)=O C(=O)(C1c2c(Br)cnn2CCN1C(=O)Cc1nc(C)c(C)[nH]1)OC C#Cc1cncc(C(=O)NC(C)C(C2CC2)NC(=O)CCc2ccccc2)c1 C1(C(=O)NCCCN(C(c2c(Cl)cc(C)s2)=O)C)Cc2nn[nH]c2C(C)C1 C(=O)(CC(C)(C)C#N)NC(C)CNC(=O)Cc1ccc(F)cc1 C(=O)(N(O)Cc1ccccn1)NC(c1ccccc1)C c1(OCC)ccc(CN2CC3C(C2)N3C(c2cc(Cl)cc(I)c2)=O)c([N+](=O)[O-])c1 CC(C)(O)C(F)C(=O)NCC(O)CC(=O)NCC(O)CNC(N)=O C1(CNC(C2CCS2(=O)=O)=O)CCC(Nc2nccc(C(F)F)n2)CC1 CC1CC(CC(N2CC(CO)C(O)C2)=O)CN1C(=O)C(N)=O Cc1ncc(C(=O)NCC2(F)CCN(C(=O)CN3CC(=O)NC3=O)C2)n1C c1(C(N(CC(O)CN(C)C(C2CCOC2)=O)C)=O)cn(C)c(=O)c2cncn12 CC1CC(C(=O)N(C)Cc2ccncc2F)CN(C(C2C=CCS2)=O)C1 OCC1(c2ccccc2)CCCN(CC2NC(=O)N(Cc3ccccc3)C2=O)C1 C(C(CO)(CO)NC(=O)C=CC=Cc1ccccc1)N(C)C(C1CCC2CC12)=O C1(NC(c2c(C)n(C)nc2)=O)CC1C1CCN(C(C2CCOC(=O)N2)=O)CC1 c1(NC)ccc(F)cc1C(=O)NC(CNC(=O)C(C)=C1CCC1)C(C)C N1(C(c2occ(C)c2C)=O)CCCC(CNC(c2cccc(C(N)=O)n2)=O)CC1 c1(C(=O)NCC2CN(C(C3(CC(C)=O)CC3)=O)CC2C)cc(F)c(F)cc1F C(CC(C(C)C)NC(C1CC1c1cccs1)=O)N(C(c1c(C)snn1)=O)C C(=O)(C(=O)CC(C)C)NC(CCOCC)C(=O)NC1CCCC1C(C)C c1(C(=O)NCCC2(CNC(C3C(CC)C3)=O)CC2)cc2n(n1)CCCC2O CCCCC(O)C(C)C(=O)NC1(CCC)CCN(C(=O)CC2(O)CCC2)CC1 N1(C(C2(OCC)CCOCC2)=O)CC2CN(C(c3cncc(O)c3)=O)CC2(C)C1 Cc1cc(C(N2CC(CC(C)NC(c3cc(CO)[nH]n3)=O)C2)=O)c(F)cc1Cl C(CCCC(=O)N(CCCN(C)C(c1scnc1C)=O)C)OCC c1(CN2CCC(CNC(C(CCC)OCC)=O)C2)ccc(Cl)nc1C c1(C(N(CCN(C(C23C(C)OC(CC2)C3)=O)C)C)=O)ccc2cccc(F)c2n1 CCCCC(CNC(=O)C(CC1CC1)NC(=O)NC(C)C)CC C1(NC(=O)CC2(O)CCC2)CCC(O)CN(C(C2OCCOC23CCC3)=O)C1 N1(C(c2nn(CC)c(C)c2)=O)CC(NC(C2CCOC(=O)N2)=O)CC1(C)CC Cc1nc(C)c(C(=O)NCCN(C)C(c2cc([N+](=O)[O-])c[nH]2)=O)c(C)n1 N1(C(C(C(C)C)CO)=O)CC(C)OC2(CCN(C(=O)CC3CC(C)(C)CO3)C2)C1 C1(C(=O)NCC(C(=O)OC)C)CCC2CCC1CN2C(=O)CCC=C(C)C c1(C(N2CCC(N(C(CCC(=C)Br)=O)C)C2)=O)cc(-n2ccnn2)ccc1F C1(C(N(c2ncccc2Br)C)=O)CC[Si]2(CCCC2)CC1 c1(OCC)ccc(Cl)nc1C(=O)NC1CCCN(C(C23CC(OC)C2C3)=O)C1C N1(C(C)=O)CC2CCC(NC(=O)C=Cc3ccc(-c4cccc(Cl)c4)s3)C2C1 c1(OC)ccc2c(CCNC(N3CCCC3c3nc(C)no3)=O)c[nH]c2c1 C1(C(=O)NC2(C)CC(F)(F)C2)CC(NC(C2CC2(F)Cl)=O)C12CCC2 N1(C(C2(NC(C)=O)CCC2)=O)CCC(CCC(C)(C)NC(=O)C(O)C(C)C)CC1 C(CNC(c1ccncc1OC(C)C)=O)(CC(F)(F)F)NC(C(C)OC)=O c1(C(=O)NC(C2CN(C(C3(F)CCOC3)=O)C2)C)cc(-n2cnnc2)ccn1 c1(C(C)NC(C=CCN(C(COCCC#C)=O)C)=O)ncc[nH]1 C1(CCC(=O)N(CC(C)O)CC(C)O)CCCN(C(c2cn[nH]c2)=O)C1 Cn1ncc2ncc(C(N3CC(CO)(NC(=O)CCc4ccccc4)C3)=O)cc12 C1(C(N(CCCNC(C2C(CCC)C2)=O)C2CC2)=O)CS(=O)(=O)CC(=O)N1 CCC(O)C(C)(C)C(=O)N1CCC1CNC(=O)CCc1c(C(=O)OC)c(C)[nH]c1 N1(C(CCC(=O)N(C)C)=O)CCC(NC(c2ccc(C3CC3)cc2F)=O)C(F)C1 N1(C(CN(C(COC)=O)C)=O)CC(CNC(C2CC(C)=NO2)=O)CC1(C)C C#CCCCCCC(=O)NC1CCC1CNC(=O)Cc1cnccc1OC C1(NC(C2(NC(C)=O)CCCCC2)=O)CC2CN(C(c3cc[nH]c3)=O)CC12 C(N=c1nc(NC2COc3cc(F)ccc32)c2c([nH]1)CSC2)c1cccc(C)n1 S(=O)(=O)(C(F)(F)F)NCCC(=O)NC1CN(C(=O)CC(F)(F)F)CCO1 C(c1ccc(F)cc1F)=CC(=O)N(CCCNC(=O)CC1CC1(C)C)C(C)C c1(C(c2nnnn2C2CC2)NCC(=O)OC)ccc(F)cc1.CC(F)(F)F c1(C(=O)NC(CC=C)CNC(=O)Cc2ncc(C)s2)cc(F)cc2cc[nH]c12 c1(OC)c(C(=O)NC2CC(CC(=O)Nc3cccnc3C(C)C)C2)cnn1C c1(CC(=O)NC2CC(F)(CNC(C(C)=C3CCC3)=O)C2)ccc(C)c(Cl)c1 C1(NC(c2ccc3ccoc3c2)=O)CC2CC1CN(C(=O)C=CCO)C2 C1(=CC(=O)NC(C2CN(C(CCCC)=O)C2)C)CN2CCC1CC2 c1(OCC(N2CC(C)C(NC(=O)CC3CC4(CCC4)C3)C2)=O)ccc(Cl)cc1Cl N1(C(=O)NC2CCC(C(N)=O)C2)CC2(CCC2)C12CCC2 C1(C(=O)NC(C)(C)C(F)F)C2CCCC2CN1C(=O)COC(C)(C)C C(=O)(CP(C)(C)=O)NCCN(CCOC)C(c1cnc(COC)nc1)=O C=CCCCCCC(=O)N1CC(NC(c2ccnc(C)c2)=O)CC1(C)CC C1(C)(C(N2CC(OC)(CNC(=O)C(C)CCN(C)C)C2)=O)C(C)(C)C1(C)C CC1(C)CCCN(C(=O)Cc2ccccc2Cl)C1CNC(c1ccccc1Br)=O c1(CN(c2ccccc2)C(C2C(C)(C(F)F)C2)=O)cn2c(n1)CCCC2 Cc1c(NC(C2CCCN(C(=O)C(C)CO)C2)=O)cccc1[N+](=O)[O-] CC1=NOC2(C1)CC(C(=O)NC(C1CN(C(C3C=C3C)=O)CCO1)C)C2 C1(C(=O)OC)C2CCC(C2)C1N(C)C(c1ncccc1N(C)C)=O C(CS(=O)(=O)c1ccc(F)cc1)NC(C(C(=O)OCC)OC)=O C1(C2CCN(C(CCCC)=O)C2)CCCCN1C(=O)COC(C)(C)CC N1(C(C2(OCC)CCOCC2)=O)CC2(CNC(C3CC(C)CO3)=O)CCC1CC2 N1(C(c2n[nH]c(C)c2N)=O)CC2CC(NC(=O)CC3CCSCC3)C2C1 C(=O)(CCCC(=O)NCCC1CCCN(C(=O)Cc2nc(C)sc2C)C1)OCC C1(C(N2CC(NC(CCc3n(C)ccn3)=O)(CO)C2)=O)C(C2CC2)C1(F)F c1(N2CCCC(COC(C)=O)CC2)nc(Cl)nc2c(F)c(Br)c(Cl)cc12 C1(c2cn(Cc3cncc(OC)c3)nn2)CCN(C(=O)CC(C)N(C)C)C(C)C1 C(N=c1ccnc(-c2ccccn2)[nH]1)C1CC(NC(C=C(C)C2CC2)=O)C1 C1(C)(C(C)C)CCN(C(=O)CONC(=O)CN2CCN(C)CC2)CC1 CC(CC(=O)N1CCC2C(NC(C34CC(CC(F)F)(C3)C4)=O)CC12)P(C)(C)=O N1(CC(=O)NCCN(C(=O)C(F)CC2CCOC2)C)CCOCC1 N1(C(c2cncc(OCC)c2)=O)CC(NC(C=CC(=O)OCC)=O)C(C)(C)C1 Cc1c(NC(C)C(C)C(=O)O)cnn1C c1(CC)nc(C(=O)NC2CC(NC(c3cnc(OCC(F)F)cn3)=O)C2)c(C)o1 C(=O)(C(CC)CCOC)N(CC(CC)NC(=O)CCc1ccc(O)c(Cl)c1)C C#CC1(C(=O)NC(C)CN(C(=O)C(CCSC)OC)CC)CCCC1 C(=O)(CC(C=C)CCC)N1CCC(C(C(=O)NCCSCC#C)C)CC1 CCC(CO)C(=O)NCC(C1CC1)N(C)C(c1ccnn1CCOC)=O CN1CCN(C2CN(CC(N3CCCCC3CC(=O)NC3CC3)=O)C2)CC1 c1(C(=O)NC2C(C)CCN(C(=O)CCc3cccs3)C2)ccc(F)c(C#N)c1 C(C)(C)(CC(F)C(=O)N(CC(=O)NC(C)(C)C)C)NC(CCC(=O)NCCC)=O C1(NC(C23CC(c4ccc(F)cc4)(C2)C3)=O)CCCC12CCN(CC#N)C2 c1(CC)nc(C)[nH]c1C(=O)NC(C)CN(C(=O)CC1CCCO1)C C1(C(N2CC(NC(c3n(CC)ccn3)=O)C(C)C2)=O)CCc2ncnc(C)c2C1 C1(CC=C)(NC(=O)CCCCCO)CCCN(C(=O)Cc2ncccc2C)C1 n1(CCC(=O)NC2CCC(C(N3CCC(CF)CC3)=O)C2)cnc2ccccc12 N1(C(CN2C(C)CCC2C)=O)CCN(C(=O)C=Cc2cccc(CO)c2)CC1C CC1(C)OCC2CC12C(N1CCCCC1CNC(C1(n2cncn2)CC1)=O)=O C(=O)(C(C)C(C)C1CCC1)NCC1(F)CC(NC(CCOC)=O)C1 N1(C(c2nccc(N(C)C)c2)=O)CC2CCC1CN2C(C1(F)CC2(CCC2)C1)=O N1(C(CC(C)SC)=O)CCC(C)(C)C(CNC(c2n[nH]c3c2CCOC3)=O)C1 C1(NC(C2C(C(=O)OCC)C2)=O)CC2CCC1CN(C(C1CC(C)(CC)C1)=O)C2 c1(OC)ccc2[nH]c(=NC(C)CCSC)[nH]c(=NC3C=CCC3)c2c1 Cn1cc(C#N)cc1C(=O)NCc1nc(C(=O)NCCCC(C)(F)F)co1 C(N=c1[nH]nc(CC(C)C)s1)C1OCCN(C(C(=Cc2cn[nH]c2)C)=O)C1 N(C1CCCc2ccc(O)cc21)CC1(C)CN(C)C(=O)CC1 Cc1cn(C)cc1C(=O)NCCC1CC(NC(=O)Cc2ccccc2CC#N)C1 c1(NC(C2CC3(CC3)CN2CC2CN3CCC2CC3)=O)ccc([N+](=O)[O-])c(Cl)c1 C1(NC(C(CC)CCOC)=O)CN(C(C2(C)CC(C)(C)C2)=O)CC2(CCC2)C1 C(=O)(C(O)CCCNC(C1(O)CC1)=O)NC1CCN(CCC)C1 CC1CC(=O)NCCN1C(c1cc(CNC(=O)CC2CCCN2C)on1)=O CC(C)CS(=O)(=O)CCC(=O)N1CCCCC1CNC(=O)CC1CCCOCC1 N1(C(c2nc(C)[nH]n2)=O)CC(NC(=O)C=Cc2cscn2)C(CC(C)(C)C)C1 c1(C(=O)NC2C(NC(c3cnc(C)o3)=O)C2)c(C)nn(C)c1C(F)(F)F C1(CN(C(c2n(CCC)ccn2)C(=O)NC2COC2)C)CCC(CNC)CC1 C1(NC(C(C)N(C)C)=O)CCCC(CNC(=O)CN2CCS(=O)CC2)C1 C(C(C)(C)CCNC(c1ccc(C)n1C)=O)NC(C1(CC)CCC1)=O c1(CC(C)NCC2(CC)CC=CCC2)ccc(OC)c(OC)c1OC CC(=O)CCCC(=O)N1CCN(C(c2ccnnc2O)=O)CC1CC(C)(C)C c1(-c2c(F)ccc(NC(c3c(OC)ccc(C)c3)=O)n2)ccc2occc2c1 N(C1COc2c1ccc(Cl)c2Cl)C(=O)NCCN1CC(C)NCC1 C12(NC(c3c(OC)ncc(Cl)c3)=O)CCCCC1N(C(=O)CCC(F)(F)F)CC2 C1(N(C(c2n(C)ncc2)=O)CCO)CCN(C(c2cnc(C(N)=O)cn2)=O)CC1 C(=O)(C(C(=O)N1CCCC(CN(C)C(C2(CO)CC2)=O)C1)C(C)(C)C)OCC c1(N(C)C)cnc(Br)cc1SCC(F)(F)F.N12CC(F)CC1CNCC2=O N1(C(c2cnc(C)o2)=O)CCOC(CN(C)C(c2ccn(C3CC3(F)F)n2)=O)C1 c1(C(=O)NCC(CNC(c2c(C)snn2)=O)CO)ccc2c(c1)CC(=O)NC2 N1(C(C=CC(CC)C)=O)CC(NC(=O)CC(C)(C)C)CC12CCOCC2 C1(CNC(CC(C=C)C)=O)Cc2ccccc2CN1C(c1cc(F)cnc1O)=O c1(C(N2CCC(N(C(C(c3ccc(C)cc3)C)=O)CCO)C2)=O)c(C)nn(C)c1Cl C(=O)(CC1=CCCCC1)NC(C)CC(=O)NC(c1c(O)cccc1F)C N1(C(c2c(C)csc2Cl)=O)CC(C2CCCN(C(c3ccc(Cl)[nH]3)=O)C2)C1 C1(C(=O)N(C)CCOC)(CC)CCNC1=O.C1(=O)C(OC)CNCCN1C C1(S(=O)(=O)N(C(C(C)C)C2CCC2)Cc2ccccc2)(CC)CC1 c1(C(N2C(CNC(=O)CCC3CCCO3)CCC2)=O)ccncc1Cl c1(C(C2CC2c2ccccc2)=O)ccc2ncccc2c1.N12CCOC(C1)C2 Cc1cc(C(=O)NC(C2CN(C(=O)C(C)OCCC(C)C)C2)C)cc(C)c1 c1(C(=O)NCCN(C(C(C(C)C)(C)O)=O)C)cc(O)nc2c1CCCC2 c1(C(c2ccccc2)OC(C2(NC(=O)OC(C)(C)C)COC2)=O)ccc(O)nn1 c1(C(N2CCOCC(CNC(CCOC(C)C)=O)C2)=O)cc2ccncc2[nH]1 c1(C(=O)NC(CNC(C(C)(C2CC2)OC)=O)(C)CC(C)C)cc2c[nH]cnc-2n1 N1(C(C(C=C)O)=O)CCC(NC(=O)CN2CCCCC2)C12CCCC2 C1(C(C)C)CCN(S(=O)(=O)NC(C2(C(F)(F)F)CCCCCC2)=O)CC1 c1(C(=O)NC2CC(C(=O)N(c3nn[nH]n3)C3CC3)C2)cc2c(C3CCCC3)cccc2[nH]1 c1(CC)cc(C(N2CCC(CC(=O)N(CC(O)CO)C(C)C)C2)=O)n(C)n1 C(=O)(CCCC(=O)NCC(C1CC1)NC(=O)CCc1ccc(Cl)s1)NCC c1(SC(C)C(=O)NCC(C)(C)CN(C(=O)CC#N)C)ccc(F)c(F)c1 c1(C(=O)NC(CC(C)NC(c2cc(CCOC)on2)=O)C)cnc2n1CCOC2 C1(CC(=O)N(CC=C)CC)CCCN(C(=O)CCC2CCCN2C)C1 C1(NC(CS(C)(=O)=O)=O)C2CC3C(C2)C13C(N1CCNC(=O)C1CCO)=O C1(C(=O)NCC2(O)CCN(C(=O)C(=Cc3cnc[nH]3)C)C2)(CC)CCOCC1 C1(N(C)C(C2CCC2F)=O)CCN(C(=O)CCNC(c2ccsc2)=O)CC1 C(=O)(CN=S(C)(C)=O)NCC(C)(CO)NC(C1CC1c1ccccc1F)=O C(=O)(C(CC(C)C)C(C)C)N1CC(OC)(CNC(=O)Cc2cccn2C)C1 C(=O)(CCCC(C)C)NC1CCN(C(C(C)OCc2cccc(C)c2)=O)C1 c1(C(CCC)NC(C2CN(C(=O)CC)C2)=O)cc2c(s1)CCC2 c1(OC)ccc(OC)c(CNC(N2CCCC2C(C)O)=O)c1 c1(OCC(=O)N(C2CCC(NC(=O)CC3(C)CC3(F)Cl)CC2)C)ccc(F)cc1 c1(SCC(n2cccn2)C)cc(C(=O)Cc2ccccc2)cn1C CC1CC=CCC1NC(=O)C(C1(O)CCC1)NC(=O)C=CC(F)(F)F CCCCCCC(C)C(=O)C(C(CCSC)NC(CC(CN(C)C)N)=O)=O.OC C1(NC(N2CCCC(CC(=O)NC3(C(C)C)CCC3)C2)=O)CCC(=O)NC1=O c1(C(=O)NC2C(CNC(c3cnc(C(=O)OC)s3)=O)C2)ccc(C)cn1 CCC(CC(=O)NC1CN(C(C2CCC=CCCC2)=O)C2(CCC2)C1)CC(C)C c1(OC)ncc(Cl)cc1C(=O)NCC(C)CNC(C1CC(N2CCOCC2)C1)=O C1(C)(NC(CSCCCC)=O)CCCN(C(c2nc(Br)c(C)s2)=O)C1 C12(NC(c3cnc(SC)n3C)=O)CC3CCC(C1C2)N3C(C1(C)CCC1)=O Cc1cn2cccc(C(=O)NC(C)CC(C)NC(=O)C(C)CC3CCCC3)c2n1 c1(COCC(=O)NC(C(C)=O)C)ccccn1 c1(C(=O)NCCNC(c2c(C)noc2C)=O)ccc2c(ccn2C)c1 c1(C(=O)NC(CC(C)C)C(=O)O)cn2c(n1)CCN(CCC(=O)NCC(=O)O)CC2 N1(C(c2scc(C(N)=O)c2)=O)CCC(CNC(=O)C(F)=CCCF)CC1 Cc1scc(C(N2CCN(C(=O)COCC3CCCO3)CC2)=O)c1C1CC1 Cc1cc(CCC(=O)NCCN(C(=O)C(C2CCCCC2)C)CC2CC2)n(C)n1 c1(NC(C2N(C(CCCSC)=O)CC(F)C2)=O)c(C)cc(C#N)cc1C C1(N(C(C=CC)=O)C)CCCC(N(C)C(c2cnc(-c3cccs3)o2)=O)C1 C1(COC)(NC(=O)Cc2nc(C3CCCC3)cs2)CCCNC1 c1(C(c2n(CC)nnn2)NCc2ncoc2C(F)F)cnn(C)c1C(C)C C=CCC(C)(CC)C(=O)N1CC(CNC(c2csc(C)n2)=O)C(F)(F)C1 N1(C(C(C)=CC)=O)CCN(C(=O)C(F)CC2CCCCC2)C2CCC12 c1(N(C)CCO)ccc(C(=O)NCC2(C3CC3)COCCN2)cc1 c1(CC(=O)NC2(CNC(C(C)c3cncs3)=O)CC2)ccnc(O)c1 C1(C(N(C)CC2CC2(C)C)=O)CC(F)(F)CN1C(c1cc(F)n(C)n1)=O Cc1ccccc1C(=O)N(C)CC1(O)CN(C(=O)CC2CCC(C)C2)C1 CC(C)(CNC(=O)CSc1ccccc1Cl)C(=O)O.c12cn(nn1)C2 c1(C(C)C(=O)NC2CC(CNC(C3CCC(C)O3)=O)C2)ccc(Cl)c(Cl)c1 C(=O)(C1=C(C2(C)CC2)N(CCC2CC2)C(=S)NC1c1cnn2c1CCC2)OC C1(CNC(CC(=O)NCC)=O)CN(C)CCN1C(C12CC=CC(C1)OC2)=O c1(C(=O)NCC2CN(C(c3ccc(C)nc3C)=O)C3C2C3)ccc([N+](=O)[O-])cn1 N1(C(C(=O)NCC(F)F)=O)CCC(N(CCC(N)=O)C(CN(C)C(N)=O)=O)CC1 C(=O)(C1CCc2c[nH]nc21)N1CC(NC(c2c(N)sc(C)c2C)=O)CC1(C)C C(C(N=[N+]=[N-])C(=O)N1CCC(NC(c2ccc(OC(C)C)nn2)=O)C1(C)C)OC C12(NC(c3ccc(OCC=C)cc3)c3nnnn3CCC)CCCC1OCC2 C1(C(=O)NCC2CC(NC(C3CC(F)(CO)C3)=O)C2)CCCCCC1(F)F c1(C(=O)NC2(C)CN(C(C3CCn4nncc4C3)=O)C2)cc2cccc(Cl)c2s1 C1(c2cn(CC(CC)C)nn2)CN(C(=O)CCCOC(C)=O)CCN1C O=C1CC2=NNC(CC(F)C)C(=O)N1CCC2 N1(C(CCOC(C)C)=O)Cc2n[nH]cc2C1C(=O)NCc1ccn(C)c(=O)c1 c1(C(N2CC3CC3(C(=O)Nc3cnc(Br)nc3)C2)=O)ccc(F)cc1Br C(C(C)(C)C(=O)NC1CC(c2cn(CC3CCO3)nn2)C1)N(C)C Cn1cc(C(N2CC(F)(CNC(C3CCC(C)(C)OC3)=O)C2)=O)n(C)c1=O c1(C(N2CC(NC(C(C)C#N)=O)C(C(F)F)C2)=O)cc2cnccc2o1 c1(C(=O)NC(CNC(c2cnc(C)o2)=O)(C)C(C)C)cccn2ncc(Br)c12 c1(OC)cccc(OC)c1CN1CCCCC1C(=O)NCCc1ccccc1Cl C12(CNC(c3ccns3)=O)CC1CN(C(=O)Cn1ncc(Br)n1)C2 c1(C(=O)OC)cc(C(N2CC(O)CC2CNC(c2[nH]nnc2C)=O)=O)cc(F)c1 Cc1ccc(C(=O)NCC(C)NC(=O)C(c2cccc(Br)c2)(C)C)c(N)c1 C(C1CC(C)Oc2ccccc21)NC(c1c(OCC(=C)C)cccc1)=O C1(O)(C(=O)NCC2C(C(=O)NCc3n(CC)cnc3)C2)CCOC1(C)C C1(C(N(CCN(C)C)CC)=O)CCN(C(c2cc[n+]([O-])cc2)=O)CC1O C1(CC(=O)N(C)CC2CCN(C(C(C)(C)SC)=O)C2)CC(F)(F)C1(F)F C(=O)(C(C)(C)CCC#N)NC12CC(NC(CCCn3c(C)cc(C)n3)=O)(C1)C2 Cc1nc(NC2CC(NC(=O)CCc3ccc4c(c3)OCO4)C2)c2sccc2n1 N1(C(CC2C=NN(C)C2=O)=O)CCCC(F)(C(=O)NCC(C)(CO)CO)C1 c1(C(N2CC(C(C)NC(C(C=CC)O)=O)C2)=O)csc(C)c1Br c1(CN(C)Cc2cc(-c3ccncc3)c[nH]2)ccc(CNC(=O)C(C)(C)CCl)cc1 C(=O)(CC1=CCCCC1)NC(C1CN(C(C2(COC(C)(C)C)CC=CC2)=O)C1)C C1(C)(C(=O)NC(C2(CNC(=O)C(C)N(CC(F)(F)F)C)CC2)C)C=CCC1 C(=O)(C(C#N)C(C)(C)C)N1C(C)CC1C(N1CC(c2ncccn2)C1)=O C=CCC(CNC(=O)CC1CCN(C(=O)C(C)(F)C(C)(C)F)C1)CC(C)C C(=O)(C(C)(C)CCC(=O)N1CCC1CNC(=O)C(C1CCCCCCC1)O)OC N1(C(C2(C)CCOC2)=O)CC2(C1)SCCC2NC(c1csc(-c2cnc[nH]2)n1)=O c1(C(=O)NC23CC(C(=O)N(c4ccsc4)CCO)(C2)C3)cc2ccccc2[nH]1 CC1CC(C)N(C(=O)CCCOC(C)(C)C)CCN1C(=O)C1=CCS(=O)(=O)C1 N1(C(C(CCC)C)=O)CCCCC(C2CN(C(C3CC4(C3)CC4F)=O)C2)C1 C1(CNC(c2c(C)n(C3CC3)nn2)=O)CCC(C)CN1C(=O)CC1(O)CCC1 C1(C(=O)NCC(CC)C#N)(CC)CCCN(C(=O)C=CC2CCC2)C1 C1(CN(C(=O)CC2(CO)CC2)C)CCN(C(c2scnc2C(F)(F)F)=O)CC1 C1(NC(C(CC=C)NC(c2nnccc2C)=O)=O)CCC(C)(C)CC1 C1(NC(c2ccn(CC#N)n2)=O)COCCN(C(=O)Cc2ccc(F)cc2Cl)C1 CC1(C)CN(C(C2CCCC(F)C2)=O)CC1NC(C1C2CCC(=O)C12)=O Cc1nccnc1C(C)NC(=O)C(C1CCCN(C(=O)CC2(C)CC2)C1)C C(C(=O)N1CCN(C(c2cc3sccc3[nH]2)=O)C(CC2CC2)C1)(C(C)(C)C)SC Cc1cccc(CNCC(=O)O)c1.c1(C2C(=O)N2)ccccc1 C1(C2CCN(C(C3CCCS3(=O)=O)=O)CC2)(NC(Cc2c(C)nn(C)c2)=O)CC1 c1(C2C(C(=O)NCC3CCN(C(c4cc(C(C)C)no4)=O)C3)C2)ccc(F)cc1 N1(C(CS(CC)=O)=O)CCC(C2CC2)(CNC(c2conc2C2CCC2)=O)C1 C1(OC)CC2CC1CN(C(=O)C(O)CNC(=O)C(C)SC)C2 C(=O)(C(C)(CCc1nccn1C)N(C)C)OCCOCCNCCOCC c1(CC(=O)NCC(N(C(C2CCN(C)C2)=O)C)C2CC2)csc2c(F)cccc12 c1(C(=O)NCC(c2ccccc2)C)cccc(NC2=NCCS2)c1 C1(C(=O)NCC(=C)C)CC2C=CC1N(C(=O)C=Cc1ccccc1)C2 C(c1cocn1)=CC(=O)N(CC(C)NC(C1CC2(CC2)C1)=O)C CCCCC(F)C(=O)N1CC2CC1CN2C(C12CC(C(C)(C)C)(C1)C2)=O c1(C(=O)NC(CC2CN(C(C(c3cccc(C)c3)F)=O)C2)C)nnc(O)nc1O C(C(O)C(=O)Nn1cnc2ccccc12)NC(C(CCC)C)=O c1(NC(C2N(C(C(C)OCC=C)=O)CC(C)C2)=O)ccc(Br)c(Cl)c1F c1(OC)ccc(C(=O)NC2CCCC(NC(c3nnccc3C)=O)CC2)cc1O c1(C(N(C(CC)CC(=O)NC2CCCC2CN(C)C)C)=O)coc2c1COC2 O=C1C2CC3C(C2)C13C(N1CCCC1C(=O)NCCO)=O Cc1cnc(NC2C=CC(C(=O)NC3CCC(Br)CC3)C2)nc1 N1(C(C2(OC)CCCOC2)=O)CCN(C(=O)Cn2ccc(C)n2)CC(C)C1 n1(CCN(C)C)nccc1C(N1CC(CNC(=O)CCN2CCOCC2)C1)=O C(=O)(N=c1[nH]oc(C(C)(C)C)c1C#N)NCC1(COC)CCCCO1 c1(OC)ccc(C2CCCN2C(c2ccccc2SCc2cccs2)=O)cc1F C1(CC(=O)NC2C3CN(C(c4c(CC)nns4)=O)C2C3)CC2(CCCC2)CO1 c1(SC)ncc(N)c(C(=O)NCC2CCCC2NC(c2cc(C)ncn2)=O)n1 C=C(Cl)CC(C(=O)NCc1ccc(C#N)o1)NC(C1(CC)CCCO1)=O c1(N2C(=O)C3C(CC3)C2)nccc(N)c1Cl.Cc1nc(N(C(C)C(CO)N)C)n[nH]1 N(C(=NCCN1CCCC1=O)NCCC(C1CCCCC1)=O)CC(C1CC1)OC C1(C(=O)OC)CC12CN(C(=O)CC(C)CNC(=O)CNC(C)=O)C2 C(=O)(C1CCCc2cccnc21)NC(CNC(CCC(=O)NCCC)=O)C(C)C C(c1ccc(OC(F)F)c(OC)c1)=CC(=O)NC1CCN(CC(=O)NCC)CC1 C1(NC(c2ccccn2)=O)CCC2CCN(C(c3ccc4cccnn34)=O)C1C2 CC1C(NC(c2cncc3sccc23)=O)CC2CCC1N2c1nnc(C2CC2)s1 C1(C(=O)NCCOC(C)C)CCCN1NC(=O)CCC1CCCN1C Cc1ccc(Br)cc1NC(=O)C(=O)NC1CCCC(CF)C1 c1(C(=O)NCC2CC(NC(c3c(NC)snc3C)=O)C2)nccn2cc(C)nc12 C1(NC(C2(NC(=O)C=CCO)CC(O)C2)=O)CC2(CNC(=O)O2)C1 c1(NC(=O)CCCOC(c2cnn(C3(C(F)(F)F)CC3)c2)=O)ccc(F)cc1 c1(-c2nc(C(CC#C)C)on2)ccc2ncccc2c1 N1(C(Cn2ccc(C)n2)=O)CC(NC(C2(C)CC2c2ccccc2)=O)C2(CC2)C1 O=C1NCC2(CCCN(C(=O)C3=CCNC3)C2)O1 c1(N2CCC(NC(=O)CC3CC4(CC4)CO3)C2)cc(C(F)(F)F)nc2ncnn12 C(=O)(CCCCC(N)=O)N(C(C)CN(C)C(c1cc(-c2ccco2)c[nH]1)=O)C c1(C(N2CC3(C(C(=O)Nc4ccno4)C3)C2)=O)c(F)cncc1F C12(NC(C3C(=C)C3)=O)CC(CNC(c3cc(C4CC4)[nH]n3)=O)(C1)OC2C CC1(C(=O)NCCCC2CCN(C(=O)CCC3CC3(Cl)Cl)CC2)CCC(=O)N1 c1(OC)ccc(NC(C2CC(NC(=O)Cc3cccc(C)c3)C2(C)C)=O)cc1C c1(C(N(C)CC2(O)CN(C(=O)CO)C2)=O)ccccc1SC(C)(C)C N1(C(C(C(C)C)NC(CCOC(C)=O)=O)=O)CC2CC1CN2C(C)C C(=O)(C(C)(C)CC#C)N1CC(OCCNC(C(CC#C)C2CC2)=O)C1.OC CC1OCCCC1C(=O)NCCCN(C(=O)CCOC1CCCC1)C C12(NC(c3n(CC)c(O)nc3)=O)CCC(C1)N(C(=O)COC1CCC1)C2 CC(CC(=O)NC1C2CN(C(C3C4CC5C(C4=O)C35)=O)CC12)CC(F)(F)F c1(C(CC)N(C2CCCN(C(c3cn(C)nc3C)=O)C2)CC)ccc(F)cc1 c1(C(=O)NC2CC(C)(NC(CCC#CC)=O)C2)ccc(OC)c(F)c1N c1(C(=O)NC2(CO)CN(C(C3(C)CC3Br)=O)C2)cc2n(n1)CCOC2 CC(C)CC(CNC(C1(CF)CCOCC1)=O)NC(c1cnn(C(F)(F)F)c1)=O C1(=O)CCCCCCN1.CC1CCCC(CNC(=O)COC2CCOC2)O1 NS(=O)(=O)c1ccc(C(=O)NCC(CO)NC(=O)Cn2cnnn2)o1 N1(C(C=CCC)=O)CCCC(O)(CNC(=O)C(c2c(Cl)cccc2Cl)C)CC1 C(=O)(C1=CCCSC1)NC1(CN(C(CC2CC(SC)C2)=O)C)CC1 c1(C(=O)NOCCC2CCCCO2)n[nH]cc1CNC(C1CCCO1)=O c1(C(C(=O)N(CC(C)NC(C2(C)CCC(C)C2)=O)C)C)cccc(F)c1 c1(C(=O)NCC(CN(C(C2C(NC)C2(C)C)=O)CC)(C)C)ccc2oc(=N)[nH]c2c1 N1(C(CCC=C)=O)CC(CNC(=O)CC2(N3CCCC3)CC2)C2(CC2)C1 c1(C(=O)NC2CCC(NC(C(C)OCC)=O)CC2)c(C)[nH]c2ccc(Cl)cc12 Cc1cc(C(N2CC=C(C(=O)Nc3cnn(C)c3)C2)=O)nnc1C N1(C(c2n(CC#C)ccc2)=O)C(C)CN(C(=O)C=C(Cl)Cl)CC1C N1(C(C(CC)(C)OC)=O)CC(CO)C2(C1)CN(C(c1cncc(Cl)c1C)=O)C2 c1(CC(C)(C)C)ccc(C(=O)NCCC(O)CNC(=O)C(CO)N(C)C)cc1 c1(CCCC)nc(C(=O)NCC2CCN2C(c2ccsn2)=O)cs1 C#Cc1ccc(NC(=O)C(CC=C)CC=C)cc1Br N1(Cc2cccc(OC)n2)CCOC2CC(CO)CCC12 c1(C(=O)NC(CCC)CNC(=O)C(CC)NC(N)=O)cc(C)n(C)c1C C=CC1(O)CCN(C(C2CCCN(C(c3cncc(OC)n3)=O)C2C)=O)C1 C1(CC)CN(C(c2c(Cl)c(C(C)C)nn2C)=O)CCN1C(=O)CCSC C1(NC(C2(CNC(CC3C(C)CC3)=O)CCC2)=O)CCN(C(=O)CC2CC2)CC1 c1(C(=O)NC23CC(NC(C(C(CC)CC)C)=O)(C2)C3)n[nH]c2nccc(Cl)c12 C=CCC(C)C(=O)NCC1(OC)CN(C(c2ccc(CN3CCCC3)cc2)=O)C1 c1(OC)cncc(CNC(C2CC(C)N2C(c2cccc(CO)c2)=O)=O)c1 C12(CNC(CSCCC#N)=O)CCCC(CN(C(c3ccc([N+](=O)[O-])s3)=O)C1)C2 C1(NC(C(COC)O)=O)CCCCC1CNC(C1CCCC1)=O c1(OC)ccc(Cc2cn(CC(O)CNC(=O)CC3CCCOC3)nn2)cc1 N1(C(C(COC)C)=O)CCCC1(C)CNC(c1ccc(C(C)C)o1)=O c1(C(=O)NC(C)CN(C)C(c2csc(=N)[nH]2)=O)cccc(CCO)c1 c1(OC)ccc2c(c1)C(C(=O)NC(C)C(C)(C)NC(=O)CCCNC(N)=O)CC2 C(=O)(CC1=CCCCC1)NCC(=O)NCC(CC(C)C)NC(C1(CO)CC1(F)F)=O C1(NC(COCCCNC(CN(C(C)C)C)=O)=O)CN(C)CCC1O C1(NC(C2C(OCC)C2)=O)CN(C(=O)CC23CC(CO2)C3)CC1C1CC1 c1(OC)ccc(F)c(CN2CC3CC2CN3C(C2CCSCC2)=O)c1F Cc1cc(C(=O)NC(Cc2ccccc2)CCNC(c2cnco2)=O)c(C)o1 CC1(NC(=O)C(=O)NCC(F)(F)F)CN(C(C2CCC2(C)C)=O)C1 N1(C(C(N2CCNC2=O)C)=O)CCC(CF)(NC(c2cncc(CO)c2)=O)C1 Cc1cc(CCC(=O)NC(C)(CNC(C2(CC#N)COC2)=O)C(C)C)cc(C)c1 C(=O)(CC(C)(C)CC(C)=O)N1CC2(CN(C(C3CCC(CC)O3)=O)C2)C1 c1(C(=O)NC2CCCC(CN(C(c3c(C)nns3)=O)C)C2)cc2n(n1)CCC2 c1(C(C(=O)N(C)CC2N(C(CCOC(C)=O)=O)CCC2)C)ccc(Cl)cc1 C1(CNC(COC(CNC(C=CC(=O)OCC)=O)(C)C)=O)CCOCC1(C)C c1(NC(CC2CCN(Cc3ccc(OC)cc3)C2)=O)c(C)nn(C(F)(F)F)c1C CC1(C)CC(CNC(c2ccon2)=O)CN1C(C1CC2CCC2C1)=O C=CCC(C)(O)C(=O)N1CCC(NC(=O)C(C)C2CC2)C(OC)C1 c1(CC)nn(C)c(Cl)c1C(N1CCC(N(C(C2CNC(=O)N2)=O)CC)CC1)=O C1(C(=O)OC)(NCCN2CCP(C)(=O)CC2)CCCC(C)C1 N1(C(CC(C)C)=O)CCOCCC1C(=O)NCC(C)(O)C1CCC1 C1(NC(CCC=C)=O)CCN(C(c2ccc(N)cc2Cl)=O)CC(O)C1 N1(C(c2ccc(OC)cc2C)=O)CC(NC(=O)CC=C(C)C)Cc2ccccc21 c1(C(N2CCN(C(c3c(C(C)C)onc3)=O)CC2)=O)cc2c(F)ccc(Cl)c2[nH]1 Cc1ccc(F)c(C(=O)NC23CCCC(NC(=O)C(C)CS(C)=O)(C2)C3)c1 C(=O)(C1=CS(=O)(=O)CCC1)NC1CC(NC(c2cc(C(C)C)on2)=O)C12CCC2 N1(C(C)C(N)=O)CCC2(CC1)CC2(C)C(N1CCN(C2CCOCC2)CC1)=O c1(C(N2CC(NC(c3c(N(C)C)nccc3)=O)C2)=O)nn(C)cc1[N+](=O)[O-] c1(CN2CC(=O)N(CCCCOCCOCC)C2=O)c(F)ccc(Br)c1Cl c1(C(=O)NCc2cn(CC(=O)NCC3CNC(=O)C3)nn2)ccncc1F Cc1[nH]c(=NCc2cccc(O)n2)sc1C(=O)Nc1cccc(Br)n1 N1(C(CCOC2CN(C(c3nc(CC)oc3)=O)C2)=O)CCCC(C#N)C1 N1(C(C(C2CCC2)OCC)=O)CCC(O)(CCNC(=O)CCCCN(C)C)C1 C1(CC)CCCN(C(c2cnc(C)nc2C)=O)C1C(=O)NCCC[Si](C)(C)C C1(CN)CC(CNC(C2CSC2)=O)CCO1 CCCC(CC)C(=O)N(C(C)CN(C)C(c1cc(=O)n(C)cn1)=O)C c1(NC(C(CC)(C)O)=O)ccc(NC(=O)CCC(=O)N2CCOCC2)c(F)c1 c1(C(N2CCCC(N(C(=O)CC3CCC(=O)N3)CC)C2)=O)ccc(S(N)(=O)=O)s1 C1(C(N2CC(OC(=N)O)C2)=O)(NC(C(C2CCC(=O)N2)C)=O)CC1(C)C N1(C(C=C2CCC(C)CC2)=O)CC2CCC1C(CNC(C1CCC(O)CC1)=O)C2 c1(C(=O)NCC2N(C(C(C)OC)=O)CC(F)(F)C2)c(C)sc2ccccc12 Fc1ccc(Cc2nc(-c3ccsc3)nn2-c2ccc(OC(F)F)cc2)cc1Cl C(c1ccc2occc2c1)=CC(=O)NCC(CNC(C1C(C(C)C)C1)=O)(C)O Cc1cccc(C(=O)NCC(CC2CC2)C(=O)NCc2ncccn2)c1N c1(OC)cc(C(=O)NC2CCC(NCc3c(F)cccc3Cl)C2)c(OC)cc1Cl c1(C(N2CCCC(O)(CNC(CCOC(C)C)=O)C2)=O)cn(C)c2ccccc12 c1(CNC(=O)Nc2c(SC)cccc2)c(C)nn(C)c1Cl C1(CC)CN(C(c2cnc(O)cc2C)=O)CCC1NC(=O)CCc1ccco1 C(=O)(CCCN=[N+]=[N-])NCC(C(C)C)NC(=O)COc1ccc(Cl)cn1 Cc1cc(F)ccc1C(N1CCCC1)=O.c12ccc(cc1)C(=O)N(C)C2 CC(CC1CC1)C(=O)NCC(c1ccccc1)CNC(=O)CCc1ccn(C)n1 C(=O)(C(CC(C)C)CC(C)C)N1CC(NC(CCCOCC=C)=O)C(C)C1 c12ccc(nc1C)N1CCN(CC1)C1CCN(CC1)C2=O.C1(N)CCOCC1.CS Cc1[nH]c(=N)sc1CC(N1CC=CC(NC(c2ccc(C(N)=O)[nH]2)=O)C1)=O CC1CC(C(N2CC(C)(NC(=O)CC3CC4CCC3C4)C2)=O)CCO1 Cc1c(Br)c[nH]c(=NCC(c2ccccc2)c2ccccc2)c1C c1(C(CC)NC(C2CCN2Cc2noc(C)n2)=O)cccc(C(F)(F)F)c1 c1(C(N2CCC(C)(NC(=O)CCC3CCOC3)C2)=O)cc(S(N)(=O)=O)ccc1N C1(C2CCCCC2)(C(=O)NC(CCNC(C(C(C)C)OC)=O)C(C)C)CC1 N(S(N)(=O)=O)CC(=O)N(CC(C)NC(c1cnc[nH]1)=O)C N1(C(C(C)(C2CC2)OC)=O)CCC2(CCC2)C(CNC(=O)CCCF)C1 c1(C(=O)OC)c(C(=O)NC(C)Cn2cc(CNC3(CO)CCC3)nn2)n[nH]c1C C1(NC(c2c(C)cc[nH]2)=O)CCN(C(C2CCC(C(C)C)CC2)=O)CC1C C1(CCC(=O)N(CC(CC)NC(c2c(CC)nns2)=O)CC)CCC(=O)NC1 c1(OC)ccnc(OC)c1C(=O)NC1CC2CC1N(C(=O)C(C#N)C(C)C)C2 CCC(C#N)(CC)C(=O)N1CCN(C(c2ccc(C3CC3)o2)=O)C(CCO)C1 CCC(CC1CCC1)N(C)N1CC(C)OC(C)C1 c1(C(=O)NCC(C)(CO)NC(C2CCC(=O)N2)=O)cccc2c(O)nncc12 c1(CC)nc2ccccc2cc1C(=O)NCC#CCNC(=O)C(C)N1CC(C)C1 c1(C(=O)NC2C=CC(CNC(C3C(C=C)C3)=O)C2)csc(=NC)[nH]1 C(=O)(C(F)n1ccnc1)NCC(=O)NCCc1ncc[nH]1 N#Cc1ccc(CC(N2CC3CC3(CNC(=O)CC3NC(=O)NC3=O)C2)=O)cc1 C1(CNC(c2n(CC=C)nnn2)(C2CC(C)(C)C2)C)C(C)(C)C1(C)C c1(C(N2C(C(C)(C)NC(CCSCCCC)=O)CCC2)=O)cccc(COC)c1 N1(CCNC(N(CC(CC)O)C)=O)CCOC(C)C1 CCC(C)C(CC(=O)NCCS(=O)CC)NC(=O)C(CC1CC1)OC c1(C(=O)NCC(C2CC2)NC(C2CCC(C(N)=O)O2)=O)ccc([N+](=O)[O-])s1 c1(C(=O)NC2C(C)CCN(C(=O)CCCC#N)C2)cnn2ccc(Cl)c(F)c12 N1(C(C(CC2CC2)NC(C(n2c(C)ccn2)C)=O)=O)CC2(C1)NC(=O)NC2=O Cn1nc(C(=O)NC2COCCC2NC(=O)Cn2cnnc2)cc1C(F)(F)F C=CCCC(C)(C)C(=O)NCCC1CN(C(=O)CC2CCN(OC)CC2)CCO1 C1(CCOC)CN(C(c2ccc(Br)cc2)=O)CCN1C(=O)COCC(C)C C1(CC(N2C(C)CC(F)C2)=O)CC2(CC2)CN1C(C1CC(C)(C)CN1C)=O Cc1nc(C2CCCC2)sc1C(=O)NCC1CC(NC(C2CN(S(C)(=O)=O)C2)=O)C1 CCCCCCC(CNC(c1ncoc1C1CC1)c1nnnn1C1(C)CC1)CC c1(C(C(=O)NCCCSCC)N(CCCN(C)C)C)nc(C)sc1C N1(C(CCCC(=C)C)=O)CCC2(CC1)CC2NC(=O)CCN(C)CCO c1(C(N2CCCC(C)(NC(C3CC4CC4C3)=O)C2)=O)cc2c(nc1N)CCCC2 c1(C(N(CC(CNC(CC(COC)C)=O)C)C)=O)cc(OC)ccc1F c1(C(N2CCCN(C(C(C)NC(=O)NC)=O)CC2)=O)ccc2nn[nH]c2c1 c1(CC=C(C)C)cc(C(=O)NC2CCN(C(C3(C)CC3C)=O)CC2O)ccc1F C1(C)(NC(C(CCC)O)=O)CCN(c2nc(OC)cc(OC)n2)CC1 CC(C)C(CNC(c1occ2c1CCC2)=O)N=c1[nH]nc(C#N)s1 C1(C(N(C2CCCC(O)C2)C)=O)CC(C)(C)CCN1C(C1CCNC(=O)C1)=O N1(C=O)CCC(c2ccc(F)cc2)CC1.CC(C#N)CN(C)C(=O)NCCSC C(C(CC(F)(F)F)NC(C1(CCF)CCC1)=O)NC(C(COCC)C)=O O=C1CN(C(=O)OCCOCCO)c2ccccc2N1C(=O)C1CC1SCCCO c1(C(=O)NCC2N(C(C3N(C(C)C)C(=O)CC3)=O)CC2)cccc(C#N)n1 c1(C(=O)NCCCCC(=O)Nc2c(C)csc2)c[n+]([O-])c(C)cn1 c1(-c2c(CN(CCN(C)C)C)cc(Cl)cn2)ccc2c(c1)C(=O)C(=O)N2 c1(C(=O)NC(C(=O)NC(c2n(C)ncc2)CO)C2(C)CC2)cc(Cl)cn1C c1(C(N2C(C(=O)Nc3cnn(CC)c3)CC(=C)C2)=O)cnc(Cl)cc1OC C1(C(N(CCN(C)C(C2CC(=O)N(C3CCC3)C2)=O)C)=O)CCC2(CCC2)CO1 C(=O)(C(C(C)O)NC(C1CCCN1C(C)C)=O)NC1CCN(CCC)C1 Cc1cn2c(n1)C(C)CC(C(=O)NCC1CN(C(C3OCCCO3)=O)CC1O)C2 c1(C(C(=O)NCCN2CCC(O)CC2)Nc2ccco2)ccc(F)c(Cl)c1 C(=O)(CCC(=O)NN(C)C)N1C(C)CN(C(c2cnc(SC)n2C)=O)C(C)C1 Cc1nc(C)c(C(=O)OCc2nc(CS(C)(=O)=O)n[nH]2)c(C)n1 c1(C(=O)NCC2C(NC(c3c(C(C)C)occ3)=O)COC2)ccn2ccnc2c1 C1(NC(=O)C(F)=C2CCCC2)CCCC(NC(c2ccc(C3CC3)nc2)=O)C1 N1(C(c2cncc(C(=O)OC)c2)=O)CCN(C)C(CNC(=O)CCC2CCC2)C1 C12(NC(=O)COc3cccnc3)COCCC1CN(C(=O)CN1CCSCC1)C2 Cc1c(C(=O)NCCC(O)CNC(=O)CC2CCCOC2)sc2[nH]cnc(=O)c12 C1(NC(CC(C)C)=O)CCN(C(=O)Cc2ccc(F)c(Cl)c2)C(C)C1 C12(C(=O)NC3CC(C)N(C(=O)CSCc4ccncc4)C3)CCCC(C1)OC2 CC(CC(=O)NCc1csc2ccc(Cl)cc12)CC(C)(C)C C1C(CO)(CO)N1C(=O)C(C)NC(=O)C(C)SC.c1(C(=O)N)ccco1.CO c1(CCC)cnnc(C(N2CC(CC(C)(C)CNC(C3CC(NC)C3)=O)C2)=O)c1 c1(C(N(C(C)C)CCNC(=O)C(c2ccccc2)F)=O)cncc(C(F)F)c1 O=C(C#CC1CCCC1)N1CC(O)CC1C(=O)N=c1ccn(C(F)F)[nH]1 C(CCCC(=O)NCCCCC(=O)NC(C)CC(C)O)OC CC(C)(C)C(=O)NC1CC1C(=O)NCC1COC(=O)N1 c1(C(N2CCC(N(C(=O)C(F)C(C)C)CC)CC2)=O)cncc(Cl)c1C C(C(=O)N1CCC(C)C1CNC(c1cc(C(N)=O)c[nH]1)=O)(C(C)C)NC(=O)OC Cc1noc(C(=O)NC(CNC(=O)CCC2CC2(F)F)C2CC2)c1C C1(NC(=O)OC(C)(C)C)CCN(Cc2cccc(CO)c2)CC1CC#N C(C1=NOC2CN(C(c3nocc3C(C)(C)C)=O)CC12)NC(COCCC=C)=O C(=O)(C(C)(C#N)CC)N1CCC(C(C(=O)NCCN(CCC)CCC)C)CC1 N1(C(CCc2cc(C)[nH]n2)=O)CCC(C(=O)NCc2cn(C)cn2)C(C)(C)C1 c1(C(=O)NC(C(C)(C)NC(CC(C)n2ccnc2)=O)C)ccc(=O)n(C)n1 C(=O)(CCCC(C)=O)NCC1(C(=O)NCCN(C)C)CC(=C)C1 N1(C(c2c(C(C)C)cccc2)=O)CCCN(C(=O)CCCCCO)C(C)C1 C(C(=O)NC1CCN(c2cc(C)ncn2)C1C)(C(C)C)NC(C)=O c1(C(C(=O)N(C(C)CNC(=O)CCN2CCOC2=O)C)C)c(C)noc1C c1(C(=O)NCC(C)(C2CC2)NC(C(C)n2cccn2)=O)ccc(C#N)[nH]1 C1(NC(C2C(C)(CC)C2)=O)CC2(CCN(C(=O)CC3=CCCC3)CC2)C1 C1(CNC(CNC(CNC(C)=O)=O)=O)(CNC(C2CCCCO2)=O)CCCCC1 N1(C(=O)OC(C)(C)C)CC2CCC(C1)C(NCC1CCC(=O)N3CCCC13)C2 N1(C(=O)Nc2n(CC)nc(C)c2-c2ccccc2)CCCNC(=O)C1(C)C N1(C(C(C(C)C)CO)=O)CCC(C)N(C(c2ccc(-c3cnn(C)c3)o2)=O)CC1 Cc1cc(C(C(=O)NCC(C)C)N(CCC(=O)N(C)C)C)c2ncccc2c1 N1(C(c2c(C)cco2)=O)CC(NC(C2CCC(N(C)C)CC2)=O)C2(CC2)C1 N1(C(c2cc(Cl)c(Br)cc2Cl)=O)CC2CCN(c3ncnc4occc34)CC2C1 c1(CC)cc(C(N2CCC(CNC(=O)C(C3CCCC3)OC)C2)=O)n(C)n1 CC(C)CC(C(=O)NCC1(F)CC(NC(=O)Cc2nc(=N)[nH][nH]2)C1)C(C)C C1(CC)(NC(C2CCC2(F)F)=O)CCN(C(c2cnn(CCOC)c2)=O)C1 N1(C(CC(C)OC)=O)CCC2(CC1)C(NC(=O)CC1(CO)CC1)CS(=O)(=O)N2C N1(C(COCCNC(c2c(CC)cncc2)=O)=O)CCCC2(CC1)CC2 c1(C(N(CC(C)N(C(=O)CCC(C)(C)C)C)C)=O)cnc(N)c([N+](=O)[O-])c1 CCC(CC(=O)NCCC1CN(C(c2nc[nH]c3ncnc2-3)=O)C1)CC(C)C C1(CN(CCc2c(C)ocn2)C)CCCN(C(=O)C(=O)C=Cc2cccs2)C1 C(S(=O)(=O)CCCC(=O)N=c1cc(C2CC2)n(C)[nH]1)C1CC(C(C)C)C1 C1(C(N(CC=C)Cc2cccc(-n3cnnn3)c2)=O)Oc2ccccc2OC1C N1(C(C2N(C)CCCC2)=O)CC2(CCC2NC(=O)CN2C(=O)CNC2=O)C1 C1(CNC(C2CN(C(C)C)C2)=O)CCOC1C(=O)NCCC1CC1 C(N=c1cccc(S(=O)(=O)N2CCOCC(C)C2)[nH]1)c1c(OC)ccnc1 N1(C(C(F)=CC)=O)CCOCC(CNC(=O)CC2(OC)CCCC2)C1 c1(OCC)n[nH]cc1C(=O)NC1(CCNC(=O)Cc2cnnn2C)CCC1 C(CC(=O)NCCn1cc(C)cn1)(CC(C)C)NC(C(C)OCC)=O c1(C(N2C(C(=O)NC(c3ccc(F)cc3F)CO)CC2)=O)c(Cl)cc(Br)cc1Cl C1(CC(C)NC(c2cc[nH]n2)=O)CCN(C(c2cncc(F)n2)=O)CC1 C(=O)(C1=CCN(C(C2(C(C)(C)O)CCC2)=O)CC1)NC(CCOC)C N1(C(C(COC(C)=O)C)=O)CCCN(C(=O)C=CC2CCCN2C)CC1C C1(NC(c2cc(Cl)cc(Cl)n2)=O)CCN(C(=O)CCC[N+](=O)[O-])CC1F C(=O)(CCCC1OCCO1)NCC1(NC(C(C)SC(C)C)=O)CCC1 c1(C(=O)NC2CCCN(C(CCCOCCC)=O)C2)ccc(O)c(C(C)=O)c1 c1(C(N2CCCC(NC(C3C(C)CC3)=O)CC2)=O)ccc([N+](=O)[O-])cc1Br c1(C(=O)NCCN(C(c2ccc(OC(C)C)o2)=O)CC)ccc2n[nH]cc2c1 N1(C(C23OCC(C)(C2)C3)=O)CCCC(F)(CNC(c2cscc2F)=O)C1 c1(C(N2CCN(C(C(c3scc(C)n3)C)=O)C(C)C2)=O)ccc(N)c(Cl)c1O C(=O)(CCCC(C)(F)F)NCCCCN(C(C(C)Oc1ccc(Cl)cc1)=O)C CON(CCO)C(=O)C1CCC(NC(=O)C2=C(C)CC2)C1 C(=O)(C1CCCc2cncn21)N1CCC(N(C(C2(OC)CCCOC2)=O)C)CC1 Cc1n[nH]c2cnc(C(=O)NC3CN(C(=O)Cn4cccc4)CC3O)cc12 Cc1ccc(S(=O)(=O)NC(=O)CCc2ccccc2N)cc1C C1(C#N)(C(N2CC(NC(c3ccc(C#C)cc3)=O)C2)=O)C(C#N)C1(C)C C=CCC(C(=O)N1CC=CC(NC(c2nnn3c2CCCC3)=O)C1)C(C)C C1(C(C)C)CN(C(C2CCC(N(C)C)CC2)=O)CCN1C(=O)C(=O)N(C)C C1(NC(C2CCCN(CC)C2)=O)CC2(CCCN(C(=O)COCCCF)C2)C1 C(=O)(C(CNC(C1CNC(=O)N1)=O)C(C)(C)C)NCC1N(C)C(=O)COC1 c1(C(=O)NC(C(C(=O)OC)(C)C)c2ccccc2)ccc2nccc(=O)n2c1 N1(C(CC(C(C)C)(F)F)=O)CC2CCCN(C(c3cn4c(n3)COCC4)=O)C2C1 CC1CCC(NC(c2ccc(C(F)F)cn2)=O)CN1C(c1ncc(Cl)nc1Cl)=O c1(CC)c(C(=O)NC2CC(NC(c3cnccn3)=O)C2)cnn1-c1ccccn1 Cc1c(CC(N2CCC(CC(=O)N(C3CC4(CC4)C3)C)C2)=O)ncn1C c1(C(=O)NCC2(O)CC(C(=O)NCC(C)C(C)(C)C)C2)ccn2cncc2c1 CCCCCCC(CC)NC(C1(C)CCCN(C(=O)CCc2csnn2)C1)=O CCC(CC(=O)NC1CC2(C1)CC2NC(c1coc(Cl)n1)=O)C1CC1 C1(CNC(c2c(C)ccc(C)c2)=O)CN(C(C2COCCOC2)=O)CCC1(F)F c1(C(=O)NCC2(NC(c3cc(C(F)(F)F)cc(F)c3)=O)CC2)cc2cccn2cn1 Cc1cc(C(=O)N(CCC(C)NC(=O)C(n2ccc(C3CC3)n2)C)C)ccc1Cl C1(C(N2CC3CN(C(C(COC)C)=O)CC32)=O)Cc2ccccc2CN1C n1(CCC)ncc(C(=O)NC(Cc2ccccc2)C(=O)N2CCCCC2)c1Cl C(C)(N(C)N1CCOC2CCN(CCO)CC12)c1nc(C)sc1 CN1CCOCC1C(=O)NCC1(C)N(C(=O)C(C)(C)N2CCCCC2)CCC1 C1(NC(Cc2ccc(C)s2)=O)CC2CCC(C1)N2C(=O)COC1CCOCC1 CC1CCCCC1(C)C(=O)NCCn1ccc(C(=O)NC2CC3(C2)CC3(F)F)c1 C1(CC(=O)NC(CN(C2CC2)CC)C)CCCCN1C(=O)CSc1nc[nH]n1 Cc1ccc(C(N2CC(NC(=O)Cc3sc(O)nc3O)C(C)C2)=O)c(O)c1 N1(C(C2CSCCS2)=O)CCN(C(c2cncs2)=O)C(c2cccc(F)c2)C1 Cc1ccnc2nc(C(N3CCCC(NC(=O)CCOCC4CC4)C3)=O)nn12 C(C(C)(F)C(C)(C)F)(c1n(-c2ccc(OC)cc2)nnn1)NCC(Br)=C(C)C N1(C(C)C(=O)NC2(CO)CCCC2)CCN(C(c2ccoc2Cl)=O)CC1 c1(C(C)C)ncc(C(=O)NC(C)CC2CN(C(=O)CC(=O)N(C)C)C2)s1 C(=O)(CC(C(F)(F)F)NC(C1(C(C)(C)O)CCC1)=O)NC(c1ncccn1)C CC1CCC2N(C1)C(=O)C(=O)NC2.c1(C2(CN)CC2)cccs1 C1(C(N2CCCC(CN(C(c3cc(C)sc3)=O)C)C2)=O)CC12CCOCC2 c1(OC)cc(C(=O)OCc2ccc(O)c(Cl)c2)nc(C(C)C)n1 CCCC(CCC)C(=O)NCC1(CNC(C2CCN(C3CCSC3)CC2)=O)CC1 C(=O)(C(CC(C)C)N(C)C)N(CCCOCCNC(CC)=O)C c1(C(N(CCC(C)NC(=O)Cc2cnns2)C)=O)ccc([N+](=O)[O-])cc1F Nc1cc2c(cc1C(N1CC3(CNC(=O)CC4CCCO4)CCC1C3)=O)CCC2 C1(C2CCCC2)(C(=O)NC(C(C)(C)O)c2ccccc2)CCNC1=O N1(C(c2oc(CC)c(C)c2)=O)CC(NC(=O)C(COC)OC)CC12CCC2 CCCCCC(=O)N1CCC(C(=O)NCCn2ccccc2=O)(C(C)C)C1 c1(OC)c(C(=O)NOCCSc2cn(C3CCCC3(F)F)nn2)ccc(Br)c1F c1(C(=O)Nc2ccc(NC(=O)NC(C)=O)cc2)c(C)cnnc1O O(NC(=O)C(=O)OCC1CC(F)(F)C1(Cl)Cl)CCC1N(C)CCC1 c1(C(CC)C(=O)NCC2(O)CN(C(=O)CCN(S(C)(=O)=O)C)C2)cccc(Cl)c1 C#CCCC(C(=O)NCC1CC2CCC(C1)C2)NC(c1nocc1Cl)=O N1(C(C(CCCCC)F)=O)C2CCCC1CN(C(=O)CC(C)F)C2 c1(CNC(c2cc(Cl)cc(Cl)c2F)=O)ccc2ccccc2n1 C(C(C)(C)CC(=O)NC1(CCCCO)CC1)NC(C1N(CC)CCOC1)=O c1(SC)cnn(C)c1C(N1CCC(c2cn(CCOCCO)nn2)C1)=O c1(CC)ccccc1OCC(=O)NCC(CNC(=O)C(c1ccc(Cl)cc1)C)OC c1(OC)nc(N2CC(CNC(N3CCCC(O)(CO)C3)=O)C2)cc(C)n1.C(C)(C)(C)O Cn1ccc2cc(C(=O)NCCC3CCCN(C(=O)COC(F)F)C3)cnc12 C#CCC(C)(CC)C(=O)NC1CCCC1C(=O)NCCC(C)N1CCC1 C1(C)(C(=O)NC(C)(C)C)CC12CCN(C(=O)Cc1ccccc1O)CC2 C(=O)(CC(C)(C)CNC(C)=O)N1CC(C(N2CCCC(C(C)O)C2)=O)(SC)C1 NC1CCc2ccc(C(=O)NCc3nccc(O)n3)cc21 c1(CNC(=O)C(=O)NCC2CCCCCCC2)ccc([N+](=O)[O-])cc1Cl N1(C(C(=O)NCCOC)=O)CC(C2(NC(c3cnn(C(F)F)c3)=O)CC2)C1 Cc1cc(C(=O)NC2CC(NC(C3(CO)CCOC3)=O)C2)c(F)cc1Cl Cc1ccc(CCC(=O)NC2CCCC2NC(C2(C)COC(=O)OC2)=O)cc1Cl N1(C(C(C)OCC(F)(F)F)=O)CC(C)(CNC(=O)COC2CCCC2)CC1(C)C CCC(C)C(O)CC(=O)NCCCN(C)C(C1(C2(O)CCC2)CC1)=O C(=O)(CC(C)(C(F)(F)F)N(C)C)NCC(CCCC)NC(=O)CCCN(C)C CCC(O)C(F)(F)C(=O)NCCCNC(=O)CCc1c(F)cccc1Cl CC1CCN(C(c2nc(Cl)cs2)C(=O)NCCCF)CC1NC(=O)OC(C)(C)C c1(C(N2C3C(NC(C(CC)CC)=O)CC(C3)C2)=O)cc2ccccc2s1 C(=O)(C(C)(O)C(C)C)NC(CC)CN(C(=O)CSCc1cccc(C)c1)C c1(CNC(C2CCN(C)C2)=O)ccc(CNC(=O)CC2CC3CC3C2)cc1F N12CCOCC(C1)C2=O.c1(OC)n[nH]cc1C(N1CCCC1CN(C)C)=O N1(C(CC(C)(O)c2ccccc2)=O)CCC(NC(=O)C=CI)C(CO)CC1 c1(C(N2CC(OC)C(NC(c3ccc(C(F)(F)F)o3)=O)C2)=O)ccc(N)c(F)n1 C(=O)(CCCn1ccnc1)NC(CNC(C1(COCC)CC1)=O)C1CC1 C1(NC(C(C2CCCCC2)NC(C(C2CCOC2)OC)=O)=O)(CO)CCOCC1 CCCC(CNC(=O)C(C1CCC1)OC)NC(c1c[nH]nc1C(C)(C)C)=O C(=O)(C1=NOC(C)C1)N1CCC(OC)(CNC(=O)CC2(OC)CCCCC2)C1 N1(C(c2cc(C)sn2)=O)CCCC2(C1)CN(C(c1ccnc(C)c1C)=O)CCO2 c1(OC)cc(C(N2CCOCC2C(N2CCCC(F)C2)=O)=O)c(C)cc1[N+](=O)[O-] C1(C(N2CCC3C2CCCN3Cc2ccccc2)=O)CCc2nccn2CC1 c1(C(=O)NCCC2N(C(C(C)=CC)=O)CCC2)cccc(OC)c1O N1(C(C(n2c(C)ccn2)C)=O)CCC(F)(C(=O)NC2(CO)CCCCC2C)CC1 c1(C(N2CCCC(NC(C3CC(=C)C3)=O)C2C)=O)cccc(SC)c1[N+](=O)[O-] CC(C)(C)CC(C)(C)C(=O)N1CCN(CCCNC(=O)C2=CCCCO2)CC1 Cc1ccc(C(=O)NCC23CC(NC(C4OCCOC4C)=O)(C2)C3)cc1C C(=O)(C(CC(F)F)NC(C1CC(C)(C)CO1)=O)NCc1cc(C)ns1 C1(CC(=O)NC2(CNC(CC3CC(C(C)(C)C)C3)=O)CCC2)CCC2(CC2)CO1 C=CCCCCCCC(=O)N1CC(OCCNC(c2n[nH]c3ncccc23)=O)C1 N1(C(CCC)=O)CCCN(C(c2nnc(S)n2C)=O)CC1C(C)C C1(C(N(C)Cc2ccc(Cl)s2)=O)C2CCC1(c1ccc(Br)cc1)C2 O=C(CC1=Cc2ccccc2C1)NC1CCCC(CNC(=O)CSC2CC2)C1 C1(CNC(CCC(=O)NC)=O)CN(C(C2CC3COCC3C2)=O)CC(C)(C)O1 c1(C(C)(C)C)cnc(C(=O)NC(C2CCCN2C(C2CCCCS2)=O)(C)C)cn1 C1(COCC)CCCN(C(=O)NCC2CCCN2c2ccccc2)C1 c1(C(N2C3CCC(NC(C(C#N)C4CC4)=O)(C3)C2)=O)cc2ccnc(Cl)c2[nH]1 N1(CCNC(C2CC(C)(C)OCC2)=O)CCN(C(C2CCC2CF)=O)CC12CCC2 O=C1NC(C(=O)NCC2CC2NC(c2cccc(Sc3ccccc3)c2)=O)CC1F Cc1cc(C(=O)NCC2(C(N)=O)CN(C(C3(C4CCCO4)CC3)=O)C2)oc1C N1(C(c2cn(CC)nc2)=O)CC(CNC(=O)C(N2CCSCC2)C)C(F)(CO)C1 C1(NC(c2cccc(N)n2)=O)CC2CCC1C(NC(=O)CSCc1cccs1)C2 c1(CN(C2CCCC(n3ccnc3)C2)CC)ccc(C#N)cc1F C1(NC(c2c(OCC)oc(C)n2)=O)CN(C(=O)C(C)(O)CC)CC1S(C)(=O)=O C1(C)(NCC(=O)N(C(CCNC(Cn2c(C(C)C)ncc2)=O)C)C)CC(C)(C)C1 c1(C(=O)NC(C2N(C(C(C=CC)O)=O)CCC2)(C)C)cnn2ccsc12 C1(C(N(C(CCC)CC)C)=O)CCOCC1C(=O)OC c1(C(=O)ON(CCCCCC)CCCC(C)C(F)F)cnc(OC)nc1 c1(N(C(CNC(CC2C(C)(C)C2)=O)=O)CC2CCCC2O)ncoc1C1CCC1 c1(NC(C)C(C)Sc2ccccc2)ccccc1C1CC1C(F)(F)F c1(COC)cc(=NCC2CCC(NC(=O)CCCC3CCC3)C2)[nH]cn1 CCCC(C)(C)CC(=O)NCC(CNC(C12CCCC1C2(F)F)=O)S(C)(=O)=O CCC(CC)C(C(=O)N1CCCOC(CCNC(C2(C)CC=CC2)=O)C1)OC C1(NC(CCc2n(C)ncn2)=O)CC2CCC1N2C(=O)COCC1CCCOC1 CN1CC(C)(C)CC1C(=O)NC1CCCCN(C(C2(C)CCC2)=O)C1 c1(C(N2CCC(C)C2CNC(C2CCC(O)C2)=O)=O)cccc(C#N)c1 C(=O)(C(C(=O)N1CCC(NC(=O)CCCc2cc[nH]n2)CC1)C(C)(C)C)OCC N1(C(COCCC)=O)CC2CCC1C1CN(C(c3csc(C)n3)=O)CC21 c1(OC)ccc(C=CC(=O)NCC2CC(NC(c3cc(CF)on3)=O)C2(C)C)nc1 CCCC(C)C(=O)NC(Cc1ccccc1Br)C(N1CCSCC1C1CC1)=O CN1CC(NC(=O)C(C2(C)CC2)NC(c2ccc(=N)[nH]n2)=O)C(=O)N1 c1(C(=O)NCCCCNC(C(CCSC)O)=O)cc2ccccc2nc1C(F)F C1(CCNC(=O)CSCCOC2CC2)(NC(C2C(=C)C2)=O)CCOCC1 C1(OC(=O)Cc2ccc(NC(=O)NCC)cc2)CCCCC(c2ccccc2)C1 CC1CCN(C(=O)CC2CCC(=O)NC2)C(CNC(=O)CCc2cnco2)C1 c1(NC)ccccc1C(=O)NCCC1CC(C(=O)Nc2ccsc2C(C)C)C1 N1(C(CSCC#C)=O)CCC(NC(=O)CN2CCn3ccnc3C2)CC(O)C1 CC(CCCCCO)NC(=O)C(C1CCCO1)NC(=O)CCc1ccccc1 c1(CC)nc(C)c(C(N2CC(CNC(c3c(Cl)cnn3C(C)C)=O)CC2C)=O)s1 Cn1cccc(C(=O)NCC2CCCCN2c2nnc(-c3ccccc3)o2)c1=O CC1C2C(CCN2C(c2csnc2Cl)=O)CN1C(=O)C(C)n1cncn1 C1(C(N2CC(C3(NC(C4C(C)C4)=O)CC3)C2)=O)CCOC2(CCCC2)C1 CC1CN(C)CC(C(N2CCC(NC(c3c(C(F)F)cnn3C)=O)C(O)C2)=O)O1 N1(C(c2ccc(C)nc2)=O)CC2CCC(CNC(C3CSCCS3)=O)C2C1 Cn1cnc2c1CCC(C(N1CC(NC(c3cccc(N)n3)=O)C(C)(C)C1)=O)C2 Cc1cc(=NCCCN2CCCC2)[nH]cc1S(=O)(=O)NCC1C(F)(F)C12CCC2 C1(NC(=O)Nc2nc(-c3cccnc3)cs2)CC12CCc1ccccc12 c1(C(C(=O)Nc2ncn(C)c2)N(C)C)ccccc1[N+](=O)[O-].N12CCC(O)(C1)C2 c1(CC(=O)N(CCC(C)NC(c2c(SC)cccc2)=O)C)cc(F)cc(F)c1 c1(C(=O)NC(CNC(c2c(OC)n[nH]c2)=O)C2CC2)ccc(C)c(Br)c1C c1(-n2c(C(C(C)C)SCC)nc(-c3ccc(Cl)s3)n2)ccc2nccnc2c1 S(=O)(=O)(c1ccc(COC)cc1)C(CSCCC(=O)N(CCC)CCC)=O C(=O)(C1=C(Cl)CCOC1)NCCC(C)(C)NC(=O)COc1ccc(C(N)=O)cc1 c1(C(=O)N(CCCNC(c2c[nH]nc2C(F)F)=O)CCO)ccc2ccnn2c1 Cc1c(C(=O)NCC2CC2NC(=O)CCSc2ccccc2)n[nH]c1C1CC1 Cc1ccc(C(N2CCN(CCNC(c3cc(C4CC4)[nH]n3)=O)CC2)=O)cn1 C12(CNC(COCCC)=O)CCC1CCN2C(c1cccc(NC(C)=O)c1)=O C(CCC(CO)NC(=O)CC1(C(=O)NCC)CC1)NC(C1(C#N)CCC1)=O Cc1cc(=O)cc(CNC(c2cn(CC(F)(F)F)cn2)=O)[nH]1 c1(CCNC(C(C)SC(C)C)=O)ocnc1CNC(C1CCC(C(N)=O)O1)=O C1(NC(CC2(OC)CCC2)=O)C2COCC1CN(C(=O)C=CC1CCCO1)C2 N1(CC(=O)NCCC)CCC2(CCN(C(c3cccc4ncccc34)=O)C2)C1 N1(C(C2OCCN(CC)C2)=O)CCN(C(c2ccn(C(F)F)n2)=O)C(C(F)F)C1 CC1CCC(CNC(C2CCSCC2)=O)N(C(c2ccc(C(F)F)c(F)c2)=O)C1 c1(OCCCC(=O)OC2CCN(CC(c3cc(C)[nH]n3)=O)C2)ccccc1Br c1(C(C(=O)NC(C)CC)N(CC(C)C)CCC)cc2c(cc1OC)CCC2 C(CN=c1[nH]nc(C2CC2)o1)(CC(C)C)NC(C1CCN(C(C)=O)CC1)=O C1(NC(c2c(C)snn2)=O)CN(C(c2cc(C3CC3)no2)=O)CC1O c1(OC)nc(Cl)ccc1C(=O)NCCC1(O)CN(C(=O)C(O)Cc2cnc[nH]2)C1 c1(C(N(CC(C)NC(C2(O)CN3CCC2CC3)=O)C)=O)cc2c(O)cccc2[nH]1 c1(NC(CC)C(C)CN(C)C)nc(=NC2CCC3(CC3)C2)[nH]c2c(C)nn(C)c12 c1(C(=O)NCC2CN(C(CCC3C(C)C3)=O)CC23CC3)nn(CCF)cc1[N+](=O)[O-] N1(C(C=C(CC)CC)=O)CCC2C(CCCN2c2cc(SC)nc(SC)n2)C1 c1(NC(C2C=CC(NC(c3c(CC)n(C)cc3)=O)C2)=O)cc(C)c(C)c(C)c1 N1(C(CC2(C)CCCC2)=O)CCCC(CNC(=O)CC2CCC23CCC3)CC1 CC(O)(CNC(=O)CCCC1CCCC1)CNC(C1CCCCC1)=O Cc1nnc2n1C(C(=O)N(C(C)CCNC(c1cccc3ccnn13)=O)C)CC2 C1(CCC)(NC(CCCC#C)=O)CCCN(C(c2cn(CCOC)nc2C)=O)C1 C1(NC(c2ccncc2)=O)CC2(C(=O)NCC3C4COCC34)COC1C2 C#CC(CNC(=O)CCCCCN(C(=O)Cc1ccccn1)C)CC(C)(C)C CC1(C)CC2(CC(C(N3C(CNC(c4ccnnc4)=O)CC4COCC34)=O)C2)C1 C1(C2=CCCCCC2)(C(=O)NCC2(F)CCN(C(C(CCC)(C)C)=O)CC2)CC1 c1(C(=O)NCC2C(NC(CC(C)CF)=O)CCCC2)cc(F)c(Cl)cc1Cl C1(CNC(C(C)Cc2ccnn2C)=O)CCN(C(=O)Cc2ccc(F)cc2)CC1 C(CC)(C(=O)NCC1(NC(c2cc(CCO)on2)=O)CC(OC)C1)SCC.C1(C)CC1 C1(NC(c2c(C)noc2)=O)CC(F)CN(C(c2ccc(NC(N)=O)cc2)=O)C1 N1(C(COCC#C)=O)CC2C3CCC(C2C1)N(C(c1ccccc1CO)=O)C3 n1(CC(=O)NC2CN(C(C(C)P(C)(C)=O)=O)C(CO)C2)cc2ccccc2n1 N1(c2cccc(S(=O)(=O)NCCN(OC)C)n2)CCc2ccc(C#N)cc2C1 c1(C(N2CCC(F)(CNC(C3(C)CCC(=O)NC3)=O)C2)=O)c[nH]c2cnccc12 N1(C(Cn2ccc(C)n2)=O)CCC(C)(C)C1C(=O)NCC1(CN(C)C)CC1 Cc1nc(C)c(CC(N2CCCC(C)(NC(=O)C(C)C3CCCO3)C2)=O)c(O)n1 c1(CNCc2ccc(C3CCN(C)CC3)cc2)cc2c(Br)cccc2s1 C1(NC(=O)CCOC2CCC2)C=CCN(C(C2CCC2)=O)C1 c1(CNC(C2(C)CCCN2Cc2nc(Cl)ccc2F)=O)ccc(F)c(C#N)c1 C(=O)(C1CCSc2ccccc21)NCC1(NC(CCC(C)(C)O)=O)CCCC1 c1(C(N2CCC(F)(CNC(C3(C(N)=O)CCC3)=O)C2)=O)ccc(Br)c(N)c1 C1(C(=O)NCC(CC(C)C)C)CC(NC(=O)C2=CCN(C)C2)C12CCC2 Cc1nccc(C(=O)NC2CC2CNC(=O)CCCSc2ccccc2)n1 N1(C(C(C2CN(C(CCCCCC)=O)C2)OC)=O)CCCC(C2(C)CC2)C1 c1(C(=O)NC2(CC=C)CN(C(=O)CN3CCCCC3)C2)coc2c1CS(=O)(=O)C2 n1(CC)c(C)cc2c1CCCC2NC(c1c(C)oc(C)c1C)C C1(NC2CCCC2)Cc2ccccc2C1.c12cc(C)nc(n1)NC(C)(C)CCN2C c1(C(N2CCCC(NC(c3ncc(Cl)nc3Cl)=O)CC2)=O)[nH]cc2c1CCCC2 c1(C(N2CCOCC(NC(C=CC(C)C)=O)C2)=O)nnc(O)c2ccccc12 C(=O)(C1CCc2c[nH]nc21)NCCCCNC(c1cncc(OC)c1)=O c1(CC=C)cccc(C(=O)N(CCC(=O)NCC2C3COCC23)CC)c1 C12(C(=O)NC3C(C(N(C4CC=CC4)CC)=O)CC3)CCC(CC1F)C2 C1(C(N2C(CCC)COCC2)=O)CC(C)(C)CCN1C(=O)Cn1ncccc1=O C1(CCC)(NC(C(CC#C)C)=O)CCN(C(C2CN(C(C)=O)C2)=O)CC1 N1(C(c2c(C)nn(C)c2)=O)CCOC2(CCC(NC(=O)Cn3cncn3)CC2)C1 C(=O)(CCCC(F)(F)C(F)(F)F)NC1COCCN(C(C(C(C)C)C#N)=O)C1 c1(CNC(=O)NCC(CC(C)O)C)coc2c1CCCC2 C1(C(N2C(C)CC(NC(COC(C)C)=O)C2)=O)CCCCC1(F)F C#CCN(OC)C(=O)C(O)CNC(=O)CCC1CC1(F)F C12(CCNC(C(F)=C(C)C)=O)CCC1CN(C(C1(c3cccs3)CC1)=O)C2 c1(CC)cnc(C(=O)NCC(C2CC2)NC(c2cc(COC)cs2)=O)cn1 C1(C(=O)NC(CC(C)(C)OC)C)CN(C(C2CCC2C#N)=O)CC12CCC2 CC(CC(=O)NC1(C2CCCO2)CC1)(C1CC1)NC(=O)CC1(C(F)(F)F)CCC1 c1(N(C)Cc2cscn2)[nH]c(=NC2CCCC(O)C2)nc2c1cnn2C C1(C)(CC)CCC(c2nnnn2Cc2ccccn2)(NCC2CCCO2)CC1 c1(C(=O)NCC(C)NC(=O)Cc2ccc3sccc3c2)cc(S(N)(=O)=O)co1 c1(OC)cnc(NC(c2ccsc2CSC(C)C)=O)nc1CO C(=O)(C(C)(C)C#N)NC1C(NC(C(C)CSCc2ccccc2)=O)C1 C(CCCN=[N+]=[N-])NC(C(c1ccco1)NC(COCCSC)=O)=O C1(CNC(C=NOC)=O)CC(C)(C)CN1C(=O)CS(N)(=O)=O c1(OC)cc(C(c2nnnn2C)NCCc2ccncc2F)ncc1C O=C(C1CCc2cccc(O)c21)NC1CCCC1NC(C1CC2(C1)CC(O)C2)=O C1(C(=O)NC2C(NC(c3c(C(N)=O)cccc3)=O)C2)COc2cc(F)ccc2O1 CCC1=NOC(CC(=O)NCCN(CC(C)O)C(=O)C=C(C)c2ccco2)C1 C1(C(=O)NCCC(=C)CNC(=O)Cc2cc(C)sc2C)CCc2nc(C)[nH]c2C1 C1(c2nnnn2C2COC2)(NC(CC=C)CC)CSCCSC1 C1(C(=O)NCCCN(CCC)CCC)(NC(=O)Cn2cccc2)CC1C C1(C)(CNCC(C)CC2CC2)C(C)(C)C1(C)C C1(CCNC(c2cnc(CC(C)C)s2)=O)CCCCN1C(C1CCC=CCC1)=O CC(C)(F)C(C)(F)C(=O)NCC1CC(NC(c2cncc3ccsc23)=O)C1 N(C1CCCc2c1cnn2-c1ccccc1)C(=O)NCc1c(C)scc1 CC1COCCCN1C(=O)C(CC(N)=O)NC(=O)Cc1ccon1 C(N=c1[nH]c(=N)[nH]c(=NCC2(c3ccccn3)CC2)[nH]1)c1c(C)nccc1 C=CCC(CNC(c1n[nH]cc1CC)=O)NC(=O)CSCC(N)=O N1(C(C2(COC)CC=CC2)=O)CC(N(C)C(C2CCCO2)=O)C(C)(C)C1 c1(C(N2C(C)CN(C(C3(C)CC3Br)=O)CC2)=O)ccc2ncsc2c1 N1(C(CCCc2nc(C)sc2)=O)CC(NC(c2cc(Cl)on2)=O)C2CCCCC12 N1(C(c2cn(C(C)C)nn2)=O)CCOCC(NC(C2(CCF)CCC2)=O)C1 S(=O)(=O)(c1csc(C(=O)N(CCNC(C23CCN(CC2)CC3)=O)C2CC2)c1)NC N1(C(C2C(C)CCC2)=O)CCCC(C)(C)C1CNC(C1CCCSS1)=O C1(NC(CCSCCC)=O)COC2C(NC(C3CNC(=O)CC3(C)C)=O)COC12 c1(NC(=O)Nc2ncccc2Oc2ccc(F)cc2)cc2cccnc2cn1 c1(C(=O)NC(C)CN(C(=O)CCc2nccs2)C)sccc1S(N)(=O)=O N1(C(c2c(CC)cco2)=O)CC2CCCC(NC(=O)COc3cnn(C)c3)(C2)C1 c12c(cccc1C)C(=O)NCCSC2.C(CCO)OCCOC N1(C(C(COCC)C)=O)CC(OC)CC1C(=O)NCc1c(C)cnn1C C1(C(=O)NCC(N(C(=O)COC2CCCCC2)C)C2CC2)(CF)CCOCC1 c1(C(N2CC=CC(C(N3CC(OC)C(O)C3)=O)C2)=O)cc(O)ccc1C c1(C(CC)O)nc(-c2nnn(CC)n2)n(C2CC2)n1 c1(OC)cc(CC(=O)N(C)CCN(C(=O)C(C)(C)CF)C)cc(F)c1 c1(C(=O)NC(C(=O)N(C)CC2(O)CN(C(CC(C)C)=O)C2)C)ccc(F)cc1F S(=O)(=O)(c1ccc(NCC#CI)cc1)N(C)CC C(=O)(CCC(=O)N1CCC(O)CC1)OCCCOCCOC c1(SC)cc(C(=O)NC2CC(CNC(c3[nH]cnc3C)=O)C2(C)C)c(C)o1 C1(CC(N2C(C)(C(C)C)CC2)=O)CC(O)CN1C(=O)C(C)CC1CC1 Cc1nnc(N2CC(c3ocnc3CNC(C3CCCC3C)=O)C2)s1 N1(C(=O)NCCCCl)CC2CC1CN2Cc1ccccc1NCCCl c1(CC)cc(C)c(C(=O)N(CCCN(C)C(C2C3CC(=O)CC23)=O)C)o1 c1(C(=O)NCC(C)NC(C(CC#C)C)=O)cnc2cnccc2c1 c1(-c2c(C)noc2)cccc2[nH]cc(CC(=O)NCc3cc(Cl)cc(Cl)c3F)c12 C1(C)(C(=O)NCC2C(C)CN(c3ncnc(=N)[nH]3)CC2)CCCNS1(=O)=O N1(C(C2(Cc3ccccc3)CCC2)=O)CCC(NC(C2CC2C2CCC2)=O)CC1 c1(C(=O)NC(C(C(C)C)C)CNC(C2(CO)CCCC2)=O)ccc(C#N)cc1F c1(C(=O)NCCCN(C(C=C(CCC)C)=O)CC2CCCC2)nn(C)cc1C C=CC(C)CC(=O)NCC(CC)(CC)NC(=O)C(CCC)NC(N)=O NS(=O)(=O)C1(C(=O)NCC2(F)CCC(NC(C3CCNC3=O)=O)C2)CCCC1 N1(C(CC)=O)CC2CN(C(c3cc(C4(C)CC4)ccc3Cl)=O)CC2C1 C(=O)(C1=C(Cl)CCOC1)N1CC(CCNC(c2ccc(F)s2)=O)OCC1 C(=O)(C1=CN=C2N=CNN2C1)N(C1CCN(C(C2CC=C(C)CC2)=O)C1)CC C1(C(=O)NCC(C(CC)C)C)CC2CN(C(=O)C=Cc3cc[nH]c3)CC2C1 C(=O)(C(C)(C)C(C)O)N1CC(C(C)NC(C2(C)CC(C#N)C2)=O)C1 Cn1c(C(N2CC3CC2C3CNC(C2C=CC=CC=C2)=O)=O)cccc1=O c1(C(=O)NC(CNC(CC2(C=C)CCC2)=O)CO)ccc(O)nc1Cl C=CC(CCC)CC(=O)NC(c1ccnn1C)C(=O)NCC1([Si](C)(C)C)CC1 C1(C(N2CCC(CNC(c3cc(F)n[nH]3)=O)C2)=O)CC2CCC(C1)S2 c1(C(N2C(C(C)NC(CC)=O)CCC2)=O)cnc2ccncc2c1 CCCC(O)C(=O)N1CCC(C(=O)NCc2c(C)noc2CC)CC1 N1(C(=O)OC(C)(C)C)CCC(NC(=O)CC2CC2(C)C)C(O)C1 C(CCC(C)(C)NC(=O)C(C1CCOCC1)C)NC(c1nc(C(C)C)sc1)=O C1(N(C)C)COCC1(c1nnnn1C(C)(C)C1CC1)NCC1(CC2CCC2)CC1 N1(CC(=O)N(CCC(=O)NCC2(CF)CCC2)C2CC2)C(=O)CNC1=O CN1CCCC(CNC(=O)C(CC2CC2)c2ncco2)C1c1ccccc1 c1(C(=O)NCC(CC=C)NC(=O)C(F)(F)CC2CCCO2)cn(C)nc1C C1(N(C(=O)CCCNC(=O)C(CO)NC(N)=O)C)CCC(C(C)(C)C)CC1 Nc1ncnc2c1ncn2CCNC(c1ccccc1-c1ccc(F)cc1)=O C(CC1=CCN(C(=O)CN2CCOCC2)CC1)NC(=O)CC(C1CC1)C1CC1 c1(OCC(=O)NC(CN(C(C(C)OCC#C)=O)CC)C)cccc(Br)c1 c1(C(=O)NC(c2cncnc2)(C)C)coc(CNC(=O)CCCN2CCCC2)n1 c1(C(N2CC3CC(NC(c4c(C)scn4)=O)C3C2)=O)cncc2c(O)nccc12 S(=O)(=O)(c1ccc(Cl)nc1)N1C(CC#N)CN(C(c2ccc(O)cc2)=O)CC1 C1(C(=O)NCC(C)(C)NC(C2CCN(CCC)CC2)=O)CCc2n[nH]cc2C1C c1(C(C(=O)NCC(C)N(C(=O)CC2CCC(O)C2)C)(C)C)cc(Cl)ccc1F N1(C(C(CC=C)c2ccccc2)=O)CCC2C(NC(c3ccsn3)=O)C2C1 C1(COC)(NC(=O)CC=Cc2ccc(C)cc2)CCCN(C(c2cnsn2)=O)C1 C1(C(=O)NCC(C)CN(C)C(C2(O)CCCC2)=O)C(c2ccccc2)C1(F)F N1(C(c2ccn(C(C)(C)C)c2)C(=O)Nc2ccccc2)Cc2ccc(Br)cc2C1 c1(OC)ccc(C(N2CC(CC(C)NC(=O)CCc3cnc(C)o3)C2)=O)c(F)c1 n1(C(C(=O)N(C(CC)C)CC(=O)Nc2snc(O)c2Cl)C)c(C)cc(O)cc1=O CC1CCC(F)(C(N2CCC(NC(c3nncs3)=O)C(C(N)=O)C2)=O)CC1 N1(C(C)C(=O)N(CCCN(C(=O)C(C)Oc2cccnc2)C)C)CCCCC1=O N1(C(c2c(CC)csc2)=O)CCN(C(=O)Cc2cccc(Cl)c2Cl)CC(O)C1 N1(C(C2NC(=O)CC(C)C2)=O)CC(C)N(C(c2cnn3c2OCC3)=O)C(C)C1 n1(C(=O)NCc2cn(C3CN(C(C(CC)OCC)=O)C3)nn2)ccc([N+](=O)[O-])n1 C(=O)(C(F)CC(C)(C)NC(=O)CC1CSCCO1)N1C(CC(=O)NC)CC1.OC Nc1ncc(Br)nc1C(=O)NCC1CCC(NC(C2CN(C3CCC3)C2)=O)C1 C(=O)(C1=CCCN(C(=O)OC(C)(C)C)C1)NC(CNC(C(C(C)C)C)=O)C N1(C(c2cnn(CC)n2)C(=O)NCCCF)CCc2oc(C)nc2C1 c1(C(N(C(C)C(C)(C)C)C)=O)cc(CNC(=O)CC(C)C2CCCO2)nn1C C1(C)(C(N2CC(C(=O)N(C)CCn3cc(C)cn3)(SC)C2)=O)CC2CC2C1 C1(NC(C(C)n2ccnc2)=O)CCC(C(=O)NC2CCCC2C(N)=O)CC1 Cc1ncnc(C)c1CC(=O)NC(CO)C(C)NC(c1ccc(N(C)C)nn1)=O C1(Nc2c(OC(C)C)cccc2)C2CCC1N(C(=O)COC(C)C)C2.C1C(=O)O1 N1(C(C2CCCN(C(C)C)C2)=O)CCC(C)N(c2cnc(C#N)cn2)CC1 N1(C(c2ccnc(Cl)c2F)=O)C2CCC1CC(O)C2.C123CC(C1)(C2)C(=O)N3 c1(C(=O)NCC(=C2CN(C(c3cnc[nH]3)=O)C2)F)cnn2ncccc12 C1(NC(CC2CN(C)C2)=O)CC2CCCC(C1)N2C(c1csnn1)=O C1(NC(c2c(C(C)C)c[nH]c2)=O)C2CC(NC(C3(C)CNC(=O)C3)=O)CC12 CC(C)CC(C(=O)NCC(O)CCNC(c1ccc(C#N)o1)=O)C(N)=O c1(C(CC)NC(=O)C(=O)Nc2nccn2Cc2cccc(Cl)c2)ccccc1Br c1(OC)cc(C)c(C(=O)N(C)CC2CCN(C(c3cnoc3C)=O)C2)cn1 C1(CCC)CN(C(=O)CC2OCCO2)CC1C(N1CC2(CC2)C1)=O C1(CC(=O)NCC2CCCC2NC(c2cncs2)=O)CC(=O)NC1=O C(=O)(CC(C(C)C)C(C)C)N1CC(OC)C(NC(=O)CCC2CCN(C)CC2)C1 c1(C(=O)NC2CCCC(NC(=O)COC(F)F)C2)ccc(C(C)(F)F)cn1 Cc1cn(C(C)C)cc1C(=O)NCCCC1(NC(=O)Cc2ccc(F)cn2)CC1 C1(C2CCN(C(C3CSCCS3)=O)C2)(NC(=O)C(F)CC2CC2)CC1 c1(C(=O)NC2CN(C(C)=O)C(C)C2)coc2c(C)cccc12 C1(CNC(c2cc(OC)n[nH]2)=O)CC12CCN(C(=O)CC1CSCCS1)CC2 CS(=O)(=O)c1ccc(C(=O)NCC2(F)CC(NC(=O)CCNC(N)=O)C2)[nH]1 O=C(CCCCCO)NCC1(N2CCOCC2)CCOCC1.C12(CC1)C(=O)N2 N1(C(C2(CF)CCN(C(C(C(C)C)O)=O)C2)=O)CC2(COC(C)(C)C2)C1 c1(C(N(CC(C)NC(C2CCC2C(F)F)=O)C)=O)c(C(F)(F)F)ncn1O N1(C(COCCCC)=O)CCN(C(C2(C#N)CC3CCC2C3)=O)CC(O)C1 CC1=CC(C)CN(C(C2C(C)CN2C(C2CCN(C)C2)=O)=O)C1 Cc1cccnc1CC(=O)NC(C1CCCN1C(C1CCC(C(N)=O)C1)=O)C C=CC1(CC(N2CCOC(CNC(=O)CCOCCOC)C2)=O)CCCCC1 N1(CC(=O)NC(C#C)C)CCN(C(c2cnccc2OC)=O)CC1 C1(NC(CSc2cccc(C)c2)=O)CS(=O)(=O)CC1NC(c1cc(C#N)on1)=O c1(OC)ccc(C)c(C(N2CCCC(NC(=O)CCc3nncs3)C2)=O)c1N N1(C(c2ccc(CC)cc2N)=O)CCN(C(c2cn(CCO)nn2)=O)C(C)C1C N1(C(c2ccc(C(C)C)cc2)=O)CCC2CCC(C1)N2C(C1(CO)COC1)=O C1(CC(=O)N(CCNC(=O)COCC2CCCC2)CC)COC2CC1C2 Cc1ccccc1C(C)CC(=O)N1CC(N(C)C(c2cc(O)n(C)n2)=O)C1 c1ccc(NC2(CNC3CCCCO3)CCC2)cc1 c1(C(=O)NCC(C2CC2)NC(C2CC(SC)C2)=O)ccc(C2CCC2)[nH]1 c1(C(=O)NCCOC(C)(C)CNC(=O)COCCF)cccc(F)c1O C1(C(=O)NCCC(C)NC(c2cnn3c2OCC3)=O)CC(S(C)(=O)=O)C1 C=CC1(CC(=O)NCCc2cccnc2F)CN(C(C2C(C)C2C)=O)C1 c1(C(N(C)CC2N(C(CCC)=O)CCCC2)C)nc(C(F)(F)F)cc(C)n1 C#Cc1cnc(C(=O)NC2(C)CC(NC(C3(CO)CC4CCC3C4)=O)C2)c(C)c1 C1(C(=O)NCC(CNC(COCCC)=O)F)CCSCC1 N1(C(C23N(C(C(N4CCOCC4)C)=O)CC(C2)C3)=O)CC2C3CCC(O3)C2C1 C(=O)(C#CC1CCCCO1)N(C1CCCN(C(c2c(C)coc2)=O)CC1)C c1(C(C)NC(C2CCCN(C(CC(C)(C)OC)C)C2)=O)nc2ccc(C)cc2[nH]1 CC1CCN(C(C2(C)C(C)(C)C2(C)C)=O)CCN1C(=O)CN(C1CCSC1)C N1(C(CN(C(C(C)C)=O)C)=O)CC2(CC2)CC1CNC(C1CC12CCSCC2)=O c1(NC(C2C(C(=O)NC3(C(=O)OC)CC3)C2)=O)cccc(C(F)(F)F)c1N CCC(CN(C)C)CC(=O)NCC(C)(C)NC(=O)C=Cc1cncs1 c1(C(=O)NC(CC)CNC(=O)C=C2CCC(C)CC2)cncc2ccccc12 CN1C(=O)NCC1C(N1CC2C(NC(C3CSC3)=O)C2C1)=O C(CCCC(=O)N1CCC(OC2CC2)C1)NC(=O)C=CC(=O)NC1CC1 N1(C(c2c(OC)n[nH]c2)=O)CCC(C)C1CNC(=O)COc1cccnc1 CC(C(C)C(=O)N1CC2(CC(NC(c3cc(C4CC4)[nH]n3)=O)C2)C1)C(C)(C)C c1(C(N2CCC(N(C)C(c3ccnn3C)=O)CC2)=O)cccc(N)c1C(F)F C1(N(C(C2CCCC2)=O)CC)CCCN(C(=O)CC2CCS(=O)(=O)C2)CC1 CCCC(C#N)C(=O)NCCCCc1cn(-c2ccc(C)c(Br)c2)nn1 c1(C(N(CCNC(C(F)(F)C2(OC)CCC2)=O)C2CC2)=O)cnc2cccnn12 C1(NC(c2cncc(C)n2)=O)CC2CN(C(C3CN(C)CC(C)O3)=O)CC12 c1(C(N2C(CNC(C3N(C(C)(C)C)CC3)=O)CC2)=O)cc2c(s1)CCOC2 C1(CC(=O)NC2(C)CC(NC(c3c(C)nc(C)n3O)=O)C2)CS(=O)(=O)CCN1C c1(OC)cccc(C2CCN(Cc3cc(Cl)ccc3N(C)C)C2)c1F c1(C(=O)NCC#CCNC(C(C)=CC2CC2)=O)nnc(O)c2ccccc12 CN1CCc2[nH]nc(C(=O)NC3C=CC(CNC(=O)C#CC4CCCO4)C3)c2C1 c1(C(N2CCC3(CCC3)C2)=O)csc2c1CCN(Cc1cccc(F)c1O)C2 C1(CC(=O)NCCN(C2CCCC2)C(c2cc(Cl)ccn2)=O)CCS(=O)(=O)C1 c1(-c2cncc(C3CCN(C(CCOCC)=O)CC3)c2)ccc2sc(C)nc2c1 C(C(C)(C)C(=O)NC1CC(CCOC)C1)N(C(=O)Cn1cnc(=N)[nH]1)C Cc1nc(C(N2CC(O)(C(F)C(=O)N(c3ccccc3F)C)C2)=O)sc1C C1(NC(C2CN(C(C(C)=C3CC3)=O)CC(C)O2)=O)CC2(CCCCC2)C1 N1(C(C=CC(C)NCCCCN2CC(C)OC(C)C2)=O)Cc2ccccc2C1 N1(C(c2nc(CCC)sc2)=O)CCCC(C2(NC(C3(OC)CCSC3)=O)CC2)C1 N1(C(C2(COC)CC2)=O)CCC(CNC(=O)CCN(CC(C)C(C)C)C)C(O)C1 O(NC(=O)C(F)C(C)(F)F)C(C(=O)NCC(NOC)=O)CC(C)C c1(CCC)nc(NC(=O)CCON)cc(C)n1 CCC(CC)(CC)C(=O)NCC(C)NC(c1ccc(CN2CCCC2=O)cc1)=O C1(NC(C(CCC)C)=O)CC2CCC(C1)N2C(C)C(=O)N(C1CCCCC1)C C(N=c1cc(C(F)F)nc[nH]1)C1CC(C)N(C(c2csc(Cl)c2)=O)C1 Cc1cccc(C(N2CCOC(C(=O)NC(c3ccc(Br)cc3)CO)C2)=O)c1O C1(CCNC(C2C(C)CC(C)O2)=O)CCCN(C(c2nnn(C)c2N)=O)CC1 C(=O)(CCCCC(C)(C)OC)NCCCN(C(C(C(=O)OC)OC)=O)CCO C1(N(C(C=C(C)C(F)F)=O)C)CCCN(C(C2CC(N3CC(O)C3)C2)=O)C1 c1(CC)cc(C(=O)NCC2(NC(c3ccc(-n4cncn4)cn3)=O)CC2)sc1C O=C(CC(F)(F)C(F)(F)F)NC1CCC12CN(C(c1cccc3[nH]ncc13)=O)C2 n1(CCC(N2CCC(N(C)C(c3nocc3Br)=O)C2)=O)ncc2c1CCCC2 C(=O)(CCCCN=[N+]=[N-])N(C1CC(C(=O)NCC2CCN(C(C)C)C2)C1)C N1(C(C(CSC)O)=O)CCC(C(O)CNC(C2CC(F)(F)CS2)=O)CC1 Cc1ccc2sc(N3CCC(CNC(=O)C(C)O)C(F)(F)CC3)nc2c1C Cc1nn(CCO)cc1C(N1CCN(CCCF)CC1)C(=O)NCC1CC1 c1(C(N(C(c2cnn(C3CCC3)c2)C(=O)NC)C)=O)csc2cncn12 C1(CC(F)F)(C(=O)NC2CC(CC(C)(C)C)C2)CCNC1 c1(CNC(=O)NC2(CCO)CCCOC2)ccc(Cl)c(F)c1F c1(CNC(C(N2CCCC(O)(CN(C)C)C2)=O)=O)cccc2c1C(=O)OC2 C(N=c1[nH]c(N2CCOC(CCF)C2)nc2c1COC2)C1(C)COCCO1 CCCC(O)CCNC(C1(CNC(c2sccc2F)=O)CC(C)(C)C1)=O N1(C(c2cnn(CC)c2C(F)(F)F)=O)CCN(C(=O)CC(F)(F)F)CC(CO)C1 C(CCC(C)(C)C(=O)NCC1(O)CCCC1(C)C)NC(C(C(=O)OC)C)=O C1(O)(C(=O)NCCN(C(C(C)CC(F)F)=O)CC2CC2)CN2CCC1CC2 c1(N2CCC(CNC(C(CC)(CC)CO)=O)C2)ncc([N+](=O)[O-])c(=N)[nH]1 N1(C(C(C(C)C)OCC)=O)CCC2CCC(C1)N2Cc1ccc(C#N)cc1F Cc1ccc(F)cc1C(=O)NC1CC(C(N2CCOC(CC(N)=O)C2)=O)C1 c1(C(=O)NC2C(OC)CC2)cn2c(n1)CN(C(c1c(F)ccc(Br)c1Cl)=O)CC2 c1(CNc2cccc(COC(c3c(C)coc3C)=O)c2)ccc2c(c1)CCCO2 C(=O)(C1=CCCCC1C)NC1CC(C)(CNC(Cc2c(C)cco2)=O)C1 CCC(CC)C(C)C(=O)N1CCC(C)(CNC(c2ncccc2SC)=O)C1 CC1N(C(C2(C(C)NC(c3ncccc3O)=O)CC2)=O)CCOC1(C)C c1(SC)ccc(CC(N2CC3CC3(CNC(=O)C=Cc3cc[nH]n3)C2)=O)cc1 c1(C(=O)NCC(O)CCNC(c2ccc(O)nc2Cl)=O)ccc2c[nH]nc2n1 C12(C(=O)NC3CC(C(C(=O)NCC(CCOC)O)F)C3)CCC(CC1)C2 CCCCCC(C(C)(C)C)NCc1cnc(CCC)s1 c1(C(=O)NCCOC2CN(C(C3C(OCC)C3)=O)C2)cc2n(n1)CCCO2 c1(C(N(C)CCNC(C2CCCC(C(N)=O)C2)=O)=O)cc(C(C)(C)C)ccc1N c1(C(N2CCN(C(CS(CCC)(=O)=O)=O)CC2)=O)cc2cccc(C)c2s1 c1(SC)ncc(C(=O)N(C2CN(C(=O)C(C)C3CCC3)C2)C)n1C c1(SCC(=O)NC(CNC2(OC)CCSC2)C)ccc(C(C)(C)C)cc1 CN1CCc2ccc(C(=O)NC3C4CN(C(c5ccc(Br)cc5)=O)CC34)cc21 C1(CC)CN(C(=O)CNC(=O)CCCc2ncco2)CC(CC)O1 Cc1ncc(CC(=O)NC2CCCC(NC(c3cc(CCO)on3)=O)C2)c(O)n1 N1(C(=O)CC2COCCO2)CCOC2(CCN(C(C3CCCCO3)=O)CC2)C1 C1(CCNC(CC2C(C)C2(F)F)=O)CCCCN1C(c1cc(C(F)F)no1)=O N1(C(=O)NC2(c3ccc(OC)c(Br)c3)CCOCC2)CCCCCCCCC1 C(=O)(CCOCCCNC(=O)C(O)C1CCCC1)NCC(=O)OC C1(C(=O)NC2C(c3n(C)ncc3)C2)CN(C(=O)C=Cc2cnccn2)C(C)(C)C1 C1(NC(CCc2cc(C)no2)=O)CC(NC(=O)CSS(C)(=O)=O)C1(C)C c1(C(=O)NCC2CCN(C(C(CC(N)=O)O)=O)CC2)[nH]nc2ncccc12 N1(C(C2(C(N(C)C)=O)CC2)=O)CC2CC2(NC(C2CCC(=O)NC2)=O)C1 C1(C(C(=O)N(C(CC=C)CC)C)Sc2cn(C)nn2)CCC2CC1C2(C)C C1(CC(N2CCC(C(C(N3CC(N(C)CC)C3)=O)F)C2)=O)CCC(=O)NC1 N1(C(CN2CCC(OCC(C)C)CC2)=O)CCc2ccccc2C1 C1(CN(C(CC2CC(SC)C2)=O)CC(=O)O)CCc2ncnc(C)c2C1 Cc1ccc(C(=O)NC2CCC2NC(c2ccccc2Cl)=O)c2c1NCCC2 Cc1cc(=NC(=O)C=CCCCNCCC2CCC(C)(C)C2)[nH]n1CCO C(=O)(C1=NOC2(CCC2)C1)N1C2CC(NC(c3ccc(C)cc3O)=O)CC1CC2 CC1(C)COC(CCC(=O)NC2CC3(C2)CC3NC(c2coc(CO)c2)=O)C1 c1(C(N(C)CC2CCN(C(CSCC#C)=O)CC2)=O)cc(C(=O)OC)ccc1Cl N1(C(c2c(CNC(C3(CC#C)CCOC3)=O)ocn2)=O)CCCC2CC12 C(CCCC)(CC=O)CC=C1CCN(C)C1.C(C(=O)N)SCC#C C1(NC(CC2(CSC)CC2)=O)C(C)CCN(C(c2cc(Br)co2)=O)C1C C(C(=O)Nn1cnn(CCOC)c1=O)N(C(=O)CC1CCOC1)CCC Cc1nc(Cl)sc1C(=O)N(C1CCN(C(c2nccnc2Cl)=O)C1)C C12(C(=O)NC3CC(C(N4CC(C(F)(F)F)C4)=O)C3)CCCCC1C2 c1(C(=O)Nc2nccc(OCCC)n2)cc(N)cc(F)c1.C12CCCC(C1)N2C N1(C(C(CCC)OC)=O)CC2CC(CNC(C3(N(C)C)CCC3)=O)C2C1 CC(Cc1ccco1)C(=O)NCC1CC(CNC(C2CCCN2C)=O)C1 c1(COC)cccc(NC(=O)NCC(c2cccc(OC)c2)SC)c1 c1(C(N(c2cccc(NC(=O)C(F)(F)F)c2)C)=O)cccc(N=c2nn[nH][nH]2)c1 N12C(CCC1(C)C)C2.C(CC#N)NC(=O)NCCN(S(C)(=O)=O)C c1(C(N2CCC(C(=O)NCCC(C)(O)C3CC3)(CC)C2)=O)ccn2cncc2c1 n1(CC)ncnc1C(N1CC(O)(CCNC(C2(C3CCCO3)CC2)=O)C1)=O CC1(C)CC(=O)NCC1C(=O)NCC=CCNC(c1ocnc1C1CC1)=O c1(C(=O)NC(C(=O)NC(C#C)C(C)C)CO)cnn(C)c(=O)c1 c1(CC)noc(CC)c1CC(N1CCC(NC(C2(CO)CCC2)=O)C1C1CC1)=O C1(NC(c2nc(COCC)sc2)=O)CC12CCN(C(C1CC13CCC3)=O)C2 CN(C)S(=O)(=O)NC1CC1NC(=O)C(c1ccc(F)cc1)O C(CC(C)(C)C(=O)NC1(C2CCCN2C(c2ccc(C(=O)OC)s2)=O)CC1)OC N1(C(C(C2CCCCC2)OC)=O)CCCC(CC(N2CCC(C(C)O)CC2)=O)C1 O=C1Cc2cnc(N3CC4CC4(C(=O)Nc4cc(Br)ncc4F)C3)nc2N1 CCCCCC(O)C(=O)NCC12CCC(CC1)N(C(=O)CC(C)(C)O)C2 c1(C(N(CC(C)NC(C(C)C2CCC2)=O)C)=O)sc(Cl)cc1Br C1(CC(C)C)CCCCN1C(C1(C(F)F)CCCO1)=O c1(C(=O)NCC2(C)OCCN(C(C(C)OCOC)=O)C2)cccc2c1CC(=O)N2 c1(C(N2CCC(NC(c3nc(C)oc3)=O)C(F)C2)=O)[nH]nc([N+](=O)[O-])c1Cl C1(CCCC)CCCN(C(c2ncoc2C2CCCNC2)=O)C1 Cc1c(C(=O)NC(CO)C(C)NC(c2cc(C3CC3)no2)=O)nn2ccccc12 c1(C(=O)NCC(=O)NC)ccc2c(n1)CCN(C(=O)C(O)C(C)C)C2 c1(OC)cncnc1C(=O)N(C)CC1(O)CN(C(=O)C(C)(C)c2ccno2)C1 C1(CNC(C(CC)OC)=O)CC(C(=O)NCc2nc(C)sc2C)=NO1 C1(CC(=O)NCC2COCC2O)CCN(c2ncccn2)CC1 Cn1cc2c(n1)CC(C(=O)NCC(C(C)(C)C)NC(=O)Cc1ccoc1)CC2 c1(N(C)CC2CCN(C(=O)CC3CCCOCC3)CC2)nc2ncc(Cl)cc2o1 C1(CC#C)(C(=O)NC(C(C)OC)CO)CCN(C(=O)COC2(C)CCC2)C1 C1(CCC(=O)N(CC(CC)NC(=O)C(C)(C)n2cnnn2)C)CC(C)(C)CO1 c1(C(=O)NCCC(C(C)C)NC(CSCC(C)C)=O)c(N)nn2ccccc12 c1(OC)ccccc1C(C(C)NC(=O)C(=O)NCC1CC1)NC(=O)CCC1CC1 CC1(C(N2CCC2C(=O)NC2COC(C(F)F)C2)=O)CCCCO1 C(=O)(CCC(C)(C)C)N1CCC(CC=C)(NC(C2CC(=O)N(C(C)C)C2)=O)C1 N1(C(c2ncc(OC)nc2)=O)CC=C(C(=O)NCC2(O)CC(O)C2)CC1 c1(NC(C(C)OC(=O)C(=O)Nc2ccccc2)=O)ccc(Cl)cc1NCC1CC1 CCC(C)CC(C(=O)NCCC1(OC)CCC1)NC(c1ncccc1CC)=O C=Cc1ccc(C(=O)NC(CN=[N+]=[N-])C(=O)NCCC2CCCC2(C)C)cc1 CC(CC(=O)NC1CC2CC(NC(=O)CCCN3CCCC3)C2C1)C(C)(C)C C(N=c1[nH]c(=NCc2cncs2)c2ncccc2[nH]1)C1CCCC(C)O1 N1(C(c2n(C)nc(O)c2)=O)CC(N=[N+]=[N-])CC1C(=O)NCCCCCN=[N+]=[N-] c1(SC)nc(C(=O)NCCCCCNC(c2nn[nH]c2Cl)=O)c2ccccn12 CC(F)(F)C(F)(F)CC(=O)N1C2CCC1CN(C(=O)C(C)(C)C13CC(C1)C3)CC2 c1(NC(C(N2CC(O)CC(C)C2)=O)=O)cc(F)c(Br)cc1F N1(C(C(=Cc2cnc[nH]2)C)=O)CCCC(O)(CNC(=O)CN2CCS(=O)CC2)C1 N1(CC)CCCC1CC(=O)NCCC(C)NC(c1nc(C)cs1)=O N1(C(C2(S(C)(=O)=O)CCC2)=O)CCN(C(c2ccc(O)cc2F)=O)CC12CCC2 O=C(CC1OCc2cc(Cl)ccc21)NC1CN(C(=O)C=C2CCC2)C2(CCC2)C1 C1(NC(c2cc(CCNC(=O)CC3OCCO3)on2)=O)CCCC1C1CC1 N1(C(c2n(C)cc(F)c2)=O)CC(NC(c2ccnc(Cl)c2)=O)C(C#N)C1 c1(OC)cc(C(=O)NCCN(CC(C)O)C(=O)Cc2cn(C)nn2)cc(Cl)c1 c1(C(=O)NC2CCC(NC(c3ccn(CC)n3)=O)C2)noc(C)c1C(=O)OC C(=O)(CCCCCC#N)NC1CCN(C(c2cnc(C)c(N)c2)=O)CC1C c1(C(N2C(CCNC(C(COC)C)=O)CCC2)=O)cccc(S(=O)(=O)CC)c1 c1(CCC(N2CC(C(=O)OC)C(N)C2)=O)c(I)ccnc1O C(CC)(CCCC(=O)NCc1nn[nH]c1C1CC1)NC(CSCCC)=O c1(C(C(N2CCC(NC(CC(=C)Br)=O)C2)=O)OC)c(F)cccc1F C(=O)(CC(C(F)F)NC(C1(C)CCN1C(=O)C(=O)NC)=O)OC C1(n2cc(-c3c(C)nn(C)c3)nn2)CCN(C(=O)Cc2cccs2)CC1O N1(C(c2ncn(CC)c2)=O)CC=C(C(=O)NC(CO)CCC2CC2)CC1 Cc1cn(C)cc1C(=O)NCc1cccnc1CNC(c1ccc(=N)[nH]c1)=O CC1CC(NC(=O)CN(C)C(c2ccoc2)=O)CN1C(=O)C=Cc1cnn(C)c1 C(=O)(C1CCCn2cnnc21)NCC(CO)NC(CCNC(=O)NC)=O C1(NC(C2(SCC)CC2)=O)CN(C(=O)CNC(c2ccnc(O)c2)=O)CCC1C N1(C(C(CC=C)C)=O)CCC2(CC1)CCN(C(=O)C=C(C)C1CCCCC1)C2 Cc1nc2c(N3CC4CN(S(=O)(=O)CCCl)CC34)ncnc2[nH]1 C(C)(CO)(C(=O)NC(CCC)CCO)NC(c1ccc(CC)s1)=O C1(CNC(C2(C=C)CCCC2)=O)CCC2(CCC2)C1NC(c1cccnc1O)=O c1(C(=O)NCc2ccc(Cn3cc(Br)cn3)o2)csc(-c2ccncc2)n1 c1(OC)cc(OC)nc(CC(N2CCC3C(NC(c4cn(C)cn4)=O)CC23)=O)n1 C(CN=c1ccc([N+](=O)[O-])c[nH]1)N(C(NNC(C)=O)=O)CCO C(=O)(CC(C)(C)C)ONCC(C)(CC)NC(C(F)=CC)=O C1(NC(CCC=C)=O)CCS(=O)(=O)C12CN(C(c1c3c(nn1C)CCC3)=O)C2 C1(C(=O)NCC(C)CN(C)C(c2ccco2)=O)CCS(=O)(=O)C1.C1(=O)C(C)(C)N1 N(C(=NCCCc1nnc2ccccn12)NC1C(C)(C)C1(C)C)C(CC)C c1(C(=O)NCC(CCNC(c2cc(C)nc(C)c2)=O)O)nccc2nn[nH]c12 N1(C(CCC2N(C)CCC2)=O)CC2CC1CN2c1nc(C2CCCCC2)ns1 C=CCCC(C(=O)NC1(c2ncc[nH]2)CC1)NC(C1CC(=O)N(C)C1)=O CN(C)S(=O)(=O)N(C)CC(N1CCC(CO)C(NC(=O)C2=NOCC2)C1)=O c1(C(N2C(C)(OC)CC2)=O)ccc(Cn2nccn2)cc1 N1(C(c2ccc(C=C)cc2)=O)CCCC2CN(C(c3cccc(=O)n3C)=O)CC12 C1(COC2CCN(C(C3(C)N(C(CSC)=O)CC3)=O)CC2)CCC(C2CC2)C1 C1(CNC(=O)CC2CC=CC2)CC2COCC2N1C(c1ccc2cc[nH]c2c1)=O C(C1CCCCCC1)=CC(=O)N(CC(C)NC(c1cnn(C)c1)=O)C N1(C(C(C)Cc2ccco2)=O)CCC2(C1)CN(S(=O)(=O)c1ccn(C)n1)C2 c1(OC)ccc(C(=O)NC2CC2NC(C2(F)CCC2)=O)c(Br)c1 N1(C(CC(C=C)C)=O)CCC(NC(c2cn(C)nc2C)=O)CC1c1ccccc1 c1(N2CC(CC)SCC2)ncnc(NC(COC(C)C)C(C)(C)C)c1C C(=O)(CCC(C)(F)F)N1CCC(CN(C(c2cc(C)nc(C)n2)=O)CC)CC1 C=CCC(C(=O)NCC(CO)NC(=O)CCC1CCCCCC1)c1ccccc1 c1(C(=O)NC2CC3C(NC(=O)CCn4ccnn4)C3C2)ccnc2ccsc12 c1(CC(=O)NC2CCCN(C(c3cccn3C3CC3)=O)C2)c(Cl)ccc(O)c1Cl c1(NC(C2(c3ccc(F)cc3Cl)CCC2)=O)cnc2c(c1)CCC2 C1(C(=O)NCCC2CCN(C(C3(CCC)CCC3)=O)C2)CC2COCC(C1)C2 N#Cc1ccc(CCC(=O)OCC(N2CCN(C(CCCC)=O)CC2)=O)c(F)c1 C12(CNC(c3cc(Cl)cs3)=O)CCCC1CCN2C(=O)CC(C1CC1)C1CC1 CCCCCCC(F)C(=O)NC1CN(C(=O)Cn2cc(F)ccc2=O)CC1F N1(c2ccccc2)CCN(C(=NCCc2ccccn2)NCCC2CC2)CC1 c1(C(=O)OCC)ccc(C(N2CC3C(C2)C3(C)C)C(=O)NCCOC)c(Cl)c1 c1(C(=O)NC(CCC)C(=O)NCC(C2CC2)SC)nccc(C)c1F N1(C(C2CCN(C)C2)=O)CCOCC(C)(CNC(=O)C(C)(C)c2cccnc2)C1 C(CC(C(=O)NC1(CCNC(=O)CCc2cn(C)nc2C)CCC1)N(C)C)SC N1(C(C(C)OCC(C)C)=O)C2CCC1C(CNC(=O)Cc1ccsc1Cl)C2 O=C(C1=CSCCO1)NC(C1CCCCCC1)CO Cc1ccc(C)c(C(=O)NCC2CCN(C(=O)C(O)Cc3ccccn3)C2)c1 c1(C(=O)NC(C)CN(C(=O)CCSc2ccc(Cl)cc2)C)cccn(C)c1=O c1(C(=O)NCc2c(=N)cc[nH]c2)cnn2cnnc2c1 C12(C(=O)NC3C(C)CN(C(=O)CCC(C)(C)C#N)C3)CCCC1CC(F)(F)CC2 CN=c1[nH]c(=NCC2C3COCC23)[nH]c(=NC2COC(C)(C)C2)[nH]1 Cc1ccc(NC(=O)CCNC(=O)C(C)N(C)Cc2ccc(F)nc2)cc1 C1(C(=O)NCCC)CCCN1CCC(=O)NCCC(C)(F)F C12(CC)CN(C(=O)C(C)C)C(CNC(c3coc(CC4CC4)n3)=O)(C1)C2 N1(C(C(C(C)C)NC(C2(F)CCC2)=O)=O)CCCNC(=O)C1C(C)C C(C(C)(O)CNC(c1cnn(C2CC2)c1)=O)NC(C(C1CCCOC1)OCC)=O c1(OCC)cccc(C(C(=O)NCCC2(C)CC2)N(C(C)(C)C#N)CC)n1 CN1N=C(CC(=O)N(C)CC2CN(C(c3ccc(F)c(C#N)c3)=O)C2)CC1=O N1(C(C(=O)Nc2ccc(O)cc2)C2(CC)CC2)CCCC(C#N)C1.C1CC1 C1(CCNS(CCOC)(=O)=O)CCCN(C(=O)Nc2ccn(C3CC3)n2)C1 C1(F)(CNC(=O)C=CCn2cncn2)CCCN(C(C2CCS2(=O)=O)=O)C1 C1(C)(C(=O)NCCC2N(C(c3cccc(OC)n3)=O)CCOC2)CCC(=O)NC1 c1(CCC)ccc(C(=O)N(CC(CC)NC(=O)C(C)C2(O)CCC2)CC)cc1 Cn1nc(O)cc1C(N1CC(CCCCNC(C2CCC(=O)NC2)=O)C1)=O C1(CC(N2CC3C(C(=O)OC)(C3)C2)=O)C2CCCC2N1C(=O)Cc1ncoc1C CC(C)CC(C)CC(=O)N1CCC(C(=O)NCCC2(O)CCCC2)O1 C1(CCC(=O)NCC2(NC(C3CNC(=O)N3)=O)CCOCC2)CCC(F)(F)CC1 CCCCC(COC)NC(=O)CNC(=O)CNC(c1nnn(C)c1CC)=O C(=O)(CCC(=O)C(C)(C)C)NCCN(CCC)C(c1ccc(CN(C)C)nc1)=O N#Cc1cccc(Cl)c1C(=O)OCc1ccnc(O)c1 c1(C(N(CCNC(=O)CCCc2ccc(F)cc2)C2CC2)=O)cc(Cl)ccc1F CC1CC(NC(C2COC3(CCC3)C2)=O)CCN1C(=O)CC(F)(F)F N1(C(c2c(OC)cc(F)cc2)=O)CC2CCC1C(CNC(C13CC(C)C1C3)=O)C2 C1(C)(CC)CCCN1N(CC1CCCO1)Cc1ccc2c(c1)OCO2 c1(CCC(=O)NC2CCCC(NC(=O)C(c3ccccc3)O)C2)ccc(Cl)cc1 CCC(CC)(CC)C(=O)NCC(C)NC(c1sc(-n2cccc2)nc1C(C)C)=O c1(C(N2C(CNC(=O)CCNC(C3CCC3)=O)CCCC2)=O)cc2scnc2[nH]1 Cc1nn(C)c(=O)c(C(N2CCC(NC(=O)CN3C(=O)CCCC3=O)C2)=O)c1C c1(C(=O)NC2CCCC(NC(C3C(=C)CC3)=O)C2)ccc2c(c1)CCCO2 n1(C(C)(C)C)cnc(C(N2CC(NC(=O)C(F)=CCCF)C2)=O)n1 c1(C(N(CCC(C)NC(c2cnc3c(c2)CCC3)=O)C)=O)cc2c(nn1)CCC2 C(N=c1nc(N2CCC(C)S(=O)CC2)c2c([nH]1)CSC2)c1cccc(C)c1N C1(C(=O)NC2CC(CNC(c3cnc(C(N)=O)s3)=O)CC2O)CC12CCOCC2 N1(C(CC(CC)O)=O)CCCC(CNC(c2ccc(-c3cnco3)cc2)=O)CC1 C1(C(=O)NCC(CNC(COCC(=C)C)=O)CO)CC2CC(=O)C1C2 c1(C(C2CCC2C(=O)NCC2CCCC(CC)C2)=O)snc(C)c1C(N)=O C(=O)(CC1CCc2cc(Br)ccc21)NCC(CNC(CCCC=C)=O)CO N1(C(c2cccc(SC)c2)=O)CCCN(C(=O)C(C)n2cccn2)CC1C c1(NC(C)=O)ccc(C(N2CCN(C(=O)Cc3c[nH]nc3C)C3CC23)=O)cc1C C(C)(CCNC(=O)COCC(F)(F)F)N(C(C=CCC)=O)C N1(C(c2n(C(C)C)ccn2)=O)CCC2(CCCN2C(c2cc[nH]n2)=O)CC1 C1(C(=O)NC(C(C)C)CNC(C2C3CCCOC23)=O)CC(C)(C)CC(C)(C)C1 c1(C(=O)NCCC(C(=O)NC2C(C)(C)C2(C)C)O)cc2occc2[nH]1 c1(C(=O)NCC(CNC(c2c(C)c(Br)no2)=O)C)c[nH]c2cccnc12 c1(C(=O)NCCC2CCCN2C(=O)Cc2cc[nH]n2)sc(F)cc1Br Cc1ccc(NC(=O)C(C)NCCC2CCCC2(F)F)cc1 N1(C(C(C(CC)O)C)=O)CCC2(CCN(C(=O)CN3CCc4ccccc43)C2)C1 C(C)(CN=c1[nH]c(=N)[nH]c(=NC2CCCC(CO)C2)[nH]1)n1c(C)cc(C)n1 c1(NC2(CO)CCCN(C(C3CC(CCC)C3)=O)C2)cc(C#N)nc(C)n1 S(=O)(=O)(c1cc(CNc2nc3ccc(C#N)cc3[nH]2)ccc1OC)NCC CC1CCC(C)N1CC(N1CCCC1CN(C(=O)CCSc1ccccc1)C)=O c1(C(=O)NC(CCCNC(CSCCC(C)C)=O)(C)C)ccc2occc2n1 Cc1ncc(Cl)cc1C(=O)NCC(O)CCNC(=O)C(C)Cc1ccccc1 C(CCN=C(NCc1ccc(SC)cc1)N1CCC(F)(C(F)(F)F)C1)SSC c1(NC(C(N2CC(COC)OCC2)=O)=O)cnc(OC)nc1C(F)F C1(C)(CNC(C(C)CF)=O)COCCN(C(c2cnc(=N)[nH]c2)=O)C1 C1(CC(N2CCCC(N(C)C)C2)=O)CC(C)(C)CN1C(c1c[nH][nH]c1=N)=O N1(C(=O)C=CC2CC2)CCC2(C1)c1[nH]cnc1CCN2C(C1CCCOCC1)=O c1(C(C)F)ccc(C(=O)N(C2CN(C(=O)C=Cc3ccncn3)C2)C)cc1 c1(C(N2CCC(C)C2CNC(=O)C2=CCSC2)=O)ccc2c(c1)C(=O)NC2 c1(C(=O)NCC2N(C(CCOC)=O)CC2)cccc(Cc2nc[nH]n2)c1 C1(CNC(C2OCCN(C)C2)=O)CN(C(C2CCCCCC2)=O)CCC1(F)F O=C(C1=CCCSC1)NC1CC(NC(C2CCCCN2CC(F)F)=O)C1 c1(CC(N2CCCC(NC(C(CC)OC)=O)(CC)C2)=O)noc2ccccc12 C1(C(N(C(CNC(c2c(F)ccc(C)c2)=O)C)C)=O)CCN(S(=O)(=O)N(C)C)C1 c1(CNC(N2CCC(CO)C2)=O)nc2ncc(Br)cn2n1 c1(C(C)C)ccc(C(N2CCC(CF)(NC(C3CCCC3)=O)C2)=O)c(O)c1.CO C1(C(=O)OCC)C2CC(CN(C(=O)C(C)(C)O)C2)N1Cc1csnc1C C#CCCN=C(NCCCCCC)NCC1CCCN1CCC c1(C(=O)NC2CC(CNC(CC3C(C)CCC3)=O)C2)cccc(=O)o1 C1(NC(C=CCC)=O)CCC2(CCN(C(c3n[nH]cc3C)=O)C2)C1 C1(C(N(C)CCNC(=O)CC2COCC2O)=O)CCCCC1c1nc[nH]n1 c1(C(=O)NC)cncc(CNC(C2(C(=O)OCC)CCC2)=O)c1.N12CCC1C2 c1(CC(=O)NCC(CC)(C)NC(c2ccc(C)c(Cl)c2)=O)ccc(Cl)cc1N N1(C(CN(C)C)=O)CCCC(CN(C)C(C2CCN2S(C)(=O)=O)=O)C1 c1(C(=O)NCC(CC)(C)NC(C2(N(C)C)CCC2)=O)cc(OC)cc(OC)c1 C(C(CC(C)C)C(=O)NC1CC2(C1)CC2C(=O)N(C)Cc1cccc(F)c1)OC CCC(C)C(C(=O)NC1CNC(=O)C12CC2)NC(c1csc(=N)[nH]1)=O C1(C(=O)NCCC(C)NC(=O)OC(C)(C)C)(Cc2ccccc2)CC1(F)F C#CCCC(C(=O)NOC(CO)CO)NC(=O)C(C)OC(C)=O C1(OC)(CNC(C2COCCN2C)=O)CCN(C(c2nc(Cl)cs2)=O)CC1 Cc1ccc(F)c(C(N2CCC3C(NC(=O)Cc4c[nH]nc4C)C3CC2)=O)c1F c1(C(=O)NCC(CC)NC(CCC(CC)C)=O)cc(C)c2c(O)nc(O)nc2n1 CC1(C)CN(CCC(N2CC(O)(CCNC(=O)Cn3cnc(=N)[nH]3)C2)=O)CCS1 N1(C(C2N3CC(C)N(CC3)C2)=O)CC2(CCCCN2C(C2CCCN2N=O)=O)C1 c1(C(=O)NCCNC(CC2N(C(C)=O)CCC2)=O)cccc2c1CCC2 N1(C(c2c(C)con2)=O)CCCC2(C1)CN(C(=O)Cc1ccns1)C2 N1(c2cc(SCC)ncn2)CC2CN(C(c3ccncc3O)=O)C2C1 CC1(C)OC(C(N2CC(NC(c3cnc(O)o3)=O)C3(CCC3)C2)=O)C(C)(C)O1 C(=O)(C(CCCC(C)C)N1CCC(c2cccc(I)c2)C1)NCCCOC C1(CC(=O)NCCCNC(=O)OC)COCCN1C(=O)CC(C)SC CC12CC(C(N3CCC(CCCN4CCOCC4)CC3)=O)(C1)C1(CCC1)O2 C1(C(N(CC(CC)(C)OC)C)=O)CC12CCN(C(c1sc(F)cc1C)=O)C2 N1(C(c2ncc(OC)cn2)=O)CC(NC(c2cc(Br)c(C)o2)=O)C2(CC2)C1 CCCCC(CNC(=O)Cc1ccccc1OCC(F)(F)F)NC(=O)CCF C(=O)(CCCCCC#N)NCC(C(=O)NCCN1CCC2CC12)N(C)C C1(C2CCN(C(c3ccc(N)cc3O)=O)C2)(NC(CCC#C)=O)CC1 C(=O)(CCC(C)(C)O)NC1CC(Nc2nccc(OCCOC)n2)C1(C)C CC1(CNC(=O)C(CNC(c2cn[nH]c2)=O)CC2CCCC2)CCCC1O C1(CNC(CC(c2ccc(C)cc2)C)=O)CC(F)(F)CN1C(=O)C(C)CF N1(C(c2c(=O)ccn(C)c2)=O)CCC2(NC(c3ccc(O)nc3)=O)CCCCC12 C1(CNC(C(C)c2ccsn2)=O)(NC(=O)CC2=CCCCC2)CCC(C)(C)CC1 CC1(C(=O)NCCc2ccc(F)cc2)CCCN(C(=O)C(F)F)C1 N1(C(c2cc(C)on2)=O)CC2CCC(NC(=O)Cn3cccn3)CC2C1 c1(C(=O)NC(C2CCCN2C(=O)CCOC2CC2)(C)C)nc2cccnc2s1 N1(C(C(c2cccnc2)C)=O)CCCCC(NC(=O)CC23CC(C2)C3)C1 n1(CC)nc(C(=O)OC)cc1C.c12cn(nn1)CCOC(=O)C1CC21 CCCCC(C)C(=O)N(C1CN(C(c2cnc(Cl)cn2)=O)CC1(C)C)C N1(C(C23CC(C(C)(C)C)(C2)C3)=O)CC2CN(C(C3(C)COC3)=O)CC2C1 C12(C(=O)NC3C(CNC(=O)CCCCC4CC4)CCCC3)CCCC1OCC2 CCC(CC)C(O)CNC(C1COCCC1NC(c1coc2c1COC2)=O)=O Cc1cc(C(N2CCCC(CO)(Nc3ncnc4sccc34)C2)=O)cc(C)c1F CN1CCCCC(C(=O)NCC(O)CNC(c2cc(C(F)(F)F)ncn2)=O)C1=O C(=O)(C(CCC(C)(C)C)N(C1CCOC1C)C1CC1)NCCOCC Cc1cc(=NC2CCCN(CP(C)(C)=O)C2)[nH]c(NCCn2ncc(Br)n2)n1 Cc1nccc(C(=O)NC(C)CCNC(c2ncsc2Br)=O)c1Cl C1(C(=O)NC2CC(CNC(c3ncccn3)=O)C2)CCn2ncnc2C1 C(CC(C)N=c1cc(C)nc(CC2CC2)[nH]1)NC(c1ccc(OC)cn1)=O CCC(CC)(CCNC(c1ccsc1)=O)NC(=O)CC1C=NN(C)C1=O N1(C(C2(COC)CCOCC2)=O)CC(NC(=O)CC2CC(C)=NO2)CC(F)C1 n1(CCNC(C(N)=O)=O)cc(C(N2CC(n3ccnc3)C2)=O)cn1 c1(C(=O)NCCOCCC(=O)NCCS(CC)=O)sc(C)cc1C c1(C(N2CCC(C(N3CCN(C4CCOCC4)CC3)=O)C2)=O)ccc(Cl)nc1O N1(C(C(=O)Nc2cc(F)cc(Br)c2)=O)CCc2nc3ccccn3c2C1 Cn1c(=O)c2sccc2n2c(CNc3ccc(Cl)c(-n4ccnc4)n3)nnc12 CN1C(=O)COCC1CNC(C1C(NC(C2CCCCC2F)=O)C1(C)C)=O Cc1nc(N2CCC(NC(C3NC(=O)CC3C)=O)C2)cc(O)n1 c1(CCC(=O)NCC(CNC(Cc2ccc(C)o2)=O)C)ccc(=N)[nH]c1 C=CCCCCCCC(=O)NCC1CCCCN1C(=O)CC1CC2CCC1C2 N1(C(c2c(C)[nH]c(=N)s2)=O)CCC2(CCC(NC(C3CC3c3ccco3)=O)C2)C1 C(=O)(C(N)CN1CCCC1)NCC(C)Cc1cccs1 C(C(C)(C(=O)N1CC2C=CC2C1)NC(C1CC(C)=NO1)=O)SC C=CC1CN(C(c2cccc(N)c2C(F)F)=O)CC1NC(c1ccnc(C)n1)=O c1(CC)cc(N2CCC(N(C)C(c3noc(CC)c3C)=O)C2)nc(CC)n1 C1(C(=O)NCC(CNC(c2n(C)ncc2)=O)(C)O)CC2(CO1)CC(F)(F)C2 C1(C(C)C)CN(C(=O)C(O)C(F)(F)F)CCCN1C(c1ns[nH]c1=O)=O C(=O)(C(F)(F)CC)NCCN(C(C12CC(CCC)(C1)C2)=O)C1CC1 c1(C(C(=O)NC(CSC)C)(C)N(C)CCC2CC2)n[nH]c2c1CCCC2 C1(CN(C(C2C(C=C)C2)=O)C)CCCN(C(=O)C(c2cccc(OC)n2)(F)F)C1 c1(NC(C2(CNC(c3cccc(OC)c3F)=O)CC2)=O)cc(Cl)c(N)c(Cl)c1 N1(CC(=O)NC)CCC(c2nc(CC(=O)N(c3cccc(Cl)c3)C)no2)CC1 CC1CN(C(=O)C2=C(Cl)CCC2)CC(CCNC(=O)CCc2cnn[nH]2)O1 c1(OCC)ccc(-c2ccc(SCc3nnc(C)n3C)cc2)cc1OC Cc1nc(C(=O)NC(C(N2CC(S(C)(=O)=O)C2)=O)C2CCC2)ccc1C#N c1(CC)oc2ccccc2c1C=CC(=O)NCCNC(=O)C=C(C)C1CC1 C(C(C)(O)C(=O)N1CCC(CF)(NC(=O)CSc2ccncc2)C1)OC C1(CC(=O)NCC(C)(CO)NC(Cc2c(C)scc2)=O)CCCN(C)C1 c1(CN(C2CC(C)OCC2)C)cc(Cl)cnc1O Cc1cccc(C(N2CCOCC(CNC(c3ccc(F)nc3F)=O)C2)=O)c1C c1(C(N2CCCC(CCC)(NC(=O)CC(C)CF)C2)=O)nccc2occc12 C(=O)(C(C)(C)CCC#N)N1CC(C)C(CNC(c2cc(C3CCC3)no2)=O)CC1 C(=O)(CCCCCCNC(C1CCCS1)=O)NCC(C)Cn1cccn1 Cc1nn(CCO)cc1C(=O)NC1(C)CC(NC(=O)C(C)CN2CCCCC2)C1 N1(C(C(N2CCCC(C)C2)=O)=O)CCN(C(C2(O)CCOCC2)=O)CC1CO N1(C(C(C(CC)CC)C)=O)CCC(NC(=O)CCn2ccnn2)C(F)(F)CC1 N1(C(C(C)=O)=O)CCn2c(C(N3CCC4(CNC(=O)O4)C3)=O)cnc2C1 N1(C(C2(C)ON=C(C)C2)=O)CCC(C)(NC(C2CCCC(C(F)(F)F)O2)=O)CC1 C(=O)(C1CCc2c[nH]nc21)NCC1C(C(=O)NCc2cncc(Cl)c2)CCO1 N1(C(CN(CC(C)(C)C)C)=O)CC2(CCCCN(C(C3CC34CCC4)=O)C2)C1 Cc1c[nH]c(C(=O)NCC2(CN(C)C(c3c[nH]nc3C(F)(F)F)=O)CC2)c1 N1(C(c2ccncc2Cl)C(=O)NC)CCN(C2=NCC(C)S2)CC1 Cc1ccc(CCC(=O)N(C)CCN(C(=O)Cc2ccc(Cl)c(F)c2)C)cc1Cl c1(NC2CCC(NC(C(C)C3CCCC3)=O)CC2)ncc2c(n1)CCCC2 C=C1CCC(CNC(C2CC2c2cnn(C(C)C)c2)=O)C1 N1(C(C=CC(C)(C)SC)=O)CCC(C)C(CNC(c2ccnc(C)c2O)=O)C1 c1(C(=O)NCC=CCNC(C(CC)N(C)C)=O)cnn2c1CCCC2 N1(C(c2c(C(c3ccccc3)C)cns2)=O)CCC(C)(CCNC(N)=O)C1 c1(CN(C(=O)CC2(C)CCN2C(=O)CSC(F)(F)F)C)ncccn1 c1(C(N(C)CC2CCN(C(C=CCN(CC(F)(F)F)C)=O)C2)=O)scc(C)c1Cl C1(C(=O)NCC2CC3CN(C(c4scc(C)c4C)=O)CC32)CN2CCN1C(C)C2 Cc1cn2c(C(=O)N(CC(C)NC(C3(N(C)CCOC)CC3)=O)C)c(C)nc2s1 C1(NC(c2c(CC)c[nH]c2)=O)CC2C1CCN2C(=O)CCC1C(=O)ON=C1C c1(C(=O)NC2CCCCN(C(C=C(COC)C)=O)C2)c(Cl)ccc2ncccc12 Cn1nnc2cc(C(=O)NCC(F)CNC(c3ccc(N)c(F)c3)=O)sc12 CCCCCC(CC)C(=O)N1CCCN(C(=O)CN2CCNC(=O)C2)C(CO)C1 c1(OC(C(=O)NC(CC=C)CNC(c2ccoc2Cl)=O)C)ccccc1OC C1(C(C)(C)O)CCCCN1C(=O)NC1CC1F C(=O)(C(C)OC)N(CCNC(=O)CCNC(=O)OC)CC N1(C(=O)CCF)CC(O)(C2CCCN2C(=O)C(O)Cc2ccccn2)C1 Cc1ccc(C=CC(=O)NC2C3CN(C(=O)CCc4nc(=N)[nH][nH]4)CC23)o1 c1(C(N2CCC(NC(CCCOC)=O)C(CO)CC2)=O)nn(C)c2ccccc12 C=CC1(CC(=O)NCCN2C(=O)CCC2=O)CN(C(=O)COC2CN(CC)C2)C1 N1(C(C(c2ccc(Cl)s2)C)=O)CC(F)(CNC(=O)C=CC2CCCO2)C1 C=CC1(CC(=O)NC2CC(NC(c3cc(OC)no3)=O)C2)CCOCC1 C(C(=O)Nc1cc(C)ccc1C)(C(C)(C)C)NC(c1c(CC)[nH]cc1)=O N1(C(c2nc(C)oc2C)=O)CCC(C)(C)C1CC(=O)Nc1ccc(O)c(Cl)c1 C1(C(=O)NCc2cc(C)on2)CCCC12CCN(c1ncnc3sc(Br)cc13)C2 c1(NC(=O)NCC2CC(=O)NC2)ccc(F)c(OC(F)(F)F)c1 C1(CNC(C(CC)(C)CO)=O)CCC2(CN(C(C3CSC3)=O)C2)O1 N1(C(=O)C=CC2CCCCC2)CCN(C(c2cncnc2C2CC2)=O)C(CO)C1 C1(CNC(CC2CC(SC)C2)=O)CCN(C(c2cc[nH]c(=N)c2)=O)CC1C C1(C(=O)OC(C)(C)C)CCC(C(C)(C)C)N(C(N(C2COCC2F)C)=O)C1 CCC(O)C(C)C(=O)N(C(C)CNC(c1cc(C)n(C)c1C)=O)C c1(C(=O)NC2CC3CN(C(CCCC(C)=O)=O)C2C3)cc2n(c1)CCCNC2=O c1(C(N(CC(CC)(C)OC)C)C)cccc(F)c1F n1(CC(=O)NCCCC2CCCN2S(=O)(=O)CCBr)ncccc1=O C12(C(=O)NCC3CC(NC(Cc4c(C)noc4Cl)=O)C3)CCC(F)(CC1)C2 C12(C(=O)NC(CNC(c3cccc(CC)n3)=O)(C)CC)CCC(C1)C2(C)C c1(CC(=O)OCC(c2ccsn2)=O)c(F)ccc(Cl)c1Br c1(C(C)OCC)ncc(C(=O)OCc2csc(OCC)n2)s1 C(C1CCOCC1)=CC(N1CC(C)(C(=O)NCCOCC#C)C1)=O C1(C(N2CC3(CN(CC)C3)C2)=O)CCN(C(=O)CCS(C)(=O)=O)O1 CC1(C(=O)NC(CC(=O)NCC2(C)CC2(F)F)C2CC2)CC(=O)C1 C1(C(N(CC(C)(C)O)CCC)=O)C(NC(=O)C(C)OCCOC)C1(C)C c1(C(=O)NCC(C)NC(C(CC)NC(N)=O)=O)ccc(-c2nnc(C)n2C)cc1 N(C(=NCCSC)N1CCC(c2ccc(F)cc2Cl)CC1)C1C(OCC)C1 c1(OC(C)C)ccc(F)c(C(N2CCC(N(C(=O)C(C)C(F)F)C)C2)=O)c1F C(C(C)N=c1[nH]ncs1)(c1ccccc1)N(C1(O)CN(C(C)=O)C1)C CCCC(C(=O)N1CC(OC)C(NC(c2cc(F)n[nH]2)=O)C1)OCC CCCC(C)(C)CC(=O)NCCCOCCNC(C1(CO)CCCCO1)=O CN1C(=O)OCC12CCN(C(=O)Nc1cnn(C3CC3)c1)C2 C12(NC(c3c(C)nc(O)[nH]3)=O)CCCN(C(C3(CC(C)C)CC3)=O)CC1C2 c1(-c2n(C(CC)CC)cnn2)ccc(-c2noc(C3CCCS3)n2)cc1 N1(C(C(C)NC(=O)Cn2cnnn2)=O)CC=CC1CNC(=O)Cc1ccon1 C1(CC)C(NC(c2occc2C)=O)CCCN1C(=O)COCc1cccc(C)c1 Cc1n[nH]c(C)c1CCC(=O)NC1CCCC(CNC(=O)CC2CCC(C)C2)C1 C1(CN(C(c2c(CC)csc2)=O)C)CCCCN1C(=O)Cc1nncn1C(C)C Cc1nc2cc(C(N3CCN(C(C)CC(=O)O)CC3)=O)cc(Br)c2o1 c1(CC(C(=O)NCC(CN(C(=O)COC2CC2)C)(C)C)(C)C)ccc(C#N)cc1 N1(C(CC)=O)CCC(C)(CNC(C2CC(NS(C)(=O)=O)C2)=O)C1 N1(C(C2(NC(CCOCCOC)=O)CCCC2)=O)CC2(CC(CO)CO2)C1 CC1CN(C(=O)C(c2ccccc2)O)CC(C)C1N=c1nc[nH]s1 C1(C(=O)NC(CNC(Cn2c(C)ncc2)=O)C)CC12CCC1(CC1)CC2 CC(C)CS(=O)(=O)CC(=O)N1CCC(NC(C2(F)CCCN(C)C2)=O)C1C Cc1ccc(C)c2c1OCCC2Nc1ccc(Br)cc1C(F)(F)F N1(C(CCNC(COC)=O)=O)CC2CC(NC(=O)CCc3ccncc3)C1C2 C1(C(N2C(C(=O)O)C(NC(=O)C(F)(F)F)CCC2)=O)CC2(CCOCC2)C1 C(=O)(C(F)(F)Cc1ccc(Cl)cc1)N1CC(C(C)N)C1 N1(C(C)C(=O)NCc2ccccc2Cl)CCC(Cc2ccc(O)nn2)CC1 CCCC(CCC)CC(=O)NCCN(C(=O)CCc1ncc[nH]1)CC1CC1 C(CCC(N)=O)(C(=O)NC1CC(N(C(=O)CCCCCF)C)C1)NC(C)=O c1(C(=O)NC23CC(NC(=O)C(O)CC(F)F)(C2)C3)cc(F)cc(F)c1O C1(NC(C(C)SCCCC)=O)CC(NC(C2CC=CCO2)=O)C(O)C1 Cc1c(C(=O)NCCN2CCN(C(c3cc(F)ncc3Br)=O)CC2)cncc1Br N1(C(C=CC=CC)=O)CCCC1(C)CNC(=O)CC(OCC)OCC c1(OCC)nc(N2CC(C(C)NC(=O)C(C)(C)c3ccccc3)C2)ncc1Cl N1(C(C(n2cc(CC(C)C)nn2)C)=O)CCCN(CCOC2CCCCC2)CC1 c1(CC)c(NC2CC(CNC(c3cnn(CC4CCOC4)c3)=O)C2)ncnc1Cl N1(C(C(C)=CC2CC2)=O)CCC2CCCC(C1)N2C(=O)CCc1cnn(C)c1 C1(CC(=O)NC(C(C)NC(CC(CC=C)(C)C)=O)(C)C)Cn2ccnc2NC1=O c1(C(N2CCN(C(c3c(CC)[nH]c(=N)s3)=O)CC2)=O)cc(C)ncc1C CS(=O)(=O)c1c[nH]c(=NC2CN(C(=O)COC3CCCC3)CC2C#N)cn1 C(=O)(C1CCc2c(Cl)cccc21)NCC1CC=C(C)CC1.N12CCCC1C2 N1(C(C(CC)(C)OC)=O)CCN(C(c2ccc(-c3ccco3)o2)=O)CC12CC2 C1(NC(c2c(Br)ccc(OC)n2)=O)C2CCC1CN(Cc1ccnn1C)C2 N1(C(c2cccc(F)c2F)=O)CCN(C(C2OCC3COCCC23)=O)CC(O)C1 Cc1ccc(S(N)(=O)=O)c(C(=O)NCC2C3CN(C(C45CC(CO4)C5)=O)CC23)c1 N1(C(c2cscn2)=O)CCOCC2(COCCN2C(C2(CC3CC3)CCC2)=O)C1 c1(C(=O)NCC2CC(NC(CC(=C=C)C)=O)C2)cc(Br)cc2scnc12 CC1(C)C(CC(=O)NCC2(NC(C3CNC(=O)N3)=O)CCC2)CC1O N1(C(C)=O)CS(=O)(=O)CC1C(N1CCC(CNC(C2(C)CC2C)=O)C1(C)C)=O C1(C(=O)NCCN(C(c2cc3cnccc3[nH]2)=O)CC)OCC2COCCC12 C(CCC(O)C(=O)NOC1CCC1)NC(c1c(OC)cnnc1)=O CC(C)CC(C(=O)N1CCN(C(c2sccc2C#N)=O)CC1C)C(C)C C(=O)(C(C)(O)Cc1ccccc1)NCC1C(NC(c2n(CC)ccc2)=O)C1 CCC(CC)C(C)C(=O)NC(C1CN(C(=O)Cc2cc(F)ccc2OC)C1)C Fc1ccc(F)c(CNCC2CC2c2cccnc2)c1F N1(C(c2c(C)nc(C(C)C)cc2)=O)CC2CN(C(c3cnoc3C)=O)CC2(C)C1 N1(C(CC(CC)C)=O)CCCC(N(C(c2ccc([N+](=O)[O-])[nH]2)=O)CC)CC1 C1(C(N2CC(CC#C)OCC2)=O)N(C(c2cc[nH]n2)=O)CC12CCCC2 C1(CC(=O)NCC(CC)N(C(c2cn(CCC=C)nn2)=O)C)CCCC(=O)C1 Cc1cc(C)n2ncc(NC(N3CCSc4ccccc4C3)=O)c2n1 c1(CC(=O)NCCCN(C(CC(C(C)C)OCC)=O)CC)ccccc1[N+](=O)[O-] C(=O)(C1=C2CCN=C2NC=C1)N1CC2OCC(NC(C(C)CN(C)C)=O)C2C1 N1(C(=O)OC(C)(C)C)CC(C(=O)N(N2CC(c3cccnc3)C2)C)C1C1CCC1 C1(F)(CNC(C(C)NC(CC)=O)=O)CCC(NC(=O)C=Cc2cccn2C)C1 N1(C(C2(CC)CC2)=O)CCC(C)C(NC(c2cc(C3CCCCC3)[nH]n2)=O)C1 c12ccc(cc1)CN1CCC(C1)CNC(=O)CCO2.CCCCCOC(F)(F)F c1(CC(=O)NCC(N(C(C2C(=C)C2)=O)C)C2CC2)c[nH]c2cccc(OC)c12 CC1(C(N2CCN(CCO)CC2)=O)CC(O)CN1C(C1CC(N2CCCC2)C1)=O CCCC(CC)C(=O)N1CC(CNC(=O)CNC(C)=O)C(C)C1 C1(CNC(c2c(CC)occ2)=O)CN(C(=O)CSc2n[nH]c(O)n2)CCO1 C1(C(=O)NCCc2ncoc2CCNC(C2(CC)CC2)=O)CC2(C1)CC21CCC1 CCCCC1CC(=O)N1.C12(NC(=O)C=C(C)COC)CC(C1)C2 c1(OC)ccc(Br)cc1NC(=O)NC(c1nc(C2CC2)no1)(C)C N1(CN=C(NCC(CC(C)C)(C)N(C)C)NC(C)COC)CCc2sccc2C1 N1(C(C(C)n2cnnn2)=O)CC2(CCC2CNC(c2cc(Br)no2)=O)C1 c1(C(C)C)ncoc1C(=O)NC(C1CCOC1)CNC(c1cc(Cl)ns1)=O C(=O)(C(O)C(C)(C)CC)N(C1CC2CN(C(C3(C(=O)OCC)CC3)=O)C1C2)C C12CCCCC1CN2C.c1(C(=O)NC2CCNCC2)cc(-c2cccs2)[nH]n1 CCCCC(F)C(=O)NCC1(C)CCN(C(C2CCCCC2(C)C)=O)C1 C=CC(CC)CC(=O)NCC1CCCN1c1nnco1 Cc1c(C(=O)N(C)CC2C3CN(C(=O)C(O)C(C)(C)C)CC23)cccc1F C1(CC(=O)NC23C(CN(C(c4cc(OC)ncn4)=O)C2)C3)C(=O)N(C)N=C1C CC(CC(F)(F)F)C(=O)NC1CCC(CNC(c2ccc3[nH]ccc3n2)=O)CC1 c1(C(=O)NCCC(C)N(C(c2ncc(C)cc2F)=O)C)ccnc2cc[nH]c12 Cc1nc(=NCC2CCCC2NC(C2C(C(F)(F)F)C2[N+](=O)[O-])=O)s[nH]1 C#Cc1cccc(OCC(N2CCCC(NC(=O)CCCc3cccs3)C2C)=O)c1 N1(C(C=Cc2ccn(C)c2)=O)CCCC12CCN(C(C1CCC(C)(C)CO1)=O)C2 N1(C(c2[nH]cc(C#N)c2)=O)CCC(O)CC1CC(=O)NC1CCC(F)(F)CC1 C1(C(=O)NCC2(OC)CC2)COCC1NC(C1(CO)CCCO1)=O C1(C)(NC(CC(C)C2CCCO2)=O)CCN(C(=O)C2=CSCS2)CC1 c1(C(=O)NCCCC2(NC(c3cncc(F)c3)=O)CC2)cnc2[nH]cnc2c1 N1(C(C2N(C)CCC2)=O)CCCC(O)(CNC(c2ccc(C(F)F)cc2)=O)CC1 C1(CNC(CC(C=C)C)=O)(CO)CC12CCN(C(c1coc(N(C)C)n1)=O)CC2 c1(C(=O)NC2CN(C(c3sccc3Cl)=O)CC23COC3)cc(Cl)c2cc[nH]c2c1 c1(C(N2C(C)CC(NC(=O)CCOC3COC3)C2)=O)cc2c(F)cccc2s1 Cc1cccnc1CSC1CN(C)C(=O)N1.N12CCCC1C1(O)CN(C1)CC2=O c1(CC)cscc1C(=O)NC1CCCC1CC(=O)NCC1SCCS1 C1(CN(C(C(Cn2ccc(C)n2)C)=O)C)COCCN1C(c1cc(Cl)cn1C)=O C1(NC(c2ccc(COC)o2)=O)CN(C(=O)C(F)CC2CCOC2)CC1C c1(C(=O)NCC(CO)NC(c2ccc(C)cc2O)=O)cc([N+](=O)[O-])c(C)cc1C C1(C(N2CCN(C(=O)NC3(C)CNC(=O)C3)CC2)=O)CCC(F)(F)CC1 c1(C(N(CCNC(=O)C(c2ccccc2)O)C2CC2)=O)c[nH]cc1Br C12(NC(=O)C=C3CCCC3)CCCC(CN(C(C3CC4(C3)CC43CC3)=O)C1)C2 c1(C(N2CC(C)C(NC(=O)CN(C)C)C(C)C2)=O)cc2cccc([N+](=O)[O-])c2[nH]1 N1(C(c2cc(CC)on2)=O)CCOCC(NC(C23CCC(CC2)O3)=O)C1 N1(C(C(C)N(C(C2C(C)(C)C2(F)F)=O)CC)=O)CC2(CC(CO)CO2)C1 Cc1[nH]c(Cl)nc(=NC2CN(C(=O)CS(=O)(=O)C(C)(C)C)CC2(C)C)c1C#N N1(C(=O)Cc2cc[nH]n2)CCC2(CC1)CN(C(c1cc(F)cc(Cl)c1O)=O)C2 Cc1cc(C(=O)NC(c2cccc(C(=O)O)c2)Cc2ccccc2)nn1C Cc1cc(NC(=O)C(=O)NC(c2cnn(C)c2)CN(C)C)c(C)s1 CCC(C(=O)NCc1csc(C(=O)NC(c2ccncn2)C)c1)OC N1(C(CCC(CC)OC)=O)CCC(C2CC2)(CNC(c2cccs2)=O)C1 N1(C(C(=O)NCC(F)F)C2C(CC)C2)CCC(c2cccnn2)C1 C1(C(F)(F)C(=O)NC2CCC2NC(=O)CSCC(C)C)(OC)CCCC1 N1(C(C2(C#C)CCCC2)=O)CC2CC(NC(C3(C)CCN(C)C3)=O)C1C2 C1(CC)CCN(C(=O)C(C)N=[N+]=[N-])C(C(=O)NCCOC(C)=O)C1 C(=O)(C(C(C)C)n1ncc(N)n1)NCC(=C)CCNC(C1CN(C)C1)=O c1(C(=O)NC2C(C)N(C(c3ccno3)=O)CCC2C)cnc2ccccn2c1=O C1(C(=O)NCC(CC)(CC)NC(=O)C(C)N2CC(C)C2)CC2C=CC1C21CC1 C1(CNC(C=CCOC)=O)CN(C(c2sc(OC)nc2Cl)=O)C2COCC2O1 Cc1ccc(C(N2CCC2(C)CC(=O)NC23CCC(CC2F)C3)=O)c(C)c1 C(=O)(C1Cc2ccc(Cl)cc21)NCC1N(C(c2ccc(OC)cc2O)=O)CCC1C N1(C(c2c(N)non2)=O)CCOC(CCNC(C2CC3CC3C2)=O)C1 C(CC(CNC(=O)C(C)(C)NC=O)NC(=O)C(Cc1ccsc1)NC=O)OC c1(C(=O)NCC23N(C(CCCSC)=O)CC(CCC2)C3)ccc2cnccc2c1 C12(NC(CC3(C=C)CN(C(=O)CCN4CCOC4=O)C3)=O)CCCC1OCC2 CC1=NOC(C(=O)N(C2CC(C(=O)NCCc3cnc(C)[nH]3)C2)C)C1 CC(C)C(C)CC(=O)NC1CCC(=O)NC1C1CCN(c2cc(Cl)ncn2)CC1 N1(C(c2cccc(C)c2O)=O)CCC(C2(NC(=O)C(n3cc(Cl)cn3)C)CC2)C1 Cc1cc(C(N2CCN(C(C3(C(=O)N(C)C)CC3)=O)CC2)=O)c2c(c1)CCC2 c1(CC)nn(C)c(C(N2CC3CN(C(=O)C(C)(C)NC(C)=O)C3C2)=O)c1Cl CC1CN(C(=O)CC2CC2C(F)(F)F)CCCN1C(=O)C=CCO Cc1cc(C)c(C=CC(=O)NCCCC(C)NC(C2CC(CF)C2)=O)c(C)c1 CCC(CC(=O)N1CCC(C(=O)N=c2cc(C)n(C(C)C)[nH]2)(CF)C1)C(C)(C)C C12(C(=O)NC3CCC(NC(CC(CN(C)C)O)=O)CC3)CC3CC1C2C3(F)F n1(CCC)nccc1C(=O)NC1CCCC1CNC(=O)C(C)Cc1cnc[nH]1 c1(C(=O)NC(CCNC(c2cc(OCC)no2)=O)C)cnn(C2CC2)c1Cl c1(C(N(CCC(C)NC(=O)Cc2cc[nH]n2)C)=O)cc(Cl)c(F)cc1N O(N(C(=O)C1CC(C)CN1C(=O)CCn1cncn1)C(C)C)CC N1(C(C2(COC)CC2)=O)CC(C(F)(F)F)C(CNC(=O)CN2CCCCC2C)C1 C1(CCNC(c2n(CC(=C)C)nnn2)c2cscc2F)CCCS1(=O)=O Cc1ccc(C(CCO)Nc2cc(NCC3CCCS3(=O)=O)ncn2)cc1 CC1(C)CC=C(C(=O)NC2CC3(C2)CC(NC(=O)CSCC(N)=O)C3)CC1 CCC(C)CC(C(=O)NCc1ccc(SC)o1)NC(C1CCCC(=O)C1)=O c1(CCC(=O)NC(C)C(C)NC(=O)Cn2ccc(C3CC3)n2)ccc(F)cc1F C12(C(N(CCOC)C)=O)CC(C)(C1)OC2(C)C c1(OC)ccccc1NC(=O)C(c1cccc(Br)n1)N1CC=CCC1c1cccnc1 c1(C(=O)NC2(CNC(C3C(CCO)CCO3)=O)CCC2)ccc2n[nH]cc2c1 N1(C(C(C(C)C)O)=O)CCC(n2cccn2)(CNC(c2cc(C#N)no2)=O)CC1 N1(C(c2ccc(C(C)=O)s2)=O)CCOCC1CNC(=O)C(C1CCOCC1)C c1(C(=O)NC(CC)C(OC)OC)cc(S(=O)(=O)N2CCCCC2)ccc1F c1(C(N(CCNC(C=CC(=O)OC)=O)C2CC2)=O)cc(S(=O)(=O)N(C)C)c[nH]1 c1(-c2nnc(C)o2)ccccc1C(=O)NC(CNC(=O)C(C)NC(N)=O)C(C)C N1(Cc2nccc(C)c2)CC2(CN(C(=O)Cn3cc(CO)nn3)CC2C(=O)O)C1 C1(C(N2CCCC(CCNC(C3(C)CC3(F)F)=O)C2)=O)CCCC12CCOCC2 C(CN=C(NC1CCS(=O)(=O)C1)NCC=C)NC(c1cscc1C)=O c1(CNCC(CN(CC)CC)O)cccc(C#N)c1 c1(C2C(C(=O)NC(C(C)NC(C3CCOCC3)=O)(C)C)CCC2)ccc(F)cc1 N1(C(c2cnc(CCC)s2)C(=O)NC(C)C)CCc2cc(F)c(F)cc2C1C c1(NC(CC2(OC)CN(C(C34CC(CO3)C4)=O)C2)=O)nnccc1C Cc1cc(C(=O)NC(Cn2cccn2)C(N2CCN(CCF)CC2)=O)ncn1 C1(NC(C(C)C(F)F)=O)CN(C(c2ccnc(OC3CC3)c2)=O)CC(C)(C)C1 C1(C(N(C)Cc2c(C)occ2)=O)COCCC1NC(c1csc(F)c1)=O c1(CC)n[nH]cc1C(=O)NC1CCC(N(C)C(c2cc(-c3ccco3)on2)=O)C1 c1(N(C)Cc2cc[nH]n2)[nH]c(=NCCCC(F)F)nc2c1cnn2C C1(C(=O)NC2(CC=C)CCCN(C(=O)CCC)C2)CC2(CCCC2)CO1 Cc1sc(-c2ccncc2Cl)nc1CN1CCN(C(c2ccccc2)=O)CC1 C(CCCCCCO)(C(=O)NC1CC(C(=O)OC)C1)N1CCC(CC(=O)OC)C1 c1(C(=O)NC(CN(C(C2N(C(C)=O)CC2)=O)C)C)cccnc1 C1(C(=O)NC2C(F)CCN(C(Cc3c(C)scc3)=O)C2)CCc2[nH]nc(O)c2C1 c1(C(=O)NC2C(NC(C3(OC)CC(C)(C)C3)=O)CCOC2)cn(C)c(=O)n1C c1(CC)cc(C(=O)NC(C)(CNC(C2CCS(=O)(=O)N2)=O)C2CCC2)ccc1F N1(C(c2cnc(C(C)C)s2)=O)CCC(NC(=O)CCCN2CCCCC2)C(O)C1 CC1(C)CCC(CC(=O)NC2CCOC3(CCC3)C2)N(C(=O)OC(C)(C)C)C1 C1(NC(CCC(=O)NC)=O)CCN(C(=O)Cn2cnc(C(N)=O)c2)C12CC2 C(=O)(CCCCCCCCCO)N1CC2CN(C(c3c(CC)onc3)=O)C2CC1 CC1CN(C(=O)CSc2ccccc2)CC1NC(=O)Cc1nncn1C Cc1nn2c(c1C(=O)NCC1CCN(C(=O)CN3CC=CC3)CC1C)CCCC2 c1(C(=O)NCCCN(C)C(C2CCC(C)(C)OC2)=O)ccc(Cl)c(C#N)n1 C1(C(N(C2CCN(C(CCN(C)CC)=O)CC2)C)=O)CCCC2(CCCCC2)C1 c1(C(N2CCC(C(=O)Nc3ccc(O)nc3)C2)=O)cccc2ncccc12 N1(C(C(Cc2cn[nH]c2)NC(c2cnccn2)=O)=O)CC(F)(F)C1C1CC1 CN1CCN(C(C2CN(C(=O)COc3ccc(O)cc3Cl)CCO2)=O)C(CO)C1 C12(C(C)C)COC(C(=O)NC(C)CC(C)NC(c3cnc(N(C)C)s3)=O)(C1)C2 C1(C(=O)NCC(=C2CN(C(C3CCCN3C3CC3)=O)C2)F)CC2CCC1C2 C1(CNC(C(=O)N(C)Cc2ccno2)=O)CCCC(F)(F)CC1 Cn1cnnc1C1CCN(C(c2csc(Cl)c2)C(=O)NC2CCOCC2)C1 C1(C(=O)NC2CCN(C(=O)CN3CCCC3CO)CC2)CCCC2(CC2)C1 CC(F)(F)C(C)(C)C(=O)NC1COCCC1NC(c1coc(C(F)F)n1)=O c1(-c2ccc(SCC)s2)ccc(-c2cnoc2)c(C)c1.N12OCC(C1=O)C2 C(C)(C)(CC(F)C(=O)NC(c1cccnc1)C)NC(C(C(C)C)SC)=O c1(C(N(C(C)C(N2CCC(CCOC)C2)=O)CC)=O)cc2ccccn2c1 Cn1cc2c(C(=O)NCC3(F)CN(C(=O)C4=CC5C=CC(C4)C5)C3)cccc2n1 Cc1ncccc1CC(=O)NCCCOCCNC(=O)CN1CCCC1=O C1(CNC(c2cccc(C)c2Cl)=O)CN(C(=O)CC(C)C2CC2)CCC12CCOC2 C1(C)(C(=O)NC(CN(C(CCSC)=O)C)C)CCN(C)C1=O C1(NC(NCC2CCC(CC)O2)=S)CCC(=O)NC1 c1(C(N2CC(O)(CNC(C(C(C)(C)C)OC)=O)C2)=O)c(C)cc(O)cc1C C1(NC(C(Br)=C(C)C)=O)CC2(CCN(C(c3cccc4nncn34)=O)C2)C1 c1(OC)ccc2nc(NC(C(=O)N3CCCC3)=O)[nH]c2c1.c1(C(CN)=O)ncoc1C C(CC(=O)NNC(=O)C(C)(C)CCCCNC(=O)CCCCC1CC1)OC C1(N(C(=O)CN2CCCC2)C)CCN(C(=O)NC2CC2Cl)CC1O C(CCC(=O)NC(c1n[nH]c(CO)n1)C)(C(C)C)NC(C(c1ccc(C)o1)C)=O C1(C(C)=O)(C(=O)NCCOC(C)(C)C)CC1.C1(C)COCCN1CCCF CC1CCCC(C)C1NC(c1cc(CNC(c2cc(Cl)cn2C)=O)no1)=O C1(C(N2CC3C(CC(=O)NCC4(C)CCOC4)(C3)C2)=O)CC2CCCC2C1 C1(C)(NC(C2C3N(C(c4c(C)csn4)=O)C(CC3)C2)=O)CN2CCC1CC2 C1(CCNC(c2nc(C)sc2)=O)CCCCN1C(c1cnnn1C)=O Cc1cn2c(n1)CC(C(N1CC(NC(c3c[nH]cc(F)c3=O)=O)CCC1C)=O)C2 N#Cc1ncc(Br)cc1NC(C1CCN(C(=O)C=Cc2cccnc2)C1)=O CCCC(CNC(c1c(C)nsc1N)=O)C(=O)NC(c1nc[nH]n1)C1CC1 c1(Oc2cccc(C(=O)OCC(=O)NCCC(C)N(C)C)n2)ccc(Br)cc1F N1(Cc2ccc(C)cc2)CCc2c(n(C)c3ncccc23)C1.N12CC=CC1C2=O CN1CC(C(=O)N(CCCNC(c2ccccc2)=O)CC2CCCCC2)NC1=O C(CC(C(C)(C)C)NC(c1c[nH]nc1Cl)=O)N(C)C(C1CCCC1C1CC1)=O C12CCCN1C(=O)OC(C)(C)COCCC2.C1(OC(C)(C)C)CCOC1 N1(C(C(C2CCC2)OC)=O)CC2(C(N3CC(S(C)(=N)=O)C3)=O)CC1CO2 CC1OC(=O)NC1C(N1CCCC(C(=O)NCC2C(CO)C2(C)C)C1)=O c1(NC2CC(NC(c3c(C)[nH]nc3Cl)=O)C2)ncnc2cccc(Br)c12 C1(C(=O)NC(CC=C)C2CC2)CC12CCN(C(=O)C=Cc1cc[nH]n1)C2 c1(C(=O)NCCN2CCN(C(CCCC=C)=O)CC2)cnc2nc(Cl)ccc2c1 N1(C(C2CC(C(=O)OC)C2)=O)CCN(C(=O)C=C(C2CC2)C2CC2)CC(C)(F)C1 N1(C(C(F)=CCC)=O)CC2CCC(C1)N2C(c1cc2c(ccn2C)[nH]1)=O CP(C)(=O)c1cccc(S(=O)(=O)NC2(C(F)(F)F)CC3C=CC2CC3)c1 Cc1cc(C)c(C(=O)N(C(CNC(c2ccc(C(N)=O)[nH]2)=O)C2CC2)C)c(S)n1 C1(C(N2C(C)(C(=O)Nc3n(C)ncc3)CCC2)=O)CSC(c2ccccc2)=N1 C1(NC(CCC)=O)CCCN(C(c2ccnn2C)C(=O)NCC(F)F)C1 CCC(CC(=O)NC(C(C)C)C1CC1)N(C(=O)CC1CCOC1(C)C)C c1(-c2cc(C(=O)NCC(CN(C(CC(C)N(C)C)=O)C)O)n[nH]2)cccc(Cl)c1 NS(=O)(=O)c1ccsc1C(=O)NCC1CCC(NC(C2CC(F)(CO)C2)=O)C1 Cc1cccc2c(C(N3CC4(C3)CN(C(=O)Cc3csc(S)n3)C4)=O)cnn12 C1(C(=O)NC(C2CCN(CC(=O)NC3CC3)C2)C)COC(C)C1 c1(N2CCCCC(NC(C3(C)CC=C(C)CC3)=O)C2)cc(C#N)ccc1[N+](=O)[O-] c1(C(=O)N)ccc2nc(C)cn2c1.C1(N)CC(CO)N(C(c2nc(CC)sc2)=O)C1 N1(C(c2c(CNC(C3CC(C)(C)C3)=O)ccs2)=O)CC2CC=CC1C2 C1(C(N2CC(NC(c3cc(O)ccc3F)=O)C(F)C2)=O)CCCCNC1=O N1(C(C(CCC)NC(N)=O)=O)CC2CN(C(c3ccc(N)cc3C)=O)CC2(C)C1 c1(C(=O)NCC2COCCN(C(C3(C)N(C)CCC3)=O)C2)coc(S(C)(=O)=O)c1 CCCCCCN(CC(=O)NC1CC(NC(=O)Cn2cc(C(=O)OC)cn2)C1)C C1(C(C(=O)NC2(CC(C)C)CC2)C)CCN(C(=O)C(C)(C)N2CCCC2)C1 N1(C(CC)C)C(=O)NC(c2cn(C)nc2C)C(C(=O)N(C)C)=C1C1CC1C CON=Cc1ccc(C(=O)NCC2CN(C(=O)CC=C(C)C)CC23CC3)cc1 C1(NC(c2cscn2)=O)(CF)CCN(c2ccnc(CO)n2)C1 C(=O)(C1Cc2ccc(Cl)cc21)N1C2CN(C(C3N(S(C)(=O)=O)CC3)=O)CC1CC2 C12CC(C1(C)C)NC(=O)C2.C1(C)(CC(N2CC(C(C)C(=O)O)C2)=O)CCOC1 N1(C(Cc2ccc(C)o2)=O)CCCC2(NC(c3cnn(C)c3F)=O)CC2C1 C1(NC(C(C)Sc2ccc(Cl)cc2)=O)CC2C1CCN2C(=O)Cc1c[nH]nc1O N1(C(c2cc(COC)sc2)=O)CCC2C(CCN2C(c2ccc([N+](=O)[O-])o2)=O)C1 C1(OC)CC(CC(=O)NC2(C)CN(C(=O)C(F)(F)CN(C)C)C2)C1(C)C C12(C(N3CCC(CN(C(=O)CC4(C)CC4(F)Cl)C)C3)=O)CC(CO)(C1)OC2C Cc1cc(C(=O)NC2CN(C(c3c[nH]nc3C3CCOCC3)=O)C2)c(N)c(F)c1 CC(C)C(CN(C)C)N=c1[nH]c(=NCc2c(Cl)cnn2C)[nH]c2cccnc12 C1(C(N2CCC(NC(CCc3ccc(SC)cc3)=O)C2)=O)CN(S(N)(=O)=O)C1 c1(C(N2CC3N(C(C(CC#C)C)=O)CC(C3)C2)=O)[nH]c2ccc(OC)cc2c1C C(=O)(N=c1ccn(CC(N)=O)[nH]1)C1N(C(C2N(C(=O)OC)CC2)=O)CC(O)C1 C(=O)(C(C(C)C)NC(=O)OC)N1CC(O)(C(C)NC(C(C)OCC)=O)C1 C1(=CC(=O)N(CCOCCCNC(C2C(C)OC(C)C2)=O)C)CCC(C)(C)CC1 N1(C(c2c(NC)ccs2)=O)CCN(C(=O)C2=CCC(C(F)(F)F)OC2)CC(O)C1 C1(C(=O)NCC)(CC)CCCN1C(=O)C(C1CCC1)OCC(N1CCCC1)=O N1(C(C(COC)OC)=O)CC(OC)CC1CCNC(=O)CCCn1ccnc1 CC1(C)CC(CC(=O)NCC2CCN(C(c3cnc(C(F)(F)F)s3)=O)C2)CCO1 O=C(C1=CCN(C(C2CCCC2)=O)CC1)NCC12CCCCC1C2 C1(CCNC(CSC)=O)CN(C(c2cnn(-c3ccc(F)cc3)n2)=O)CCO1 O(S(=O)(=O)c1ccccc1)c1cn(N2C(=O)N(c3ccc(Br)cc3)CC2)nc1 c1(C(=O)NCCC(C)N(C(c2c(CC)noc2)=O)C)cc2c(cc1F)NCCC2 C1(NC(CCCC(N)=O)=O)CN(C(=O)CNC(c2ccncc2)=O)C2CCCC12 c1(C(N(CC(C)NC(=O)C(N2CCNC2=O)C)CC)=O)nnccc1C Cc1cc(C(=O)N(C)CC2COCCN2C(=O)CCCC2CC2)ccc1F C1(NC(C=C(C)C(F)F)=O)CCN(C(c2cccc(C3CC3)c2)=O)CC1C(C)C N1(CCC(=O)N(C(CC)CF)C)CCCCC1c1nc(O)n[nH]1 C(=O)(C(C)(F)CCCC)N1CCC(CN(C(C(C=C)(C)C)=O)C)C1 c1(C(=O)NCC2CCC(NC(C3C(C)OC(=O)N3)=O)C2)ccc(C(N)=O)cc1F Cc1nccc(C(N2CC(NC(=O)C(C(C)C)C3CCCCC3)C(O)C2)=O)n1 C1(C(N(CCC(=O)NCC(c2nccs2)C)C)=O)CC1C1CCCC1 C1(CNC(c2n(C)ncc2)=O)CN(C(=O)CONC(=O)OC(C)(C)C)C2CC12 N1(CC(=O)N(CCCCCNC(=O)COCc2ccccc2)CCl)CCOCC1=O C1(C(=O)NCC(C)(CO)NC(c2coc3c2COC3)=O)CCc2[nH]nc(O)c2C1 c1(C(=O)NCCC(CNC(c2cncc(OC)c2)=O)O)ccc2oc(C)nc2c1 N1(C(C(C)C#N)=O)CC(C(=O)Nc2cc(C#N)ccc2F)C2(CCC2)C1 c1(OCC)ncc(C(=O)NCCC2CC(NC(=O)CCCOC(C)C)C2)s1 CC(C(Cc1ccncc1)CO)N(C(C(=O)NC(c1ccco1)C)=O)C1CC1 CC(C)(CO)C(C)(C)NC(C1CC(=O)CN1C(C1OC2CCC1C2)=O)=O C1(OC)CC(F)CN(C(=O)CC2CCCN2C(=O)CC2(C)CC2)C1 N1(C(C2N(CC)CCC2)=O)CCC(C(N2CC(CO)C(C)C2)=O)(CF)C1 C1(=CC(=O)NCCC2(C)CCN(C(C(=O)NCC)=O)C2)CCC(C)(C)CC1 c1(OC)ccc(NC(C2(NC(=O)CC3CCOC3)CCSC2)=O)cc1 N1(C(C(C)(C2CC2)OC)=O)CCC(CNC(c2c[nH]cc2C(C)(C)C)=O)C(C)C1 C1(C(=O)NCCN(C)C(C2(F)CS(=O)(=O)CC23COC3)=O)CCOCC12CCC2 C#CC1(C(=O)NC2CCOC(C)C2)CCN(C(=O)Cc2csnn2)C1 c1(OC)ccc(O)c(OCC(O)CNCC2C3COCC23)c1 C(=O)(C(N=[N+]=[N-])C(C)C)N1C(C(=O)NC2CC(CC(=O)OCC)C2)CCC1 N(C1CC2(CN(C(c3c(C)cnn3C)=O)C2)n2ccnc21)C(CCCC(=C)C)=O Cc1cc(C(=O)NC2CC(CNC(=O)C(F)=C3CCC3)C2)c2[nH]cnc2c1 CC1(C)CN(C(C2CCC2CF)=O)CC(C)(C)C1NC(c1nnc(O)cc1O)=O C1(C(=O)NC(C)CC#N)CCCC(Nc2cc(-c3cccs3)ncn2)C1 c1(C(=O)NC2(C3CCN(C(C4(CC)COC4)=O)C3)CC2)cnnc2ccccc12 C(=O)(C(=O)CC(C)CC)NC1CCCC(C(=O)NC(CC#C)CO)C1 c1(C(=O)NCC(CC)NC(=O)C(O)CCC(C)C)c(C)cc(C)cc1C CCCCCC(O)C(=O)N1CC(C)(CNC(=O)COC)NN=CC=C1 CC1CC(=O)NCC1C(=O)NCCN1CCC(NC(=O)Cn2cnnn2)CC1 C=CCC(C)C(=O)NC1(CO)CN(C(C2(CCOC)CC2(F)F)=O)C1 C1(NC(c2ccc(Cl)cn2)=O)C2CC3C(C2)C13C(=O)NC1CCCC(CO)C1 c1(C(=O)NCCOCCN(C(=O)Cc2cnccn2)C)ns[nH]c1=O Cc1nc2cc(C(=O)NCC(C)(CO)NC(=O)CC3CCC(=O)N3)cnc2[nH]1 Cc1cc(CC(=O)NC2CCC2NC(=O)CCCc2ccccc2)ccc1O c12ccc(cc1)o2.c1(C(N2CC(N(C(=O)CC3CC3)C)C2)=O)cccc(CO)n1 C(=O)(C(O)CC[S+](C)C)NC12CC(NC(c3nccc(N(C)C)c3)=O)(C1)C2 n1(C(COC)C)nc(CC2CCCC2)nc1-c1ccc(-c2cccc(Cl)c2)cn1 N1(C(c2c(COC)cccc2)=O)CC2CN(C(C3CC3(F)F)=O)CC2(C)C1 C#CC1(C(=O)NCCc2noc(=O)n2C)CCN(C(c2ncccc2F)=O)C1 c1(SC)ncc(Cl)c(C(N2CCN(C(c3cc4ncsc4[nH]3)=O)CC2C)=O)n1 N1(C(=O)NCC(C)(C)Oc2ccc(Br)cc2)C2CCC1C(N)C2 c1(C(N(C)CC)=O)ccc(C)cc1.c12cn(nn1)CCC1CN(C1)C(=O)C2=O CCC(C)C(O)C(C)C(=O)NC1CC2(C(=O)NCCC3COCCO3)COC1C2 N1(C(c2c(CC)cccn2)C(=O)NC(C)CC)CC2CC(O)CC2C1 C1(NC(C(C)N(C(CC)CO)Cc2cccc(Br)c2)=O)CC2CC3C(C2)C13 N1(C(C2(C)CN(C(CCn3ccc(C)n3)=O)C2)=O)CCC(F)(COC(C)C)CC1 C1(C(=O)NCC(CC(=O)NCC2COCCO2)C2CCC2)CC2(CCO1)CC2 c1(C(=O)NCC2C(NC(c3ccc(NCC)cc3)=O)C2)ccc2nncn2c1 c1(N2CCC(NC(CC)=O)C2)nc(N2CC3(C)COCC3(C)C2)nc2c1COC2 C1(C(=O)NC(CC#C)CC)CN(C(=O)C(F)n2ccnc2)CC1OC N1(C(CN(CCCCCC)C)=O)CCC(CNC(=O)CC2OCCC2C)C(C)C1 N1(C(COCC=C)=O)CCN(C(=O)Cc2ccsc2C)C(COC)C1 C1(NC(c2c(C)n(C)c(C3CCCC3)c2)=O)CC(=O)N2CCCCC12 C1(CC)CN(C(c2sc(C(C)OC)nc2C)=O)CCC1NC(=O)CCF O=C1NCCc2occ(C(N3CCCC3CCNC(C3CC4CCC3C4)=O)=O)c21 Cc1nc(Cl)ccc1S(=O)(=O)N(C1CN(CC2COCCN2)C1)Sc1ccccc1 S(=O)(=O)(c1ccc(N2C3CCCC2CC(O)C3)c(F)c1)NCc1ccc(C)cc1 C(=O)(CCCC(CC)NC(=O)C(CC1CCCC1)OC)N1CCC(OCC)C1 N1(C(c2oc(CC)c(N(C)C)c2)C(=O)NC2CC2)CCC2C(C(=O)OC)C2C1 N1(C(C(C=C)(C)O)=O)CCC(C=CC(=O)NCC(C)(O)CCO)CC1 Cc1nccc(C(=O)NCC2CC2NC(=O)COCC2CCCOC2)c1N N1(C(C2ON=C(C)C2)=O)CCC(NC(c2cc(Br)c[nH]2)=O)C(C)(C)C1 CCCC(C(=O)NC(CCC(C)C)C(=O)NCCN(CC(F)F)C)C(C)C c1(CN2CCC(C(N3C(CNC(CCC=CC)=O)CC3)=O)C2)ccccc1Cl C(=O)(C(C)CC(C)C)NC1CN(C(CCCOCCOCCOC)=O)CC1C C1(C(C)C(=O)N2CC(CC(C)(C)CNC(=O)CC3CCC3)C2)CCC(C)(C)CC1 N1(C(C2C(CCC)CCC2)=O)CC(C)(C)CC1CNC(=O)CC1CC(O)C1(C)C C(=O)(C(O)P(C)(C)=O)N(CC(C)NC(=O)COCCOC)CC c1(N2CC(C)(CNC(c3c(OC)cc(Cl)nc3)=O)C2)ncc2cn[nH]c2n1 C1(CNC(=O)CCCN2CCCC2)C2CC1N(C(C1(N3CCOCC3)CC1)=O)C2 Cn1cc(C(=O)NCCN(C(C2C3COCC23)=O)C2CC2)c(C(F)(F)Cl)n1 c1(C(=O)NC(CCCC)CNC(=O)CC2(C)CC(F)(F)C2)cc(O)nc(O)n1 Cc1nc2ccc(C(N3CC4CCCN(C(C5CC(C)CO5)=O)C4C3)=O)cc2o1 C1(CC(=O)NCC(CN(C(c2cnc(CCCC)s2)=O)C)(C)C)CCCCC1F c1(C2(C(=O)NCCC3CCN(C(=O)C(F)(F)CO)C3)CC2)ccc(F)c(Cl)c1 N1(C(C(=O)NCCC2(O)CN(C(C3N(C(C)=O)CCC3)=O)C2)C)CCCC(O)C1 c1(NCc2cccc(C(=O)OCC)c2)cc(-c2n[nH]c(C)n2)ccc1C c1(C(N2CCC(NC(C3(F)CC3)C3CC3)C2)=O)cccc(C(F)(F)F)n1 N1(C(C2CN(C(c3n(CC)ccn3)=O)C(C)CC2)=O)CC2CC(OC)C(C2)C1 C(COCc1ccccc1)(C(=O)NC1CC(F)(CNC(C2CCCO2)=O)C1)OC C1(C(=O)NC(C(CO)NC(Cc2c(C)cccn2)=O)C)COc2ccccc2O1 C1(OC)CC2CC1CN(C(C1CCC(C)C1)C(=O)Nc1ccc(F)cc1C)C2 C(=O)(C1CCCc2n[nH]cc21)N1C(CNC(c2ccc(C(C)C)cc2F)=O)CC1 CC1c2ccccc2CC1C(=O)NC1(CO)CN(C(c2cc[nH]c2)=O)C1 C1(C2CC(NCc3nc(C4CCC(C)N4C)on3)C2)SC2C=CC1CC2 N1(C(C(CC(=C)C)C)=O)CC(NC(=O)Cc2ccccc2Cl)CC2(CC2)C1 c1(NC(COc2cc(C)cc(C)c2)=O)nc2ccccc2n1C(C)C CCC(C(=O)N1CCCC1CN(C(C1CC1C)=O)CC)N(C)C c1(OC)ccnc(C(=O)NCC(C)CC(=O)N2CCC2CO)c1 CC#CC1CCN(C(=O)CC2CCCN(C(=O)CC=CCC)C2)C1 N1(C(C(CCC(C)C)F)=O)CCCC2C1CCCN2C(=O)CCN1CCCC1 CC1=C(C(=O)N2CC(F)(C(=O)NCC3CCOC3)C2)CCC1 n1(CC(=O)N(C2CCN(C(C3CCC(F)(F)C3)=O)C2)C)ccc2ccc(F)cc12 c1(C(N2CC3CC(C2)CN(C(=O)C(F)(F)F)C3)=O)nc(C2CC2)n2ccccc12 C1(CNC(CC2CCCN(C)C2)=O)CN(C(c2ccnc(S)c2)=O)CC12CCC2 C12(NC(COCC=C)=O)CCC(CN(C(c3cc(C)c(C)s3)=O)C1)C2 CCCCCC(=O)NCC(=O)NC(CNC(=O)C=CCN1CCC1)CC(C)C N1(C(CCCC(C)NC(=O)C2=NN(C)C(=O)CC2)=O)CCC2(CCN(C)C2)C1 CC(O)(CC(=O)N1CC2=C(C1)CN(C(=O)COC(F)(F)C(F)(F)F)C2)C(F)(F)F N1(C(C(C)S(C)(=O)=O)=O)C2CCC1CC(F)(CNC(=O)CCCNC(N)=O)C2 c1(C(=O)NC2CCN(C(C3C(CC)N(C)CC3)=O)C2)cc(O)nc2cnccc12 Cc1cc(N)ccc1C(N1CC(NC(=O)Cc2cnc(Cl)cc2C)C2(CC2)C1)=O C1(CNC(C(C)(C)C2CCCCO2)=O)CCN(C(C2CSC2)=O)CC1 C1(CNC(C2(C=C)CC2)=O)COCCN(C(=O)C(C)(C)c2cncs2)C1 Fc1ccc(Br)c(CNCC2C3CCC4C(C3)CC24)c1 c1(CNC(C2CCN(C(CC3(NC(C)=O)CC3)=O)C2C)=O)ccc(F)nc1C C1(C(N2C(COC)C(C)(C)C2)=O)CNC(=O)CN1C(=O)C(=O)C(C)C c1(C(N2C(C)CC(NC(=O)CC3CCC(=O)N3)C2)=O)ccn2nncc2c1 N1(C(COCCC)=O)CC(F)(C(=O)NCC(C)OCCO)C1 c1(C(C2(C)COC2)NCCSCC(C)Cn2cccn2)nnnn1C1CCC1 C1(CCNC(c2cn(C(F)F)cn2)=O)CCCN1C(=O)CNc1ccccn1 C(=O)(C1CCc2sc(C3CCCCC3)nc21)NC(CN(CC(=O)NC)CC)C CC(C)C(N=[N+]=[N-])C(=O)NCC1COC(CNC(=O)C(C)c2ccco2)C1 C1(NC(=O)Cc2ccsc2Cl)CCC12CN(C(c1cccn(C3CC3)c1=O)=O)C2 c1(C(N2CC(C(C)NC(C(CCOC)(C)C)=O)OCC2)=O)cc(C)c(F)cc1Cl c1(NC(C2CC(NC(C(C)C)=O)C2)=O)cc(Cl)c(C#N)cc1[N+](=O)[O-] N1(C(c2cc(C)[nH]n2)=O)CCC2CN(C(c3c(Cl)ccnc3C)=O)CC12 Cc1cc(C(=O)C(=O)NCC2CCC(F)C2)c(C)o1 N1(C(c2ccc(C)s2)=O)CCC2(CCOCC2)C(CNC(=O)C(C)CC(C)C)C1 C(=O)(CC(C(F)F)NC(=O)CCC(N)=O)N1CCC(NC(C)=O)CC1 c1(-c2ccc(CN(C3CCCC3)C(C3CCCO3)=O)cn2)ccc(F)c(F)c1 c1(C(N2CCC(N(C(c3csc(C(F)(F)F)n3)=O)CC)C2)=O)ccc(F)nc1F c1(COC)c(C(=O)NC(CNC(c2cnc(N(C)C)s2)=O)CC(C)C)cnn1C C1(C(N2CC(C(Cn3cc(COCCC#N)nn3)F)C2)=O)CC(=O)CC2CC12 C1(C(=O)NCC(C)(C)OCCO)CCN(C(C2CC2Cl)=O)C1 C(c1cccc(Cl)c1)=CC(=O)NC1(CO)CN(c2nc(C3CC3)ns2)C1 C1(NC(CCC2(NC(c3c(CC)nco3)=O)CCC2)=O)CCC(CC)CC1 c1(OC)ccc(CC(=O)NC2CC(NC(c3cc(Cl)nc(Cl)c3)=O)C2)cc1Br C1(NC(C(CC)(C)C)=O)CN(C(C2CN(S(N)(=O)=O)C2)=O)CC1C1CC1 Cc1nn2ccccc2c1C(=O)NCCCN(C(=O)C(C)(C)C(C)(C)C)C c1(C(N2CC(C)(NC(C=Cc3scc(C)n3)=O)C2)=O)nccc2ccsc12 C(=O)(C(C)C(=O)N1CCOCC1)NCC(Cc1ccccc1)NC(COCC)=O C(=O)(CC(C)CC(=O)NC(CC1CC1)C(=O)Nc1cccc(F)c1)OC C1(C(N2CCC(N(C(C(C)OCC=C)=O)CC)C2)=O)SC2C=CC1CC2 C(=O)(CCCn1cc(CCN)nn1)N(C(C)(C)C)CCF c1(CNC(C2(C)CC=C(C)CC2)=O)nc2c(s1)CN(C(c1ccoc1)=O)CC2 N1(C(CC=CCNC(C2C(CCC)C2)=O)=O)CC2C(C(=O)OC)C2C1 C1(NC(C(c2cccc(C)c2)C)=O)CCC(C)N(Cc2cc(C)on2)C1 C(=O)(C1Cc2c(Cl)cccc21)N1CCC(CCNC(CCC=C)=O)C(F)(F)C1 c1(C(=O)NCC2(F)CN(C(C34CCC(CC3)CO4)=O)C2)cc2ccc(Cl)cc2o1 N1(C(CCCN(CCC)CCC)=O)CC2(CC(NC(C3CCN(C)C3C)=O)C2)C1 C1(C(=O)NC(CNC(C2(CCCC)CCC2)=O)(C)CO)CS(=O)(=O)CC(=O)N1 CC(C)(C)C(=O)C(=O)NCC1CCCN1C(C1(Cl)CC12CCC2)=O C1(CCOC)(C(N2CCC(O)(CCNC(=O)C(C)(C)CF)C2)=O)CCN(C)CC1 S(=O)(=O)(c1cc(C(F)(F)F)ccc1C(=O)O)NC1CC2(CC(OC)C2)C1 C(=O)(C(CC)C(=O)N(C1CCCCC1NC(=O)C(F)=C1CCC1)C)OCC N1(C(c2cn(CCOC)nc2)=O)CC2C3CCC(C2C1)N(C(C1(Cl)CC1)=O)C3 CCC(C)(C)CC(C(=O)NCc1ccco1)N1CCC(CO)C(O)C1 C=CC1(CC(=O)NC2(C(=O)O)CCC2)CCC1 C1(C(N2CC(NC(C(C)(C)N(C)C)=O)C(F)CC2)=O)Cc2ccccc2C1 S(=O)(=O)(c1nc2c(s1)CCCC2)NC(C1(C2CC2)CC1)=O C(=O)(C(C)N(OC)C(=O)CCN(OC)C(=O)C1CN(CCC2CC2)C1)OC C=CCC(C(=O)Nc1nnc(C)n1CC)NC(=O)CCCNC(C)(C)C c1(C(N2CCC(=C)CC2C(N2CCCC(CCC)C2)=O)=O)cccc2ccnn12 C(COC(=O)C(Cc1ccccc1)C(=O)OC(C)(C)C)(CC(C)C)OC c1(C(=O)NCC2CCN(C(c3[nH]c(CC)c(Cl)n3)=O)C2)cc2cccn2cn1 CC(C)C(=O)NC(CNC(C1CCC1C(C)(C)C)=O)CO N1(C(c2cc(C)cc(Br)c2)C(=O)NCCCOC)CCc2ccc(F)cc21 N1(c2n(CCC#C)c(C3CCCCCC3)nn2)CCC(F)(F)CC12CCC2 N1(C(COCC)=O)CCC(C)(C)CC1C(=O)Nc1cnc(CO)nc1C C1(C(N2CCN(C(c3cc(O)cs3)=O)CC2)=O)CC12CCC(F)(F)CC2 CC(C)(O)C(O)C(C)(C)NC(=O)NCCOC1CCN(S(N)(=O)=O)C1 c1(C(C)=O)ccc(CC(=O)NCCC(C)(C)NC(=O)C(=Cc2ccco2)C)cn1 CCCCCCC(C)C(=O)NC12CCC(C(=O)NCCCn3cnnc3)(CC1)C2 C12(NC(CCCC)=O)CCCC1N(C(c1ccn(C3CCC3)n1)=O)CC2 C=Cc1cc(C(N2CC(NC(=O)CCCN3CCCC3)CC2C)=O)cc(F)c1 N1(C(C2(CC=C)CC2)=O)C2CCC1CC(C(=O)NOCCCC)C2 Cc1ccc(NC(c2ccc(C3(F)COC3)cc2)=O)c(CO)c1 CC1CCCC(CC(N2CCC(CC(=O)NC34CCN(CC3)C4)C2)=O)O1 C1(C(N(CC(C)NC(c2nccc(C)n2)=O)C)=O)CC(C2CCC2)C1 C1(NC(CCCOC(C)C)=O)C2CCC1N(C(=O)CC1CCCCN1C)C2 c1(CNC(=O)C(O)Cc2ccccn2)cccc(NC(C2CCC3(CC3)C2)=O)c1 C(CCNC(=O)CC1(CSC)CC1)(CNC(=O)C(C1CCCCC1)F)OC CCC1=NOC(C(=O)NC2(CNC(c3cc(C)c(C)[nH]3)=O)CCC2)C1 c1(OC)ccc(C(C)=CC(=O)NC(C)CN(C(=O)CSCCN(C)C)C)cc1 C1(OC)(CNC(c2csc(-c3cnn(C)c3)n2)=O)CCN(C(=O)CNC(N)=O)C1 C1(CC(=O)NC2CN(C(COCc3cc(OC)no3)=O)C2)CCCC(OC)C1 c1(SC)nn(C)cc1C(=O)NC1CCN(C(C2CCC(O)CC2)=O)CC1 Cc1cnccc1N1CCN(C(=O)NC(c2ccc(Br)cc2)C(F)(F)F)CC1 CC(CC(=O)N1CC(S(C)(=N)=O)C1)CC(C)(C)C.C12CC(O)C1CC(=O)N2 c1(C(=O)NCC(CN(C(C(C)CS(C)=O)=O)C)(C)C)ccc(F)c(O)c1F C(=O)(C(C)(O)CC(C)C)NC1CCN(C2CCN(Cn3c(C)ncc3)C2)CC1 c1(C(=O)NCC(CC(=O)OCC)C)cc(I)ccc1O Cn1nnc2c1CC(C(=O)NCCC1(NC(=O)CC3(O)CCOC3)CCC1)CC2 CC1CC(NC(C23CC(C)(CN2C(c2ccco2)=O)C3)=O)C(C)CN1C C(N=c1[nH]c(=NCC(F)F)[nH]c2c1COCC2)c1cccc(OCC#N)c1 C1(F)(C(=O)NC2CC(NC(C3CCC(C)CC3)=O)CC2O)CCCN(C)C1 CCS(=O)(=O)N1CC(C(=O)N(CCCC(=O)CC2CC2C)C)C1.C1(C(=O)N)(C)CC1 C(=O)(CCCS(C)(=O)=O)N1CC(NC(C2(CCCC)CCC2)=O)C2C1C2 C1(NC(C2(NC(c3cccc(F)c3F)=O)CCOCC2)=O)CC2OC(=O)CC12 c1(CC)cnccc1C(N1CC(NC(c2nc(Cl)sc2C)=O)C1)=O C(=O)(C(CC(F)F)NC(C1C=CCC1)=O)NCC(C)(O)CO C(=O)(CC(C)NC(N)=O)NC(C(=O)NCCC(=O)NC(C)C)c1cccs1 C1(C(N2CC(OC)C2)=O)C(C)CCN1C(c1cnccc1C)=O c1(C(N2C3CC(CN(C(=O)CCCC4CC4)C3)C2)=O)cnc2ncccc2c1 c1(NC(C)Cc2ccc(I)cc2)ccc(Cl)c(F)c1C(=O)N(C)C C#CCC(CC(F)F)NC(C1(F)CN(C(=O)C(C)(O)CCC)C1)=O n1(CC(=O)NCCN(CC(C)O)C(C2CCCSC2)=O)cc(C#N)c(O)nc1=O Cc1cc(=NCc2ccccc2CNC(c2c[nH]nc2C2CC2)=O)[nH]c(Cl)n1 N1(C(C(C(C)(C)O)NC(C(C)OCCOCC)=O)=O)CCC12CCOCC2 C1(C(=O)NC2C(NC(c3ccc(C(F)F)nc3)=O)CC2)CCc2nc(O)[nH]c2C1 c1(C(=O)NCC(C(C)C)NC(C2CCOC2=O)=O)cc(F)c2[nH]nnc2c1 C1(CNC(c2ccc(CCF)cc2)=O)COCCN(C(=O)CC2CCCC2)C1 C1(NC(C2C(C)OCC2)=O)CCOCC1NC(c1coc(Br)c1)=O CC(C)C(=O)C(=O)N1CC2C(NC(=O)C(C)Oc3ccc(Br)cc3)C2C1 C=C1CCN(C(=O)Cc2nc(=N)[nH][nH]2)C(C(=O)NCC2CC(O)C(O)C2)C1 c1(C(N(C2CCN(C(C3(CSC)CC3)=O)CC2)C)=O)ccc(S(C)=O)cc1 c1(NC(=O)NCC2CCC(NC(=O)COC3CC=CC3)C2)ccc(F)c(F)c1 c1(C(=O)NC2CN(C(c3ccc(C(OC)OC)o3)=O)C2)nccc2n[nH]cc12 C1(CNC(c2n[nH]c(C)c2Cl)=O)CN(C(C2COC(=O)N2)=O)CCC1(C)C C(CN=c1[nH]c(=NCC2CC3CCC(C2)S3)c2cc(Cl)ccc2[nH]1)CCN(C)C CC1CN(C)CCCN1C(C1CC2CC1CN(C(C1SCCS1)=O)C2)=O C1(C(N(C2CC(C#N)C2)CC(=O)NCC2CC(F)(F)C2)=O)CCC(CO)CC1 C1(NC(CC2(CC)CCC2)=O)CC(C(=O)NC2CC2CCOC)CC1O CN1CCCCC1C(=O)NCCC1CCCN1C(c1ccc(OC(F)F)cn1)=O C1(C(=O)NC(c2nc(C)[nH]n2)(C)C)(NC(=O)C(C)C2CC2)CCN(C)C1 N1(C(=O)CCC=CBr)CCN(C(c2cc(F)c[nH]2)=O)C2CCCCC2C1 C(=O)(C1CCCc2ncnn21)NC1C(CNC(=O)CCn2cccnc2=O)CC1 N1(C(C2CCN(CC)C2)=O)CC(C)C(C)(CNC(c2[nH]cc(C)c2C)=O)C1 C1(NC(C2C(C(C)(C)C)C2)=O)CCN(C(c2c(N)cccc2F)=O)CC(C)(C)C1 C1(NCCC2(C)CCNC2)C=CC2(CCCCCC2)CC1 Cc1ccccc1-c1nc(COCCC(=O)NCCCCCN(C2CC2)C)cs1 C1(C(=O)NC2C(OC)CN(C(=O)Cc3c[nH]nc3C)C2)COCC2(CCC2)O1 C1(C(N2CC(=C)C2)=O)CCC(C2CC2)N1C(C1(n2cnnn2)CC1)=O C1(CC(N2C3C(NC(=O)COCCF)C(C3)C2)=O)CCn2cncc2C1 c1(C(N(CC(CN(C(=O)CC2CCCN(C)C2)C)O)C)=O)cccc(C(F)F)c1 Cc1c(Cl)c(C(=O)NC2(CNC(C34COC(CF)(C3)C4)=O)CCOC2)nn1C Cc1cc(Cl)c(C(N2C3CCC2CC(NC(C2(C(C)C)COC2)=O)C3)=O)cc1C N1(C(c2cc(CCC)nn2C)=O)CCN(C(C2(CC)CCCC2)=O)CCC1C CC(=O)CCCC(=O)N1CCC(C)CC1CNC(c1cc(F)n[nH]1)=O Cc1cccc2cc(NC(=O)NCC(O)COc3c(F)cccc3F)c(O)nc12 N1(C(CSCCOC)=O)CC(NC(c2c[nH]c(Br)c2)=O)C2CC12 c1(C(=O)NC(CC)CN(C(=O)C(C)OCC2CC2)C)cccc(CC(F)(F)F)c1 n1(CCCC)nc(-c2ccccn2)nc1-c1csc(-c2csc(C)n2)c1 CC1CN(C(C2(C)CC3CCC2C3)=O)CCC1NC(=O)CCCc1ccccc1 c1(C(N2CCCN(C(c3cc(C)sc3C)=O)C(C)C2)=O)cnn2c1C(=O)CCC2 N1(C(C(CSCC)C)=O)CC2CC(CNCC3(C(=O)OC(C)(C)C)CC3)CC2C1 Cc1cc(F)c(C(N2C(C(=O)Nc3cnn4cccnc34)CCC2C)=O)c(F)c1 n1(C(C)C)ncc(C(=O)NC(C)C(C)NC(=O)CSCc2cccnc2)c1N C1(NC(CC=C)=O)CCCN(C(=O)C(O)Cc2ccccc2Cl)C1C c1(C(N(C2CCN(C(c3ccnnc3)=O)C2)CC)=O)ccnc2cc(Cl)ccc12 c1(C(n2ccnc2)CN2CC(O)(c3nccs3)C2)cccc(Cl)c1 c1(CSCC(=O)NCC2CC(NC(=O)Cc3cc(Cl)cs3)C2)ccc(F)cc1 N1(C(C(N)Cc2csc3ccccc23)=O)CC2(CCC2)CCC1CO C(=O)(C(C)(C)CNC(C1C2CC1N(C(C1(F)CCOC1)=O)C2)=O)NC C(=O)(C(C)(C)CC(C)C)N1CC(C(C(=O)NCC2CC(C)(C)CCO2)OC)C1 N#Cc1ccc(C2CCN(C(C3CC3C(=O)O)=O)C2)s1.c12ccc(cc1)s2 c1(C(N(C2CCN(C(c3cc(C(N)=O)cs3)=O)C2)C)=O)c[nH]c2ncnc(O)c12 C1(CNC(C(C=C)(C)O)=O)CC(C)(C)CN1C(=O)C(c1ccc(Cl)cc1)C c1(C(=O)NC2C(NC(C3CC(=C)C3)=O)CS(=O)(=O)C2)cccc2c1oc(=O)n2C C1(NC(c2c(C)noc2)=O)CCCCN(C(C2CCC2)=O)C1 N1(C(C(N2C(CC)CCC2)=O)=O)CCOC(c2ccc(NC(=O)COC)cc2)C1 Cc1sc(NCCN(CCCNC(c2cc(C(C)C)nc(C)n2)=O)C)c(C)c1C c1(CNC(C(CNC(C2(Cl)C(C(C)=O)C2)=O)O)=O)ccc(C)c(O)c1 n1(C(C)C)cccc1C(=O)NCC(C)(O)CNC(C1(C(N2CCCC2)=O)CC1)=O CC(C)CC(O)C(C)C(=O)NCc1cc[nH]c1C(N1CC(O)CC1(C)CO)=O N1(C(c2nc(OCC)sn2)=O)CCC2CCN(C(c3cc(CC)no3)=O)CC12 c1(C(=O)NCC(C(C)(C)C)NC(C2(OC)CCCSC2)=O)cc(Cl)c(C)cn1 CC1OC2(C)CC1(C(=O)NC13CCC1CN(C(c1ccc(N)c(Cl)c1)=O)C3)C2 c1(SCC)cccc(CC(=O)NC(C)Cn2cc(Cn3cc(Cl)cn3)nn2)c1 N1(c2nnc(CC)n2C(C2CC2)OCC(=O)N(C)C)CCC2C(C1)C2(F)F C(=O)(C1=NN(CC)C(=O)CC1)NC1N(C(CC(=O)NCC)=O)CC2(CC2)C1 C1(NC(C2C(C=C)C2)=O)CC(NC(C23CCC(OC)C2C3)=O)C(O)C1 C1(C(=O)OCC)CCC2(CC(C(=O)NCC3(OC)CCCCC3)C2)N1 C1(NC(c2ccc(F)s2)=O)CC2(CCN(C(=O)C3=CCCOC3)C2)C1 N1(C(C2C(OC)CCC2)=O)CCCN(C(c2cnc3nccn3c2)=O)CCC1 c1(OCC(=O)NCc2cn(C(CCCC)CC)nn2)ccc(F)cc1N c1(C(=O)NCCOC2CCN(C(c3c(CC)nc[nH]3)=O)C2)ccc(C)nc1O C1(CC)C(C(=O)NC(c2ncccn2)CC)CCCN1C(c1c[nH]c(=O)cn1)=O CC1=C(C(=O)N2CC3CN(C(=O)CCCC(C)C)CCC23)COCC1 N1(CC(=O)Nc2n(CC)nc(C(C)(C)C)c2)CCc2cccc(O)c21 O=S(=O)(c1cccc(N2CC=CCC2)n1)NCC(C(F)F)c1ccccc1 C1(O)(C(C)NC(C=CCCC)=O)CCN(C(=O)CC2CCC(C)CO2)CC1 Cc1cc(C(=O)NC(C(N2CC3(CCCO3)C2)=O)C2CCCC2)ncc1N C1(NC(=O)Cc2cc[nH]c2)(CO)CCCN(C(=O)CCF)C1 c1(C(=O)NC2CN(C(C3N(C)CC(O)CC3)=O)CC23CC3)ccnc2c1CCO2 C(=O)(C(C)CC(C)C)N(CC(C)NC(C1CC(OC)C1)=O)CC C(C)(C)(C=CC(=O)OC)NC(C1(C(=O)OCC)C(CCC)C1)=O.c1(CN)ccccc1 C(=O)(C1CC(C)(C)Oc2ccccc21)NC1(C)CN(C(C(COC)OC)=O)C1 c1(C(=O)NC23CCN(C(c4c(C)nc[nH]4)=O)CC2C3)cc2c(o1)CCCNC2=O c1(CC(=O)NCC2CCCN2C(=O)CCN2CCOC2=O)ccc(CO)cc1 C1(C(=O)NC(C)CSC(F)F)CCCCCC1NC(c1cc(O)nc(O)n1)=O C1(CCNC(C2CCCC2(F)F)=O)CSCCN1C(c1cnsc1)=O c1(OC)nc(C)c(Br)cc1C(C(=O)NCC(C)C)N(C)CC1CCCC(F)(F)C1 c1(NC(C2CCC(NC(=O)CCC3CC3)CO2)=O)cc(F)c([N+](=O)[O-])cc1F c1(OC)ccccc1-n1nnnc1C(c1nccn1CC)NC1CC12CC(O)C2 c1(C(N2CCC(NC(C(c3ccc(Cl)cc3)C)=O)CC2)=O)c(Cl)nn(C)c1Cl C1(NC(C2N(CC#C)CCC2)=O)CC2CC(C1)N(Cc1csc(C3CC3)n1)C2 c1(C(=O)NCC(CC=C)NC(=O)CC2CCCCN2C)c(F)ccc2n[nH]cc12 N1(C(C2(C#N)CCCC2)=O)CC(F)(F)CC1C(=O)NCCCN1CCCCCC1 c1(CC)c[nH]c(C(=O)NC(C)CNC(C2(c3ccccc3)CC2)=O)c1 N1(C(CC(C=C)C)=O)CCC2(CC2NC(c2cc(C3CC3)no2)=O)C1 c1(OC)ccccc1C(CNC(C1(CCO)CC1)=O)NC(c1nc(C)sc1C)=O c1(OC)cc(CN(C)C(=O)NCc2ccc(C(F)(F)F)nc2C2CC2)ccc1C c1(CNC(C(C)Oc2c(C)cccc2)=O)ccc(Cl)c(OC(F)F)c1 C(CC(C)(C)CNC(C1C=CCN1C(=O)C(C)NC=O)=O)OC N1(C(C(n2cc(CC=C)nn2)C)=O)CCCC(CN2CC3CC2(C(F)(F)F)C3)C1 Cc1cc(S(=O)(=O)N2CCOCCC2)ccc1-c1cc(F)ccc1C C#Cc1ccc(C(=O)NCC2CCN2C(=O)C(C)N(C)C(C)=O)cc1 N1(C(Cc2ncc(C)[nH]2)=O)CCC2(CCN(C(c3cnc(N)c(Cl)c3)=O)CC2)C1 c1(C(N(C2CC(NC(C3C(=C)CC3)=O)C2)C)=O)cc(Cl)cs1 Cn1ccc(CNC(N2CC(c3nc[nH]n3)C2)=O)cc1=O N1(CCNC(C2CC(CNC(C3C(=C)C3)=O)OC2)=O)CCCC(O)C1 c1cc2n[nH]cc2cc1-c1nnc(CC2CC2)o1 c1(C(=O)NC(c2nc(-c3cccc4c3COC4=O)no2)C)ccc2c(c1)C(=O)NCC2 C1(C2CN(C(C3CC3Cl)=O)C2)(NC(C2CCCCC2)=O)CC1 C1(OCC)COCC1N=c1[nH]c(=NCC2CCCN(C)C2)[nH]c2ccsc12 CCCC(C(=O)NC1C2CN(CC(CC)OC)CC12)S(N)(=O)=O c1(CN)cccc2c1CCN2C(c1cnnn1-c1cc(Cl)ccc1Cl)=O c1(N(C(=O)CN2CCCC2)C(=O)OCC)cccc(F)c1N c1(COC)cc(C(=O)N(C(C)CNC(=O)CCN2CCCC2)CC)c(C)o1 c1(C(N2C(CNC(C(CCCOC)C)=O)CC(F)(F)C2)=O)cc(C)c(O)c(C)c1 C(CCC)(CC(=O)NC(C)CC(C)C(F)F)NC(CCC)=O N1(C(CCCN(C(C)C)C)=O)CCN(C)CC1C(=O)NC1CN(C(N)=O)C1 N1(C(CC(CCSC)O)=O)CC(CNC(=O)CN2C(=O)CCC2=O)CC12CCC2 c1(C(=O)NC(c2cnn(C)c2)C(=O)NC(c2cncnc2)C)cnn(C)c1N c1(C(N2CC(O)CC(NC(C3CC4(CCC4)C3)=O)C2)=O)c(Cl)ccc2ccoc12 C=CCCC(C)(C)CNC(c1cncnc1-c1ccccc1)=O N1(C(Cc2ccc(C(C)C)cc2)=O)Cc2[nH][nH]c(=NC(=O)c3cnco3)c2C1 c1(C(=O)NC2(CNC(COCCOC)=O)CC2)cccc(CN(C)C)c1 N1(S(Cc2cccc([N+](=O)[O-])c2)(=O)=O)CC2CCCN2Cc2ccccc21 Cc1cc(Cl)c(C(=O)NC2CN(C(=O)C(C)n3ccnn3)CC2O)cc1C C1(C(C2CCCC2)C)CCCN(CC(=O)NCCNC(=O)OCC(F)(F)F)C1 Cc1cc(C(=O)NCCC(O)C(=O)NCC2(C)CC=CCC2)c(C)cn1 CC1NC(=O)CCC1CNC(C1CCN(C(C2CCCCC2)=O)CC1)=O CC1CC2(CC(C(N3CCCC(NC(C4(Cl)CCC4)=O)C3)=O)C2)C1 C(C(C)(CC(=O)O)NC(=O)C(C(C)C)OCC1CC1)OC c1(C(=O)NCCC2CC(C(=O)NC(CSC)(C)CO)C2)nc(C)ccc1C C#CCCCCS(C)(=O)=NC(=O)CC1CC(C)(C)OC(C)(C)C1 CC1CC(NC(=O)C=CC2CCCN2C(=O)CN2CCCCC2)CCC1(C)C C1(C(=O)NC2CON(CC)C2=O)CN(C(=O)CSC(F)F)CCC1(C)C C1(NC(C2C(NC(C(CCC)OCC)=O)CCOC2)=O)CCC(N=[N+]=[N-])CC1 c1(C(c2n(CC(=C)C)nnn2)NCCCC(C2CC2)OC)ccccc1C(C)C Cc1ccc(-c2nc(C)c(NCC3OCCC3C(=O)OC(C)(C)C)s2)cc1 c1(-c2cc(C(=O)NC3C(NC(C(CSC)O)=O)C3)on2)ccc(Cl)cc1 N1(C(c2n(C)ccn2)=O)CCC2C(CCN2C(=O)Cn2cnc3ccccc23)C1 S(=O)(=O)(c1c(F)cc(F)cc1F)N1C(C(N2CC(O)C2)=O)CC(F)C1 CC(CCCN=c1[nH]c(=NC(CF)CF)c2c(F)cccc2[nH]1)c1ccccc1 C1(CN(C=O)Cc2cccc(OC(F)(F)F)c2)CC2OCCC2O1 c1(OC)cc(N(C2CC3CNC2C3)C(c2[nH]ccc2C)=O)c(Br)cn1 c1(C(N(C2CCN(C(c3nc(CCC)oc3)=O)C2)CC)=O)nnn2c1CCC2.CC N1(C(c2c(F)ccc(OC)c2)=O)CCCCC(NC(=O)CC(C)SC)CC1 c1(C(=O)NCCCN(C(CCCCC=CC)=O)C(C)C)nnn2c1CCCC2 N1(C(Cc2c(C)n[nH]c2C)=O)CC23CCCC2(C1)CN(C(=O)CSC(F)(F)F)C3 C(=O)(CC(C)(C)C(F)F)N1CC(C)C(CNC(=O)CSc2nncs2)CC1 C1(C(C)C)CCC(C(=O)NCC(C)NC(C2(CSC3CCCO3)COC2)=O)CC1 Cc1cccc2nc(CC3CCCN3C(=O)CSC3(C)NC(=O)NC3=O)[nH]c12 Cc1nn(C)c2cc(NC(N3CC(=O)N(Cc4cnc5c(c4)CCCC5)C3=O)=O)ccc12 C1(COC)(CNC(c2n[nH]c(C)c2C)=O)CCCN1C(c1[nH]cnc1C)=O Cc1cc2[nH]c(C(=O)NC3C4CC3CN(C(c3ccc(F)cc3Cl)=O)C4)cc2o1 C=CC1OCCCC1C(=O)NCC1CCN(C(=O)C(CC)=CC)C(C)C1 CCC(CCC(=O)NC(C)CC(C)O)NC(c1cccc(OC)c1)=O c1(SC)nc(N2CCC(NC(C3CCN(C)C3=O)=O)C(C)C2)cc(Cl)n1 c1(CN(CC(=O)NC(C)CCc2ccncc2)C)ccc(N(C)C)cc1 C(CC(=O)NC1CC1c1cncs1)(CC(C)C)NC(c1c(C)nncc1)=O C(c1ccccc1C#N)=CC(=O)NCC1OCCCN(C(C(CC)O)=O)C1 c1(OC)ccc(CNC(Cc2nonc2C)C(C)C)cc1O C=CCC(C)C(=O)NCCCC1(NC(=O)CCc2nc(-c3ccco3)no2)CC1 c1(C(=O)NCC2N(C(C(N3CCCCCC3)C)=O)CCC2)cncc(N)n1 CC(C)(C)CC(F)C(=O)NC1CCCC(C(N2CC(=O)NC(=O)C2)=O)C1 c1(C(=O)NC2C(NC(C(C)OCC(F)(F)F)=O)C2)ncc(F)cc1N c1(CC(=O)N(C2C(N(C(=O)C(O)C(F)F)C)CCCC2)C)ccn2cncc2c1 C1(CNC(c2cnc(CC)s2)=O)CCN(C(C2CC2c2cccnc2)=O)CC1C C=C1CC(C)(C(=O)NCC2OCCC2C(=O)Nc2csc(C)c2)C1 Cc1csc(CC2(C(N3CCC(Cc4cccs4)C3)=O)CC2)n1 c1(C(C(=O)NC2C(NC(C(CSC)(C)C)=O)C2)C)ccc(F)c(Cl)c1 Cc1nc(C)n(CCCC(=O)NCCC(C)NC(=O)C=CC(=O)N(C)C)n1 c1(C(N(C(C(=O)OC)CCF)C)=O)cc(C)nc(C)c1.C12(CC1)C(=O)N2 C(=O)(C#CC1CCOC1)N1C(CCC(=O)NCC(c2cnn(C)c2)C)CCC1 C1(C(=O)NCC(CCC)(C)O)CC(C)CN(C(=O)C(C)(C)CCSC)C1 c1(NCc2c(C)ncs2)[nH]c(=NCC2CCCC3(CC3)C2)nc2c1ncn2C(C)C CC(C)(O)C(C)(O)CNC(=O)CC1CC(C(F)(F)F)C1 CC(F)(F)C(C)(C)CC(=O)N1CCC2CC1CN(C(c1ccc(Cl)c(F)c1)=O)C2 N1(C(CN(C)S(N)(=O)=O)=O)CCOC2(CCN(C(C3CCC(CO)CC3)=O)C2)C1 Cc1c(C(N2CCC(CCCNC(=O)C(CO)NC(N)=O)CC2)=O)ncn1C C1(CC)CN(C(c2ccc(OC)nc2Cl)=O)CCN1c1ncccn1 CC1CCCCC1CC(=O)NC1CC1(Cl)Cl.N12CCN(CC1)Cc1cn(nn1)CC2 c1(OC)cc(C(=O)NCC2CN(C(c3cnc(C)[nH]c3=N)=O)C2)ccc1[N+](=O)[O-] c1(C(C(=O)NCC=C)N(CCC(N)=O)CC)cncn1C N1(C(C2CC3(CC3)C2)=O)CCC2(CCC(NC(C34CCCN3CCC4)=O)CC2)C1 CC(C)(CNC(C1CCCO1)=O)CCNC(c1ncoc1C1CC1)=O C#CCC(C(=O)NC(CCF)C(=O)NC(c1ncc(C)cn1)C)C1CC1 c1(C(=O)NCC(c2ccc(C)cc2)NC(=O)C(C)(C)C(C)C)cncc(C#N)c1 C12(NC(Cc3c(C)cccc3Cl)=O)CCCN(C(C3CCCC3)=O)CC1C2 C(=O)(C#CC(C)(C)O)N(C)CC1CCCCN1C(c1cn(C(F)(F)CO)nn1)=O c1(CC)ncc(C(=O)N(C2CCC(NC(c3nc(O)sc3C)=O)CC2)C)c(O)n1 C(N=c1[nH]cnc(Cl)c1OC)C1CCC(NC(=O)CC2CC3CC3C2)C1 C1(C)(CNC(C2(NC(=O)OC)CCCC2)=O)CCN(C(c2cnn(C)n2)=O)C1 c1(C(N2CC(C(C)NC(C(C)OCC)=O)C2)=O)cc(C#N)c(F)cc1F C1(NC(C=CSC)=O)(CNC(=O)CCC2CCCC(O)C2)CCCCC1 C1(C(=O)SCC)CCCCC1NCCOC1CN(C(=O)C(CCSC)N(C)C)C1 C1(C)(C(NOCCC=C)=O)CCCN(C(C2CC(=O)OC2(C)C)=O)C1 N(C(=NCCc1ccsc1)NCC(C)(C)C)Cc1n(C)nc(C(F)(F)F)n1 C(=O)(CC(C)C(F)(F)F)N1CCC(OCCNC(C2(COC)C=CCC2)=O)C1 CCCC(O)C(CO)NC(=O)C1=CCN(C(c2n[nH]c(C)c2C)=O)C1 N1(C(c2n(C)c(S)nc2)=O)CC(NC(=O)Cn2cnnc2)C2CCCCC12 N1(C(c2c(CC)n(C)cc2)=O)CC2CCCC1CN(C(=O)Cn1cnnn1)C2 C1(NC(C2C(C)C2C)=O)CC2(CCN(C(C3C4CCCCCCC34)=O)C2)C1 N1(C(c2ccn(C)c2CC(=O)O)=O)CCn2cc(C(=O)NC3CCOC3)nc2C1 N1(C(C2(CCC)CCCC2)=O)CC2(C)CN(C(C3(NC(N)=O)CC3)=O)CC2(C)C1 N1(C(CC=C=C)=O)CCC2(C1)CN(C(c1cn3cccc(C)c3n1)=O)CC(C)O2 N1(C(CC(C)C2CC2)=O)CCC(CNC(c2ccn3ncnc3c2)=O)C12CCC2 N1(C(c2cc(Cl)ns2)=O)CCC2(C1)CN(C(C1CCC1c1nc[nH]n1)=O)C2 C1(NC(=O)CCc2cc(Cl)cs2)CC2CCC1(NC(=O)C(C1(O)CCCC1)F)C2 N12CCC(CC1)NC(=O)C2C.n1(CC#C)cc(C(=O)NCCOC(C)(C)C)cn1 C1(CNC(c2nccc(C)n2)=O)COCCN(C(=O)C(C)C2(O)CCC2)C1 c1(CC(=O)NC2CC3CC2N(C(c2ccco2)=O)C3)ccc(Br)cc1F Cc1ccc(CC(=O)N(C)CC2C3CN(C(=O)C(C)(C)CO)CC23)cc1Br CCC(CCC(=O)N1CC(C(F)Cn2cc(C(C3CCOCC3)C)nn2)C1)OC c1(CNCc2cc(Br)sc2)cc(N2CCCC2)ccn1 C(CCN=C(NCCCN(C)C)NCC1CCC(C)O1)SC N1(C(c2ccc(OCC)nc2O)=O)CCC(=C(F)F)CC1 N1(C(C=CC(CC)=CC)=O)CC(NC(C2(OC)CCSCC2)=O)CC1C N(C1CCCn2cnnc21)C(=O)Nc1c(OCC)nccc1 N1(c2nc(C)nc(Cl)c2)CC(NC(=O)C2=C(Cl)CC2)C2CCCCC12 C1(C#C)(C(N2C(C#C)CC2)=O)CCN(C(=O)C(C)C(C)COC)C1 C1(N(C(c2c(C)nco2)=O)C)CCCN(C(C2CCCS2)=O)C1 N1(C(CCC(C)(C)NC(C(n2ccc(C)n2)C)=O)=O)Cc2cccc(F)c2C1 c1(N(C(C2C(NC(CCOC)=O)CCC2)=O)C)cc(C)cc(F)c1 C#Cc1ccc(C(=O)NC2(CCOC)CCN(C(c3conc3CC)=O)C2)cn1 c1(CC(=O)NC2(CO)CCC2)ccc(CN2CCC(c3ncc[nH]3)CC2)cc1 C1(NC(c2oc(C)c(CO)c2)=O)CC2CCC1N2C(=O)C(O)C(C)(C)C C1(CNC(CSC)=O)CN(C(=O)C(c2c(C)cccc2C)O)CC12CCOCC2 N1(C(c2cc(C)[nH]n2)=O)CCN(C(=O)C(c2ccc(Cl)cc2Cl)O)CC1C(F)F N1(C(C=CC)=O)CCC2C1CCCN2C(=O)C(C)NC(=O)C(C)(C)C C1(C(=O)NCC(C)N(c2ncc(C)c(O)n2)C)CC2(C1)NC(=O)NC2=O N1(C(CC(C(=O)OC)(C)C)=O)CCC2(CCC(NC(C3CC4(CCC4)C3)=O)C2)C1 N1(C(C(C)N(C(c2ccn(CCF)n2)=O)C2CC2)=O)CCCC2(CC2)C1 N(C)(S(=O)(=O)N(C)C)CC(=O)NC1(CCO)CN(C(C=Cc2nc(C)sc2)=O)C1 C1(N(C(C(C(C)C)SC)=O)C)CCCCN(C(c2ccc(C)nc2O)=O)C1 C1(C(=O)OCC2CCN(c3ccccc3F)C2=O)CCN2CCOCC12 c1(C(=O)NCC(=C)CCNC(=O)C(C)(c2cccs2)N(C)C)ccc(Cl)c(F)c1 C12(CC(N3CCC(OC)C3C(C)C)=O)CCC1CN(C(C1CCC1C#N)=O)C2 c1(NC=O)ccc(C(=O)NC2CN(C(c3cc[nH]n3)=O)CC2F)cc1 N(C1c2ccccc2CC1NC(=O)C=CC1CCC1)C(c1cncn(C)c1=O)=O N1(C(CC2(OCC)CC2)=O)CC(O)CCC1C(=O)NC(c1nncn1C)CO c1(C(=O)NC(CN(C(C(C2CC2)OCC)=O)CC)C)cc(I)c[nH]1 C(N=C(NCC1(O)CCOC1)NC1CCCCC1)c1ccc(CN(C)C)s1 N1(C(c2n(CCOC)ncc2)=O)CCC(C)(NC(c2cc(Br)ccc2F)=O)CC1 c1(C(=O)NCC(CCOC)NC(=O)CCC2CCCN(C)C2)cncc(C)c1C N(C1CCCc2cc(Nc3ccnc(C#N)n3)ccc21)C(=O)OC(C)(C)C C12(NC(CC3CC(SC)C3)=O)CCCCCC1N(C(=O)C=Cc1ccn(C)c1)CC2 CCCC(CCCNC(C1CC1C)=O)NC(=O)C=Cc1cncs1 c1(C(=O)NC2CN(C(CCCCC)=O)C(C)(C)C2)cnc2n1CCOC2 N1(C(CSC)=O)CCC2(CCOC2)C(CNC(c2n[nH]c3cc(C)ccc23)=O)C1 c1(C(=O)NCC2(NC(CN3C(C)CC3)=O)CCOC2)ccc(Cl)cc1Br CC1(CCNc2cc(C(F)F)ncn2)CCN(C(=O)Cc2cccc(Cl)c2)C1 n1(CC)nc(C(C)C)cc1C(=O)NCCC(C)NC(C1CCC1n1ccnc1)=O CC(CC(=O)N1CC(C)(NC(C2CCN2C)=O)C1)C(F)F N12CCCCCC1C2=O.c1(CC)[nH]ccc1C(=O)N(CC)Cc1ncnn1CC C(C)(C)(C(C)CC(=O)NCc1noc(C(C)C)n1)NC(CC(CC)SC)=O C1(C(N2CC(CNC(C(C)OCC3CCCCO3)=O)C2)=O)CCC(C)(C)CC1 CCCCC(CCCC)NC(C1C(C)OCCN1C(c1ccnn1C(C)C)=O)=O N1(C(CCCOCC=C)=O)CC2(CC2)CC1CNC(=O)C(C)(C)c1cnn(C)c1 C1(C(=O)NCCNC(=O)NC2(OCC)CCCC2)CCCC(C)(C)CC1 N1(C(C2=C(C)CC2)=O)CC(O)C(O)C1CNC(c1cccc(C(N)=O)n1)=O c1(C(N2CC(O)(Cc3cn(CC(=O)OCC)nn3)C2)=O)cc2c(Cl)cccc2[nH]1 c1(C2(CNC(N3CC4C(C)(COC4)C3)=O)CCCC2)ccc2c(c1)OCCO2 C1(N(C(C2N(C(c3c(C)cco3)=O)CCSC2)=O)C)CN2CCC1CC2 N1(CC(=O)NCC(n2cc(CC3CCNCC3)nn2)C)CC2C(N(C)C)C2C1 c1(CC(=O)N(CCNC(=O)CNS(=O)(=O)NC)CC)c(C)[nH]c2ccccc12 CCC(C)C(C(=O)N1CCC(NC(=O)CC2(C(=O)OC)CCCCC2)C1)OC CC1CN(C(C2CC2c2cn[nH]c2)=O)C(C)CN1C(=O)CC1CC2C=CC1CC2 C1(NC(C(=Cc2cnc[nH]2)C)=O)CCC(F)(CNC(=O)Cn2cnc(C#N)n2)C1 CON1CC(C(N2CC(F)CC2CC(=O)NCC2CC3(CCO2)CC3)=O)CC1=O c1(C(C(=O)NCCC2(C)CC2)N(C2C(C)CCC2)C)cccc2c1OCC(=O)N2 c1(C(=O)NCC(CN(C)C(c2ncoc2C2CC2)=O)O)sc(F)cc1Br S(=O)(=O)(CCC(F)(F)F)N1CC2CN(C(C=CCCCCC)=O)C2C1 N1(C(C(CCC)c2ccc(Cl)cc2)=O)CC2(CNC(=O)C=C(C)C)CC1CCO2 c1(CCCNC(=O)C(=O)NC2CCCC2)ccc(F)cc1Cl N1(C(C(C)OC)=O)CCCCC1C1CCN(C(C2CN(C)C2)=O)CC1 C12(CCCSC1)NC2.S(=O)(=O)(CCN(C)C)N(CC)CC C1(CC(=O)N)CN(C)C(=O)N1.C1(CNC(=O)C(=O)NC)CCCC1NC(CCN)=O CC(F)CC(=O)NCC(Cc1ccccc1)NC(c1csc(Cl)n1)=O CCCC(C)C(=O)NCCN(C(C)C)CC1CCCCCC1 CCC(CC(=O)N(C1CCN(C(C2CC2C(=O)OC(C)(C)C)=O)C1)C)OCC C1(O)(CNC(c2nccc(CC)c2)=O)CCCN(C(c2ccncc2)=O)CC1 c1(OC)ncc(C(=O)NC(C)CCCNC(c2coc(C(C)=O)c2)=O)c(C)n1 c1(C(=O)NCC2(NC(CC3CCCN(C)C3)=O)CCOC2)cc(F)c(Cl)cc1Cl c1(C(N(CC(N2C(C)(CCCO)CC2)=O)C2CC2)=O)cc(CO)ccn1 N1(C(C2N(C(c3ccn(C)c3)=O)CC(O)CC2)=O)CC2(CCCCC2)C1 N1(C(C)=O)CC(O)CC1C(=O)NCC1(F)CN(C(=O)CCC(=O)C2CC2)C1 N1(C(C(CC#C)NC(c2ccc(CF)cc2)=O)=O)CCN(CC)C(C)C1 CCC(C)C(=O)NCC(C)(C)CC1CN(C(=O)Cn2cncn2)C1.C1(=O)CN1 N1(C(COCC)=O)CCC2C(CCN2Cc2ccc(C)nc2Br)C1 S(=O)(=O)(c1ccc(NCC2CC=CC2)cc1Br)NCc1c(C(C)C)noc1 C1(C(=O)NCCN(C(=O)C(C)(C)C2CCOC2)C)CC(=O)OC1(C)C C1(CNC(c2cnc(C(C)(C)C)s2)=O)CC(F)(F)CN1c1nnc(C2CC2)s1 N1(C(C2N(C(C3N(C)C(=O)CC3)=O)CC=C2)=O)CC(F)(F)C(F)(F)C1 C1(C(N(C2CCCN(C(C3CC(=C)C3)=O)C2)CCO)=O)CCc2ccccc2C1 c1(NC2C(CC=C)CCCC2)cc(N2CCCC(F)(C(=O)NC)C2)nc(C)n1 CC1CCCn2c(C(=O)NCC3CC(NC(=O)Cc4cnc[nH]4)C(O)C3)cnc21 C1(CC(=O)NC2C(CC(C)(C)C)CN(C(=O)CC(C)(C)F)C2)CC2CCC1CC2 C(=O)(CC(CC1CC1)NC(=O)CC(Cl)Cl)NC(C#C)(C)C1CCC1 Cc1nn(C)c(C(=O)NC23CC2CN(C(=O)CNC=O)C3)c1[N+](=O)[O-] c1(C(N2CC(CNC(c3ccc(CC)o3)=O)C(C)CC2)=O)ccc2ccsc2c1 c1(CC(=O)NCC=CCNC(C(c2n(C)ccc2)=O)=O)ccc([N+](=O)[O-])cc1Cl N1(C(=O)NCC23CC2CN(Cc2cccc(C4CC4)c2)C3)CCS(=O)(=O)CC1 N#Cc1c[nH]c2c(F)cc(F)cc2c1=NCC(O)COc1ccc(F)cc1 c1(OC)c(C(=O)N(C)CC2CCCN2C(C2CC23CCOCC3)=O)cccc1Cl C1(NC(c2cn(CCC)nc2)=O)CC2CCC1N(C(=O)Cc1ccncc1Cl)C2 n1(C2CC2)ncc(-c2ncno2)c1Nc1ccccc1.C(COCCS)OC C(=O)(CCCC(=O)N(CC)CC1(F)CCN(CC(=O)N(C)C)CC1)NCCC c1(C(N2CC(n3cc(CCCCC)nn3)C2)=O)cccc2nnn(C)c12 c1(CN2CCC(NC(c3n[nH]cc3[N+](=O)[O-])=O)C(F)C2)cc2ccccc2cn1 C(=O)(C(C)C(O)C(C)C)NC1C(C(=O)NC2CCN(CC)CC2C)CC1 C1(C(C(=O)N(CC(C)NC(C2(CCC)CCC2)=O)C)C)CCOCC1 Cc1cc(N)c(C(N2CCCC(NC(=O)CC3CC3(Cl)Cl)C2C)=O)cc1C C1(NC(C2CC(OC)C2)=O)CC(C)(NC(=O)C=CC2CCC2)C1 c1(OC)cncc(C(=O)NC2CC(N(C)C(c3ccc(C(N)=O)nc3)=O)C2)c1 Cc1ccc(C(=O)NCC(C)CNC(=O)COc2cccnc2)nc1 C1(CNC(C(C)(C)OCC)=O)CC(NC(=O)C=CCOCCOC)C1(C)C c1(OCC(=O)OC)ccc(NC(c2ccc(-c3n[nH]c(O)n3)cc2)=O)cc1OC N1(C(c2cnc(OC)nc2C)=O)CC(C)CN(C(c2csnn2)=O)CC1C C1(CNC(COCCN(C)C)=O)(CO)CCCN(C(C2CCCO2)=O)C1 C1(OC(C(=O)NCC(C)NC(c2cnn(-c3ccccn3)c2)=O)C)CCCCC1 c1(N2CCCC(C(C)C)CC2)nc2c(c(=NC3CCN(C)C(=O)C3)[nH]1)SCC2 CC1CCC1C(=O)N(CCC(=O)N1CC(c2nn[nH]n2)C1)C1CC1 CCCCCC(C)(C)C(=O)NCC(C)(O)CNC(c1c(C)[nH]c2ccccc12)=O c1(N2CCN(C(COC)=O)CC2)[nH]c(=NCc2cnc(C)cn2)nc2sccc12 C1(C(=O)NCCN(C(C(C)NC(C2CCOCC2)=O)=O)C2CC2)CCS(=O)(=O)C1 C1(N(C(C2CCC(C)(CC)O2)=O)C)CCC2CN(C(c3ccc(F)s3)=O)CC12 C1(CC(=O)N(C)CC2(CNC(=O)Cc3ccccn3)CC2)CCCCCCC1 N#Cc1cc(C(F)(F)F)cc(CN(CCS(=O)(=O)N2CCCC2)C(C)(C)C)n1 Cc1csc2ncnc(NCC3CN(C(C4CCNC4=O)=O)CC34COC4)c12 CC1=NNC(=O)C1CCC(N1CCC(NC(=O)C(C)C(C)C)CC1)=O CCCCCC(CC)C(=O)N1CC(NC(c2ncsc2CC)=O)CC12CCCC2 c1(C(=O)Nc2c(OCCC)cccc2)ccc(S2(=O)=NCCC2)cc1 CC(C)(O)C(F)CNC(=O)C(C1CC=CCC1)NC(=O)Cn1[nH]cnc1=N CS(=O)C=CC(=O)N(CCNC(C1CSCCS1)=O)Cc1cccc(Cl)c1 Cc1cc(C(N2CCC(N(C(=O)COC(F)(F)F)CCO)CC2)=O)c(C)s1 N1(C(Cn2c(C)ncc2)=O)CCC2C1CCCN2S(=O)(=O)CCC(F)(F)F N1(C(C=CC=CCCCCC)=O)CCC(C2(NC(C3CN(C(C)=O)C3)=O)CC2)C1 C1(CCOC)(NC(=O)C(F)C(F)(F)F)CCN(C(c2coc(N(C)C)n2)=O)CC1 c1(Nc2ccc(NC(C3N(C)C(=O)OC3)=O)cc2)ncc2ccsc2n1 c1(-c2cccc(C(=O)NCCCCN(C)C)c2)cccc2c([N+](=O)[O-])cccc12 c1(OC)nccc(I)c1CNCC1(NC(=O)CN2C(=O)CSC2=S)CCC1 N1(C(CCC=C)=O)CC(NC(=O)Cc2c(CC)noc2CC)C(F)(F)C1 c1(C(=O)NCC2C(NC(c3cncn(C)c3=O)=O)C2)cn2cccc(F)c2n1 Cc1ccc(NC(C2CN(C(c3cc4sccc4s3)=O)CCC2O)=O)c(C)c1 C(C)(C1=CCN(C)CC1)NC(CN(C(=O)Cc1cn(C)cn1)C(C)C)=O C1(NC(CNC(C2C(C)C2)=O)=O)CC=C(C(=O)N2CC(O)(C(N)=O)C2)C1 N1(C(C2C(C)=C2)=O)CCN(C2CCN(C(c3cnc(Cl)cc3Cl)=O)CC2)C(=O)C1 C1(O)(CNC(CN(CCC#C)C)=O)CCCN(C(c2cc(CSC)on2)=O)CC1 N1(C(C2N(C)C(=O)CC2)=O)CC(NC(c2nocc2C(C)(C)C)=O)CC1(C)C C=CC1(CO)CCN(C(=O)C(CCC)NC(c2cn(C)nc2CC)=O)CC1 c1(NC2(CNC(c3ccc(O)nc3Cl)=O)COC2)ccc([N+](=O)[O-])c(O)n1 N1(C(c2ccn(C)c2)=O)CCC2(CC2C(N2CCS(=O)(=O)CC2)=O)C1 CCCC(C(=O)NC1CC(CN)C1)OC.C12(CC=O)CCC(CC1)C2 C(C(=O)N(O)Cc1cn(C(C)C(=O)N2CCCC2)nn1)NC(CC)=O c1(C(N(C2CN(C(C(C)SC)=O)CC2(C)C)C)=O)c(C)ccc2n[nH]cc12 CS(C)(=O)=NC(=O)C(=O)N1CC2(C1)CN(C(c1cc[nH]c1C1CC1)=O)C2 N1(CCOCC)CCN(C(c2ccn(C)c2)C(=O)NCC2CCCO2)CC1 CN1CCN(C(c2cc(=O)n(C)cn2)=O)CC1CNC(=O)Cn1cccnc1=O C1(N(C(c2c(CC)cc[nH]2)=O)C)CN(C(C2C3CC4C(C3)C24)=O)CCC1C N1(C(Cc2c(C)ncc(Cl)c2)=O)CCN(C(c2c[nH]c(C#N)c2)=O)C(C)C1C N1(C(=O)COCC2CCCC2)CCC2CN(C(c3ccc4[nH]ccc4n3)=O)C2C1 C1(NC(CC2CC(CC)OCC2)=O)CC2(CCN(c3nc(C(=O)OC)ns3)C2)C1 CN1CC2(CCN(C(c3cccnc3CNC(C3CC(O)C(F)C3)=O)=O)C2)C1 N1(C(c2ccn(C(F)F)n2)=O)CCC(C(N2CCOCC2CO)=O)(CCF)C1 c1(C(N(C2(CC(=O)N(C3CC(O)C3)C)CC2)C)=O)ccc(C#N)[nH]1 c1(C(=O)NC2CCCC(CC(=O)NC(CCC)CO)C2)cc(C)ccc1NC N1(C(C(C)CC2CCC2)=O)CCN(C(c2cc(O)cnc2N)=O)C(C)C1 C1(NC(=O)CNCC2CC2)CC(F)(F)C1.C1(N2C(C3CCCS3)C2=O)CCCC1 c1(NC(C2N(C(c3cccc(N(C)C)c3)=O)CC(F)C2)=O)c(F)ccc(Br)c1F N1(C(c2c(C)oc(CO)c2)=O)CCOC2(CCN(C(=O)C#CC3CCOC3)C2)C1 C1(C(N2CCC(COC)CC2)=O)C2CCC1CN(C(C1(F)CCCC=C1F)=O)C2 N1(C(c2cnc(CC)nc2C)=O)CCC2CC1CN(C(=O)C(C)(C)C)C2 C1(NC(c2n(CC)ccc2)=O)C2CCN(C(C3SCCCS3)=O)CCC12 C1(NC(C)=O)CN(C(c2cc(F)cc(Cl)c2C)=O)CC(F)(F)C1 C1(C(N2CC(CC(C(=O)NCc3cc(C(C)C)n[nH]3)F)C2)=O)COCCN1C C(=O)(C(C)(C)CN(C)C(C1CCC(O)CC1)=O)NC(c1nc(C)[nH]n1)CO CC(CF)CC(=O)NCC1(C(F)F)CCNC1=O C(=O)(C1c2c[nH]nc2CN1C(=O)CC1CCC(O)C1)N(CC(C1CC1)OC)C c1(CNC(C(C)C2CCCO2)=O)nc2c(s1)CN(C(c1cnc(N)cn1)=O)CC2 c1(NC(CNC(C2CCCC(OC)C2)=O)CO)nc2c(cc1[N+](=O)[O-])CCCC2 n1(CC)cc(C(=O)NCC(CC)(CC)NC(=O)C#CC(OC)OC)c(=O)cc1C c1(-n2c(C(c3c(OCC)nsc3)NCC=C(C)C)nnn2)ccc2c(c1)OCO2 C(C)(CCCC(=O)N1CCN(C)CC1)NC(C1(SC)CC(=O)C1)=O N1(C(CCC(C)(F)F)=O)CC2(CNC(=O)C(CO)C(C)(C)C)CC1CCO2 C(=O)(C(F)C(C)(C)O)N1C(C2(O)CN(C(Cn3c(C(C)C)nnn3)=O)C2)CCC1 Cn1ncc(S(C)(=O)=NC(=O)C2CC3CC2(c2cccnc2)C3)c1CN Cc1cnccc1C=CC(N1CCCC1CN(C)C(c1nccc(Cl)c1O)=O)=O c1(OC)c(Cl)cc(C(=O)NC2CCN(C(C3COC(=O)O3)=O)C2)nc1Cl Cc1ncc(C(N2CCC=CC2C(N2CCC(C)(N(C)C)C2)=O)=O)cc1C#N C1(CNC(=O)C(C)(C)C)(NC(C(C)NC(c2nncs2)=O)=O)CCCCC1C N1(C(C2(OC)CC2)=O)CCN(C(=O)CCCc2ccc(Cl)c(Cl)c2)C(C2CC2)C1 c1(OC)ccc(C(=O)NC2CC(C(=O)Nc3ccnc(C)n3)C2)c(F)c1F C(=O)(CC(F)(F)CC(=O)N1CC2CC(C1)CN(C(=O)CNC(C)=O)C2)OC C1(CNC(=O)C(c2ccccc2)O)CC2(CO1)CN(C(=O)Cc1cc[nH]c1)C2 C(c1ccccc1)=C(C)C(N1CC2CC1C2C(=O)NCc1nnc(C)n1C)=O c1(C(N2CC3C(C(=O)Nc4cc(OC)c(Br)cc4)(C3)C2)=O)cc(F)cc(C)c1O C(CC(F)(F)CC)NC(C1(NC(C(C=C)O)=O)CCSC1)=O Cc1c(C(=O)NCC2C(C)CCN2C(c2c[nH]c(C#N)c2)=O)ccc2cncn12 C(=O)(CC(C)(C)CC(F)F)N1CCC(C2(NC(CCS(C)=O)=O)CC2)C1 CC1(C)CCC(CNC(c2cncnc2C2CC2)=O)N(c2ccnc(C3CC3)n2)C1 c1(OC(C)=O)ccccc1C(c1nnnn1C1(C)CC1)Nc1ccccc1OC c1(C(=O)NCC2C(NC(CCCC(N)=O)=O)CCC2)coc2c1C(O)CCC2 CCC(C)CCCCC(=O)NCC1CC1C(=O)NCCc1ccnc(O)c1 O=C1Nc2cc(C(N3CCOCC(CNC(C4C=CCC4)=O)C3)=O)ccc2C1=O N1(C(C2(CC)CCC(O)CC2)=O)CCC2(CCC2CNC(=O)C(C)(C)CF)CC1 C(=O)(C(F)C(C)(C)O)N(CC(N1CCCC(OCC)C1)=O)C1CC1 Cc1csc(C(N2CC(CNC(=O)C=C3CCCCC3)C3CC23)=O)c1C C1(C(C)C)CCCCN1C(=O)C=CCN(C)C(c1ncn(C)n1)=O N1(C(c2c(C)cnn2C)=O)CC2CCC2(CC(=O)NCCC(=O)NC(N)=O)C1 N1(C(CCC=C=C)=O)CCC(NC(=O)COc2cncc(Cl)n2)C(CO)CC1 C(=O)(C1=CCc2ccccc21)NC1CC2CN(C(C(=O)NC(C)C)=O)CC(C1)C2 c1(C(=O)NC(C)CC(C)N(C(C2(N(C)C)CCC2)=O)CC#N)cccc(=O)n1C c1(CNC(=O)Cc2ccccc2)cn(CC(C2CC2)NC(c2cnc(O)s2)=O)nn1 N1(C(C(C(C)O)C)=O)CCN(C(c2nccc3cc[nH]c23)=O)C2(CCC2)C1 N1(C(C2CC(CCC)OCC2)=O)CCCN(c2ccccc2)CC1 C1(NC(CC2C(C)C2)=O)CC2CC(C1)N(C(c1cc(O)c(F)cc1N)=O)C2 Cc1cc(C(=O)NCc2ccc(CNC(C3(C)CCCO3)=O)cc2)cc(N)c1O C1(C(=O)NC(CC=C)CO)CC2CC(C1)N(C(C)=O)C2 Cc1ncc(C=CC(=O)NC2CN(C(=O)Cn3cnnc3O)CC2C)c(O)n1 c1(C(CNC(c2c(CCC)n[nH]c2)=O)NC(=O)C(C)SC(C)C)cccc(C)c1 c1(CNC(C(C)CN(C(=O)CCN2CCCC2=O)C)=O)ccccc1C#N C(=O)(CC(C1CC1)C1CC1)NCCC(C)N(C(=O)CC1CCCN1C)C c1(OCCOC)ccc(SC)cc1.c12cnc(nc1)CCNC(=O)C(=O)N2 CC1CN(CC(=O)N(C)CC2(CNC(C3(C#N)CC3)=O)CC2)C1 N1(C(c2ccc(CC)cc2F)=O)CCCC(C)(C)C1CNC(=O)CN1CCC1 N1(C(C=C(CCC)CCC)=O)CCOC2(CCN(c3ccc(C#N)nc3)C2)C1 C1(C(N2C(CNC(CCOC)=O)CC(F)(F)C2)=O)CC2CC1C1C2C1(F)F N1(C(CSc2ccc(C)cc2)=O)CCN(C(C2CC3CCC3C2)=O)C(C2CC2)C1 c1(C(=O)NC2(CNC(C3CCN(C4CC4)CC3)=O)CC2)cc2n(c1)CCC2 C1(C(N(C2CCN(C(c3nc(CCC)sc3)=O)C2)CC)=O)CCC(=O)NC1 c1(C(=O)OC)ccc(CN2CCC2C(=O)Nc2c(Cl)cccc2Br)c([N+](=O)[O-])c1 N1(C(C(C(C(C)C)O)(F)F)=O)CC2CS(=O)(=O)CC2(NC(c2ccn(C)n2)=O)C1 Cc1ccc(-n2nc(C)cc2-n2cc(-c3ccnc(CNC(C)C)c3)nn2)nn1 C=CCC(CC=C)C(=O)NC(CC=C)C(=O)NCCC1CC=CC1 c1(C(N(CC(C)(C)NC(C2CC(C)(C)CCO2)=O)C)=O)n[nH]c2ccccc12 c1(CNC(=O)CC23CC(C2)C3)cccc(NC(=O)C(O)C2CCCC2)c1 c1(NCC(CC)(CC)CO)[nH]c(=NCC(C)(C)NC(C)C)nc2sccc12 C1(CNC(C(C)CN(C(=O)CC2(O)CCCC2)C)=O)CC12CCOCC2 C#Cc1ccc(C(=O)NC(CC#CC)C(=O)N2CCCCC2CO)cc1C S(=O)(=O)(CCCC)NCCC(=O)NCCN(C(C1CC(COC)CO1)=O)CC C(=O)(CCC(C)(C)C(=O)OC)NC1CC(C)(CNC(CC(CCC)C)=O)C1 N1(C(COC(C)=O)=O)CCC(O)CC1C(=O)NCC1CCCCN1C C1(NC(C=CC(C)C)=O)CCCC(CC(=O)NCC2(F)CCOCC2)C1 C=C1CC(C(C2CC2)OC2CCC2)C1.O(NC(=O)C1(N(C(=O)CO)C)CC1)C S(=O)(=O)(c1ccc(C(=O)NCC2CC2NC(=O)C2=CCCS2)cc1)NC(C)(C)C C1(C)(C(=O)NCC(C(C)C)NC(c2ccccn2)=O)CC(C2CC2)=NO1 c1(-c2scc(C(=O)NC(c3ncc(F)cc3F)C)n2)c(Cl)cccc1Cl CC(F)(F)CC(=O)NC1CCC(NC(=O)CC2CCC23CCC3)C1 Cc1cc(C2CC2)ccc1C(=O)N(C)CC1CCCN1C(c1ncoc1C)=O Cc1c[nH]ccc1=NC(=O)C1CCC(NC(C2CCC(CO)CC2)=O)C1 C(CNC(=O)Cn1nnc(C2CC2)n1)(CC(F)(F)F)NC(Cc1c(C)n[nH]c1C)=O c1(C(=O)NC2C(C)CCN(C(c3cccn3C)=O)C2C)cccc2c1nnn2C c1(CC(=O)N(C2CC(N(C(C(C)C3CC3)=O)C)C2)C)ccc(C(=O)C(C)=O)cc1.O C1(C)(C(N2CC(O)(CCNC(C3(OC)CCCOC3)=O)C2)=O)CCC(C)C1(C)C C(=O)(C1CCCn2nccc21)N1C2CN(C(c3cccnc3)=O)C(C2)C1 c1(CN2CCC(C#N)(NC(=O)Cc3ccc(Cl)cn3)C2)cc2ccoc2cn1 CC1(C)C(CNC(C2CC(=O)CN2C(=O)CCc2nc(=N)[nH][nH]2)=O)C1(C)C c1(-c2nc(NC(c3ccc4c(c3)OCO4)=O)sc2)cccc2ccnn12 c1(C(=O)NC(CNC(c2ccc(C#C)cn2)=O)CCOC)cnc2ncccn12 C1(CNC(c2c(CC)nco2)=O)CN(c2ccnc(Cl)n2)CCN1C C1(N(C)C(C2CCC=CO2)=O)CCCN(C(=O)CC2CCC3CC23)CC1 Cc1sc(C(=O)NC(c2ccc(N3CCN(C)CC3)cc2)C)cc1[N+](=O)[O-] CCC(CC)(CO)C(=O)NCCCCCN(C)C(C1CCCN(C(=O)NC)C1)=O N1(Cc2c(C)nc(CCC)o2)CCC(NC(=O)Cc2nonc2C)CC(C)(C)C1 c1(C(=O)NCC(C)(C2CCC2)NC(C2Cc3nccn3C2)=O)cc2n(n1)CCC2 c1(C(=O)NC2CC3CN(C(c4cn(CC=C)nn4)=O)CC32)cnn2ccn(C)c12 CC(C(=O)N1CCN(C(C2CCCCN2C)=O)CC1)S(C)(=O)=O N1(C(C2CN(C)C(=O)CC2)=O)CCC2C(CCCN2C(c2cnccn2)=O)C1 c1(C(=O)NC(C(=O)N2C(CC)CC2)CO)ncncc1OC C1(CN2CCCN(C(C)=O)CC2)Cc2ccc(C(=O)O)cc2O1 O=C1C2Cc3ccc(F)cc3N2C(=O)N1CC1(Br)CCOCC1 N1(C(CC2C(CC)C2)=O)CCOC2(CCC(NC(=O)C(C)(C)OC(C)C)CC2)C1 CC(=O)CCCC(C)C(=O)NC1CCCC(NC(C2CC(C)CCO2)=O)C1 C(C)(CCC(=O)N1CCC(OCC(=O)NCCc2cccnc2Cl)C1)OC c1(C(N2C(CC)CC(C)(C)C2)C(=O)NCCCSC)cc(S(N)(=O)=O)cs1 C1(C(=O)NCCCNC(CC(c2cccs2)NC(C)=O)=O)(C(F)F)CCOCC1 C1(C(N(CCS(=O)(=O)NCC)CC)=O)C2CCC1(c1ccnn1C)C2 C12(SCC(=O)NC(C3CCCCS3)=O)CCC(C1)N(C(c1ccc(N)cc1)=O)C2 C1(NC(CCC2N(C(C(CC=C)OC)=O)CCCC2)=O)CCn2cnnc2C1 c1(C(N(C(C)C(=O)NC(CO)CCCO)CCC)=O)ccc(=O)n(C)c1 C1(N(C2(C(=O)NOCCCF)CCCC2)C(c2ccncc2)=O)CCCCCC1 C(=O)(CCCCNC(=O)CCC1CC(F)(F)C1)N(C)Cc1cncn1C Cc1ccc(C(=O)N(C2CC2)CC2CCCN2C(c2cnsn2)=O)cc1Br c1(C(N(CC(C)N(C(CCN(C(CCC)C)C)=O)C)C)=O)cc2ccncc2s1 CC(F)(F)C(=O)NC1CCCC1CNC(=O)C(c1cccnc1)N1CCCC1 Cc1ccc(C(=O)NCC(C)(F)CNC(=O)C(C)C#N)cc1F C12(NC(=O)Cc3cnns3)CCCCC1N(C(=O)CS(=O)(=O)C1CC1)CC2 c1(C(=O)NC2CC(NC(=O)CC(c3ccc(F)cc3)O)C2)ccnc2ncnn12 N1(C(CCN(CC)CC)=O)CCc2nnn(C3CCN(C)CC3)c2C1 C(=O)(C(O)CCC(C)C)NC1(C(N2CC(CCCCC)C2)=O)CCSC1 CC(C)C(CNC(C1(C)CC1(C)C)=O)C(=O)N(C(C)CCO)C C1(CNC(CS(CC)=O)=O)CC12CCN(c1snc(Cl)c1C#N)CC2 c1(OC)ccc(Cl)cc1C(N1CC2CC1CC2NC(=O)Cc1cnnn1C)=O C=CCC(CNC(C1CCCN1CC(C)C)=O)NC(c1cc(CC(C)C)[nH]n1)=O c1(CC(=O)NCCN(C)C(c2ccc3nonc3c2)=O)cncc2ccccc12 C1(SC)CN(C(C2CC(n3cccn3)C2)=O)CC1NC(=O)CNC(C1CCC1)=O C(=O)(CCCCCSC)NC(C1N(C(C2C(=C)CC2)=O)CCC1)(C)C C1(NC(CC(n2ccc(C)n2)C)=O)CN(C(c2cc(C#N)cs2)=O)CC(C)(C)C1 C1(NC(CCCOCC=C)=O)CCC(C)N(C(=O)Cn2ccsc2=N)C1 C1(O)(C(C)NC(c2occc2CO)=O)CCN(C(=O)CCSc2ccccn2)C1 C1(CNC(C(C=C)O)=O)CC12CCN(C(=O)CCCCC#N)CC2 C1(NCCCNC(=O)NC(CCSC)C)CC2CC1C1CC21 Cc1ncnc(O)c1C(N1CCC(CCCNC(C2(CO)CCCO2)=O)CC1)=O Nc1ccc(C(=O)NC2CCCC2NC(=O)CC(F)(F)Br)nc1 n1(CC)cc(Br)c(C(=O)NCC2(NC(=O)CCOc3cccnc3)CC2)n1 C1(C)(C(=O)NCCCN(C(CNC(CC)=O)=O)C2CC2)CCSCC1 c1(CC)cccc(OCC(N2CC(O)(CN(C(=O)CCC(C)OCC)C)C2)=O)c1 Cc1cc(C(=O)NCC(CC(F)(F)F)NC(=O)CC2CCCCN2C)cc(C)n1 N1(C(C(C)(C)CF)=O)CCC(C2(O)CC(NC(C3C=CCCC3)=O)C2)CC1 N1(C(C(CCCC)O)=O)CCN(C(c2cc(C(F)F)ncn2)=O)CC(C)(F)C1 c1(CC2C(C(=O)NC(c3n(C)ccn3)C(F)F)C2)cccc(I)c1 c1(C(=O)N(C(C)(C)C)CC#N)ccc(-c2cncnc2C(N2CCOCC2)=O)cc1F CC(C)CC(CNC(=O)CCc1ccc[nH]1)NC(=O)CC1CCN(C)C1 Cc1cc(Cl)n[nH]c1=NCC12CC(C1)C(C#N)N2 C1(NC(C2CCCN(CC(F)F)C2)=O)CCN(C(C2CC3(CCC3)C2)=O)CC1F c1(COC)ncc2n1CCCC2.n1(CCC=C)c(NC)nnc1CC1CC1 N1(CC)C(=O)CCC1CC(=O)NC1CCN(C(c2sc(C(C)C)nc2C)=O)C1C C1(NC(c2c(C)cnn2C)=O)CC2CCC1N2C(=O)C(c1ccc(F)cc1)F N1(C(C2C(CC)CCO2)=O)CC2(NC(=O)COCc3ccnn3C)CCC1CC2 C1(CNC(c2c(C)oc(-c3cnn(C)c3)n2)=O)C(C2CC2)CCN1C(=O)C(F)F Cc1c(CNC(c2nccc(Cl)c2F)=O)oc2ccccc12 C(=O)(C(C)(C)CCC(C(=O)NCCC#N)N1CCOCCC1C(C)C)OCC c1(COC(CN(CCOC)C(=O)N(CC(O)CO)C)=O)ccc(OC(F)F)cc1 c1(CC)ccc(F)cc1NC(=O)CCCCNC(=O)C=Cc1ccn(C)c1 C1(NC(CC2(CS(C)(=O)=O)CC2)=O)CCCN(C(=O)C2=C(Cl)CC2)CC1 c1(C(=O)NCC(C(C)(C)C)NC(CNS(CC)(=O)=O)=O)cc(N)c(F)cc1F c1(CNC(c2n(CC(=C)C)nnn2)C2(CF)CC2)ccc(-n2cncn2)c(F)c1 N1(Cc2ccc(N(C)C)cc2O)CC2CN(C(c3ccc(F)c(Cl)c3)=O)CC2C1 c1(C(=O)NCC(CNC(C2CCC(C(=O)OC)C2)=O)F)c(C)nc(C)nc1C C1(CC(=O)NC(CC#C)(C)C)N(C(c2c[nH]nc2OC)=O)CCC1(C)C c1(C(=O)NCC2CCN(C(Cc3cccc(OC)c3)=O)C2)nc(Br)cnc1N N1(C(C2(CSC)CC2)=O)CCC(C(C)C(=O)NC2CC(C)C2)CC1 c1(C(=O)NC(CC(C)NC(c2cn(CCF)nn2)=O)C)cccc2nnn(C)c12 CCCCCCC(F)C(=O)NC(CN(C(=O)CS(=O)(=O)N1CCCCC1)C)CC Cc1c[nH]cc(C(N2CCC(NC(C3CN(C4COC4)C3)=O)CC2)=O)c1=O C1(CC(N2C(C)CC2)=O)COCCN1C(C1CCCC(=O)C1)=O c1(N2CCN(C(C(C)Sc3ccccc3O)=O)CC2)ncnc2cc[nH]c12 c1(CC)ncc(C(=O)NC(C2CN(C(=O)CCc3cc[nH]n3)CCO2)C)c(O)n1 c1(C(C)C(F)(F)F)cccc(CNC2CCCC(CN)C2)c1 C1(NC(C2C(C)(C(C)C)C2)=O)C=CCN(C(=O)Cc2nccs2)C1 c1(C(N(CC(O)CNC(=O)CN(C2CCCC2)C)C)=O)cc(=O)n(C)cn1 N1(C(c2cc(Br)n[nH]2)=O)C2CCC1CC(O)(Cc1ccccc1)C2 c1(CC(C)C)cc(C(=O)NC2CCC(NC(C3(C(N)=O)CC3)=O)CC2)cc(O)n1 O=C(CCCCC(F)(F)F)NCC1(F)CCN(C(c2ccc[n+]([O-])c2)=O)C1 C12(NC(CC=C)=O)CCN(C(c3cccs3)=O)CCC1C2 N1(C(C(CCC)n2cc(COCC)nn2)=O)CCOC(C(=O)OC(C)(C)C)CC1 c1(NC(C(N2CCC(F)(C(=O)OC)C2)=O)=O)ccc(F)cc1C(F)(F)F C1(CNC(=O)Cn2cccn2)CCN(C(=O)CCNC(C2CCC2)=O)CC1(F)F c1(NC(N2CC(C(C(=O)OCC)F)C2)=O)ccccc1OCC c1(N2CC(C)(CNC(Cc3n(C)cnc3)=O)OCC2)ncc([N+](=O)[O-])cc1CO N1(C(C(CC)Sc2nc(=N)[nH][nH]2)=O)CCN(C)c2ccc(C)cc21 N1(CCc2c(C)cccn2)C(=O)CN(Cc2cccc(OCC(F)(F)F)n2)C1=O C(CCN(C)C(c1ccc(C(F)F)o1)=O)(C(C)C)NC(c1cn(CC=C)nc1)=O N1(C(C(C(=O)OCC)F)=O)CCC(C)(C)C1CNC(=O)CC(=O)N(C)C C1(NC(C2CC(C3CCC3)C2)=O)CCCCN(C(c2ccco2)=O)C1 Cc1cc(C(N2CCC(C(C)NC(c3cc(C#N)[nH]c3C)=O)C2)=O)cc(C)c1F C1(NC(CC2N(C)CCC2)=O)CCC12CCN(C(c1cscn1)=O)CC2 CC1(C)NC(=O)CC1C(N1CCCCC1CNC(c1nc(Cl)c(Cl)s1)=O)=O c1(C(C)C)ccoc1C(=O)NCC(O)C(=O)N(C)CC1CC1(F)F c1(C(=O)NCC2(O)CCN(C(CCCCOC)=O)C2)cc(Cl)c2ccccc2n1 C12(CNC(CC3OCC(C)(C)OC3)=O)CCCC1N(C(c1csc(Cl)c1)=O)CC2 CC(C)COC(=O)CNC(N)=O.C1C(=O)N1C(C)C1CC1.C1(CC)CCC1 C(=O)(CC(C)(C)CCOC)N1CC(N(C(c2c(CC)[nH]cc2)=O)C)C1 C(=O)(CC=O)N(C(C)C(=O)N(C)C)C.C(C(C)(C)CC1CC1)C1CCCCC1 N1(C(C(n2ccc(C)n2)C)=O)CC(O)CC1C(=O)NCC(C)(C)CC1CC1 C(C)(C(C(=O)NCCC1CCOC1)NC(c1cc(C)sc1N)=O)OC c1(C(N2CC(C(C)NC(c3ccc(Cl)s3)=O)C2)=O)cn2c(n1)CCCC2 c1(CC)cc(F)cc(NCC#Cc2cnn(-c3ccccc3)c2)c1C N1(C(C2CN(C(N)=O)C2)=O)CCCCC1C1CCN(C(=O)CCc2cn[nH]c2)C1 C1(C(N2C(C)(CCC)CC2)=O)CN(C(C2CC(=O)C2(C)C)=O)CCN1C C(=O)(CCCCCC#N)NCC1CCN(C(C(CC)C(C)C)=O)CC1 Cn1cnc(C=CC(=O)NCCCCC2CN(C(c3cc(C(F)F)cs3)=O)C2)c1 C1(CN(C(=O)C(Cl)=CCl)C)CC(F)CN1C(=O)CSCc1cccs1 CN1CC2CCC(NC(=O)NC(Cc3ccccc3)CCC3CC3)C2C1 c1(NC(=O)NCC2N(C)CCCC2)c(C#N)cnn1C1CCCC(C(F)(F)F)C1 N1(C(C2CCC(C)O2)=O)CC2CCC(C1)C2CC(=O)N1CCC1 C1(NC(c2csc(O)n2)=O)CC2(C1)CN(C(c1cnc(-n3cccn3)cn1)=O)C2 c1(-n2ccc(C(N(CCNC(=O)C(C)(C)SC)CC)=O)n2)ccc(F)c(Cl)c1 C1(NC(C=CC)=O)C(C)(C)CN(C(C2CN(C(=O)C(C)(C)C)CCO2)=O)CC1(C)C c1(C(=O)NC(CNC(C2CN(CC)C(=O)N2)=O)C(C)C)cccc2c1CNC2=O N1(CCNC(c2cc(CC)on2)=O)CCCN(C(C2NC(=O)OC2(C)C)=O)CC1 c1(OC)cc(SC)ccc1CNC(N1CC(CO)OCC1C)=O N1(C(c2c(CC)scn2)=O)CCOC2(CCN(C(c3cc(Cl)cnc3C)=O)C2)C1 C1(C(N(CC#CC)C)=O)(NC(=O)C(=Cc2ccco2)C)CCSC1 Cc1cncc(C)c1C(N1CCC(C(=O)NC2CN(C)CC2O)C(C)C1)=O c1(OC)cc(F)c(C(N2CC(NC(c3c[nH]c(=O)cn3)=O)CC2C)=O)cc1N S(=O)(=O)(c1ccc(=NCc2ccno2)[nH]c1)NCc1cccc(OCC)c1 c1(C(N2CCC(NC(=O)C(Cl)=CCl)CC(O)C2)=O)cncc2cnccc12 C1(C)(CNC(CS(=O)(=O)N(C)C)=O)CN(C(=O)COCC(F)(F)F)CCO1 C(=O)(C1=NN(C(C)C)C(=O)CC1)NC(C1CN(C(C(CC)CO)=O)C1)C C12(C(=O)N(C3(C4CN(C(C5CC6CCCC56)=O)C4)CC3)C3CC3)CCCCC1C2(F)F N1(Cc2n(C)ccn2)CC(Cc2ccc(Cl)cc2OCCO)C2(CC2)C1 C1(C(=O)NCCC2(NC(C3NC(=O)OC3)=O)CC2)CCC(C2CC2)C1 CC1CN(C(c2ccc(SC(F)F)cc2)=O)CC1NC(c1coc(O)n1)=O C1(OC)CN(C(=O)CC(=O)N(C)C)CC1NC(=O)C(O)CC1CCCCC1 C(=O)(CC(O)CNC(=O)CCC1CCC1)N(C1CCCC1C#N)C CCC(C(=O)NC1CCC(NC(C2(OC)CCCCC2)=O)C1)C(C)C c1(C(N2CC(O)(CCNC(C(C)OCC=C)=O)C2)=O)cc(O)c2ccccc2c1 C(=O)(CC(C)(C)C(F)F)N1CCC(C(N(CC)CC2CC2)=O)OCC1 Cn1c(=O)oc2cc(C(N3CC4COC(=O)C4C3)C(=O)NCC3CC3)ccc12 N1(C(C2(N(C(c3nc(C)c(C)s3)=O)C)CC2)=O)CCCC2(CCC2)C1 N1(C(C(c2ccncc2)OC)=O)CCCC2(CCN(C(C3(F)CCCC3)=O)C2)C1 N1(C(C2(NC(C3CN(C)C3)=O)CC(O)C2)=O)CC(CO)C2(CCC2)C1 Cc1cccc(C)c1OCC(O)CNC(c1ccnc(NC(=O)C2CC2)c1)=O C1(CNC(=O)C(N2CCC(CO)C(O)C2)c2ccnc(Cl)c2)CCC(F)(F)CC1 CCCCC(C(=O)NC)NC(=O)C(O)C1CN(C(=O)C(C)OC(C)=O)C1 N1(C(C(N)=O)=O)CCN(C(C2CC3CCC3C2)=O)CC1c1cn[nH]c1 C(CCC(C)(C)O)NC(C(CNC(CC(C)C1CC1)=O)O)=O N1(C(c2c(Cl)cc(C)s2)=O)CC(NC(=O)C(Cl)=CCl)C(C)(C)C1 CC1CC(CCNC(C)=O)CCN1C(=O)OC(C)(C)C.c1(O)nc(C(C)(F)F)cs1 N1(C(C)C)CCC(N(C(=O)C(C2CCN(C(=O)Cn3cnnc3)C2)C)C)C1 c1(-c2cn(C(C)C)c(=O)cc2)ccc2cc(C(=O)NCCC(O)CO)cn2c1 N1(CC)CCOC(C(=O)NCC(C)(C2CC2)NC(c2ccc(C(F)(F)F)[nH]2)=O)C1 CC1CN2CCN1CC2C(=O)NCCCCCN(C(=O)Cc1ccsc1Cl)C CC1(C)COC(C(=O)NC2(C)CN(C(C3COCCO3)=O)C2)C1 N1(C(C2ON=C(CC)C2)=O)CCCC2(NC(=O)CCC[N+](=O)[O-])CCCC12 c1(C(N(C2CC2CNC(c2cccc(OCC(F)F)c2)=O)C)=O)ccc(N)c(N)n1 C1(NC(C(n2c(C)ncc2)C)=O)CCN(C(c2cn(C3CC3)cn2)=O)C12CC2 c1(NC(C2CC2C(=O)Nc2ccc(I)nc2)=O)cc(Cl)c(Br)cn1 CC(C(=O)N1CC(OCCOC(=O)C=CBr)C1)c1cncs1 c1(-n2c(C(C)Oc3cccc(OCC)c3)nc(COCC)n2)ccc(F)c(F)c1 C1(Cn2cc(C3CCN(C(c4c(C#N)csc4)=O)C3)nn2)CCC(F)(F)CC1 c1(C(N2CC=CC(NC(C3CCCCS3)=O)C2)=O)ccc(F)c(O)c1 c1(C(=O)NCC(C(C)(C)C)NC(CCC#C)=O)cc2n(n1)CC1(CC1)C2 C(=O)(CC1=CCN(C(=O)C(C)S(C)(=O)=O)CC1)N1CCCC(C)(OC)C1 c1(C(=O)NCC(C(=O)NCC2(C)CC3CC3C2)N(C)C)cc[n+]([O-])cc1 Fc1ccc(C(C2CC3CC3C2)Nc2nnnn2CC2CC2)nc1 N1(C(CCCOCC)=O)CCN(C(=O)COc2ccc(OC)cc2)C2CC12 CC(C(C)C(=O)NC1CC2(CCN(C(c3cocn3)=O)CC2)C1)S(C)(=O)=O CCC(CNC(c1c(CNC(c2cc(C3CC3)no2)=O)nnn1C)=O)CCO C(CCCCC(=O)N1CC(C)OC(C)C1)N(C(CC(C)OC)=O)C c1(N(C2CCN(C(c3ccc(SC)s3)=O)CC2)C)ncncc1C#N n1(CC2CCN(CCCN3C(=O)CCCCC3)CC2)cnc2cc(Cl)ccc12 c1(C(=O)NC2(CC)CN(C(C34CCC(OC)C3C4)=O)C2)ccc(F)cc1 CCC(C)C(C(C(=O)Nc1cccc([N+](=O)[O-])c1)N(C)CCOC1CC1)OC CC1=CCC(C(=O)NCC(O)CN(C(=O)C(C)(C)c2ccsc2)C)CC1 Cc1nnccc1C(=O)NC(C1CCCC1)CNC(C1(C2(C)CC2)CC1)=O N1(C(c2cc(C)c(Cl)cc2)=O)CCC(C)N(C(c2nocc2Br)=O)CC1 C(=O)(C1=C(Cl)CCCC1)NCCC1CN(C(C(C)NC(c2ccccc2)=O)=O)C1 c1(OCC)cc(C(c2nnnn2CCC2(C)CC2)NCCCS(C)=O)sn1 C1(NC(COCCC#C)=O)COCC1C(=O)NC1(C(=O)OC)CC1C c1(N2C(CNC(C(c3cccc(OC)c3)C)=O)CCC2)ccc([N+](=O)[O-])c(C)c1 CCC(C)(CC)C(=O)NCC(C)(CO)NC(=O)Cc1cc(Br)ccc1Cl c1(NC(CCN2C(C)CCCC2C)=O)cnc2cc(Br)ccn12 C1(OC)(CNC(=O)CN2CCNC(=O)C2)CCN(C(=O)CCCn2ccnc2)C1 c1(CCCC(=O)NCC2(C)CCN(C(C=C(C)C(F)F)=O)C2)ccc(O)c(F)c1 c1(SC)ncc(C(=O)NCCC2CCC(NC(=O)CCC3CC3)C2)s1 C1(N(C(=O)CCCn2cncn2)CC)CCN(C(=O)C(F)C2CCC2)CC1 Cc1ccc(C=CC(=O)NC2CC(N(C)C(C3CCCN3c3nccs3)=O)C2)s1 c1(-c2cc(C(=O)NCc3nc(NC)sc3)no2)c(Cl)cccc1Cl C(=O)(CCC(CF)CF)NC(CC(=C)Cl)C(=O)N1CC(F)CC1C O=C(CC(F)(F)C(F)F)NC(CNC(c1ccnn1C1CC1)=O)CO N1(C(C2C(OCC)CCC2)=O)CCCCC(NC(c2nccc(N)c2Cl)=O)C1 C1(C(=O)NCC(C)(C2CCC2)NC(CC=CCC)=O)Cc2nn(C)cc2C(=O)N1 C(=O)(C(C)CCC(C)(C)C)NC1CC2(CC(C(=O)NCCNC(C(C)C)=O)C2)C1 N1(C(c2cccc(C)c2N)=O)CC2CCCC2(C(=O)NOC(C)C)C1 C1(C(NOCCC#C)=O)C(C)OCCN1C(=O)C(C)OC(C)=O Cc1ccc(C(=O)NC2(c3cc(N)ccc3O)CC2)c(N2CCNC2=O)c1 N1(C(C(=O)NCCCC=C)=O)C2CCC1CC(F)C2 C1(C(=O)NCC(CO)NC(c2cc(C(F)(F)F)n[nH]2)=O)CCn2ncnc2C1 C1(C(N2CCCC(C(=O)NCCC)C2)=O)COCCN(C(C2CNC(=O)O2)=O)C1 C#Cc1cnc(N2CCC(CNC(c3cnc(F)c(F)c3)=O)C2(C)C)nc1 C1(C2CN(C(=O)CCCCc3cnc[nH]3)C2)(NC(C2C(C)CCC2)=O)CC1 N1(C(C(CC)COC)=O)CCCN(C(c2cc3sccc3[nH]2)=O)C(C)C1 c1(N2C(C)(CNC(C3(C)CCCS3(=O)=O)=O)CCC2)nccn2nnnc12 N1(C(C=CC=CC)=O)CCC(C2CC(NC(c3cc(SC)c(C)o3)=O)C2)C1 c1(CN(CCOC)CCOC(=O)CCC2CCOC(CF)C2)c(Cl)cncc1Cl N1(C(c2ncc(C)cc2C)=O)CC(C)(C)OC2(C1)CN(C(c1[nH]cnc1C)=O)C2 C(c1ccc(C)nc1)=CC(=O)N(CC(CC)NC(C1CCC=CCCC1)=O)CC Cc1ccc(F)c(C(N2CC(NC(=O)COC3CCOCC3)CC(O)C2)=O)n1 CCCCC(CNC(c1sccc1C#N)=O)NC(=O)CC1CC2CC2C1 CCC(CC(=O)NCC(C)(C)COC)N(C)C(c1ccnc(CO)c1)=O C1(C(N2CC(F)(CNC(CCSCC(C)C)=O)C2)=O)CCC(C(N)=O)CC1 Cc1ccn(C)c1C(=O)NC(CNC(=O)CCSc1c(C)n[nH]c1C)C(C)C Cc1cc(CC(N2CC(CNC(c3conc3C3CC3)=O)C2)=O)no1 N1(C(COC)=O)CC(CC(=O)N(CC(C2CC2)OC)C)CC1(C)C Cc1nnn(CCNC(=O)NC(c2ccccc2)c2ccccn2)n1 C1(NC(C2CCC(CC)CC2)=O)CC1C1CCCN(C(c2ccc(C#N)[nH]2)=O)C1 N1(C(CN(C(=O)OC)C)=O)CCC(F)(CNC(C2(N3CCCC3)CCC2)=O)C1 C12(NC(CC=C)=O)CCCC1CN(C(c1ccc(C(N)=O)cc1)=O)C2 N1(C(Cc2nc(C)[nH]n2)=O)CCC2CN(C(=O)Cc3cc(C)sc3C)C2C1 CCCCS(=O)(=O)CC(=O)NC1(CNC(=O)C(C)C2(O)CCC2)CCC1 C12(NC(COCCC#C)=O)CCC(C(=O)NCC3CCCC3CF)(CC1)C2 C(CCN=c1[nH]c(=NCc2cccnc2N(C)C)[nH]c2ccsc12)N(C(C)=O)C N1(C(C(c2cnccn2)C)=O)CC(NC(=O)CN(C)Cc2ccco2)CCC1C c1(CC(C)C)ncc(C(=O)NCC2CCN2C(c2cn(CC(N)=O)nn2)=O)s1 c1(C(N(CCC2N(C(C=CC(CC)C)=O)CCCC2)C)=O)cc(Cl)ccc1C c1(C(=O)NCC2C(C)CN(C(=O)Cc3cc[nH]n3)C2)ncc(N)cc1Cl N1(C(C(CC)OCC)=O)CCN(C(=O)CN2CC(=O)NC2=O)CC1CCO c1(C(=O)NC2CCCC(N(C(CCOCC#C)=O)C)C2)ccc([N+](=O)[O-])cn1 C1(OC)CN(C)C(C)(C(=O)N(C2CCN(C(c3ncc(Cl)s3)=O)CC2)C)C1 C1(NC(C23CC(CNC(C(C)(F)F)=O)(C2)C3)=O)CCN(C2CC2)C1=O c1(N(CC)CC)ccc(C(=O)NC23CC(C(=O)NC4CCO4)(C2)C3)cc1 N1(C(Cc2c(C)noc2C)=O)CCC2(CCCN2C(=O)CC2CCC(C)(C)C2)C1 c1(C(N2CC3N(C(C(CC)=O)=O)C3C2)=O)cc(F)c(Cl)c([N+](=O)[O-])c1Cl Cc1cc2[nH]c(C(N3CCCN(C(=O)COc4cnn(C)c4)C(C)C3)=O)cc2o1 c1(CC(=O)OCC)cc(Cl)ccc1NC(c1csc(N(c2ccccc2)C)n1)=O C1(CNC(CSS(C)(=O)=O)=O)CC(NC(=O)CSCC(N)=O)C(O)C1 c1(-c2cn(CC)nc2)cc(C=O)ccc1C(=O)OC N1(C(c2ccc(O)nc2)=O)CCN(C(c2cncnc2)=O)C2CCCCC2C1 CC(C)C1=CCC(C(=O)NC2CCN(C(c3ccc([N+](=O)[O-])o3)=O)C23CC3)CC1 C1(NC(c2c(OCC)cccn2)=O)COC2(CCCN(C(=O)CC3(C)CC3)C2)C1 C1(NC(C=CC(=O)OCC)=O)CCC(NC(c2ccnc(O)c2)=O)CC1 c1(C(=O)NCC(CN(C(c2nc(C)n(C)c2C)=O)C)C)c[nH]c2c(F)cccc12 c1(NC(c2cnn(CC(C)C)c2C(F)F)=O)cccc([N+](=O)[O-])c1Cl N1(C(c2n(CC#C)ccc2)=O)CCCC2(C1)CN(C(=O)C(=O)C(C)CC)CCO2 N1(S(CC)(=O)=O)CCOCC1C(=O)NC1CN(C(=O)C=Cc2ccco2)CC1C N#CC1CC(F)(F)CN1C(C1CCCN(C(C2CCC(CO)CC2)=O)C1)=O c1(NC)ccccc1C(=O)Nc1ccccc1CN(C1COC1)C1CC1 C(c1c(C)nn(C)c1Cl)=CC(=O)NCC(C)(C)NC(CC1CC(CC)OCC1)=O CCC(CSCC)N=c1[nH]c(=NC)[nH]c(=NCC2(CS(C)(=O)=O)CC2)[nH]1 N1(C(C2CCC(NC(CN3CC(C)(C)C3)=O)CC2)=O)CCC(O)C12CCCC2 C(=O)(CC1=CCN(C(=O)COc2ccon2)CC1)NCC1N(C(C)=O)CCC1 c1(C(=O)NC(CC2CN(C(C(CC)C)=O)C2)C)cc(Br)c(Cl)s1 C1(C(=O)NCC(C2CCCC2)NC(C(C(C)C)(C)C)=O)CCCCN1S(N)(=O)=O N1(C(=O)Nc2ccc(OCC)cc2)CCC2(CC1)CN(Cc1cscc1OC)C2 C1(NC(C2CCCC23CCC3)=O)CC2CCC(C1)N2Cc1cc(C2CC2)no1 c1(C(=O)NCC2N(C(C3(OC)CCCCC3)=O)CCC2C)cn2c(n1)SCC2 c1(C(=O)NCCCCC(C)NC(=O)C=C2CCN(C)C2)ccn2ccsc12 C12(C(=O)NCC3CC(C)N(C(C4C(C)(C)C4(C)C)=O)C3)CCC(F)(CC1)CC2 N1(C(C2C(C)=CCS2)=O)CCCC(CCNC(=O)C=Cc2cnc(C)s2)C1 C=C=C(C)CC(=O)N(C)CCNC(c1cccc(Oc2ccccn2)c1)=O C1(CNC(CC2ON=C(C)C2)=O)COCCN(C(c2cc(O)nc(O)n2)=O)C1 c1(OC)cc(NC(c2n[nH]cc2NC(=O)Cc2ccc(Cl)c(F)c2)=O)cc(Br)n1 Cc1cc(=NCc2cccc3sccc23)[nH]c(N2CCC(N(C)C)C2)n1 Cc1nn(C)c(C)c1C(=O)NCC1(F)CCCN(C(C2C3CCC(=O)C23)=O)C1 c1(N2CCN(C(C)=O)CC2)nc(=N)nc(N(CCC#N)C)[nH]1 CC(C)=C=CC(=O)N1CC(O)CC1C(=O)NCC1CC2(CC2)CO1 CCC(CC)CC(=O)NC1(CNC(C2CC23CCCOC3)=O)CCCC1 Cc1cc(F)c([N+](=O)[O-])cc1C(N1CC(NC(=O)CCS(C)(=O)=O)C(O)C1)=O Cc1cc(C(=O)NC2CN(C(=O)C(C)C#N)CC2S(C)(=O)=O)c(S(N)(=O)=O)s1 N1(C(C2CCN(C(CC(CC(C)C)O)=O)C23CCC3)=O)CCc2cccnc2C1 Cn1cc(C(F)(F)F)c(NC(C2CC2NC(C2(c3cn[nH]c3)CC2)=O)=O)n1 N1(C(C(C=C)O)=O)CCCC2C1CCN2C(c1cc(Br)cn1CC)=O Cc1nc(C(=O)NC2CC(NC(C3CCOCC3)=O)C23CCC3)c(C)n1C c1(C(N2CC(NC(=O)Cc3ccc(Cl)cc3Cl)C3C2C3)=O)cncc2[nH]ccc12 N1(C(C(CCC=C)NC(C23CCCC2C3(F)F)=O)=O)CCOC2COCC12 C#Cc1cc(C(=O)NC2(C)CCN(C(c3ccnn3C(F)F)=O)C2)cc(F)c1 C1(NC(Cn2nc(C)c(Cl)c2)=O)C2CC1N(C(c1cc(C3CC3)nn1C)=O)C2C CC(C(=O)N1CCC(NCCC2CN(C)C2)C1)P(C)(C)=O.C(C)(C)(C)NC(=O)O CC1CCCCN1CCNC(N1CCC(Nc2ccc(C(F)(F)F)cc2)C1)=O CCCC(C)(O)C(=O)N(CCCCN(C(=O)C(n1ccc(Br)n1)C)C)C c1(CCC)ccc(C(=O)NC2CCC(NC(=O)CCc3ccc(Cl)cc3)C2)cc1 C1(NC(C2(C)CCN(C)C2=O)=O)CC2CCC(C1F)N2C(c1cc[n+]([O-])cc1)=O c1(CC(=O)NCC2(F)CC(NC(CCCN(C)C)=O)C2)c[nH]ccc1=O N1(C(C2(C)C(C)CCCC2)=O)CC=C(CC(=O)NC2CC(CCO)C2)CC1 N1(C(CC2OCCN(C(C(C3CC3)OCC)=O)C2)=O)CCC2(CCOC2)CC1 Cc1cccc(CC(=O)NC(CCN(C(=O)C(C)C(F)(F)F)C)C(C)(C)C)c1F c1(SCC(N2CC(CCC(F)(F)F)C2)=O)scnc1C1CCCC1 CC(C)C(CCC(=O)N1CCCC(C(C)(C)C)C1)NC(c1ccn(C)n1)=O N1(C(CC2N(C(C(C)C3(O)CCC3)=O)CCC2(C)C)=O)CC2CSCC(C2)C1 N1(C(C2(CCC)CC2)=O)C2CCCC1CN(C(=O)CC1CCC3CC13)C2 c1(C(=O)NCCOCCN(C(c2c(CC)nco2)=O)C)cc(N)ccc1Cl c1(OC)c(F)cc(N)c(OC)c1F.c1(C(N(CC2=CCSC2)C)C)ccccc1Cl c1(C(=O)NC(C)CCCNC(=O)C(F)=C2CCC2)ccc(C(F)F)cc1Cl c1(C(=O)NCCCN(C(C=CC(CC)C)=O)C)cn(CCN2CCCC2=O)cn1 N1(Cc2cccc(C(=O)Nc3ccc(C)cc3)c2)CC2(COC(C)C2)C1 S(=O)(=O)(c1cccnc1N(C)Cc1cn(C)cn1)N1CCCC(CC)CC1 N1(C(c2cn(CC)nn2)=O)CCC(C2(O)CN(C(=O)C3=C(C)CC3)C2)CC1 N1(C(C(C(=O)OC)C)=O)CCC2(CCCN(C(=O)Cc3ccnc(F)c3F)C2)C1 CC(O)(CNC(=O)CC1CCCO1)CNC(C1(C(N)=O)CC1)=O CCCCC(CNC(C1CC1C(N)=O)=O)NC(c1oc(CCC)nc1C)=O c1(C(=O)NCC(CNC(CCCOCC=C)=O)C(F)(F)F)cnc2n1CCOC2 C12CCCC(C1)S2.n1(CCC(=O)N(C)CC)cc(COC)nn1 c1(C(=O)NC(CNC(c2c(C)n(C(C)C)nc2)=O)CC(C)C)cc(O)nc(O)n1 C1(C(=O)NCC2(COC)CCCN2C(c2cccnc2)=O)CC(C)CC(C)(C)C1 N1(C(c2c(C(C)C)ocn2)=O)C(C(=O)NCCNC(=O)C(C)C)C2CC(O)C1C2 Cc1c(C(N2CCC(CNC(=O)CCCF)C(F)(F)CC2)=O)[nH]c2c1CCCC2 C(N=c1cccc(C(=O)OC)[nH]1)c1ncn(CC)n1 N1(C(C(C2(C)CC2)NC(=O)Cc2coc(C)n2)=O)CCCC(F)(CO)C1 N1(C(c2c(Cl)cn(CC)n2)=O)CC2(CCCC2NC(C2CCCCO2)=O)C1 N1(C(CC2(C)CCN(C(c3ccc(C=C)cc3)=O)C2)=O)Cc2ccnn2CC1C N1(C(c2n(C=C)ncc2)=O)CC2CC(C(=O)NCc3cnc(O)nc3O)CC2C1 C1(CNC(=O)CSCC(N2CC(F)C2)=O)CCCC(F)C1 N1(C(c2nccc(CNC(CCCC3C(C)C3)=O)c2)=O)CC2C(C1)C2(C)C c1(OC)ccc2oc(C(=O)N(CC(C)NC(=O)C(C)C#N)C)c(C)c2c1 C(CNC(c1ccncn1)=O)(CC(=O)Nc1ccc(CO)nc1)OC c1(CCC(=O)NCCN(CCOC)C(C2COCC(C)O2)=O)ccc(C)cc1C CC1CC(C)CN(S(=O)(=O)NC(c2cccc3cc[nH]c23)C)C1 c1(SC)ncc(Br)c(N(C(=O)Cc2ccc(Cl)cc2F)CC2CCCNC2)n1 c1(C(N2C(CC)C(NC(=O)CCC3CCCO3)CC2)=O)ccc(OC)cc1O N1(C(c2n(C)cnc2)=O)CCC2(CC(NC(C3CCC3)=O)C2)C1 c1(C(=O)NC2CCN(C(c3c(C)c(Cl)ccc3)=O)C(C)C2)cc2cnccc2[nH]1 c1(C(=O)NC(C2CCCC2)CNC(=O)CCOC2CC2)ncoc1C1CCCO1 N1(C(CCOC)=O)CC2CC1(CNC(c1ccc(-c3nc[nH]n3)nc1)=O)C2 CC(C)C(F)(F)CC(=O)NC1CCN(C(c2cn(C3COCC3F)nn2)=O)C1 c1(C(N2CC3C(NC(C(CC(C)C)F)=O)C3C2)=O)cccc2nccnc12 C1(CC)CN(C(c2ccc(C3CC3)cc2)=O)CCN1C(=O)C(CC)N(C)C CC1CCN(C(=O)CCC2CC2)C(CNC(c2ccc(C(C)(C)C)o2)=O)C1 N1(C(C(CC)OC)=O)CCC2(CCCN(C(=O)CNC(C3CCC3)=O)C2)CC1 c1(OCC(CNC(c2cc(-c3cccc(F)c3)on2)=O)O)ccc(Br)cc1 c1(C(=O)NCC2(NC(C3CC4CC4C3)=O)CC2)ccc(CO)o1 C1(C(=O)NC(C)C(CO)NC(=O)Cc2ccsc2C)(CC)CC(C)(C)C1 C1(NC(C(=O)OCC)=O)CC(F)C(C(=O)Nc2nc(C)sc2C(=O)NC)C1 CCC(CCC(=O)NCc1cccc(CNC(=O)C=CC(=O)N(C)CC)c1)OC Cc1cc(C(=O)NCC2CC(CNC(=O)Cn3ccnn3)CO2)ncc1F Cc1ccc(C)c(C(N2CCC(CNC(C3CCCN3N=O)=O)C2(C)C)=O)c1 c1(OC)c(C)cc(CN(C)CC2CCCN2C(C2CCC3(CCC3)O2)=O)cc1Cl N1(C(c2c(N(C)C)nccc2)=O)CC(NC(c2cnc(O)o2)=O)C(C2CC2)C1 c1(C(N(C=O)CC2CN(C)C2)C2CC2)ccc(F)cc1 C1(N(C(=O)CCn2cccn2)CC)CCCN(C(c2ncccc2C)=O)C1 C=CC(CCC)CC(=O)N1CCC(NC(c2ccccc2N2CCCC2=O)=O)C1 C#Cc1ccc(C(N2CCCC(CC)(NC(=O)CCNC(N)=O)C2)=O)nc1 N(C1COc2cccc(F)c21)S(c1ccc(NCc2c(C)ocn2)nc1)(=O)=O C1(CC)CN(C(C23CC2COC3(C)C)=O)CCC1NC(=O)C=C(Cl)Cl CCCC(O)C(CO)NCc1ccc(CCC)cc1 N1(C(CNC(c2c(C(C)C)onc2)=O)C)CCN(C(=O)CC2(O)CCOC2)CC1 c1(-c2cn(CCCOCC(=O)NC(CC)(C)C3CC3)nn2)scc(C)c1C(=O)O N1(C(C=Cc2c(N)cccc2)=O)CCC2(CCN(Cc3cncc(O)c3)C2)C1 C=CCC(CC(C)C)C(=O)N1CCCC1CN(C(=O)CC1CC(N(C)C)C1)C C1(OCC(=O)NCC23C(CN(C(C(C)c4cncs4)=O)C2)C3)CCC(F)(F)CC1 N1(C(c2c(C(C)C)[nH]cc2)=O)CCCCC1C1(NC(C2CCN(C)C2=O)=O)CC1 C(=O)(C(C)(CNC(c1n[nH]cc1CC)=O)CC)N1C(C#C)CCC1 Cn1ncc(C(=O)NC2CN(C(=O)Cc3cccnc3O)C3CC23)c1Cl N1(C(CCS(C)(=O)=O)=O)CC2CCC(C1)N2C(c1ccc(F)cc1Br)=O n1(CC)cc(CC(C(=O)NCC(=O)NC2(CC)CC2)C2CCC2)nn1 c1(C(N(C2CCCC(NC(Cc3c(C)scc3)=O)C2)C)=O)ccc(N)c(F)c1 C1(C(=O)NC2CN(C(c3c(OC(C)C)nccc3)=O)C(C)C2)CC2CC2CC1C N1(c2nccc(C(=O)OCC)n2)CCS(=O)(=O)C(CCNC(=O)CN(C)CC)C1 c1(C(=O)NC(C2N(C(C(=O)NC(C)C)=O)CCC2)C)ccnc2c1nnn2C CCC(CNC(c1sc(NC2CC2)nc1C)=O)(CC)NC(C1CC=CCO1)=O N1(C(=O)C2=CCOCC2)CC2CCC(NC(C3CC4CCC(C3)S4)=O)CC2C1 c1(CC)c(C(N2CCCC(C(C)(O)CNC(=O)C=CSC)C2)=O)cccc1C c1(C(=O)NCC(CNC(CC=CC=C)=O)C)cc2cccnc2s1 C(=O)(C(CC=C)C(C)C)N1C(CN(C(c2nccc(C#C)c2)=O)C)CCC1 C1(NCC2(NC(C3CCN(C(=O)NC)C3)=O)CCC2)C2CCC(F)(F)C12 C1(C(N2CC3C(CNC(c4ccccc4O)=O)C3C2)=O)CC2(CCC2)CO1 Cc1n[nH]c(C)c1S(=O)(=O)NC1CN(c2ncnc3c(Br)csc23)C1 c1(C(=O)NC2CCC(C(N=c3cc(C)o[nH]3)=O)CC2)c(F)ccc([N+](=O)[O-])c1F N1(CC(C)C)CCCC1C(N1CC(C(C)NC(=O)C=CSc2ccccc2)C1)=O c1(OC)ccc(C(=O)N(C(=O)CC2CCC(C(F)(F)F)N(C)C2)C2CC2)nc1Br c1(C(N2CCC(COC)(CNC(c3ccc(C)o3)=O)C2)=O)cc(F)c(F)cc1O C(C(C)(C)CC(=O)N1CC(n2cnnc2)C1)NC(Cc1cc(C)nn1C)=O c1(C(=O)NCC2CCC(NC(C3(CC)COC3)=O)C2)ccc(-c2ccsc2)cc1 C1(C(N2CCC(NC(c3cnn(CCC)c3C)=O)C2C)=O)Cc2ccccc2C1 Cc1nc2c(n1C)CN(C(=O)NCc1ccc(C3CCCCC3)o1)CC2 O=C(C1=CCOC1)NC1CN(C(c2cccc(-c3ccccc3)n2)=O)C2CC12 Cc1csc(=O)n1CCC(=O)NCC1CCC(NC(=O)CSC2CC2)C1 CC1=C(C(=O)NCC2CN(C(=O)C(C)CC3CCCO3)C(C)(C)C2)CCO1 c1(N(C)C)ccc(-c2cc(CN3CCCCC3)[nH]n2)cc1 C1(NC(c2ccc(C(F)F)cc2)=O)CN(C(=O)Cc2sc(O)nc2O)C2CC12 CC(C)C(C)(CNC(c1cc[nH]c1)=O)NC(C1CC1F)=O C1(CCOC)(C(=O)NCCN2CCC(C)C2)CCN(C(=O)C=CC(C)(C)C)CC1 Cn1nc(Br)cc1C(=O)NCC1(C)CCCC1NC(C1CC1(C)C)=O C1(C)(C(NOCCCOC)=O)CC(O)CN1C(c1c[nH]nc1C1CC1)=O c1(C(N(C(C)CNC(=O)CCN2CCCCC2)C)=O)cc(N)cc2ccccc12 C1(CNC(C#CC(C)(C)C)=O)CN(C(=O)CC2CCSC2)C2(CCC2)C1 C=CCCC(=O)N1CCCC1C(C)(C)CNC(c1cnn(CC=C)c1)=O c1(CC(=O)NCC(C)N(C(C2(C)CC(F)(F)C2)=O)CC)c[nH]c(=N)nc1O C1(NC(=O)C=Cc2ccoc2)CCN(C(C2(F)CC2)=O)CCC1c1ccccc1 N1(C(C(CCC)CCC)=O)CCc2sc(CNC(=O)COCC3CC3)nc2C1 N1(C(C(COC)(F)F)=O)CCC(CNC(c2cn(C)cn2)=O)C(F)(F)CC1 N(C(=NCC1C(C)(C)C1(C)C)NCC1(C#N)CC1)C(c1cccs1)C c1(C(C)NC(C(=O)Nc2c(C(=O)OC)cccc2)=O)nc(Cl)ccc1Cl CCN=c1nc(NNC(=O)Nc2cccc(C(O)CC)c2)[nH]c(=NCC)[nH]1 c1(OC)ccc(Cl)c(C(=O)N(C(C)CNC(c2csnc2C)=O)C)n1 C=CC(C)(O)C(=O)NC(c1ccc(F)cc1)CNC(=O)C(C)(C)N(S(C)(=O)=O)C c1(C(=O)NCCC(C)NC(c2cc[nH]c2-c2ccccc2)=O)ccc(F)cc1Cl C(=O)(CC1=Cc2ccccc2C1)NC1(CCOC)CCN(C(C=CCC)=O)CC1 N1(C(c2[nH]ccc(=N)n2)=O)CCN(C(=O)C2=C(Cl)CC2)C2CCCCC2C1 C(=O)(CC(CC(C)C)NC(=O)Cc1ccc(C#N)cc1)NC1CCN(C(C)=O)C1 N1(C(C(CC(N)=O)O)=O)CC2CN(C(c3scnc3Cl)=O)CC2C1 N(C1CCCn2cnnc21)C(=O)CC1CCN(C(C2CC3CCCC3C2)=O)CC1 c1(NC(C2N(C(c3ccc(C(C)O)cc3)=O)CC2)=O)ccc(S(N)(=O)=O)cc1Cl C=CCCC(CC(C)C)C(=O)N1CCCN(C(c2ccc(C(N)=O)s2)=O)C(C)C1 C(CCCC(=O)NC(C)CCC1CC1)N(C(C(C)C1CCOC1)=O)C C(=O)(CC(C(F)(F)F)n1cccn1)OCc1c(F)ccc(CC)c1 C1(COC)(NC(=O)CCc2cnn(C)n2)CN(C(=O)Cc2ccc(C)o2)C1 c1(C(=O)NC2C(CNC(c3cc(N)c(Cl)nc3)=O)CCC2)ccc2cnnn2c1 C1(CNC(c2cc(C)ncn2)=O)N(C(=O)CN2CCCS2(=O)=O)CCC1(C)C N1(C(C(c2ccccc2)OC)=O)CCC(C2CC(NC(c3cc(C)c[nH]3)=O)C2)C1 C12(C(=O)NCCN(C(CCCNC(=O)OC)=O)C(C)C)CCCCC1NC(=O)C2 C1(C(=O)NCCCC(C)NC(c2c(C)ccs2)=O)COCCN1CC(F)(F)F c1(C(=O)OC)cc(-c2ccccc2OC(F)=C(F)F)c2cc(C(F)(F)F)[nH]c2c1 Cc1cccc2cc(C(=O)NCC3CN(c4cncc(Cl)n4)CCC3(F)F)[nH]c12 N1(C(C2(CC#C)CC=CCC2)=O)CCN(C(c2ncc(Cl)n2C)=O)C2(CCC2)C1 N1(C(CC2CCC(OC)CC2)=O)CCC(C)(NC(C2CCCS(=O)(=O)C2)=O)CC1 O=C(Cc1csc(C(=O)O)n1)NNC(=O)N=c1cc2n([nH]1)CCCC2 CCC(O)C(C)C(=O)NCC1(O)CCN(C(c2cnc(C(C)=O)s2)=O)C1 N1(C(c2c(C)csc2Cl)=O)CC(CNC(C2(C)CCC(=O)NC2)=O)C2(CC2)C1 C(N=c1[nH]c(N2CCC3(C2)CN(C)C3)nc(=N)[nH]1)C1CCC(C)(CC)O1 N1(C(c2ncccc2Cl)=O)CCC2C(C1)CN2C(=O)CCSCc1ccccn1 N(C(=NCCc1cccs1)N1CCC(N2CC=CC2)C1)CC(CC)(C)Cl N1(C(c2cc(C)c(C)o2)=O)CC(N(C)C(C2CCCC(O)C2)=O)C(C)(C)C1 C(CC(C(=O)NCC1(C(C)(F)F)CC1)NC(C12CC(F)(C1)C2)=O)N(C)C c1(NC(CC2CCN(C(c3cc(OC)c(I)cc3)=O)C2)=O)ccc2c(c1)OCC2 c1(OCCCCNC(=O)C(N)=O)cnc(O)cc1C(=O)O.CC(C)(C)O C(C)(C)(C(C)CC(=O)N1CCC(C2CC2)CC1)NC(C1CN(CC)C(=O)C1)=O CC(=O)CCCCC(=O)N1CC2(CCCC2)C1C(N1CCN(CC2CC2)CC1)=O N1(C(C(CCOCC)NC(C2C=CCC2)=O)=O)CC2(CC=CC2)C1 C1(CNC(C2C(CC)C2)=O)C(C)CCN1C(=O)CCN1CCNC(=O)C1 Nc1cccnc1C(=O)NC(CC1CCCC1)C(N1CCCC(F)C1)=O c1(OC(C)C(=O)NC2CN(C(c3c(Br)nnn3C)=O)C2)ccc(F)cc1 C(=O)(C(F)(F)CO)N1CC(CC(C)NC(c2cnc(-c3ncccn3)s2)=O)C1 CCCS(=O)(=O)C(C)C(=O)NC1CCC(NC(c2cncc(C3CC3)c2)=O)C1 C(=O)(CCCC(=O)NC1(C)CC(NC(=O)CC(O)CC)C1)NCC C(C(C)S(=O)(=O)c1ccccc1)NC(C1=C(C)OCCS1)=O C12(CNC(C(C=C)(C)CC)=O)COCCN1CCN(C(C1(Cl)CC1)=O)C2 C(=O)(C(Cc1cccnn1)NC(c1ccsn1)=O)OC C(=O)(CC(C)(O)CCC)N(C1CCN(C(=O)COCCSC)C1)CC c1(CN(C(CC2CCN(C(C(CC)C)=O)C2)=O)C)ccc(OC)nc1 C1(C(N2CCC(C=C)CC2)=O)CCN(C(=O)C(C)=CC(C)(C)C)O1 CCCC(O)CC(=O)NCCCCNC(=O)C(F)(F)C(O)c1ccccc1 N1(C(C(C2CCCC2)NC(CC(C)C2CC2)=O)=O)CC(O)C(O)C1 Cc1n[nH]cc1CCNC(C1(NC(c2csnn2)=O)CC1(C)C)=O c1(N(C)CC2CC2)nc(N2CCS(=O)C3(CCC3)C2)nc2c1CCCCCC2 C1(C(=O)NC(C2CCCN2C)C)CC2CC2N1C(C1CCN(C)CC1)=O C12(CC(=O)NC(C)C(CO)NC(=O)C(C)OC3CCCCC3)CCC(CC1)CC2 c1(CC)c(C(=O)NC2CC(CNC(=O)C(C)C(C)(C)C)C2)cccc1F Cc1nc(C(=O)NCC2CCCCCN2C(=O)CC2COC(=O)C2)cn(C)c1=O N1(C(C(CC=C)NC(C)=O)=O)CCC2(CC1)CC2C(=O)N(CCCF)C N1(C(C2(C)CN(C)C(=O)C2)=O)CCN(C(C2CC(F)(F)CS2)=O)CC12CC2 C=CCC(C(=O)NCC=CCNC(=O)CCOCC1CCCO1)c1ccccc1 CCC(C)(C)C(O)C(=O)NCC(CC1CC1)C(=O)N1CC(C(F)(F)F)C1 C1(C(=O)NC2C(NC(=O)CCc3ccsc3)C2)CCC2CC2CC1 Cn1cc2c(NC(=O)CC3CCN(c4ncnc5c4CCC5)C3)cccc2n1 N1(C(C2(COC)CCOC2)=O)CCC2C(C1)CN2C(c1cccc2scnc12)=O C1(NC(C=C(C)C(F)F)=O)CN(C(c2ccc(C3CC3)c(F)c2)=O)CCC1C C1(C(=O)NC(C)CNC(c2ccc(CC(F)(F)F)cc2)=O)CC2C=CC1CC2 Cc1ccc2occ(C(=O)NCC34CC3CN(C(c3ccc(Cl)cc3)=O)C4)c2c1 CN1CC(O)CC1(C)C(N1CCCC(NC(c2cc(O)ccc2F)=O)CC1)=O N(C1CCc2cccnc21)C(CNC(CC(CCCC)O)=O)=O C1(CNC(C(c2c(C)cccc2C)O)=O)CC2CC(C1)N(C(=O)CC#N)C2 N1(C(C23CN(C(=O)CSC4CC4)C(C2)CCO3)=O)CCN2C(=O)NCC2C1 c1(NCC2OCC(CNC(c3c(C)cc(CC)o3)=O)C2)cnc(C#N)cn1 C1(C(C)=O)CC(C(=O)NC2CC(NC(=O)C(C)(C)c3cccs3)C2)C1(C)C C1(O)(CN(C(COC)=O)C)CCCN(C(C2CCC(=O)N(C3CC3)C2)=O)C1 CCC(CCC(=O)Nc1cnn(C)c1C)NC(=O)CCc1ccco1 c1(CC(N2CC(F)CC(NC(c3n[nH]cc3Cl)=O)C2)=O)coc2ccc(F)cc12 N1(C(C2C(c3n(C)cnc3)C2)=O)CCC(F)(NC(c2cccc(Br)c2F)=O)CC1 N1(C(C2CC(N(C(=O)CC3(O)CCCC3)C)C2)=O)CCc2ccsc2C1 CC1CC2(CCN(C(=O)C3=COCCC3)CC2)CN1C(C1CCCC(C)(C)O1)=O c1(OC)c(NC(C2C3CCC2(c2ccccn2)C3)=O)cccc1C(=O)O c1(CC)cn2c(n1)CC(C(=O)NCC(C1CCC(F)(F)CC1)C)CC2 C1(SC)CCCC1n1cc(C2(C)CN(C(C3CCCN3C(C)C)=O)C2)nn1 C1(CN(C(C(C)n2cccc2)=O)C)CN(C(c2cc(C(N)=O)c[nH]2)=O)CCO1 C1(NC(C(CCCC)=O)=O)CN(C(c2cn(CCC)nn2)=O)C2(CCC2)C1 C1(NC(c2n(CC)nnc2)=O)CC2(C1)CC(C(=O)N(CC(C)C)CC(C)C)C2 O=C(C1=C(c2cccc(F)c2)CCC1)NCC1(c2cccc(F)c2)CCC1 C1(C(N2CC(NC(C(C)(C3CC3)OC)=O)C(SC)C2)=O)CCC(C)(F)CC1 c1(C(=O)NCCN(C(C(N)=O)=O)CCc2ccccc2)[nH]cc2c1CCCC2 CN1N=C(C(=O)NC2CC(NC(c3cnc(Cl)c(O)c3)=O)C23CCC3)CCC1=O CC1(C(F)(F)F)CCN(C(=O)COC(C2(c3ccccc3)CCC2)=O)C1 C(C)(CCC(=O)N1CCOC(CNC(c2cn(CCC(C)C)nn2)=O)C1)OC N1(C(C(C)NC=O)=O)c2ccccc2CC1C(F)(F)F c1(CNC(c2cccnc2O)=O)cc(O)nc(CNC(C2(CO)CCC2)=O)n1 c1(OC)ccc(C(=O)NC(C)CC2CCN(C(c3cccs3)=O)CC2)c(C)n1 N1(C(c2nc(C)oc2)=O)CCC(NC(=O)C=CC(c2cnn(C)c2)=O)CC1C c1(OC(C(=O)NCC(C2CCN(CC)C2)OC)F)ccccc1COC(F)(F)F c1(C(=O)NC(C2N(C(=O)NCc3cc(OCC)n[nH]3)CCC2)=O)cncc(C)n1 C1(C(N2C(CNC(CCN(C)CCO)=O)CCCCC2)=O)CCc2nccn2C1 C1(CNC(C2=NOC(C)C2C)=O)CN(C(C2(F)CCC2)=O)CC12CCC2 CN1CC=C(CC(=O)NCC(C)(C2CC2)NC(c2cc3cnccc3o2)=O)CC1 C12(C(=O)NCCS(CC)=O)CCNCCC1C2 N1(c2snc(CCC)n2)CCC(C)C(NC(=O)C(C)(c2ccccc2)N(C)C)C1 Cc1csc(C=CC(=O)NC23CC2CN(C(C2(c4ncco4)CC2)=O)C3)n1 N(C1CCOc2cccc(Cl)c21)C(C(n1cc(-c2cccc(Cl)c2)nn1)C)=O c1(SCC(C)=O)cccc(NC(=O)NC(c2nnc(C)o2)CC)c1 C(=O)(C1CCCc2ncnn21)NC1(C)CCCN(C(CCC#C)=O)C1 c1(-c2n(-c3ccc(C(=O)OCC4CCN(C)C4)cc3)cnc2)cc2ccccc2o1 CCCC(C#N)C(=O)N1CC(NC(c2cc(-c3cnn(C)c3)on2)=O)CC1(C)C N1(C(COCC#C)=O)CC(NC(=O)C(CC#C)C2CC2)C(O)C1 N1(C(C(CC=C)CC)=O)CC2CCC1C(CNC(c1ccc(=O)n(CC)n1)=O)C2 N1(C(C2CCN(C(CCC3CC(C)C3)=O)C2)=O)CCc2cc(F)ccc21 c1(OC)ccc(C(=O)NCC2CC(OC)CN2C(C2CNC(=O)N2C)=O)cc1F c1(-c2ncc[nH]2)ccc(Cl)cc1.C1(CN(C(c2ccsc2)COC)C)(OC)CCCC1 CC1(C)CCC(C(=O)NC2(C(=O)Nc3cc(F)ccc3O)CCSC2)CO1 N1(C(CCOCC)=O)CCCC12CCN(C(c1cc(N)c(Cl)c(O)c1)=O)C2 N1(C(CC(C)(C)NC(=O)CCCC#N)=O)CCC12CCC(O)CC2 Cc1ccc([N+](=O)[O-])cc1C(=O)NC1CCN(CCC(F)(F)F)C(C)C1 C(C)(c1ccccc1C)=CC(N1CC(COC)N(C(C2CC(C)=NO2)=O)CC1)=O CC1(C)COC(CCNC(C2(NC(=O)C(F)F)CCCC2)=O)C1 C(=O)(C(COC)COC)N(CC(C)NC(CC(n1c(CC)ncc1)C)=O)CC Cc1cccnc1C=CC(=O)NCCN1CCN(C(C2(C)C=CCCC2)=O)CC1 N1(C(CNC(c2n(CC)ncc2)=O)C(F)F)CCN(C(=O)CC2CCOC2)CC1 c1(OC)cc(N2CC3CC(NC(=O)C(C)=C4CCC4)C3C2)ccc1[N+](=O)[O-] C1(C(=O)NC2CCC23CN(C(c2cc(Cl)c[nH]2)=O)C3)CCc2nccn2C1 C1(COC)CN(C(c2ccnn2-c2ccccc2)=O)CCN1C(C1CC1(F)F)=O CC(O)C(C)(C)C(=O)NCC#CC(=O)NC1CC(=O)N(C2CC2)C1 NS(=O)(=O)c1n[nH]cc1C(N1CCC12CN(C(c1ccnc(Cl)c1O)=O)C2)=O C1(F)(C(=O)NC(CC)CNC(=O)Cc2ccc(Cl)s2)CC=CCC1 N1(C(c2cccc(NC(C)=O)n2)=O)CC2(CCC(CNC(C3CC3CF)=O)O2)C1 C(c1cncc(F)c1)=CC(=O)NC1CC(NC(c2cccc(Br)c2)=O)C1 C(C)(C)(CC(=O)NCC1CC2CCC1C2)NC(Cc1c(C)ncs1)=O N(C(=NCCc1ccccn1)NC(c1ccc(N(C)C)cc1)C1CC1)C(C)CF c1(C(N(C2CC(NC(CCOC)=O)C2)C)=O)cnc(-c2ccoc2)s1 C(=O)(CCC(=O)N1CCC(F)(CNC(C2CCC(C)(C)O2)=O)C1)NC N1(C(C2N(C(C3C(c4cccc(C)c4)C3)=O)CC2)=O)CCCC2(COC2)C1 N1(C(C2C(CC)CCO2)=O)CCN(C(=O)CC=Cc2ccc(F)cc2)CC1CO C1(CC(=O)NCC(COC)NC(=O)C=Cc2ccncc2)CCCC(OC)C1 C(=O)(CCC(C)(C)C)NC1C(CNC(C2CCCN(C(C)=O)C2)=O)C1 N1(C(C2CCC(C(C)(C)C)CC2)=O)CC2CCC(NC(=O)C=C3CCC3)CC2C1 C12(CC(n3cc(C4CN(C(=O)Cn5ncnn5)CCO4)nn3)C)CCC(CC1)C2 C1(NC(C2(CCCC)CCC2)=O)CCCCCC1NC(=O)CC1CCN(C)CC1 c1(OC)nscc1C(=O)NC1CC(O)C1CC(=O)NC1(C(=O)OC)CC1 C1(NC(c2cn(CC=C)nn2)=O)CCN(Cc2nc(CCCC)no2)C(C)C1 CCC(CC)(CC(=O)OC)C(=O)NCC(C)CSC C(=O)(C(O)C(F)(F)F)NCC(C)(C)CNC(C1(n2cccn2)CCC1)=O c1(CC)ccc(C(=O)NCCC(C)C(OC)OC)cc1Cl c1(C(=O)NCC2(NC(CNC(=O)OCC)=O)CCCC2)ccccc1CC(C)C N1(C(C(C2CC2)OC)=O)CC(C2CN(C(c3ncc(Cl)cc3Cl)=O)C2)C1 CCC(C)(CNC(=O)C(F)(F)c1nc(C)cs1)NC(c1nocc1C)=O C1(CC(=O)NC2(CF)CCN(C(c3c(C)ccnn3)=O)C2)CCC2CC1C2(C)C Cc1ccnc(CNC(=O)N(C)Cc2nnn(C(C)C)n2)n1 CC1(C)CCOC1C(=O)NCCC1(C)CCN(C(c2cccc[n+]2[O-])=O)C1 CCCCC(CC)C(=O)N1CC(C2CCCCN2C(c2cc3n(n2)CCO3)=O)C1 O=C1COc2cc(F)c(C(N3CCCC(NC(C4CNC(=O)N4)=O)C3)=O)cc2N1 C1(C(=O)NCC(C)NC(=O)C(=O)NCC(F)(F)F)CCCN1C1CCCC1 C1(CNC(c2c(C)nc(C(C)C)s2)=O)CN(C(c2cc(N)ccn2)=O)CC12CC2 c1(CN(C2CCC3(CCC3)C2)C=O)ccc(F)c(C(F)(F)F)c1 c1(OC)c(C(N2CCC(CNC(c3cccnn3)=O)C23CC3)=O)ccnc1Cl C1(C2CCN(C(=O)CCc3cc(Cl)cs3)C2)(NC(=O)CN2CCCC2=O)CC1 O=[N+]([O-])c1cnn(CCN2CCOC(c3cn(CC(F)(F)F)nn3)C2)c1 c1(C(=O)Nc2c(F)cc(I)cc2F)n[nH]c2c1CN(c1ccnc(Br)n1)CC2 c1(OC)ccc2ncc(C(=O)NC3CN(C(=O)CN(C)S(N)(=O)=O)CC3F)n2n1 N1(C(C(C)OC2CCCCC2)=O)CC(C2CN(C(=O)C(C(C)(C)C)C3CC3)C2)C1 c1(C(=O)NCc2cc(C(=O)NC(C34CCC(CO3)C4)C)on2)ccnc(CO)c1 Cc1cc(-c2cn(CCCC(=O)NC3CCCOC3(C)C)nn2)c(C)cc1Cl CCC(C)(COC)CNC(=O)C(c1cn(C)nn1)NC(=O)C(C)=CC1CC1 C(=O)(C1CCc2cccnc21)N1CCCCC(N(C)C(c2csc(CO)n2)=O)C1 C1(C(=O)NCC(C)(C2CCC2)NC(=O)CC23CC(C2)C3)CC2(C1)CC(F)(F)C2 N1(C(Cc2ccn(C(C)C)n2)=O)CCN(C(=O)CC2CCCC2)CC1C1CC1 C1(C)(C(=O)NCC2CC(NC(c3c(OC)nccc3)=O)C2)CCCC1(F)F C(=O)(C(C)Cc1ccncc1)NC1C(NC(CCOCCC)=O)CC1 CC1CCC(C(=O)NOCCCCF)CN1C(C1(C)CCCN(C)C1)=O CCCC(C)(C)CC(=O)N(C(C)CC(N1CCN(C)C(=O)C1C)=O)C c1(C(=O)NC2CC(F)(CNC(CC(C)C)=O)C2)cnn2c(=O)cc[nH]c12 C(C(C(C)(C)C)NC(c1cc[nH]n1)=O)NC(C(n1ccc(C(F)(F)F)n1)C)=O C(C)(C)(CCN=c1[nH]cnc2cccnc12)NC(c1nc(C(C)C)sc1)=O C1(CNC(C(n2ccc(C)n2)C)=O)CC2(CCC2)CN1C(=O)OC(C)(C)C N1(C(C=C(C)C(C)(C)C)=O)CCC(O)(CNC(=O)CCc2ccnc(Cl)c2)C1 C1(NC(=O)C(c2ccc(F)cn2)(F)F)CC12CCN(C(c1coc(Cl)n1)=O)CC2 c1(CN2CCCC(OC3(CO)CC3)C2)cccc2ncnn12 c1(C(C)C)ccoc1C(=O)NC(Cc1cnc[nH]1)C(=O)NC1CCCSC1 c1(C(=O)OC)ccc(NC2CC2C(=O)NCc2cccc(C(=O)OC)c2)cc1Cl C1(C(=O)NCc2cccnc2F)CCC2(CC2)N1C(c1csc(Cl)c1)=O CC1(C)CN(C(=O)CCc2ccncc2)C(CNC(=O)CN2CC=CC2)CO1 N1(C(c2c(CC)cco2)=O)CCC(C)CC1C(=O)NCC(C)(F)C(C)C N1(C(C2C(C)(C)CC2)=O)CCCC(F)(CNC(c2ccccc2C(F)F)=O)C1 C#CC1(C(=O)NCCCC(O)CO)CCN(C(=O)C(C)CSC)C1 C1(CNC(C2C(C)N(C)CC2)=O)CC2(CCN(C(c3csc(Cl)n3)=O)CC2)C1 N1(C(CC2C(C)(C)C2)=O)CC(C2CN(C(c3ccc(C(F)F)c(F)c3)=O)C2)C1 C1(NC(Cc2cn(C)nc2)=O)CCN(C(=O)CN2C(=O)CNC2=O)CC12CCC2 C1(C#N)(C(=O)NCCN(C(c2c(N(C(C)=O)C)cccc2)=O)C)CCCOC1 N1(C(C(C)=C(C)C)=O)CCCCC1CC(=O)NCc1nn[nH]n1 c1(C(N2CCCC(C(=O)Nc3ccc(SC)cc3)C2)=O)cc(Cl)cc(Cl)n1 C1(NC(=O)COC2CCOC2)CC(NC(c2cc(C3CC3)cs2)=O)C(O)C1 c1(CC(=O)NC(C)CCCNC(c2c[nH]cc2Br)=O)noc2ccc(F)cc12 c1(C(=O)NCC2N(C)CCN(c3ncnc(Cl)c3F)C2)cc2cccnc2s1 N1(C(=O)Cc2cccnc2Cl)CC2CC(Nc3cc(C4CC4)ncn3)CC1C2 C1(CC=C)(C(N2CCOCC2C)=O)CCCN1C(=O)C(O)C=CC C1(C(=O)NC(C=C)C2CC2)C2CCCC2CN1C(c1nccnc1N)=O CC1(C(=O)NCC2(CCNC(c3cc(F)ccc3F)=O)CC2)CCC(=O)CC1 C(=O)(C1=CC2CCC(C1)C2)NC(c1cn(C)nn1)C(N1CC(C)CN(C)CC1)=O c1(CC)ocnc1C(=O)NC(C)C(=O)NCCCN1CCOCC1 c1(C(CNC(C(=O)N(CC#C)CC2CCCO2)=O)C)cccc(F)c1 C(C(O)CN(C(=O)CCC1CCCO1)C)N(C(=O)CC1(CO)CCC1)C C1(C2CC2)(CNC(C(c2n(C)ncc2)NC(C2C3CCC(F)C23)=O)=O)CCC1 c1(C(=O)NC2(CO)CCN(C(=O)CCCC3CCCCC3)C2)n[nH]c2c1COC2 C1(CNC(CC2CC(CC)C2)=O)CC12CCN(C(=O)COc1cncc(C)n1)CC2 N1(C(c2c(C)nncc2)=O)CCC2CN(C(c3oc(Br)nc3C)=O)CC12 N1(C(COCC=C)=O)C2CCC1(CNC(=O)Cc1c(C)cccc1C)CC2 c1(C(=O)NC(CCCC)CNC(C2C3CCCCC23)=O)ccc2nccnc2n1 N1(S(C)(=O)=O)CCCC1C(=O)NC1CCCC1NC(=O)CCCF c1(OCCC(=O)N(CCNC(C)=O)CC2CC2)ccccc1C#N C1(CN(C)C)CC(O)CN1C(C1CCOCC1NC(c1cnn(CCO)c1)=O)=O C(C)(CCCC(C)C)C(C=C1CCN(C(=O)N(c2cc(C)[nH]n2)C2CC2)CC1)=O N1(C(c2c(C(=O)O)cn[nH]2)=O)CCC2CC1CN(Cc1ccccc1)C2 Cc1cc(C(N2CCCC(CNC(=O)C(C(C)C)N3CCCC3=O)C2)=O)n(C)n1 c1(C(N(C(C(C)C)C)C)=O)occc1CNC(=O)CN(C1CCCC1)C C1(NC(C(C)CO)=O)CCN(C(=O)C(c2ccc(F)cc2F)(C)C)CCC1CO Cc1csc(C(=O)NCCC(O)CNC(c2ccccn2)=O)c1 C1(C(N(CCCCCCCC)C)=O)CN(C(=O)COC(C)CC)CC12CCC2 C(=O)(C1=NOC(C)C1C)NCC1CN(C(c2c(C)n(C)c(C(C)C)c2)=O)C1 CC1(C)CCN(C(=O)CP(C)(C)=O)CC1C(=O)NC1CCCSCC1 N1(C(c2ccc(NC)cc2Cl)=O)Cc2ccc(CNC(=O)C(C)C(C)O)cc2C1 N12CCOCC1C2.c1(C(C)C)ocnc1C(=O)OC(=O)C(Cl)(Cl)Cl CC1CC(NC(C2CCC(F)CC2)=O)CN1C(=O)Cc1ccccc1Cl C(=O)(C(CC1CCCC1)NC(=O)C(F)C1CCCC1)NCC(C)N(C)C C1(CNC(C(=O)N(C)Cc2ccccn2)=O)CN(S(=O)(=O)C2CC2)CCS1(=O)=O C(CCCCCCNC(=O)Cc1ccsc1C)n1cc(CSC)nn1 N1(C(C(C)c2cncs2)=O)CC2(CNC(=O)CCCOC(C)(C)C)CC1CO2 C1(CCNC(=O)CCc2cnoc2)CN(C(=O)CC2CCSC2)CCO1 c1(N(C2CN(C(C3CCCN3C3CC3)=O)C2)C)ncnc2c(Br)nn(C)c12 C=CCC(C)(C)CC(=O)N1CCCC(C)(C)C1CNC(c1cc(=O)n(C)cn1)=O C(CC(C)C)(C(=O)NCC(C)C)N(C(COC)=O)C N1(C(c2scc(C)c2)=O)Cc2c([nH][nH]c2=NC(=O)c2ncccc2Br)C1(C)C N1(C(C(C)Oc2ccccn2)=O)C(C(=O)NC(c2cnc[nH]2)C)C2CC(F)C1C2 N1(C(CC(CCCC)O)=O)CCC2(CCCN2C(=O)C(C)c2ccsn2)CC1 n1(C(C)(C)C)ccc(C(=O)N(C2CC2)CC2CC2NC(=O)CC2CCOCC2)c1 C1(NC(C2C3CCCC23)=O)CC2(CCN(C(c3cc(CO)ccc3O)=O)CC2)C1 CC1ON=C(C(=O)N2CCN(C(=O)CNC(C3CCCCC3)=O)CCC2C)C1C Cn1ncc(Cl)c1CC(=O)NC1CCC(CN(C(=O)C(O)C(F)F)C2CC2)CC1 C1(NC(C(C#C)(C)C)=O)CCN(C(=O)CCCCOCC)CC1(C)C Cc1ncc(Cl)c(C(=O)NC2CCC(N(C(=O)CC3CC4(CC4)C3)C)C2)n1 N1(CC(=O)N(CC#C)C)CCCC(CCNC(=O)NCCOC(C)(C)C)C1 C#Cc1ccc(C)c(NC(=O)C(C2CCCN(C(C3CCCOC3)=O)C2)(C)C)c1 CC(CCNC(=O)CCc1cccc(F)c1)CCNC(C1CC1(C)C(F)F)=O c1(OCC)ccc(I)cc1NC(=O)CNC1CC(=O)N(c2cc(F)ccc2F)C1 CC(C(=O)N(C)CCN(C)CC1CC(CN=[N+]=[N-])C1)=CC(C)(C)C N1(C(c2ccn(CCC)n2)=O)CC2CCC(C1)N2C(c1cncc(CC)c1)=O CCC(CC)CC(=O)NC1CCC(NC(c2cccc(C3(O)COC3)c2)=O)CC1 Cc1ccc(O)c(CCC(=O)NC2CCN(C(=O)Cn3cc(CON)nn3)C2)c1 CON=CC(=O)N1CCC(OCCNC(=O)C(C)=C2CC2)C1 c1(NC(C2C(C(C)NC(C(C)N(CC)CC)=O)C2)=O)cc(C)cc(Cl)c1 N1(C(COCc2c(C)cccc2)=O)CCC(NC(=O)CN=S(C)(C)=O)C(C)C1 Cc1cc(C)c(NC2C3CC4C2C4C3C(=O)NC(=O)C(C)C(O)C(C)C)cc1N C12(C(=O)NCCCC(c3ccccc3)NC(C(C)SC)=O)CCCC1C2(F)F C1(NC(c2cc(C3CC3)no2)=O)CC2CCC1CN(C(C1CSCCS1)=O)C2 C(C)(CC(=O)NC1CCCC1CC(=O)N(CC(C)C)C(C)C)SC C1(NC(C(N)=O)=O)CC2CN(C(c3coc4c3CSC4)=O)CC12 C1(NC(C(c2cccc(O)c2F)(C)C)=O)CN(C(C2CC2F)=O)CC2(CCC2)C1 N1(C(C2CC(OC)(OC)C2)=O)CCC(CC(=O)NCC(F)(F)Cl)CC1 N1(CC(=O)NCC2CN(C(c3cnccn3)=O)CCO2)CCCCCCC1=O c1(C(=O)NCC2N(C(C(C)=O)=O)C3C(C2)COC3)cnc2c(Cl)cccn12 Cn1nc2c(c1C(=O)NCC1(CNC(=O)Cc3cccs3)CC(F)(F)C1)CCC2 c1(NCCC=C=C)cc(Br)ccc1S(=O)(=O)NC1CCOC(c2ccncc2)C1 c1(C(=O)NC2C3CCN(C(Cc4n(C)ncc4)=O)C3C2)cnc2c(c1)COC2 N#Cc1cccc(C(=O)NCc2cc(C(N3CCC(O)CC3)=O)no2)c1Cl C(=O)(CCCCN=[N+]=[N-])N1CC2C(CC(=O)NC(c3nc[nH]n3)CC)(CC2)C1 c1(OC)nccc(NCC2CCCC(CNC(C3CC(=C4CCC4)C3)=O)C2)n1 C(F)(C(=O)N(C1(C(=O)NCC(COC)OC)CC1)C)=CCC Cc1cccc(CCC(N2CCOC(CCNC(C3CC4CC4C3)=O)C2)=O)c1 N1(C(C2N(C(c3cn(C)nn3)=O)CC2)=O)CC(C)CS1(=O)=O.C1(C(=O)OC)(CC)CCC1 C1(CNC(c2cc(C#N)c[nH]2)=O)CN(C(c2c(C)cccc2)C)CC1(C)C C1(C(=O)NC(C2CN(C(=O)CC(C)(C)O)C2)C)CCC2(CC1)CC2 n1(CCC)c(-c2cscn2)nc2ccccc12.C1(N2CC2=O)CNC(CC(=O)O)C1 N1(C(CCC=C)=O)CCC(C)C1CNC(c1cnccc1OC)=O N1(C(=O)OC(C)(C)C)CC2(C1)CN(C(C1(Oc3ccc(C#N)cc3)CC1)=O)C2 C1(CNC(=O)CCOCC(F)(F)F)CCCN(C(=O)CC2CC(F)(F)C2)C1 c1(N(C(=O)CCC=CBr)C(C2CN(C(C)=O)C2)C2CC2)ccccc1[N+](=O)[O-] C1(CCC)CC(NC(C)(CCC2CC2)c2nnnn2CCCOC)CCO1 c1(CC(=O)NC(C(=O)N(C(C)CNC(=O)NC)CC)C)csc(C(N)=O)n1 c1(C(N2CCC(C)(CNC(CCC3C(C)C3)=O)C2)=O)ccc(C(F)(F)F)nc1N N1(C(C(C)=C(C)C)=O)CCC(CNC(=O)Cc2sc(O)nc2O)C12CCC2 C(CC(F)CN=[N+]=[N-])NC(C(CC=CC)NC(C1CCCCN1C)=O)=O C1(C(N(CCCNC(C(CCCC)(C)F)=O)CCO)=O)CCOC2(CCCC2)C1 C1(C)(CNC(CCCC=C)=O)CN(C(=O)C=Cc2cncs2)CCO1 C(=O)(C1=CC(C)(C)C1)N(CCN(C(Cc1ccn(CC)n1)=O)C(C)C)C C1(C(=O)NC2CCN(C(CCCCC(N)=O)=O)CC2)CC(=O)c2ccccc2C1 N(C1CS(=O)(=O)c2ccccc21)Cc1nc(-c2ccc(SC)s2)sc1 C1(CC(=O)NCc2ccc(C)cn2)N(C(=O)Cc2c(C)noc2C)CCC1(C)C C=CC1COCC1NC(=O)C(C(C)C)NC(C1C2CC(=O)CC12)=O C(C(C)(C)CC(=O)N1CCCCC1C(N1CC(C(N)=O)C1)=O)OC C=C(C)CC(=O)N(CC(CC)NC(C1CCCC1)=O)C N1(CC(=O)NCc2ccccc2)CCCC(NC(c2ccc(C(=O)O)[nH]2)=O)C1 N1(C(CC(C)(C)OC)=O)CC(C)N(C(=O)CC2(n3cccn3)CC2)CC1C C1(N(C(c2ccc(C)n2C)=O)C)CN(C(=O)C(O)C2CCCC2)CC1(C)C CC(C(=O)NN1CCCC1C(=O)NOCc1nc[nH]n1)n1cccn1 c1(CN2c3ccc(cc3)C2)ccc(C)cc1.C1(C(=O)OC)C=CC(OC(C)=O)C1 C1(C2CCN(C(=O)CC3CC=CC3)C2)(NC(c2c(Cl)ccc(OCC)n2)=O)CC1 C12CCCN(C1)CC(=O)N1CC(C1)CCCCNC2=O.C1(SCC)(CC)CC1 C1(C(=O)NC(CC)(C)CNC(=O)Cn2ncnn2)CNC(=O)C(C)(C)C1 n1(CC)nnc2c(NC3CCN(c4ccc(Cl)c(C)c4)CC3)ncnc12 C(=O)(C1CCc2cccnc21)N(C)CC1(O)CN(C(C2CC(F)C2)=O)C1 CS(=O)c1cc(C(=O)NC2CC(O)(CNC(C3CC(F)C3)=O)C2)ccc1F C1(C)(CCN(C(=O)C(CC2CCCO2)NC(=O)OCCl)C)CCOCC1.C(C)(C)C Cc1cc(C(N2CCC(NC(C3CC(C)(C)C3)=O)C2C(C)(C)C)=O)ncc1C#N N1(C(C(C)NC(=O)NC)=O)CCC(NC(C2(C)CC3CCC2C3)=O)C(F)C1 CC(C)(CCc1ccccn1)n1cc(C2CNCCO2)nn1 CC(C(=O)NCCCCC(C)NC(C1CCC2(CCC2)O1)=O)S(C)(=O)=O CN1CCN(C(C2(C)CCCC2)=O)CC1C(=O)NC1CCCC1C#N N1(Cc2n(C)cnc2)CC(=O)N(Cc2csc(N3CCOCC3)n2)C1=O C(=O)(C(C)C(O)C(C)CC)N1CCCC(F)(CNC(CC(=O)NCC#C)=O)C1 C(=O)(C1CCCc2nc[nH]c21)NCC#CCNC(C1=NOC(C)C1)=O C1(NC(=O)C2=COCCC2)CCOC2(CCN(C(C34CCC(C3)C4)=O)CC2)C1 C(C(C)(O)CC(=O)N1CCN(CC(=O)Nc2c(C)cccc2O)CC1)OC c1(C(N2CC(C)(C)C(CNC(c3cncs3)=O)C2)=O)ccc2c(c1)CCC2 N1(C(CC2(C)CC2)C(=O)NCc2cc(F)cc(Br)c2)CCCC12CCCC2 N1(C(CCC=CCC=C)=O)CC2CC2(NC(=O)CSc2ccccc2Cl)C1 C=CCCC(C(=O)NCCCCCN=[N+]=[N-])NC(=O)C(C)NC(C)(C)CC N1(C(c2csc(C)c2C)=O)CC(C)(C)CC1CNC(c1ccc(C(N)=O)s1)=O CC1(C)C2CC(C(N3CCCC3(C)Cc3ccccc3Cl)=O)CC12 C1(C(=O)NCCC2CCCCN2C(=O)CSCCC(C)C)(CC)CCC(O)CC1 c1(C(N2CCC(=CCNC(C(C)SCCCC)=O)CC2)=O)coc2c1CCCC2 N1(C(CC(CC)C)=O)CCC2(CCCCC2NC(=O)Cc2csc(S)n2)CC1 Clc1ccccc1C1(SC2CN(c3nccc(-c4ccc(Br)cc4)n3)C2)CCC1 C(CC(C(=O)NC(C)C(=O)NC1CCC(CCOC)CC1)OC)OC c1(C(N2CCN(Cc3cccc(OC)c3)CC2)C(=O)NCCC)cccnc1C C1(CC(=O)NC(C)C(N2CCCC2)=O)N(C(C2CC(N(C)CC)C2)=O)CCC1(C)C c1(C(=O)NCC2CCN(C(C3(O)CCOC3)=O)C2)c(Cl)sc2nnsc12 C(C(=O)NCC(F)CNC(=O)CNS(N)(=O)=O)(C(C)C)OCC Cc1noc(C)c1C(C)Cn1cc(CN2CCC(Cn3cncn3)CC2)nn1 O=C1OCC2CCN(C(c3cc(C4CCCN4)[nH]n3)=O)C12 c1(C(N2CCSC3CCC23)C(=O)NCc2ccccc2)cn2cc(F)ccc2n1 c1(NC(C(CCCOC)NC(C2OCCC2(C)C)=O)=O)cnc2ccnn2c1 C12(NC(c3n(C)nnc3)=O)CCOCC1CN(C(c1cc3scnc3[nH]1)=O)C2 CCCCC(=O)C(=O)Nc1cccc(NC(=O)C=CSCc2ccco2)c1 CC1CCn2cc(C(N3CCC(O)(CCNC(=O)CCN4CCC4)C3)=O)nc2C1 C(=O)(C(C)(C)N=[N+]=[N-])NCC(CC(=O)N(CC(C)(C)O)C)O c1(CC)cnc(C(=O)NC(C(=O)N(C2CC3(CSC3)C2)CC)c2ccco2)nc1 c1(NC(N2CCC(CC3CCCCO3)CC2)=O)cc(-c2cccc(F)c2)ccn1 C1(C(=O)NCCOCC=C)CN(C)CCN1C(c1cnc(O)c(C)c1)=O C1(OC)CCCC(NC(=O)CC2(OC)CN(C(=O)Cn3ccnc3C)C2)CC1 C1(NC(=O)NC(C2CCCCC2)COCCCC)Cc2nccn2C1 N1(C(c2cn(C)nc2)=O)CC2CCC1C(NC(C1(C)C=CCCC1)=O)C2 c1(CNC(C2CCC(CC)C2)=O)ccc(C(=O)NC2CCSC2)nc1 C(C(C(C)(C)C)NC(=O)C(C)(C)N(C)C)NC(c1ccc(C(C)=O)o1)=O N1(C(C=Cc2n(C)ncc2)=O)CCC2CN(C(c3nocc3Cl)=O)CCC2C1 c1(C(N2CC(C)C(NC(c3cccc4nonc34)=O)C2)=O)cc2ccncc2s1 c1(C(=O)NC2C(SC)CN(C(=O)C(C#N)C(C)C)C2)cc2cccc(N)c2cn1 N1(C(c2[nH]cc(C)c(=O)c2)=O)CCN(C(C2CCCCC2F)=O)CC(C)C1 N1(C(c2cc(SC)oc2)=O)C(C(N2CC(C)(OC)C2)=O)CCC1C1CC1 N1(C(C2(C(CC)=O)CC2)=O)CC2(C)CC1(C(N1CC3CC3C1CO)=O)C2 C=C(Cl)CCC(=O)NC1C(C(N2CCCC2C(C)(C)CO)=O)C1(C)C N1(C(Cc2nc(CC)sc2)=O)CCOCC1CN(C)C(C1(C)CCCOC1)=O N1(C(c2ccc(C#C)o2)=O)CCC(NC(=O)C2=CCCCC2C)C(CO)CC1 C(=O)(C1=CCOCC1)N(CCN(C(c1cnc(C(C)C)nc1)=O)CC)CC N1(C(CC(C)n2ccnc2)=O)CCN(C)C(C(N2CCCC2CF)=O)C1 N1(C(c2c(COC)noc2)=O)CCC(C)C1CNC(=O)COC1CCOCC1 Cn1ncc2ncc(C(=O)NCC34CCC(NC(=O)CC5CC5)(CC3)CO4)cc12 C1(C(N2CCC(N(C(=O)Cc3cscn3)C)C2)=O)CCS(=O)(=O)N1 N1(CC)C(C)CN(C(C2CCOCCN2C(=O)C(c2ccn(C)n2)C)=O)CC1C c1(C(=O)NC2C(CNC(CCSC)=O)CC2)ccc(C2(F)CC2(F)F)cc1 CC1(C)C2CCC1(C(=O)NC1CC(CNC(C3CC(OC4CC4)C3)=O)C1)CC2 c1(C(N2CC(NC(CCN(CC)CC)=O)C2)=O)noc2cc(Cl)ccc12 CC1(C)CC2(CC(C(=O)NCCC3CN(C(C4CC5CCCC(C4)C5)=O)C3)C2)C1 c1(CC)ccccc1C(=O)NC(C)C(C(C)C)NC(c1cnc(C)s1)=O C1(NC(c2cc(CC)on2)=O)CN(C(=O)OC(C)(C)C)CC(C)(C)C1 C(=O)(CC(O)CC(C)(C)C)NC1COCCN(C(C=Cc2occ(C)n2)=O)C1 c1(CC(=O)NCC2CCCCC2NC(c2ccon2)=O)ccc(F)cc1C(F)F CC(CF)N=c1ccn2ncc(S(=O)(=O)N3CCOC(C)CC3)c2[nH]1 CS(=O)(=O)c1cccc(Cl)c1C(=O)NC1CCCC(NC(=O)Cc2cscn2)C1 Cc1cncc(C)c1C(=O)NC1C2CN(C(C3CCCN3C=O)=O)CC12 C1(O)(CC(C)C)CN(C(C23CC(NC(C)=O)(C2)C3)=O)C1.C(C)(C)(C)OC=O N1(C(C2C(C3C(C)C3)C2)=O)CCN(C(=O)C(C)O)CC(C)(C)C1 c1(C(=O)NC2CC(=O)N(C)C2c2ccc(Cl)c(F)c2)ccc2c(c1O)CCCC2 c1(C(=O)NC2C(C)N(C(c3ccc(C(C)(C)C)nc3)=O)CC2)ccc(F)cc1F C1(NC(CP(C)(C)=O)=O)CN(C(=O)C=Cc2ccccc2F)CCC1CO c1(C(=O)NC(CCN(C(CC(C=C)CC)=O)C)C)ccn2cc(C)nc2c1 Cn1ncc(OCC(N2CC(n3cc(-c4cccc(F)c4)nn3)C(O)C2)=O)c1C#N Cc1cccc(Cl)c1C(N1CC(NC(c2cncc(Cl)c2)=O)C(C)(C)C1)=O c1(C(N2CC(NC(CCC)=O)CC2(C)C)=O)ccc(Br)c2c1OCCC2 c1(C(N(CCOCCN(C(c2cc(C)ns2)=O)C)C)=O)nc(Cl)c(Cl)s1 C1(NC(CCOCCN(C)C(C2CCS(=O)CC2)=O)=O)CCCC(O)C1O C(CC(O)C(=O)NC(C1CCOC1)C)NC(Cc1cnc(C)s1)=O C(N=C(NC)NC1CCOc2ccccc21)c1cc(C)nn1C.C1(OCC)CCCO1 c1(C(N2CCC(C(N3CCC(COC)C3)=O)(CF)C2)=O)cccn(C)c1=O c1(CC(C(=O)NCC(CC)NC(=O)C(C)CC(C)C)C)ccc(F)c(Br)c1 C1(CNC(N(c2ccc(Cl)cc2)C(C)C)=O)CCCC(C)CC1 N1(C(=O)OC)CCC(N=c2[nH]c(N(C)Cc3c[nH]nc3C)nc3c2COC3)C1 C(=O)(C#CC1CCOC1)N1CCC(CC(=O)NC(c2nncn2C)C)CC1 C1(NC(C(=Cc2cccnc2)C)=O)CC(NC(c2cnn[nH]2)=O)C12CCC2 C1(F)(C(=O)NCC2C(CNC(C3C(c4n(C)cnn4)CC3)=O)C2)CC=CCC1 N1(C(c2ccc(C)c(O)n2)=O)CC(C)CN(C(=O)CN2CC3CC3C2)C(C)C1 CC1=C(CNC(C2CC(F)CN2Cc2c(Cl)cccc2Cl)=O)CCC1 c1(OCC#C)ccc(Cl)c(OC(CCC=C)C2CC2)c1 c1(C(=O)NC(C)CCN(C(=O)CNC(c2cccs2)=O)C)cccc2c1CCN2 N1(C(C(C(CC)C)O)=O)CCC2CN(C(c3cc(C(N)=O)co3)=O)CC2C1 CC1(C)CCN(C(C2CCOC2(C)C)=O)C1C(=O)NCc1ncc[nH]c1=O CCCN=C(NCc1cc(C)cc(Cl)c1)NC1CC(=O)N(c2ccccc2F)C1 CC(C)CC(C(=O)NCC1CCC1CO)ONC(C1(C)CCC(=O)C1)=O c1(C(N2CC3C(C(=O)NCCS(C)(=O)=O)(C3)C2)=O)ccc2nc(Cl)ccc2c1 N1(C(c2ncc(C3CC3)cn2)=O)CC2CC(C(N3CCCC3)=O)(C2)C1 N1(C(Cc2nnc(C)o2)=O)CC2CCC2(CNC(C2CC(C(C)C)=NO2)=O)C1 C1(n2cnnn2)(C(=O)NCC(CO)NC(=O)C(C2CCCCC2)O)CCOCC1 C(=O)(C(O)CC(F)(F)F)NCC(CC)NC(c1cc2sc(C(=O)OC)cc2[nH]1)=O C=C1CN2C(=O)CCC2(C(=O)Nc2cccc(NC(=O)C(C)c3cccs3)c2)C1 C(=O)(C(CC(F)F)N(C)C(c1coc(C(F)F)c1)=O)NCC(COCC)C Cc1csc(C(N2CCCC(CC(=O)Nc3cnccc3C3CC3)C2)=O)c1C c1(C(=O)OC2CCN(c3cccc(C)c3)C2=O)cc(C)c(Br)c(C)c1 N1(C(C(C)OC2CCOC2)=O)CCCC(NC(C2(C)CSC2)=O)C1C N1(C(C2(C)ON=C(C)C2)=O)CCCC2(C1)CN(C(=O)CC1OCCCO1)CCO2 N1(C(c2nc(C)[nH]n2)=O)CCC(C2CCN(C(=O)C=C3CCC(C)(C)CC3)C2)C1 N1(C(C=Cc2ccc(C)o2)=O)CCC2(CC1)CCN(C(=O)C(C)CS(C)(=O)=O)C2 C1(CNC(CC=CC=C)=O)CN(C(=O)CC(c2ccc(F)c(F)c2)C)CCN1C c1(C(=O)NCC(C)NC(c2cc(C(F)(F)F)no2)=O)cn2c(n1)SCC2 c1(C(N2CC(C)(NC(=O)CC3(C)CCS(=O)(=O)N3)C2)=O)cc(Cl)c(F)cc1O C1(C(N(C)CC2CC2(C)C)=O)N(C(c2cnn[nH]2)=O)CCC1(C)C CC1CCn2cc(C(N3CCCC(F)(CNC(C4CC(O)C4)=O)CC3)=O)nc2C1 C#CCC(C(=O)NC1CC1C(F)(F)F)NC(=O)C=CC(C)C C1(CC(N2C3CN(C(c4n(C)ncc4)=O)C(C3)C2)=O)Cc2cccc(Cl)c2O1 C(C(=O)NC(C1CCCN1C(=O)CCn1ccnc1)C)(C(C)C)OCC(C)C N1(C(C(CCC)C(C)C)=O)CCC2CCN(C(c3nn[nH]c3Cl)=O)CC12 c1(NC(C(C)S)=O)n[nH]c2c1CN(C(=O)CN1CCNC1=N)CC2 Cc1c(F)ccc(C(N2CCC3C(NC(=O)CCCCC(N)=O)C23)=O)c1C#N c1(N2CC(CN(C(c3c(C)nc(O)nc3C)=O)C)C2)nc(Cl)nc2ccccc12 c1(-n2cc(C(O)C(F)(F)F)nn2)cn2c(n1)SCC2.C12(COC)CCN(C1)C2=O Cc1ccnc2nc(C(=O)NCCCCCCNC(C3CCNC3=O)=O)nn12 Cc1ccc(C(N)=O)cc1C(N1CCN(C(=O)C(O)Cn2cncn2)CC1C)=O Cc1cc(C2CC2)ccc1C(=O)NC1CC1NC(C1CN2CCC1CC2)=O N1(C2(c3ncc(-c4ccccc4)o3)CC2)CCCC1(C)C1CCCCC1 C1(C(N2CC(CNC(CC(C=C)(C)C)=O)C3C2C3)=O)Cc2cncn2C(=O)N1 CCC(CC)CC(F)C(=O)N1CC(NC(c2cncnc2)=O)CC(F)C1 c1(C(=O)NC(C(C)C)CNC(=O)CCNC(=O)CO)c(Cl)cc([N+](=O)[O-])cc1Cl C1(NC(C(CCSC)O)=O)CCN(C(c2cc(N)cc(O)n2)=O)C(C)C1 C(=O)(C(C)CC1CCCCC1)NCC(C)NC(c1coc(-c2cnn(C)c2)n1)=O C1(C(=O)NC2CCCN(C(c3csc(C)c3C)=O)C2)SC2C=CC1CC2 C1(C(NOCCC(C)C)=O)CCCN(C(=O)Cn2cnnc2O)C1 Cc1cc(F)ccc1NC(=O)C(CC(C)C)ONC(c1ccc(F)s1)=O CCC(C(=O)OC)C(=O)N1CSCC1C(=O)NC1(C)CCC(C)(C)C1 C12(CNC(c3c(C)noc3)=O)CCCCC1N(C(c1ccn(C(F)F)n1)=O)CC2 N1(C(C(C)(CO)NC(C)=O)=O)C2CCC1C1CC1(NC(c1cc[n+]([O-])cc1)=O)C2 C1(CC)(CC)CCCN(C(C2CCOCC2)C(=O)NCCCOCC2CC2)C1 C(CCCC(CO)NC(=O)C(COC)COC)NC(CCSCCC)=O c1(NC(c2n(CC)ncc2)=O)ccc(NC(C2(F)CC2)=O)c(F)c1 c1(C(=O)NCC(CN(C)C(C2CCC(F)(F)C2)=O)O)cc2cccnc2nc1O CCC(C(=O)N1CCN(CC(=O)NC2C(C)(C)C2(C)C)CC1)C(C)(C)CC C1(NC(Cc2cnc(C)s2)=O)CC(CNC(=O)C(C)c2ccsc2)C(O)C1 c1(COC(C(N2CCN(c3ccccc3)CC2)CC)=O)c(Cl)nc2ccccn12 n1(CCCCONC(=O)NCCC(c2ccc(Br)cc2)=O)cccnc1=O N1(C(CCCOC)=O)CCN(C(c2ncc(C(F)F)s2)=O)C(C(C)(C)C)C1 c1(NC(CCOC)Cc2cccc(Br)c2)cc(C(N)=O)ccc1NC(C)=O N1(C(C(CNC(=O)OC)(C)C)=O)CC(C(=O)NCC(C)(C2CC2)OC)CC(C)(C)C1 CCCCCC(C)(C)C(=O)NCC1CN(C(=O)Cc2cc(F)ccc2Cl)CC1C C1(NC(C2CC3(CC(=O)N3)C2)=O)CCCC12CCN(C(c1ncccn1)=O)CC2 c1(CC(=O)OCC(=O)S(=O)NOc2ccc(OBr)cc2)cc(F)cc(Cl)c1.OC(F)F C(=O)(CC(C)CNC(=O)C=Cc1cccnc1)NCC1(COC)CCCC1 N12Cc3ccc(cc3C1)N(C1CCNC1c1ccccc1)C(=O)C2=O.CC(C)C C12(NC(C3CN(C)C3)=O)CCC1CN(C(c1ccc(NCC(N)=O)cc1)=O)C2 C(=O)(C(CNC(=O)CC1OCCCO1)CC1CC1)NCC1C(CC(N)=O)C1 C1(C(=O)NC2C(SC)COC2)CCCCCCN1C(=O)CCCc1cnn[nH]1 C1(C(=O)OC)CN(C(=O)Cn2cc(CN)nn2)C2(CCC2)C1.C1(C)CCCCN1C c1(CSc2cccc(COC(NOC3CCC(C)C3)=O)c2)cc(O)nc(CN)n1 CCC(O)(C(=O)NCCC1(C)CCN(C(c2cc(Cl)cs2)=O)C1)c1ccccc1 CCCCC(CN(C)C(C1CC(N(C(=O)CC2CCOC2=O)C)C1)=O)CC C1(N(C(c2occ(C)c2)=O)C)CCC(NC(C2CC2c2ccsc2)=O)CC1 C(=O)(CC(C)(C)C)NC(C)C(=O)NC1(c2cn(Cc3ccccc3)nn2)CC1 c1(CC)ccc(C(=O)NC(CNC(c2cnn(C)c2C)=O)CC(C)C)c(Cl)c1 C(=O)(C(O)CCC(C)C)N1C(C(=O)NCCN(CCC)CCC)CC(OC)C1 c1(NC(c2cc(Cl)ccn2)=O)cnc(F)c(Br)c1 C1(C)(COC)CC(NC(=O)CCn2cccn2)CN1C(c1c[nH]cc(Cl)c1=O)=O C1(N(C(=O)C=CCN(C(=O)CC2(n3ccnc3)CC2)C)C)(CO)CCC1 Cc1c(Br)ccc(-c2noc(CSc3cccc(F)c3Br)n2)c1F O=S(=O)(c1ccc2[nH]c(=NC(CO)c3ccc(Cl)c(Cl)c3)sc2c1)NCCF O=C(C(O)CC(F)F)NCC1(F)CCCN(C(=O)COC2CCCC2)C1 Cc1ccc(NCC(=O)NCC(O)CNC(=O)COC2CC2)c(C)c1 C12(NC(c3n(C)c(S)nc3)=O)CCC(CC1)N(C(C1CCC3C(C1)C3(F)F)=O)C2 N1(C(=O)NCCCN2Cc3ccccc3C2)CC2CS(=O)(=O)CC(C1)O2 S(=O)(=O)(c1c[nH]c2ncncc12)N1CCN(CC23OCCC(N)(C2)C3)CC1 C#CC1(C(=O)NCC2CC(C(C)C)C2)CCN(C(C2(C(F)(F)CC)CC2)=O)C1 c1(-c2cn(C3CCN(C(C4CCS(=O)(=O)C4)=O)C3)nn2)ccc(F)nc1 C1(NC(c2n[nH]cc2F)=O)CN(C(c2cnn3c2CCC3)=O)CC12CCOCC2 N1(C(CS(CC)=O)=O)C2CCC1CN(C(=O)Cc1cnns1)C2 c1(C(C)OC)nc(C(=O)NCC2(OC)CN(C(c3conc3C)=O)C2)co1 CC1(CNC(C2CCC(OC(F)F)CC2)=O)CCCN(C(c2c[nH]c(=N)s2)=O)C1 c1(C(N2C(CN(C(C(CC)N(C)C)=O)C)CCC2)=O)c(OC)cc(OC)cc1F Cc1ncc(C(=O)NC2(C3CCCN3c3nc(C(C)(C)C)ns3)CC2)cn1 CC1CN(C(c2cscc2C#N)=O)CCC1C(=O)N(C1CC(C(=O)OC)C1)C S(=O)(=O)(c1ccc(Cl)c2nonc12)NC1C(C)CN(C(C2CC3CCC2C3)=O)C1 C1(NC(C2CC3CC3C2)=O)CCC2CN(C(c3ccc4cnsc4c3)=O)CC2C1 c1(C(=O)NC2CC(NC(C(CC)(F)F)=O)C(O)C2)ccc2cc(C#N)ccc2c1 N1(C(C2(C(=O)OCC)CCC2)=O)CC2CCC2(CCNC(c2cscn2)=O)C1 N1(C(CCC)=O)CCC2(CCCC2NC(=O)Cc2ccc3c(c2)CCC3)CC1 c1(OC)cc(N2CCC(C)C(NC(C3CC(C)CO3)=O)C2C)c(Cl)cc1[N+](=O)[O-] CC(C)C(C(=O)NCC1CCC1NC(C1CCC(F)(F)C1)=O)C1CCC1 C1(CNC(=O)CCc2ncccn2)CCC2(CCC2)CN1C(=O)C=CCF C(=O)(CC(C(F)F)n1ccnc1)NC(C)CNC(C1(c2ccnc(O)c2)CC1)=O Cn1ccc(=O)c(C(=O)NCCCOCCNC(=O)OC(C)(C)C)c1 C1(C(N(CC(C)NC(C(C=CCCC)O)=O)C)=O)CCc2nc(O)[nH]c2C1 C1(c2noc(CCC(=O)NC3(F)CCC(=O)CC3)n2)(NC(C)=O)CCC(C)(C)CC1 N1(C(C)C(N2CCCCC2)=O)CCN(C(=O)Cc2ccc(F)cc2)CC1=O N1(C(=O)CCN2CCCCC2)CC2=C(C1)CN(C(C13CCOC1CCOC3)=O)C2 C1(C(N(C(CC)CC)C)=O)C(C)CCN1C(=O)C(C)N(C)C(C)=O c1(NC(C23CC(NC(COc4cccc(C)n4)=O)(C2)C3)=O)cnc(C)c(Br)c1 c1(CC)cc(Cl)ccc1C(N1CCCC1CCNC(c1cnnn1C)=O)=O C1(C)(OC)CC2CC1CC2NCC1CC2(C1)NCCNCC2 N1(C(C2(NC(=O)CN3CC(C)(C)C3)C(C)CCC2)=O)CCCNC(=O)CC1 C1(CC)CCN(C(=O)CCC2CCC(NC(C3(OC)CC(C)(C)C3)=O)C2)CCO1 Cc1csc2nc(CC(=O)NCC3(O)CC(CNC(C4CCC5CC45)=O)C3)cn12 c1(NC2C(C)C2)nc2c(c(=NCC3Cc4ccccc43)[nH]1)CCC2 C1(CNC(CNC(C)=O)=O)CN(C(=O)COc2cncc(Cl)n2)C2CCCC2O1 N1(C(=O)NC2C=CC(NC(=O)OC(C)(C)C)C2)CCc2c(F)cc(F)cc21 c1(CC2C(CNC3(c4n(CC)nnn4)CCC3c3ccccc3)C2)ccc(C)cc1 Cc1cc(C)c(C(N2CC(C(=O)OCC(N3CCC(CC(C)C)C3)=O)C2)=O)s1 C(=O)(CC1=CCCCC1)NC(C(=O)NC(C1CCOCC1)C)c1cccs1 N1(CC)CCOCC1C(=O)NCCCN(C(=O)C(n1ccnc1C)C)C(C)C C1(CNC(=O)COC2CCCCC2)C(C2CC2)CCN1C(=O)C(F)C1CCC1 c1(C(N(CCN(C(=O)CCC2CCOCC2)C)C)=O)cn(C)c(=O)n1C c1(C(=O)NCC2(F)CCC(NC(C3(C)ON=C(C)C3)=O)C2)cccc(N)c1O C1(C(=O)NCCC(O)CNC(C2CC23CC3)=O)(OCC)CCCCCC1 CC(C)CCC(O)C(=O)N1CCC2(CC2C(=O)NCCOC(C)C)C1 c1(C(=O)OC)cc(NC(=O)NC2(CO)CC(C)C2)c(C)s1 c1cn(CCN(C)C)nn1.N1(C(C(C2CCC(=O)N2)C)=O)CCC(OCC(=O)O)C1 c1(C(N2CCC(CNC(C(CN(C)C)N(C)C)=O)C2)=O)c(F)cccc1[N+](=O)[O-] Cc1cc(C(N2CC(F)(C(=O)Nc3cccc(N4CCCC4)c3)C2)=O)cnc1O c1(C(=O)NCCCN(CCCNC(=O)COC2CC2)C)cnn2ccccc12 C#CCCCC(=O)N1CCC(NC(c2cn(-c3ncccn3)cn2)=O)C1C Cc1conc1C(=O)NC(CNC(c1cc(-c2ccccc2)[nH]n1)=O)CO c1(CC)nc(C)c(CCC(N2CC(CNC(C3(F)CC3)=O)CC2C)=O)c(O)n1 Cc1nnccc1C(=O)NC(C)C(C)C(=O)N(CC(C)C)CCO C1(C(N(CC=C)CCC)=O)CCCN(C(=O)CS(=O)CC)C1C c1(C(N2C(CNC(C(CCC)OC)=O)CC(O)C2)=O)sc2ccc(Cl)cc2c1C c1(C(N2C3CC(NC(C4CCNC4=O)=O)CC2CC3)=O)cc([N+](=O)[O-])ccc1O c1(C(=O)NCC(C)CNC(=O)CNC(=O)Cn2cncn2)cnc(N)c(CO)c1 N#Cc1cccc(C=CC(=O)NCc2ccc(Br)nc2)c1.C12CC1C(=O)N2 C=C(Cl)C(C)(C)C(=O)NC1CCC(NC(C2(F)CC=CC2)=O)C1 C=C(Cl)CCC(=O)NCC(O)CN(C(=O)C(CC1CCCC1)CC)C c1(C(N(CC(C)N(C(=O)C=CC(=O)N(C)C)C)C)=O)ccnc(N2CCCC2)c1 c1(CN2CC(CNC(=O)CSCC(F)(F)F)OCC2)cc(C(F)(F)F)cnc1O CC(C)C(CCC(=O)N1CCCC(F)C1)NC(c1cc(C(N)=O)[nH]n1)=O c1(C(=O)NCC(CCOC)NC(c2[nH]c(C3CC3)nc2C)=O)ccc(C)nn1 C(CC(=O)N1CCCC1(C)C(=O)OC)(C(F)(F)F)NC(C1(CC#C)CCC1)=O N(C(=NCC(C)C)N1CN(C)C(=O)C1C)Cc1c(C)ccc(F)c1 c1(OC2(C(F)(F)F)CCN(C(c3cc(OCC)sc3Cl)=O)C2)cccc(Cl)c1Cl O=C1NCCCC1C(N1CC2CC2(NC(c2cnc(-c3ccncc3)s2)=O)C1)=O CC(c1ccsc1)=CC(N1CCC1CNC(c1cn(C2CCC2O)nn1)=O)=O N1(Cc2cc(-c3c(OC)cccc3)no2)CC(=O)N(C2CC2C)C1=O c1(OC)cc(C(=O)NCC2CN(C(c3c[nH]c(C#N)c3)=O)C2)cnc1O C=CCCCC(=O)NC(C)CCCNC(C1(CC(F)F)CC1)=O c1(CC)cccc(F)c1C(N1CCC(C(F)(F)F)C(CNC(=O)C(C)O)C1)=O Cc1ccc(N)c(C)c1C(=O)N(CCCCNC(=O)C(C)C(F)(F)F)C CC1=C(C)CC(C(=O)NC2CCCCN(C(=O)CN(C)C(=O)C3CC3)C2)CC1 c1(C(=O)NC(C(=O)NCc2c(OC)cccc2)CC2CC2)cc(F)cc(F)c1 c1(CC(=O)NCC2CCN(C(C(CC)O)=O)CC2)cc(C(F)(F)F)cc(CC)c1 N1(C(C(COC(C)C)NC(C)=O)=O)CC2CC(C1)N(C(C1(C)CCCC1)=O)C2 CC(CC(F)F)C(=O)N1CCC(NC(=O)CCOc2ccccc2Cl)C1C N1(C(CCC=CCC=C)=O)CC(NC(c2conc2C2CCCO2)=O)C(C)(C)C1 C1(NC(C2CCCC(C)(C)C2)=O)CCN(c2nc(Cl)c(C#N)s2)CC12CCC2 CCC(CC)CCCC(=O)N1CC(NC(c2ncc(Br)cc2F)=O)C(O)C1 N1(C(COc2c(C)occc2=O)=O)CC23CCCCC2(C1)C(=O)NC3=O c1(C(C)OC(=O)C(F)CC2CCOC2)c(F)cccc1F c1(C(=O)NCCN(C(c2cnn(C(C)C)c2Br)=O)CC)cnc(NC)cn1 C1(CCOC)(C(N2CC(C)C(F)(F)C2)=O)CCN(C(c2c[nH]nc2OC)=O)CC1 c1(C(N2CCC(CC(=O)NC(C)C(F)(F)F)C2)=O)cc(Cl)nc(Cl)c1F c1(CC)[nH]nc(C(N2CCC(O)(CCNC(=O)CCCC3CC3)C2)=O)c1Br C(N=c1nc2sccc2c(N2CCCCC(C)(F)C2)[nH]1)c1nn(C)c(Br)n1 C1(C(NOCC=C(C)C)=O)CN(C(=O)CC23CCCC2C3)CC1C(C)C C(=O)(C(C(C)(C)C)NC(=O)CCCC)NCC1(CO)C(C=C)C1 N1(C(CC2(C(=O)OC)CCOCC2)=O)CCCC(CNC(c2ccns2)=O)CC1 C1(NC(=O)NCC(C)Cn2cccn2)CCCC1P(C)(C)=O CC1CN(C(C2C3CC4C(C3)C24)=O)CC2(CCN(c3nccnc3F)C2)O1 C1(CC)CN(C(=O)C(C)CC(=O)OC)CCN1C(c1cccc(C)c1F)=O c1(C(=O)NC2CCCN(C(CC(C)O)=O)CC2)cccc2c1OC(F)(F)O2 N1(C(C(CC)NC(N)=O)=O)CCC2(CCC(NC(=O)C(C)(C)S(C)(=O)=O)C2)C1 C=CCCC(O)CN(C(=O)CC1(OC)CN(C(c2c[nH]c(=NC)s2)=O)C1)C C1(NC(CCN(S(C)(=O)=O)C)=O)COCCN(C(c2cncnc2)=O)C1 CC1(C)CCN(C(=O)CSC(F)(F)F)C1C(=O)Nc1ccc(CO)nc1 CC(C)C(CNC(C1CN(C(C)C)C1)=O)C(=O)NCCCN1CCCC1C c1(C(=O)OC)nn(C)c2c1CCN(CCC1CCN(C)C1)C2 C1(N(C(C(C)OCCC=C)=O)C)CN(C(=O)Cc2c(C)noc2Cl)CC1(C)C C12(NC(CC)C(=O)NCC(C)C)CC(CN1C(=O)C(C)(C)COC1CCCC1)C2 CC12CC3CC(CC(C(N4CCCC(O)(CNC(C5CC5F)=O)CC4)=O)(C3)C1)C2 c1(C(N2C3C(NC(C(C)NS(C)(=O)=O)=O)CC(C3)C2)=O)ccc([N+](=O)[O-])cc1N c1(C(=O)NC(CCCNC(C=CC(=O)OCC)=O)C)c(C)cccc1Cl N1(C(c2ccc(C(=O)OC)c(Cl)c2)=O)CCCN(C(=O)CC2CC2)CC1C Cc1cnc2n1CCCC2C(=O)N(C)CC1(O)CCN(C(=O)CSC2CC2)C1 CC(CC(C)NC(=O)C=CCN1CCOCC1)NC(c1ccc(CO)o1)=O c1(CC)c(C(C)NC2CCCC(CCC(=O)OC)C2)oc2ccccc12 c1(C(C)=O)c(C)[nH]c(C(=O)NCC(C)NC(c2ncc(F)c(OC)n2)=O)c1C C1(CCNC(N2CCC(OCc3ccccc3)C2)=O)(CN)CCCC1O N1(C(C=COCC)=O)CCC2CC1CN(C(c1scnc1COC)=O)C2 CP(C)(=O)CCC(=O)N1CCC(C(=O)Nc2ccc(C3CC3)nc2)C1 Cn1c(=O)[nH]c(NCCNC(=O)Cc2cncnc2)c(C#N)c1=O C1(C(N(C)Cc2ccc(CNC(C(C)(C)OCC)=O)cc2)=O)CC(=O)N(OC)C1 c1(C(N2CCN(CC3NCCC34CC4(F)F)CC2)=O)ccc2c(c1)CCCO2 C1(C(=O)NCC2CN(C(c3cc(F)c[nH]3)=O)CC2(F)F)(OC)CCC(C)(C)CC1 C1(CC)(CC)CC(NC(=O)C2=NNC(=O)C2)CN1C(=O)C(C)Cc1ccncc1 N1(C(C)C(=O)NC2COCC2CNC(c2cc(Cl)cs2)=O)CCCCC1=O C(CC(CC)C(=O)N1CCC(CNC(=O)Cc2ccsc2)C1(C)C)=CC Nc1ccc(CCNC(=O)C(F)CC2CCOCC2)cc1 Cc1noc(N)c1C(=O)NC1CCN(C(c2coc(-c3ccccc3)c2)=O)CC1 C(CC1CCCC1)(C(=O)N1CC(OCCO)C1)NC(CN(C)C1CC1)=O N1(C(C2(CC)CCCNC2)=O)CCNC(=O)CC1c1ccccc1 Cc1cccc(C(C)C(=O)NCC2CCCN(Cc3ccc(C4CC4)cc3)C2)c1 N1(C(c2cc(COC)no2)=O)CC2(CCC(NC(C3CC4CC4C3)=O)CC2)C1 N1(C(C(C)OC)=O)CCN(C(=O)C(F)(F)CCn2ccnn2)CCC1C Cc1nc(C(=O)NC(C)CCNC(c2csc(Cl)n2)=O)c(C(F)(F)F)[nH]1 c1(NCC(C)CCO)cc(Br)ccc1S(=O)(=O)NCCCCCF c1(C(=O)NCC2(C)CCCN(C(=O)CC3C=CCC3)C2)cc(C#N)ccc1O N1(C(C(CO)NC(N)=O)=O)CCN(C(c2ccc(F)cc2)=O)CC12CCC2 c1(CNC(C(CN(C(c2n(CC)ccc2)=O)C)C)=O)ccc(C)nc1 c1(C(=O)NCC2C(CNC(Cc3cn(CC)nn3)=O)C2)ccc2nn[nH]c2c1 C1(CC(N2C(Cc3cn(CCC(C)C)nn3)CCCC2)=O)SC(=S)N(C)C1=O CC1(C(=O)NCc2ccc(C(=O)NCCc3cccnc3)s2)CCC2CC2C1 c1(OCCCCC)cc(C)ccc1CNc1ccc(NC(=O)C2CC2)cn1 C1(CNC(C(C)Nc2scc(C)n2)=O)CCCN(C(C2(CC(C)C)CCC2)=O)C1 C1(NC(CCc2c(C)ncs2)=O)CCN(C(C2(COC(C)C)CC2)=O)CC1C c1(CC)ccc(C(=O)NC(C)C(CO)NC(C2(C(F)F)CCC2)=O)c(C)n1 c1(-c2n(CC)c(COC)nn2)cn2cccc(N3CCC(N)CC3)c2n1 C#CCC(C(=O)NCC1CCOC1)NC(c1csc(CO)n1)=O Cc1nc2c(o1)CCN(C(=O)NCc1noc(C(N)=O)n1)C2 C1(NC(CCC(C)C(=O)N(C2CC2)NC(CC)(C)C)=O)(CO)CC2CCCC12 c1(C(=O)NC2(CCNC(C(C)n3ccnn3)=O)CCC2)ccc(N)c(F)c1F N1(C(Cc2c(C)cco2)=O)CCC2(C1)CN(C(C1CCCC1C1CC1)=O)CCO2 N1(C(CCC(C)(C)C)=O)CCCC2(CCN(CC(=O)Nc3cccc(Cl)c3)C2)C1 CCC(C)(CNC(c1ncoc1C1CC1)=O)NC(c1cc(C2CCC2)[nH]n1)=O C1(NC(c2cc(-c3cn(C)nc3)no2)=O)CCN(C(C2(C)CC=CC2)=O)CC1O C1(NC(C(N2CCOCC2)C)=O)CC2CC(C1)N(C(C1CC1C)=O)C2 C(=O)(C(C)CC(C)(C)C)NC1COCCN(c2nnc(CC)o2)C1 c1(CCN(C)C)nc(CCc2cnn(C)c2)n(-c2ccnc(Br)c2)n1 C1(O)(C(CNC(C2(COC)CC=CC2)=O)C)CCN(C(c2csc(C)n2)=O)C1 C1(C)(CNC(C(C)Cc2cccnc2)=O)CCN(C(C2CCCCS2)=O)C1 S(=O)(=O)(c1cccc(CBr)c1)N1CC2(C(C)CN(c3nccc(N(C)C)n3)C2)C1 N1(CCCCCCC)CC2CCC(NC(C3CCc4nnc(C)n4C3)=O)CC2C1 N1(C(CC(C)n2ccnc2)=O)CC2CC2(CNC(C2CC(O)CN2C)=O)C1 N1(C(CCCC=C)=O)CC(NC(C2(C)CC2C(=O)OC)=O)CC12CCOCC2 C1(C(N2C(COC)(CNC(=O)C3=NOCC3)CCC2)=O)CC2CCCCCC12 c1(CC(=O)NCCCC(C)NC(Cn2cc(C(=O)OC)nn2)=O)ccc(C)cc1F Cc1ccc(-c2noc(C3CCCCN3C3CN(C(=O)OC(C)(C)C)C3)n2)nc1Br C1(CC(=O)NCCCN2C(C)CCC2)CCN(C(c2scnc2Cl)=O)C1(C)C CC(C)CC(CNC(C1(C)CCC(=O)N1)=O)NC(=O)CCSCc1ccccn1 Cc1ccc(C=CC(=O)NC(C)C(C)NC(c2ccc(Br)s2)=O)cc1C C(C1CCOCC1)=CC(=O)N(C)CC1CCCN1C(C1CCC1(F)F)=O c1(CCC(=O)NCC2(O)CN(C(C3C(C)CC3)=O)C2)ccc(Br)c(Cl)c1 C(CCCCn1cc(C(C2CC2)N(C)C)nn1)NC(C1CC2CC2C1)=O c1(CNC(=O)C(N2CC(O)C(F)C2)CC2CCCO2)ccc(F)cc1 N1(C(C(C)N(CC)CC)=O)CCOCC(NC(=O)C(C2CC(F)(F)C2)OC)C1 C1(CC=C)(C(=O)NCc2cscn2)CN(C(c2nocc2C)=O)C1 c1(C(=O)NC(C(C)NC(=O)C(c2cccnc2)O)CO)cc(Cl)ccc1O N1(C(C)=O)CCCC(C(=O)NC(CNC(=O)C=CSc2ccccc2)CO)C1 N1(C(C(C)N2CCC2)=O)CC2CCN(C(C3CCOC3c3ccncc3)=O)CC12 c1(C(=O)NC(C(=O)N(C)CC2CCSC2)CCF)cc2occc2[nH]1 C1(COC)CC(CNC(c2csc(C)c2C)=O)N(C(=O)CCc2cncn2C)C1 c1(C(=O)NCC(C)CC2CC2)ccc(CNC(=O)CCOC2CC2)nc1 c1(C(N2CCC3C(NC(C(C)C(C)(C)C)=O)C32)=O)cccc2sncc12 C(CCCC(C)NC(C1(F)CCCCC1)=O)NC(CC=C(C)C)=O O=C(C1=C(Cl)CC1)NC1CCOC(C(=O)NCCC#CCO)C1 c1(C(N2CC(CNC(C(C3CCOCC3)C)=O)C(C)C2)=O)ccn(O)c(=O)c1 C=C=C(C)CC(=O)NCC1CCCCC1C(=O)Nc1cnc(C)nc1 C#Cc1ccnc(C(=O)NC2CN(C(=O)CNS(=O)(=O)N(C)C)C(C)(C)C2)c1 C1(NC(c2[nH]cc(C#N)c2)=O)CCC2CCN(C(c3ccc4cnnn4c3)=O)C12 c1(OC)nc(C)cc(=NC(COC(c2cccc(Cl)c2Cl)=O)C2CCC2)[nH]1 C1(C(C)=O)CC(C(=O)NC2CCN(C(=O)COCP(C)(C)=O)C2C)C1(C)C N1(C(C(=O)NC(c2ccncc2Cl)C)=O)CCC(C)C(N)C1 c1(C(N2CCC(F)(CNC(c3n(C)ccn3)=O)CC2)=O)ccc2ncncc2c1 c1(CC)nc(N2CCCCC(NC(=O)Cc3cccnc3C)C2)c(F)c(Cl)n1 C1(C(=O)NCC(CC)NC(C=CC(=O)OCC)=O)CCC(CN2CCOCC2)O1 N1(C(C(C)OCOC)=O)CCCN(CCNC(=O)CCc2csnn2)CC1 c1(SC)ccc(N2CC(C(=O)NC3CCN(C(=O)C=C4CCC4)C3)CC2=O)cc1 C1(C(N(C(C)CNC(=O)C(C)(C)n2cc(Br)cn2)C)=O)CC2CCC1C2 C12(NC(=O)C=Cc3ccsc3)CCC(CC1)N(C(=O)CCc1cncc(F)c1)C2 N1(C(CC2(OC)CC2)=O)CC(CNC(c2ccc(F)s2)=O)C(c2ccccc2)C1 C(N=c1[nH]nc(C(N)=O)s1)C1CN(C(CN2C(C)CCC2C)=O)C(C)C1 c1(C(=O)OC(c2cc(F)cc(F)c2)C(=O)OC)cc(C2CC2)ccc1I N1(C(CCC)=O)CC2(C1)CN(C(=O)CC1CC3CC3C1)C2 C1(C)(C(=O)NC)CCN(C(=O)N(C)CCF)CC1 C1(NC(=O)CSc2nnc(S)s2)CCCC(NC(=O)CN2CCCC2)C1 C1(C(=O)NC(C2CCOC2)CNC(=O)C(F)=CCCF)(NC(C)=O)CCCC1 C(=O)(C(CC(C)C)C(C)C)NCC1C(NC(C(C)N(C(C)=O)C)=O)C1 C(=O)(CCCCCCCCCO)N(C(C)CN(C(=O)C(Cl)=CCl)C)C c1(C(=O)NC2CN(C(C=CC=CCC)=O)CC2O)ccc2ccc(Cl)cc2n1 N1(C(c2c(OC(C)C)nccc2)=O)CCCN(C(=O)C(C)n2cncn2)CCC1 c1(C(C)C)ccc(F)cc1CN1CCNCC1NC(=O)NCCc1ccccc1 c1(CCC(=O)NC2(C)CCN(C(C(C=C=C)C)=O)C2)c(C)nc(O)nc1C C1(CNC(CCOC)=O)(NC(=O)CN(S(C)(=O)=O)C)CCCCC1C.C(C(C)C)N CCCC(C(=O)NC(CO)C(C)NC(c1ncn(-c2ccccc2)n1)=O)OC N1(C(c2cn(C(C)C)nc2)=O)CCC(C(=O)NCCn2ccnn2)C1C c1(C(=O)NCC2CCC(NC(C3(C4CCC4)CCC3)=O)C2)cc2c[nH]cnc-2n1 N1(C(c2c(CCC)nns2)=O)CCC2CN(C(C3CCSC3)=O)CC12 N1(CC)C2CCC1CN(c1ncnc(N3CCN(C4CCCC4)C(C)C3)c1C)C2 c1(SCC(=O)NC2(C)CC(NC(CCSC)=O)C2)nn(C)c(=O)n(C)c1=O N1(C(c2nnn3c2CCC3)=O)CC2CCN(C(C3CCCCC3)=O)CC2C1 c1(C(c2n(CCSC)nnn2)NCCc2nc(C)cs2)cncc2ccccc12 C1(NC(C(C)(C)C2CCOC2)=O)CCCCCC1NC(C1CS(=O)(=O)C1)=O C(=O)(C1=CCCOCC1)N1CC(C)(C)C(NC(=O)Cc2ccc(Br)s2)C1 Cc1nc2sccn2c1C(=O)NC(C1(O)CN(C(=O)Cc2c(C)noc2C)C1)C CCC(CC)CCC(=O)NCc1ccc(C(N2CCc3ccsc3C2)=O)nc1 C1(C(=O)NCC(C2CC2)NC(c2ccc(CO)o2)=O)CC2CCC1C2 c1(C(N2CCC(CCNC(c3nc(C4CC4)cs3)=O)C2)=O)ccc(O)cc1 C1(N(S(=O)(=O)Cc2ccccc2)C(C)=O)CC2(C1)CN(Cc1ccc(O)nc1)C2 Cc1ccc([N+](=O)[O-])c(-n2cc(CNC(c3ccccc3)C)nn2)c1 N1(C(C=CC)=O)CCCC2CN(c3ncc(C#N)cc3Cl)CCC12 C1(NC(c2cnc(Cl)s2)=O)(CF)CCN(C(=O)Cc2cccc(F)c2)C1 C(=O)(CC1OCc2ccccc21)NCC(C)(C1CC1)NC(=O)C1=CCS(=O)(=O)C1 C#Cc1ccc(C(=O)NC2CN(C(c3ccc(SC)s3)=O)CCC2C)nc1 C1(NC(c2ccc(N(C(C)C)CC)cc2)=O)CCOC(C)(CC(=O)NC)C1 N1(C(c2scc(C#N)c2)=O)CC2CC1CN2C(c1cn(CC(F)(F)F)cn1)=O C1(CNC(C=COCC)=O)CCCC(NC(c2cc(Br)oc2C)=O)C1 c1cnc2[nH]cc(CN=c3ccn(-c4ccnc(C(F)(F)F)c4)[nH]3)c2c1 C1(N(C(C2(NC(C)C)CC2)=O)C)CCCN(C(C2CCNC2=O)=O)CC1 CC#CCCCC(=O)NCC1(OC)CCN(C(=O)CC(=O)OCC)C1 N1(C(C2CC(C)CN(C(=O)C3=CC(C)(C)C3)C2)=O)C2CCCC1COC2 C1(C2CC(OC)C2)NC(=O)N(CCc2ccccc2)C2=C1C(=O)N(OC)CC2 N1(C(C2C(C)(C)CCN(C(=O)CC3=CCOCC3)C2)=O)CCC2CCNC(=O)C12 c1(C(=O)NC(CNC(C(COC)(C)OC)=O)(C)C)ccc(F)c(OC)c1 Cc1ccc(CNC(C)(C(C)C)c2nnnn2C)c(=O)n1C C1(CNC(c2c(C)ccn2C)=O)C(O)C(O)CN1C(c1cnc(CC(C)C)s1)=O c1(CN2CCN(C(C(CC)C)=O)CC2)nc2ccccc2n1Nc1ccccc1 O=C(CCCC1CCCO1)NC(c1ccccc1)C(=O)NC1C=CCC1 C12(C(N3C(C4CCN(C(c5nncc(C)c5)=O)C4)CCC3)=O)CCC(F)(CC1)CC2 C1(C2CCOCC2)(C(N2C(CN(C(C(C)C3CCC3)=O)C)CCC2)=O)CC1 N1(C(C(CC)n2nccc2C)=O)CC(C)N(C(C2CCCCC2(C)C)=O)CC1C N1(C(C(C)(C)SC)=O)CC2(NC(c3cc(N)cnc3Cl)=O)CCC1CC2 CC(CC(=O)NC1CC(O)(CNC(c2cc(C(N)=O)co2)=O)C1)N1CCCC1=O C1(C)(C(N(CCN(C)C(c2ccnn2C2CC2(F)F)=O)C)=O)CCNC1=O CCC(COC)C(=O)NCCCC(=O)Nc1cnn(C(C)(C)C)c1 O=NN1CCCC1C(=O)NCC1CN(C(=O)CCc2cnc(C3CC3)o2)CCO1 N1(C(C2N(CC)CC2)=O)CC2CC1C2CNC(=O)CCC(C)N(C)C c1(C(N2CC(N3CCN(C(C#CC(C)(C)C)=O)CC3)C2)=O)cc2sccc2n1C c1(C(C)C(=O)NCCOC2(C)CC2)ccccc1S(N)(=O)=O C1(CCC)(NC(c2cn(C)cc2C)=O)CCN(C(c2cnnn2CC)=O)CC1 C1(OC)CCN(C(=O)CSCCNC(c2ccnc(CO)c2)=O)CC1C C1(C(=O)NCC(C2CCC2)NC(C(C)(C)N2CCCCC2)=O)CCC2(CC2)C1 N1(C(CCN(CC(F)(F)F)C)=O)CCC(CO)(NC(c2cnc(Cl)[nH]2)=O)C1 c1(C(=O)NC2C(C(N3CC(C)(C)OCC3)=O)CCC=C2)ccc2[nH]ccc2c1 CC1CC(C(=O)N(C)CCOCCC(=O)NC2CC(C)(C)OC2=O)=NO1 c1(CC(=O)O)coc2c1CN(C(C1CCC(Oc3ccncc3)C1)=O)C2 c1(C(N2C3CN(C(c4c(CC)nns4)=O)C(C3)C2)=O)nnc2ccccc2n1 C1(C)(NC(c2c(C)c(C(=O)OC(C)(C)C)on2)=O)CC2(C1)CC2(F)F n1(CC(=O)N(C)CC2N(C(C3C(C)=C3)=O)CCC2)ccc2c(N)cccc12 Cc1ncc(Br)c(C(=O)NCCCN2CCN(C(C3CCCCCC3)=O)CC2)n1 C1(NC(CCc2c(C)nccc2)=O)CC(C(=O)O)C12CCC2 c1(NC(N(CCC)C(c2ccccc2)C)=O)c(Cl)cc(Cl)nc1C c1(OC)ccc(C(=O)N(CC(Cc2ccccc2)NC(C23CCC2C3)=O)C)nn1 C(=O)(CCCC(=O)NCC1CN(C)CCN1C(C1CC1[N+](=O)[O-])=O)OC c1(C(=O)OC)cc(NCCN(C)Cc2ncc[nH]2)cc(Br)c1[N+](=O)[O-] c1(SC)cc(C(=O)NCc2ccccc2CNC(=O)CC(F)(F)Cl)c(C)o1 NC(=O)CCC(=O)NCC(C1CCCC1)NC(C1C2CN(CC(F)(F)F)CC12)=O c1(C(N2CCN(C(c3[nH]cc(C)c3)=O)CC2CCO)=O)ccc2nc(O)sc2c1 C1(NC(CSCCC)=O)CC(c2ccccc2)(NC(C2(c3cccs3)CC2)=O)C1 c1(C(N2CC(OC)C(NC(=O)C(F)C3CCCC3)C2)=O)nnn2c1CCCC2 c1(CC(=O)NC(CNC(c2cnc(OCC)s2)=O)(C)C2CC2)cc(O)nc(O)n1 C(=O)(C(F)C(C)C)OCc1nnc(CC)s1 C(C(=O)N(C)CCN(C(=O)C(C)OCC1CCCO1)C)(SC)SC C1(NC(Cc2c(C)cco2)=O)CN(C(=O)C2=C(Cl)CCOC2)C2(CCCCC2)C1 C1(C)(NC(c2nccc(CC)c2)=O)CCCCC1C(=O)Nc1cnn(CCOC)c1 N1(C(C(C(C)(C)O)F)=O)CCC2CC(NC(c3ccn(CCF)n3)=O)CCC2C1 N1(C(c2cn(CCOC)nc2)=O)CC2(C)CN(Cc3noc(C)n3)CC2(C)C1.C1CC1 c1(C(=O)NC(C)CNC(=O)C=Cc2ccco2)cc(Cl)c2n[nH]cc2c1 c1(C(N2CC(CNC(c3cc(OC)cc(OC)c3)=O)C2)=O)cc2sc(F)cc2[nH]1 CC(CC(=O)NC(C1CCN(C(c2scnc2C(C)(C)C)=O)CC1)C)P(C)(C)=O CCC(CC(C)C)C(=O)N1CCC(C2CCCN2C(=O)CC2(CC)CCC2)CC1 C12(NC(CN)=O)CCCCC1N(C(=O)C(C)CCOC)CCC2.N(CCO)(CC)CC Cn1cnc(C=C(F)C(N2CCCC2CC2C(C)(C)C2(C)C)=O)c1 c1(CNC(C2CCCN(C(=O)Cc3cccs3)CC2)=O)cccc2occc12 C12(C(CNC(Cn3ncc(C)c3)=O)NC(=O)CC3CC3(Cl)Cl)CCC(CC1)C2 Cc1nn(CC(C)C)c(C)c1CN1CCN(C(=O)NC(C)(C)C)CC1C(F)F c1(C(c2nnnn2C2CCCC2)NC(CCCC)C)cc([N+](=O)[O-])ccc1Cl CC1CC(C(=O)N2CCC(C)(C)C2C(=O)N(C)CCN2CCCC2=O)=NO1 CCCC(C)(O)CC(=O)N1CCOC(C(=O)NCCc2ocnc2CO)C1 c1(NC)cnncc1C(=O)NC1CC1C(=O)NCCSc1ccccc1 C12(C(=O)NC(c3ccc(CNC(CCSC)=O)cc3)C)CCC(O)(CC1)CC2 N1(C(C(CC=C)CC)=O)CC2CCN(C(c3nonc3CC)=O)C2C1C Cc1nocc1C(=O)OCC(=O)NC(C(C)(C)C)c1cccs1 C(=O)(CC(C)CC(C)C)NCC1(OC)CN(C(c2nnsc2N)=O)C1 c1(C(=O)NC2C(NC(c3cnn(CC)c3C)=O)CCCC2)ccc(C#N)cc1C c1(C(N(CCCNC(CCNC(C)=O)=O)C(C)C)=O)cc2c[nH]nc2s1 C1(C(=O)NC2(C(=O)NC3C(C)CCC3C)CC2(C)C)CC(=O)OC1(C)C CC1CN(C(=O)CN(C)CCO)CCCN1C(c1ccc(OC(F)F)nc1)=O c1(OC)cc(C(=O)Nc2cccc(F)c2Cl)c(NCc2cc(Cl)cnc2C)cn1 N1(c2ccnc(NCCCc3c(OC)cccc3)n2)CC2(C1)CN(C)CCO2 CC1CC(C(=O)NC(C)(C)CF)CN(C(=O)Cc2ccnc(O)c2)C1 CC1(C)CCN(C(c2nc(Cl)cs2)=O)C1C(=O)NC1CCCC1N=[N+]=[N-] Cc1ccc(N(S(=O)(=O)C(C)C)C2CC3CC2CN3)c(C)c1 Cn1cc(C=CC(=O)NC2(C)CC(NC(c3cn(CC(F)(F)F)cn3)=O)C2)cn1 N1(C(C2N(C(CC)=O)CSC2)=O)CCCC(NC(=O)C=C(C)C2CC2)C1 C(=O)(C(C(C)CC1CC(F)(F)C1)N1CCN(C)C(c2ccc(F)cc2)C1)NCC C=CC(C)(CC)C(=O)N1CC(CNC(C2CCC3(CC2)CC3)=O)C(F)(F)C1 C=CC(CC)CC(=O)N1CCCC(NC(=O)COc2cccc(F)n2)C1C CC(O)(Cc1ccccc1)C(=O)NCCCN(C(=O)CN1CCOCC1)C1CC1 N1(C(c2cccc(SC)c2)=O)CCN(C(=O)C(C)(C)N(C)C)CC1CC(F)(F)F C1(OC)CN(C(=O)C(C)(CSC)NC(C2CC(SC)C2)=O)CC12CC2 Cc1cc(Cl)c(C)c(C(N2CC(CO)(NC(=O)CCC=CC(C)C)C2)=O)c1N CC1(C)CN(C(C2CCNC(=O)CC2)C2CC2)CC1c1cc[nH]n1 c1(CNC(C2C(NC(c3ccoc3)=O)C2)=O)ccc(Br)nc1 c1(NCC2(SC)CCCCC2)nc[nH]c(=NCC2(F)COCCOC2)c1C Cc1cn2c(C(=O)NCC3CCN(C(C4CCCS(=O)(=O)C4)=O)C3)c(C)nc2s1 CC(=O)CCCC(C)C(=O)N(CCC(=O)NCCOC1CC1)C NS(=O)(=O)c1ccc(F)c(NC(c2ccccc2CF)=O)c1 C=C(Cl)CCC(=O)NC1C2CC(NC(c3cn(CCC)nn3)=O)CC12 C(=O)(CCC(CF)CF)N1C2(C(N3C(CC)CC(O)C3)=O)CC2CC1 C#Cc1cccc(C(N2CC3CC2CCN3C(=O)C=Cc2sccc2C)=O)c1Cl NC12CCOCC1CN(C(=O)C(=O)NCC(N1CCOCC1)=O)C2 C1(C)(NC(c2nc(COC)sc2)=O)CCN(C(=O)C(C)C#N)C1 N1(C(Cc2ccc(C)o2)=O)CC(CCNC(=O)CC2(C#N)CC2)OC(C)C1 C12(CNC(c3ccc(CC)cc3)=O)CC(NC(c3ncccc3Br)=O)(CCO1)C2 C1(NC(C2(N(C)C)CCC2)=O)C2CC1N(C(C1CC1c1cccc(Cl)c1)=O)C2 CCC(C)C(O)CC(=O)N1CCCC(C)(C(=O)NC2CCN(C)C2)C1 c1(C(N2C(CNC(C3N(C(C)=O)CCCC3)=O)C=CC2)=O)nccc2n[nH]cc12 N1(C(C(C)=CC2CC2)=O)CCC(F)CC1C(=O)N(C1CC(C)C1)C N1(CC(C)NC(C(COC)O)=O)CCN(C(=O)CC2CCC(=O)N2)CC1 S(=O)(=O)(c1cccnc1NCc1csc(O)n1)NC1C(CCCC)CCC1 C(=O)(C1=CC2(CCOC2)C1)NC1CN(C(Cc2nc(CC)sc2)=O)CC1C1CC1 Cc1ccc(C2(C(=O)NCC3CC(C)N(C(C45CC(C4)C5)=O)C3)CC2)cc1 CCCCCCCC(F)C(=O)N1CCN(C(C2COc3ccccc3C2)=O)C(C)C1 C1(NC(c2nc(C)oc2)=O)CN(C(c2cnsc2)=O)CCC1C C(=O)(C(C)(CC)C(N)=O)NCC1N(C(CS(=O)(=O)N(CC)CC)=O)CCN(C)C1 C(C)(C)(C(C)CC(=O)N1CCSCC1)NC(c1nc(C)oc1)=O C1(CNC(CC=C)=O)CC(C)CN(C(=O)CSCCC(C)C)C1 c1(C(N2CC=C(CCNC(CS(=O)(=O)NC)=O)CC2)=O)ccc2cn(C)nc2c1 C(CC(C)(C)C)(C(=O)Nc1cnc(F)c(C)c1)NC(CCNC(=O)NC)=O c1(CC(N2CCC(CNC(C(F)=CC)=O)C23CC3)=O)ccc2nc[nH]c2c1 c1(N(CCCC(F)(F)F)C)cccc(S(=O)(=O)NCC2CCS(=O)(=O)C(C)C2)n1 CC(C)CCC(=O)NC(C)(C)CNC(=O)Cc1cn(C)nc1C(F)(F)F c1(OC)ccc(CC(C)C(=O)NCCC(C)NC(C2CCCC2)=O)cc1OC C12(NC(C3C(C)CCO3)=O)CC1CN(C(=O)Cc1ccccc1OC(F)F)C2 C(=O)(CCC(=O)NN(C)C)N(CCCCCCNC(CC(C(C)C)C)=O)C C1(C(N2C(C)(C(=O)OC)CC2)=O)CC(NC(=O)CNC(=O)CC(C)C)C1(C)C CN1CCC(C(=O)NCCC2(O)CN(C(c3[nH]ccc3-c3ccccc3)=O)C2)C1 c1(C(N)=O)ccc(CCC(N2CCCC2c2cccc(Br)c2)=O)cc1 C1(NC(C(C)NC(C)(C)C)=O)CC(CNC(c2cc(=O)n(C)o2)=O)CC1O c1(CC)c(C(=O)NC2CCN(C(C34CCCC3CC4)=O)CC2)oc2ccccc12 N1(C(c2c(CCOCCCC)ocn2)=O)CCC(NC(=O)C2=CCSC2)CC1C Cc1nc(NC2(C3CNC3)CC2)ncc1[N+](=O)[O-] C=C(Cl)CC(C(=O)NCCCCN(C)C1CC1)NC(=O)CC1CCC(C)(C)O1 C(=O)(CS(=O)(=O)C(C)(C)C)NCC1CCC(NC(CCSCCC)=O)CC1 c1(CN(C2CC2C2CC2)C)ccc(NC(=O)C(F)=CC2CC2)cn1 C12(C(=O)OC(C)(C)C)CCC(CNC(=O)NCCCC3CCCO3)(CC1)O2 c1(NC(=O)NC(CCC=C)CO)cc(NC(C)=O)ccc1C C(=O)(C1CCc2nnc(C)n21)NCCC1N(C(Cc2cc(C)no2)=O)CCSC1 c1(CC)cccc(NC(c2ccc(NC(=O)C(=O)N(C)C(C)C)nc2)=O)c1C C(=O)(C(F)(F)C(F)(F)C(F)F)NCC(CNC(CCC(CC)OC)=O)C N1(Cc2cc(C(=O)OC)n[nH]2)CCC2C(C1)NC(=O)CCN2C C(CNC(C1COC(C)(C)C1)=O)(CC)(CC)NC(c1nc(CC)oc1)=O C1(CC(=O)OC)COC(C)(C)CN1C(=O)Nc1ccc(-n2cnnn2)c(C)c1 c1(C(=O)NC2C(NC(=O)CCC3CCCC3)C2)cc2c(s1)CCCCCC2 C#Cc1cccc(CC(=O)NC2CC3C(NC(C4(OC(C)=O)CC4)=O)C3C2)c1 C(=O)(CC(C)C(C)(C)C)NCC(C)(CC(C)C)NC(c1c(SC)scc1)=O C(=O)(C1=CCc2ccccc21)NC1C(C)CN(C(c2ccn(C(F)F)n2)=O)CC1 N1(C(CCC)=O)CCCC(C(N2CCCC2CN(C)C)=O)C1CC C=CC(C)CC(=O)NC(CCOC)C(=O)NC1(C(=O)NCC)CC1 c1(C(C)NC(C(=O)Nc2ccc(OC)c(F)n2)=O)c(O)cc(F)cc1F C1(C(N2CC(OCCOC)C2)=O)CC12CCN(C(c1ccsc1C)=O)CC2 C1(C(=O)NC(C)CC(N)=O)CCC(C2CC2)N1C(=O)C(C)C1(O)CCC1 CC1(C)C(CC(N2CC(CCCCNC(c3ncsc3C3CC3)=O)C2)=O)C1(C)C CC1CC(C(=O)NC2CC3CN(c4ccnc(C#N)n4)CC23)=NO1 C12(C(=O)NCC(C3CCC3)NC(C3(SC)CC3)=O)CC(C)(C1)OC21CCOCC1 N12CC(CCC1C)NC(=O)c1ccc(cc1)C2C.Cc1ccccc1CO N1(C(C2(CSC)CC2)=O)CCC(F)(C(=O)NC2(CF)CC2)C1 C12(CCN(C(=O)C(C)SC(C)C)C1)C(=O)N2.C1(CCOC)CCCC1(C)C c1(CC(=O)NC2CN(C(Cn3ncc(C)c3)=O)C2)ccc2ncnn2c1 N1(C(CC=C(C)C)=O)CCC(C)(CNC(c2c(C)nsc2Br)=O)C1 c1(C(=O)NCC2CCCC(NC(C3(C)CCCC3)=O)C2)cc(O)ccc1Cl N1(C(c2ccccc2)C)CCC(C)(Cc2cccc(Br)c2)C1.c12cn(nn1)C2 CC(C)(C(=O)NC1CCCC(CNC(c2c[nH]nc2Cl)=O)C1)C(F)F C(=O)(C(C)(C)CCCO)NC1(CC=C)CN(C(c2coc(C(F)F)c2)=O)C1 c1(OC)cc(C(=O)NCC(C)CNC(C2(c3cnccc3C)CC2)=O)ccc1C c1(C(=O)NCC2N(C(C(C)CSC(F)(F)F)=O)CC2)ccc(-c2ncc[nH]2)nc1 C1(C(N2C(CNC(C3C(C4C(C)C4)C3)=O)CC2)=O)CNC(=O)CC12CCOC2 c1(SC)ncc(N)c(C(=O)NCCCCNC(c2cc(F)cnc2O)=O)n1 C(=O)(N=c1cc(C2CC2)[nH][nH]1)c1c(NC(C2CCC3(CC2)CC3)=O)cncc1 CC(C)CC(=O)C(=O)NCCC1(C(N2CCC(C(C)C)C2)=O)CCC1 C1(NC(=O)NCC2CN(C(=O)OC)C2)CCCC(c2ccccc2)C1 C(N=c1ccnc(CO)[nH]1)C12OCC(CNC(C3(c4ncccc4F)CC3)=O)(C1)C2 C(=O)(CC(C)(O)C=C)NC1CN(C(Cn2ncc(C#C)c2)=O)C(CO)C1 c1(C(=O)NCC(CO)NC(c2ccccc2F)=O)ccc(Br)c(F)c1F c1(OCCC)ccc(N(C(c2ccnc(F)c2)C(=O)NC)C)cc1 O=C(CCS(=O)(=O)C(F)(F)F)NC1CC(CNC(=O)CCC(F)(F)F)C(O)C1 C1(C(=O)OC)CCC2(CC2)N1C(=O)C(=O)NCC1CCC12CCC2 N1(C(C(C(C)(C)C)C2CC2)=O)C2CCC1CN(C(=O)C#CC1CCOC1)C2 Cc1cc(C(=O)NC2(CNC(=O)C(C)NC(=O)C(C)(C)C)CCC2)c(C)n1C1CC1 C1(OC)(CNC(=O)C=CCCc2ccccc2)CCN(C(C2(C)CC2C)=O)C1 C1(C(N2CC(C(=O)NCC(=O)N(C)CC)(COC)C2)=O)CC2CC(=O)C1O2 c1(CC)cc(C(=O)NCCc2ocnc2CNC(c2nnsc2SC)=O)on1 c1(C(=O)NCCC(C)NC(=O)COC2CC2)ccc(Cc2cccs2)cc1 c1(NC(CCCCC)c2ccccc2)nc2ccccc2nc1NCC1CC1 C1(C(N2CC(OC)C(NC(c3cnc(SC)s3)=O)C2)=O)CC(S(C)(=O)=O)C1 C1(NC(C(CC2CCC2)NC(C)=O)=O)CCCCN(C(c2ccncc2N)=O)C1 c1(OCC)cccc(NC(C2CC2C(=O)NC2CC(F)CN2C(C)=O)=O)c1 c1(N2CC3CN(C(C(c4cccc(OC)c4)O)=O)CC32)ncnc2c1cnn2C c1(C(=O)NC2CN(C(c3c(SC)csc3)=O)CC2(C)C)cccn2nncc12 C1(C(=O)NCCc2ncn(C)n2)CC(NC(=O)CN2CCC(=O)CC2)CCO1 c1(C(=O)NC(CN(C(=O)CC2CC3CC3C2)C)(C)C)ccc(S(N)(=O)=O)s1 C1(NC(CSc2ccc(OC)cc2)=O)CN(C(=O)CC2CCN(C)C2)CCC1F Cc1ccc(CC(=O)NC2CC2CNC(c2cn(C(C)(C)C)nc2C)=O)c(C)c1 c1(N(CCCC)C)nc(-c2ccccc2)nc(=NCCCOCCO)[nH]1 C1(c2nnnn2C2(C)CC2)(NC(c2cccc(NC)c2)=O)CCOCCC1C c1(CN(C(C(=O)NC2CCCCC2)c2ccon2)C)ccccc1 CC(C(=O)NC1(C)CC(NC(=O)CCOc2ccc(F)c(F)c2)C1)S(N)(=O)=O CCCC(C)(CC)C(=O)NCC(C)(C)CNC(c1ccc(=O)n(CC(C)O)c1)=O N1(CC(=O)NC(CCNC(C2(C(CC)(F)F)CC2)=O)(C)C)CCc2ccccc21 C#Cc1cncc(C(=O)NCC2CCC(C(=O)NC(c3nc(C)cs3)C)O2)c1 C1(CNC(CC(C)SC)=O)CCN(C(c2cc(Cl)nn2C)=O)C1(C)C N1(C(C(C)(F)F)=O)CCC2CN(C(c3ccc(F)c(Br)c3F)=O)CC12 c1(C(C)=O)ccc(CC(=O)NC2CCC2CNC(=O)C(=O)N(C)C)cc1 n1(CC)cnc2[nH]c(=NCc3cc(Cl)no3)nc(NCc3cc(OC)ccn3)c12 C1(NC(C(C)NC(N)=O)=O)CCC(CNC(=O)CCCn2ccnn2)CC1 C(C)(CN=c1nc(C2CCCCC2)nc[nH]1)N(C(C(C)CN(C)C)=O)C c1(C(=O)NC2C(NC(C=CCC)=O)CCC2)ccc(C)c(C(=O)OC)c1 c1(C(C)C)n[nH]cc1C(=O)NC1COCC1C(=O)N(C)Cc1ccon1 CCC(CC(F)F)C(=O)N1CCOCC(NC(C2(C)CCC2)=O)C1 C1(NC(c2c(C)nc(CO)s2)=O)COC2(CCN(C(c3ncn(C)c3C)=O)C2)C1 C(CCCCCCCC1CC1)(N(C)Cc1ccc(F)cc1)C1CC1 C1(C)(NC(c2nc(C(C)C)oc2)=O)CCN(C(c2nc(Br)c[nH]2)=O)C1 N1(CC)CCN(CCC(=O)NCC#CCNC(=O)CC2CCCO2)CC1 C(C)(C)(C(=O)NCCCCCN(C)C(C1CC(F)(CO)C1)=O)OCC C1(CNC(C2CN(C(C)=O)C2)=O)CC(C)CCN1C(=O)C(O)C1=CCCC1 c1(NC(c2ccc(NS(=O)(=O)CCCl)cn2)=O)cc(Cl)nc(Cl)c1 c1(C(N2CCCCC(CNC(=O)Cn3cncn3)C2)=O)ccn2c(O)nnc2c1 C1(C(N(CCCC)CC)=O)(NC(c2cncn2C)=O)CC(O)C1 CCC(C)C(CC(=O)N(C)C(C1CCCC1)C)NC(C1CCC(C)=C(C)C1)=O C1(C)(C(=O)NC2C(NC(C3(CN(C)C)CC3)=O)CCC2)CC2(C1)CC(F)(F)C2 c1(CC(N2CC3C(C(=O)NC4CCOCC4)C3C2)=O)ccc(Br)cc1I N1(C(C(C)NS(CC)(=O)=O)=O)CCCC(NC(=O)CC2(O)CCOCC2)CC1 CCCCC(CNC(c1sc(CC)nc1C)=O)NC(=O)Cc1cccc(OC)c1 C1(NC(CC2CC(C)C2)=O)CN(C(C2CC(C)CC(=O)N2)=O)C(C)(C)C1 Cc1cc(C(=O)NCC2(NC(=O)CSc3cn[nH]c3)CC2)c(C)n1C(C)C c1(OCC)ncccc1C(N(C1CC(NC(=O)CCCCOC(C)=O)C1)C)=O.OCC N1(C(=O)NC2C=CCN(C(C(C=C)O)=O)C2)CCC(C)(C)CC1C(=O)OC(C)(C)C C1(C(C)CO)CCN(C(C2C3CN(Cc4cc(Cl)ccn4)CC23)=O)CC1 C1(C(CNC(C=C(CCC)C)=O)(C)C)CCN(C(=O)CCC(C)SC)CC1 C1(C(C)(C)C)CN(C(c2ccc(=O)n(C3CC3)c2)=O)CCN1C(C1CCOC1)=O C#CCC(O)C(=O)N(CCCOCCNC(c1n[nH]c(C)c1Br)=O)C N1(CCCC)CCCCC1C(=O)N(C(C)C)CC1CCCCO1 C1(C(=O)NCC(C)(C)NC(C2(C)C(C(=O)OC)C2)=O)(N(C)C)CCCC1 Cc1cc(C(N2CC(NC(c3c(C)ncn3C)=O)CC(C)C2)=O)ncc1N N1(C(c2cc(C)n(C)n2)=O)C2CCCC1CN(C(=O)C(F)CC1CCOC1)C2 c1(C(=O)NC2(COC)CN(C(C3CCCS3)=O)C2)ccc2nnc(S)n2c1 C(CO)(C(=O)NCC1CCCN1C(C1CC1(C)C)=O)NC(=O)OC(C)(C)C N1(C(c2c(CCC)[nH]cc2)=O)CCC(C(=O)NCCc2ncccn2)C(O)C1 c1(C(N2CCC2CNC(C2C(=O)NCCC2C)=O)C)cccc2ccccc12 N1(C(c2nccc(N)c2)=O)CCC2(CC1)CC2NC(C1CC12CCCCC2)=O C#CCC(C)(CC)C(=O)NCC(C)(C)C#CC(=O)Nc1ccc(F)nc1 CC1SCCCC1C(=O)NC(C)(C)CN(C)C(c1cc(-c2cnn(C)c2)on1)=O c1(C(N2CC3CCN(C(=O)CC4COCC4O)CC32)=O)cccc2nc(Cl)cn12 C(=O)(CC(C)(C)CC(=O)OC)N1C2C(NC(C(CCC)NC(C)=O)=O)CC(CC2)C1 c1(C(N2CC3C(N(C(C=CC=CC)=O)C)C3C2)=O)cc(O)ccc1CC C1(CN2CCC(c3c(F)ccc(Br)c3)CC2)CC2(CCN1)CCOCC2 CCCCS(=O)(=O)CC(=O)NC1CCCC(NC(c2nc(C)c(N)cc2C)=O)C1 C1(CNC(CC=CCC)=O)CN(C(=O)COc2cc(C)on2)CC1(F)F C(C1(C)COc2ccccc21)CNC(N(c1ccc(C(F)(F)F)cc1)C)=O C(c1ccncc1)=CC(N1CC2C(C(=O)OC(N3CCC3)=O)C2C1)=O C1(CNC(CCCNC(C)=O)=O)CCN(C(c2cc(C(F)F)nn2C)=O)CC1C C(=O)(C1CCc2nccn21)N1CCN(C(C2(C)CSC2)=O)CC1CO C#CCC(C)(CC)C(=O)NC1CCOCC1NC(c1cc(C)no1)=O C(=O)(CC(C)(C)CC=C)NCC1(C(=O)NCC=C)CC12CCC2 c1(C(=O)NC2CC(CNC(COc3cccc(C)c3)=O)C2)cn(C)c(=O)nc1O C(=O)(CCC1(NC(c2ccon2)=O)CCC1)NC(C1(C)CC1)CO C1(NC(COC(C)=O)=O)CCCC12CCN(C(c1cccc3nsnc13)=O)CC2 N1(Cc2c(C)ccnc2)CC2CCC(C1)C2NC(=O)C(N)=O C(=O)(C1=NNC(=O)CC1)N1CC(C2OCCN(C(Cc3nn(C)c(Cl)c3)=O)C2)C1 c1(C(N2CC(C(=O)NCC3CC34CCC4)(COC)C2)=O)cc(OC)ncn1 Cc1ccccc1C(C)CC(=O)NC1(CN(C(=O)C(C(C)C)N(C)C)C)CC1 N1(C(C2C3(CC(NC(=O)CCn4cccc4)C3)C2)=O)CCC(=C(F)F)CC1 CN1C(=O)CSC1=CC(=O)N1CC2C(CNC(C3CCCS3(=O)=O)=O)C2C1 CCCC(CC(C)C)C(=O)N1CCOC(C(=O)NCCCCCCF)CC1 c1(C(N2CCC(C)(CNC(C(C)SC(C)C)=O)C2)=O)cc(S(N)(=O)=O)c[nH]1 c1(C(=O)NC(CNC(CCOCCC)=O)(C)C)ccnc(OCCOC)c1 c1(N(CC(=O)OC(c2cccc(Cl)c2Cl)C)S(C)(=O)=O)cccc2ccccc12 N1(C(COCCNC(=O)C2=COCCC2)=O)CCC2C(C1)C2(F)F c1(OC)ccc(-c2cnccc2CN2CCN(c3ncccn3)CC2)c(OC)c1 c1(C(=O)NC(C(=O)NCP(OCC)(C)=O)CC(C)C)cc2cccnc2[nH]1 N1(C(C2N(C(Cn3ncc(C#N)c3)=O)CC2)=O)CC(=O)NC(=O)C1 n1(CCC)cc(Cl)c(C(=O)NCCC(C)CCNC(c2cnn(CCC)c2)=O)n1 C1(c2cccc(F)c2)(NC(=O)CCF)CCN(C(=O)CC(O)C2CCCC2)C1 C1(NC(c2c(C)c[nH]c2)=O)CC(O)CN(C(c2cn(C)nc2-c2ccoc2)=O)C1 c1(C(N(CCNC(C2N(CC)CCCC2)=O)C)=O)c(Br)nc2n1CCC2 N1(C(C(CC)Sc2nc(=N)[nH][nH]2)=O)CC(CNC(=O)Cc2cn[nH]c2)C2(CC2)C1 C(C1CC1)(C1CC1)=CC(=O)NC(C(=O)NCc1nncn1C1CC1)C1(C)CC1 C(C1CCCc2ccccc21)c1cn(-c2nccs2)nn1.OCC(F)CO c1(C(n2cc(C3(C)CN(C(=O)CCC#N)C3)nn2)CC)ccccn1 c1(C(N2C(C(C)(C)NC(=O)CC3CC=CCC3)CCC2)=O)ncncc1Cl N1(C(CC2N(C(CC(C(=C)C)OCC)=O)CC2)=O)CCCN(C)CC1CC c1(C(=O)NC2CC2CNC(=O)C(F)F)nc2c(cc1Br)OCCO2 C=CCC(CC(C)C)C(=O)Nc1ccccc1OCc1cccs1 c1(N2CC(C)(CNC(=O)CC(=O)NC3CC3)OCC2)cnc2[nH]ccc2n1 Cc1cc(C)n(C(C)CC(=O)NC(CCNC(=O)Cc2cnc(C)s2)C(C)C)n1 CC(CC(=O)N1CC=CC1CN(C)C)C(=O)c1cccc(F)c1 c1(C(=O)NCCN(C(=O)C(C)C2CC2)CCC)cc(F)ccc1NC Cc1cc(F)c(CNCC(CO)CC(C)(C)C)c(Br)c1 Cc1ccc(OCCC(=O)NC2C=CCN(C(C3CCCCN3C)=O)C2)c(C)c1 N1(C(c2ccn(C)c(=O)c2)=O)CC2=C(C1)CN(C(C1CCc3ncsc3C1)=O)C2 CC1CC(=O)NCC1C(=O)NC(CNC(=O)CCC(C)O)C1CC1 C(=O)(C(C)(C)C(F)(F)F)NC(CC1CN(C(CC2CC(OCC)C2)=O)C1)C c1(CCNC(C(C)NC(C)=O)=O)nc2cc3ccccc3cc2[nH]1 c1(C(=O)NCCC(C)N(C)C(C23CCC(CC2)C3)=O)cc(N)cc(S(C)(=O)=O)c1 N1(C(CN(C(C)=O)C)=O)Cc2n[nH]cc2C1C(=O)NCC1C2CCCC12 c1(C(N2CCC(CNC(C(C)NC(C)(C)C)=O)CC2)=O)csc2nccn12 C1(C2(NC(CCNC(N)=O)=O)CC2)CCCCN1C(=O)CC1CC2(CC2)CO1 C12(CCCCC1)CC(=O)O2.C(=O)(C(C)N=[N+]=[N-])N(CC)CC1CCOC1 c1(C(=O)NC2(C)CN(C(=O)CC(=O)NCC(F)(F)F)C2)ccnc(OC2CC2)c1 c1(C(=O)NC2C(NC(c3cc(OC)ncn3)=O)CCCC2)cc2sccc2[nH]1 c1(C(=O)NC(C)(C)CNC(=O)CC2CCOC(C)(C)C2)c[nH]c(=N)c2[nH]ccc12 Cc1sc(C(=O)NC2CC(C)(NC(=O)Cc3c(Cl)cnn3C)C2)cc1[N+](=O)[O-] O=C(C1=CNC2=NCCCN12)N1CC2CCN(C(C3CC4CCC(C3)O4)=O)C2C1 c1(C(N2CC(O)CC(NC(c3csc(C)c3C)=O)C2)=O)nccc2ccncc12 c1(C(=O)OC)sc(Cl)cc1S(=O)(=O)NCC1(CO)CC(C)(C)C1 N1(c2snc(C)n2)CCCC2(CCN(C(=O)C3CCCc4c3ncn4C)C2)C1 C(=O)(CCC(C)(C)SC)NCC(C)(C(N)=O)OC.C1(=O)COCCCN1 N1(C(=O)Cc2ccc(O)cc2)CCCC2(C1)CN(C(c1cnn[nH]1)=O)C2 CCCCC(CC)CC(=O)NC1CC(CC(=O)NC)C1(C)C.C1C(=O)N1CCC N1(C(=O)OC(C)(C)C)CCC(C(c2ccc(F)cc2)CC(=O)O)CC1 C(=O)(CCCC(=O)N(C1CN(C(C2CC(F)(CO)C2)=O)CC12CC2)C)OCC C1(CC)CC(CC(=O)NCC2CCCN2C(=O)CNC(=O)C(F)(F)F)CCO1 N1(C(C2N(CC)CCC2)=O)CCC2CN(C(c3cc(C)cnc3N)=O)CC2CC1 CN1CCC2(CC1)CC2C(N1CCOCC(C(=O)NCCC(=O)N(C)C)C1)=O Cc1ccnc2nc(C(=O)NCC(C3CCN(C(=O)C4=CCC4)CC3)(C)C)nn12 N1(N(C2CCSC2)C)CCN(C(=O)CNC)C(C2CC2)C1.C1(C=O)CC1CF c1(OC)noc(C)c1NC(C1CC(NC(=O)CNC(C2CC2C)=O)C1)=O C1(NC(CCC)=O)CCCN(N(C)C2CN(C)CC2O)C1 N1(C(CC(C=C)C)=O)CCC2(CC1)CN(C(=O)CCc1cc(Cl)no1)C2C(C)C Cc1ccnc(N2CCCC2c2cccnc2)c1-c1ccc(CO)cc1 C(=O)(CC(CC)NC(c1ccn(CC)n1)=O)N(CC)Cc1ccoc1 c1(C(C(=O)NC(CC)CNC(=O)CCc2cnco2)C)ccc(OC)cc1C c1(C(=O)NC2CC(CNC(C(C)(C)OC(C)=O)=O)C2)n[nH]c(C)c1Cl CC(CC(N)=O)C(=O)N1CCC(CCN(C)C(c2ncncc2N)=O)CC1 C1(CNC(c2nc(C)sc2C)=O)CCC2(CN(C(C3CCC(C)(C)O3)=O)C2)O1 c1(COC)ccnc(C(=O)N(C2CCN(C(=O)C(C)SC3CCCCC3)C2)C)c1 c1(CNC(C2(N)CCC(C)C2)=O)cc(F)ncc1Br C(=O)(CCCC(C)C)NCC(c1c(OC)cccc1)NC(=O)CC1(C)CC1(Cl)Cl N1(C(C(C)(F)F)=O)CCCC(N(CCO)C(C2CCN(S(=O)(=O)C(F)F)CC2)=O)C1 N1(C(CCCCCC)=O)CCc2nc(CNC(=O)C(CC(C)C)C(C)C)sc2C1 c1(C(=O)NC2CN(C(COCCC#C)=O)C(C)C2)cc(Cl)c2ccccc2c1O N1(C(C2(CC=C)CCC2)=O)CC2CC(NC(c3ccc4sccc4c3)=O)C(C2)C1 c1(C(N(CC(CC)NC(c2cc(C)c(CC)o2)=O)CC)=O)cc(C)n(C)n1 C1(NC(c2cc(C)oc2)=O)CC(NC(c2ccc(C(C)C)cc2)=O)C12CCC2 C1(=CCNC(C2(CC#C)CCOC2)=O)CCN(C(=O)Cc2cc(C)no2)CC1 Cc1cccc(CC(=O)NCCOCCOCCCNC(C2CC2(F)Cl)=O)c1F CC(C)C(C(=O)NCC(CC1CC1)C(=O)N(CC(F)Cl)C)C(C)C C1(CCC#C)CCN(C(c2cn(CCNC(c3cncc(O)c3)=O)nn2)=O)CC1 C(=O)(C1=C(Cl)CCCC1)NC(CNC(c1ccc(C#C)nc1)=O)CC=C N1(C(Cc2cc(C)no2)=O)CC(N(C(=O)Cc2c(C)n[nH]c2C)C)C2(CC2)C1 C1(c2cn(CCC(C)(C)C)nn2)CCCN(CC(=O)NC2CCOC(C)C2)C1 c1(C(=O)OC)cc(C)nn1CC(N1CCC(C)(CNC(=O)CC2CC23CC3)C1)=O c1(N(CC2CCCOC2)CC)nnc(-c2cccn2C)n1C CC(C(=O)NCc1ccc(C(NCP(C)(C)=O)=O)o1)C(C)(C)C C(CC(C(=O)NCCNCCN=[N+]=[N-])NC(=O)C(C)CC1CCC1)SC C1(NC(C2C(c3c(C)occ3)C2)=O)CCN(C(=O)C=C(Cl)Cl)CC1C c1(OC)ccc(C(N2CC3CC(NC(=O)C(C)c4cccs4)C2C3)=O)cc1O CN1CCCC(C)(C(=O)NC2CC=CCC2C(=O)NCc2ccc(Cl)o2)C1 O=S(=O)(c1ccc(Cl)cn1)N1CC2CN(Cc3ccc(Cl)o3)C2C1 C1(C(=O)NCC2CCC(NC(CCC(=C)C)=O)C2)CN2CCN1CC2C C(=O)(C(CC(C)C)CC(C)C)N(CC(CNC(CCOC(CC(C)C)C)=O)O)C CC1(O)COCCN(C(=O)C(CC2CCC2)NC(C2CCC(F)CC2)=O)C1 c1(C(=O)NCC2(C)CCN(C(c3c(CC)[nH]cc3)=O)CC2)cc(F)c(F)cc1N Cc1nc2ccc(C(=O)NC3CCN(C(C4(CC5CCC5)CC4)=O)C3)cc2n1C Cc1c(C(=O)NC(C)CCCCNC(C2CCS(=O)(=O)C2)=O)sc2cncn12 Cc1ccncc1C(=O)N(C1CCCN(C(=O)Cc2ccoc2)C1)C c1(OC)ccccc1SCC(N1CCCC(C(C)NC(=O)CN2CCCC2)C1)=O C(=O)(C(O)CC(C)(C)C)NCC(CC)NC(c1nc(CC)oc1C)=O N1(C(CC=CC=C)=O)CCN(C(c2[nH]cc(C)c2C)=O)C(c2cccc(Cl)c2)C1 C(C(C)(CC)CC)(c1n(CCOC)nnn1)NCC1(NC(=O)OC)CC=CCC1 c1(C(=O)NCC2(C)CCCN2C(=O)Cc2cscn2)c(F)cc(C#N)cc1F c1(C(N2CC(N(C(C(C=C=C)C)=O)C)C(O)C2)=O)ccc(Cl)c(OC)c1F C1(C(=O)NC(C2CN(C(C(C3CC3)SCC)=O)C2)C)CCN(C(N)=O)CC1 C12(NC(CCC)=O)CN(C(c3cccnc3-c3cnn(C)c3)=O)C(COC)(C1)C2 Cn1nc([N+](=O)[O-])cc1C(N1CCC2CCCC12CNC(=O)CC1=CCCC1)=O C1(C(N(C(c2ccc(C(F)(F)F)cc2)C)CC)=O)Cc2c[nH]cc2S1(=O)=O N1(C(C2CC(OC)C2)=O)CCSCC1C(=O)N(C1CC1(C)C)C c1(NC(CCN(C(=O)C2=C(C)CCOC2)CC=C)=O)cc(C#N)ccc1F C(C(CC(F)(F)F)NC(c1cccc(CO)n1)=O)NC(c1nocc1C1CC1)=O c1(C(N2C(C3(NC(C4CC5CC5C4)=O)CC3)CCC2)=O)nc[nH]c2ncnc1-2 N1(C(C=CSC)=O)CC2(C1)CN(C(=O)Cn1cnc([N+](=O)[O-])c1)CC2CO C(C1=CCCN(C(=O)Cc2ccc(OC)cc2)C1)NC(CC=CC=C)=O C1(CNC(C(CC)(C)C)=O)(NC(C2CCC(C#N)C2)=O)CCC(C)(C)CC1 O=C1NCC(C(=O)NC2CC(CCC(=O)NC3CC(F)(F)C3)C2)N1 C(CC(=O)N1CCC(NC(c2cccc(N)c2O)=O)CC1C)(C(F)(F)F)OC c1(NC(CCOC2CN(C(CC)=O)C2)=O)cc(C(=O)NOCCOC)co1 N1(C(COCC)=O)CC2CN(C(=O)C(c3cccc(C)c3)C)CC2C1 C(C(C)(C)CC(F)F)c1onc(CN2C(c3cccc(OC)c3)(COC)CCC2)n1 c1(CNC(C2CSCCN2)=O)cccc(F)c1Br C1(C(=O)NCCCN(C(=O)CN2CCCCCCC2=O)C)OC(C)(C)OC1(C)C c1(C(N2CCC(CNC(COC)=O)C2)=O)c(N)ccc2nccnc12 c1(C(=O)NCC(C(C)C)NC(CC(c2ccc(C)cc2)C)=O)cc(Cl)ccc1F C12CCN(CC1)CCN(C1CC1)C2=O.c1(SC)cscn1 c1(NC(C2C3(CN(C(c4ccnc(C)n4)=O)C3)C2)=O)cc(F)c(F)cc1[N+](=O)[O-] C1(C(=O)NCCCCNC(c2ccc(C#N)o2)=O)CCC(N=[N+]=[N-])CC1 c1(C(C(=O)N2C3CCN(C3)CCS2(=O)=O)(F)F)ccccc1C.CCC(=O)O C(N=c1ccnc(CO)[nH]1)C1C(CNc2cc(CC)nn2Cc2ccccc2)C1 C=C(C)CCCC(=O)NC(CC1CC1)CC(=O)NCC1CC(C#N)C1 C12(C(N(CCCCNC(C(C)Cc3ccccn3)=O)C)=O)C=CC(CC1)C2 Cc1c(Br)sc(CNC(c2cc3n(n2)CCC3)c2nnnn2CCC2CC2)c1C C1(CNC(CN(C2CCSC2)C)=O)COCCN1C(=O)Cc1cncc(F)c1 C12(NC(C3CCOCC3)=O)CCCC1N(C(C1CC3(CCCO3)C1)=O)CCC2 c1(C(N2CC(O)(C(C)NC(C3CCC3(F)F)=O)C2)=O)cccc(C(F)F)c1F C(CC)(CC)(CCNC(C1(CF)CC1)=O)NC(C1CC(O)(CC#C)C1)=O c1(C(=O)NC(CC#C)(C)C)cc(Br)ccc1CC N1(CC)N=C(C(=O)NC2(C3CC3)CCN(C(=O)Cc3cc(Cl)cs3)C2)CCC1=O c1(CC(=O)NC(C)CCNC(C2CC(F)C2)=O)ccnc(O)c1 C(CCCNC(=O)C(C)N(C)C(C)=O)(c1ccccc1)NC(C1C(CC)C1)=O N1(C(C=CC(C)(C)C)=O)CCC2CCCC12CNC(c1ncc(C(F)F)s1)=O C1(C#N)(C(N2CC(CCC=C)(CC(=O)NC3C(C(=O)OCC)CC3)C2)=O)CC(C)C1 c1(C(=O)NCCN(CC(=O)NCCCC)C(C)C)cc(C(F)(F)F)nn1C Cc1oc(C#N)cc1C(=O)NC(C)C(=O)NC1(C)CS(=O)(=O)C1 c1(C(C)C)ccc(NC(=O)C(=O)NC(C2CCCCO2)C2CC2)cc1 C1(C)(CNC(c2n(C(CC)(C)C)nnn2)c2cc(COC)on2)C=CCCC1 CC1(CNC(C2CCCN2C(=O)CCc2nccs2)=O)CCCCCC1 c1(C(=O)NC2(C)CN(C(C(C)Cc3ccccc3F)=O)C2)cc2cccnc2o1 C(=O)(C1=CCCOCC1)NC1CCN(C(c2n(CC#N)ncc2)=O)CC1O CCCCCC(=O)NC1CCN(C(=O)C(c2ccc(F)cc2)C2CC2)C1CC C1(C(N(C)CC2(Br)CC2)=O)CCCCC1CNC(=O)CN1CCSCC1 C1(C(N2CC(C)C(CNC(=O)C(C)(C)C)CC2)=O)CC2C=CC1C21CC1 C1(C(=O)NCC2(F)CC(CNC(c3c(OC)n[nH]c3)=O)C2)CCC(C2CC2)CC1 C1(C(=O)NCC(CCC)NC(=O)C(C)(C)O)CCCC(F)(F)C1 C(c1ccccn1)=CC(=O)NCC(C)(C)NC(C1C(C)(C)C1(F)F)=O C12(C(N3CCC(NC(C(c4ccccc4)N(C)CC)=O)C3)=O)CC(C1)C(C)O2 C1(NC(CC2C(C)(C)OCC2)=O)C2CC3C(C2)C13C(=O)N1CC(O)CO1 CC1(C)CC(C(=O)NCCOCCC(=O)NCC2CC3CCCC3C2)CCO1 c1(C(N(CC)CC2CCN(C(=O)Cn3ccnn3)CC2)=O)ncc(Cl)cc1F c1(OCCNC(C(=O)OC)Cc2ccc(F)cc2)cc(C)nc2cc(Cl)ccc12 CN1Cc2c(CNC(c3nn(-c4ccccc4Br)cc3O)=O)cccc2C1=O N1(C(C2N(C(C(CCOC)OC)=O)CCC2C)=O)CC2(CCOCC2)C1 N1(C(CC2(C)OCCO2)=O)CC2CCN(C(=O)C3=NNC(=O)CC3)C2C1 c1(N(C)C(C2CN(C(C3CC3C(=O)N(C)C)=O)C2)=O)c(Br)cc(C(F)(F)F)cc1I O=C(CCC(=O)N1CCCC1C1CCCCCC1)c1ccncc1 CC1(C(N2CCC(CNC(C3CCC(F)C3)=O)C2)=O)C=CCCC1 C(=O)(CC(C)C(F)(F)F)N1CCCC(C)(NC(Cc2ccc(SC)cc2)=O)C1 c1(C(=O)NC(C(C)C)C(C)NC(=O)CC2C(C)(C)C2(C)C)noc2ncccc12 N1(C(=O)OC(C)(C)C)CC2CC(C(N3CCCC(C(C)(F)F)C3)=O)CC(C1)C2=O c1(C(=O)NC(CC2CN(C(C3CC=C(C)CC3)=O)C2)C)cc2n(n1)C(C)CCC2 C1(C(=O)NCCSC)CN(CC2(N3CCN(C)CC3)CCCCC2)CCC1O C1(NC(=O)NCC(CCSC)N)CCC(C)(C)CC1CSc1ccccc1 N#CC1CCN(c2cc(CNc3ccccc3)ncn2)C1 c1(C(=O)NC2CCCN(C(C3CC34CCSCC4)=O)CC2)scc2c1CCCC2 C1(NC(C2CCC(C(C)C)CC2)=O)CCCCN(C(C2(F)CCOCC2)=O)C1 C1(C)(CNC(c2c(C)onc2)=O)CCN(C(C2CCC(CC(C)C)CC2)=O)C1 N1(C(C2CCN(CCO)CC2)C(=O)NCC)CCCCC1c1ccco1.C(C)S c1(OC)cccc(CCCNC(=O)C(=O)NCc2ccc(C)n2C)n1 C1(CNC(C(C)NC(C)=O)=O)(CO)CCN(C(c2cc(C(N)=O)c[nH]2)=O)C1 N1(C(C)=O)CCOc2cc(Nc3cnn(S(C)(=O)=O)c3)ccc21 N1(C(C(c2cccc(Cl)c2)(C)C)=O)CC2CC1CN2CC(=O)C1CC1 CC1(C)CCCC(CNC(=O)CC2CCC(NC(C3(C)CC(F)(F)C3)=O)CC2)O1 c1(NC(=O)C2CC2)ccc(Cl)c(C#N)c1.CN1CC(N2C3(CCC3)CC2=O)C1 CC1CCCN(C(c2cc(CF)on2)=O)C1CCNC(c1ccc(N)c(N)n1)=O c1(OC)c[nH]c(C(N2CCC(CNS(C)(=O)=O)CC2)C(=O)NCC(F)F)cc1=O N1(C(c2cccc(CNC(C3C(C)OCC3)=O)n2)=O)CCOC2(CCC2)C1 C(=O)(C(O)CCC(C)C)NCC(C)(C1CCC1)NC(c1nc(OC)c(F)cn1)=O CCCC(CC)CCC(=O)N1CCC(OCC2CC2(C#N)C(=O)OC)CC1 n1(CC(C)(F)F)ccc(NC(N2CCC(N)C2)=O)n1 c1(C(=O)OCC)cc(C)c(O)nn1.C1(=O)CCC(=O)CSC2CN1CCO2 C(N(O)C(=O)Cc1cccc(Cl)c1)c1cn(C(C)(C)C)nn1 N1(C(CCCNC(C2N(C)C(=O)CCC2)=O)=O)CC2C=CCC(C2)C1 CC1(CC(N2CC(=C(F)CNC(=O)C=C3CCCC3)C2)=O)CCCCC1 C1(OC)CCCC(NC(c2nc(-c3cnccn3)no2)C(C)C)C1 CC12CCC(C(=O)NC(CNC(=O)C=C3CCC3)CO)(CC1)CO2 N1(C(CCN(CCOCCOC)C)=O)CC(NC(=O)C(F)(F)CO)C(C)(C)C1 C1(C2CC2)(NC(CC(C=C)C)=O)CCN(C(c2noc3c2CCCC3)=O)C1 CC1(C)CCC(CNC(=O)CC2CSCCO2)(NC(C2CCC3(CCC3)O2)=O)C1 Cc1ccnn1C(C)CNC(C1(O)COC1)C c1(CC)ccc(C(N2CCCC2C(=O)NC2(COC)CC2)=O)cc1 C1(CNC(C(F)=CC)=O)CCCC2(CN(C(=O)C(C(C)(C)C)N(C)C)C2)O1 C12(CNC(COC(C)=O)=O)CC(NC(=O)Cc3csc(C4CCCC4)n3)(CO1)C2 c1(-c2nc(-c3nccc(OC)c3)nn2C2CS(=O)(=O)C2)onc2ccccc12 C1(C(C)C)CN(C(N)=O)CCN1C(=O)C(Cc1ccc(O)cc1)NC(N)=O CC1(C)CC(CC(=O)NCCCNC(c2cccc(C(C)(C)C)c2)=O)NC1=O C1(CNC(C(C(C)C)NC(COC)=O)=O)COCCN(C(c2cc(C)c[nH]2)=O)C1 N1(C(CC(C)OC(C(=O)NC(C)C)=O)=O)CCC(OC2CC2)CC1 C1(NC(c2ccc(CO)o2)=O)CCCN(C(C2CC(n3ccnn3)C2)=O)CC1 c1(C(N(C2CN(C(Cc3cc(C)[nH]n3)=O)CC2F)C)=O)cc2nccn2c(O)n1 C(=O)(CCCc1sccc1C)NCC(CC)NC(C1(n2ccnc2)CCCC1)=O C12(CNC(CC(CC)CC)=O)CCCC1N(C(=O)C=C1CCCC1)CCC2 C(=O)(C1=NOC(C2(O)COC2)C1)NCC(C1CCCC1)NC(c1cnsc1)=O CC(C)S(=O)(=O)C(C)C(=O)N1CCC2(C1)CN(C(c1cc(Cl)c(F)c(Cl)c1)=O)C2 Cc1cccc(C)c1C(=O)NC1CC1C(=O)OC(=O)C(C)N(C)C CCC(C(=O)NC(c1ccccn1)C)N(C(=O)Cc1cnsc1)C C(CCCC(=O)NCc1ocnc1C(N1CCOC(CCF)C1)=O)OCC C1(NC(c2c(OC)cc(C)cn2)=O)CC2CC1CN(C(C1CCC(C)C1)=O)C2 C1(C(=O)NCC2(O)CCN(C(=O)CNS(=O)(=O)C3CC3)C2)C2CCCCCC12 c1(CC)nc(C)c(C(=O)NCC2CC(NC(=O)C(F)(F)Cn3cccn3)C2)s1 c1(OC(CC)C)ccc(C(N2CC(NC(=O)CC)C(C(F)(F)F)C2)=O)cc1 c1(CC)nc(C)oc1C(=O)NC12CC1CN(C(c1csc(C(C)C)n1)=O)C2 C(=O)(CCC(F)(F)F)N1C(C(=O)NC(COC)C2(C)CC2)CCC1 C(=O)(CCCC(CC)NC(=O)Cc1c(C)cnn1C)NCCCC=C C1(O)(CN(C)C)CCN(C(=O)CC2C=CC(NC(C3CC4CCC4C3)=O)C2)C1 c1(CN2CC(C(=O)NC(c3ccccc3)C(N)=O)OCC2)cc(Cl)c(F)c(Cl)c1 c1(C(N2CC(CCNC(C(COCC)C)=O)C2)=O)cc(Cl)c2n[nH]cc2c1 c1(C(=O)NC(C)CCNC(=O)C(c2cccc(F)c2)C)cnc2n(c1=O)CCS2 c1(C(N2C(CNC(c3ccc(C=C)cc3)=O)CC3CC32)=O)cncc2[nH]ccc12 C=CCCCC(C(=O)NCC(C)C(F)(F)F)NC(C1COCOC1)=O c1(C(=O)NC2CC(NC(c3ccc(C#C)cn3)=O)C2)n[nH]c2ccc(Br)cc12 c1(CC(N2C(CNC(CC=C)=O)C=CC2)=O)ccc(F)c(Br)c1 c1(NCCN(C(=O)CC2(O)CCCCC2)C)nc(O)n(C)c(=O)c1[N+](=O)[O-] c1(C(C(=O)NCC)N(c2ccccc2)C(C)=O)cccc(Cl)c1 C(c1ccc(OC)c(F)c1)=CC(=O)OC.C1(=O)C(Cc2ccccc2)N1CC1CC1 CC1=C(C(=O)N2CCCOC(CNC(C3(F)CCC3)=O)C2)CCO1 N(C1CCc2cc(NC(=O)COCC(=O)OC(C)(C)C)ccc21)C(CSC)=O N1(C(CC(=O)N(C)C)=O)Cc2ccccc2C1CNC(=O)CCC(C)(C)[N+](=O)[O-] c12c(cnn1CC)C(=O)NC2.c1(OCCNCC(=O)NC)ccc(OC)cc1 C(C)(C(=O)NCCCCO)N(CCC)C(C1CCO1)=O C1(NC(C(C=CC)O)=O)CCCCC1NC(c1cn(CC2CC2)nn1)=O C1(NC(Cn2ncc(CC)c2)=O)CCC(C)(C)CC1CNC(c1nnsc1C)=O C(=O)(C1CCCCc2ccccc21)NC1CC(CNC(=O)C2=CCOC2)C1 C12(CNC(C(C)(C)CF)=O)CCC(C1)N(C(=O)C(F)CC1CC1)C2 CC(=O)C(C)CC(C)C(=O)N1CC(C(=O)N(C)Cc2cccnc2)CC(C)C1 C1(CNC(C(CCOC)C)=O)CCCCN(C(c2cc(-c3ccco3)c[nH]2)=O)C1 c1(OC)ccc(-c2n[nH]cc2C(N2CC(NC(=O)CSCCC#N)C2)=O)cc1 c1(C(=O)OC)nc(CCN(c2ccccc2)C(=O)C(C2CCCCC2)F)oc1C C(=O)(CC(C)(C)C)NC(N1CC(C(C(=O)NCCC2CN(C(C)=O)C2)OC)C1)=O C(CCCCCNC(C1CCOC(=O)N1)=O)NC(C(C1CC1)OCC)=O Cc1cc(C(N2CC(O)CC2CNC(C23CCC2C3)=O)=O)ccc1[N+](=O)[O-] c1(C(C)NC(C2(CC(N)=O)CC2)=O)nocc1C(=O)NCCC(C1CC1)C1CC1 C1(NC(C(=O)NCC2CC2)=O)CCCC2CN(C(c3nccc(Cl)c3F)=O)CC12 N1(C(c2c(CC)c[nH]c2)=O)CCN(C(=O)CC2=CCN(C)CC2)C(C)CC1C CC1(C)CC(NC(c2cccc(Cl)c2F)=O)CN1C(C1CCC(=O)C1)=O CCS(=O)(=O)CC(=O)NCC(CC)CC(=O)NC(CF)C(F)(F)F c1(CNC(C2(NC(c3n[nH]c(C)c3Cl)=O)CCOCC2)=O)ccnc(F)c1F C(C)(C(CC(=O)Nc1cnc(C)c(Cl)c1)NC(=O)CCC1(C)N=N1)OC CC1CN(C(c2ccnc(N(C)C)c2)=O)CCC1C(=O)N(CCO)C1CC1 C(C(=O)N1CC=CCO1)C1(CNC(C2C(C)CC2)=O)CC1 N1(C(C2CC(CNC(C(C)OC)=O)OC2)=O)CCCN(C)CC1 c1(C(=O)NC(CC)CC(=O)NC(c2ncnn2CC)C)ccnc2cc[nH]c12 Cc1n[nH]c(=NCC(C)(C(C)C)NC(=O)CC2CCNC2=O)s1 c1(-c2onc(C)n2)ccc(C(=O)NC(C)CN(C)C(c2nocc2Cl)=O)cc1 CC1CN(Cc2ccccc2)CC(C)N(C(c2ccc3ocnc3c2)=O)C1 C1(NC(c2cc(-c3ccn(C)c3)[nH]n2)=O)COCCN(C(=O)CC2CCCC2)C1 CC1CC(NC(c2ccno2)=O)CCN1C(c1ncccc1Cl)=O CC1=NN(C)C(=O)C1CC(N1CCC1CNC(=O)CCOC1CCC1)=O C(=O)(CCCCC(=O)NC)N1C2C(N(C(C(C=C)C)=O)C)CC(C2)C1 C12(CCNC(C3C4CN(C(c5cnc(Cl)s5)=O)CC34)=O)CC3CC(CC(C3)C1)C2 CC1(C(N2CCC(OC3CN(C(=O)CCF)C3)CC2)=O)COCCO1 c1(C(=O)Nc2c(C(F)(F)F)ncc(COC)c2)cnc2c(Br)n[nH]c2c1 C(=O)(C(O)CC(C)(C)C)N1C(C2CCCN(C(CCC(=C)Cl)=O)C2)CCCC1 C(=O)(CCCC(=O)N(C)C)NCC(C(=O)NCC1(O)C(C)CCC1)N(C)C c1(OCCC(=O)N(C(C)C=CC(=O)N(C)C)C2CC2)ccc(F)cc1Cl Cc1cc(Nc2ccc(C(=O)Nc3ccc(Br)nc3)cn2)cc(C#N)c1 c1(OC)cnc(F)c(C(=O)NCC(n2cc(-c3cnccc3Cl)nn2)C)c1 C1(C(N2CCC(CCCC)C2)=O)CCN(C(c2sccc2CC)=O)C(CC)C1 C1(NC(C2C(CNC(Cc3cnc(C)s3)=O)CC2)=O)CCCN(C)C1 C1(CC)C(NC(c2cccnc2C)=O)CCCN1C(=O)CN1CCC(OC)C1 C1(C(N2C(COC)C=CC2)=O)CC2CC2N1C(=O)C(n1ccnc1C)C c1(SC)nc(N(C2CCNCC2(C)C)C(=O)CN2CC(=O)NC2=O)cc(C)n1 C1(NC(c2c(CC)cccc2)=O)CC2CCC(C1)N2C(C1(Br)C(C)C1C)=O N1(C(C(C)CCO)=O)CCN(C(=O)CSc2n[nH]c(O)n2)CC(O)C1 C1(C(=O)N(CCCCNC(c2c[nH]nc2C)=O)C)(OC)CC(C)CC(C)C1 Cc1cn2c(C(=O)NCCN(C)C(c3ccnc4ccccc34)=O)c(Cl)nc2s1 C(=O)(C(C)CCO)NCC(CN(C(C(C)OCCN(C)C)=O)C)(C)C c1(C(=O)NCC(C)N(C)C(C2COC3(C)CC2C3)=O)cccc(C(F)(F)F)c1O C1(CC(=O)NC(CN(C(c2ccoc2CC(N)=O)=O)CC)C)CCCS(=O)(=O)C1 C1(CCNC(C2CC(OC(F)F)C2)=O)CCN(C(=O)CSC2CCCCO2)C1 C1(C(=O)NCC(C)CNC(C2(C)CC2C(F)(F)F)=O)CS(=O)(=O)CC(=O)N1 C1(NC(c2ccc(SC)cc2)=O)CN(C(=O)Cc2nonc2C)C2CCCCC12 S(=O)(=O)(c1c[nH]ccc1=NC(C)C1CCCCN1CC)N1CCC(CC)(CO)C1 N1(C(CC(=O)OCC)=O)CCC(NC(C23CC(CF)(CO2)C3)=O)C1(C)C C1(N(C(c2c(CC)nco2)=O)C)C2CN(C(=O)CCOc3ccccc3F)CC12 N1(C(C(N2CCSCC2)C)=O)CCC(NC(C2CN(C)CC(C)O2)=O)CC1C CC(C(=O)NNc1ccc(Br)nn1)c1c(F)cccc1Cl c1(-c2onc(C(=O)O)n2)ccc(Oc2ccc(Cc3ccccc3)cn2)cc1Cl C1(C(c2cn(Cc3c(C(=O)O)cco3)nn2)O)CCN(C(C2(Br)CCC2)=O)CC1 C1(NC(c2ccc(CC)cc2)=O)CN(C(c2cccnc2)=O)CCC1(F)F N1(C(Cc2cn(CC)nn2)=O)CCC(C)(CNC(=O)CSCCN(C)C)CC1 C1(O)(CC(=O)NC2C(C)(C)C2C(=O)NC2CC(CO)(CO)C2)CCCOC1 CN1CCN(C(C2OC3CCC2CC3)=O)CC1CNC(=O)CSc1ccccn1 c1(C(=O)NC2C3CN(C(CCC=C)=O)C(C3)CC2)cc(S(N)(=O)=O)c(Cl)cc1Cl c1(CNC(C(C)C2CC2)=O)ccc(CCNC(C2(C)CCC(=O)N2)=O)cc1 C#Cc1ccc(OCC(N2CCN3CC2C(=O)NC(C)C3=O)=O)cc1.C(C)(=O)OC CCCCC(CNC(=O)C(C)CCOC)NC(c1ocnc1C1CC1)=O C1(C(=O)NCCNC(Cc2cn(CC)nc2)=O)CCCS1(=O)=O N1(C(c2cc(C)sn2)=O)CCN(C(=O)CC2CC(C)(C)CO2)CC1C CCC(CC(F)F)C(=O)N1CCCC(CCNC(c2cc3oc(Cl)cc3[nH]2)=O)C1 N1(C(CSC)=O)CC2CCC2(CC(N2CCCC2CCO)=O)C1 c1(C(=O)NCCCC(c2ccccc2)NC(C(C=C)O)=O)c(F)c(N)cc(F)c1F C1(C(=O)NCC2N(C(C3(F)CC3)=O)CCC2)CC12CCOc1ccccc12 c1(NC(c2ccccc2I)=O)cc2ccc(C(=O)O)cc2cn1 c1(C(=O)Nc2ccc(-c3cnn[nH]3)cc2)ccc(O)cc1Cl c1(OCC=CC)cccc(CC(=O)NC2CCN(C(=O)CCC(=O)NC)C2C)c1 c1(CC)ccc(F)c(C(N2C3CCC2CN(C(=O)C=CCF)C3)=O)c1F c1(C(N2CC(OC)CC(NC(C(C=C)(C)C)=O)C2)=O)ccc2nn[nH]c2c1 N1(CC(=O)NCC(N(C(=O)Cc2ccon2)C)C2CC2)C(=O)CCC1=O CC(C)(C)CS(=O)(=O)NCCc1c(Cl)cccc1Cl C1(C(=O)OCc2nnco2)CCCC12OCCO2.CC(C)(C)N1C(=O)C1 N1(CCNC(Cc2cc(C)no2)=O)CCN(C(C2CCCC23CC3)=O)CC1 c1(C(=O)NCCCC2N(C(CC(COC)C)=O)CCC2)n[nH]c2ccc(Cl)cc12 c1(CC)ccc(C(N2CCC(NC(c3cc(COC)no3)=O)C2(C)C)=O)cc1F N1(C(C2CC3(ON=C(C)C3)C2)=O)CCCCC2(C1)CN(C(=O)C(C)SC(C)C)C2 NS(=O)(=O)CCC(=O)NCCCC1CCCN1C(c1ccc(NC=O)cc1)=O C1(C(=O)OC(C)(C)C)C(C(=O)NCCNC(C23CCC2CC3)=O)C1(C)C CC(C)(C)S(=O)(=O)CC(=O)N1CCN(C(C2COCCOC2)=O)C2CC12 c1(C(N2CC(C(C)NC(c3c(C(C)C)nns3)=O)C2)=O)cc2ccsc2[nH]1 Cc1ccc(C=CC(=O)NCC(C)CNC(=O)CC2CCCS(=O)(=O)C2)cn1 N1(C(C=Cc2cnc(C)s2)=O)CCCC2(NC(C3CCC=CCC3)=O)CCCC12 Cc1cc(F)cnc1C(=O)NC1CCN(C(=O)CCC(C)C#N)CC1O N1(C(C23CCC(OC)C2C3)=O)C(C(N2CCOCC2CN(C)C)=O)CCC12CC2 N(C1CCc2c(Cl)ccc(Br)c21)Cc1cnc(OC)nc1 C1(C(=O)NCCC2CCN(C(C3CC(C(=O)OC)C3)=O)C2)CCC(C)(C)OC1 c1(NCC(C)C(F)(F)F)ccc(S(=O)(=O)NC2CC2C2CCOCC2)c(Br)c1 C=CC1(CC(=O)NCC23CCC(CC2NC(=O)Cc2cn[nH]c2)C3)CCCCC1 c1(NC(C)=O)ccc(C(=O)NC(C)CNC(C2(C#N)CC(C)C2)=O)c(Cl)c1 C1(C2(NC(Cc3ncc(C)s3)=O)CC2)CCCCN1C(C1C2CCCC12)=O N1(S(c2ccc(C(=O)OC)cc2)(=O)=O)CCCC2(CCN(C(=O)CN(C)C)C2)C1 c1(NCCCC(N)=O)nc(N2CCSCC2)nc2scnc12 C1(NC(CCC2(C)CC2)=O)CC2CCC1N2C(=O)Cc1ccc(NC(N)=O)cc1 C(=O)(CCCS(C)(=O)=O)NC(C1N(C(CC(CC)C2CC2)=O)CCC1)(C)C CC(C)C(C(=O)NC1CN(C(C2CCC2)=O)CC1C)NC(c1cccs1)=O N1(CCCNC(C2C(OC(C)(C)C)C2)=O)CCN(C(c2ccc(F)s2)=O)CC1 CCC(C)(C(=O)NC(C)CCCCNC(=O)CCc1ccc(O)nn1)OC N1(C(c2c(C)n(C)nc2)=O)CC2CN(C(c3ccnnc3S)=O)CC2(C)C1 c1(C(=O)NC2C(NC(c3cn[nH]c3)=O)CC2)c[nH]nc1-c1ccco1 c1(OC)cc(Cl)c(C)cc1CN1CCN(C(=O)C(F)(F)CC(C)C)CC1 c1(-c2nc(C(C3CC3)OC)nn2-c2ccnc(Cl)c2)c[nH]c2nc(Cl)ccc12 Cc1cnc(Cl)c(NC(C2CN(C(=O)C(C)(C)Cc3ccccc3)C2)=O)c1 N1(C(c2cc(C#N)sc2)=O)CCCC2(CCCN2C(c2ccc(Cl)nc2O)=O)C1 N1(C(Cc2ncc(C)s2)=O)CC(C2CN(C(c3cc(F)c(F)cc3O)=O)C2)C1 Cc1cncc(C(N2CC(CCNC(=O)C(O)CN(C)C)C(C)C2)=O)n1 CCCC(C)(C)C(=O)N1CCC(C)(NC(C2CCC23CCOCC3)=O)C1 CCCC(CCC)CCCC(=O)N1CC(CCNC(=O)CN(C2CCSC2)C)C1 C1(C(=O)OC)CC(=O)CN1CCc1c(O)n[nH]c1C c1(C(N2CC(C)C(CNC(C3CCCCO3)=O)CC2)=O)cccc([N+](=O)[O-])c1 Cc1cc([N+](=O)[O-])cc(Br)c1NC(=O)NCCC1CCOC(C)C1 CCC(C(=O)OC)C(=O)NCC(CNC(c1cccc(C(N)=O)c1)=O)CO CN1CCc2c(NC(=O)NC3(c4cc(O)ccn4)CC3)cccc2C1=O Cc1ncc(CCNC(=O)C(C2(O)CN(C(C3CC3[N+](=O)[O-])=O)C2)F)[nH]1 C1(CCC(=O)N(C2CCCC2)CCNC(C2(C(N)=O)CC2)=O)CCC(=O)N1 C(=O)(C1=CCCOC1)NC(C(C)C)CCN(C)C(c1cnc(C(F)(F)F)cn1)=O c1(N2CCCC(CCNC(=O)C=Cc3nccs3)CC2)c(Br)cccc1[N+](=O)[O-] c1(NCc2cc(C)ns2)cc(NCC(Cl)=CCl)ncn1 c1(CCC(N2CC(C)C(NC(=O)Cn3nnc(=O)[nH]3)C2)=O)ccc(F)cc1Cl CC(O)(CC(=O)N1CC(NC(=O)COc2cccc(F)c2)C(O)C1)C1CC1 C(=O)(C(C)(C)CC(=O)NC(C)CNC(c1ccccc1C(C)(C)C)=O)OCC CCC(C)CCCCC(=O)N1CCC(N(C(=O)CCCN(C)C)CCO)C1 CC1(C)C2CCC1(C)C2C(=O)NC1CN(C(c2cc(F)ccc2F)=O)CC1F c1(CC)cc(C(=O)NCC2CCC(C(=O)NCCC(C)(C)F)O2)n[nH]1 O(C=C(C#N)C(=O)N1CC(NC(c2cc(C3CCC3)no2)=O)C(C)(C)C1)CC C1(C(N2CCCC(O)C2Cc2ccccc2)=O)COc2ccccc2C1 c1(C(=O)NCC(C)NC(C(C(=O)NCC)(C)C)=O)nc(C)nc2sc(C)c(C)c12 N1(C(c2cccc(C#N)c2)C(=O)NCCSC)c2ccc(Cl)cc2CC1C C(C(COC)C(=O)N(CCNC(C1CC2CCC1C2)=O)C(C)C)OC c1(OC)ccc(C(C(=O)NCCC(F)F)N(C)C(C2CCCO2)C)c(Cl)c1OC C1(NC(C(=O)Nc2nc(C)sc2C)=O)CCCC2CN(CCCCCF)CC12 c1(C(=O)NC2C(NC(COCCCC(C)C)=O)CCOC2)cn2c(n1)CCC2 C(C)(C(=O)N(CCCNC(=O)CNC(=O)Cn1cncn1)C)=CC Cc1ccc(NC(=O)CN(C2CCC2)C(C2CN(C3COC3)C2)=O)c(C)n1 C#Cc1ccc(C(N2CCC3CC23C(=O)NC(CC2CC2)C(=O)NC)=O)cc1 N1(C(C2CC3(C2)CC32CC2)=O)CC2C3CCC(C2C1)N(C(=O)COCCCF)C3 N#CCCCC(=O)N1CCCC1C1CCN(C(C2CC(F)(CO)C2)=O)C1 CC1CC(C(=O)NCC2CCN(C(=O)CCc3cn[nH]c3)CC2)Cc2nn[nH]c21 C1(C)(C(=O)NCCC(CC)(C)NC(C2COCCO2)=O)CCCN(C)C1 C1(OC)CCCN(C(=O)C(CC(C)C)ONC(c2cccc(F)c2)=O)CC1 C1(NC(C2CCC3(CCC3)O2)=O)CCC12CCN(C(=O)C1=CCCOC1)CC2 c1(N(CC)CC)nc(N(C)C2CC2NCc2cccc(CO)c2)c2c(n1)CCC2 c1(OC)cccc(-c2cc(N3CC4CC(C3)N4C(=O)CN(C)C)ccn2)c1OC CCC(CC(F)F)C(=O)NCC1(NC(c2ccn(C(C)(C)C)n2)=O)CCOC1 C1(CNC(C(=O)NCC)=O)C(C)CCN1C(c1ccc(CO)o1)=O N1(C(C2(OCC)CCOC2)=O)CCCC(C2CN(C(=O)C=CC3CCC3)C2)C1 C1(NC(CN(C2CCSC2)C)=O)CC(C2CCN(C(C3CC3F)=O)C2)C1 CC1C(C)N(C(c2cccc(C#N)c2Br)=O)CCN1Cc1ccccc1 c1(C(C(=O)NCC2CC2)N(CCCOC)CC(C)C)nc(Br)ccc1OC n1(CC2COC(C)(C)O2)cc(Br)cc(I)c1=O C1(CNC(c2[nH]cc3c2CCC3)=O)CN(C(=O)C(F)(F)CO)CCC1(F)F C1(CNC(N(C)CC2CC2C)=O)C=CCC1 O=S(=O)(c1ccc(NCCF)cc1Br)NC(c1ccc(F)cc1F)c1nncs1 C(=O)(C(O)CCC(C)C)NCC1C(N(C)C)CN(C(C2COCOC2)=O)C1 C1(OC)CCCCC1C(N1CCC1CNC(c1nc(=O)n(C)[nH]1)=O)=O Cn1cc(-c2nnc(CO)o2)c(Oc2ccccc2)n1 c1(C(N2CC(N(C)C(c3cccnc3)=O)C3(C2)CC3)=O)cccc([N+](=O)[O-])c1 CCCCC(C)(c1nnnn1CCOC)NCc1nnc(C)o1 C1(CC(=O)NC(C2CCN(C(C3(C(C)(C)C)CCC3)=O)CC2)C)CCC(=O)NC1 Cc1n[nH]c(=NC2CC(F)(CNC(=O)C=Cc3ccc(F)nc3)C2)s1 C1(NC(C2CCCN(C(c3ccc(C(=O)OC)s3)=O)C2)=O)CCNC(=O)CC1 c1(C(=O)OC)cccc2[nH]c(CNC(=O)CC3CC(C(=O)OC)C3)cc12 c1(C(N2C(C)CC(NC(c3c(C)c(N)n(C)n3)=O)C2)=O)ccc2cncn2c1C c1(C(=O)NCC2CC(F)CN2C(c2cc(Br)n[nH]2)=O)csc2ccncc12 C1(C(=O)NCCC(C)(C)NC(c2cc(C(C)(C)C)ccn2)=O)CCC2C1C2(F)F C1(C)(CC(N2CCC(COC)C2)=O)CCN(C(=O)CCC=C(C)C)C1 C1(OC)C(NC(C2(CNC(=O)Cn3cncn3)CC=CC2)=O)CC12CCC2 N1(C(CCCOCC)=O)CC2(CCCCN(C(C3(Cl)CC3(F)F)=O)C2)C1 CC(C)(C(=O)N1CCC(NC(c2cnn(C(F)(F)F)c2)=O)C(CO)C1)S(C)(=O)=O N1(C(C2CC(=C)C2)=O)CCC2CCN(C(c3csc(C(F)(F)F)c3)=O)C2C1 C1(CCN(C)Cc2cnc(Br)c(N)n2)CN(C(=O)OC(C)(C)C)CCS1(=O)=O CC1(C)CC(=O)NC1CNC(C1(C)CCN(C(c2c[nH][nH]c2=N)=O)C1)=O CC1CCCC=C1C(=O)NC1C=CCN(C(c2ccc(F)o2)=O)C1 C1(CN(C(=O)Cc2ccccc2C2CC2)C)CCCCN1C(=O)C(F)C1CCC1 C1(NC(CC2N(C(c3c(C)n(C)cn3)=O)CCCC2)=O)CC1C1CCCC1 C1(C(=O)Nc2cnn(C3CCCCC3)c2)(CC)CCNC1 N1(C(COCCC=C)=O)CCCC(CCC)(NC(c2cccn2C)=O)C1 n1(CC2C(CC)C2)c(N2CC3CC2C3)nnc1C(C)C C1(NC(C(=O)NC(C)Cc2ccncc2)=O)CCCN(Cc2cccc(F)c2)C1 Cc1sc(C)c(C(=O)NCC2(C)CCC(NC(c3cnc(N(C)C)s3)=O)C2)c1C#N C(=O)(C(F)(F)c1cscc1Br)NC(C)CNC(C1(C)CCC1)=O C=CC(F)(F)C(=O)NCCC(C)NC(C1C(CN=[N+]=[N-])C1(C)C)=O Cn1cncc1CC(=O)NC1CCCC1NC(C1CSCCS1)=O N1(C(C(C)=C(CC)C)=O)CC(OCC)C(NC(=O)CNC(=O)C(C)(C)C)C1 Cc1ccc(CCC(N2CC3CC3(NC(C34CCC3C4)=O)C2)=O)cc1Cl c1(CC(=O)NC2CC(C(F)F)C2)ccc(Cl)cc1S(=O)(=O)N.CF CCC(F)(F)CC(=O)N1CCSCC1CCNC(c1ccc(OC(C)C)cn1)=O C1(C)(NC(C(CCSC)NC(COCCOCC)=O)=O)CN2CCC1CC2 c1(OC(CC)C(=O)NC(C)(C)C(C)NC(=O)C(C)NC(=O)NC)cccc(C)c1 c12ccc3c(c1)n(CCC#N)c(=O)n3CC2.C=CCSC.CC=C c1(NC(N2C(C)(CNC(=O)OC(C)(C)C)CC2)=O)ccc(-c2nn[nH]n2)cc1 N1(C(c2c(C)nc(COC)s2)=O)CCN(C(=O)CC(C)SC)CC1CO C1C(OCC)CC2C(CCC(CCC(=O)NC)C(=O)N)(CC(=O)N2)C1 N1(C(c2conc2C2CC2)=O)CCN(C(C2(C(F)F)CCC2)=O)CC1CO C1(C)(C(N2CC(n3cc(C(C)(C)NC(C4CC(O)C4)=O)nn3)C2)=O)COCCO1 N1(C(C2(C=C)CCN(C(=O)Cn3cccc3)C2)=O)CCCC(C)(C)CC1 C(C(N=c1cc(Oc2ccc3c(c2)CC3)n(C)[nH]1)c1nnnn1C)(OC)OC c1(C(=O)NCC(CCCC)NC(=O)C(C(C)C)NC=O)nc(C)c(C)nc1C C1(CC)CN(C(=O)COC(C)(C)C)CC1C(=O)NCCc1noc(C)n1 CC1CCC(NC(=O)CC2(C(F)(F)F)CCC2)CN1C(C1CCCN1C(N)=O)=O Cc1c(-c2noc(-c3cc(-c4ccco4)on3)n2)oc2ccccc12 C#CCCC(O)C(=O)NC1(CNC(c2cc(C(=O)C(F)(F)F)c[nH]2)=O)CCOC1 c1(C(C)C(=O)NC2(CNC(C3CSCN3C)=O)CCCCC2)ccc(F)cc1 c1(C(N2C(C)CC(CNC(c3cccc(OC)n3)=O)C2)=O)ncc(Cl)cc1Cl C#CC1CCC(C(=O)NC2CN(C(C3OCCC3C)=O)CC2(C)C)CC1 N1(C(c2c(C)[nH]c(=N)s2)=O)CC(NC(C2CCCN2C(N)=O)=O)CC(C)(C)C1 c1(OC)nccc(C(=O)NC23CC(NC(=O)C(C)CC(F)F)(C2)C3)c1F c1(C(C)C)ccc(C(=O)NCC2CN(C(=O)C(C)OCCN(C)C)CCO2)cc1 C1(CC)(CC)CN(C(=O)C(n2cc(-c3ncc(C)cc3C)nn2)C)CCS1(=O)=O C1(CNC(c2c(OC)nsc2)=O)N(C(C2CC2F)=O)CCCC1(C)C C=CCC(CC(C)C)C(=O)N1CCCC1(C)C(=O)N(C1CCC1C)C c1(CNC(c2n(C)ccc2)=O)nc(CNC(C2C(C3CC3)C2(F)F)=O)cc(O)n1 Cc1cc(C)c(C(c2nnnn2C2CC2)NC2CCn3nnnc3C2)c(C)c1Br N1(C(=O)CCC2CC2C2CC2)CC2(CCCCN2C(=O)COC)C1.C1(O)CCCOC1 Cc1cc(CN(C=O)Cc2ccc(O)c(Br)c2)ccc1N(C)C Cc1ccc(C)c(CC(=O)NC(C2CCCCN2C(=O)C(C)OCC2CC2)C)c1 N1(C(c2nc(OC)c(C)s2)=O)CCc2sc(CNC(c3ncoc3C)=O)nc2C1 c1(C(=O)NCC(C)(C(C)C)NC(C(C)SC)=O)cccn2nnnc12 c1(C(N2CC(O)(C(C(=O)N(C3CCCOC3)CC)F)C2)=O)cccc(NC)n1 c1(C(=O)NCC2(OC)CCN(C(c3cncs3)=O)C2)cc2c(F)cc(F)cc2[nH]1 C=CC(C)(CC)C(=O)NCc1cn(C2CN(C(=O)CSCC(N)=O)C2)nn1 N1(C(CNC(=O)OCC=C)=O)CCC(NC(C2CCCCN2N=O)=O)C(C)C1 C1(C(=O)NCCC2CCN(C(C(COC)N(C)C)=O)CC2)CCCCCN1C c1(C(=O)OC)ccc(C)nc1NC1CCN(C(c2cc(C)cs2)=O)C1C CC1CCCCN1C(=O)C=CC(C)NC(=O)C(CO)N(C)C N1(C(CN(CC)CC)=O)CC(NC(C2CCC2C(=O)OC)=O)CC(C)C1 C#Cc1cccc(C(=O)NCCCCN(C(=O)C(C)(C)CO)C)c1Cl c1(CNC(C(C)(C2CC2)OC)=O)ccccc1CN(C)C(c1c(C)cnn1C)=O Cc1cnncc1SC(N1CCOCC1c1ccccc1Cc1ccccc1)=O c1(C(N2C(C)CCN(C(=O)C(F)OC(F)(F)F)CC2)=O)c[nH]c2cc(F)ccc12 Cc1nc2ccccn2c1CC(=O)NCC(C)NC(=O)C(C)C(C)(F)F N1(C(CCS(C)(=O)=O)=O)CCC2CCN(C(C3CCCC3O)=O)CC12 c1(C(=O)NC2(C)CCCN(C(C3C(CC)CCC3)=O)C2)cccc2ccncc12 c1(CC)cc(C(=O)NC2CC(CO)N(C(C3CCC(=O)O3)=O)C2)ncn1 Cc1ccc(-c2nc(C)c(C(C)NC(C)C(=O)OC(C)(C)C)s2)cc1 c1(C(=O)NC(C2CCN(C(C(C)SC)=O)C2)(C)C)cc(Cl)c(F)c(Cl)c1 CC1CN(S(=O)(=O)N2CCN(Cc3n[nH]c4cc([N+](=O)[O-])ccc34)CC2)CC(C)O1 C12(C(=O)NCC3C(CC)CCN3C(=O)CC(F)(F)F)CCCC(CO1)C2 C1(C2CCC2)(CNC(C=Cc2cn(C)nc2)=O)CCN(C(c2cscn2)=O)CC1 C12(CN(C(C(c3ccc(C(=O)O)cc3)C)=O)C3CC3)CCCC1OCC2 Cc1nn(C2CC2)c(C)c1S(=O)(=O)NC(C1(C)Cc2ccccc2C1)=O C1(n2cc(-c3ccc(C(=O)OCC)o3)nn2)CCN(S(=O)(=O)CC(C)C)CC1 N1(C(C2CC(=O)NC2)=O)CCC2CCCC12C(=O)NCC(O)C1(Cl)CC1 C1(C(N2CC(CNC(c3cn(CCC)nc3C)=O)C2)=O)CCc2[nH]nc(O)c2C1 c1(OC)ccc(CN(C(=O)C(n2cc(C(O)CC(C)C)nn2)C)C)cc1O c1(C(=O)NC2CC3(C(C(=O)NC(C(=O)OCC)C)C3)C2)cnc(C)nc1C C1(NC(C2(OC)CCCC2)=O)C2CN(C(c3ccc(C(C)C)nc3)=O)CC12 N1(C(c2scc(C(=O)OCC)n2)=O)CCC(C(=O)NC2C3CCCCC23)CC1 c1(C(=O)NCC2C(NC(C)=O)CCC2)ccc(-c2cncnc2)cc1F c1(C(=O)NCC(N(C(C(C2CCC(=O)N2)C)=O)C)C2CC2)cncc2[nH]ccc12 C(=O)(CCS(C)(=O)=O)NC(C)C(C)NC(=O)C(F)(F)c1ccsc1Cl C(=O)(C(CC(=O)O)n1cc(-c2cn(CCC)nc2)nn1)OC.N12CCOC(C1)C2 C1(C(N2CCC(NC(CCC3CC(C)C3)=O)CC2)=O)CC(O)c2ccccc2O1 c1(C(=O)NC2CCC(N(C)C(c3sccc3F)=O)CC2)c(Cl)nn(C)c1Cl c1(NC(C2(C)N(C(c3c(C)ccc(OC)c3)=O)CCC2)=O)ccc2scnc2c1 n1(CC(=O)NCCCN(C(=O)OC)C)nccn1.C1C(=O)N1 C1(NC(CN2CCN(C)CC2)=O)CCN(C(=O)Cc2cccc(Cl)c2)C12CC2 Cc1ccc(C(N2CCN(C(C3CCC(C)(C)CC3)=O)C3CC23)=O)cc1O O=S1(=O)CCC(NC(=NCC2CC23CCSC3)NC2CCOCC2)C1 Cc1ccccc1NC(=O)NCCNC(=O)CCC1CCCN1 C1(CC(C)NC(=O)C#CC2CC2)CCN(C(=O)C2CC2)CC1 c1(NC(=O)CC2CCCN(C(=O)CC3CCOC3=O)C2)cccc(F)c1F CCC(C(=O)NC1CC(CCNC(=O)CCc2cncn2C)C1)OC C12(NC(c3c(Cl)cncc3Cl)=O)CCCC1N(C(=O)CC1CC1)CCC2 c1(C(N2CC3C(CCNC(C=CC)=O)(CC3)C2)=O)cc(C)c(Cl)c(C)c1 C1(C(N2C(C(=O)Nc3cc(O)nc(O)n3)CC(O)C2)=O)CCc2nc[nH]c2C1 c1(N2CC3(C(NC(C4CC45CC5)=O)CCS3)C2)c(Cl)cncc1[N+](=O)[O-] CC1CN(C(=O)CC2CCCC2)CCC1C(N1CCCC1)=O.C1(=O)CCCCN1 N1(C(C2C(CC)N(C(=O)Cn3cccc3)CC2)=O)CC(O)CC1(C)C C(=O)(C(=O)C(F)(F)F)NCCC1CCN(C(C(C)CC2CCC2)=O)CC1 c1(C(N2C(C)C(NC(c3n[nH]cc3Cl)=O)CCC2)=O)cc([N+](=O)[O-])ccc1O c1(C(=O)NCCCN(C(=O)Cn2cnnn2)CC)cnn(CCC(F)(F)F)c1 C1(C(=O)NC2(C(F)(F)F)CS(=O)(=O)C2)CCn2c(O)nnc2C1 C1(NC(c2nnc(C)s2)=O)CCCC2CN(C(=O)C(c3ccccc3Cl)C)CC12 C12(C(=O)NC(C3CN(C(c4c(OC)nccc4)=O)C3)C)CC3CC(C(=O)N1)C2C3 c1(NC(=O)NC(C)(CN)C2CC2)ccc2cccnc2c1 N1(C(=O)CC23CCCCC2C3(F)F)CC(N=c2[nH]c3cccc(F)c3o2)C1 C1(C(=O)NC(C)(C)CCNC(c2csc3nnsc23)=O)COCC2(CCC2)O1 C#CC1(O)CCN(C(C2CC(F)(F)CN2C(c2coc(C)c2)=O)=O)C1 c1(C(=O)OC)ccc(NCCCNC(=O)CC2CC3(CCC3)CO2)c([N+](=O)[O-])c1 c1(C(=O)NC(CC)(C)CNC(C2CC2COC)=O)ccc(F)c(C)c1C#N N1(C(c2ccc(C#C)o2)=O)CC(F)(F)CC1C(=O)NC1(C)C(C)(C)C1(C)C c1(C(=O)NC(C)C(CO)NC(=O)CCS(C)(=O)=O)cccc2[nH]nc(O)c12 c1(C(C)NCCC2CC(=O)N(C)C2)cc(Cl)ccc1OC(F)F CC(C)CCCC(C)NC(c1cnn(CCNC(c2cnco2)=O)c1)=O c1(C(N2C(C)CC(O)C2)=O)ncc(Cl)cc1C(=O)O O=C1NCC2(CCN(C(=O)CC3(NC(C4CC(O)C4)=O)CCCCC3)C2)O1 N1(C(C2(C)C(C)C2)=O)CCCC(CCCCNC(=O)CC2(C)CCCC2)C1 C1(CNC(C2=CCC(C)CC2)=O)CN(C(c2cc(Cl)cn2C)=O)C2COCC2O1 N#Cc1cn(CC(N2CCCC23CCN(C(=O)C2=CCCC2)C3)=O)c(=O)nc1O c1(C(N2CCC(C(=O)NC)C2)C(=O)NC2(C)CC2)cc(Cl)ccc1C C(=O)(C(C)C(F)(F)C(F)F)N1CCC(CNC(C2(CC)CCOCC2)=O)C1 C1(NC(c2c(CC)nns2)=O)CCN(C(C2(N=[N+]=[N-])CC2)=O)CC1CC N1(C(CCCC=C)=O)CC(C)CCC1CNC(=O)Cc1cnc(COC)nc1O c1(CNC(COCC(=C)C)=O)cn(C2CN(C(=O)CCc3ccncc3)C2)nn1 c1(C(C)OCC)nc(C(=O)NC2(C)CC(NC(c3snnc3C)=O)C2)cs1 C(c1ccc(C(=O)OCC(=O)NC2C3CCC(O3)C2N)cc1)=CC(=O)OC c1(C(=O)NC(CNC(C(C)NC(C2CCCC2)=O)=O)C2CC2)ncc(F)cc1N C(=O)(CS(=O)(=O)CC(=O)NCC12CN(C(=O)Cn3cccn3)CC1CCO2)OC N1(C(Cc2cnc(C)[nH]2)=O)CCCC(C)C1CNC(=O)CCc1ccn(C)n1 C1(NC(c2n(CC)ccn2)=O)C(CNC(=O)C(C)=CC2CC2)CCC12CCC2 c1(OC)sc(C(=O)NCCCCN(C)C(c2cc[nH]c(=N)c2)=O)cc1Br N1(C(c2[nH]cc(C(C)=O)c2)=O)CCCCC(N(C(=O)C(C)NC=O)C)C1 c1(C(=O)NCc2c(C)cccc2)csc2c1CCN(C(=O)C(C)(C)F)C2 C1(NC(c2nc[nH]c2C(F)(F)F)=O)CCCCCN(C(C2CC2F)=O)C1 c1(C(=O)NCC(C)CNC(=O)COCc2nc[nH]n2)ccc(F)c(N)c1 c12ncccc1C(=O)NCC1(O)CC(C1)CNC2=O.C1(COC)CC1.C(C)=O N1(c2nc(=NC)[nH]c(=NCc3ncc(C)cn3)[nH]2)CCOc2ccc(Br)cc2C1 N1(C(CNS(C)(=O)=O)=O)CCOC2(CCCN(C(C3CCC=CO3)=O)C2)C1 Cc1cc(=NC(=O)C2CCN(C(c3cc(Br)cc(I)c3)=O)CC2O)[nH]c(Cl)n1 Cc1ncc(CCC(=O)NC2(CNC(C3CCCN3C3CCCC3)=O)CC2)s1 C(=O)(CCC1=CCCCC1)N1CC(C#C)(C(N2CCc3c[nH]nc3C2)=O)C1 C(CCCCC(=O)NC1CN(C(=O)Cc2nccn2C)CC1(C)C)NC(C)=O S(=O)(=O)(c1ccc(C#N)cc1Cl)N1CC2C(CNC(C)=O)(C2)C1 c1(C(=O)NC(CC)CNC(=O)C=C(Cl)Cl)ccc(C(=O)CF)cc1 CC1C(C)N(C(c2cc(Cl)cc(Cl)c2OC(F)F)=O)CCN1C(=O)C=C1CCC1 C1(N(C(=O)CC2(OC)CCC2)CC)CN(C(c2cc(=O)cc[nH]2)=O)CC12CC2 C1(CNC(c2c(OC)nsc2)=O)COCCN1C(=O)CC(C)c1ccco1 N1(C(CC2C(C)CCC2)=O)CCCC2(CCN(C(=O)CS)CC2)C1 c1(OC)ccc(O)cc1C(N1CC(O)(C(C)NC(c2csc(Cl)c2Cl)=O)C1)=O c1(N2CCC(CNC(c3cc(CC)cc(F)c3)=O)C2)ccc([N+](=O)[O-])cc1F CCC(CN(C)C)CC(=O)NCC1C2CN(C(c3ccnc(Cl)c3OC)=O)CC12 C(C(C(=O)NCCC(F)F)NC(=O)Cn1ccnc1C)SCC C1(C(=O)NC2(CC=C)CCN(c3nnc(C(N)=O)s3)C2)CCC(C)(C)CC1 N1(C(C2CC(OCC)C2)=O)CC2CN(C(c3ccc(O)cc3)=O)CCC2(CO)C1 CC(C(=O)NCC1CC2CCC1N2C(c1cc(C(F)F)ccc1F)=O)C(C)(F)F C(=O)(C(C)CC(F)F)N1CCC(CN(C(=O)C(C)Cc2ccccc2)CC)CC1 N1(C(C(C)=C(C)C)=O)CCN(C(C2OCCC2C(F)(F)F)=O)C(CS(C)(=O)=O)C1 c1(C(N2CCC(C)(CNC(C(c3ccc(C)cc3)=O)=O)C2)=O)ccc(F)cc1C c1(CC(=O)NCCCN2CCN(C(C)C)CC2)ccc(C#N)cc1 C1(OC)COCC1n1cc(C(=O)NCCCNC(c2ccnn2C)=O)nn1 c1(C(=O)NCC(C)CNC(c2cn(C)c(O)n2)=O)cc(Cl)cc(F)c1N Cc1cc2c(C(N3CCCC(CO)(NC(c4cnns4)=O)C3)=O)ccc(C)c2[nH]1 C1(C(N2CC(NC(CC3(C)CC3)=O)(CO)C2)=O)COC2(CCC2)C1 c1(C(N(C(C)CNC(=O)CSC2CC2)CC)=O)ccc2nc(O)[nH]c2c1 c1(CNC(CC=CC=C)=O)nocc1C(=O)NC(C)CC(N)=O C1(C(=O)NCCCC(C)NC(c2ncc(Cl)nc2Cl)=O)CCCC(F)(F)C1 N1(C(C2(C)CCCN2C(c2cc(Br)cnc2F)=O)=O)CCC(O)C(C)(CO)C1 C1(CC(=O)NC2(CNC(c3cnn(C)c3N)=O)CCC2)CCC(C)(C)CO1 c1(C(=O)OC)ccc(C#N)c(N2CCC(NC(=O)C=C(C)C(C)(C)C)C2)n1 N1(C(C2(COC)COC2)=O)CCC(CO)C(NC(=O)C=CC2CCCN2C)C1 CS(=O)CCC(O)C(=O)N1CCC(NC(=O)Cn2nnc3ccccc23)CC1 N1(C(c2c(C)ccs2)=O)CC(CNC(c2cc(CO)c(C)o2)=O)C2(CCC2)C1 CS(=O)(=O)c1cccc(Cl)c1C(=O)NCC1CCN(C(C2CC3C=CC2C3)=O)C1 CC1(NC(=O)OCc2cnn(C(F)(F)F)c2)CCNC1=O C1(C)(C(=O)NCC2C(CC)CN(C(c3cc(C)ns3)=O)CC2)CC(C)OC(C)C1 C1(C(=O)NCC2(C3CC3)CCCO2)CC=CCC1C(=O)Nc1cncs1 N1(C(=O)C=Cc2cccc(F)c2)CCN(C(=O)CN2CC=CC2)CC(CO)C1 C(=O)(CCCCCC#N)N(C(c1ccccc1)CNC(C1CC=CCO1)=O)C c1(C(N(C2CN(C(C3CCSCC3)=O)C2)C)=O)cccc(Cn2ccnn2)c1 Cc1nc(C(=O)N(CC(O)CNC(=O)CCNc2ccccc2)C)cs1 c1(C(=O)NCC2CC(NC(C=CC(=O)NC)=O)C2(C)C)cc(Br)c2c(c1)OCO2 C1(C(=O)NC(C(=O)NC2CCC=CCCC2)CC2CC2)Cc2ccccc2C1 O=C(C(O)C(F)(F)F)NCc1cccc(-c2cc[nH]n2)c1 N1(C(C(c2ccco2)NC(CC=CCC)=O)=O)CCCC(CCO)CC1 Cc1noc2ccc(N3CCC(NC(=O)NCCC4CC(=O)N(C)C4)CC3)cc12 C1(OC)CCCC1C(=O)NCC(C)N(C)C(C1CC(C)(C)C1)=O c1(C(C(=O)NCC(=C)C)N(C)CCC2(C)OCCO2)nc(Br)cs1 C1(CNC(C2CC(OCC)C2)=O)COC2COCC12.C12(C)CCCN1C2=O CC1(C)c2ccccc2NC1C(=O)Nc1cnc2ccc(Br)cc2n1 C(=O)(CCS(=O)(=O)NC)N(CC(C)NC(=O)C1=CCCSC1)C.C(C(N)=O)NCC#N CCC(C)C(O)C(=O)Nc1cccc(NC(=O)CN2CCCC2)c1 c1(NC(C2CCN(Cc3c(C(=O)OC)cccn3)C2)=O)cc(F)c(Cl)cc1F Cc1nc(C(C)(C)C)nc(O)c1C(=O)NCCCCC(C)NC(=O)CC(F)F Cc1nc2c([nH]1)CC(NC(c1c(I)ncn1C)c1nnnn1CCCF)CC2 Cc1c[nH]c(C(=O)NCCC2(C(=O)NC3CC(CC(N)=O)C3)CCCO2)c1C c1(C(N2CC3(CC(C(=O)Nc4c(SC)cccc4)C3)C2)=O)cc(Br)cc(Cl)c1F C(C)(C(CC(=O)N(C1CCN(C(C)C)C1)C)NC(C1CCOC1C)=O)OC N1(C(COC(CC)(C)C)=O)CC(N(C(=O)CN2CCC(O)CC2)C)C(O)C1 C(=O)(CCC(N)=O)NCC1(NC(c2n(COC)ncc2)=O)CCOC1 N1(C(C2(SC)CCC2)=O)CCC(C2CCN(C(c3cc4scc(C)c4[nH]3)=O)C2)C1 c1(C(=O)OC)ccc2c(c1)C(NC(=O)NC(C)C(=O)N(C)C1CC1)CC2 N1(C(c2c(OC)scc2)=O)CC2(NC(C3OCCC3C)=O)CCCC2(F)C1 C1(CN(C(=O)C(N2CCCC(F)CC2)=O)C2CC2)CCC2(CCCCCC2)O1 N1(C(c2c(Cl)cn(CC)n2)=O)CCC(C2CCN(C(=O)C3=COCCC3)CC2)C1 CS(=O)c1ccc(CC(=O)NC2CC(NC(c3ccc(N)c(Cl)c3O)=O)C2)cc1 C=C(F)C1(CC(N2CCN(CCNC(=O)CSc3n[nH]c(O)n3)CC2)=O)CCC1 C(=O)(C=C1SCC(=O)N1C)N1C(COC)(CNC(=O)C2=CC3CCCC23)CCC1 c1(OCCC(=O)NCCCCNC(c2ccc(C)cn2)=O)ccccc1[N+](=O)[O-] N1(C(C(C(C)C)F)=O)CC(NC(=O)C=CSCc2ccco2)CC1(C)C c1(CC(=O)N(CC(CNC(C(CC)C)=O)(C)C)C)c[nH]c2cc(F)ccc12 c1(CCC(=O)NCC2CC(CNC(C=CCCC)=O)OC2)ccc(O)cc1 C1(C)(C(=O)NCC(n2cc(C3(C)CCCC3)nn2)C)CCCS1 N1(C(=O)C=CC2CCCCCC2)CC2CCN(C(C3C=CCS3)=O)C2C1 Cc1cc(C(=O)NC2(C(=O)N(C3CCN(C4CC4)C3)C)CC(F)C2)sc1C c1(CCc2c(C)c(N3CCC(C4CCCC4)C3)ncn2)ccc2oc(=O)n(C)c2c1 c1(C(=O)NCCCOCCCNC(C(C(C)(C)O)F)=O)cn2cccnc2n1 Cc1cc(C(=O)NCC(C)CC(=O)NC2CC3CC3C2)nc(O)c1 n1(CCC(=O)NCC(C)NC(=O)CC2CCC3CC23)cc([N+](=O)[O-])cn1 N(C(=NCCC(C)C)NCc1ccnc(N2CC=CC2)c1)CC1CCC(=C)CC1 c1(C(N2C(CNC(c3ccc(=N)[nH]n3)=O)CC(OC)C2)=O)cc(C)c(C)c(F)c1 C=CCCCCCC(=O)N1CCN(C(=O)COCCOCCOC)CC(O)C1 N1(CCCCn2cc(C(=O)NC(CNC(CN(C)C)=O)=O)nn2)CC2CCC1C2 N1(C(C(c2cccc(C)c2)O)=O)C2CCC1CC(O)(CNC(=O)CCF)C2 c1(OC)ccccc1CC(=O)NCC(CO)NC(=O)COCP(C)(C)=O C1(C)(OCC)CCCN(C(=O)CCC(c2nn[nH]n2)NC(c2ccc(C)cc2)=O)C1 C1(C(=O)NC2(CC)CCN(C(C3CC34CCC4)=O)CC2)CCCCN1S(N)(=O)=O CC1=C(C)CC(C)(NC(C2(C(C)NC(c3cc(C(C)C)[nH]n3)=O)CC2)=O)CC1.CO C(=O)(CC(C)C(C)(C)C)N1CCC(C=C)(C(=O)NCC(c2cnc[nH]2)C)C1 C1(C2CCN(C(=O)Cc3cc[nH]c3)C2)(NC(c2cc(CCC)c(C)s2)=O)CC1 N(C(=NC)N1CCC(SC(C)(C)C)C1)Cc1[nH]nc(COCC)n1 C1(c2nnc(C(=O)OCCOCCOCC(C)C)o2)CN(C(C)(C)C)CC(C)O1 CC(C)CC(O)CC(=O)NC(C)(CNC(=O)C=CCO)Cn1cccn1 Cc1cc(F)sc1C(=O)NC(C)C(=O)NCC1CC12CCC2 CC(C)C(O)C(=O)N(CC(C)CNC(=O)Cc1ccc(SC2CC2)cc1)C C1(NC(=O)CN2CCCC2=O)CCN(C(c2ccc(F)cc2O)=O)C12CCC2 N1(C(C2C(C)C2C)=O)CCCC1CNC(=O)C(C)n1ccnc1 C1(c2ccc(C)cc2)NC(=O)N(CCC(=O)N(c2nnnn2C)C2CCC2)C1=O c1(C(N2CCN(C(C=CC=CC)=O)CC(O)C2)=O)ccnc2c1ccn2C c1(C(=O)NCCN(CC(C)O)C(=O)CC2C=CCC2)ccc(CCN(C)C)cc1 N1(C(c2cc(OC)c(O)c(Cl)c2)=O)CC(NC(C2(C)CC2)=O)CC12CCOCC2 CC1CCN(C(c2cccc3c2CCO3)=O)C(C)C1NC(c1nc(Cl)cs1)=O C1(C(=O)NCC(CNC(c2cc(C)c(Br)o2)=O)C)C2CCC1(C)C2(C)C c1(C(=O)NCC(CC)(CC)NC(c2cc(C)cc(C)n2)=O)cc(C)nc(Cl)c1N C1(c2nnnn2CCOCC2CC2)(Nc2c(CC)cns2)CCCC(C)C1 C=C(C)C(CC(=O)NCCOCCS)OCC.C(=O)(CS(=O)CC)N1CC(N)C1 CN(CCCC(=O)NCC1(C)CCCC1NC(c1cc2ccccc2o1)=O)N=O C1(CC=C)(C(=O)Nc2ccc(SC)nc2)CCCN(C(=O)C(O)C=CC)C1 CC(F)(F)C(F)C(=O)NCCCC1CN(C(C2CCC(CN=[N+]=[N-])C2)=O)CCO1 N1(C(C2CC(F)CN2C(c2cc(F)c(F)c(Cl)c2)=O)=O)Cc2ccc(F)cc2C1 C1(CC(=O)NCC(CC)NC(c2ccc(OC)c(C)c2)=O)CCCC2(CCC2)O1 c1(C(=O)NC23C(CN(C(C(C)(C)c4ccccc4)=O)C2)C3)cc(N)c(Cl)cn1 N1(C(C2(CC)CCC2)=O)CC(NC(c2cc(N)ccc2Cl)=O)C2(CC2)C1 N1(C(C2(CCNC(C(C)C)=O)CCCO2)=O)CCC(C)(CN(C)C)C1 C1(NC(CCC)=O)CCN(C(=O)CC2CC3(CCCC3)CO2)CC(O)C1 CC(CCN=c1ccc(Br)c(S(=O)(=O)CN(C)C)[nH]1)N(CC(O)C1CCC1)C O=C(C1=C2CCN=C2NC=C1)NCCN(C(C1CCCCC1)=O)Cc1cccs1 C1(C)(NC(CC2C(NC(C3(OCC)CC3)=O)CC2)=O)CCCC1O N(C1CCCc2occc21)C(c1cc(CNC(C(C=C=C)C)=O)sc1)=O N1(C(c2cc(C)[nH]c2)=O)CCCC(C(=O)NCCc2cc(C)ns2)CC1 C(=O)(C1=CCCN(C(=O)CC2C=NN(C)C2=O)C1)NCC(C#C)C(C)C C1(C(N(CCC(C)NC(c2sccc2Cl)=O)C)=O)Cc2c(F)cccc2O1 C1(C(F)F)(NC(C2CCCN2C(=O)Cc2ccc[nH]2)=O)CCCCC1 N1(C(COCCCC)=O)CCC(C2CC2)C1CNC(c1cncn1C(F)(F)F)=O Cc1c(C(F)(F)F)cc(C(N2CCN(C3CCOC3)CC2)=O)cc1[N+](=O)[O-] C1(NC(c2cc(C)sc2)=O)CCCN(C(C2CN(c3nnnn3C)C2)=O)CC1F Cc1cc(NC(=O)C(C)(C2CC2)N(C)C(c2ccc(F)cc2)=O)cnc1C c1(C(=O)NC2C(CNC(CCC(C)OC)=O)CC2)sc(C#N)cc1Cl N1(C(C(C)OCCOC)=O)CCCC(CO)(NC(=O)C(C)c2cccs2)C1 c1(N2CC3N(C)C(CC3)CC2)nc(=NCC23CCC(CO2)C3)[nH]c2ccsc12 c1(C(=O)OC)cnn(C(C)(C)C)c1Cl.C12COC(C1)CNC(=O)C(=O)N2 C1(C(CNC(COCCC#C)=O)(C)C)CCN(C(C2CCCC2OCC)=O)CC1 c1(C(=O)OCC)c(N2CCCC(NC(=O)CC3(O)CCCC3)C2)cc(C)nc1O CCCCC(=O)C(=O)N(CCCN(C(=O)C(C)c1cc[nH]n1)C)C N1(C(C2CC(SC)C2)=O)CC2CC(NC(=O)C(C)(O)C3CC3)C(C2)C1 c1(SCC(N2CCCC(CNC(C3(SC)CC3)=O)C2)=O)ccsc1[N+](=O)[O-] N1(C(c2cc(C)ncc2C)=O)CC2CCC1C(CNC(C1CC1F)=O)C2 C12(CN(c3cccn3C)CCNC(C)=O)CC3CC(C1)CC(O)(C3)C2 c1(CN2CC(C(=O)OC)C(C#N)C2)ccc2[nH]c(C(=O)NCCC#N)cc2c1 Cc1cc(C)c(C(=O)NCC2(NC(=O)CCOc3ccc(Cl)cc3)CCC2)s1 C1(c2cn(CCC3CN(C(C4OCC(C)C4)=O)C3)nn2)CCCC(F)(F)C1 CCC(CCC(=O)OCC)OC(=O)Cn1cc(F)ccc1=O N1(C(C=CC2N(C(c3c(CC)cnnc3)=O)CCC2)=O)CCCC(CCO)CC1 NS(=O)(=O)CCCC(=O)N1CCC(O)C(NC(=O)C(O)c2ccsc2)C1 CCC(CC(=O)N(CC(C)(C)NC(=O)CCC1(C)CCC(=O)N1)C)C1CC1 Cc1cn(C)nc1C(=O)NC1(C(=O)NC(C(N)=O)C2CCCC2)CC1C Cn1[nH]c(C2CCCN(C(=O)CCN3CCOCC3)C2)nc1=N N1(C(CC2(C)OCCO2)=O)CCC(CF)(NC(=O)Cc2cc(C3CC3)no2)C1 Cc1ccc(SCC(N2CCN(C(c3cn(C(C)C4CC4)nn3)=O)CC2)=O)cc1 Cc1cc(C(=O)NC(C)CC(C)NC(=O)Cn2ccsc2=N)c2c(c1)CCO2 CCC(C)C(O)C(C)C(=O)N1CCOC(CN(CC(=O)NC)C2CC2)C1 c1(CC)cccc2c(F)c(C(N3CC4C(NC(=O)C=C(Cl)Cl)C4C3)=O)[nH]c12 Cc1ccc(Cl)cc1C(=O)NC1(CNC(C2CCN(CC(C)C)C2)=O)CCCC1 N1(C(c2c(F)ccc(N)c2)=O)CCCC(C2CCCN(C(=O)C(F)(F)CO)C2)C1 c1(C(N2CC3C(NC(c4n(C(C)C)cnc4)=O)C3C2)=O)n[nH]c(C(C)C)c1[N+](=O)[O-] C=CCCC(C(=O)NCC(CC)(CC)OC)NC(=O)C(O)CC1CCCC1 c1(NCCC)ccc(C(=O)NC(C)C(C)NC(=O)C(C)SC)cc1[N+](=O)[O-] N1(C(CCCc2ncc(C)o2)=O)CCC(CNC(=O)CSCC(C)C)C(C)C1 C1(NC(c2ccc(SCCCN(OCC)CC)c(Br)c2)=O)CCCCC(F)(F)C1 c1(C(N2CCC(F)(CNC(C3(CO)CCC3)=O)C2)=O)cccnc1F C=CCCCC(C)(C)C(=O)N1CCC(C)N(C(=O)CC2CCS(=O)(=O)CC2)CC1 C1(C)(CCNC2C(CC)CCC2)COCCN(C(=O)Nc2cn(C3CC3)nn2)C1 c1(CC(=O)NCC2N(C(C(CSC)OC)=O)CCCC2)ccc2ccccc2c1 C(=O)(CC(F)(F)C(F)(F)F)NC(C1CCCN1C(=O)C1=CCOCC1)C C1(C(C)NC(c2ccc(C3CCCCC3)o2)=O)CN(C(=O)C2CC2)CCO1 CC(CS(C)(=O)=O)C(=O)N1CC(O)(CN(C)C(C2(CO)CCOCC2)=O)C1 c1(C(N(C2CC(NC(C3CC4(CSC4)C3)=O)C2)C)=O)nnc2ccccc2c1N C1(CNC(C(COCC)C)=O)CN(C(c2ccccc2OCC#N)=O)CCN1C c1(C(N2CC(NC(CC3(C)CC3(F)F)=O)C2)=O)ccc(C(=O)CF)cc1 c1(C(N2CCC(OCCNC(C(C)n3cncn3)=O)C2)=O)cc(C2CC2)nn1C c1(C(N(CC(C)N(C(=O)CC2CCN(C)C2=O)C)C)=O)cc2n(n1)CCC2 Cc1nc(N2CC3CCCC(NC(C4CC(C(C)C)C4)=O)C3C2)ccc1[N+](=O)[O-] N1(C(CN(C(C(C)C)=O)C)=O)CCC2CN(C(=O)CN3CCN(C)C(=O)C3)C2C1 C1(C2CC(=O)NC2)CC(NC(=O)COC2CC(F)(F)C2)CCO1 CC1(C)COCC1C(=O)NC1CN(C(=O)CC2CC3CCC(C2)C3)CC1O CCC(C)(CNC(C1CCC(=O)O1)=O)C(=O)N(C)Cc1nnc(C)o1 C1(CC(=O)NC(C2CN(C(C3C4CCC(=O)C34)=O)CCO2)C)CC2(CCC2)C1 c1(OC)cc(C(N2CCC(F)(CNC(=O)C=Cc3nc(C)co3)C2)=O)c(F)cn1 c1(OC)ccc(C2CCN(C(c3csc(-c4cccc(F)c4)n3)=O)CC2)nc1 CCC(CC(F)F)C(=O)NCC1CN(C(=O)CC(C)C(=O)OC)CC(C)(C)O1 C(CC(C)(C)CC(=O)N1CC(Nc2snc(C)c2C#N)C(C)(C)C1)OC C1(C(=O)NCCC2CC(NC(CC(C)O)=O)C2)CCC(C)(C)OC1 c1(CCC)nc(=NCC2(O)CCCN(C(=O)CC(=O)N(CC)CC)C2)s[nH]1 Cc1cc(C)c(C(=O)NCCC(C)N(C(=O)CCC(F)F)C)cc1N C1(CC(=O)NC(C=CC(=O)NC(COCCOC)C)C)NC(=O)NC1=O Cc1cccc(CC(=O)NC(C)CCNC(C2(S(C)(=O)=O)CC2)=O)c1Br Cc1ncc2n1CCC(C(=O)NC(C)C(C)(C)NC(=O)Cn1cnnn1)C2 N1(Cc2ccc(SC)s2)C2CCC1CC(NC(c1ccc(I)c(O)c1)=O)C2 c1(C(=O)NC2CC3CN(C(C(C)=CC)=O)CC32)cccc2[nH]nc(O)c12 N1(C(C(=Cc2cn[nH]c2)C)=O)CCOC(CCNC(=O)CC2CCC(=O)N2)C1 C(=O)(CCCCCC(=O)NCC1CC1NC(c1nc(OC)c(C)s1)=O)OCC C(CC(C(C)(C)C)NC(C1CC1c1ccco1)=O)N(C(C(C=C)(C)C)=O)C C(CCC)(C(=O)NC1CCC(OCC)C1)NC(CSCCCC)=O C(=O)(C1CCCc2n[nH]cc21)N(CC(C)CNC(=O)Cc1cccnc1Cl)C c1(C(N2CCN(Cc3c(C)nn(C)c3Cl)CC2CC#N)=O)nc2ccccn2n1 Cc1nc(C)c(C(=O)NCC(O)CN(C)C)o1.C(COCCOC)S c1(C(C)=O)ccc(NCC2CN(C(C3CC3(Cl)Cl)=O)CC2C)c([N+](=O)[O-])c1 C=CCC(CC)C(=O)OC.c12cc(cc(F)c1)NC(=O)C1CC13CC23 c1(OC)ncccc1N(C(=O)CSc1cccc[n+]1[O-])C c1(CCC(=O)NCC(CO)NC(CC=C(C)C)=O)cc(Br)cs1 CCC(C)C(O)CC(=O)N1CC(F)(CNC(=O)CNS(=O)(=O)c2cccnc2)C1 CC1(C(=O)NCC2(NC(=O)CN3CCS(=O)CC3)CC2)CCc2ccccc2C1 C(C(CC(C)C)C(=O)NCc1ccc(C(=O)NC(C2CCCO2)C)nc1)OC c1(C(=O)NC(CNC(Cc2c(C)n[nH]c2C)=O)CO)onc2ccccc12 N1(C(C(C)(C)CC2CC2)=O)CCC2(CC1)CC(Nc1snc(Cl)c1C#N)CO2 c1(CC(=O)NC2C=CCN(C(c3cc(O)ncn3)=O)C2)cc(F)cc(Br)c1 C(C(=O)N1CC(C2CC2)(OC)C1)(C(C)(C)C)NC(C(COCC)C)=O CC(CCC(=O)N1CCC(CNC(=O)Cc2cncnc2)C12CC2)S(C)(=O)=O C1(C)(CC)CN(C(c2[nH]cnc2C)C(=O)Nc2ccc(F)cc2C)CCO1 CCCC(C(=O)N1CCN(C2CCN(C(=O)Cn3cnccc3=O)C2)CC1)OC C1(CNC(CCCC(C)=O)=O)COC(C)(C)CN1C(=O)CC1CCOC1=O C(C(O)C(=O)NC(C)CC(=O)NCCc1ccon1)=CC N1(C(CCC2(NC(=O)CCc3ccsc3)CCC2)=O)CC(O)(C2CCC2)C1 C(=O)(C(CC1CCCC1)NC(=O)CC(C)C1CC1)NCCCNC(N)=O c1(OCc2cn(-c3ccc(OC)c(Br)c3)nn2)ccnc2ncnn12 N1(C(C2(OC)CCC2)=O)CC(CCNC(=O)C(O)Cn2cncn2)C(C)C1 N1(C(=O)CC2CCCO2)CCC(O)(C2(NC(C34CCCC3C4(F)F)=O)CC2)CC1 CC1(C)CCC(CNC(C2CC(C)(C)CN2C(c2cnn(C3CC3)c2)=O)=O)OC1 Cc1cnc(C(N2CCOCC2CNC(=O)CCS(C)(=O)=O)=O)c(C)c1 N1(C(C(COC)OC)=O)CCCC(CO)(NC(=O)Cc2cccnc2)C1 C1(NC(c2csc(Cl)c2Cl)=O)CC2CCC1CN(C(=O)C1CCc3c[nH]nc31)C2 N1(C(C(C2CCCCC2)C)=O)CC2CC(NC(c3ccc(Cl)s3)=O)CC1C2 c1(OC)cnc[nH]c1=NCC1(O)CCCN(C(c2ccccc2SCCO)=O)C1 C(=O)(C(C)(C)C(=O)N1CCCCC1CNC(c1csc(C)n1)=O)NC n1(CC(N2CC(N(C(C(C(C)C)C)=O)C)C(C)CC2)=O)nnc2ccccc12 Cc1cc2nc(NC(=O)Cn3cnc4sccc4c3=O)sc2cc1C O=C(C#CC1CCCO1)NCC1CCCN1C(c1scnc1C1CC1)=O c1(N(CCC(N)=O)C)nc(N2CCN3CCCC3C2)c2cccc(F)c2n1 n1(CC(=O)NCC2(F)CCC(NC(C(CCCC)O)=O)C2)ncc2ncccc12 N1(C(c2[nH]cc(C)c2)=O)CC(NC(C2CCCCS2)=O)CCC1C C(C(F)(F)C(F)(F)F)Oc1ccc(NC(C2CC(CO)CO2)=O)cc1 N1(C(c2c(C)cn(C)n2)=O)CC2CC1CCC2NC(=O)Cc1c[nH]nc1C Cc1cnc(C(N2CC(NC(C3CC4(CCC4)C3)=O)CC23CCC3)=O)cc1C#N N1(C(C(C)Cc2ccc(Br)cc2)=O)CCOC2C(C(=O)OC(C)(C)C)CC12 c1(CC(=O)NCCN(C(=O)C(C)CC2CCCO2)CC)nc2ncc(C)cn2n1 N1(c2ccnc(SC)n2)CCC2C(CCN2C(c2cccnc2F)=O)C1 NS(=O)(=O)CCc1cn(C2CCN(C(c3ccn(CC(F)F)n3)=O)C2)nn1 C1(NC(C(C)OC)=O)COC2(C1)CN(C(c1c(N)cccc1F)=O)C2 N1(C(CNC(CNC(C)=O)=O)=O)CCOC(CNC(C2(CO)CCOC2)=O)C1 C1(NC(c2c(NC)cncc2)=O)CCN(C(=O)C(F)(F)COC)CC1F c1(CCC(=O)NCCC2CCN(C(C3(F)CCOC3)=O)C2)ccc(F)cc1 c1(OC)ccc(-c2csc(C(=O)Nc3ncc(Br)cc3Br)c2)cc1OC C1(NC(C2C(=C)CC2)=O)CC2CC(NC(c3cnc(Cl)cc3N)=O)C1C2 C(=O)(C(C)C(C)COC)NCC1(F)CC(NC(c2cc(CCC)ncc2)=O)C1 Cn1cncc(C(N2CC=CC(NC(=O)CC3CC4CC4C3)C2)=O)c1=O Cc1cccc2c(N(C(=O)C=Cc3ccc(F)cc3)CC3CCNC3)ncnc12 C(=O)(CC1=CCCC1)N(C(C)CNC(=O)C(c1cc(Cl)ccc1F)(C)C)CC C1(N(C)C(c2ccc(C(F)F)s2)=O)CCCC(NC(c2ccccc2O)=O)C1 Cc1cc(C)nc(N2CC(NC(c3cn(CC4CCCO4)nn3)=O)CC2C)n1 N1(C(c2ncc(OC)c(Br)c2)C(=O)NC2CCCC2)CC2CC(O)C(O)CC2C1 C1(CNC(c2c(CCC)[nH]cc2)=O)CCN(C(c2c(C)nsc2C)=O)CC1C C1(NC(C(C)NS(C)(=O)=O)=O)C2CC3CN(C(C4CCCC4(C)C)=O)C1C3C2 c1(C(=O)NC2C(C)N(C(=O)CC3CC3(C)C)CC2)c(Cl)c([N+](=O)[O-])nn1C C1(NC(c2cc(Cl)no2)=O)CC2CC1CN2C(C1(C(c2ccccc2)=O)CC1)=O CCCCN=C(NCC(c1cccc(C)c1)O)NCC1(C)CCC(OC)CC1 C(=O)(C(CC(C)(C)C)NC(c1cc(O)n(C)n1)=O)NC1CN(C)C(=O)C1 C(C(=C)C1CCOCC1)NC(C1(C)N(C(C2C(C(=C)C)OCC2)=O)CC=C1)=O C1(N(C(=O)COCc2ccccn2)C)CN(C(=O)CN2CCSCC2)CC1(C)C C1(N=c2[nH]nc(CC)o2)(CCC)CCN(C(=O)C(C)C2CCCC2)CC1 C(CC1=CCCCC1)N(C(C1CCCN(C(CCSC)C(=O)O)CC1)=O)C c1(CC(=O)NC(C2CN(C(C(COC)(C)OC)=O)C2)C)cc(F)ccc1C C1(C(=O)NCC2(NC(C(C=C)O)=O)CC3CCC2CC3)Cc2c(C)cccc2O1 c1(C(N(C2CCN(C(c3ccc(CCC)s3)=O)CC2)C)=O)cc(C)c(O)c(C)c1 CN1C(=O)CCC1CC(=O)NCc1ncccc1C(N1CCC(C)(F)C1)=O c1(C(=O)NC2CC3(C(NC(C4CN(C)C(=O)N4)=O)C3)C2)[nH]nc([N+](=O)[O-])c1Cl C1(CC(=O)N(C)CC2CCCN(c3nnn(C)n3)C2)CCOC(C)(C)C1 C1(C(=O)NC(Cn2cc(C(C=C)(C)O)nn2)C)CC2(CCNCC2)CO1 Cc1cc(C(=O)NCC2CC2NC(=O)CC2(n3cncn3)CC2)cnc1C(F)F C1(NC(Cc2c(CC)cccc2)=O)CC2(CCCN(C(=O)C(C)C)C2)C1 C(C(C)N=c1nc2scnc2c(N2CCNC(=O)C2)[nH]1)(c1ccccc1F)OC C1(NC(C2CC2)=O)C(C)(C)C(O)C1(C)C.N1(C(C(C)OC)=O)CCC(CO)(CF)C1 C1(C2CCN(C(=O)CN3CC=CC3)C2)(NC(C=C(CCN(C)C)Cl)=O)CC1 C(=O)(CCCC(C)=O)N1C(C(=O)NCC2(F)CCCCC2)(COC)C=CC1 c1(OCC)cccc(C(=O)NC2CCC(CNC(=O)CNC=O)C2)c1N C1(NC(c2cnc(OCC)nc2)=O)CN(C(=O)CC(=O)OC(C)(C)C)C(C)(C)C1 C(C1=CCN(C(=O)CCCC(OC)OC2CCCC2C)CC1)OC c1(C(N2C(CC(=O)NCCC(CC)CO)CCCC2)=O)cccc(C#N)c1 C1(C(C)N(C)C(C2CC(CCNC(=O)CC(C3CC3)C3CC3)C2)=O)CCOCC1 CC1CN(C(=O)CCC2(C)CN(C(C3CCN(C)CC3)=O)C2)CC1(F)F CC1COc2c(C(=O)NC3CCCC3NC(=O)CCCC(N)=O)cccc21 CC1(C)C=C(C(=O)N2CC(NC(c3cc(-c4cccs4)[nH]n3)=O)CC(F)C2)C1 c1(C(N(CCN(C(=O)C(O)CSC)CC)CC)=O)sc2cccc(C)c2c1Cl C12(C(=O)NCCOCCCNC(c3nn(C)c(F)c3)=O)CCC(CC1)CC2 c1(C(N2CC(O)(CN(C(=O)CCCCO)C)C2)=O)coc2c1C(=O)NCCC2 C1(C(=O)NC2(CSC)CCC2)CCN(C(c2cnnc(O)c2)=O)CCO1 C1(OC)CC(CNC(C2CCN(S(C)(=O)=O)CC2)=O)N(C(=O)CC2CC(F)C2)C1 C1(C(N(C2CC(C(N)=O)C2)C)=O)CN(C(C2(C#N)CCCO2)=O)CCN1C c1(OC)cccc(CCC(=O)NC(C)CC(C)NC(c2ccsn2)=O)c1F N1(C(Cc2ccc(C)c(C)c2)=O)CCC2CN(C(c3nc(Br)cs3)=O)CC2C1 C1(C#N)(C(=O)NCC(C(=O)NCCCC#C)C)CC(=O)C1 c1(SC(C(=O)OC(CCC)C)C)ccc(Cl)cc1 C1(C)(NC(C(CNC(C2N(CC)CCC2)=O)N(C)C)=O)CC(C)(C)C1 C1(NC(CC2(C)N(C(c3cc(C)cc(O)n3)=O)CCC2)=O)CCn2nccc2C1 c1(C(=O)NCC(CC(C)C)NC(C(C(CC)O)C)=O)nc(N)cc2ccccc12 CC1(CNC(=O)Cc2cc[nH]n2)CN(C(=O)CNC(=O)CCCCO)CCO1 C1(NC(C2CCN(C)C2)=O)CN(C(c2cc(C(C)(C)C)on2)=O)CC2(CC2)C1 C1(C(=O)NCC(CSC)(C)C)C2CCC(C2)N1C(=O)C(C1CCCCC1)C c1(NC(C2CCC(NC(c3cccc4cc[nH]c34)=O)C2)=O)c(Cl)cc(Cl)cc1Br C#CCCCCCC(=O)NC(C1CCOC1)CNC(c1cc(F)ccc1CC)=O N1(C(c2c(C)c(Cl)ccn2)=O)CCC2(CCCCC2NC(c2cc(Cl)no2)=O)C1 N1(C(C2C=C(C)CS2)=O)CC(C(=O)Nc2cc(C)cc(O)c2)CCC1(C)C c1(N2CCCC(CSC)C2)nc(N(CCS(N)(=O)=O)C)nc2ccc(Cl)cc12 c1(CC(C(=O)O)NC(CC2C(C)(C)COCC2)=O)ccc([N+](=O)[O-])cc1F N1(C(CCc2nc(C)sc2)=O)CC(NC(=O)CCc2scnc2C)CC12CCC2 C1(NC(c2c(SC)ccs2)=O)CCN(C(C2(C)COCCO2)=O)CC1CO Cc1cc(C(N2CCOC(C(=O)NC(C)C#N)C2)=O)c(F)cc1F C1(SC)CN(C(=O)CC2(CO)CC2)CC1c1c(SCc2ccccc2)cccc1 c1(C(=O)NC2C(NC(C3(C(C)C)COC3)=O)C2)cccc(OC(F)F)c1 O=C(CCCC(=O)C1CC1)NCc1cc(C(=O)NCc2cncs2)on1 C1(C(=O)NC2CN(C(=O)CC3CNC(=O)O3)CC2CO)(CC)CCCC1O C#CCC(C)(C)C(=O)N1CC(CNC(c2ccccc2C(C)C)=O)C(O)C1 Cc1ccc(F)c(CC(N2CCC(C)(NC(C3CC34CC4(F)F)=O)CC2)=O)c1 c1(C(=O)NCCOCCNC(CC2(C)CCCO2)=O)cc(Cl)ccc1-n1cncn1 Cc1cc(C(=O)NCC2(CNC(c3cc(C)cnc3N)=O)CC2(F)F)c(C)cn1 CC#CCCCC(=O)NC(CC#CC)C(=O)NCCC(=O)NC(C)CC N1(C(c2cnc(C(C)O)s2)=O)CCOC(CN(C(=O)C=Cc2nccs2)C)C1 Nc1cc(F)cnc1C(N1CCN(C(=O)CSc2ccccn2)C(CCO)C1)=O C1(CSC)CN(C(=O)COC2CCCCC2)CCO1.C12CCCC1NC2=O CC1(C)CCCC(C(=O)NCC2CN(C(c3ccnc(F)c3N)=O)C2)CC1 C1(CNC(C2CCCO2)=O)(NC(c2cn(C3CCCC3)nn2)=O)CCOCC1 c1(C(CC)C)ccc(CNC(=O)CC(c2ccccc2)C)nc1 C(=O)(CCCNS(C)(=O)=O)NCCN(C(C(C)OC1CCCC1)=O)CC(C)O C1(CC=C)(C(=O)NCCCC)CN(C(=O)C(C)OCCOCCc2cnn[nH]2)C1 C(C)(C(=O)N1CC(NC(=O)C(C)(C)CO)CC(F)C1)(C(C)C)OC N1(C(C(C)OCCC#C)=O)CCC(CCCCNC(C2C3CC4C(C3)C24)=O)CC1 c12nc(cs1)C(=O)N(CC1CC1)CCN2.C(=O)(C(C)=C1CC1)C(C)=O CCC(C)C(C(=O)NCc1cncc(OC)c1C)N(C)C N1(C(CCOCCC)=O)CC(CNC(c2cncn2C)=O)C(C)(C)C1 Cc1cc(=O)oc(C)c1C(N1CC2CC1C2NC(C1CCC(C)(C)O1)=O)=O C1(O)(CNC(=O)CC(F)F)CCN(C(c2ccccc2-n2cncn2)=O)C1 C1(OC)CC2(C1)CN(C(=O)CNC(=O)C(F)CC1CCC1)C2 C(C(C)(C)CC(=O)NCC(CO)NC(c1cnc(C2OCCO2)s1)=O)OC(C)=O N1(C(C(C(C)C)(C)C)=O)CC(NC(=O)CC2(C)CCOCC2)CCC(O)C1 c1(OCCNC(=O)COC(F)(F)F)cc(OCF)cc(F)c1 c1(C(N(C2CCCN(C(c3cocn3)=O)CC2)CC)=O)nn(C)c2c1CCCC2 c1(C(=O)NCC2C(C)CCN2C(c2cnc(C(N)=O)cn2)=O)csc2nnsc12 N1(C(CC2CNC(=O)O2)=O)CCN(C(c2cccc3nccn23)=O)CC(O)C1 N1(C(c2n(COC)ncc2)=O)CC=C(C(C)(C)C(=O)N2CCC(F)(C#N)C2)C1 c1(SC)cc(C)c(C(=O)NCC(CC(C)C)NC(=O)Cn2nnc(=O)[nH]2)o1 N1(C(Cc2ncc(C)s2)=O)CCC(NC(C2CC23CC3)=O)C(O)C1 c1(C(=O)NCCCC(C)NC(C2=C(C)CCC2)=O)n[nH]c2c1CCSC2 C1(C(=O)NC2CCN(C(C(C)OCCOC)=O)CC2C)CCC(C2CC2)CC1 c1(SC)ccccc1C(N1CC(CCCCNC(C2CN(C)CCO2)=O)C1)=O N1(C(C2C(NC(C(C)=CC3CC3)=O)CCC2)=O)CCOC(C)(C(C)C)C1 Cc1cc([N+](=O)[O-])nn1C(C)C(=O)NCC(C(C)C)NC(c1cn[nH]c1)=O Cc1cccc2cc(C(=O)N(C)CC3CCCN3C(c3nnn(C)c3C)=O)sc12 CCC(O)C(=O)N1CCC(NC(c2ccc(C(F)(F)F)s2)=O)C1 c1(SC)ccc([N+](=O)[O-])c(NC(c2cn(CCC(C3CC3)N(C)C)nc2C)=O)c1 c1(CC)ccc(C)cc1NC(=O)C(O)C(C)(C)NC(=O)OC(C)(C)C N1(C(=O)COCCc2nccc(-c3ccccc3)n2)CCN(CC(O)CO)CC1 c1(CC(N2CC3CN(C(CC(CCC)O)=O)C3CC2)=O)c[nH]c2cccc(Cl)c12 C1(C(=O)NCCCC2CN(C(C3(F)CC3)=O)CCO2)CC2(C1)CC21CC1 C1(NC(C2C(C=C)C2)=O)(CNC(c2cnc(Cl)[nH]2)=O)CCOCC1 C1(CNC(c2ccc(Cl)nn2)=O)CCN(Cc2cc(Cl)c(O)cc2F)CC1(F)F C(=O)(C1=Cc2ccccc2C1)N1CC(C(=O)NCC(COC)(F)F)CC12CCC2 CC1C(C(=O)NCCC2CC2)CCCN1C(c1cc(F)cc(Cl)c1)C(=O)N(C)C C1(C(N2CCC3(CC3NC(=O)C(F)OC(F)(F)F)C2)=O)CCn2ccnc2C1 Cn1cc2c(n1)CC(C(=O)NC1CCC(CCNC(=O)CNC=O)C1)NC2=O CC(F)CC(=O)N1CCCC1C(=O)NCC1(C(C)O)CC1 c1(C(N(C2CCCOC2)CC)=O)ccn(CCNC(c2cnn[nH]2)=O)c1 CC1CCC2(CC1)CCC(CNC(C1CNC(=O)O1)c1nnnn1C(C)(C)C)O2 c1(C(=O)NCCCN(C(=O)C=Cc2ccc[nH]2)CC)cc2cccn2c(O)n1 C#CCC(C)C(=O)N(CCCNC(c1ccoc1I)=O)C c1(N2C(C(C)(C)NC(C(C)NC(COC)=O)=O)CCC2)nc(Cl)nc2[nH]cnc12 c1(CC)nocc1C(=O)NCC(CCNC(=O)Cc1ncoc1C)OC N1(CCNC(CCn2cc(-c3cccc(N)n3)nn2)=O)CC2COCC2C1 CC1(C)COCC1C(=O)NC1CC2(C1)CC2NC(C1CC1c1ccccc1)=O C1(NC(Cc2n(C)cnc2)=O)CCCN(C(=O)C(O)CC(F)F)CC1 CN1CCOc2ccc(-n3cc(CC4(C(=O)O)CCC(C(=O)O)CC4)nn3)cc21 c1(C(=O)NCCC2N(C(CN(C(=O)OC)C)=O)CCC2)cc(SC)oc1C CON=Cc1ccc(C(N2CCC(C)(NC(=O)C#CC3CCCO3)CC2)=O)cc1 C(=O)(C(CCOCCO)NC(C12CCCC1C2)=O)NC1CC(CCOC)C1 Nc1cc(C(=O)NC2CCC2NC(c2n[nH]cc2Cl)=O)c2ccccc2c1 N1(C(Cc2ccc(C)cc2)=O)CCC(NC(c2cc([N+](=O)[O-])c[nH]2)=O)C(C)C1 C1(C(=O)NCC2(C(N3C(CCC=C)CCC3)=O)CC23CCC3)CC(=O)CC(=O)N1 c1(OCCC)cccnc1CC(=O)NCCC1(O)CN(C(=O)CCC=C(C)C)C1 N1(C(C(CC)CC)=O)CC(NC(=O)NC2CCc3ccnn3C2)CC12CCC2 c1(C(=O)NC2C3CN(C(CC(C)SC)=O)CC2C3)ccc2[nH]c(C)c(C)c2c1 c1(C(=O)NCC2(C)N(C(=O)CCCN=[N+]=[N-])CC(OC)C2)cc(C)nc(Cl)c1N c1(CCC(=O)Nc2c(OCCNCC)cccc2)ccc(Cl)c(Cl)c1 CC(C)(C)S(=O)(=O)CC(=O)N1CC2CCC1CN2C(=O)CC1CCOC1=O N1(C(c2scc(C(N)=O)c2)=O)C2CCC1CC(CNC(=O)C(O)C(F)(F)F)C2 C1(O)(C(=O)NCCCNC(=O)Cc2cncs2)CCC(C(F)(F)F)CC1 c1(CN2CC(NC(CCC(C)C)=O)C(F)(F)C2)ccc2ccccc2n1 C1(NC(C2CC(C)(CC)C2)=O)CCN(C(c2ccc(C(N)=O)cc2)=O)CC1 C(CC(=O)N=c1ccn(C(C)C)[nH]1)C1(OC)CN(C(C(CCC)=CCC)=O)C1 CCC(C)(C(=O)N1CC2(CNC(=O)C(C)(C)C)CC1CO2)C(N)=O C12(NC(C(CC)=CCCC)=O)CCCC(CN(C(c3cnc(C4CC4)s3)=O)C1)C2 N1(C(C(C(C)C)NC(C)C)=O)CC2CCC1C(NC(C1(O)CC1)=O)C2 C=CC(C)CC(=O)NC(Cc1ccccc1Br)C(=O)NCC(=O)N(C)O c1(OC(C)C(=O)NCC(F)CNC(=O)CC2CC(=O)C2)ccc(Cl)cc1Cl C1(C(=O)NCC2CC(NC(=O)COCC3CC3)C2)CNC(=O)CC12CCOC2 C1(NC(c2c(CC)nco2)=O)CCN(C(=O)Cc2ccoc2)CC1C(C)C C(=O)(C(C)(C)C(=O)NCC(C)N(C(=O)CC1CC1(Cl)Cl)C)OCC C1(NC(C(c2ccnn2C)C)=O)CCC(NC(c2cn(C(C)(C)C)nn2)=O)CC1 n1(CC)cc(C(=O)NC2CC(CNC(C3CCC(OC(F)(F)F)C3)=O)C2)c(C)n1 CCC(CNC(=O)C(C(C)O)NC(=O)C=CC1CC1)C(C)(F)F c1(C(N2CCC(O)(CN(C(c3c(OC)noc3C)=O)C)C2)=O)cc(C)cc(C)c1 C(=O)(CS(=O)(=O)c1ccccc1C)NC1CC(NC(CC2CC(CC)OCC2)=O)C1 c1(CNC(C2C(C(N3CCN(CCCC)CC3)=O)C2)=O)ccnc2[nH]ccc12 C1(C(N2CC(CC=C)(NC(=O)C(CCC)=CCC)C2)=O)CCc2nnnn2CC1 Cc1nc2ccccc2cc1NC(C1CC12CN(C(c1cnc(Br)s1)=O)C2)=O CC(C)(O)C#CC(=O)NCCCNC(C1CC1(c1ccccc1F)C)=O C1(NC(C(Cc2ccc(C)cc2)C)=O)CCN(C(=O)CCc2ccco2)C(C)C1 C1(O)(C(=O)NC2(CCNC(c3cnn4c3CCCC4)=O)CC2)CN2CCC1CC2 c1(N2C(C(=O)Nc3nccc(SC)n3)CC(=C)C2)ncnc2n[nH]cc12 c1(OC)cc(C(=O)N(C)CC2(O)CN(C(=O)C(O)CN3CCCC3)C2)ccc1C N1(C(C(=O)NCCC)=O)CCC(OCC(=O)Nc2sccc2C)C1 N1(C(c2c(C)c[nH]n2)=O)CC2(CCCN(C(c3ccc(C(C)F)cc3)=O)C2)C1 N1(C(c2ccc(COC(C)C)cc2)=O)CCC(O)(CNC(=O)C(C)O)CC1 C1(CNC(C(C)N(C)C)=O)CCN(C(=O)C(CO)N(C)C)C(C)C1 N1(C(c2ncc(OC)nc2)=O)CCCCC(C(=O)NC(C)C(C)SC)C1 C1(NC(CC(=C)C)=O)CCN(C)C12CCCN(c1ncnc3sccc13)C2 C1(NC(C(C(C)C)CO)=O)CN(C(c2ccc(=O)n(C3CC3)c2)=O)CC2(CCC2)C1 NC(=O)CCCCC(=O)N1CCC2(CC1)CC2NC(c1ccc(=O)oc1)=O C(=O)(C(O)CCC(C)C)NCC1C(CC(=O)NCc2ncc(C)[nH]2)C1 c1(C(N2CCN(C(C=CSC)=O)C(C)CC2)=O)ccc(C#N)c(F)c1Br Cn1cc(S(=O)(=O)NC(C2(C)C=CCCC2)=O)ccc1=O N1(C(c2cc(CC)c(CC)o2)=O)Cc2nccn2CC(NC(C2CC2(Cl)Cl)=O)C1 CC(C)CCCCC(=O)NC1CN(C(=O)C(c2ccc(Cl)cc2)(C)C)C1 N1(CCNC(C#CCNC(C=CCOC)=O)=O)C(=O)CNC1=O c1(C(N2CC(N(C(C(C(C)C)n3cnnc3)=O)C)C2)=O)cc(F)cc2nn[nH]c12 C(=O)(C(C)(C)C(C)C)N1CCC(CC=C)(NC(=O)C=Cc2ccc(C)s2)C1 S(=O)(=O)(c1ccccc1F)N1CCC(N(C)Cc2ncsc2Br)C1 N1(C(c2nnc(C)o2)C)CCC2(CC1)CN(C(=O)CC1Cc3ccccc3O1)C2 Nc1ccc(F)c(F)c1C(N1CC(NC(=O)CC2(O)CCOCC2)C(F)C1)=O Cc1sc(Br)cc1C(=O)NCC#CCNC(C1CCS(=O)CC1)=O C1(C(N(CC(C)NC(c2cnnn2C)=O)CC)=O)CC2(CCCC2)CO1 c1(C(=O)NCCCC(=O)NC)ccc2nnc(C(F)F)n2c1 Cc1c(C(=O)NC2(CO)CN(S(=O)(=O)c3cccs3)C2)cc(Cl)cc1[N+](=O)[O-] CC(CC(C)(C)O)C(=O)NC1CCC(N2CCN(C)CC2)C1 C#CCC(C)(C(=O)Nc1cccc(C(C)C)c1)NC(C1CC(=O)CCO1)=O N1(C(C2(C(C)C)CC2)=O)CC(F)(CNC(=O)C(F)(F)Sc2cnn(C)c2)C1 N1(C(CSCCCC)=O)CC2CC2(CNC(C2CC2F)=O)C1 CC(C)(Cc1nn[nH]n1)C(=O)NC1CC(c2cccc(Br)c2)C1 Cc1cccc(CCNC(=O)Cn2cc(-c3cncc(C(N)=O)c3)nn2)c1C S(=O)(=O)(c1cccc(=NCC(C)OC(F)F)[nH]1)NCC1N(S(N(C)C)(=O)=O)CCC1 C1(CNC(Cc2c(C)ncs2)=O)CCCC12CCN(C(=O)C=CCF)CC2 N1(C(Cc2c(OC)cccc2OC)=O)CC2CCC1CN2Cc1ncsc1Br CCC(CC)C(C(=O)NCC1COCCN1C(C1OCCCO1)=O)OC c1(C(=O)NC23CN(C(CCOC)=O)C(C2)C3)ccc(Oc2ccccc2)cc1 C1(O)(C(=O)NC2CC3CC2N(C(=O)CC2CCCC2)C3)CC2(CCOCC2)C1 c1(NC2CC(F)(CNC(C3CCCC(C)C3)=O)C2)ncc2c(n1)CCOC2 C(C(C)(O)CC(=O)NCCC(C(F)(F)F)N1CCOCC1)OC(C)=O CC1CC(NC(c2cc(OCC(F)F)ccn2)=O)CN1C(C1CC(O)C1)=O C1(CC)CCC(C(N2CCOC(CNC(=O)C(O)CSC)C2)=O)CC1 C1(NC(=O)CC2C=CCCC2)COC2(C1)CN(C(C13CCCN(CCC1)C3)=O)C2 N1(C(Cc2c(C)ccc(F)c2)=O)CC(C2CN(C(=O)C(c3ccccn3)O)C2)C1 C=C=C(C)CC(=O)N1CCC(C2CCCCN2C(=O)CCC2CCC2)C1 C(=O)(CC1=NNC(=O)C1)NC1(CNC(CCC(=O)N(C(C)C)C)=O)CCCC1 CC1CN(C(=O)C(C2(C)CC2)NC(C2CCC2C)=O)C(C)C(C)(C)O1 C(=O)(C(F)(F)C(F)F)NC1CN(C(C2C(C(=O)OCC)C2)=O)CC1C(F)F CCC(CC(C)C)C(=O)OC(c1nc(-c2ccccc2)no1)C c1(OC(C)C(=O)NC2CC2CNC(C2CC(C)(C)C2)=O)cccc(Cl)c1Cl c1(CNC2CC3CC(CC(=O)OC)C2C3)c(C)cc(CN)cc1C C1(CC(=O)NCC2CC(O)CN2C(c2cccc[n+]2[O-])=O)(COC)CCOCC1 C1(NCc2c(Br)coc2)CN2CCCC1C2 C=CC(C)(C)NC(=O)CCC1CC(NC(C2(COC(C)C)CC2)=O)C1 c1(C(N(CCNC(=O)CC2(C)CCOC2)CC)=O)cnnc(-c2ccccc2)c1 CCC(CC(=O)NCCCc1cccs1)N(C(=O)C(CSC)OC)C c1(-c2cncc(C)c2)ccc(NC(=O)Nc2ccnn2Cc2cccs2)c(C)n1 c1(NC(C(CC)NC(C2C3CCC(C3)C2C)=O)=O)cccc2c1OCO2 C(=O)(C1=CCS(=O)(=O)C1)N1CC2(CC(NC(=O)C(F)CC3CCCCC3)C2)C1 c1(C(=O)NCCCN(C(C=NOC)=O)C(C)C)ccncc1N1CCOCC1 C(C(CC(C)C)NC(=O)CCc1ccoc1)NC(C1C(C)=CCS1)=O c1(N2CCCCC(NC(c3ccc4cncn4c3)=O)C2)ncc2cccnc2n1 Cc1cc(C)c(C(=O)NCC2COCCN2C(c2cnc(O)n2C)=O)s1 CC(C)(CCCNC(C1CCCO1)=O)C(=O)NC1C2CCCCC12 Cn1c([N+](=O)[O-])cnc1COC(=O)Cc1ccc(F)cc1 Cc1ccncc1C=CC(=O)NC(C1(O)CN(C(C2CC3CC3CC2C)=O)C1)C N1(C(C(CSC)C)=O)CCN(C(=O)Cc2ccccc2C(C)C)CC(O)C1 c1(SCC(=O)NCCC(O)CNC(C2CCCCO2)=O)ccc(F)cc1 C#Cc1ccc(NC=O)cc1.C12(C3(O)CN(C3)C(=O)C(C3CC3)OC1)CC2.OCC C(C)(N=c1nc2sccc2c(NCC2CSCCS2)[nH]1)c1c(SCC)cccc1 c1(C(N(CC(CN(C(CC(C(=O)OC)C)=O)C)O)C)=O)cnc2cc[nH]c2c1 c1(NC(=O)NCC(CC)CCC2CCCC2)ccc(F)cc1C#N c1(C(N2C(C)CCC(NC(c3cc(OC)ns3)=O)C2)=O)cccn2nccc12 c1(C(=O)NC2CN(C(C3CNC(=O)O3)=O)C(CO)C2)cc2ncsc2[nH]1 c1(C(C)C)cccc(F)c1C(=O)NCCNC(=O)Cc1ccco1 C1(C(NOCCC=C)=O)(CNC(c2cc(Cl)ns2)=O)CCCO1 C1(CNC(c2nnc(CC)s2)=O)CCN(C(=O)CSC(F)(F)F)CC1C C1(NC(Cc2scc(C(C)=O)c2)=O)CN(CCN(C)C2CC2)C(C(=O)O)(C(C)C)C1 C(C)(C)(CCCN=c1[nH]c2c(c(=NCC3CC(N(C)C)C3)[nH]1)CSC2)OC CCCCC(O)CC(=O)N1CCC(F)(CNC(=O)CCc2cc[nH]n2)C1 c1(C(C(=O)NC(C(CO)NC(C=CC(=O)OC)=O)C)N(C)C)ccccc1C c1(C(=O)NCC(CNC(c2cc(Cl)cc(C)c2N)=O)O)ccc2c(c1)CCC=C2 CCC(C)CC(C)C(=O)N1CCC(CCNC(C2CC(C)(C)C2)=O)CC1 c1(C(N2C(C(=O)Nc3cc(OC)ncc3)CCCC2)=O)ccn2cncc2c1 Cc1cc(N)c(C(=O)NC2CCC(NC(C3(C)CC4CC4C3)=O)C2)c(F)c1 CCCC(C(F)(F)F)NC(C1CCCN(C(c2cc(C)nn2C2CC2)=O)CC1)=O C1(C#N)(C(=O)NC(C2CN(C(c3cnn(CCN(C)C)c3)=O)C2)C)CCC1 C1(C(N2CC(OCC)C(CNC(=O)C(C)OC)C2)=O)CC2(CC2)CN1C N1(C(C(CC)OCC)=O)CCC(N(C(c2cnoc2-c2cccs2)=O)CC)CC1 c1(C(N2CC(CNC(C(=C(C)C3CC3)F)=O)C2)=O)c(N)sc2c1CCSC2 Cc1cc(CC(=O)NC(C)CCCNC(=O)C(C)Cc2cnco2)c(C)s1 S(=O)(=O)(c1ccc(Cl)c2cccnc12)NC(C(c1ccc(C(C)(C)C)cc1)N)=O CC1CCc2[nH]nc(C(N3CC4CC(NC(=O)CCCC(N)=O)C3C4)=O)c2C1 C1(C(=O)NC(CC2CN(C(C(C)N(C)C)=O)C2)C)CCCN1CC(F)(F)F C(=O)(C1=Cc2cc(Cl)ccc2OC1)NC1C(NC(COCCCCCC)=O)COC1 C1(C(=O)NC(C)CCNC(=O)C(C)CCO)CC(=O)CC1(C)C c1(Cn2c(-c3cc(C)c(Cl)c(N)c3)nc(COC(C)C)n2)cccc2cccnc12 S(=O)(=O)(c1nccs1)N1CCC(NC(c2cccc(Br)c2F)=O)C1 N1(C(CC(CC)OC)=O)C2CCCC1CN(C(=O)C(C)CC(C)C(C)=O)C2 C(=O)(CCS(=O)(=O)CC(C)C)N1CCC(CCOC)(NC(C2CCCSC2)=O)C1 N1(C(C2(C(N(C(C)C)C)=O)CC2)=O)CC(NC(c2cnn[nH]2)=O)CC2(CC2)C1 C12(CNC(c3ccc(C)s3)=O)CCC(NC(c3cc(=O)cc(Cl)[nH]3)=O)(CO1)C2 c1(C(c2nnnn2Cc2ccccc2)NCCSCC)ccc(F)c(Br)c1 N1(CCNC(CCC2(NC(C(C)c3cccs3)=O)CCC2)=O)CCCCC1 c1(C(N2CC(NC(C(C)C3CCCO3)=O)(CO)C2)=O)cc2c(Cl)cc(F)cc2[nH]1 C(=O)(C(CCC(N)=O)N(C)C)NCC1(CNC(=O)CCC(=O)N(C)C)CCCCC1 C=C(C)CN=C(NCCC1CCOC1)N(C)CC(C1CC1)OC C1(CC)CN(C(c2nn(CC)cc2Cl)=O)CCC1NC(C1(O)CCSCC1)=O N1(CC)CC(C(=O)NC2CN(C(=O)CCc3nc(C)no3)C2)CCC1=O c1(C(=O)NCCC(C(C)C)NC(c2cscn2)=O)c(F)cccc1[N+](=O)[O-] N1(C(c2cc(C)nnc2)=O)CCN(C(=O)CCCCCF)CC1CF C(=O)(CC1=CCCC1)NC1C(C)CCCC1.C1(=O)CCN1CC1CC1 CC(=O)CC(C)(C)CC(=O)NCC(C)NC(=O)CC1(O)CCCOC1 C12(CCNC(=O)CC3CCCCC3)CCC1CN(C(=O)CCc1ccco1)C2 c1(NC(CCSC)C)ccc(S(=O)(=O)N(C)CCc2c(F)cccc2Cl)c(Cl)c1 C(COC)(C(=O)NCCCN(C(=O)CCSCc1ccccc1)C(C)C)OC CCC(C(=O)NCC1CCCCN(C(=O)C(=O)NC)C1)C(C)(F)F c1(C(N2CC3C(NC(c4cc(Cl)nc(Cl)c4)=O)C3C2)=O)ccc([N+](=O)[O-])c(Br)c1 N#CCCCCC(=O)N1CCC(NC(C2CC3CCC2O3)=O)CC1 c1(CC)nc(C)sc1C(N1CCSC(C(N2CC(O)C(O)C2)=O)C1)=O CCCCCCCCCC(O)C(=O)NCCOCCN(C)C(c1ccc(Cl)o1)=O N1(C(c2nc(NC)c([N+](=O)[O-])cc2)=O)CCc2ccc(Cl)c(F)c2C1C c1(C(=O)NCC2C(C(N(CC(COC)(F)F)C)=O)C2)cccc(C)c1N N1(C(C2CCN(CC(C)C)CC2)=O)CCN(C(=O)CC2CC2(C)C)CC(CO)C1 CCCCC(C(=O)NC1CCC(NC(=O)C(C(C)(C)C)OC)C1)N(C)C c1(C(=O)NC(CN(C(=O)CCn2cccn2)CC)C)cnn(C(C)C)c1Br C(CC(C)C)(C(=O)NCC(O)C(=O)NC)N(C(C1CC(=C)C1)=O)C N1(C(C2CC(CCC(C)(C)C)(O)C2)=O)CC2(CN(C)C)CC2(CO)C1 O=C1C2CC3C1C3C2C(=O)NC12CCC(C(=O)NCC3C=CCOC3)(CC1)C2 c1(C(N(CCC(C)NC(c2cc(N3CCCC3)ccn2)=O)C)=O)ccncc1O C1(N(C)C)CC2(C1)CN(C(c1ccncc1)C(=O)Nc1ccc(F)cc1)C2 C1(CCC)CN(C(=O)Cc2csnn2)CCN1C(=O)Cc1c(C)n[nH]c1C CN1CCC(C(=O)NCC2CCC(NC(c3cc(C(F)(F)F)cs3)=O)C2)CC1=O N1(C(C(CC)CC2CCCC2)=O)CC2CN(C(=O)Cc3nnc(C)s3)CC2C1 c1(N2CCC(CNC(C#CC(C)(C)C)=O)C2)ccc([N+](=O)[O-])cc1F C(CNC(C12CC(F)(C1)C2)=O)(C(C)(C)C)NC(Cc1cc(C)no1)=O N1(C(C2(C#N)CC2)=O)CCC(NC(=O)Cc2ccc(F)cn2)C2(CCC2)C1 CC(C)CCCC(C)CNC(=O)C(c1ccnn1C)NC(C1(O)CCSC1)=O c1(NC(C(c2cccc(N)c2)(C)C)=O)ncc2cc(Br)ccc2n1 N1(C(c2cccc(C)c2)=O)CC2CC(CNC(=O)CN3CCOCC3)CC1C2 c1(C(C(=O)N(C(=O)C=Cc2ccc(Br)s2)CC)(C)O)ccc(F)cc1 C(CC1=CCCCCC1)NC(CC1CC(NC(C2(CC(C)C)CC2)=O)C1)=O c1(CC(=O)N(C2CCCN(C(c3c(CC)nns3)=O)C2)C)ccc(C#N)cc1 C=C=CCC(=O)NC1COCC1NC(=O)C(F)F c1(C(=O)NC2C(NC(C(C=C)(C)C)=O)CC2)c(F)ccc(C)c1Cl C1(C(N(C2CCN(CCc3noc(CC)n3)CC2)CC#C)=O)CCCC(F)C1 CC1(C(=O)NCC2(NC(c3cccc(CC(F)(F)F)c3)=O)CCC2)COCCO1 Cn1ccc(C(=O)NC(CNC(c2csc(Cl)n2)=O)CO)n1 c1(CNC(=O)NCC2(C(=O)OCC)CC2C(F)(F)F)c(C)ccc(C)c1O N1(C(C2CCN(C)C2=O)=O)CC2CCCC2(C(N2CCCCC2)=O)C1 Cc1cc(NC(c2ccc(NC(C3(n4ccnc4)CC3)=O)cn2)=O)ccc1Br c1(C(N(CCCNC(=O)COc2ccsn2)C2CC2)=O)ccn2ccnc2c1 N1(C(CCNS(CC)(=O)=O)=O)CC(C)CN(C(c2ccc(Cl)c(O)c2)=O)CC1C c1(NC(=O)C(C)S)ccc(F)cc1.C(C(=O)N(CCCNC(C)=O)C1CC1)=CC C1(NC(=O)OC(C)(C)C)CC2CC(NC3CCN(C4CC4)C3=O)CC12 c1(SC)ccc(C(N2CC3C(NC(c4cn5c(n4)SCC5)=O)C3C2)=O)c(Cl)c1 CC1(NC(c2ccncn2)=O)CN(C(=O)C(F)=C2CCC2)C1 C(C(O)CC(F)(F)F)NC(C(C(C)NC(c1cccc(CO)n1)=O)C)=O Cc1nc(CNC(C2CC(NC(C3CC(CF)C3)=O)CCO2)=O)sc1C CCCCC(CNC(c1ccc(C(F)(F)F)nn1)=O)NC(C1CC1F)=O c1(C(=O)Nc2ccc(COC)c(Cl)c2)ccc2c(C)c[nH]c2c1 CCCC(CNC(=O)C(C)(C)C(=O)OC)C(=O)NCc1n[nH]c(C)n1 c1(COCC(=O)NCCC2(NC(=O)C(=Cc3c[nH]cn3)F)CCC2)ccccn1 C1(NC(c2ccc(OC)s2)=O)CCCCC1CNC(c1c(C)[nH][nH]c1=N)=O c1(C(N2CCN(Cc3ccc(OC)cc3)CC2)=O)ccnc(Cl)c1OC c1(C(N2C(CNC(c3c(C)snc3)=O)CCCC2)=O)cc2c([nH]1)CCC(C)C2 c1(C(=O)NCC2CC(CC(=O)OC)C2)c(Br)ccc(F)c1I C12(C(=O)NC3CCN(C(=O)Cn4nccn4)CC3)CCCC1C2(F)F C1(C(N2CC3(CCNC3=O)C2)=O)N(C(C2CC23CC3)=O)CC12CCCC2 C(C)(CNC(c1ccsc1)=O)(CC(C)C)NC(c1cccc(SCCC)c1)=O N1(C(c2nc(CNC(C(N3CCOC3=O)C)=O)oc2)=O)CCC2(CC1)N=N2 c1(C(C)=O)cc(C(=O)NCC(n2cc(CC(C)O)nn2)C)c[nH]1 C1(NC(CSCCC(C)C)=O)C=CC(CC(=O)NC(C)CC(C)O)C1 CCC(C)(C)CC(C(=O)NCC1CC1)N1CCC(CO)CC1 c1(C(=O)NCC(c2ccccc2)C)c(-c2cnc(N)nc2)cncc1F.C(F)(F)F N1(C(C2(CC)CCOCC2)=O)CCC(C)C(NC(c2ccncc2)=O)C1 CCC(CC(=O)N(CC(O)CN(C(=O)C(F)n1ccnc1)C)C)OC C1(NC(C2(CNC(C(CC=C)NC(C)=O)=O)CC3(CC3)C2)=O)CCOC(C)(C)C1 C1(C(=O)OC(C(CF)C2(C)N=N2)=O)CN(C(C)(C)C)CCC1c1ccc(F)cc1 c1(N2CC(=C(CNC(C(C(COC)C)C)=O)F)C2)ncnc2c1CCCC2 c1(C(=O)NC2CCCN(C(CSCCC)=O)C2)ccc(C(C)CC)nc1O C1(=CC(N2CC3C(NC(=O)C=CCn4cncn4)C3C2)=O)CN2CCC1CC2 c1(C(N2CCC(CC=C)(NC(=O)C(O)CCSC)C2)=O)cccc(Cl)c1[N+](=O)[O-] C1(NC(CC2N(C)CCC2)=O)CCCCN(C(c2cncnc2)=O)CC1 CC(CN(C(=O)C(F)C(C)(C)O)C)N=c1ccn2c(Br)cnc2[nH]1 c1(OC)cc(Cn2nc(C(C)O)nc2-c2ccc(OC)cn2)cc(OC)c1OC c1(C(C(=O)NCC2N(C(C(CC)=CC)=O)CC(OC)C2)(F)F)ccc(F)cc1C N1(C(c2[nH]cc(CN(C)C)c2)=O)Cc2ccccc2C(NC(=O)C=CCF)C1 c1(CC=C)ccccc1NC(c1ccc(C)nn1)c1nnnn1-c1ccccc1 C#CC1(C(=O)NC2CN(C(c3ccncc3Br)=O)CC2C)CCCC1 Cc1noc(Cl)c1CCC(=O)NCc1csc(CNC(C2CC(F)(CO)C2)=O)n1 c1(NC(C2N(C(CNC(Cc3cc(C)on3)=O)=O)CC2)=O)cnc2[nH]nnc2c1 C1(OCC)COCCC1CC(N1CC(CNC(=O)CC2CCOC2C)C1)=O CN1CCC(C(=O)NCCCCNC(C2NC(=O)C3CCC23)=O)c2ccccc21 c1(C(=O)NC(C)CN(C)CCOC2CCOC2)ccc2ccc(Cl)cc2n1 C=CC1CCCCN1C(=O)C(C(C)(C)C)NC(C1CC(C)N(C)C1)=O c1(OC)ccc(C2(C(=O)NC(CNC(c3c(CO)n[nH]c3)=O)C)CC2)cc1OC Cc1oc(CNC(=O)CCCC#N)nc1C(=O)NOCC(C)C Cc1cn(C(C)(C)C(=O)N(C2CCC(NC(=O)C(F)(F)F)C2)Cc2cnsn2)cn1 C(CC(O)CCO)NC(C(C1CCCC1)NC(=O)CCc1ccccc1)=O c1(C(=O)NCC2CCN2C(=O)C=C(Cl)Cl)ccc(=O)n(CC(F)(F)F)c1 CC(C)(CCCF)C(=O)NC1C2CC(NC(C3CS(=O)C3)=O)CC12 [N-]=[N+]=Nc1cc(F)ccc1C(=O)NCCC1=CCCCCC1 CC(O)(CC(F)F)C(=O)N1CC2CCC2(NC(c2ccco2)=O)C1 C(CC(C)C(=O)N1CSCC1C(N1CCCC1C1(C)CC1)=O)=CCC c1(CC(=O)N(C)CCOCC(F)(F)F)ccc(Cl)nc1 c1(C(N2CCCC(CNC(C(C)OC3CCCC3)=O)C2)=O)ccc(O)nc1Cl N1(C(CC#N)=O)CCC2(C1)CN(C(=O)Cc1csc3cccc(F)c13)CCO2 C1(NC(C2CN(C)C(=O)CC2)=O)CCC2CN(C(=O)CN3CCOCC3=O)CC12 c1(COC)ncc(C(N2CCCC(NC(c3n[nH]c(SC)c3Cl)=O)C2)=O)c(O)n1 Cc1cc(C(=O)NCC23CCC2CN(C(C2C=CCCC2)=O)C3)cc(F)c1 CC(F)(F)C(=O)NCC1(CNC(C2CC2(C)C(F)F)=O)CC1 CC(C)C1=CCC(C(=O)NCC2CC(CNC(c3ccc([N+](=O)[O-])s3)=O)C2)CC1 C1(Nc2ncn(C)c(=O)c2)(CNC(=O)C(=O)NC2CC2)CCC(F)(F)CC1 CCCCCC(c1nnnn1C1CCOC1)Nc1cccc(N2CCOC2=O)c1 n1(CC(=O)NC2(CNC(C3(C(F)F)CC3)=O)CCCC2)ncn(O)c1=O N1(C(=O)OC(C)(C)C)CCC(C(=O)NCCc2ncco2)CC12CC2 N1(C(CNC=O)=O)CCC(C2(O)CCN(C(c3cc4cscc4s3)=O)C2)CC1 C(C(=O)O)(C(O)c1cccnc1)NC(=O)C(n1cc(Cl)cn1)F c1(C(=O)NC(C2(O)CN(C(C=CCC)=O)C2)C)cc(C)c(Cl)cc1C N1(Cc2cccc(OCC)n2)CC2(CCC(NCc3cc(C)cc(Cl)c3)C2)C1 c1(C(c2n(CCCCCC)nnn2)NCC(=O)NCCC)ccc(Cl)cn1 C=CCCCCCC(=O)N1CC(C(=O)N(C(C)CO)CC)C(C(C)C)C1 C1(NC(c2cn(CCOC)nn2)=O)C=CCN(C(=O)C(F)C2CCC2)C1 Cc1c(C(N2CC(NC(=O)CCN3CCC(O)CC3)C(C)(C)C2)=O)nn(C)c1N C1(c2ccc(CC)cc2)CN(C(C2(CCF)CC2)=O)CCN1C(C1SCCS1)=O C1(C)(CCNC(C(c2ccc(OC)cc2)C)=O)CCN(C(c2cnsc2)=O)CC1 c1(CC)c(C)nc2scc(C(N3CCCC3CNC(C)=O)C(=O)NC3CCC3)n12 C(=O)(CCC(C)(C)C#N)N1CCC(C(C(=O)N(CC(C)C#N)C)(C)C)C1 Cc1ccc(C(F)(F)F)cc1C(=O)NCC(C1CC1)NC(=O)CN1CCCCC1 C1(C(N2CC(NC(c3ccncc3O)=O)C3(C2)CC3)=O)Cc2cc(Cl)ccc2O1 c1(C(=O)NCC2CCC(NC(=O)CCCCF)C2)noc2ccc(Cl)cc12 Cc1cccc(C(=O)NCC(C)C(=O)NC(C2CCC2)C2CC2)c1F N1(C(=O)OC(C)(C)C)CC(C2CCCCC2CNS(=O)(=O)N(C)C)CC1C(=O)O C1(CCNC(c2cc(C)on2)=O)CSCCN1C(=O)COc1ccsn1 c1(C(=O)NC2CN(C(c3cncc(OC)n3)=O)C3C2C3)cc2n(c1)CCSC2 n1(CC)nc(C(=O)NCC(CO)NC(=O)CCc2csc(=N)[nH]2)c(Br)n1 c1(C(=O)NCC2OCCN(C(C=CCCC)=O)C2)cc2nc[nH]c2cc1F c1(C(=O)NCC(CC(=O)N(CC(CC)CC)C2CC2)C2CCC2)ccc([N+](=O)[O-])o1 c1(CC(N2CC3CN(C(c4c(C)c[nH]n4)=O)CC3C2)=O)ccc([N+](=O)[O-])cc1F N1(c2nccc(=NCc3c(N)cccc3)[nH]2)CCCC1C1OCCO1 c1(C(N(CCC)CCNC(=O)C=CCF)=O)c(CC)cccc1CC.O c1(C(N2CC(CNC(CCC=C)=O)N3CCC2C3)=O)ccc(=O)n2c1CCC2 c1(NC(c2ccc(OC)cc2)=O)scc(O)c1C#N.c12ccc(cc1)C(=O)NC2 C#CCCCC(C)C(=O)NC1C2CC1N(C(c1cnc(C3CC3)nc1)=O)C2 c1(C(C(=O)NC(CNC(c2nc(C)[nH]n2)=O)C)(C)O)ccc(F)cc1 CCC(Cc1cccc(F)c1)C(=O)NCC(c1cn(C2CC(O)C2)nn1)(C)O c1(CC(=O)NCC(CC(C)C)NC(=O)C(C)(O)C2CC2)ccc2nc(O)[nH]c2c1 C#CC1(NC(=O)C=CC(C)NC(c2cccc(COC)n2)=O)CC2CCCC12 N1(C(=O)NC(c2cc(O)n(C)n2)C)CC2(COC)CC(c3ccccc3)(C1)C2 CC(C)(CNC(=O)C(C1CCOCC1)N1CCCC1)Cn1cc(C2CC2)nn1 CC1(C)CC(NC(=O)C=CCO)CCN(C(C2CC3(CCCC3)CO2)=O)C1 C(=O)(C(C)C(F)(F)C(F)F)NCC(CC)(CC)NC(C1CC1(C)C(F)F)=O c1(C(N2CCN(C(CSCCCC)=O)C(C)CC2)=O)c[nH]c2c(CC)cccc12 N1(C(C(CC)C)=O)CC2(C1)SCCC2NC(c1nc(Cl)ccc1F)=O C1(NC(=O)Cn2ccnn2)CN(C(C2CC2c2ccncc2)=O)CCC12CCC2 Cc1ccc(O)cc1CN1CC2(CC2)CC1C(=O)OC(C)(C)C Nc1c(C(=O)NC(c2ccccc2Cl)CCO)cc(F)cc1Br C#CCCCC(C)C(=O)N1CC(NC(=O)C(C)CN2CCOCC2)C(CO)C1 O=C(C1=CCCCO1)NC1CCN(c2ncnc(O)c2Br)C1 C(=O)(C1COc2ccc(Cl)cc21)N1CCCC(CN(C)Cc2ccco2)C1 c1(OC)nc(N2CCCC(CCNC(=O)CCC3CCOC3)C2)cc(C)n1 C1(NC(=O)C(F)C2CCCC2)CCOC(C(N2CCC3(CC3)C2)=O)C1 C=CC1(C(N2CCC(C(C)C(=O)NCC(C)(C)C3CC3)C2)=O)CCOCC1 c1(C(=O)NC2C(NC(CN3CC(C)C3)=O)C2)ccc(-c2cn[nH]c2)cc1 N1(C(C2C(OC)(OC)CC2)=O)CC(CNC(c2ncoc2C)=O)CC1(C)C CC1CCN(C(=O)CCCc2ccsc2)C(CNC(=O)CCC2CCCCO2)C1 C1(C(=O)NCC(CNC(=O)CC(C2CC2)C2CC2)CO)CCCC2(CCC2)O1 c1(C(N2CC(C(N(C)CC3C(C)C3)=O)OCC2)=O)cc(F)ccc1F c1(C(N)=O)ccc(C(=O)NCC(O)CNC(c2ccc(C3CCOC3)s2)=O)[nH]1 c1(CN(C)CC2(C)CC2(F)F)cc2cc(Cl)ccc2s1 CC(C)CCCN=c1[nH]c(N2CCC3(CCCN(C)C3)C2)nc2ccc(Cl)cc12 c1(OC)cc(CN=c2[nH]cc(C(c3cccs3)=O)s2)ccc1C(N)=O C1(C)(CC)C=C(C(=O)NCC2CN(C)CCN2C(c2csc(C(C)=O)n2)=O)C1 C(C(=O)NC1CC(N(C(=O)Cc2ccccc2C)C)C1)(C(C)(C)C)OC C=C(C)CC(C(=O)NCCCNC(c1ccc(CC2CC2)s1)=O)NC(C)=O c1(C(=O)NCC2(F)CC(NC(c3c(N)ccc(O)c3)=O)C2)ccnc2c1CCC2 N1(C(C(n2c(C)cc(C)n2)C)=O)CCCC(C)(C(=O)NCCSc2cccs2)C1 N1(C(C2(F)CCN(C(c3ccc(SC)o3)=O)C2)=O)CCc2nc(O)[nH]c2C1 C1(CNC(CNC(=O)OCC)=O)CCCC1(C)NC(C1CC1C)=O C1(OC)CC(C)CN(C(c2ccnc(CNC(C3CCCC(OC)C3)=O)c2)=O)C1 N1(C(CC(C)O)=O)CC2(C(N3CCCC(N=[N+]=[N-])C3)=O)CCC1CC2 C1(NC(CNC(c2ccc(C)s2)=O)=O)CC2CN(C(C34CC(C3)C4)=O)CC12 C1(NC(c2n(C)cnn2)=O)CN(C(c2cc(O)ccc2F)=O)C2(CCOCC2)C1 N1(c2snc(SC)n2)CCCC(C)(C)C1CNC(=O)CN1CC2CC2C1 C1(NC(c2c(OCC)n[nH]c2)=O)CN(C(C2CC2C(N)=O)=O)C(C)(C)C1 N1(C(CCC2N(C)CCC2)=O)CCC2(CC1)CN(C(c1c[nH]c(=N)s1)=O)CCO2 C(=O)(C(C#N)CC)NC(CCC)CNC(c1ccncc1OC(C)C)=O CCC(C(=O)OC)C(=O)NC1(CO)CCN(C(=O)C(=O)NCCOC)C1 c1(C(=O)NCC(C)O)cccnc1CNC(=O)CCOCCSC1CCC1 N1(C(c2ccc(-c3nc(C)[nH]n3)cc2)=O)CC2(CCOCC2)C1C1CC1 c1(C(=O)NC(C(C(C)C)C)CNC(c2ccc(Cl)cn2)=O)cnc2[nH]ncc2c1 C(C(O)(C(=O)NC1CC(NC(=O)CN2CCCCCC2)C1)C(F)(F)F)N(C)C C1(NC(C(F)=C(C)C)=O)CCN(C(=O)C(C)C2CC2)CC1F c1(CC(=O)NC2C(NC(=O)COCCOCCO)C2)csc(C(F)(F)F)c1 C1(NC(Cc2c(C)cccn2)=O)CC(F)CN(C(C2CCC(=O)N2)=O)C1 CC1C(=O)N(C)CCN1C(C1CCN1Cc1ccncc1O)=O C(=O)(C(C)(C)C(=O)NCC(C1CCN(C(c2cnc(O)c(C)c2)=O)CC1)O)NC N1(C(c2c(CC)ncs2)=O)CCCC2CN(C(=O)C(c3ccccc3C)C)CC12 c1(C(=O)NCC2C(NC(COCC=C)=O)CCC2)cc(=O)c2ccccc2n1C C1(NC(=O)CC2CCCO2)CCN(C(c2ccc(Cl)c(Cl)c2)=O)CC1O c1(C(=O)NC2C(NC(C3(C(F)(F)F)CC(=C)C3)=O)COC2)cc(F)cnc1OC N1(C(C#CCNC(C2CCCCCC2)=O)=O)CCOC2CCCCC12 c1(C(=O)NCCCOCCN(C(C(C2CCCCC2)C)=O)C)cscc1Cl Cc1ncc([N+](=O)[O-])n1CC(=O)NC1CN(c2cnn(C)n2)C1 CC1=C(C)CC(C(=O)N(CC(C)(C)C(=O)NC2CCN(C(N)=O)CC2)C)CC1 CC1Cc2cc(CC(=O)NC34CC(C3)N(C(=O)CSCC(N)=O)C4)ccc2O1 C1(CN(C(=O)COCCCF)C)CCCC(NC(c2ncccc2F)=O)C1 c1(C(=O)NC(C2CCN(C(c3c(C)c[nH]n3)=O)C2)(C)C)nn(C(F)F)cc1Cl C(=O)(C(CCC=C)CC(C)C)NC1CCN(C(C2(C#C)CCC2)=O)CCC1(F)F C1(CN(CC)CC)CCCCN1C(=O)CCc1ccc(N(C)C)nc1 N1(C(C(C)(C)OC(C)C)=O)CCN(C(C2(C)CCCS2)=O)CC12CCC2 n1(CC)cc(Cl)c(C(=O)NC(C(C)NC(c2conc2COC)=O)C(C)C)n1 c1(C(=O)NCC(CCOC)NC(c2cc(C3CC3)nn2C)=O)cc2occc2[nH]1 c1(CC(=O)NCCN(C(=O)C2=C(C)CCC2)CC)ccc2ocnc2c1 c1(Oc2c(CN(C(C(c3cnn[nH]3)SC)=O)C(C)C)cccc2)ccccc1Br CC1CC(C(=O)NCC(CO)NC(=O)Cn2cccc2)C1 n1(CC)ncc(C(=O)OCCNC2(C(C)(C)O)CC2)n1 c1(CC(N2CC(CC(C)NC(c3c(CC)cno3)=O)C2)=O)ccc(F)cc1 c1(C(=O)NC2CN(C(C(CC)C(C)O)=O)CC2(C)C)ccnc2[nH]ncc12 N1(C(C(C=C)(C)C)=O)CCC2(CC1)CN(C(=O)C(F)C1=CCCCC1)CC2CO N1(C(C(CCC)=CCC)=O)CCn2c(CNC(C3CC3(C)C(F)F)=O)nnc2C1 C1(NC(c2c(CC)nc(C)o2)=O)CN(C(=O)Cc2ccccc2O)CCC1C C#Cc1ccc(F)cc1C(=O)NCCCC(C)(C)NC(c1oc(C)cc1C)=O C1(CNC(c2ccc(SCC)nc2)=O)CCC(C)CN1C(=O)CNC(N)=O c1(SC)cc(C(=O)NCCC2(O)CCCNC2)cc(SC)c1 N1(C(CSCCC#N)=O)CCN(C(=O)CON=C2CCCCCC2)C2CCCC12 C1(CCNC(c2cc(OCC)no2)=O)CC(F)(F)CN1C(=O)C(N)=O C1(NC(C2(CC)CC2)=O)CC2CC1CN2C(C1(c2ccccc2)CC1)=O C1(C(=O)NCC2CCCN(C(c3ccc[nH]3)=O)C2)CC12CCC(F)(F)CC2 C1(c2cccs2)(N(C(N2CCC(Cc3ccccc3)C2)=O)C2CC2)CCOCC1 C1(C(=O)NCC2CC23CCC3)(CNC(C(C)C2CCCC2)=O)CC(C)(C)C1 C(=O)(C(C)C(O)C(C)C)NCCN(CC(C)O)C(c1nc(C(C)C)oc1)=O CC1(C)CCC(CC(=O)Nc2cccc(NC(=O)CC3C=CS(=O)(=O)C3)c2)C1 CCC(CC)C(C)C(=O)N1CC2(CCC(CNC(C3(C(C)C)COC3)=O)O2)C1 c1(C(N(C2CC(NC(CC3(CC)CCC3)=O)C2)C)=O)nc(C)oc1C N1(C(C(CC(C)C)C)=O)CCCN(C(c2csc(-c3ncc[nH]3)n2)=O)CC(CO)C1 c1(C(=O)NCC2(F)CN(C(C3C(CC)CCC3)=O)C2)cccc(C(C)(F)F)n1 N(C1CCCc2sccc21)C(CCCCCO)c1n(CC(=C)C)nnn1 C1(C)(CC)CC1C(=O)NCC1CC(C(=O)NCC(C)(C)n2ccnc2)C1 CCC(CC(=O)NCC1CN(C(C2OCCC2(C)C)=O)CCO1)OC C1(OC)(CNC(C2CC(F)(CO)C2)=O)CCN(C(=O)CC2OCCC2(C)C)C1 C(=O)(C(C#N)C(C)C)NCC(c1ccccc1)N(C(c1[nH]cc(C)c1)=O)C c1(OCC)cnc(C(=O)NC(CNC(=O)CCCOC2CC2)CC(C)C)cn1 c1(OC)nccnc1C(=O)NC1CC(C)(NC(C2CCCN2C(=O)C(C)C)=O)C1 C1(C(=O)NCc2cn(-c3ccccc3C(F)(F)F)nn2)CNC2(CC2)CO1 CC(C)CC(C(=O)N(c1ccccc1)CCCN1CCC(O)C1)NC(N)=O Cc1c(F)cc(C(=O)NC2CCCCN(C(=O)C=Cc3cscn3)C2)c(F)c1N Cc1ncsc1C=CC(=O)Nc1cccc(NC(=O)C(F)(F)c2cncs2)c1 C1(CN(C)C)CCC(C(N2CCC(N(C(=O)Cc3nc[nH]n3)C)C2)=O)O1 N1(C(c2nn(CC)c(C)c2)=O)CC2(NC(C3CC(C)(OC)C3)=O)CCC1CC2 N1(C(C(C)=NOCC#N)=O)CCCC(CC(=O)N(C(C)CO)C2CC2)CC1 C(=O)(C(C)(C)CC(=O)N1CC2CCCC2(NC(c2ccoc2C)=O)C1)OCC C#CC(C)(C)C(=O)N1CC2CC2(CNC(C2(COC(C)C)CC2)=O)C1 c1(C2(C(=O)NC3C(NC(C(C)SC(C)C)=O)C3)CC2)cc(F)cc(C#N)c1 c1(CC(=O)NC(CC)CN(C(=O)CCN(C(=O)CO)CC)C)c(C)cc(O)cc1C c1(C(N2CC(CNC(CSCC=C)=O)C3C2C3)=O)nc(C)ccc1C C1(CN(C)C)CCC(C(=O)NCC(O)CCNC(c2csc(Cl)c2)=O)CC1 N1(C(COCCCC#C)=O)C(CNC(=O)C2=C(Cl)CCOC2)CC2CCCC12 N1(C(C2CC(NC(CCC(CC)CC)=O)C23CCC3)=O)CCc2c(O)noc2C1 C1(C(=O)NCC(CN(C)C(c2ccoc2C(F)(F)F)=O)(C)C)CCCCS1(=O)=O CCN=c1ccc(C(=O)NCC(C)(C(C)C)NC(=O)CC2CC23CC3)c[nH]1 C1(NC(C2C(CC)OCC2)=O)CC12CCC(NC(=O)C=C1CCN(C)CC1)CC2 Cc1cc(C)c(C(=O)CCCC(=O)OCC2CC2C2CC2)c(C)c1 O=[N+]([O-])c1ccc(C(N2CCN(OCc3c[nH]c4cnccc34)CC2)(CC)OC)c(F)c1 N1(C(CC(c2ccc(Br)cc2)C)=O)CC2C(C(=O)NOCC(O)CO)C2C1 c1(NC(CCC2CC(NC(CC(C(=C)C)OCC)=O)C2)=O)cc(C)c(C)c(C)c1 Cn1nc(C(F)(F)F)cc1C(c1ccccc1)NC(N1CCC(O)(C(F)(F)F)C1)=O [N-]=[N+]=NCC(C(=O)N1CCSC2(CC2)C1)NC(=O)C(O)C1CCCC1 CC1CC(CNC(=O)C(C)NC(=O)COCc2nc[nH]n2)C1 c1(OC)ccccc1C(CNC(=O)CC1CCC1)NC(c1ncc(F)cn1)=O N1(C(C(=O)NCCC)C(C)C(C)(C)C)CCn2c(nc3ccccc23)C1 CCC(CC(=O)NCCC1(OCCOC2CC2)CCOCC1)NC(=O)COC C1(C(N2CC(O)(CCNC(COC3(C)CCC3)=O)C2)=O)CC(C2CCCC2)C1 c1(C(=O)OC)cnc(C(=O)NC(C)CCCNC(=O)C(C)n2cncn2)cn1 C(=O)(CC(C)(O)C(F)(F)F)NC(C)CN(C(=O)C(C)CCc1cccc(F)c1)C c1(C(=O)NCCN(C(C(c2ccccc2)SC)=O)C)cc2cc(Cl)ccc2s1 C(=O)(C#CC1(C)CCCO1)N1CCCC(N(C(c2c(OC)cccc2Cl)=O)C)C1 C1(NC(c2cnc(C3CC3)s2)=O)COCCN(C(c2ccccc2Br)=O)C1 c1(C(C)NC)cn(C2CN(C(c3scnc3C3CCCC3)=O)C2)nn1 C1(CC(=O)NCCCC2N(C(CCC(=O)OC)=O)CCCC2)CCCCC1(F)F c1(CC(=O)NC(C(C)NC(C2CC2(F)F)=O)CO)ccc(Cl)c(Cl)c1 c1(C(=O)NCC=C(C(=O)NCc2c(CC)noc2)C)cccc2cncn12 C#Cc1ccc(C(=O)NC(CC(=C)C)C(=O)NCC(C)(C)C2CCCO2)cn1 c1(C(C)O)ccc(C(N2CCC2C(N2CCOCC2CO)=O)=O)cc1 C=C(C)CCCC(=O)NCc1nc(C2CCN(C(C3CC3(F)F)=O)CC2)n[nH]1 N1(C(C=Cc2c(C)n[nH]c2)=O)CCC2(CCCN2C(=O)COCC(F)F)CC1 CC(C)C(C)(CNC(=O)CC12COC(CF)(C1)C2)NC(=O)Cc1cncs1 CC1CC(=O)NCCN1c1nnnn1C1CCC2CC2CC1 C1(CNC(CC(=O)OC)=O)CC2CC(C1)N(C(=O)C(c1cc(F)cc(F)c1)C)C2 C=C=CC(C)C(=O)N(C)CC1COCCN1C(c1cn(CCO)nc1C)=O c1(N(C)CCC2CC2)ccc(S(=O)(=O)NCC(O)CCC2CC2)c(Br)c1 C=C(CNC(=O)COCc1ccccc1)CCNC(C1CSCCS1)=O c1(OC)ccc(Cl)c(C(N2CCC3C(NC(=O)Cn4cnccc4=O)C23)=O)c1 C=CC(C)(CCOC)C(=O)NC(C)CCCNC(=O)CC1CCCNC(=O)C1 C1(CNC(c2c(COC)cc[nH]2)=O)CN(C(C2CCCNC2=O)=O)CCCO1 N1(C(C2C(=C)CC2)=O)CCCCC1CN(C(=O)C(CC)=CCCC)C C=Cn1nccc1C(=O)NC1CC(CNC(c2ccc(C(C)(F)F)nc2)=O)C1 c1(-c2nccc(C(C(C3CCN(C)CC3)C#N)=O)c2)ccc(Cl)c(Cl)c1 C(=O)(CCCN=[N+]=[N-])NC(C=CC(=O)Nc1c(C)n(C)nc1)C C1(C(N2CCC(N(C(c3ccc(F)s3)=O)CC)C2)=O)CCCC(OC)C1 N1(CC(=O)N(CC(O)CNC(C2C=CCC2)=O)C)CCC(c2ccccc2)CC1 CCC(CC)CC(=O)NCC1CCC1NC(=O)COC(F)(F)F c1(NC(C2(NC(CCOCC)=O)CC(F)(F)C2)=O)ccc(OC)c(OC)c1 CCC(C(=O)NC(C1CCN(C(c2cnc3n2CCC3)=O)C1)(C)C)C(C)C C1(C(N2CCC(c3nn[nH]n3)C2)=O)C2CCC(C2)N1C(=O)Cc1ccccc1F C(=O)(CCCCCn1cc(-c2ccnn2C)nn1)NC(C(=O)OC)C1CC=CC1 CC(C)C(C)(CN=c1[nH]c(=N)[nH]c(Cl)c1[N+](=O)[O-])NC(c1coc(C(N)=O)c1)=O CC1(C)CCN(C(=O)C(N2CCCSCC2c2cnn[nH]2)=O)CC1CO c1(OC)cccc(C(CNC(C)=O)NC(C2C3CCC2(c2ccncc2)C3)=O)c1 c1(C(N2CCN(C(C3=C(C)CCC3)=O)CC(O)C2)=O)cc2c(cc1C)OCO2 c1(C(=O)OC)ccc2c(c1)CN(N1CCC([N+](=O)[O-])CC1)C2 O=C1NCCN(C(C2CCN(C(C3(CC4CC4)CC3)=O)C2)=O)C1CCO C1(C(N2C(CN(C(c3c(CC)ocn3)=O)C)CCC2)=O)CCCCC(C)(C)C1 N1(C(C2CCC=CCC2)=O)CC(C2CN(C(c3cnc4n3CCS4)=O)C2)C1 CC(CC(=O)N(CCCCN(C(=O)CN1CC2C=CC1C2)C)C)CC(C)(C)C c1(C(=O)NC23CC(CNC(CC(C)CF)=O)(C2)C3)cc(F)c(O)c(F)c1 c1(C(N2CCCC(c3cn(CCO)nn3)C2)=O)n[nH]c(=O)c2ccccc12 c1(C(N(CCCNC(CCN(CC)CC)=O)CC)=O)ccc(C)c(P(C)(C)=O)c1 c1(NC(c2nccc(-c3cccc(OCC)c3F)c2)=O)cc(OC)ccc1C#N C1(NC(C(=O)N(C)Cc2ccc(C)cc2)=O)CC(O)CN(C(=O)OC(C)(C)C)C1 CC(C)CC(C)(C)C(=O)NCC1CCC(C(N2CCCCCC2C)=O)O1 O(NC(=O)CC=Cc1ccccc1)CC(=O)NCc1c(CC)nn[nH]1 C12(CNC(CC(C)SC)=O)CC1CN(C(c1cnn(CCO)c1)=O)C2 Cc1cc2c(N3CCCC3C(=O)NC3CSC(C)C3)ncnc2s1 [N-]=[N+]=NC1CCCN(C(c2cccc3c[nH]nc23)C(=O)NC2COC2)CC1 N1(C(C2C(=C)C2)=O)CC2CCN(C(=O)Cc3csc(-c4cccnc4)n3)CC2C1 C1(CNC(C(C)=CC)=O)CN(C(c2ccnc(C)c2)=O)CC(C)(C)O1 C1(O)(CN(C(=O)CC2CCCN(C)C2)C)CCN(C(=O)CC2CC2)C1 N1(C(c2c(C#C)c[nH]n2)=O)CC2CC(NC(c3ccn4ccnc4c3)=O)CC1C2 c1(CCC(=O)NCc2cccc3cn[nH]c23)ccc2ncsc2c1 N1(Cc2cc(C(=O)OC)cc(F)c2)CCC2(CC1)CC2CO C(CC(C)(C)CC(=O)NC1CCC(N(C)C(c2nnc(O)cc2C)=O)CC1)OC c1(C(=O)NCC2CCCCN(C(C(C)=CC3CC3)=O)C2)cc(C)cc([N+](=O)[O-])c1 c1(C(=O)OC(c2ccc(CC(F)(F)F)cc2)C)cccc(C(=O)NCC)c1O c1(OC)ccc2c(=NCCC3CC=CC3)[nH]c(=NCc3cccc(O)n3)[nH]c2c1 C1(CNC(c2cn(C)nn2)=O)CC(O)CN1C(c1csc(CC(F)F)n1)=O N(C1CCc2c1ccc(F)c2Br)C(c1cc2c(cc1Br)OCO2)=O c1(C(N2CCN(C(CS(CC)(=O)=O)=O)CC2CCO)=O)nccn2cnnc12 C1(C(N2C(C(C)NC(c3ccc(Cl)cc3Cl)=O)CCC2)=O)CS(=O)(=O)CC(=O)N1 C1(CNC(c2cnc(C)nc2)=O)COC(C)(C)CN1C(C1CCCN(C)C1)=O C(=O)(C1=C(Cl)CC1)NC(CC)(C)CNC(=O)CCc1ncc[nH]1 N1(C(c2ccco2)=O)CCC2CCC(C1)N2C(=O)CCc1ccc(O)c(Cl)c1 N1(C(N)=O)CCCC(C(N2CC(O)(CNC(C34CC(CCO3)C4)=O)C2)=O)C1.C(C)N CC1CN(C(c2cncc(C(C)(C)C)c2)=O)CC(C)CN1C(=O)C(CO)C(C)C N1(C(Cc2cnc(C)s2)=O)C2CCC(C(N3CCCCC(CO)C3)=O)C1CC2 Cc1nc(=N)[nH]c(=NCC2CC(CNC(c3ccncn3)=O)CO2)[nH]1 N1(C(C2CCCN(S(CCC)(=O)=O)C2)=O)CCOC2(C1)CN(C(=O)CN(C)C)C2 C1(N(C)C)CCCN(C(=O)CONC(C2CCOC2(C)C)=O)C1 C1(OC)CC(C)CN(C(C2CCCN(C(=O)CC3CCC(=O)C3)C2)=O)C1 N1(C(CC2CC(=C)C2)=O)CCC(C)C(CC(=O)Nc2ccsc2OC)C1 CC1(C(=O)NCc2ccc(C(=O)NCC3CC4C=CC3C4)cn2)CCC(O)CC1 C1(C(N2C(CC(N3CC=C(C)CC3)=O)CC2)=O)CC12CCCCC2 Cc1nn(CCO)cc1C(=O)NCCC1CC(NC(C2CC3CCC2C3)=O)C1 c1(OCCOCCNC(C2(N(C(=O)Cn3ccnn3)C)CC2)=O)cccnc1 C(N=c1[nH]c(=NCC(CC)C(C)(F)F)c2cccc(F)c2[nH]1)C1C(C(=C)C)OCC1 Cc1ncsc1C=CC(N1CCCCC1CCCNC(C12CC(F)C1C2)=O)=O O=c1ccc2cc(S(=O)(=O)NCC(Cc3ccccc3)C3CC3)ccc2[nH]1 N1(C(c2ccc(I)s2)C(=O)NCC(=C)C)CCC(C(F)(F)F)CC1C(=O)OC CN1CC=C(CC(=O)N2CCCC(C(N3CCC4NCCC4C3)=O)CC2)CC1 c1(C(N(C2CCCN(C(COCCC=C)=O)CC2)C)=O)cnn2c(=N)[nH]cnc12 N1(C(CCOCCOC)=O)CCN(C(=O)COC2CCC2)CC1c1ccccc1 C1(CNC(C2CCS(=O)(=O)N2)=O)CC2(CCC2)CN1C(c1cn2ccsc2n1)=O N1(C(C2CC(N(C)C)C2)=O)CC2(C1)CN(C(C1CN=C3N=CNN3C1)=O)CCO2 C1(NC(Cc2ncn(C)c2)=O)CN(C(=O)CC2=CCCC2)CC2(CC2)C1 C=CC(C)(C)CC(=O)NC1CCN(C(c2ccc(CN(C)C)nc2)=O)C1(C)C N1(C(C=C(CC)CC)=O)CCc2[nH]nc(CNC(c3ccncc3Br)=O)c2C1 c1(-c2nnc(NC(c3ccc(F)cc3F)=O)s2)cc([N+](=O)[O-])ccc1F Cc1cc(C(N2CC3(C2)CN(C(C2Cc4nncn4C2)=O)C3)=O)ccc1C#N n12cc(cn1)C(O)CC2.c1(C(=O)NC(C)=O)cocc1Br.C1(=O)CCN1 c1(C(=O)NC(c2nocc2C(=O)NC2(CO)CCOCC2)C)n[nH]c2c1COC2 CCCC(C)C(=O)NCCCCCN1CCN(C(=O)CC2CCCN2CC)CC1 c1(C(=O)NC2CCCN(C(C3CCN(C)CC3)=O)CC2)ccc2nccnc2c1 C1(C(=O)NCCC(C)NC(C=C(C)Cl)=O)(Cc2ncn(C)n2)CCCC1 C1(C(=O)NCC2(F)CCC(NC(c3c(COC)ncs3)=O)C2)CC12CCOCC2 N1(C(CCC(=O)OC)=O)CC(CNC(=O)C(C)CN2CCCCC2)OC(C)(C)C1 Cn1nnc(C(=O)NC2CCN(C(C3CC(O)(c4ccccc4)C3)=O)C2)n1 c1(C(=O)NCC2N(C(c3c(C)ncc(Br)c3)=O)CC2)ccc2nn[nH]c2c1 C1(O)(C(=O)NCC2C(NC(c3cnc(CC)s3)=O)CCC2)CCCC(C)(C)C1 CC1(CNC(=O)CC2(NC(c3ccncc3F)=O)CCC2)CCC(=O)N1 c1(C(=O)NC2(C)CC(NC(COC(CC)C)=O)C2)cccc(C)n1 N1(C(=O)NCCCOC(C)(C)C)CC(F)(F)C1C1CC1 c1(OC)ncc(Cl)c(=NCC2CC(NC(c3cccc4cnccc34)=O)C2)[nH]1 C(=O)(CCCC(F)(F)C(F)(F)F)N(CCCNC(c1c(C)con1)=O)C CCC(C)(C)CC(=O)NCC(CC(=O)NCC1(CC(N)=O)CC1)OC CC1(NC(=O)NCC2CC(O)(C(c3ccccc3)O)C2)CCC(=O)NC1=O C(CCC(C)C)(C(=O)N1CCC(NC(c2cnc(S(C)(=O)=O)s2)=O)C1)NC(C)=O C(N=c1nc2c(c[nH]1)CCCC2)c1c(C)nc(-c2ccc(C)c(Cl)c2)s1 N1(C(c2nccc(CC)c2)=O)CCC2CN(C(=O)CSCCC(C)C)CC12 n1(C(C)C(=O)NCCC2CC2(Cl)Cl)cc(C2(C)CCCO2)nn1 N1(C(COCC(=C)C)=O)CCCCC(NC(c2ccnn2C(C)CC)=O)C1 CCCC(C(=O)N1CCCC(CCNC(C2(CO)CCOCC2)=O)C1)S(N)(=O)=O N1(C(C(CC(=C)C)C)=O)CCCCC(C2CN(C(c3cncc(Cl)c3Cl)=O)C2)C1 c1(C(=O)NCC2C3CN(C(C(C)=CC)=O)C2C3)cnc2c(n1)CCCC2 N1(C(Cc2ccc(C)nc2)=O)CCC2(CC2)CC1C(N1CCCCC(CO)C1)=O C12CC3(CCN(C3)C(=O)C=CCN3CCC3C(=O)N1)C2.c1(CC)cccc(OC)c1 N1(C(CC)=O)CCN(C)CC1CNC(c1sc(CC2CC2)nc1C)=O c1(C(=O)NC(C)CCCNC(=O)CC#N)ccc(-c2ccccc2)cc1F C1(NC(C(C2CN(C(=O)CCC3CCCC3)C2)OC)=O)CC12CCCCCC2 CC1=C(C(=O)N2CCC(CC(C)C(C3(C(=O)N(C)C(C)C)CC3)=O)CC2)CCC1 c1(C(=O)NCC(NOCC(=C)Cl)=O)ccc(NC)cc1 C12(CC(C(=O)C(O)Cn3cncn3)=O)CC(N(C(=O)C3=C(Cl)CC3)CCC#N)(CO1)C2 n1(COC)ccc(C(=O)NC(c2ccccc2)C(=O)NCC2(N(C)C)CCC2)n1 C=CCN(OC)C(=O)c1cn(CCN(C(=O)C(CCC)OCC)CC)nn1 C(CCC(C(=O)NC(C)CC(C)(C)OC)NC(C1CCC2(CC1)CC2)=O)OC c1(C(N(C)Cc2cn(Cc3cccc(C)c3)nn2)=O)cc2c(C)sc(C)c2s1 C(=O)(C(C)C(C)C(C)(C)C)N1CC2(CC(NC(c3cc(C)c(C#N)cn3)=O)C2)C1 C1(NC(C2C(C)OCC2)=O)CN(C(c2cnn3cccnc23)=O)C2CCCC12 N1(C(N2CCC(CCC)C2)=O)CCC=CC1C(=O)OC(C)C.CCO C1(CC)CC(NC(=O)C(c2ccc(-c3ccccc3)cc2)(C)C)CCN1 N1(C(c2cnn(C)c2C2CC2)=O)CCCOC(CNC(=O)COC2(C)CCC2)C1 Cc1cc(C(=O)NC2CC(C)CN(C(=O)C(C)NC=O)C2)cc(O)n1 N1(C(C=CCC)=O)CC(C2CCN(C(=O)CC3CCOCC3OC)CC2)C1 C=CCN=c1[nH]cc(C(=O)NC(CN(C(=O)Cn2ccc(C)cc2=O)C)CC)s1 CC1=C(C(=O)NC2CCC(NC(c3cncc(C(F)F)c3)=O)C2)CCO1 C(=O)(C1=CCC2(COC2)OC1)NC(C(C)NC(=O)Cn1ccc(C(F)(F)F)n1)C N1(C(C=CCOC)=O)CC2CC3CC2C1C3NC(=O)CCC1C(=O)ON=C1C N1(C(c2c(OC)cncc2)=O)CCC(CNC(=O)COC(C)(C)C)C(O)C1 CC1CN(C(=O)C2=NOCC2)CC(c2nc(N(C)Cc3ncc(F)cc3N)n[nH]2)O1 c1(OC)c(F)ccc(C(N2CC3CN(c4nccc(C)n4)CC3C2)=O)c1F N1(c2n(C)c(=O)nc(O)c2)CCC2CCC(C1)N2C(=O)CCCC1CCCCC1 c1(C(N(C)C2CC2)=O)cc(NC(=O)CC2CCC(C3CC3)O2)ccc1Cl C1(CC)C(=O)NCCCN1C(=O)CC=CCNC(c1cc(C)c[nH]1)=O Cc1ccc2ncc(CNC(=O)C(=O)NC3CCC(N4CCNCC4)CC3)n2c1 C(=O)(CC(C(=O)NCCC(C)CCNC(c1cnsc1)=O)NC(C)=O)OC c1(SC)ccc(C(=O)N(C(C)CCNC(=O)C(C)(C)c2cnco2)C)s1 C(c1ccc(F)cc1)=CCC(N1CC2C(CNC(CCSC)=O)C2C1)=O N1(C(CCN(C)CCO)=O)CCC(C2CC2)C1C(=O)NC1CC2(CCOC2)C1 C1(CNC(c2ccc(COC)o2)=O)CCN(C(C2(C#N)CC2(C)C)=O)CC1(F)F N1(C(c2cc(C)[nH]n2)=O)CCC(NC(=O)Cc2ccns2)C(O)C1 N1(C(Cc2c(C)n[nH]c2C)=O)CCCN(C(C2CCN(C3CC3)C2=O)=O)CC1 c1(OC)ccncc1C(N1CCCC1C(C)NC(c1nccnc1N)=O)=O CC(O)C(C)(C)C(=O)Nc1cccc(NC(C2(n3cncn3)CC2)=O)c1 CCCC(CCC)=CC(=O)N(C)CC1(NC(=O)C(C)OCc2ccccc2)CC1 c1(C(N(C2CC(C#N)C2)CC(=O)NC(c2ncc[nH]2)CC)=O)ccc(Cl)o1 C1(C(=O)NC(C)CCCNC(=O)C(C)(F)F)CCC2CCCCC2C1 c1(C(=O)NCC2(NC(=O)COc3ccccn3)CC2)coc2cccc(Br)c12 C1(CNC(C(C)(C)SC)=O)C2CCC1CN(C(C1CCS(=O)(=O)CC1)=O)C2 N1(C(C=COCC)=O)CCC(c2ccccc2)(NC(=O)C(C2CC2)OC)C1 C(=O)(C1CCN(C)c2ccccc21)NCC1C(NC(c2c(OC)ccnc2)=O)C1 O=C1CN(CC(=O)NC2CCCCC2NC(C2CC3CC2CO3)=O)C(=O)N1 C1(c2cn(CCC=C)nn2)CN(C(C2CC=CCO2)=O)CCO1 C(=O)(C(C)(C)N(C)C)NC(C1(O)CN(C(=O)CCCc2ccsc2)C1)C C(=O)(CCC(C)NC(c1ncn(C)n1)=O)NCc1ncc(C)o1 C=CCCCCCC(=O)N1CCCC(NC(=O)CC2CCCCO2)C1C C1(NC(c2csc(-c3nc[nH]n3)n2)=O)CN(C(=O)CC23CC(F)(C2)C3)CC12CC2 N1(C(C(CC)C)=O)CCCC2(CCCN2C(c2n[nH]c3c2CCC3)=O)C1 C1(C(=O)NCCC(C)NC(=O)Cn2[nH]cnc2=N)(CC)CCCO1 CC1CC(=O)NCC1C(=O)NCCC(C)(C)NC(=O)CCOC1CCCC1 C1(NC(CC2(C)CC2(F)Cl)=O)CCC(NC(=O)C=CCOC2CCOCC2)CC1 C1(C)(C(N2CCCC(C)C2)C(=O)NCC(C)C)CC(F)(F)C1 c1(C(N2CC3CN(C(CC(C)CN(C)C)=O)CC3C2)=O)cc2c(=O)[nH]ccn2n1 N1(C(C2CC=C(C)CC2)=O)C2CCC1C(NC(c1cc(C)n(CCO)n1)=O)C2 c1(CC(N2CC3(CN(C(=O)CCc4cnn[nH]4)C3)C2)=O)cncc2ccccc12 C1(CNC(c2c(C)nc[nH]2)=O)CC2CCC1N(C(c1cc(C3CC3)nn1C)=O)C2 c1(C(=O)NCC2CCCN2C(=O)CC2CC3CCC2O3)cccn2ncnc12 C1(CC)CN(C(c2cc(C)c[nH]2)=O)CCC1NC(C12CC3CC1C2C3)=O N1(C(c2c(COC)nn(C)c2)=O)CCOCC(C(=O)NC(CO)C(C)(C)C)C1 N1(C(c2ccc(N)cn2)=O)CCC(NC(=O)CC2CC(O)C23CCC3)C(O)C1 c1(C(N(C)CC2CCN(C(c3c(C)nc(CC)o3)=O)C2)=O)cc(F)cc(Cl)c1N O=C(C#CC1CCCCO1)N1CCC(CCCO)CC1 CCCC(C(=O)NC(CN(C)C)C(=O)NCc1ccncc1F)C(C)C N1(C(COCCOC)=O)CC(C(=O)NC(C2CCCO2)(C)C)C(C(C)C)C1 C1(NC(C(C)=C(CC)C)=O)CCN(C(C2CC(NS(C)(=O)=O)C2)=O)CC1C C(CCO)(C(F)F)NC(=O)CC(=O)Nc1ccccc1.CC12CN(C1)C2=O C1(NC(C2CCOC2)C)CCCN(C(=O)CN2CCOCC2)C1 N1(C(C2(OCC)CCCC2)=O)CC2C(CC(=O)NCC3COCCN3C)C2C1 N1(C(C(C)NC(CC)(C)C)=O)CC(NC(=O)Cc2ccn(C)c2)CC1(C)C C12(NC(CCNC(=O)OC)=O)CC(C(=O)NCCCc3cc[nH]n3)(C1)C2 C(CN=c1[nH]c(=NCCc2nc(-c3ccncc3)n[nH]2)[nH]c2ccsc12)OCC N1(C(=O)CN(C(=O)CSC2CC2)C2CC2)CCC(c2ccco2)C1 c1(C(=O)NCC2(F)CC(NC(C3C(C(N)=O)CCC3)=O)C2)c[nH]ccc1=O C1(N(C)C(c2cscc2F)=O)CCCC(NC(=O)Cn2nnnc2C2CC2)C1 c1(NC)ncc(C#N)cc1Cl.c1(CN2C(=O)Cn3cc(nn3)C2)cc(Cl)cs1 Cc1ccc(C=CC(=O)NCC(C)CNC(c2c(Br)nnn2C)=O)s1 C1(C)(CC)CCC(C(=O)NC2CC2CNC(=O)CCc2cn[nH]c2)O1 c1(OC)ccc(Br)c2c1C(NCC1CCNC3(CCC3)C1)CC2 C(=O)(C(C)CS(C)=O)NCC=C1CCN(C(C2(C(=O)NCC)CC2)=O)CC1 Cc1cc(C(N2CCCC(N(C(=O)C3=CCOCC3)C)C2)=O)cc(C)c1Cl CC(C)CCC(=O)O.C1(CC(=O)NCO)CCOC1=O.C1C(=O)N1.C1C(=O)N1 c1(C(N(CCNC(C(C(C)C)SCC)=O)C)=O)cc(F)cc2cnccc12 O(NC(=O)C(CCC(C)C)NC(=O)C(C)NC(N)=O)C(CC)CC c1(OC)ccc(C(CN(C)C)NC(=O)NC(C(F)(F)F)C2CC2(C)C)cc1 C=CCC(C(=O)OC)NC(=O)Cn1cc(-c2cccc(SC(F)(F)F)c2)nn1 C=CC1(C(=O)NCc2cnns2)CCN(C(=O)CC(C)C(F)F)C1 N1(C(C(COC)(C)C)=O)CCN(C(=O)CSCCc2ccccc2)C(CO)C1 N1(C(C(CCC)CNC(C2(CCOC)CCC2)=O)=O)CCC2(CC(CO)C2)C1 Cc1cc(=NC(=O)CN2CCC(F)(F)C(CNC(=O)CC3CC3(C)C)C2)[nH]o1 C1(C(=O)NS(=O)(=O)CCCCCl)CCC2(CCOCC2)O1 N1(C(C(C)(C)CO)=O)CC2CN(C(C3(S(C)(=O)=O)CC(O)C3)=O)CC2(C)C1 CC1CN(C(c2ccccc2-n2cc(CO)nn2)=O)CC1(C)C(=O)OCC(N)=O c1(C(C(=O)NCCOC)N(C2CNC(=O)C23CC3)C)c2ccc(Br)cc2nn1C N1(C(C(COCC)N=[N+]=[N-])=O)CCCC(C2CN(C(c3cc(=O)cc[nH]3)=O)C2)C1 Cc1ccnc(C(=O)NCC(C)C(F)C(=O)N2CC3(CCC3)C2)c1F c1(CC(=O)N(C(CCNC(C(C)OCCC#C)=O)C)C)cc(C)n(C)n1 n1(CCN(C)C)cc(C(=O)NC2CC2CNC(C2(N3CCOCC3)CC2)=O)nn1 C1(C(=O)Nc2cc(F)ncc2F)CC12CCN(C(C1(C3CC3)CC1)=O)CC2 CCCC(CCC)C(=O)N(CCNC(C1CCCC1C1CC1)=O)CCOC c1(C(=O)NCCOCCC(=O)NCc2c(C)n(C)nc2)cc(O)ncc1F C#Cc1ccc(F)c(C(=O)NCCC(CC)(CC)NC(=O)CC2CCOCC2)c1 c1(C(C(=O)N(C2CCN(C(=O)CC3CSC3)C2)CC)C)c(F)cccc1F C1(C(=O)NCC(CCCC)NC(CC2(C=C)CCC2)=O)CCOC(=O)CC1 C=C(F)C1(CC(N2CCC(NC(=O)CCCn3nc(C)cc3C)C2C)=O)CCC1 C12(C(=O)NC(CC=C)(C)C)CC1CN(C(=O)CC1CCCCN1C)C2 c1(NCCC(C)C)c(C(=O)NC2(C)CCN(C(=O)OC(C)(C)C)C2)cccc1Cl C1(OC)CC2(C1)CC(C(N1CC3CC(NC(=O)Cn4nc(C)cc4C)C1C3)=O)C2 C(C)(C)(CC(=O)N1CCN(CCCNC(c2cc[nH]c2C2CCC2)=O)CC1)OC C#CCCCCCCC(=O)N1CC2CC1(C(=O)NCc1nc(C3CC3)no1)C2 Cc1ccc(C(N2CC(NC(c3cc(C)n(C)c3)=O)CC(C)C2)=O)cc1CO c1(SC)ccc(Cl)c(C(=O)NCC2CCC2NC(c2cc(N)cc(O)c2)=O)c1 c1(CC(N2CCN(CCCNC(C(C)SC)=O)CC2)=O)cc(F)c(F)cc1F N1(C(c2c(CC)ccc(F)c2)=O)CCC2(NC(=O)Cc3cccnc3)CCCC12 C12(CCCC1C1CC1)C(c1nnnn1CCOC)N2.C1(C(=O)OCC)(C2CC2)CC1 C1(C(N(CCN(C(C2CCC(C(C)C)CC2)=O)C)C)=O)CC(C)CC(=O)N1 c1(C(N2CCCCC(NC(CN(C)C)=O)C2)=O)cc([N+](=O)[O-])c(Br)cc1F C1(C(=O)Nc2c(C(C)C)scc2)CN(C(=O)Cn2cc(Cl)cn2)CCC1O C1(C(=O)N(Cc2cnn[nH]2)Cc2ccccc2)CC12CCN(CCCO)CC2 Cc1nc(C(N2CC3CC3(CNC(=O)C(C#N)C3CC3)C2)=O)c(=O)[nH]c1C CN1CC(C(=O)NC2(CNC(C3(CCF)CC3)=O)CC(O)C2)NC1=O c1(C(=O)NCC2C(NC(C(n3ccc(C)n3)C)=O)C2)cc(Br)c(C)cn1 C(CCCC(=O)NCC(CC(C)C)NC(C1SCC=C1C)=O)SC c1(-n2ccc(C(=O)NCC3CCN3C(c3ccc[nH]3)=O)n2)ccc(F)c(F)c1F C12(C(=O)NC(C(C)F)C)CCCC1CCN2C(=O)C(c1cnn(C)c1)C C1(NC(c2cnc3nccn3c2)=O)COC2(C1)CN(C(C1C3(CC3)C13CC3)=O)C2 C=CC(CC)C(=O)NC(C(=O)N(C)CC1(OC)CCC1)c1ccoc1 N1(C(CCc2onc(CSC)n2)=O)CCC2(NC(=O)Cc3cnn(C)n3)CCCC12 N1(CC)CC(NC(=O)C(CC2CCC2)NC(=O)C=CC2CCCC2)CC1=O c1(C(C(=O)NC(C2(O)CN(C(C3(O)CC(C)(C)C3)=O)C2)C)CO)ccc(F)cc1 C1(NC(C(C)C2CCCC2)=O)CC2CCC1CC2NC(C1CC1C1CCCO1)=O c1(CC)ccc(C)c(NC(C23CC(CN(C(c4nocc4Cl)=O)C2)C3)=O)c1 C1(C(N(CC(C)NC(c2c(C(=O)OC)n(C)nc2)=O)C)=O)CN2CCC1(C)CC2 N1(C(C(C)(C)SC)=O)CCC2C(C1)CN2C(=O)CC(C(F)(F)F)N1CCOCC1 c1(CC(C(=O)NCC(CNC(CC(=C)C)=O)C)C)ccccc1Cl Cn1cc2c(n1)CC(C(=O)NCC1CN(CCF)CCCO1)CC2 Cc1coc(C(=O)NC2CCC(CNC(=O)C(F)(F)c3cscn3)C2)c1 N1(C(CC(=O)OC)=O)CCC(NC(c2nc(Cl)oc2C)=O)C(CO)CC1 Cc1cccc(C)c1C(=O)NCCC1CCCN(C(=O)C(C)n2cnnn2)CC1 C1(S)CNC(c2ccccc2)CO1.c1ccc(C2CNCCO2)cc1 Cc1cc2cc(C(=O)NCC3CN(C(=O)C(C)(F)C(F)(F)F)C3)[nH]c2cc1Cl C1(CC(=O)NC2C(N(C)C)COC2)CCOC1(C)C S(=O)(=O)(c1ccsc1C(N1CCC(NC(=O)C=Cc2cncs2)C(O)C1)=O)NC Cc1ccccc1C(=O)NCC(=O)NCC(F)CNC(c1sccc1Cl)=O CC1(C)OC2(C(=O)NCCCNC(C34CCCCC3C4)=O)CCC1CC2 c1(C(=O)NCC=CCC(=O)NCc2cn(CC#C)nc2)c(C)[nH]c(C)c1C N1(C(C2(C(N(C(C)C)C)=O)CC2)=O)CCOCC(NC(=O)C2=COCCO2)C1 c1(C(N2CC(O)(CNC(c3ccc(SC)o3)=O)C2)=O)cnc2c(c1)c(C)nn2C S(=O)(=O)(c1ccc(F)c(Br)c1)N1CCN(C2CCN(C(=O)C(F)F)C2)CC1 C1(CCNC(=NCCC)NCCc2cncs2)COC2(CCCC2)O1 N1(C(COCC=C)=O)C(C(=O)N(C(C)C(C)(C)O)C)C2CC(O)C1C2 C1(CC)C(NC(=O)C(C)Oc2cccnc2)CCN1C(=O)CCC=CC(C)C c1(C(=O)NC(C=C)C)ccc(Cl)c(C2=CC(=O)CC(C)(C)C2)c1 c1(C(N2C(C(C)NC(c3cnc(O)o3)=O)CCCC2)=O)cccc2oc(O)nc12 N1(C(C(c2cc(F)cc(F)c2)(C)C)=O)CCCC(NC(C2CCNC2=O)=O)CC1 N1(C(c2c(C)cccn2)=O)CC2CCC(CNC(C3(F)CCOC3)=O)C2C1 C1(C(=O)NC(CCCCNC(=O)Cc2ccns2)CO)CC2CCCC(C1)C2 c1(C(=O)NC2CC(NC(c3c(C(N)=O)nccn3)=O)C2)ccnc2c1CCO2 Cc1[nH]nc2cc(C(N3CCN(C(=O)CC(C)CF)CCC3C)=O)ccc12 c1(C(N2CCCC(NC(C3CC4CC4C3)=O)CC2)=O)c[nH]c2cc(O)ccc12 C1(NC(c2ccsn2)=O)CC(NC(c2ccnc(O)c2Br)=O)C12CCC2 CCC(CC(C)C)C(=O)NC(CN(C)C(c1sc2ccsc2c1C)=O)CC C1(NC(C2CCN(C(C)C)CC2)=O)CCN(C(c2cnc(N)c(Cl)c2)=O)C1(C)C C1(S(=O)(=O)NC(C2CNCCO2)C)(C(=O)OCC)CCC1 c1(-c2cn(C(C)CC(N)=O)nn2)cccc(Cl)c1Cl c1(CC(=O)NCCCCCCNC(CCS(=O)(=O)NC)=O)ccc(C)c(F)c1F Cc1nn(CC(=O)NC(C(C)NC(C2(O)CCC2)=O)C(C)C)c(C)c1[N+](=O)[O-] CC(C)(C)C(CNC(=O)CCC(F)(F)F)C(=O)NC1CCC2CCC12 c1(NC(c2cccc3nccn23)=O)cccc2ccoc12 C1(NC(C(Br)=C(C)C)=O)CN(C(=O)CCC(C)C#N)CCC12CCC2 CCCCCS(=O)(=O)CC(=O)NCC(C)CN(C(=O)CC12CC(C1)C2)C C(C(F)(C(=O)NC(C)C(=O)NCCF)C(C)C)NC(c1c(CC)cccc1)=O CC(C)C(C(=O)NC(C)CN(C(=O)Cc1n[nH]c(=N)s1)C)c1ccncc1 c1(OC(C)(C)C)ccc(NC(N)=O)cc1CNC1CCC(C)(c2ccccc2)C1 N1(C(C2(O)CC(C)(C)C2)=O)CCCC(C2CN(C(c3sccc3CC#N)=O)C2)C1 CN1C2CCC1CN(C(=O)C(CO)NC(c1ccncc1N)=O)CC2 Cc1cc(NC(=O)CC2(NC(=O)Nc3ccncc3)CCC2)cc(NC(C)C)c1 c1(OC)cnncc1C(=O)NC(C1CCN(C(C2CCC(=O)N2)=O)C1)(C)C CC1CCC(NC(c2cnc(-c3ccccc3)[nH]2)=O)CN1C(=O)CNS(N)(=O)=O c1(C(N2C3CN(C(CC4C(C)(C)CCCC4)=O)C(C3)C2)=O)c(F)ccc(N)c1F CCCC(C)CCCC(=O)NCCCNC(=O)C(c1cccnc1)O C(=O)(CCCCCF)N1CCC(C(C)NC(Cc2cccc(OCC)n2)=O)C1 C(CCC(C(=O)NC1CN(C(C)=O)C1)NC(c1scnc1Cl)=O)OC C(CSC1CC1)(C(=O)NCCC1COCCO1)NC(=O)OC(C)(C)C CCCC(CC(C)C)C(=O)NC1C=CC(C(N2CCC(OCC(N)=O)C2)=O)C1 N1(C(c2nccc(N)c2)=O)CCCC2(NC(c3c[nH]nc3Br)=O)CCCC12 C(CCCCCCO)NC(C(C1CCCN(C(=O)CCC2(C)N=N2)C1)C)=O Cc1cc(NC(C2(C)CCCC2)=O)ccc1NCCC(=O)NC(=O)C(C)C N1(C(c2cnn(C)c2N)=O)CC2CCN(C(C3CC(n4cnnc4)C3)=O)C2C1 c1(OC)c(C(=O)OCC2COCCN2C)c(C)nn1C Cc1cccc(C(=O)NC2(CCNC(=O)C(F)C(C)(C)O)CCCC2)c1C C(C(C)(C)C#CC(=O)Nc1ccc(O)cc1Cl)NC(CCCC#CC)=O C(=O)(C1=CCC(C)CC1)NCCC(C)NC(=O)C(O)CCc1cn[nH]c1 C(=O)(C(CCO)N(C)C)N(CCN(C(=O)CCc1nc(C2CC2)no1)C(C)C)C N1(C(c2n(CC#C)cnn2)=O)CCN(C(c2scnc2Cl)=O)C(CC)C1 C1(C(=O)OC)CC(C(=O)OC)CC(C(N2CCC(CCF)CC2)=O)C1 Cc1cc(C(=O)NCC2CCCC(NC(=O)COCc3scnc3C)C2)n(C)n1 C1(C(N2CCC(C)(CC)CC2)=O)CCC(C)(C)N(C(=O)Cc2nc(=N)[nH][nH]2)C1 C(CC(C)C)(C(=O)N(CC(C)O)CC(C)O)N(C(c1cc(CC)[nH]n1)=O)C c1(CN2C(C)CCC(C(F)(F)F)C2)cc(Cl)cc2c1CCC2 CN1C(=O)CC(NC(C2C(CNC(=O)CCc3cnn[nH]3)C2(C)C)=O)CC1=O CCC(O)C(C)C(=O)N1CCC(C(C)(C)NC(=O)Cc2cnn(CC)c2)C1 C1(C(=O)NCc2c(COC)ocn2)CCCC(NC(=O)CN(C)C(=O)OC)CC1 C(C1CCCCCC1)=CC(N1C(CO)CC(NC(Cc2c(C)noc2)=O)C1)=O C1(NC(c2cncc(CNC(=O)CCc3cnccn3)c2)=O)CCCCC1(F)F C1(CNC(CNS(N)(=O)=O)=O)CC2(CO1)CN(C(c1cc(Cl)c([N+](=O)[O-])[nH]1)=O)C2 c1(OC)ccc(C=CC(=O)NC2CCC(N(C(=O)C(C)OC)C)CC2)cc1O c1(C(=O)NCC(CC=C)NC(=O)CC2COCCN2C)cc2c(C)nn(C)c2s1 C1(CNC(COCCCCC)=O)COC(C)(C)CN1C(c1cccc(C)c1)=O C12CN(CCC1C)C(=O)C2.C1(CCC)(CC)CCCN1C(=O)CCC1CC1 Cc1ccc(C(=O)NCC2CN(C(=O)CC(c3cccc(F)c3)O)CCO2)nc1 C1(NC(C(c2c(C)n[nH]c2C)C)=O)CC2CC(C1)N(c1nnc(C#N)s1)C2 c1(CC(=O)NC(c2nn[nH]n2)C2CC2)ccccc1OCCCC#N CC(C)C(O)CC(=O)NCC(F)CNC(c1cc(-c2ccncc2)no1)=O C=CC(CC)CC(=O)N1CCCC(CN(C)C(c2coc(-c3cn[nH]c3)c2)=O)C1 C1(C)(C(=O)NCC2N(c3ncc(OC(C)C)cn3)CCC2C)CCCCCC1 c1(C(=O)N(CCN2CCN(C(c3ccncc3)=O)CC2)CCO)cc2cccnc2o1 c1(C(=O)NCC2COCCN2C(=O)C#CC2CC2)cc(=O)c2ccc(Cl)cc2o1 N1(C(c2cncc(OCC)c2)=O)CCNc2ncccc21 c1(OCCC)cccc(C(=O)NCCC2CCN(C(=O)C(C)c3ccsc3)C2)c1 C1(C(N(CCCNC(C(CSC)OC)=O)C)=O)CC2(C)CC1CO2 C1(CNC(C2CC(CN(C)C)C2)=O)C2CN(C(=O)C(F)n3ccnc3)CC12 N1(C(C2CN(Cc3c(C)cccn3)C2)=O)CCCC2CCCCC12 N1(C(C(CSC)O)=O)CCC2(CC1)CCN(C(C1CCC3(CCOCC3)C1)=O)C2 c1(C(N2CC(F)(CNC(CC(C)C(C)(C)C)=O)C2)=O)cc2c(F)c(F)ccc2[nH]1 c1(C2(CC=CC(=O)NC3(CCOCC)CCC3)CC2)ccc(C(=O)O)nc1 CC(O)(C(=O)N1CC(NC(=O)CCCc2ccc(F)cc2)C(F)(F)C1)C(F)(F)F C(=O)(C1=CCc2ccccc21)N(CCN(C(CCN(C)CCO)=O)C(C)=O)C(C)C c1(C(=O)NC2CC(NC(C3C(C)(CC)C3)=O)C2)cc(C)nn1C c1(C(=O)NC23C(CN(C(c4ncc(NC)nc4)=O)C2)C3)ccc2c(c1)CCC2 c1(CC(=O)NC2C3(CC(NC(CCNC(COC)=O)=O)C3)C2)cccc(C)c1C C1(C2(C)CC2)CC(O)CN1C(C1CCCN1C(C1CCC(F)(F)C1)=O)=O C(=O)(C(C)(C)C(=O)NCC(CC(F)(F)F)NC(=O)C=Cc1ccc(F)cc1)NC C1(N(C(C2CC(SC)C2)=O)C)CN(C(=O)C=C2CCN(C)C2)CC1F Cn1nc(C(F)(F)F)cc1NC(C12CC1CN(c1ncc(Br)cn1)C2)=O CCCC(C)(C)C(=O)N1CCCC(C)(C(=O)NCc2noc(C3CC3)n2)C1 c1(COCC)nnc(N2CCOC3CC23)n1C1CC1 c1(C(=O)Nc2ccc(-n3c(C)ccn3)cc2)cc2cccc(C)c2s1 C1(CCNC(CCCOC)=O)C(C)CCCN1C(C1CCCCC1)=O N1(C(C(CCO)N(C)C)=O)CCCN(CCNC(=O)C(F)CC2CCCC2)CC1 N1(C(=O)CC(F)(F)C(F)F)CC2CCN(C(C3(CF)CCOCC3)=O)CC2C1 C1(CNC(c2ccco2)=O)CC2(CCC2)CN1C(c1sccc1OC(F)F)=O C(C)(C(C)(C)C(=O)N1CCCC1CCN(C)C)NC(C(CO)NC(C)=O)=O CN1CC(C(=O)NC2CN(C(=O)C=Cc3ccc(=N)[nH]c3)CC23CC3)CCC1=O N1(C(c2c(C)cc(F)s2)=O)CCC2CC(NC(c3csnn3)=O)CCC2C1 c1(NC(C(n2cc(CN3CCC(=O)CC3)nn2)C)=O)cc(=O)[nH]c2cc(F)ccc12 C1(CNC(C(C)NC(C)C)=O)CCC2(C1)OCCO2 N1(C(C2CN(C(C)=O)C2)=O)CC2CC3CC2C1C3NC(c1n[nH]cc1Br)=O c1(C(=O)NCCCCC(C)NC(C(COCC)C)=O)ccc(F)c(Cl)c1N CCCC(C)(CCC)C(=O)NCCNC(C1CN(C(C2C=CC=CC=C2)=O)C1)=O N12CCCC(C)(C1)C2.N1(C(=O)OC(C)(C)C)CCC2CC12C(F)(F)F c1(NC)c(C(=O)N(C(C)CCNC(c2c[nH]cc2C(F)(F)F)=O)C)cccc1F C1(C(N(C(C)CCNC(=O)Cc2cncs2)C)=O)OCCN(C)C1=O c1(CN2CC(O)(CNC(c3c(C)cc(Br)cc3Cl)=O)C2)ccc2nc(O)[nH]c2c1 c1(NC(C2C(NC(c3c(O)ccc(C)c3)=O)C2)=O)cc(Cl)c(Cl)cc1I C12(NC(=O)C3=COCCO3)CCCC1N(C(c1nc3ccccn3n1)=O)CC2 Cc1cc(CC(=O)NCCCC2CCN(Cc3ccccc3)CC2)n(C)n1 CC(C)(CC(=O)N1CCC1CNC(C12CCC1CC2)=O)C1CCCCC1 c1(C(=O)NCC2OCCN(C(CC3(C)CCC3)=O)C2)cccc2c1CCC2 C1(OC)CC2CC1CN(C(c1conc1CNC(c1cnccn1)=O)=O)C2 N1(C(C(CSC)OC)=O)CCCC(C)(C)C1CNC(=O)C(=O)N=S(C)(C)=O C1(O)(CN(C)C(C2(F)CCOC2)=O)CCN(C(=O)CCc2ccc(Cl)cc2)CC1 c1(C(N(CC(C)N(C(c2cnc(NC(C)=O)o2)=O)C)C)=O)nn(C)c(N)c1C c1(CC)ccc(C(=O)NCC2(NC(c3cc(OC)n[nH]3)=O)CCOC2)cc1Cl C(=O)(CCC(=O)N1CC(NC(=O)Cc2c[nH]nc2O)CC1C)N(CCC)CCC C1(C(C)NC(C2(C(N)=O)CC2)=O)CCN(C(c2ccc(CCF)cc2)=O)CC1 CC1(C)CC1(c1ccccc1)C(=O)NCC1CN(C(C2(CF)CCC2)=O)C1 c1(C(=O)OC)ccc(OC(C)CCF)c(C)c1 N1(C(c2cnc(CC)s2)=O)CCCN(C(=O)CCCC(=O)N(C)C)CC1C Cc1cc(F)c(C(N2CCC(C)C(NC(c3csc([N+](=O)[O-])c3)=O)C2)=O)cc1F c1(C(=O)NCC2(F)CC(NC(COC(CC)C)=O)C2)ccc2nnc(O)n2c1 C1(O)(CCC2(C)CN(Cc3cccc(N4CCOCC4)c3)C2)CCCCC1 C(=O)(CCC(C)C#N)N(CCC(=O)OCC)C1CC1 N1(C(C2CC(NC(C(n3cc(CC4CC4)nn3)C)=O)C2)(C)C)CCCC1C(C)O C1(C)(NC(C2C(OC)C2)=O)CCN(C(c2cc(C3CC3)on2)=O)CC1 N1(C(=O)CCn2cc(-c3ncccn3)nn2)CC(CO)C(CO)C1 N1(C(C(C)(C)N(S(C)(=O)=O)C)=O)CC2CC1CN2C(c1cncn(C)c1=O)=O c1(CC(=O)OC)ccc(C(F)(F)F)c(NC(=O)NC23CC(N=[N+]=[N-])C2C3)c1 C1(S(N)(=O)=O)(C(N(C)CC2CN(C(C3CCCCN3C)=O)C2)=O)CCC1 C1(CNC(c2ccc(SC)o2)=O)CCC2CN(C(C3CCOC3=O)=O)CC12 N1(C(C(C)=C(C)C)=O)CCC(C2CCCN2C(C2CCC(C)(C)C2)=O)CC1 N1(C(Cc2c(SC)cccc2)=O)CCC2(CC1)CN(C(=O)CC1CCOC1C)C2 C#Cc1cccc(C(=O)NC2CC(CCNC(c3ncccc3F)=O)C2)c1F c1(C(N2CC(CCC)N(C(=O)C(C)=C(C)C)CC2)=O)oc2cc(Cl)ccc2c1C C1(CNC(CCCC#C)=O)C(C)CCCN1C(=O)C(C)N(CC(F)(F)F)C N12CCCN(CC1)C(=O)C2.c1(CCC(=O)OCC(=O)NC)nnc(C)n1C C1(NC(c2cc(CO)[nH]n2)=O)CCC2CCN(C(C3(CO)CCC3)=O)C1C2 N1(C(C2C(C)(COC)C2)=O)CC2CC(C1)C2NC(c1cc(O)cc(F)c1)=O Cc1[nH]nc(C(N2CCCC(C3CCCN3C(=O)C=C3CCC3)C2)=O)c1Cl C1(NC(C)Cc2cccs2)CCC(NC(C2(C)CC(C(F)(F)F)C2)=O)C1 C1(C(=O)N(c2ccncc2)Cc2ccco2)CSc2ccccc2O1 c1(C(CC(=O)N(CCCN(C(CC(C)O)=O)C)C)C2CC2)ccc(F)c(F)c1 C(=O)(CCCC(=O)NC1(C)CCN(C(C2CCC(O)C2)=O)CC1)NC(C)C N1(C(C2(CNC(=O)C=CCCC)CC(=C)C2)=O)CC2CC(OC)C(C2)C1 c1(C(N2CCN(C(CC(CCCC)O)=O)CC2CC)=O)sc2ccccc2c1Cl N1(c2ncc(C)cn2)CC(NC(=O)C(CO)c2ccccc2)CC(C)C1 CC(C(=O)NCC(O)CC(=O)N1CC(N(C)C)C(C)C1)C(C)(C)C c1(C(=O)NCC2N(C(CSCC)=O)CCCC2C)c(F)cccc1[N+](=O)[O-] c1(CC(=O)NCC2(F)CN(C(CC3(C=C)CCC3)=O)C2)cn2c(n1)CCCC2 C1(C(=O)NC(CNC(c2ccnc(C(F)(F)F)c2)=O)C2CC2)CC2(C1)CC(F)C2 C1(C(N2CC(C)(NC(C(C(C)C)C)=O)C2)=O)CC(c2ccccc2[N+](=O)[O-])=NO1 C(C(C)(COC)C(=O)N(C)CC1CN(C(c2nnn(C)c2N)=O)CCO1)OC N1(C(C(c2ccc(OC)cc2)=O)=O)CCCC(NC(c2cc(C)sc2C)=O)C1C c1(CCC(N2C(CCCNC(C3CCSC3)=O)CCC2)=O)nc2ccccc2[nH]1 N1(C(CN(C(C(C)OCC=C)=O)CC)=O)CCN(C(c2conc2CC)=O)CC1 N1(C(C(C)OCC#C)=O)CC2CCC1CN2C(c1c(C)[nH]c(C(=O)O)c1C)=O Cc1cc(C(N2CCCC(CNC(=O)C(F)C(F)(F)F)CC2)=O)c2occc2c1 N1(C(C(C)C2CC2)=O)CC2(CCN(C(c3ccc(F)cc3O)=O)CC2)C1 C1(C)(CNC(=NCc2c(Br)cn(C)n2)NC2CCCC2)COCC2CCCN12 n1(CC(=O)NC2CN(C(C3(SC)CC3)=O)CC2C)c(C)cc2ccccc12 C1(C(N)=O)CCCC(C(N2CC(O)(CN(C(=O)CC3CCOC3)C3CC3)C2)=O)C1 C(=O)(CS(=O)(=O)C1CC1)NC1(CC(=O)NC(C2CCOC2)C)CC1 C(=O)(C(F)CC(C)(C)C)NCCn1ncc(C(=O)NC(C)CC(N)=O)c1 N1(C(C(C)NC(=O)NCc2c(CC)c[nH]n2)=O)CCN(C(C)C)CC1 Cc1cnc(C)c(C(=O)NC(C2CCCN2C(=O)CC2CCCCC2)C)c1 c1(OC)ccc(CCC(N2CCC(C(=O)Nc3cnccc3Br)C2)=O)c(C#N)c1 c1(C(=O)NCCN(C(c2cnc(CCCC)s2)=O)CCC)cc(OC)n(C)n1 CCC(C)(C(=O)O)N(C(=O)CC(O)c1cn(Cc2cccc(Cl)c2)nn1)C c1(NCCNC(=O)NCC2(c3ccc(OC)nc3)CC2)cc(F)c(C)cc1Cl C(C)(CCC(=O)NC1(CCNC(=O)C(=O)NC2CC2)CCC1)OC c1(OC)ccccc1CCC(N1CCOCC1CNC(=O)C=CC1CCOC1)=O C(=O)(C1COc2ccc([N+](=O)[O-])cc21)NCC(CC)(C)NC(=O)C(C)(C)O N1(C(COC(C)=O)=O)CC2CCC(CNC(C3(C)CSC3)=O)C2C1 C(C(C)(O)CC(=O)N1CCCC(CCC(=O)NCC(F)(F)F)C1)OC N1(C(CCP(C)(C)=O)=O)CCN2C(=O)C(NC(c3cnc(=N)[nH]c3)=O)CC2C1 C(=O)(C1=NNC(=O)C1)N(CCC)CCNC(=O)CC1(c2ccon2)CC1 CC1(C)CC(C(N2CC=CCC2)=O)CCN1C(=O)CCn1cccc1 N1(C(C2CN(C(C(=Cc3ccco3)C)=O)C(C)(C)C2)=O)CC2CCC(C1)C2O c12ncccc1NC2=O.C1(CNC(C(=O)N(C)C)=O)CCCSCC1 C1(CC(=O)NCCO)CN(C(c2ccnc(CO)c2)=O)CCO1.C(CSC)OC c1(CNC(c2c(CNC(C3(COC)CCOC3)=O)cc[nH]2)=O)nn(C)cc1SC c1(C(N(C2CCC(NC(C3CC34CCC4)=O)CC2)C)=O)cc(Cl)cc(F)c1N C(=O)(CN=c1[nH]c(=NCCc2nncn2CCC)[nH]c2cccnc12)NCC=C C=C(C)C1CN(C(=O)CS(=O)Cc2ccc(Oc3cccc(Cl)c3)cc2)CCO1 CC1OCCC1CNCC(=O)NC1CC(CC(=O)N(C)C)C1 Cc1c(F)ccc(C(=O)NCC2CCCN2C(=O)Cc2ccc(Cl)cc2F)c1Cl c1(CCN(CC(CN(C(C2C(CC)C2)=O)C)O)C)nc(CC(C)C)no1 n1(C(C)C)ncc2cc(NC(=O)C(C)Cc3ccncc3)ccc12 CS(=O)(=O)c1ccnc(NCC2CN(C(C3C=CCC3)=O)C2)n1 C1(CNC(C2N(C(Cc3n(C)ccc3)=O)CC=C2)=O)CC12CCOCC2 C(C1=CCN(C(=O)CCN2CCCC2)CC1)NC(c1cncc(CC)c1)=O CC(=O)CCCC(=O)NCC1CN(C(=O)CCSC(F)(F)F)C2CC12 C1(CCN2CCN(C(=O)C(F)(F)F)C3C2C3)CCc2cccnc2C1 C1(Cn2cc(C3CCN(C(CC4(NC(C)=O)CC4)=O)C3)nn2)CC(C)(C)C(=O)O1 N1(C(C(C)=C(C)C)=O)CCC(C(=O)NCc2ccnc(O)c2)CC1(C)C N1(C(C2(F)CCN(Cc3cc(OCC)c(O)cc3)C2)=O)CCCC(F)C(F)(F)C1 C1(N(CCCN(C)C=O)C)CC2CC1CN(C(=O)CCOc1cccnc1)C2 C1(CNC(c2c(Cl)cn(CCC)n2)=O)CC(C)CN(C(C2C=CCS2)=O)C1 c1(C(=O)NC2CCC(CNC(Cc3nn(C)c(Cl)c3)=O)C2)cnn2c1CCCC2 c1(C(N2C(CC(=O)N(CC)Cc3cnn(C)c3)CCC2)=O)ccc(C)nc1N c1(CC=CC(=O)OCCN2CCOCC2)cccc(Br)c1.C12CCCN1OC2=O CCC(C(=O)N1CCC(n2cccn2)(CNC(=O)C2=COCC2)CC1)C(C)C c1(OC)c(C(=O)NC2CC(CC(=O)NC3CC(NC(=O)CO)C3)C2)cnn1C C1(C(=O)NCCC2(O)CCN(C(=O)C(O)CCSC)C2)(CC)CC(C)(C)C1 N1(C(C2(CCC)CC(=O)C2)=O)CCC(F)(C(N2C(CO)CC2C)=O)C1 Cc1cccc(C(C)(C)C(=O)NCC2CCCC(NC(=O)C3=NOCC3)C2)c1 c1(C(N2CCC(CNC(C34CCCC3NCC4)=O)CC2)=O)cccc(Cl)c1F N1(C(C2=C(C)OCC2)=O)CCn2ncc(CNC(c3ccc(Cl)c(Cl)c3)=O)c2C1 C1(CNC(CCOCCOCC)=O)(COC)CCN(C(C2OCC2(C)C)=O)CC1 N1(Cc2cnc(C#N)cn2)CC2CCCC2(NC(c2cn(C)nc2C2CC2)=O)C1 C1(NC(c2[nH]cc3c2CCS3(=O)=O)=O)C2CC3CN(C(c4cc[nH]n4)=O)C1C3C2 CC(Cc1cnc[nH]1)C(=O)NCC1CN(C(c2ncoc2C2CCC2)=O)C1 C(=O)(CCCC(=O)NCCCNC(C1CCCCN1C)=O)N(C)C C1(Cl)(C(N2CCCC(CNC(CCCCOCCC=C)=O)C2)=O)CC2CCC1O2 CCC(CC(F)F)C(=O)NCc1cn(C2CCCCN2c2ncc(Br)cn2)nn1 N1(C(CCc2n(C)cnc2)=O)C2CCCC1CN(C(C1CCCCS1(=O)=O)=O)C2 Cc1nc(C2CCN(CC(C)Cn3cccn3)CC2)sc1C(=O)Nc1nn[nH]n1 N1(C(c2nc(C)co2)C(=O)NC(c2ccccc2)C)CC(CO)OCC1C C1(C(N(C2CN(C(CCCOC)=O)C2)C)=O)Cc2cccc(F)c2O1 Cc1[nH]nc2c1CCC(C(N1CC(NC(c3ccn(CCF)n3)=O)C(O)C1)=O)C2 c1(C(=O)NC(C)CN(C(=O)CC2(O)CCCOC2)C)cc2cscc2s1 c1(C(N2CC(C)C(CNC(=O)CC3CCOCC3)CC2)=O)c(N)cc(Cl)cc1F CCCCCCC(=O)NCC1C2CN(C(c3nc(C)oc3C)=O)CC12 C(=O)(C(C)CC(C)(C)C)NC1CCCN(C(c2nc(CCC)sc2)=O)C1 Cc1cnc2n1CCN(C(=O)C(c1ccnn1C)NC(=O)CCn1cnnn1)C2 N1(C(c2cc(NC(C)=O)ncc2)=O)CCC2(CCCC2NC(c2cscn2)=O)C1 Cc1ccc2nc(C(=O)NC3CN(C(=O)CN4CCC4C)CC3C)ccc2c1 c1(C(N2CC(O)(C(C)NC(CC3(C=C)CC3)=O)C2)=O)cc(C)c2c(c1)CCCN2 c1(CC)cncc(CNC(C2(NC(=O)Cc3c(C)noc3C)CC(F)C2)=O)c1 C1(C(N2CCC(C)(CNC(c3cncnc3C)=O)C2)=O)(CC)CNC(=O)C1 Cn1ccc2[nH]c(C(=O)NC3CC(NC(c4c[nH]c(=O)cn4)=O)C34CCC4)cc12 N1(C(C(CNC2CCN(CC)CC2)O)=O)CC2CC1CS2=O c1(CC)ccc(C(=O)NN(C(=O)C(C)OCCOC)C(C)CSC)c(N)c1 C1(c2n(-c3c(OC)cccc3)nc(C3CC34CC4)n2)CC2(CCC2(OC)OC)C1 C12CCN(CC1)C2=O.C1(C(C)(C)C)(CN(C(=O)Cc2cn(C)nn2)C)CCCC1 c1(CC)ccc(C)c(C(=O)NC(C2CCCC2)CNC(c2cc(Cl)no2)=O)c1 C1(C2CC2)(NC(COCCC#C)=O)CCN(C(=O)C(C)SC(C)C)C1 c1(CC)conc1CC(=O)NCC1CCCN1C(=O)CC1CCC1 n1(CC)ccc(CC(=O)NC2CCC2CC(=O)N(CC(CC)OC)CC)n1 C#CCC(C)(C(=O)N=c1cc(OC)n(C)[nH]1)NC(=O)CC1CCC(C#N)C1 C1(C)(C(=O)NC2(C)CN(C(C3CC3F)=O)C2)CCN(C(=O)C(C)(C)C)C1 c1(C(=O)NCC(CC)NC(=O)C(F)(F)c2nc(C)cs2)ccccc1C(C)(F)F C1(CN(C(c2cc(OC)n[nH]2)=O)CC)CCCCN1C(=O)CCCF CCCCCCCCCC(=O)NCC1CCC(N(C)C(C2CC(C)CO2)=O)CC1 C1(C(C)CNC(=O)Cn2ccnc2)CCN(C(=O)C(C2(O)CCCCC2)O)CC1 C1(COC)(CNC(=O)CCn2ccc(C)n2)CCCN1C(c1ccccc1)=O c1(C(=O)NC(C(=O)N(CC(C)N(C(C)=O)C)C)C(C)O)ccc(=O)n(C)n1 c1(C(=O)NC(CNC(c2cc(C)ncn2)=O)C(C)C(C)C)ccc(C)c(Cl)c1Cl C1(O)(CNC(c2c(CC)nn(C)c2Cl)=O)CCCN(C(=O)CCC(C)OC)CC1 C1(C(=O)NOCCCF)(CC)CCN(C(=O)C(C)(C(C)C)OC)CC1 N1(C(C2(OCCOC)CC2)=O)CC2CC1CN2C(=O)C=Cc1ccnn1C C1(C(=O)NCCNC(CC(C)C(F)F)=O)CC2CCC(C1)C2F c1(C(N2C(CC(=O)NC(C(C)C)c3ncc[nH]3)CCC2)=O)cccc[n+]1[O-] C#CCCC(C(=O)NCCc1ccc(C)nc1)NC(C1C=CCC1)=O C1(C(=O)NCCCN(C(CN(CC)CC)=O)CC2CCCC2)CCSC(C)C1 C1(COC)(OC)CCN(C(c2cc3n(n2)CCO3)=O)CC1 C1(O)(C(C)NC(C=CSC)=O)CCN(C(C2CC(C)CO2)=O)CC1 C(=O)(C(CC(C)C)n1ccnc1)NCCCCN(C(C(F)=CCC)=O)C c1(C(N(CC(CN(C(C(COC)C)=O)C)O)C)=O)cn(CCC#N)c(=O)nc1O C(=O)(C1=C(c2ccccc2)CCCC1)N(CCNC(=O)Cc1conc1C)CC CC(CNC(N1CCOCC(C(=O)O)C1)=O)CC(F)(F)F c1(CSC)cc(C(N2CC3CC2CN3C(=O)CC(C)(C)CCOC)=O)ccc1F N1(C(C2CC3(C2)CC(F)(F)C3)=O)CCC2OCCN(C(=O)C(O)C3CCC3)C2C1 CC1=C(C(=O)NC2C=CCN(C(c3oc(C)nc3C)=O)C2)CCC1 C1(NC(CC2CC(=C)C2)=O)CC2CCC1CN2C(c1cnc(OC)nc1C)=O C1(OC)C(O)CC1N=c1[nH]c2ccccc2nc1N1Cc2ccncc2C1 CC1(C)CCC(C)(C)N(C(C2CCC(CC(F)(F)F)CC2)=O)C1 C1(N(C)C(C2CCC(NC(=O)CC3(C#N)CC3)C2)=O)CCCC1(C)O C(CCC(=O)NC(C)(CNC(=O)CSCC(N)=O)C1CCC1)OCCOC CCC(O)C(C)(C)C(=O)N1CCN(C(c2ccnc(S)c2)=O)C(CO)C1 N1(C(CS(=O)(=O)NCC)=O)CCN(C(=O)CCC2CCOC2)CCC1C CC(C)C(O)C(C)C(=O)NCCC(C)(C)C(=O)N1CCC(CO)C(C)C1 N1(C(C(C(COC)C)C)=O)CCCN(C(=O)Cc2cc(OC)ccc2Cl)CCC1 C1(CC(=O)NCC(CC)NC(c2cnc(C3CC3)s2)=O)(OC)CCOCC1 C1(C(=O)NC2CCCN(C(C3(CC(=O)OC)CC3)=O)CC2)CCN2CCOCC12 CC1(C)NC(=O)CC1C(N1CCCC(C)(CNC(c2ccnc(S)c2)=O)C1)=O N1(C(C2CC(C#C)(O)C2)=O)CC2CCC(CNC(c3cc(O)ncn3)=O)C2C1 CCC(CC(=O)NCCCCC1CN(C(=O)CNc2nccs2)C1)C(C)C N1(C(C(=O)NC2(C)CC2)CCc2ccco2)CCCC(CO)(CO)C1 c1(C(N2CCC(C)C2CNC(=O)CC(Cl)Cl)=O)ncc(F)cc1F C(C(C)(COC)C(=O)N1CCC(C(C)C(=O)NC(c2nccs2)(C)C)C1)OC N1(C(C(C)NC(c2ccco2)=O)=O)CCC2CCN(C(=O)CSC3CC3)CC12 CCC(CC(=O)N(CC(C)(C)CNC(C1CC(=C2CCC2)C1)=O)CC)SC C1(NC(C=CCC)=O)COC2C(NC(c3c(F)ccc(F)c3OCC)=O)COC12 S(=O)(=O)(c1ccc(Br)c(Cl)c1)N1CCC2(C(C(=O)NCc3ccc(Br)cc3)C2)C1 C(CCC1CC1)(C(=O)NCc1ccc(O)cc1)NC(c1cn(CC)nc1)=O Cc1nn(C)c(Cl)c1CC(=O)Nc1cccc(NC(c2cc(C(N)=O)c[nH]2)=O)c1 N(C(=NCCOC1CCSCC1)NCc1ccccc1)C1CC(C(N)=O)C1 CC1(C)CC(C(=O)N2CCCC2(C)CNC(c2cc(O)ncn2)=O)=NO1 c1(C(N2CC(C)(CCC(=O)NC3C(C)C3)C2)=O)cc(O)cc(F)c1 c1(NCC2(CNC(C3(C)CC4CCC(C3)S4)=O)CC2)nccc(S(C)(=O)=O)n1 N1(C(C(=O)NCCOC(C)C)=O)CC2CC2(NC(=O)C(C)C2CCC2)C1 C(=O)(CCCC(C)=O)NC(COC)C(=O)N(C)CC1CCC(C)CC1 c1(C(=O)NCC2(F)CC(NC(C=C(CC)CC)=O)C2)cnc2c(c1)ncn2C C1(CCNC(CNC(N)=O)=O)CC(F)(F)CN1C(C1OC2CCC1CC2)=O C1(CNC(=O)Cc2cncnc2)CC2CCC(C1)N2C(=O)C1=C(Cl)CCCC1 C1(C2CCC2)(C(=O)NC2C(OC)CN(C(=O)C(C)(C)COC)C2)CC1(F)F Cc1ccc(C(O)C(=O)NCCC(O)CNC(=O)C=CC2CCCC2)cc1 C(=O)(C#CC1CCOCC1)NCC1(NC(C2C(OC)C2)=O)CCC1 N#CC1CCCC(C(N2CCCC(C(=O)NC3CCC=CCC3)C2)=O)C1 c1(C(N2CC(O)(C(C)NC(C3CCCN(C(N)=O)C3)=O)C2)=O)ccc(=O)n(C)c1 Cc1cc(CC(=O)N(CC(O)CNC(C2(O)CC2(C)C)=O)C)ccc1Cl N1(C(CCCOCC=C)=O)CCC(O)(CNC(c2cccc[n+]2[O-])=O)C1 N1(C(Cc2ccc(C)nc2)=O)CCN(C(c2n[nH]c(C)c2Cl)=O)CC1C c1(C(N2CCCC(NC(C(C)(C)NC(=O)OC)=O)C2)=O)cc2n(n1)CCNC2=O c1(COC)cc(Cl)c(Cl)cc1Nc1cc(C(=O)OC)ccc1C.C12CC1C(=O)N2 c1(CCCC(=O)N2CC(=C(CNC(C3CC(C)(F)C3)=O)F)C2)ccc(F)c(F)c1 Cc1ccc(CCC=O)cc1Cl.N1CCN(C(=O)Cc2ccsc2)C(C2CC2)C1 CON1CC(C(=O)NCC2(O)CC(CNC(=O)CC(C)(C)C3CC3)C2)CC1=O N1(C(CC(C)OC)=O)CCC(C)(C(=O)NCCC(F)(F)F)C1 CC1CCN(C(=O)C=Cc2cnc[nH]2)CC1NC(=O)C=CCN1CCCC1 c1(C(N(C2CCN(C(Cc3c(C)n(C)cn3)=O)CC2)C)=O)ncc([N+](=O)[O-])n1C c1(C(N(CCN(C(CC(CC)C)=O)C)C)=O)cccn(CC(C)C)c1=O C(C(F)C(=O)NCC(CNC(C1(c2cccnc2)CCCC1)=O)OC)N(CC)CC C1(C)(C(=O)NCC2(COC)CCCN2C(=O)CCCC2CCC2)CCCNC1=O C1(NC(CCC(=O)NC)=O)CCC2CN(C(c3ccn(C)c3)=O)CC2C1 N1(C(C(C)Sc2ccccn2)=O)CCC2C1CCN2C(=O)CNc1ccccn1 C12(C(=O)NC(CC)C(=O)OC)CC(CN(C(c3cc(OC)cs3)=O)C1)C2 c1(C(=O)NC(CCCNC(Cc2c(C)non2)=O)C)cc2c(C)ccc(F)c2o1 Cc1cc(CC(=O)NCC2CN(C(C3(C#N)CC3C)=O)C2)nn1C C=C(Br)CC(C)(C)C(=O)NCC1CC1NC(c1ccn(CC(C)C)n1)=O CC(C)(CNC(=O)CCCNC(C1CCCC(=O)N1)=O)C(N)=O C1(NC(CC(CC)(C)C)=O)CC2CN(c3cc(C)c([N+](=O)[O-])cn3)CC2C1 n1(CCC)cc(C(N2CCC(N(C(=O)C(C)CC(C)C)C)C2)=O)c2ccccc12 c1(C(=O)NCC2C(NC(C(C)c3cccs3)=O)COC2)cnn(C)c1Cl c1(C(=O)NCC(CNC(c2c(CCC)nsc2N)=O)C)cccc2cncn12 N1(C(C(CCCC)N(C)C)=O)CCC2(CCN(C(c3ccnnc3)=O)C2)C1 c1(C(=O)NC2CCCN(C(c3cnc(CC)[nH]3)=O)C2)cnc2ccnn2c1N N1(C(CCC=C)=O)CCOC2(CCN(C(c3cnc4cc(C)nn4c3C)=O)C2)C1 c1(C(=O)NC(C(=O)OC)C)n[nH]cc1CNC(=O)CCOC1CCCC1 C(C)(C)(CC(F)C(=O)NCC(C)(O)COC)NC(C=C(CCC)CCC)=O C1(CCNC(c2c(CC)cccn2)=O)CC(F)(F)CN1C(=O)CC1CC(C)(C)C1 c1(OC)cc(N2CC(C)CCC2c2ccccc2)cc(OC)n1 C1(C(=O)NC(C)CNC(c2ocnc2C2CC2)=O)(N(C)C)CCCOC1 CCCC(O)CC(=O)NC1CCN(C(=O)Cn2ccc(C)n2)C1 CC1CCC(=CC(N2CCOC(CCNC(=O)CC3(O)CCCOC3)C2)=O)CC1 N1(C(c2cc(C)cc(C)c2O)=O)CCCCC12CN(C(c1nc(Cl)sc1C)=O)C2 c1(C(=O)NC2CC(CCNC(C(C)CC(C)(C)C)=O)C2)ccc([N+](=O)[O-])c(N)n1 n1(C(C)C)ncc(C(=O)NC2CCCN(C(=O)CC3SC(=N)NC3=O)C2)c1Cl N1(C(CC)CC)C(=S)NC(c2cc(OC)c(O)cc2F)C2=C1C1(CCC1)NC2=O N1(C(C2OCCN(C)C2)=O)CC2CCCC2(C(=O)NCc2ncnn2C)C1 C(C(=O)NC1(CNC(=O)C2=CSCCO2)CCC1)(C(C)(C)C)OC O=S(=O)(c1nc(N2CCC3(CCCCC3)C2)ccc1Br)N1CCSCC1CCO N1(C(c2c(C)c(Br)no2)=O)CCOCC(NC(C2(C)CCCS2)=O)C1 N1(C(CCC(C)C)=O)CCC(C2CC2)C1C(=O)N(C(C)C(N)=O)C N1(C(CCC2OCCN(C(CCC(=O)NCCC)=O)C2)=O)CCCC(C)(O)CC1 c1(CC)c(C)[nH]c(C(=O)CN(CCO)CC)c1C N1(CC(=O)N(CC(CN(C(C(c2ccc(N)cc2)C)=O)C)O)C)CCNC(=O)C1 CCC(CC(=O)OC)NC(c1oc(CNC(=O)Cc2ccn(CC)n2)cc1C)=O c1(C(N2CC(CNC(CNC(CCC)=O)=O)N(C)CC2)=O)cc2nnn(C)c2s1 C#Cc1cn(C)nc1C(N1CC2(C)CC1(C(=O)NC1CCC(C)(C)C1)C2)=O C1(NC(CCC=C)=O)CCN(C(=O)C(c2ccc(F)cc2)F)C(C)C1 c1(C(=O)NCCC2(CNC(c3n(CC)nnc3)=O)CC2)cc2c(s1)CCCC2 CC1CN(C(=O)CCCN2C(=O)CCC2=O)Cc2cccc(Br)c21 c1(C(N(C)CC2CCN(C(C3CCC(=O)N3)=O)C2)=O)cc2c(cc1Cl)NC(=O)C2 C1(N(C(CCC#CC)=O)C)CCN(C(c2ccc(C)cc2Cl)=O)CC1C c1(N2CCOCC(C)(O)C2)ncc2c(=N)[nH][nH]c2n1 C(CCC(C)C)(C(=O)N(C)CC1CCOCC1)NC(CC(CC)C1CC1)=O C1(C(N(CC(O)C(F)(F)F)C)=O)CC2CCC(C1)N2C(C1(F)CCCC1)=O c1(C(N2CC(NC(CC(CC)O)=O)C(F)(F)CC2)=O)ccc(C)cc1[N+](=O)[O-] C=CCCCCCCC(=O)NCCOCCC(=O)NCCc1cnc(C)[nH]1 C(=O)(C(C)(C)CNC(=O)CN(C(C1CCSC(C)C1)=O)C1CC1)NCC C(=O)(C1CCc2cc(F)ccc21)N1CCC(NC(c2n(CC)nnc2)=O)CC1C CCCCCCNC(C1(NC(=O)CC2C=CCCC2)CC(F)C1)=O c1(C(=O)NCCCN(CCC)C(c2cc(C)nn2CC)=O)ncc(C)cc1C N1(C(c2c(C)cc(CC)o2)=O)CCCC(C(N2CCCC(CO)C2)=O)(CC)C1 c1(CNC(C(CC)SC)=O)cncc(NC(=O)C(=O)Nc2ccccc2F)c1 Cc1ccc2sc(C(N3CC4CC(C3)C4NC(=O)CC3CCCO3)=O)c(C)c2c1 C(=O)(C1=C(Cl)CC1)N1CCC(OCCNC(=O)C(O)CN2CCCC2)C1 N1(C(CC2(NC(C)=O)CC2)=O)CCC(C(=O)NCC(O)C(C)(C)C)(CO)CC1 C#Cc1cccc(NC(C)C(N2CCN(C(=O)C(F)n3cccn3)CC2)=O)c1 C1(NC(COCCCOC)=O)CCC12CN(C(=O)C=C(F)c1ccccc1)C2 N1(Cc2cn(C(C(=O)N(CCC)CC3CC3)C)nn2)CCCCC1C(=O)O O=C1CC(=O)NC(C(=O)NC2CC(C(F)C(=O)NCc3ccncc3Cl)C2)C1 Cc1cc[nH]c1C(=O)N(C1CN(C(=O)C(F)n2cccn2)C1)C c1(CNC(=O)C(N2C3COCC2C3)c2cn(C3CCOC3)nn2)ccccc1F C1(CNC(c2cocn2)=O)C(C2CC2)CCN1C(c1csnc1Cl)=O C12(CNC(c3ccc(C)cn3)=O)CCC1CCN2C(=O)CSc1nncn1C C=CC1CN(C(=O)CNS(=O)(=O)CCCC)CC1NC(=O)Cc1ncccc1C c1(CC)cccc(CC(=O)NCCN(C(c2cc(C)c(Br)o2)=O)C2CC2)c1 c1(C(N2CC(NC(Cc3c(C)noc3)=O)C(C)CC2)=O)cnc2cccc(C)n12 C(=O)(C1CCCc2nc[nH]c21)NCC1(F)CC(CNC(=O)CCOC2CC2)C1 CC1C(=O)CC1C(=O)NCC1(NC(=O)CC2CCSC2)CCC1 C1(CNC(CCc2ccn(C)n2)=O)CC2COCC2N1C(c1cc(O)cs1)=O Cc1ccc(C(=O)NC(C)C(N2CC3(CC3)CC2C)=O)cc1O C(CCC(=O)N1CCCC1CC(=O)NCC(C1CC1)SC)OC C1(CNC(C(n2ncc(C)c2)C)=O)CC(O)CN1C(=O)C=CCCC(C)C N1(C(C)=O)CC2CN(Cc3cc(-c4cc(C)c(O)nn4)cs3)CC2(C)C1 c1(OC)c(C(=O)NC(CNC(=O)C=C(C)C2CC2)CC(C)C)cccc1C(F)F c1(OC)ccn2c(C(N3CCC4CC3CN(C(=O)C(C)(C)C)C4)=O)cnc2c1 N1(C(C(CC)CC)=O)C2CCC(C2)C1CNC(C1C=CC=CC=C1)=O Cc1nn(C(N2CC(NC(C3(n4nccn4)CC3)=O)CC(O)C2)=O)cc1[N+](=O)[O-] C1(C(=O)NCC2CC(NC(C(CC(C)C)C)=O)C2)CN2CCN1CC2C C1(NC(C2CC3CCC2O3)=O)CCN(C(c2ccnnc2O)=O)CC1 c1(OC)ccc(CC(=O)NC(C)CNC(=O)CC2CC(C)(C)CCO2)c(C)c1 c1(C(=O)NCC2CC(NC(c3cnn[nH]3)=O)C2)c(Cl)ccc2c[nH]nc12 C(=O)(C(O)(CN(C)C)C(F)(F)F)NC1CC(NC(C(CC)(C)CO)=O)C1 FC(F)(F)CNC(c1ccccc1)CC1CCNC1 C1(C2N(C(C3C(C)C3)=O)CCC2)CCN(C(=O)CCN(C)CCO)CC1 CC1(C)CCCC(C(C)(O)CNCc2cccn2-c2c(Cl)cccc2Cl)C1 C1(NC(C2C(CC)CCC2)=O)CCN(c2ncncc2Cl)CC1F C(=O)(C1=CCCCO1)NC1CN(C(=O)C2=CCCC2)CC1c1cccc(F)c1 C(=O)(C1=C(C#N)CCC1)N1CC(NC(c2c(C)cccc2F)=O)CC(OC)C1 c1(OCC)cccc(CC(=O)NC2CCCC(NC(c3n[nH]c(CC)n3)=O)C2)c1 C1(CC)COCCN1C(=O)C(C)N(C(=O)C1=CCSC1)C N1(C(C2C(OC)CCC2)=O)CCC(=CCNC(C2(C(F)F)CCOCC2)=O)CC1 Cc1ccc2[nH]c(C(=O)NC3(C)CCCN(C(c4sc(F)cc4C)=O)C3)cc2c1 CC(=O)CCCC(C)C(=O)NCC1(C(N2CCC3(CCC(O)C3)C2)=O)CCCC1 c1(CC)cnc(O)c(C(=O)N(C)CC2CCN(C(C3CC3C)=O)C2)c1 C1(C(=O)NCC2CN(C(Cc3cccc(C)c3)=O)C(C)C2)COC2COCC2O1 C1(NC(N2CCC(CC)CC2)=O)CC(C2CNC2)C1 n1(CC(=O)N(CC(C)CNC(=O)C2=COCCO2)C)sc2ccccc2c1=O C1(C)(C(=O)NCCC2CCCN(C(C3C(C)OCC3)=O)C2)CCN(C)C1=O N1(C(C(Br)=C(C)C)=O)CCC(C(C)CNC(=O)C(C)Cn2cccn2)CC1 c1(C(N2CCC(C(C)N=c3nc(C(C)(C)C)[nH]s3)C2)=O)ccc2ccncc2n1 C1(NC(c2ccc(C)nn2)=O)CCC12CN(C(=O)CC1CCCC(=O)N1)C2 N(C1CCCc2c1cnn2-c1ccccc1)C(C1CC(CS(C)(=O)=O)C1)=O CC1=C(C(=O)N2CC=CC2Cn2cc(CC(C)(C)O)nn2)S(=O)(=O)CCO1 CCC(CC)(CC(=O)OC(C)(C)C)C(=O)N1CCC(OCC(F)(F)F)C1 C(C(C)(F)C(C)(C)F)n1cc(CNC(C2(C)CC3(CC3)C2)=O)nn1 c1(C(C(=O)NCCCC2CC2)N(CCCO)C(C)C)ccc(C2CC2)cn1 c1(COC)ccc(C(=O)N(C2CCN(C(C3C=C(C)CS3)=O)C2)CC2CC2)s1 CC(C)CCCC(C)C(=O)NCC(C)(C)C(=O)NC(C1CCOCC1)C C1(NC(CCCCN(C(C)=O)C)=O)C2CCC1CN(C(=O)C(=O)N(C)C)C2 N1(C(=O)Cc2cn[nH]c2)CC2(CO)CC1(C(=O)NC(CO)CCC1CC1)C2 CCC(CCC(=O)N(C)CCOCCC(=O)N(CC(O)CC)C)OC n1(CC)nc(C)c(NC(C2CC23CCN(C(=O)CN2CCCCC2=O)C3)=O)c1C C1(NC(c2c(CC(C)C)nc(C)s2)=O)CC(O)CN(C(=O)COCCF)C1 C(=O)(C1Cc2ccc(Cl)cc21)N1CC(CNC(=O)Cc2cncs2)OCCC1 Cc1ccc(F)cc1-c1nnc(CN2CCCC2c2ccco2)o1 C(C1CC1)(C1CC1)=CC(=O)N(CC(C)C(=O)NC1CCN(CC2CC2)C1)C Cc1cccc2c(C(N3CCC(CNC(=O)CC(C)(C)C)C3)=O)cnn12 CC1CN(C(=O)C(F)(F)c2cccnc2)CCN1C(=O)CC1CCCC1 N(C1CCCc2ccoc21)C(C1=CCN(C(CCC=CC)=O)C1)=O c1(C(=O)NC2CCC2NC(c2cccc(C3CC3)c2)=O)ccc2oc(S)nc2c1 CC(CC(C)(C)C)C(=O)N1CC(C)(C)CC1C(N1CCOCCC1C)=O C(=O)(C(C)(C)CS(=O)(=O)N1CC(N=[N+]=[N-])CC1C(=O)O)OCC C1(NC(CCOC)=O)CCN(C(C2(C3CCCO3)CC2)=O)CCC1(F)F n1(C(CC)C)nc(C(N2CCCC(NC(=O)C(C)N(C)C)C2)=O)cc1C C12(Nc3ncc(C)c(C)n3)CCCC1CN(C(c1cc(C)c(C)nc1O)=O)C2 CC1CC(NC(c2cc(C(F)F)nn2C)=O)CN(C(c2nn(C)cc2N)=O)C1 C(CSC)(CCNC(C1(C(C)(C)OC)CC1)=O)OC C1(C(C)NC(=O)C(C)(C)c2cn(CCCSC3CCOC3)nn2)CCCC(=O)C1 N1(C(c2c(C)nnn2C)=O)CCC2(CC1)CN(C(=O)Cn1cccc(N)c1=O)C2 Cc1cc(NC(=O)C(O)CCNC(C2(C)CCC(=O)NC2)=O)cnc1O C(=O)(C(O)CC(C)(C)C)NCC1N(C(c2nc(C)c(C)s2)=O)CC1 C1(C#N)(C(N2CC(C(C)NC(=O)Cn3cc(Cl)cn3)C2)=O)CC1(C)C CCCCC(CC)C(=O)N1CC2(CCC(CNC(c3ncc(C)cc3F)=O)O2)C1 N1(CC(=O)NC(CNC(C2(CSC)CC2)=O)C2CC2)CCOCC1 N1(C(C(CC=CC)C)=O)CC2(CC(NC(C34CCC(OC)C3C4)=O)C2)C1 CCCCC(CNC(=O)CC(C)n1cc(Br)cn1)NC(=O)CCSC Cc1[nH]c(C#N)cc1C(N1CCC(CF)(NC(=O)Cn2cccn2)C1)=O C1(O)(CC(=O)Nc2nccs2)CCN(Cc2ccc(F)c(Br)c2)CC1 c1(OC(CC)C)ccccc1C(N1CC(NC(c2cc[nH]c2C)=O)C(C)C1)=O N1(C(C2C3C(NC(c4ncc(C)[n+]([O-])c4)=O)C4C(C3)C42)=O)CC2(CNC(=O)N2)C1 C1(CNC(COC2(C)CCCC2)=O)CCCC(NC(c2cccnc2)=O)C1 Cc1ccn(C)c1C(N1CCCC(CN(C)C(c2cc(Cl)ccn2)=O)C1)=O Cc1nc(NCCc2ccc[nH]2)cc(=NC(C)c2nc3ccccc3s2)[nH]1 Cc1cnc(NC(C2CC2NCc2cc(Br)ncc2Br)=O)c(Cl)c1 C1(C(=O)NCC2(O)CC(NC(=O)CSC(F)F)C2)CN2CCC1(C)C2 c1(C(N2CCC(C(=O)NCC(CO)CO)C2)=O)ccccc1-n1cccn1 C12(CC(=O)N(C3CCCN(C(c4snc(C)c4N)=O)C3)C)CCCN1CCC2 N1(C(C2CC3(CC3)CO2)=O)C2CCC1CC(NC(=O)C(F)(F)C(O)C1CC1)C2 Cc1cc(C(=O)N(CCCC(=O)NC2CCN(C(C)(C)C)C2)C)c(C)n1C CC(N=c1[nH]c2c(c(=NCc3cncs3)[nH]1)SCC2)c1ncnn1C c1(C(=O)NC2(C)CCCN(C(C3(CO)CC(F)(F)C3)=O)C2)cnn2cnnc2c1 c1(C(N2CCC(CCNC(C(CC)OC)=O)C2)=O)ccc(OC2CC2(F)F)cc1 c12cnc(Cl)cc1NC2=O.c1(-c2cc(NCCN(CC)CC)n[nH]2)ccc(Cl)cc1 C1(CNC(C(F)=CC)=O)C(C)CCN1C(=O)CCc1cn[nH]c1 N1(C(CCCOC)=O)CC(CNC(=O)C(C)Cc2ccccc2)CC(C)(C)C1 Cc1ccc(C(=O)NCCOCCNC(=O)CC=C(Cl)Cl)c(Cl)c1 CCC(CC)C(=O)NCC1CCCN1CC.c12ccccc1CNC2=O C1(CC=C)(C(N2CC(NC(=O)CO)C2)=O)CCOC1.C12C=CC(C1)CC(=O)N2 c1(C(N)=O)cocc1C(=O)NCC1CCCN1C(=O)CC1CC2(CC2)C1 C1(O)(CCNC(CCC(C)OC)=O)CCCN(C(c2cnccc2C(F)F)=O)C1 C#CCCCCCCC(=O)NCC(CC=C)C(=O)NCCNS(C)(=O)=O C1(NC(c2c(OC)ccs2)=O)CCCC(C(=O)NCC2(CCO)CCCC2)CC1 C(N=c1nc2sccc2c(NCC(Cl)Cl)[nH]1)c1onc(-c2c(F)ccc(C)c2)n1 CCCCCCCC(=O)NCC(c1ccccc1)NC(=O)C(c1cccn1C)=O Cn1cc(C(O)C(N2CCCC2CCCNC(C2(F)CC=CC2)=O)=O)cn1 N1(C(C(CCC)NC(C)=O)=O)C2CCC1CN(C(C1CC(OC)C1)=O)C2 c1(CC(=O)N(CCC(=O)NCCSC)C)ccc(O)cc1 C1(NC(C2(SCC)CC2)=O)CCN(C(c2cccc(C#N)c2)=O)CC(C)(C)C1 c1(CNC(C2CC(F)CN2C(c2ccc(I)c(Cl)c2)=O)=O)csc2ccccc12 C(=O)(C1CCCn2cnnc21)N1C(CN(C)C(C2CCC(C)(C)C2)=O)CCC1 c1(OC)cc(C(N2CCCC2CCCNC(=O)CSCC2CCCCO2)=O)sn1 C1(C(=O)NC(c2c(C(=O)O)cccc2F)C)CC2COCC(C1)C2 O=[N+]([O-])c1c(Br)cccc1S(=O)(=O)N1CCC1CO c1(C(N2CCC(C(C)C(=O)NCc3cscn3)C2)=O)ccc(O)c(F)c1 C1(c2nnnn2C)(NC2(CCOC)CCOCC2)CC2CC(O)C(C1)N2C c1(NC(=O)NCc2ccc(OC(F)F)nc2)ccc(-c2cscn2)cc1 C1(C(C)C(=O)Nc2[nH]cc(C(N3CCCC3)=O)c2)CCN(C(C2(C)CC2)=O)CC1 N1(C(CCS(=O)(=O)NC)=O)CCC(C)(C)C(NC(=O)Cn2nnnc2C)C1 C(=O)(C(C)(C)COCC)NCCN(C(=O)C(C)CN1CCOCC1)CCC C(=O)(C1CCc2c[nH]nc21)N1CC(CC(CNC(c2c(C)sc(O)n2)=O)(C)C)C1 C1(NC(C(=CC2CCCC2)C)=O)CC2CC(NC(c3cc(F)n[nH]3)=O)CC12 c1(C(=O)NC23C(CN(C(C4(C)CC(F)C4)=O)C2)CC3)cc([N+](=O)[O-])cnc1N c1(C(C(=O)NCCOCC(F)(F)F)C2C(CC)C2)cccc(Cl)c1 C1(OCCCN(C)C(c2cnc(Cl)[nH]2)=O)CCN(C(C2CCC(=O)NC2)=O)CC1 CC(=Cn1ccnn1)C(=O)NCCC1CN(C(=O)CC2CCCCN2C)CC1C C#Cc1cccc(NC(=O)CCCN2CCOCC2(C)Cc2cccc(Cl)c2)c1 C12CN(CC1c1cncn1C)C(=O)CN(C)N(CC)C(CC)C(=O)NC2.CC.OC C(CCCC(=O)NC(C1CCCN1C(=O)C(C)C)C)(OC)OC C1(NC(c2cc3cnccc3o2)=O)CCN(C(C2(CCF)CC2)=O)C12CCCC2 CC1CC(=O)NC1C(=O)NCC1(CNC(c2cccc(Cl)c2)=O)CC1(F)F C1(OC)CCCN(C(C2CCCC2CNC(=O)C(C)(C)n2cccn2)=O)C1 C(=O)(C(O)C1=CCCCC1)NC(CCC)C(=O)NCC(C)(C)C1CC1 N(C1CCC(NC(=O)C(CC)(CC)OC)c2ccccc21)C(CSCC#C)=O C1(C(=O)NC(C2CCC2C(=O)NCC(O)CC2CCCC2)C)CCC(C#N)CC1 N1(C(C(C)OCCC(C)C)=O)CCC(C2(NC(C3CC4(CC4)CO3)=O)CC2)CC1 N1(C(C2CCCC(C)C2)=O)CC2CC(NC(c3cc(N(C)C)ccn3)=O)C(C2)C1 C1(C(=O)NCC(CO)NC(C2OCCO2)=O)(OC)CCCOC1 C1(NC(C2(CC)CCCC2)=O)CCCCC1NC(C1CCC(C)CC1)=O C1(CC)CN(C(c2ccc(C#N)[nH]2)=O)CC1NC(c1nc(Cl)sc1C)=O c1(C(=O)NC(CNC(CC(=C)C)=O)(C)C2CCC2)cc(=O)n(C)cc1Br C1(CNC(C(C)C#N)=O)CCCN(C(=O)C(C)(C)OCC(F)(F)F)C1 c1(C(N2C(C)(CNC(c3c(OCC)cccc3)=O)CCC2)=O)oc(C)nc1C#N C(CCCCC(=O)NC1CCCC1NC(C1CCCC1C1CC1)=O)OCC C1(N(C(c2c(COC)noc2)=O)C)CN(C(c2c[nH]c(C#N)c2)=O)CC1O c1(CNC(=O)NC(c2ccccc2F)C)ccc(C(C)(C)C)cn1 c1(NCc2cc(C)[nH]n2)nc(N2CCC(N(C)C)C(C)C2)nc2c1cnn2C NC(=O)C1=NOC(CNC(=O)C(C2CCC2)NC(c2cccc(F)c2)=O)C1 N1(CCNC(C(C2CCSC2)N(C(C)=O)CC2CC2)=O)CCCCCC1 c1(CC(=O)OCC(C)(CC)OCC)ccc(F)cc1[N+](=O)[O-] c1(CC(C(=O)NCc2ccc(N3CCCC3)cc2)O)c(F)cccc1Cl Cc1ccc(C)c(C(=O)NCC2(CNC(c3oncc3C)=O)CCC2)c1C c1(CC(=O)NCC(C2CC2)NC(C=CC2N(C)CCC2)=O)ccc([N+](=O)[O-])c(N)c1 CN1CC(C(N2CCOCC2C(=O)NCCC2CC(C)(C)C2)=O)CCC1=O C(N=c1cc(C)nc(N(C)CCC2CCCCN2C)[nH]1)C1(OCC)CCCSC1 C1(O)(CN(C(c2c(C)nns2)=O)C)CCN(C(c2ccncn2)=O)C1 C1(OC)CN(C(c2cn(CCO)nn2)=O)CC1C(N1CCC1C1CCCC1)=O C1(CNC(=O)C=C(C)CNC(C2(COC)CC(=O)C2)=O)(OC)CCCCC1 C1(NC(C=CSC)=O)CCOC2(CCN(C(C3CC3CC(C)C)=O)CC2)C1 c1(C(N2CC(CO)CCC2C)C(=O)NC)nc2ccc(Br)cc2s1 c1(C(=O)NCC2C(C)CN(C(C3CNC(=O)N3)=O)CC2)cnn2ccccc12 C(C(C(=O)N(C)Cc1cnc(C)s1)NC(=O)Cc1cnnn1C)OC c1(CC)cnccc1C(=O)N(C)CC1C2CN(C(=O)CSCC(N)=O)CC12 c1(C(=O)NC(CCOC)CCC(=O)Nc2c(C#N)cnn2C)ccc(=O)n(C)c1 N1(C(COCCCCCC)=O)C(CNC(=O)CCOCC)CC2COCC12 N1(c2n(C)c(Cc3ccc(Cl)cc3)nn2)CCC(C2CC2)C1c1nnc(O)n1C C(CCCC(=O)N(C1CCN(C(=O)CC2CCCC(C(F)(F)F)O2)C1)C)OC C1(CNC(c2scnc2C(F)F)=O)CCC2(CCN(C(=O)C3=CCSC3)CC2)O1 CCC(C)(CO)C(=O)N1CC(NC(=O)COc2ccc(F)cn2)C2(CC2)C1 C12(C(=O)NC(CC)C)CC(CO1)N(C(c1c(C)coc1CO)=O)C2 CC1C(C(=O)NCc2nc(N(C)C)n[nH]2)CCCN1C(c1cccnc1)=O CC(C#N)C(=O)N1CC(N(C)C(c2cc(C3CC3)no2)=O)C1 C1(NC(=O)Cc2ccc(Cl)nc2)CN(C(=O)CC(F)(F)F)C2(CCC2)C1 C1(NC(CN(C)CCO)=O)CCCCC12CCN(C(=O)Cc1cnccc1Cl)C2 C(CNC(C1(c2ccccc2)CC1C)=O)(CC)(CC)NC(C(C)OCC=C)=O c1(N2CCN(C(C3CCC(C(C)(C)C)CC3)=O)CC2)ncnc(C2CC2)c1Br C1(CNC(c2ccc(OC)c(N)n2)=O)CC2CCC(C1)N2C(=O)Cc1ccns1 C1(CCC)CN(C(c2cnc(C(N)=O)s2)=O)CCN1C(=O)Cc1ccn(CC)n1 c1(NC)cncc(C(=O)NCCN(C2CCCC2)C(C2CCNC2=O)=O)c1 CC1CCC(NC(C2(C#N)CC2)=O)CN1C(c1cc(-c2cccs2)n(C)n1)=O N1(C(CCCCOCC)=O)CC(C)(C)OC2(C1)CN(C(C1CCC(F)CC1)=O)C2 C(=O)(C(C)(F)C(=O)NCCC(C)(C)NC(=O)COC1CCOC1)OC c1(C(CNC(c2n(CC#C)cnn2)=O)NC(=O)CC(C)OC)cccc(OC)c1 c1(N(CC(=O)OCC)CC2CCCO2)nccc(=NCCC#N)[nH]1 c1(CNC(C2C(C)(C)C2(C)C)c2n(C)nnn2)csc2ccccc2c1=O C1(NC(C2CCC(NC(C3(C=C)CCCC3)=O)C2)=O)CCCCNC1=O n1(CCC(=O)N(C)CC2CCCN(C(c3csnn3)=O)C2)ccc2ccccc12 c1(C(N2CC(NC(=O)Cc3cnc[nH]3)C2)=O)cnc(COc2ccccc2)s1 N1(C(C(=O)NC2CCC(C)CC2)=O)CC2(C1)CN(C(=O)CC1=CCCC1)C2 C1(CNC(c2c(C)coc2)=O)(NC(C2CCNC2=O)=O)CCCCC1 CC1(C)CCC(NC(c2ccc(Br)cc2NS(C)(=O)=O)=O)C(CN)C1 CCCC(C(=O)N(C(C)CNC(c1nsnc1O)=O)C)S(N)(=O)=O CS(=O)(=O)c1cc(C(N2CCC(C3CC3)(NC(c3csnn3)=O)C2)=O)cc(N)c1 C(=O)(CCCCCNC(c1coc2c1COC2)=O)N(CC(C)(C)C)C1CC1 O=C(CCC#Cc1ccccc1)NCC1COCC1NC(C1(CO)CC1)=O C(C)(CCC(=O)NC(C)C(CO)NC(=O)Cc1ccnn1C)SC C(C(=O)N(C)OCC)N(C(CCCC)=O)C(=O)CC1CCCC1O c1(C(=O)NC2CCN(C(C(CC)C(C)C)=O)CC2)cc(N)c(Br)c(F)c1 N1(C(C2CC3CC3C2)C(=O)NCCCSC)C2CCC1CN(C(C)C)C2 c1(CN(C(C)C(O)Cc2ccccc2)C=O)ccc(C(F)(F)F)c(F)c1 C(=O)(C1CCCc2nn[nH]c21)NC1C(CNC(C(CC)(C)CC)=O)CCCC1 C1(CC(=O)NC(C(=O)NCC2C(OC)CCC2)CC2CCC2)CCC(C)(C)O1 CCN(OC)C(=O)C(C)N(C)C(c1nscc1C)=O c1(OC)ccc(C(N2CCCC(O)(CCNC(=O)Cn3cnnn3)C2)=O)c(O)c1 c1(-c2cn(CCC)nc2)cccc2[nH]c(C(=O)Nc3coc(Cl)n3)cc12 N1(C(C(=Cc2ccccn2)C)=O)CC2CCC1C2NC(=O)C1=CSCS1 CCCCC(CNC(=O)C=C(CC)CC)NC(=O)CC1(O)CCOC1 c1(C(=O)NCCC2CN(C(CCC=CC)=O)CC(C)O2)ccc(Cl)c(C)c1Cl c1(C(=O)NC(CCNC(c2cc(C)nc(O)c2)=O)(C)C)cc(F)c(C#N)c(F)c1 c1(C(N(CCNC(C2CC2C(F)(F)F)=O)CC)=O)sc2ncccc2c1Cl C12(CNC(CCCCCSC)=O)CCC(CN(C(=O)C3=CCC(C)CC3)C1)C2 N1(C(C)=O)CC(NC(=O)NCCCCc2cnn(C)c2O)C(C)(C)C1 C1(CC)(CC)CC(C(=O)NC(COC(C)C)C(=O)NC2CCN(CCCO)C2)C1 c1(CNC(C(=O)Nc2cccc(C3CCCN(C)C3)c2)=O)ccc(F)c(N)c1 Cc1cccc(Cl)c1CC(=O)N(C1CCC(NC(c2cc(Cl)cn2C)=O)CC1)C Cc1cnn(C(C)C)c1C(=O)NCC1(C)CCCN1C(=O)C(C)N1CC(C)C1 c1(C(=O)O)cc(C(=O)NC2CC2c2cccc(F)c2F)cc([N+](=O)[O-])c1 C1(CNC(C2C(C(C)(F)F)C2)=O)CCCC(NC(=O)CCc2csnn2)C1 N1(C(CCCOCC)=O)CCCC(NC(c2cn3ccsc3n2)=O)C1C N1(C(CCC(=C)Cl)=O)CCN(C(C2CCC3(CC3)C2)=O)CC1C1CCCC1 N1(C(c2cccn3c(CO)nnc23)=O)CCn2c(n[nH]c(=O)c2=O)C1 Cc1nc(C(C)NC(=O)CC(C2CC2)NC(c2cc(Cl)cs2)=O)n[nH]1 c1(OC)ccc2cc(C(=O)NC3CN(C(c4cnn(C)n4)=O)CC34CC4)[nH]c2n1 C1(O)(C(N(C)CC2CCCN(C(C3(CSC)CC3)=O)C2)=O)CCC(C)(C)CC1 C=C(Cl)CCC(=O)NC(CN(C)C(c1coc(-c2ccccn2)n1)=O)CC CC1COc2c(C(=O)NC(C3CCN(C(=O)CC4(C#N)CC4)CC3)C)cccc21 C(=O)(CCCC(C)N(C)C)N1C(CN(C(CNS(CC)(=O)=O)=O)C)CCC1 Cc1cccc(C(O)C(N2CCC(NC(c3nccn3C)=O)C2)=O)c1 C(c1nc2ccccc2s1)=CC(=O)NC1CCC1NC(C1CCCCC(=O)N1)=O N1(CC(CC)CC)CCCC(C(=O)NC2CCSC2)C1 Cc1cc(F)c(C(=O)NC(CO)CCCNC(c2ccn(C(F)F)n2)=O)cc1F c1(C(=O)NC(C2CC3CC3N2C(=O)C(O)C(C)(C)C)C)c(F)cc(Cl)cc1F CCC(C)(C)C(O)C(=O)NCC(C)NC(c1coc2c1CCCC2)=O c1(C(N2CCCC(C(=O)NCc3cc(C)no3)C2)=O)cc2c(Cl)cncc2s1 C1(C)(CNC(c2c(C)n[nH]c2)=O)CN(C(C2CCOC2=O)=O)C(C)(C)C1 C1(CNC(COCCCCC)=O)CN(C(c2cc(CC)[nH]n2)=O)CCC1(F)F NS(=O)(=O)c1n[nH]cc1C(N1CCCC1CNC(c1cncs1)=O)=O N1(CCC(CC)(C)C)CCCC(N=[N+]=[N-])CC1 N1(C(CC2(C)CCCO2)=O)CCN(C(=O)C(F)n2cccn2)CC1.O=C N1(C(c2nccc(CC)c2)=O)CCC2C(CCCN2C(c2ncnn2CC)=O)C1 c1(NC(CC2C(C(=O)OCC)C2)=O)cccc(NC(c2c(C)coc2CC)=O)c1 C1(C(C(=O)N(C2CCCC2)CCNC(=O)COCC(F)F)F)CCCCC1 C=C(Cl)C(C)(C)C(=O)N1CC2(C1)CN(C(=O)C(C)CSC(F)(F)F)C2 N1(C(c2c(C)ccc(=N)[nH]2)=O)CCC2C(CCCN2C(c2ccc(CO)s2)=O)C1 c1(C(N(C2CCN(Cc3nc(CC)sc3)C2)C)=O)cnn2cccnc12 c1(CC(=O)NC2C(CNC(CC(=C)C)=O)CC2)c(F)cccc1Br c1(C(=O)NCCCOCCN(C(COCCC=C)=O)C)cnc(C(F)F)s1 c1(C(N2CC3(CC(NC(C4CCCCS4)=O)C3)C2)=O)cc(Cl)cc([N+](=O)[O-])c1O C(C(C)(C)C(C)(F)F)NC(C1(NC(CCSC)=O)CC1)=O.C(C)(=O)O Cc1nn(C)c(C(=O)NCCNC(C2CC2c2ccc(Br)cc2)=O)c1Cl C=CCC(C)(C)CNC(=O)CCC1CCN(C(C2CC(N(C)CC)C2)=O)C1 C1(N(C(=O)C(C)(C)C2CCOCC2)C)CCN(C(c2ccc(Cl)o2)=O)CC1 c1(C(C)C(=O)NC2(C)CC(NC(C3CCC3)=O)C2)ccc(-c2ccccc2)cc1 N1(C(CSc2n(C)cnn2)=O)CCCC12CCN(C(c1c[nH]c(C(N)=O)c1)=O)C2 c1(C(N2C3CC(CNC(C=CC=CCC)=O)C2CC3)=O)cc2nccc(Cl)c2s1 c1(NC2C(=C)C2)nc(=NCc2nc3cc(Cl)ccc3s2)nc(N2CCOCC2)[nH]1 N1(C(C(CC)C)=O)CC2(C)CC1(C(=O)N(C)CC)C2 N1(C(Cc2c(C)non2)=O)CC(NC(=O)C(C)OCC2CC2)CC12CCCC2 C1(NC(c2cc(C)c(C)[nH]2)=O)COCCN(C(C2CC23CC(O)C3)=O)C1 c1(N2CCN(C(CNC(C)=O)=O)CC2)nc(=N)[nH]c(=NCCC2CCCN2)[nH]1 C1(CNC(c2c(CC)scc2)=O)CC2(CCC2)CN1C(=O)C(C1CCOCC1)C C1(NC(CC2C=CC(NC(CC=CC=C)=O)C2)=O)CCCCNC1=O C#CCCCC(=O)NC1C2CN(Cc3scnc3Cl)CC12 Cc1c(C(=O)NC2CCCCC2NC(c2cn(C)nc2CN)=O)cnn1C1CC1 c1(C(N2CC=CC(NC(CCc3c(C)n[nH]c3C)=O)C2)=O)ccc2nccn2n1 c1(C(=O)NC2C(CNC(CCNS(CC)(=O)=O)=O)CC2)ccc(C2CC2)nc1 N1(CCC#C)CCC(C(=O)NC2C3CN(C(C4(C)CC4(F)F)=O)CC23)CC1 c1(CC(=O)NC2C3CCC2N(C(=O)C2=CCCC2)C3)ccc2nc(O)[nH]c2c1 N1(C(C2N(CC)CC2)=O)CC(CO)(NC(c2n[nH]cc2SC)=O)C1 CC(C)C(O)CCN=c1[nH]c(=NCc2ccnc(OCCO)c2)c2[nH]ccc2[nH]1 c1(C(C(=O)NC2C(n3cc(-c4c(C)ocn4)nn3)CCC2)O)ccc(Br)cc1 c1(C(=O)NC(CC(C)NC(Cc2c(C)n(C)nc2)=O)C)n[nH]c2c1CCSC2 Cc1ccc(C(=O)NCC2C=CCN2C(=O)CCc2nncn2C)cc1C C1(C(=O)NCC2(CO)C(C=C)C2)CCN(C(c2c[nH]c(=NC)s2)=O)C12CC2 C(=O)(C1=CCCN(C(=O)CC=CCNC(c2cnc(C(C)C)o2)=O)C1)OC c1(C(C(=O)NCC2C(NC(CCC3CC(OC)C3)=O)C2)OC)ccccc1Cl C1(NC(C2(N(C(c3cc(OC)no3)=O)C3CC3)CCC2)=O)CC(C)OC1=O N1(C(CC2C3CN(C(C=COCC)=O)CC2CC3)=O)CC(F)(F)OC(F)(F)C1 C1(CNC(C=C(CCC)C)=O)CC(CNC(c2cnc(CC(C)C)[nH]2)=O)CO1 c1(CC)cc(C(=O)NC23CCN(C(c4cc(F)ccc4C)=O)CC2C3)cc(O)n1 C(=O)(C(C(=O)CC)C(C)(C)C)O.N1(n2cc(CC(=O)NOC)nn2)CCC(F)(F)C1 C1(C(N(C)CC2CN(C(C=C3CCC(C)C3)=O)C2)=O)CC(C2CC2)=NO1 CCCCCC(C)CC(=O)NCC1CC(O)(CNC(=O)CCF)C1 N(C1CCCn2ccnc21)CC1N(Cc2ccccc2)CC1C1CC1 N1(C(CC(=O)NCC#C)=O)CC=C(CNC(C2CNC(=O)N2C)=O)CC1 Cc1oc(C2CCOCC2)nc1C(=O)NCC1CCCCN1C(=O)CS(N)(=O)=O c1(C(N2CC3C(CNC(C(CC=C)C)=O)(CC3)C2)=O)nc2ccccc2cc1Cl C(C1(C)CCOCC1)=CC(=O)NCC1C(C)CCN1C(=O)CN(C1CCC1)C Cc1nccc(C(=O)NC2C=CC(CC(N3CCC(C)(C(N)=O)C3)=O)C2)n1 C1(N(C(c2cncnc2)=O)CC)CCCN(C(=O)C(C2CC2)C2CC2)C1 c1(C(=O)NC(CCCC)C)oc(CNC(=O)CCc2nc[nH]n2)cc1C c1(C(=O)NC(CN(C(C2C(C)OCC2)=O)C)(C)C)ccc(C#N)[nH]1 c1(C(C)C(=O)N(C2CC(NC(=O)C(F)(F)c3ccnn3C)C2)C)ccc(F)cc1 Cc1cc(C)c(-n2cc(CCN(C)C(C3CNC(=O)N3)=O)nn2)c(C)c1 Cc1cc(CNC(C2CCCC(NC(=O)Cc3cnoc3)CC2)=O)cc(C)n1 CC1(C)CCC1C(=O)NCC1C=CCN1C(=O)COc1ccccc1 c1(C(=O)NCC23C(CN(c4cc(N(C)C)ncn4)C2)C3)ccc(C#N)c(Cl)c1 C1(NC(CC(=O)N(C)C)=O)CCCN(C(c2c(Cl)ccnc2F)=O)CC1 c1(C(C)(C)C(=O)NC2CCC(NC(=O)Cc3csc(Cl)n3)C2)cccc(O)c1 c1(C(=O)NCC2(O)CN(C(C3CC(=O)N3)=O)C2)ncc(Br)cc1F C#CC1CCC(NC(C2C3CN(C(c4ccc(F)c(O)c4)=O)CC23)=O)CC1 N1(CCC)CC(C(=O)N(CC(C)(C)NC(C23CCC2C3)=O)C)CC1=O c1(C(=O)NC2CCC(C)N(C(c3nccnc3N)=O)C2)c[nH]c2cc(Cl)ccc12 N1(C(CCSCC(C)C)=O)C2CCC1CC(CCNC(=O)C(F)n1cccn1)C2 c1(NC(C23CC(C(N4CC5CC4CO5)=O)(C2)C3)=O)ccc(Br)c(C(F)(F)F)n1 C(=O)(C1=C(C)OCCS1(=O)=O)N1C(CC)CN(C(=O)CN2CCOCC2=O)CC1 Cc1cccc(CC(=O)NCC2CC(F)(CNC(=O)CC3CCCSC3)C2)c1C CC(C)C(O)C(C)C(=O)N1C2CCC(C(=O)NCC3CCC(C)C3)C1CC2 C1(NC(c2c(C)cno2)=O)Cc2ccccc2C1NC(=O)C(C)CS(C)(=O)=O CCC(C)CC(=O)C(=O)NC1CCCCCC1C(=O)NOC1CC2CCC1C2 C1(NC(C(CC2CN(C(C3(OC)CCCCC3)=O)C2)F)=O)CCC(=O)N(C)C1=O C(=O)(C(O)CCNC(=O)CSCC(F)F)NC1(CCC)CC1 C1(NC(CC2C(C)CCO2)=O)CCC(C)(CNC(=O)CN2CCN(C)CC2)CC1 c1(C(=O)NCc2cc(C)c(O)c(C)c2)ccc2c(c1)CCCC2=O C12(CNC(CC3(C=C)CC3)=O)CC3CC(CC(C3)C1NC(=O)C(F)CC1CC1)C2 Cc1cc(C(=O)NC2CCN(C(C3(O)CCCC(C)(C)C3)=O)C2)c(F)cc1F C1(C(N2CCN(CCN(C(c3c(C)occ3)=O)C)CC2)=O)CCC2(C1)CC2(F)F c1(C(=O)NCC(CCC)NC(C2CCC(NC(N)=O)CC2)=O)cccc(Cl)c1 N1(S(C)(=O)=O)CCN(CC(=O)NC2CC(NC(C3(N=[N+]=[N-])CC3)=O)C2)CC1 S(=O)(=O)(c1c(Cl)cc(Cl)cc1Cl)N1CCC2(CCCN(C(C(CC)C)=O)C2)C1 N1(CCNC(C2CCC(F)C2)=O)CCN(C(=O)CCC=CBr)CC1 c1(C(=O)OC)ccc(C(=O)NCC(O)CNC(c2csc(C3CC3)n2)=O)[nH]1 Cc1ccc(F)c(-c2cccnc2C(=O)Nc2c(F)cc(Br)cc2Br)c1O CCCC(C)(CCC)C(=O)NC(c1ccc(C)cc1)CNC(c1cocn1)=O NC1CCCC12CCN(C(=O)CN1CCc3[nH][nH]c(=N)c3C1)CC2 C1(CNC(=O)CCF)CC=CCN1C(=O)C(O)CC1CC1 c1(NC(C(N2CCC(C#C)C2)c2cccs2)=O)ccc(OC)c(OC)c1 C=CCCCCCC(=O)N1CCC(C(=O)Nc2cnccc2CO)C(CC)C1 N1(C(c2cnc(OCC)s2)=O)CC(NC(=O)CCCc2cnn[nH]2)C(C(F)F)C1 C=CCCCC1C(=O)N1.C1(C(=O)N(CC(C)(C)COC)CC)CC12CCCCC2 c1(C(N2CC3(CCN(C(c4cccc(C)n4)=O)C3)C2)=O)cc2ccc(Cl)cc2o1 c1(C(=O)NC2C3CN(C(C4(CC#C)CCCCO4)=O)CC32)cc2c(s1)CCOC2 C1(NC(C=CSC)=O)CC(NC(C2CC2c2cn[nH]c2)=O)C(O)C1 C(=O)(C(CC1CC1)NC(c1ncoc1C)=O)NCC(C1CCC1)OC N1(Cc2c(OC)cccc2)CCC(C)C(CC(F)(F)F)C1.C1CC(=O)O1 C1(CC(=O)NCCOC2CC2(F)F)CCC(CNC(C2C3CCC(F)C23)=O)CC1 N1(C(c2cc(C)c(N)cn2)=O)Cc2nccn2CC(NC(=O)CC=C(Cl)Cl)C1 Cn1cc(C(=O)NCCN(C(C2CCO2)=O)CS(C)(=O)=O)c(C2CC2)n1 Cc1ocnc1CC(N1CC(C(=O)N(CCN(C)C)CC2CC2)C1)=O c1(N)cc(CC2(CN(C(CC)C(=O)NCC3CC3)CC)CC2)nc(OC)n1 CC1(C)CC(C(=O)N(C2CC2)CC2COC(=O)C2)CO1 N1(C(c2occ(C)c2)=O)CC2(CCN(C(=O)C=Cc3ccccc3Cl)C2)C1 N1(C(C(c2ccccc2)N(C)C)=O)CCC(CNC(=O)CC2CC=CC2)C1 CN1CCOC(CONC(c2cccc(CN(C)C(N)=O)n2)=O)C1 C(=O)(CN=c1[nH]c2ccccc2s1)NCCOCCN(C(C(COC)C)=O)C CC1CC(NC(=O)CSc2ccccc2)CN(C(=O)Cc2n[nH]c(=N)s2)C1 C(CCCCC(=O)N1CCN(C(c2n[nH]cc2C(C)C)=O)CC1)SC C(CCC(=O)N(CC(O)CN(C(=O)Cc1ccon1)C)C)OC O=C1NCC2CCC1N2N1CCCC(C(c2cc(F)ccc2F)=O)C1 n1(C(C)C)cc(C(c2nnnn2C2CCCC2)NCCc2cnn(C)c2)cn1 N1(C(COCCCC#C)=O)CCC(C2CCCN(C(=O)C(C)CC(N)=O)C2)CC1 CC(O)C(C)(C)CNC(=O)C(=O)Nc1ccc(-c2cccnc2)cc1 c1(SC)cc(N2CCN(C(c3sc(C)nc3C)=O)CC2)nc(-c2ccncc2)n1 C(=O)(C(CC(F)F)NC(=O)C=Cc1cnccn1)NCC(C)(C)n1cccn1 O=C(CCS(=O)(=O)c1ccc(F)cc1)OCc1cscc1C(F)(F)F C1(CNC(C(C)=C2CCCC2)=O)CC12CCN(C(c1ccoc1Cl)=O)CC2 C1C(C(F)F)CC(=O)N1.C1(C)(C)C(=O)O1.S(=O)(=O)(Cc1ccon1)N(C)C C(=O)(C1Cc2c(Cl)cccc21)NC(CNC(C1=C(CC)OCCC1)=O)(CC)CC C(Cc1ccccc1)(CC(F)(F)F)N(C(c1cnn(C)c1CCC(F)(F)F)=O)CC N1(C(C(C)(C)NC(C)=O)=O)CCC(N2CCC(C3CC3)CC2)C2(CC2)C1 N1(C(c2ccc(SCCC)cc2)=O)CC2CCC1C2NC(=O)C(O)C(F)F Cc1nc(NC(CNC(C2CCCC3C2C3(F)F)=O)C(C)C)c(C)c(Cl)n1 C(C)(c1ccccc1OC)=CC(N1C2C(CNC(C(CC)(C)CO)=O)C(C2)C1)=O C=CCCC(C(=O)NCC(C)CC(=O)NC)NC(c1cnc2n1CCC2)=O c1(CC)sc(C(N2CCCC2C2CCCN(C(=O)C=CCOC)C2)=O)cc1C N1(C(C=COCC)=O)CCC(C2CCN(C(c3cn(C4CCC4)nn3)=O)C2)C1 CCC(C)(CN=c1[nH]c(-c2ccccc2)nc(=NCCCC2CC2C)[nH]1)C(N)=O c1(C(N(CC(C)O)CCNC(C2(C)CCCCC2)=O)=O)ccc2c(c1)nnn2C C(C1=Cc2cc(Br)ccc2OC1)NC(C)(C)CS(C)(=O)=O C1(NC(Cn2c(C)ccn2)=O)CCCC(NC(=O)C(c2ccc(Cl)s2)C)C1 O=C(CS(=O)(=O)CCO)NCCC1CCCN(C(C2CC3CCC2O3)=O)C1 c1(OCC)cc(N2CC(=C(F)CNC(=O)CCC3CCOCC3)C2)ccc1[N+](=O)[O-] CC1(C)CC(C(N2CC(OCCNC(C3CC=CCC3)=O)C2)=O)CNC1=O N1(C(C(c2c(C)n[nH]c2C)C)=O)CCN(C(C2CC2(C)C(C)C)=O)C(C)C1 C(CC(=O)NCC1(C(C)C)CC1)(C(F)(F)F)NC(CCC=CC)=O S(=O)(=O)(c1cnn2ccc(NCC3CCOCC3C)nc12)N(CCCC(C)C)C C1(C(=O)NC2(C(=O)NCCN(C(=O)CCCc3ccco3)C)CC2)CC2CCC1C2 C1(CCCNC(CCNC(C)=O)=O)CCN(C(c2ncsc2N(C)C)=O)CC1 CN=c1[nH]cc(C(N2CC(OC)CC2CNC(=O)C2=CCOC2)=O)o1 c1(N(S(=O)(=O)c2ccc(Cl)s2)Cc2cc(C)ncc2)c(C)ccc2ncccc12 c1(C(=O)NC2CCCN(C(CC=CCC)=O)C2)ccc2c(c1)oc1ccccc21 c1(C(N2CCC(C(CNC(C(CC)O)=O)(C)O)CC2)=O)ccn2cncc2c1 N1(C(c2c(C)con2)=O)CCN(C(c2ncncc2Cl)=O)C2COCC12 CCC(C)(O)C(=O)NCc1c[nH]nc1C1CCN(C(c2cc(C(C)(C)C)n[nH]2)=O)C1 C(=O)C(C)CS(C)(=O)=O.C(=O)(CS(=O)(=O)CC)OC(CC)CC N1(C(c2cnn(C)n2)=O)CCC2CC1CN(C(=O)CCn1cncn1)C2 C(=O)(C(CCS(C)=O)N(C)C)NCC1CCC(CN(C(C(C)C2CC2)=O)C)CC1 c1(NC(C2CCN3C(C2)C3)=O)c(O)cc(F)cc1F.Cc1nn(C)c(C(=O)O)c1F CCC(CC)(CN=c1[nH]c(C(C)(C)C)nc(=N)[nH]1)NC(c1cscn1)=O C1(C(N(CCCn2cc(CCNC(C)=O)nn2)C)=O)CC2CCC1O2 O=C1Cc2c(C(=O)NCC(F)CNC(=O)Cn3cnnn3)ccnc2N1 N1(C(C(C)NC(=O)NC)=O)CC(O)CC1C(=O)NCC1(NC(C)=O)CCCCC1 c1(CN(CC(=O)OCC)C(c2ccc(OC)cc2)C)ccc(Cl)cc1 N1(C(C2=C(C)CCC2)=O)CC2=C(C1)CN(C(=O)C(C)(C)C(C)C)C2 C(=O)(C1CCCc2sccc21)N(C1CN(C(CC=CC=C)=O)C(C)(C)C1)C1CC1 C(CC(N)=O)(C(=O)NCCOCCN(C)C(C1(F)CCCN(C)C1)=O)NC(C)=O c1(C(=O)NCC2C(NC(c3c(C)nn[nH]3)=O)C2)c(OC(F)F)cccc1Br C1(CC)CN(C(=O)Cc2ccc(F)nc2)CC1C(N1CC(O)CC1C(C)C)=O S(=O)(=O)(c1ccc(Br)cc1NCCN1CCP(C)(=O)CC1)NCc1c(C)ocn1 c1(OCC)ccc(NC(C2CCC2NC(C2CC(O)CN2C)=O)=O)cc1 C#CCCCCCC(=O)NC1CCN(C(c2cnoc2C)=O)C1(C)C c1(C(=O)NC(C)CCCNC(c2ncc(F)cn2)=O)ccc2occc2n1 N1(C(C(CCC#C)O)=O)CC(NC(c2ccc([N+](=O)[O-])s2)=O)C(C2CC2)C1 C1(NC(C2CCN(C(C)=O)C2)=O)(CF)CCN(C(c2cncnc2)=O)C1 C(=O)(C1Cc2c(Cl)cccc21)N1CC(C)(CNC(CC2(CSC)CC2)=O)OCC1 C1(CNC(C2(C#C)CCCC2)=O)CC2COCC2N1C(c1ccco1)=O C1(CCC)CCCN(C(C2CC23CC(NC2(C(=O)OCC)CCC2)C3)=O)CC1 c1(C(N2CCOC(C3CC3)C2)C(=O)NCCCF)cnn(C(C)C)c1F C1(C(N2CC(CCNC(C3C(OCC)CC3)=O)C(C)C2)=O)CC(=O)NC(=O)N1 C(=O)(C(O)C(C)(C)CC)NCC1(OC)CN(C(C(CC)NC(=O)OC(C)(C)C)=O)C1 N1(C(=O)NOCC(F)(F)C(F)F)CCCc2ccc3ccccc3c21 N1(C(c2cc(OC)ns2)=O)CCC(C2CCN(C(c3ccnn3C)=O)C2)CC1 N1(Cc2csc(OCc3ccccc3)n2)CC(C(C2(CN(C)C)CC2)C)OC1=O N1(C(C(C2CC2)SC)=O)CC(CC(=O)NCCC2CCOC2(C)C)CC1C c1(C(c2nnnn2-c2ccccc2)NCC(COC)C)cc(F)c(F)c(F)c1 c1(OCC)ccc(NC(=S)Nc2cnc(C(F)(F)F)cn2)cc1OC(C)C c1(-c2nc(CC(CC)C)nn2CC2CCOC2)ccc(F)cc1Cl c1(C(N2CC(CC(=O)Nc3nn[nH]c3C(F)(F)F)C2)=O)occc1Br c1(NC(C(CC)(C)O)=O)ccc(CNC(=O)C(C)(C)N2CCOCC2)c(C)c1 N1(C(C2(OC)CCC2)=O)CCC(COC2CCN(C(C3(Cl)CC3)=O)C2)CC1 Cc1ccc2c(N3CCCOC(CNC(c4ccc(CO)o4)=O)C3)ncnc2c1 C1(NC(c2cccc(OCCF)n2)=O)CN(C(=O)C=Cc2cccs2)CC12CC2 N1(C(C(C)Cc2cnco2)=O)CCCCC(CNC(=O)COC2(C)CCOC2)C1 Cc1cc2c(CC3SCCC3c3noc(C4CCCO4)n3)csc2s1 c1(N(C(=O)CNC2CC(NC(=O)C(F)C3CCCC3)C2)CC)ccc(C#N)cc1 Nc1c(C(=O)NCC2(NC(C3CC4(CCC4)CO3)=O)CCCCC2)cccc1F N1(C(C2N(CC)CCC2)=O)CCCC1(C)CNC(=O)Cn1ncn(C)c1=O c1(-c2cnc(C3N(C(CCS(C)=O)=O)CCC3)[nH]2)ccc(Cl)cc1Cl C12(C(=O)NC3CCN(C(C(CC)C(C)C)=O)C3)CCC(C(=O)OCC)(CC1)CO2 c1(C2N(C(c3n[nH]c(-c4ccccc4)n3)=O)CCC2)nnc2n1CCC2 Cc1scnc1C(=O)NCc1ncoc1CCNC(=O)CC1(C)CC1F CC(C)CC(C)(CO)NC(=O)COC1CN(C(C2CCCCCCC2)=O)C1 Cc1oc(-c2ccccc2)nc1C(N1CCOC(CS(N)(=O)=O)C1)CN(C)C c1(C(=O)NCCN(C(c2cn(CCC)nc2C)=O)C)cnc(O)c2cccnc12 N1(C(C2CCN(C)C2=O)=O)CCC(CO)(CNC(c2ccn(C3CC3)n2)=O)CC1 c1(OC)ccc(C(N2CCOC(CNCc3ccc(OC(F)F)cc3)C2)=O)c(C)c1 C1(C(N2CC(O)CC2CO)=O)(COC)C=CCN1C(c1sccc1C)=O C#CCCC(=O)NC(C1CC1C(=O)NC(c1nn[nH]n1)C1CC1)C N1(C(CN(S(C)(=O)=O)C)=O)CCCC(NC(C23CC(C)(C2)C3)=O)CC1 C1(NC(c2ccc(SCCCC)cc2)=O)CCN(C(=O)C(C)(C)F)CC1CC C(=O)(C(O)CC1CCOCC1)NC(CN(C(=O)C(O)CC1CC1)CC)C c1(C(N2C(CCOC)CN(C(=O)C=C(C)Cl)CC2)=O)cnn2cc(C)cnc12 O=C1CC(CC(=O)NCCCn2cc(CN3CCCC3CO)nn2)CO1 C1(NC(c2c(OC)ncc(Cl)c2)=O)CN(C(=O)CSCCC#N)C2(CCC2)C1 N1(CC#CC)CCC2(CCCCN(C(=O)CC3CCCCCC3)C2)C1.C(CC#N)N c1(OC)csc(C(=O)NC2CCC(C)(CNC(c3ccncc3N)=O)C2)c1OC C(CC(O)C(=O)NCC(CC(C)C)NC(C1(C)CC(C(=O)OC(C)(C)C)C1)=O)SC c1(-c2nn(-c3c(C)ccc(F)c3)c(CC3CCOC3)n2)ccc2ncccc2c1 N1(C(C(N2CCNC2=O)C)=O)CCN(C(c2ccc(N(C)C)c(F)c2)=O)C(CF)C1 N1(C(c2ocnc2C(F)F)=O)CC2CCC2(CC(N2Cc3c[nH]nc3C2)=O)C1 N#Cc1cccc(S(=O)(=O)Nc2cc(C(N3CCC(O)(CF)CC3)=O)n(C)c2)c1 CC1CN(C(=O)CNC(=O)Cc2ccccn2)CCS1=O C1(C(=O)NCC(CNC(c2cnn(CCN(C)C)c2)=O)OC)CCCCO1 c1(N2CCC(NC(C3CN(C)C3)=O)C(F)C2)nc2ccc(O)cc2s1 Cc1cc(C(N2C3CCC2(CNC(c2nc(Cl)sc2C)=O)CC3)=O)cc(N)c1 N1(C(c2nc(C(C)C)oc2)=O)CC2CC1CC2NC(=O)COc1ccsc1Cl c1(CCC=C)ccc(-c2nc(-c3ccc(COC)cc3)nn2CC)cc1 C12(NC(C=CC=CCC)=O)CCC(CC1)N(C(c1cccc(C)c1Br)=O)C2 c1(C(=O)NCC2(NC(C3C(C(C)(C)C)C3)=O)CCC2)ccc2nccn2c1 C(c1ccncn1)=CC(=O)NCC(CC(C)(C)C)(C)O.c12csc(n1)CC(=O)OC2 C1(C(N(C2C3CC2N(C(c2noc(C)c2C)=O)C3)CC)=O)CCS(=O)(=O)C1 C1(OC)CN(C(=NCCNS(C)(=O)=O)NC2CC2)CC1NCC1CCCCN1C c1(OC)cc(O)ncc1C(=O)NCC(C)CNC(c1cccc(C2CCC2)c1)=O C12(NC(C(CC)CC)=O)CCCCCC1N(C(=O)Cc1csc(C3CC3)n1)CC2 c1(SCC(=O)NC2(CCCNC(C3(CC)CC3)=O)CC2)ccc(O)cc1 Cc1nncn1NC(=O)C1C(C)CCN1C(=O)Cn1cc(Cl)cn1 c1(C(N(C2C3CN(C(=O)CN4CCOCC4)CC23)C)=O)cnc(S)n1C C1(C(=O)NCC2(CC(=O)NCCCCC#C)CC2)CCCCC1O C(CC(=O)N(C)Cc1cccc(C)n1)(C(C)CC)NC(c1c(C#C)c[nH]n1)=O c1(SC)ccc(C(=O)NC2CC2NC(c2n[nH]cc2C(F)(F)F)=O)s1 N1(C(C(C(=O)OCC)CC)=O)Cc2cccc(O)c2C1 CCCC(CC(C)C)C(=O)N1CCC(C(=O)N(C2CCCCCCC2)C)C(C)C1 C1(NC(c2sc(CC)c(C)c2)=O)CCN(C(=O)COCC2CCCCO2)C1(C)C c1(-c2nc(CCCO)nn2CCC(F)(F)F)[nH]c2ccc(Br)cc2c1Cl c1(CN2CC(NC(c3ccc(O)c(O)c3O)=O)C(O)C2)cc(F)c(Cl)c(Cl)c1 N1(C(C=CC(C)C)=O)CC(NC(c2ccc3nn(C)cc3c2)=O)CC12CCCC2 c1(C(=O)NC2(CNC(=O)CC3(O)CCOCC3)CC2)ncnc2c1CCCC2 C1(CC)CCc2[nH]nc(C(N3CCOC(CN(C)C(=O)C4CC4)C3)=O)c2C1 CN1C(=O)CCC1C(=O)NC1C2CC1N(C(C1CC1(C)C(F)F)=O)C2 c1(C(=O)NC2CCC(CN(C(C(CCC)O)=O)C)CC2)c(C)cccc1Cl C1(C(N(CC(CC)C)C)=O)CCN(C(C2CCCOCC2)=O)CC1 c1(OC)ccnc(C(=O)NCC2(F)CN(C(C3CCCC(C4CC4)O3)=O)C2)c1 C1(OC)CN(C(C2NC(=O)OC2C)=O)CCC1NC(c1scnc1C1CC1)=O C1(CNC(CCSC)=O)CCC(C(=O)NCC2CC2C(F)F)CC1 O=C(C1=CCCOCC1)NC12CCCC1N(C(c1cnns1)=O)CC2 O=C1CCN(C)C2CCCCCN12.c1(CC)ccc(F)c(I)c1 C1(OC)CC(CC(=O)NC(C(=O)NCCC(=O)NC(C)(C)C)C2CC2)C1 c1(C(N2C(CNC(CC3(C)CC3)=O)COC(C)(C)C2)=O)cc([N+](=O)[O-])ccc1N N1(C(c2cc(CC)[nH]n2)=O)CCCC(O)(CCNC(c2cn3c(n2)SCC3)=O)C1 c1(C(=O)NC2C(NC(C(c3ccccc3O)OC)=O)COC2)ccc([N+](=O)[O-])[nH]1 C1(CCC)CN(C(C2(Cl)CC2(C)C)=O)CCN1C(c1cc(OC)no1)=O C(=O)(C1=NOC2COCC12)NC(CCN(C(C=C(C)Cl)=O)C)C(C)C C(=O)(C#CC1CCOC1)N1CCC(C(N(c2cccc(F)c2)C)=O)OCC1 C1(CC=C)(NC(=O)Cn2cnnn2)CCN(C(=O)CSc2ccccc2Cl)C1 CC(CC(=O)NCC12CC=CC(C1)OC2)C(C)(C)NC(c1ccn(C)c(=O)c1)=O CC1CCC=C1C(=O)NC(C)CCc1ccccc1.C12CSCN1C2=O c1(CN(CCNC(c2cc(COC)[nH]n2)=O)C2CC2)ccc(OC)c(Cl)n1 CCC(CCC(=O)NCCOCC1CC1)NC(=O)C(C)NC(C)(C)C C1(CC)CNC(=O)CN1C(=O)C(CC(C)C)NC(=O)CC1CCCSC1 CC1=C(C)CN(C(=O)CC2CC3(C2)CN(C(c2ccoc2Cl)=O)C3)CC1 c1(C(=O)Nc2c(C(C)(C)C)cccc2)ccc2c(=O)c(C(C)(C)C)c[nH]c2c1F CS(=O)(=O)c1ccc(C(F)C(=O)NOCCCC(F)(F)F)cc1 C(=O)(C(O)(C(F)(F)F)C1CC1)N(CCCN(C(C(CCCC)N(C)C)=O)C)C Cc1nc(C2CC2)ncc1C(=O)NC1CCN(C(C2(C3CC3)CC2)=O)CC1O C1(CC(=O)NCCN(C(C2CCCCCC2)=O)CC)CCC(F)(F)CC1 C(=O)(CCCCC(=O)NC(C1CCCCN1C(c1nnc(S)n1C)=O)C)NC c1(CC2(CNC3CCN(C(=O)C=Cc4cn[nH]c4)C3)CCOC2)cccc(Cl)c1 c1(C(=O)NCC(CC=C)NC(c2c[nH]cc(C)c2=O)=O)c(F)ccc(C#N)c1F C1(CC)CC(O)CCN1C(C1(C)CC(O)CN1C(=O)CSc1nc[nH]n1)=O c1(OCC(=O)NC2(CCO)CN(C(c3c(C)noc3)=O)C2)nn(C)cc1[N+](=O)[O-] C(=O)(C(CCF)NC(c1nc[nH]n1)=O)NC(C)CN=[N+]=[N-] N#Cc1ccc([N+](=O)[O-])cc1C(=O)NC1CN(C(=O)CCCOCC2CC2)C1 C1(C(N(CCNC(c2ccc(F)c(O)c2)=O)CCOCCO)=O)CCCC12CCC2 C1(NC(C2(C=C)CCOCC2)=O)CCN(C(=O)CC2CCCN(C)C2)CC(O)C1 CCCC(C(=O)NC1CCOCC1NC(C1(C(N)=O)CC1)=O)C(C)C C1(OC)CC(NC(=O)C=C(Cl)Cl)CN(C(c2nn(C)cc2Cl)=O)C1 c1(C(=O)NCCOCCNC(C(C2CC2)OC)=O)ccc(CN(C)C)o1 C(=O)(C(CCc1ccccc1)C(F)(F)F)N(CC(CC)C)CC(F)(F)F C1(CNC(c2c(COC)cc[nH]2)=O)CCCN(C(c2c(Cl)cnn2C)=O)C1 CN1CCn2nc(C(=O)N(C3CC3)Cc3nn[nH]n3)cc2C1 N1(C(C2C(NC(c3cnn[nH]3)=O)C3CCC2C3)=O)CCC(C2CCC2)C1 c1(C(N2CC3CC(NC(C4(CCF)CCC4)=O)CC3C2)=O)ccn2cncc2c1 Cc1cc(CC(N2CCN(C(=O)CC3(O)CCCN(C)C3)C(C)C2)=O)ccc1Br c1(C(=O)NCC2C(CNC(c3ncn(CC)c3)=O)C2)cccc(N2CC=CC2)c1 Cc1cc(C=CC(=O)NCC(C(=O)N2CC(c3nn[nH]n3)C2)N(C)C)on1 N1(C(C(C)CSc2ccccc2)=O)CCCC(CO)(NC(=O)C2=CSCCO2)C1 C1(C)(CC)CC(NC(C2CC=CC(NC(=O)CCC3CC3(C)C)C2)=O)CCO1 C1(N(C(C(CCC)N(C)C)=O)CC)CCCN(C(c2nn(C)cc2C)=O)CC1 c1(OC)ccc(C=CC(=O)NC(C)CN(C(=O)C(F)CC2CC2)C)c(OC)c1 c1(N2C(C)CC(F)C2)ccc(S(=O)(=O)NCCCCN2CCOCC2)cc1Cl Cn1ncc(C(N2CC(NC(=O)C(O)CC(F)F)C3(CC3)C2)=O)c1S(C)(=O)=O C(=O)(C(F)(F)C(F)(F)F)N(CC(C)(C)NC(c1cc(C)[nH]c1C)=O)C CC(CO)C(=O)N(C(CNC(c1csc(-c2ccccc2)c1)=O)C1CC1)C c1(C(C(=O)NCC(CC)NC(c2cocn2)=O)(C)C)ccc(Cl)cc1 N1(C(C2C(C)CC2)=O)CCC(C)(C)C(C(=O)NCC2(O)CCSC2)C1 c1(C(N(C2CCCC(NC(c3cc(C)c(C)[nH]3)=O)C2)C)=O)cnc2nccn2c1 Cc1ncc(CCC(=O)NC2(c3ccc(Br)cc3)CCCOC2)c(O)n1 C(=O)(CC1=CCCC1)NCC1C(C)CCN1C(=O)CCOC1CC1 c1(C(N2CC(NC(c3cccnc3F)=O)C(F)C2)=O)ccc2c(Cl)ccnc2c1 C1(NC(CCc2cc(C)n(C)n2)=O)CCN(C(c2nnn(C)n2)=O)C12CC2 C1(C(=O)NCc2ccc(NC(C)=O)cc2)CC12CCCCC2 C1(C(=O)NC2(C)CCN(C(c3ccn(CC#N)n3)=O)C2)CC12CCOCC2 C1(NC(=O)CC2CCOC2)CCN(C(=O)CNC(C2CCC2)=O)CC1CO N1(C(C(n2cc(SC)nn2)C)=O)CC2(CCN(N3CC4CCCC3C4CO)C2)C1 N1(CCC(CC)(C)C)CCC(=O)N(Cc2ccc(CC(C)C)cc2)C1=O CCCCN(C(=O)CN(C)C1CC1)C1CCC1 N1(C(CC(C)(C)N(C)C(C2(C)CCCOC2)=O)=O)CCn2ccnc2C1 C#CC1CCN(C(=O)C(CC)NC(c2c[nH]c(C(N)=O)c2)=O)C1 c1(C(=O)NCC(CNC(Cc2c(C)ccnc2)=O)F)c(F)ccc(F)c1Cl S(=O)(=O)(CCC(=O)NCC(F)CNC(=O)COC1CC1)NC c1(OCCNC(=O)NCc2n(C)ncc2)ccc2c3c(c(=O)oc2c1)CCC3 C#Cc1ccc(C(=O)NCC2CC2CNC(=O)Cn2cc(Br)c(C)n2)c(C)c1 CCC(C)C(=O)C(=O)NC1CCCCC1NC(C1CC2(CC(=O)C2)C1)=O N1(C(C2(COCC)CCC2)=O)C(C(=O)NCC2CCCS2)CCC12CC2 C1(NC(C23CC(NC(C(CC)OC)=O)(C2)C3)=O)CCCC(CO)C1 N(C(=NCCCC(F)F)N1CCC(OC)C(C)C1)Cc1nc(CC)on1 N1(C(CCC)=O)CCCCC1C(N1CCC(N(C(c2ccncc2)=O)CC)C1)=O C(=O)(CC1OCc2ccccc21)N1CC(C(N)=O)(CNC(CC(C)O)=O)C1 N1(CC(=O)NCCC(C)NC(=O)C(F)=CC2CC2)CC(=O)Nc2ccccc21 N1(C(C2C3CCCCC23)=O)CC(C2CC2)(C(N2CCOC3CC23)=O)C1 C1(C(=O)NCCCCC2C(C)C2)CCCCC1NC(c1cc[nH]c1)=O c1(C(=O)NC2C(NC(C(C(C)C)NC(COC)=O)=O)C2)c(O)nnc(C)c1C C(=O)(C1=CCCCC1)N1CCC(=CCNC(CN(c2ccccc2)CC)=O)CC1 C1(C(=O)NCCCC(C)NC(C(C)Cn2cccn2)=O)CCC(O)CC1 CC1(C)CC2(CC(NCC3CCCC4CC4C3)C2)C1 N1(C(C(CC(N)=O)O)=O)CCOC2CN(C(C3CCC(F)(F)C3O)=O)CC12 C1(c2onc(-c3c(C)cnc(O)n3)n2)Cc2c(F)ccc(F)c2C(=O)O1 Cc1oc(C(N2CCC(CN(C(=O)C(O)Cn3cncn3)C)C2)=O)cc1Br Cc1cc(C#N)cnc1C(=O)N(C(C)C(=O)NC(C)CC(C)(C)O)C N1(C(c2ccccc2Cl)C(=O)NC)CC2CC(C1)C2NC(=O)OC(C)(C)C c1(-c2cn(C(C(=O)NCC(CC)(C)CO)C)nn2)ccc(C)c(F)c1 CC1=C(C(=O)N2CCC(CNC(=O)CN(c3cnccn3)C)C2(C)C)CCO1 N1(C(=O)NCCCC(=O)N(C2(Nc3ccccc3)CC2)C)CCC2CNCC12 c1(C(=O)NC2C(NC(C3(COC)CCCO3)=O)CCCC2)cc(F)c(C)cc1F N1(C(C2C3CN(C(c4n[nH]c5c4COC5)=O)C2C3)=O)CC(O)C2(CCCC2)C1 C12(CC=C)CCN(C1)C(=O)CCCOC(=O)CNC2=O.C(CC)SC N1(C(C(=O)NCCOCC)C(C2CC2)OC)CCC2OCCCC2C1 N1(C(C(c2cncnc2)C)=O)CCC2(NC(=O)Cc3ccc(O)nc3)CCCC12 Cc1ccc(Cl)cc1NC(=O)C(C1CCN(C(C2C(C)(C)C2(F)F)=O)C1)F C1(NC(CC(C)CF)=O)CCC2(CC1)CC2NC(=O)CCN1CCC(O)CC1 c1(C(=O)NC23CC(NC(c4c(C)cc(F)cc4)=O)(C2)C3)cnc2ncc(Cl)cn12 N1(C(c2sccc2I)C(=O)NC(CC)(C)C)CC(=O)NC(C(C)C)C1 c1(N2CCC(NC(c3cc(SC)c(F)cc3)=O)C(O)C2)ncc2c(n1)COC2 c1(C(N2C(C)CN(C(=O)CS(=O)(=O)NC3CC3)CC2)=O)cnn2cccnc12 c1(C(N(CCCCNC(C(C)OCCC=C)=O)C)=O)c(Cl)cc(C#N)cc1Cl Cc1oc(-c2ccccc2)cc1C(=O)NCC(C(C)C)NC(=O)C=CC=C(Cl)Cl CCS(=O)(=O)CC(=O)NC1CCCC1(C)CN(C)C(c1ncnc(C)c1C)=O C(=O)(C(C)CS(C)(=O)=O)N1CC2(N(C(CCCCCOC)=O)CC2)C1 C1(C(=O)NCC(CCOC)NC(C2CCCC(C#N)C2)=O)CC2CCC1C21CC1 Cc1cc(C2CC2)ccc1C(N1CCC(C)(CNC(c2cnncc2O)=O)C1)=O N1(CC(=O)N(C(C)(C)C)CCO)C2CCCC1CC(=O)NC2 C1(CNC(c2c(C(C)C)occ2)=O)C2CN(C(=O)Cc3ccc(Cl)s3)CC12 C12(C(=O)NCCNC(C3CCS3(=O)=O)=O)CC1CNC2=O Cc1c(Cl)c(C(N2CCCC2(C)CNC(C2(C)CCCOC2)=O)=O)nn1C C1(CNC(C2CCC(CNC(CCNC(=O)OC)=O)O2)=O)CC(O)C(O)C1 C(CCC(=O)NC(C)CNC(=O)C(C)(C)C1CC1)NC(=O)OC CC1CN2CCN1CC2C(=O)NC1CCCCC1CNC(C12CCCC1C2)=O C1(C(=O)NOCC(O)CO)CC2CCC1CC2(F)F N1(C(=O)CCOC2CCOC2)CCCN(C(C2CC(F)(CO)C2)=O)CC1 c1(C(=O)NCCN(C(C2(CO)CC(F)(F)C2)=O)CC)cnn2c1CCCC2 C1(OC)CCCC1CNC(=O)C(C1CC=CCC1)NC(=O)Cc1nocc1C c1(C(=O)NC(C)CF)ccnc(CNC(C2CCCC(F)C2)=O)c1 c1(C(=O)NC2(C3CCCN3C(=O)CCc3nccs3)CC2)cc2n(n1)CC(F)C2 N1(C(CSCC=C)=O)CCN(C(c2conc2C)=O)CCC1C c1(C(=O)NC2(C)CN(C(C(C=C)c3ccccc3)=O)C2)c(C)cc(C)oc1=O Cc1cccc2ccc(C(=O)NC3CCC(NC(=O)C(C)O)C3)nc12 Cc1cccc(N)c1C(=O)NC1CCCC(NC(=O)C=CBr)CC1 CCCCC(CCC)NC(=O)C(=O)Nc1cccc(COCCCO)c1 C1(CNC(C(CSC)(C)C)=O)CN(C(=O)CC(F)(F)F)CCC1C c1(N2CC(COC)OC(C)C2)nc2c(c(=NCCC(F)(F)Cl)[nH]1)SCC2 Cc1cnc(C(=O)N(C)CC2(NC(=O)CC3CCCCCCC3)CC2)cc1Cl c1(OC)ccc(C=CC(=O)NC2CC(CNC(=O)CO)C23CCC3)c(C)c1 c1(CCCN(c2cncc(C(F)(F)F)n2)CC)ccc(N(C)CC)cc1 C(=O)(C(C(F)(F)F)C(F)(F)F)N1C2C(CNC(CC(C(C)C)O)=O)CC(CC2)C1 c1(C(=O)NC2CCCCN(C(CCCCC=C)=O)CC2)cnc2ncnn2c1O N1(C(Cc2c(C)cccc2C)=O)CCC2CN(C(c3ccnnc3S)=O)C2C1 N1(C(CC2CC(=C)C2)=O)CCN(C(=O)C(F)OC(F)(F)F)C(C(C)C)C1 C1(CNC(C2(OC)CCC2)=O)CCC(C)(C)CN1C(c1ccncc1)=O c1(NCC2(C)CCCN(C(CC(CN(C)C)O)=O)C2)ncc2c(n1)CCCCC2 C1(NC(c2coc(C3CC3)n2)=O)CCCCCN(C(=O)C(F)(F)C2CCOCC2)C1 Cc1cc(C(F)(F)F)cc(N2CCCC(C(N3CC(c4ccccc4)C3)=O)C2)n1 C=CCC(CC)C(=O)NCCCOCCNC(=O)CC1CCC(C)(C)CC1 C12(C(N3CC4CCN(C(Cc5c(C)nc[nH]5)=O)CC43)=O)CCC(C#N)(CC1)CC2 CC(C)C(C(C)NC(=O)COC1CCCCCC1)NC(=O)CCc1cnc[nH]1 c1(C(N(CCNC(C(C2CCC(=O)N2)C)=O)C)=O)cc(=O)n(C)o1 c1(C(=O)OC)cccc(CN2CCC(C(=O)Nc3ccc(C)nc3)C2)c1[N+](=O)[O-] C(=O)(CC(O)C(C)(C)C)N1CCN(C(c2ccc(NC(C)=O)s2)=O)CC1C C=CC(CCC)CC(=O)NCC1CCC1NC(c1cc(C#N)c[nH]1)=O C(=O)(C(F)(F)C1=CCOCC1)NCC(=C)CCNC(=O)CC1CCC(=O)N1CC N1(C(c2c(C)nc(C3CC3)s2)=O)CCN(C(=O)C2=CCCC2)C2CS(=O)(=O)CC12 c1(CNC(=O)NC(CC2(NC(c3c[nH]c(=N)s3)C)CC2)C2CC2)ccc(Br)cc1 C12(C(=O)OCC)CC(CC3CC(N4CCN(C)CC4)C3CN)(C1)OC2(C)C c1(C(=O)OC)ccc(OC)cc1NCC(C)COC(c1ccccc1)=O N1(C(CC=CC)=O)CC(OC)CC1(C)CNC(C1(CC(C)=O)CC1)=O C1(C(=O)NCCN(C(C)C)C(c2cnn(-c3ccncc3)c2)=O)CCCN(C)C1 c1(C(C(=O)NC(C)CC)N(CCCOC)C)sc(C(=O)OC)cc1C Cc1cccc(OCCC(=O)NCC2C3CN(CC4CCC(C)O4)CC23)c1C c1(CN(C(C=CC(C)NC(=O)CC(=O)NC2CCOC2)=O)C)ccncc1 C=CC(CC)CC(=O)NC1CN(C(C2CCCC2F)=O)C(C)(C)C1 Cc1cc(CC(=O)NC(C)CC(C)NC(c2cnsn2)=O)ccc1CO CCCCC(CNC(=O)C(C)=CC1CC1)NC(=O)Cc1nccn1C N1(C(C(C)N(C)C)=O)CC(C(N)=O)(CNC(C2CC2(C)Br)=O)C1 CCC(C)(C)C(C)NC(=O)C(C)(C1CCC1)NC(=O)Cn1ccnc1 c1(C(=O)NCC2(CNC(C(CSC)O)=O)CC2(F)F)cc2c(F)ccc(F)c2[nH]1 C(=O)(CC1=CCCCC1)NCCC(=C)CNC(=O)C(F)(F)c1ccnn1C C12(NC(C3C(C)C3)=O)CCCN(C(c3cc4n(n3)CCC4)=O)CC1C2 N1(C(c2c(Cl)cc(C)s2)=O)CCC(C)C(NC(C2CC3CCC2CC3)=O)C1 C1(CC(=O)Nc2cccc(-n3cc(CCO)nn3)c2)CC2OCCC2O1 S(=O)(=O)(c1ccc(NCc2csc(CO)n2)c(F)c1)NCC1C(C)OCC1 N1(C(C(C(C)C)OCC)=O)CCC(O)(CNC(C2(NC(N)=O)CC2)=O)CC1 C#CCCCCCCC(=O)NC1(CCCNC(C2CCS(=O)(=O)C(C)C2)=O)CC1 C=CC1(C(=O)N(CC(C)(C)COC)C)CCN(C(=O)C(C)CC(=O)OCC)CC1 N1(C(c2c(OC)nsc2OC)=O)CC2CC(NC(=O)C(=O)NC(C)C)C(C2)C1 C1(C(=O)NC(CN(C(c2c(CC)nccn2)=O)CC)C)CC2(C1)CC(CO)C2 CC(C)CCCCCC(=O)N1CCC(C)C1C(=O)N(C)CC1OCCC1(C)C C1(C)(CNC(C2(OC)CC(C)C2)=O)CN(C(c2cnc(C)c(N)c2)=O)CCO1 C1(C(=O)NC2CCC(O)CC2)CC2CCC1N(C(=O)Cc1ccc(F)c(F)c1)C2 C=CC(C)(C)CC(=O)NC(C)CCN(C(=O)C(O)C1CCCC1)C O=C(CC1=CCCCC1)NCC1CCCC(NC(=O)CCCc2cnccn2)C1 C1(CNC(c2cnn(-c3nccs3)c2)=O)CC(F)CN1C(=O)CO CN1CCC(C(N2CCCC(C(F)F)C2)=O)(NC(c2scnc2CO)=O)C1 C1(c2nnnn2Cc2ccco2)(NCc2ccc(CC)cc2)COC2(COC2)C1 N1(C(C(COC)OC)=O)CC=CC(NC(C2(CC3CC3)CCC2)=O)C1 N1CCOC2(CCCC2)C1.Clc1ccc(CCCc2ccccc2N)cc1 C1(CN(C(c2ccccc2OC)=O)CC)CCCCN1C(c1cnc(N)cn1)=O c1(CCN(C2CCN(C(=O)CC3COCCO3)C2)C)c[nH]c2ccccc12 Cc1cncc2nc(CC(=O)NCC3(C4=CCNCC4)CC3)cn12 CC1(C)CCC1CC(=O)NCC(C1CCCC1)NC(c1cnc(C(N)=O)s1)=O CN=c1ccc(Br)c(C(=O)NC(C)CN(C(=O)CCC(C)C)C(C)C)[nH]1 c1(C(=O)OC)c(OC)cccc1NC(=O)CCc1cnn[nH]1 C(=O)(CC(C(=O)N1CCC(C2CCCN2C(c2ccns2)=O)CC1)N(C)C)OC N1(C(c2cc(C)sc2)=O)CCN(C(c2nnn(C3CCOC3)c2C)=O)CCC1C C1(OC)CC(NC(=O)COC(C)C)CN(C(C2CC3CCC(C2)C3)=O)C1 C=CCC(CC)C(=O)N1CCN(C(c2cc(OC)nc(Cl)c2)=O)C(C2CCC2)C1 Cc1ccc2c(C)c(C(=O)NCC34CC3CN(C(=O)CC(C)CF)C4)[nH]c2c1 c1(CNC(=O)NCCC2(CC)CCC2)ccc2c(c1)oc(=O)n2C C1(C(=O)NCCCN(C(=O)Cc2ccno2)C)CC12C(=O)Nc1ccccc12 C(=O)(C(CO)C(F)(F)F)NCCC(=O)NCc1nccc(OC)n1 C(=O)(CC(C1CC1)NC(C1(CC)CCOC1)=O)NCC(=C)CC C(=O)(C(C(=O)OCC)C(C)C)NCC1(F)CN(C(C(=O)NCCN(CC)CC)=O)C1 C1(OC)CCN(C)CC1OC.c1(C(=O)O)cc(Oc2ccncc2)ccc1O C(CC(C)(C)C(=O)N1CCCOC(CCNC(c2cc(C)ncc2C)=O)C1)OC c1(CCNC(NNCCC=C)=NC)cc(OCC(=O)OC)cc(F)c1 c1(CC(=O)NC(CN(C(C2C(OC)CCC2)=O)C)C)ccc(Cl)cc1 C(C1=CCN(C(C2(C)CC2Br)=O)CC1)NC(C(CC)Oc1ccccc1)=O C(CCCC(=O)N1CCC1C(C)O)N(C(C(C)(C)OC(C)=O)=O)C C1(C(N(C(C)C)CCNC(C2CCC(F)C2)=O)=O)CCn2ncnc2C1 C1(C(=O)NCCCCCNC(c2cnc(C(C)C)[nH]2)=O)(COC)CC=CCC1 N1(C(c2ccc(CC#N)cc2)=O)CCC12CN(C(c1coc(Cl)n1)=O)C2 C1(NC(c2n(C(C)C)cnc2)=O)CCCC(NC(C2CC2c2cncs2)=O)C1 C1(C#CC(=O)NC2COCCN(C(=O)CC(C)C3CC3)C2)(CC)COC1 c1(C(C)NC2(c3nnnn3CC3CCOC3)CCCC2)csc2ccccc12 C1(C2CCOCC2)(C(N(C)CCN(C(=O)C(C)(C)C(N)=O)C)=O)CCOCC1 N1(C2CN(C(C3C(CCC)C3)=O)C2)CC(NC(=O)CCn2ccc(C)n2)CC1=O C1(CC)CCCN(C(=O)C(C(C)OC)OC)C1C(=O)NCC1CCCN1C(C)=O Cc1cccc(C(=O)NC(C2CN(C(c3cc(Cl)ccn3)=O)C2)C)c1[N+](=O)[O-] C1(NC(C(COC)(C)C)=O)CC12CCN(C(C1CC(CF)C1)=O)CC2 N1(S(c2c(CC(=O)OC)cccc2)(=O)=O)CCS(=O)(=O)N2CCOCC12 CC1(C(=O)NC2CCC(NC(=O)CCCF)CC2)CCC2(CC1)OCCO2 C12(C(=O)NCC3CCN(C(c4cc(C)ncn4)=O)C3)CC(CO)(C1)OC21CCC1 c1(CNC(c2c(C)nc(NC(=O)CN3C(=O)CSC3=S)s2)=O)ccc2cc[nH]c2c1 CCCCCCCCCC(O)C(=O)N1CCCN(C(=O)Cn2cnnn2)CCC1 C1(CC(=O)N(CCOCC=C)C)COCCN1C(=O)CC1(O)CCCOC1 C1(O)(CCC)CCN(C(c2c(CNC(=O)C(C)NC(C)=O)nnn2C)=O)CC1 N1(CC)N=C(C(=O)NCC(O)CCNC(=O)CC2CSCCO2)CCC1=O Cc1nc(N(c2cnn(C3CNC3)c2)C(c2ccc(Cl)c(Br)c2)=O)ncc1F C1(Oc2ccncc2)CCN(C(=NCC2CC3CCC3C2)NC2CCC2)C1 c1(C(N2CCC(NC(C(C)SCCCC)=O)C2)=O)cccc(C)c1[N+](=O)[O-] N1(C(C2(CSC)CC2)=O)CC2CCC1C(CNC(=O)C(O)CC(C)C)C2 CC1CCN(C(=O)C(C)N(C(C)CNC(=O)CCOC2CC2)C)CC1 c1(SC)cc(C(=O)NCC2CN(C(=O)CCC3CC3(C)C)CCO2)c(C)o1 N=c1nnn(CC(=O)NCC=CCNC(c2cncs2)=O)[nH]1 CC12CN(C(c3ccc(OC(F)F)cc3F)=O)CC1CN(C(C1CNC(=O)N1)=O)C2 C1(CNC(C(C=C)O)=O)CN(C(C2CS(=O)C2)=O)CCN1C c1(C(=O)NC2CC(N(C(CC(c3ccc(F)cc3)C)=O)C)C2)c[nH]ccc1=O CCC(C(=O)N(CCNC(=O)C(C)(C1CC1)OC(C)(C)C)CC)N(C)C c1(C(=O)NC2CCCN(c3nnc(C)s3)C2)ccc(O)nc1C N1(C(C23C(CN(C(C(C)CO)=O)C2)C3)=O)C2CCC1CC(CO)C2 C(c1ccc(F)cc1)=CC(=O)NC1CC(CNC(C(COC)C)=O)C(O)C1 N#Cc1cc(N(CCNC(c2csc(Cl)c2Cl)=O)C2CC2)nc(C2CC2)n1 Cc1ccc(C(C)C(=O)NC(C)(C)CNC(c2sccc2F)=O)s1 Nc1ccc([N+](=O)[O-])cc1C(N1CCC(NC(=O)CC2CCOC2)C1)=O C1(CNC(N(CCO)CC)=O)CCCN(c2nccn2C)C1 CC(C)CC(CC(C)C)C(=O)N(C)CC1(NC(=O)CN2CC(C)(C)C2)CC1 Cc1ccnc(CNC(C2CC3CC3N2C(=O)CC2CCOC2)=O)n1 C1CCCC(C(ONC(C2CC(OC)(OC)C2)=O)=O)C1.c1(CN)ccccc1 c1(C(C(=O)OC)NC(=O)CN2C(C)CC3CNCC23)ccc2ncccc2c1 C(CN=c1[nH]cnc2ccc([N+](=O)[O-])cc12)NC(=O)CC(C1CC1)C1CC1 c1(C(=O)NCC2(NC(C=C(C)C(C)C)=O)CCOC2)cc(C)cc2c1CCC2 Cn1ncc(C(=O)NC2CC(F)(CNC(c3ccc(CO)cn3)=O)C2)c1F C(=O)(CS(=O)(=O)C1CC1)N1C(C(C)C)C(NC(c2cc(F)cnc2O)=O)CC1 c1(C2C(NC(=O)NCC3CN(C(C(C4CC4)SC)=O)C3)C2)ccccc1F N1(C(C)=O)CC(F)(F)CC1C(=O)N(C(c1ccccc1C)=O)Cc1ccccc1 C(CCCC(C)NC(=O)CC(C)C)NC(CCN(C)CC)=O C#Cc1ccc(F)cc1CN(C(=O)C(c1ccccc1)NC(C)=O)C1CC1 C(CCC(O)CO)N(C(CCN(CC=C)C(c1scnc1Cl)=O)=O)C n1(CC(=O)NCC(CCNC(C(C)CSC(F)(F)F)=O)O)sc(=O)c2ccccc12 c1(C(N(CCCN(C)C(c2c[nH]cc2-c2cnn(C)c2)=O)C)=O)ccc(N)cn1 Cc1ncc2n1CC(C(=O)NC(C)CC1(O)CCC1)CC2 N1(C(C2(C(C)(F)F)CC2)=O)CCCCC(NC(c2ccc(CO)cn2)=O)C1 c1(C(N(CCN(C(c2sccc2F)=O)CC)CC)=O)ccc2c(c1N)CCCC2 N1(C(CCNC(N)=O)=O)CC(NC(c2ccc(CC3CC3)cc2)=O)C2CCCC12 C1(C(CC)=O)CCCCC1NC(=O)CC1(O)CN(C(=O)CCCn2cncn2)C1 N1(Cc2c(C)scn2)CC2C(C(=O)Nc3n[nH]c(C)c3Cl)C2C1 c1(C(=O)NCCNC(=O)Cc2cn[nH]c2)c(F)cccc1F c1(C(N2CC(CC(=O)NCCOc3ccccn3)C2)=O)ccc(C(F)F)cc1F c1(C(N(C)CCC2CCN(C(c3cnc(Cl)cn3)=O)CC2)=O)cnc(O)nc1O Cc1cc(Br)c2nc(C(=O)Oc3ncc(Cl)c(C)c3Cl)cn2c1 C(CNC(=O)Cc1cncc(C)c1)(CC(C)C)NC(C1(OC)CCCC1)=O C1(NC(c2ccncc2F)=O)COC2(CCN(C(=O)C3=CCOCC3)CC2)C1 c1(OC)cc(CNc2cncc(-c3cccc(C)c3Cl)c2)cc(Cl)c1OC N1(C(c2c(CC)ccs2)=O)CC(OC)CC1(C)CNC(c1cc(C)cc(C)c1)=O C1(CC)CCC(O)(C(=O)NC2CC(CNC(c3cnn(C(C)(C)C)c3Cl)=O)C2)C1 N1(CC(N2CC(O)(CCNC(c3n[nH]c4c3COC4)=O)C2)=O)CCS(=O)(=O)CC1 C(=O)(CC(C)(O)CCC)NC1CCN(c2ccc(C(C)=O)cn2)C(C)C1 CCC(C)CCC(=O)NCC1(OC)CN(C(c2c[nH]nc2Cl)=O)C1 C1(NC(CCC2CCC(=O)NC2)=O)CC2CN(C(c3ccc[nH]3)=O)CC12 Cc1cc(C(=O)N(C2C3CN(C(c4nocc4Cl)=O)CC23)C)cn1C(C)C Cc1cc(Br)cnc1C(=O)N(C)CCN(C(=O)CC1OCCC1(C)C)C C1(CNC(CC)=O)COC(C)(C)C1.C12(CCC1)C(=O)N2C1CC1 CCCCC(C)C(=O)NC1(COC)CCN(C(=O)C(C2CCCCC2)O)CC1 C=C(C)C(C)(O)C(=O)NCC1CCN1C(C1(C(F)F)CCC1)=O C(=O)(C1Cc2ccc(F)cc21)N(CCNC(C(c1cn(C)nc1)O)=O)CCOC c1(OC)ccccc1C(O)C(=O)NCC(C(C)(C)C)NC(c1cc(C)[nH]c1C)=O c1(C(C)NC(C(C)OCC)CO)nc(C)c(C)o1 N1(C(CCN(S(C)(=O)=O)C)=O)CCN(C(=O)C=CC2CCC2)C2CCCCC12 C(=O)(CCN(C)C1CC1)N(C(C#C)C1CC1)CC.C1(=O)CN1C N1(C(c2cnc(OCC)nc2)=O)CCOCC(NC(=O)CC2CC(C)C2)C1 N1(C(C2(C)CC(NC(c3c(C)cn(C)c3)=O)C2)=O)CCS(=O)CC1C c1(C(=O)NCC2CC(NC(C(c3ccnn3C)C)=O)C2)ccc(OCCF)cc1 c1(C(=O)NCc2cn(C3CN(C(C=CC)=O)C3)nn2)ccc2cnc(C)n2c1 C12(NC(C(C)OC3CCCC3)=O)CCCC1N(C(c1cc(C#N)on1)=O)CC2 C(=O)(C1=CNS(=O)(=O)N=C1C)N1C(C)CCC(CNC(CCCOCCC)=O)C1 c1(-n2cc(CN(C(c3ccc(F)c(F)c3)C)C)nn2)cc(N)ccc1Cl C(=O)(C(O)CC(F)(F)F)NC1CC(CNC(c2nsc3ccccc23)=O)C1 N1(C(C(C)(C)c2ccno2)=O)CCCC(CNC(=O)CSc2ccccc2O)C1 c1(CC)ccc(C(=O)N(CCCCCNC(=O)Cc2cnccn2)C)c(F)c1 c1(C(=O)NC2C(NC(c3cc(C)c(O)nc3)=O)CC2)cc(N)c(C)cc1Cl N1(C(=O)OC(C)(C)C)CCOC2(CCCN(C(=O)NCc3cc(F)n[nH]3)C2)C1 N1(C(C2(C)CC2(F)F)=O)CCOC2(CCCN(C(=O)Cc3cnns3)C2)C1 CCC(C(=O)NCC1CCCN1C(C1CCC=CCCC1)=O)C(C)C N1(C(C2C(C)C2)=O)CCC(C2(O)CN(C(=O)CCCc3ccc(O)cc3)C2)CC1 Cc1ccc(O)c(C(=O)N(CC(C)C(=O)NCC2CC(C)(C)CO2)C)c1 c1(C(=O)NC2CC(NC(c3c(OC)c(C)ccc3)=O)C2)cc2ncn(C)c2cn1 c1(C(N2CC(C)C(CNC(C3CS(=O)(=O)C3)=O)C2)=O)cnc(O)n(C)c1=O CCCC(O)CC(=O)NC1CC(C)CN(C(=O)CCC(=O)c2cnn(C)c2)C1 c1(CC(=O)N(C(C(=O)N(C(C(C)SC)C)C)(C)C2CC2)C)ncccc1F C=C(C)CN=C(NCc1ccnc(C)c1)N1CCC(N2CCC2)C1 c1(C(C(=O)NC2CCN(C(c3cnsc3)=O)CC2)(F)F)cc(Cl)ccc1F c1(C(=O)NCC(c2ccccc2)C)sccc1CNC(c1ncnn1C)=O c12ccc(cc1)[nH]2.N1(C(C(=O)NCCC(CC)O)=O)CCC(O)CC1 CCC(C)CCC(=O)N(C(C)(C(=O)NOCC=C(C)C)C1CC1)C c1(CC(=O)NCC2N(C(C3C(C)CCC3)=O)CCOC2)noc2ccccc12 C(=O)(C1CCC(C)(C)c2ccccc21)N(CCN(C(c1scc(C)c1C)=O)C)C C1(C#CC(=O)NCC2CCCC(NC(=O)CSCc3cccs3)C2)(CC)CC1 C1(C(C2(O)CCOCC2)C)NC(=O)N(CCc2nccs2)C1=O c1(OCCC(=O)NCc2cc(OCC)c(O)cc2)cc(C)cc(C)c1C C(=O)(C(O)CC[S+](C)C)N1CCC(N(C(=O)COCC2CCC2)C)C1 Cc1cn2c(n1)CC(C(N1CCCC(NC(=O)CSC(F)F)C1C)=O)CC2 Cc1cc(OCCC#CCN=[N+]=[N-])cc(C)c1S(N)(=O)=O c1(NC(C2(NC(C)C(=O)NC34CC(C)C3C4)CCCC2)=O)ccccc1Cl c1(C(c2n(CCCC)nnn2)NCc2cnn(CCF)c2)cnc(OC)c(F)c1 C1(NC(=O)CCN2CCC2)CC2CCC1N(C(=O)CCc1cnc(O)[nH]1)C2 C1(COC)(CNC(C2(C)CCOC2)=O)CN(C(=O)Cc2cn[nH]c2)C1 N1(C(CC(=C)C)=O)CCN(C2CCN(C(=O)C(C)Oc3ccccn3)CC2)CC1 S(=O)(=O)(c1cccc(N2CCCC(CC(F)(F)F)C2)n1)N(CCC(=O)NCC)C C1(NC(c2sc(C)c(O)n2)=O)COCCN(C(c2cc[nH]c(=N)c2)=O)C1 C1(C)(CNC(CC(=C)C)=O)CCN(C(c2ccc(NC(C)=O)cc2Cl)=O)CC1 c1(Cc2n(CC)c(N3CCC4CCCCC34)nn2)cc2ccccc2c(O)n1 Cc1ncc(CCC(=O)NC2CCCC(NC(=O)CC3CCC3)CC2)c(O)n1 C(=O)(N=c1ccn(CCCc2ccc(C#N)cc2)[nH]1)Nc1ccc(COC)cc1 C1(CCCNC(C(C2CCC2)OC)=O)CN(C(=O)CC2CCCC(C)O2)CCO1 CCCC(O)CN(C)C(C1CCC(NC(=O)CC2CN(C(C)=O)C2)C1)=O Cc1cc(C(N2CCC(C)(NC(=O)Cn3cnnc3)C2)=O)ncc1Br C1(C(=O)NC(CC)CNC(c2ccnn2CC2CCC2)=O)CC2C=CC1C21CC1 C(CCCC(=O)NC(C1CC(NC(c2cccc(-n3ccnn3)c2)=O)C1)C)SC c1(NC(C)=O)cc(C(N2CCC(NC(c3cnncc3C)=O)C2C)=O)ccc1F N1(C(CCCC(C)(C)C)=O)CC(CO)C2(C1)CN(C(c1cccs1)=O)C2 c1(OC)cccc(C(=O)NC2(C3CN(C(C4NC(=O)CC4C)=O)C3)CC2)c1O C(Cc1ccccc1)(C(=O)N(C1CCCNC1)c1ccccc1)NC(C)=O CCCCCC(C)CC(=O)NC1CC(F)(CNC(c2cnc(C(C)(C)C)[nH]2)=O)C1 Nc1nc2c(cc1C(N1CC(N3CCN4CCOCC4C3)C1)=O)CCCC2 N1(C(CC(CC2CC2)NC(c2ncc(OC)nc2)=O)=O)CC2(CNC(=O)N2C)C1 Cc1cc(C)c(C(=O)NC2CCN(C(C34CC(F)(C3)C4)=O)CC2O)c(S)n1 c1(OC)cc(C(F)(F)C(=O)NC2CC(CNC(C3CCCO3)=O)C2)ccc1C C1(CNC(c2ccc(CCC)s2)=O)CCCCN1C(=O)C(C)CC1CCCC1 C(C(C)(CC(C)C)NC(=O)Cc1ccc(C(F)F)cc1)NC(CC(=O)OC)=O Cc1c(C(=O)NC(C)(CNC(C2CC2(F)F)=O)C(C)C)nnn1C C(=O)(CCC(=O)N1CCCC(N(C(=O)CCCc2cc[nH]n2)C)C1)NCC c1(C(N2CC3C(NC(CC(=O)NCC)=O)C3C2)=O)n[nH]c2cccc(OC)c12 C(C)(CC(=O)N1CC2(C1)CN(C(=O)C(N)=O)C2)(C(F)F)N(C)C C(N=c1[nH]c(C(N2CCOC(=O)C2)=O)cs1)c1cccc(C(=O)OC)c1 c1(C(=O)NCCC(C)NC(=O)Cc2nnc(O)s2)cc(Cl)cc(Cl)c1 c1(C(=O)NC2CC(C)(C)N(C(c3ccc(=O)oc3)=O)C2)ccc2nnn(O)c2c1 N1(C(C=CC)=O)CC2CCC(C(=O)NC(C)(C)CC(C)C)(C2)C1 N1(C(CC2CC(SC)C2)=O)CC2COCC(C1)C2NC(=O)Cn1cccn1 C1(C(=O)NCC(C)(C)CNC(=O)CCC(=O)N(C)C)CCC(C(F)(F)F)N(C)C1 N#CC(C(=O)N1CCCC1CNC(=O)C(c1ccccc1)O)c1ccccc1 N1(CC(C2CCOCC2)OCC)C(=O)CN(CCc2cc(Br)cs2)C1=O C1(c2n(CC=C)nnn2)(NCc2n[nH]c(C3CC3)n2)CC2CCCCC12 N1(C(C2CCN(C(c3c(CC)n[nH]c3)=O)C2)=O)CCC2(CCOC2=O)C1 N1(S(=O)(=O)c2cc(C(F)(F)F)cs2)CCc2cc(F)ccc2C1.C1(N)CCNC1 C(=O)(CCC(C)NC(c1cnn(C)c1N)=O)NCC(C)N(C)C1CC1 c1(C(=O)NCC23CCC2CCN3C(c2cc[nH]c2)=O)[nH]nc2ncc(Br)cc12 C(c1ccccc1)=C(C(c1n(CCOCC)nnn1)NC1CCN(C)C1=O)C C1(C(N2C(C(N3CCCC4(CCOC4)C3)=O)C=CC2)=O)C2Sc3ccccc3C12 c1(C(N(CCNC(c2cnn(CCOC)c2)=O)CC)=O)cc(Cl)sc1Cl C(=O)(C1CC(=O)c2cccc(OC)c21)NCC(C)NC(CCC=C)=O c1(C(=O)NCC2(NC(C3CC(=O)NC3)=O)CCOC2)ccc2nc[nH]c2c1F c1(CC(=O)N(C(C)CNC(=O)CCC2CCOC2)C)ccc2ncsc2c1 C(=O)(C1=CCCOC1)NCC(c1ccccc1)NC(C12C(CN(C(C)=O)C1)C2)=O C1(C(N2CCN(C(CC(C)C)=O)C(C3CCC3)C2)=O)CN(S(=O)(=O)N(C)C)C1 Cc1c(C(=O)NCCC2CCC(NC(c3ocnc3C3CC3)=O)C2)c(Cl)nn1C C(=O)(CCCC(=O)N(C)C)NCC=CCNC(CCC=CC(C)C)=O S(=O)(=O)(c1cc(Br)c(F)cc1F)NC1CCN(C(c2ccc(F)c(C)c2Cl)=O)C1 c1(C(N2CC(NC(C(C)CS(C)(=O)=O)=O)C2)=O)cc(Br)c2[nH]nnc2c1 N1(C(C2(O)CCN(C(C(C)c3cccs3)=O)C2)=O)Cc2c(O)n[nH]c2C(F)(F)C1 c1(OCC(=O)NCC(C)(C)CNC(c2csc(O)n2)=O)ccc(F)nc1 c1(CC(=O)NCC2CCCC(NC(=O)CSC(F)(F)F)C2)cccnc1Cl CC(C)CC(C(=O)N(C(C)C(=O)NCC1CNC(=O)CO1)C1CC1)C(N)=O CC(C)(C(=O)NCCCC1(NC(=O)CC2(C)CC2(F)Cl)CC1)c1cccs1 C1(NC(CCCC)=O)CCCC(C(=O)N(C2CCCOC2)CC)C1 c1(C(N2C(CC(=O)NC(C)CC(N)=O)CC(F)C2)=O)c[nH]c2ncccc12 c1(NC(C(=O)OC)Cc2ccc(O)cc2)ncnc2ncnc(Br)c12 CCN=c1[nH]cc(C(N2CC(C(C)NC(c3cccc(C4CC4)c3Cl)=O)C2)=O)s1 c1(CN2C(C)CCC2C(=O)NC2CN(C)C2)ncn2ccccc12 c1(CC(=O)NCC(CC)NC(=O)CC2CC(O)C2(C)C)cccc(F)c1F C(=O)(C(O)CC(N)=O)N1CC(CNC(C2C(OC)CCC2)=O)C1 c1(SCC)ccnc(C(=O)NS(=O)(=O)CCCn2cnnn2)c1 c1(C(=O)NC2CC(NC(C3C4CNC(=O)C34)=O)C2)cc(Br)ccc1F C=CC1(C(=O)NC2CCC(C)(CNC(=O)C=COCC)C2)CCOCC1 c1(CNC(C(CSC)C)=O)ccc(O)c(C)c1C C(=O)(CCP(C)(C)=O)N(C1CCCCC1N(C(=O)C=Cc1ccc[nH]1)C)C c1(C(=O)OC)ccc2c(c1)C(NC(=O)CCCN1CCNCC1(C)C)CCC2 C1(CNC(C2(NC(CCCOC(C)=O)=O)CCOCC2)=O)CC1C1CCCC1 c1(C(=O)NC2C=CC(CNC(c3sccc3-n3ccnn3)=O)C2)cc(Cl)cnn1 c1(CC)c[nH]nc1C(N1CC(O)(C(C)(C)CNC(C2CCOC2)=O)C1)=O c1(C(N2CC3CC2CN3C(c2cnc(Cl)s2)=O)=O)cc2ncccn2n1 CC(C)C(C(=O)NCC1=NOC(C)C1)NC(=O)CCc1ccco1 c1(CC)nn(C)c(OC)c1C(c1nnnn1C1COC1)NCC1CCSC1 Cc1cn2cc(C(N3CCCC(NC(C4CC(O)C4)=O)CCC3)=O)cc(C)c2n1 c1(-n2c(CCCSC)nc(-c3ccc(C(C)C)cc3)n2)ccnc2c1cnn2C Cc1cc(C(N2CCC(O)(CCNC(c3ccco3)=O)CC2)=O)c(Cl)cc1F C(N=c1cc[nH]cc1S(=O)(=O)NC1CCN(CC2CC2)C1)c1c(OC)cccc1F c1(C(=O)NCCSCC(=O)NCC(CNC(C2(C)CCC2)=O)O)ccccc1 Cc1cc(NC(=O)CCC2CCCN2C(=O)Cc2ccccn2)cc(C)c1 N1(C(C2(C)CC(=C)C2)=O)CCC2CN(C(C3CC(N4CCCC4)C3)=O)CC12 N1(C(C2(CC)CCCN2C(c2ccc(C)o2)=O)=O)CCC(OC)C(C)(C)C1 c1(OC)nc(C(N2CCC(NC(=O)CCc3cn[nH]c3)CC2C)=O)cc(O)n1 c1(C(C)OC(c2cc(-c3ccccn3)c[nH]2)=O)cc(Br)ccc1F C(=O)(C(C)CC(C)C)NCCCN(C(C(=Cc1cnc[nH]1)C)=O)C1CC1 CCCCC(C)(F)C(=O)N(C1CC(NC(=O)CCNC(=O)OC)C1)C N1(C(CCC(=O)N(C)C)=O)CCCCC(C(=O)NCc2ccc(CO)cc2)C1 N1(C(C(COCC)C)=O)CC(C)(C)CCC1CNC(c1cscc1C(F)(F)F)=O C(CS(=O)(=O)CC(=O)N(C)CC1CN(C(=O)Cc2nnc3n2CCOC3)C1)OC N1(C(C(CC=C)(C)C)=O)CC2(CCN(Cc3ccc(C=C)cc3OC)C2)C1 C=C1CCC(C(=O)NC2CC3(C2)CC3C(=O)NCCN(C(C)C)C2CC2)CC1 CC1CC(C(=O)NCCN(C(=O)CCN2CCC(O)CC2)CC2CC2)CC(C)C1 c1(C(=O)NC(CCOC)CNC(=O)C(C)=CC2CC2)ccc2cccnc2c1 c1(N2CC3CN(C(C4CCN(C(CC)=O)C4)=O)CC3C2)ccc2nccnc2n1 CC1=C(F)CN(C(C2C=CCN2C(c2cc(C)nc(C)n2)=O)=O)CC1 c1(C(=O)NC2CN(C(COCC(=O)OC)=O)CC(F)C2)cn(C)c(=O)cc1OC CCCCC(O)C(C)C(=O)NCC(CNC(c1cnc2cc[nH]c2c1)=O)CO N1(C(C2CC(C)N2C(C2(C#N)CC(=O)C2)=O)=O)CCOC(C)(C)CC1 c1(CN2CC3(N(C(c4cc(C)c(O)c(C)c4)=O)CC3)C2)c[nH]c2ccc(Br)cc12 N1(C(c2ccc(C)nc2)=O)CC(O)CCC1C(N1CCC(CO)CC1)=O N1(C(C2CC(C(=O)OC)C2)=O)CC(CC(=O)NCCC2CCCN2C)CC1(C)C N1(C(C(c2ccc(C)s2)C)=O)CC(NC(C2(Br)CC2)=O)CC(C)(C)C1 c1(C(=O)NC2CC(CNC(C3(C)CCCCO3)=O)C2)cc(N)ccc1Br c1(C(C)CN(C(=O)CNC)C)cccc(F)c1 C1(NC(c2nc(CC)oc2)=O)CC(NC(=O)CN2CC(=O)NC2=O)CC1O N1(C(c2cnc(C)[nH]2)=O)CC(CNC(c2n[nH]c(C)c2Br)=O)C2(CCC2)C1 C1(NC(c2ccsc2Cl)=O)CC2CN(C(=O)C=Cc3ccc(Cl)cc3)CC12 N1(C(c2cc(CC)no2)=O)CCC2(CC1)CC2C(=O)N(C1CCC(CO)CC1)C CCC(COC)C(=O)NC(C)CCNCc1ccc(C(C)C)cc1.C1(=O)CN1 c1(CNC(C(c2ccsc2Br)N(C2CCC2)C)=O)cccc(Br)c1 c1(COC)nc(NCCOCCN(C)C2CC2)cc(N2CCOC(C)CC2)n1 N1(C(C2(COC)CCCCO2)=O)CC2CC(NC(=O)CC3=CCCCC3)CC2C1 CCCCC(O)C(=O)N1CCCC1CC(=O)Nc1c(OC)ncnc1OC N1(C(C(C)(C(C)C)NC(C)=O)=O)C2CCCC1CN(C(c1cnccn1)=O)C2 c1(C2C(CNC(=O)CCn3ccnc3)C2)c(F)cccc1F C1(NC(COCCOC)=O)CCC12CN(C(=O)CCn1ccc(O)nc1=O)C2 C1(C)(C(C)(C)C)CC(C(=O)NC2CC2NC(C2CC3CC3C2)=O)C1 N1(C(CCN(C(C(C)CC#N)=O)C)=O)CCCCC(C)(F)C1 C1(N(C(CCOC)=O)CC2CC2)CCN(C(=O)CC2CN(C(C)=O)C2)CC1 C1(NC(C2C(=C)CC2)=O)CC(CNC(c2c[nH]nc2OCC(F)F)=O)C12CCC2 c1(C(N2CCC(NC(C(CC#C)C)=O)(CO)CC2)=O)cc(OC)cc([N+](=O)[O-])c1 c1(C(N(C2CCN(C(C(COC)C)=O)C2)C)=O)cncc2[nH]ccc12 CC(C)(CC(F)(F)F)C(=O)NCC(C1CCCN1C(=O)CN1CCOCC1)(C)C C(=O)(CC(C)C(C)(C)C)N1CCC(O)(CNC(c2c(CC)ccs2)=O)C1 C1(C)(C(N(C(CF)CF)C)=O)CC(O)CN1C(c1cc([N+](=O)[O-])n[nH]1)=O C(=O)(C1=NOC2COCC12)N(C1CN(C(=O)CCn2cccn2)CC1(C)C)C N1(C(C=CCC)=O)CCCCCC1CNC(C1(C=C)CC1)=O C1(NC(CCNC(CC(C)C)=O)=O)CC(CNC(=O)CC=C(Cl)Cl)C12CCC2 c1(C(N2C(CNC(c3cnn4cc[nH]c34)=O)CCC2)=O)cccn(O)c1=O c1(C(N(C)Cc2nc(C(C)(C)C)cs2)=O)ccc2c(c1)NCCNC2=O N1(CCCC=C)CC2CCC1C1CN(C(c3cc(C)ccc3[N+](=O)[O-])=O)CC21 c1(N2C(=O)CC(C(=O)NCC(COC)(C)C)C2)ccc2nc(C(C)C)oc2c1 C1(O)(CNC(C2(C)CC2(Cl)Cl)=O)CCCN(C(=O)C(F)(F)C(F)F)C1 CCC(CC(C)C)C(=O)NCCN(C(C1C(F)(F)C12CC2)=O)CC1CC1 N1(C(C(CC)c2cccnc2)=O)CCCC(CNC(c2ccn(C)n2)=O)C1 C1(C(N2CCC(NC(C34CCC(F)(CC3)C4)=O)CC2)=O)CCCCC(F)(F)C1 c1(COC(C(C2CC2)NC(C)=O)=O)ccc(CS(C)=O)cc1 C(=O)(CC1COc2ccccc21)NC(CNC(C(C(=O)OCC)(C)C)=O)C c1(NC(C23CC(Cl)(CO2)C3)C)nccc(C(F)(F)F)n1 c1(C(N2CC(C(C(C)NC(c3ccco3)=O)OC)C2)=O)cc(CC2CC2)on1 c1(CCC(=O)NCC2N(C(c3cnc(C)o3)=O)CC2)c(C)noc1C CC1=C(C(=O)N2CC(NC(=O)Cc3ccc(O)cc3)CC2(C)CO)SCCO1 C1(C(=O)NCC2C=CC(NC(Cc3n[nH]c(=NC)s3)=O)C2)CCCC12CC2 c1(C(C)C)nc(C(=O)N(C(C)C(=O)NC(c2nncs2)C)C)co1 c1(C(N2C(CNC(CCCCCOC)=O)CC(F)C2)=O)sc2ccccc2c1C CCCCC(CNC(=O)C(c1ccc(Cl)cc1)=O)NC(c1cnn(C)c1)=O CC(C)C(C(=O)Nc1ccc(C(=O)NC(C2CCOC2)C)cn1)c1ccccc1 CCCC(CC)CC(=O)NCC(CNC(c1ccc(CO)c(Cl)c1)=O)CO c1(C(N2CCC(NC(=O)C=CSCc3ccco3)(CO)C2)=O)c(F)ccc(F)c1Cl N1(C(CCCC(C)=O)=O)CCC(O)(C2(NC(c3cc(Br)no3)=O)CC2)CC1 C1(NC(C(C)OCC#C)=O)CC2CCC(C1)N2c1ncns1 C1(OC)CC(CNC(=O)CC2CCC=CCC2)N(C(=O)C(C(C)OC)N(C)C)C1 CNS(=O)(=O)N1CCC(C(=O)NCc2ccc(CC(F)F)cc2)CC1 N1(C(C2N(CC)CC2)=O)CCCC(C2CC2NC(c2ccsc2)=O)C1 C1(NC(C=CCNC(Cc2ccn(C)c2)=O)=O)CCCC(C)(C)C1 C1(CC(=O)NCC#CCC)CN(C(c2cc(F)ccc2O)=O)CC12CC2 c1(C(=O)NC2C(CNC(CCN(CCC)C)=O)CC2)sc(=N)[nH]c1CC c1(CCC(=O)NC2C(NC(C(C)NC(CC)(C)C)=O)C2)ccc(OC)c(O)c1 C1(NC(c2cc(SCC)ncc2)=O)CCCCN(C(C2(CO)CCOCC2)=O)C1 C(=O)(C1CCc2nccn21)NC(C(=O)N(CC(CC)C)C)C(C)(C)O NS(=O)(=O)c1cccc(CC(N2CC3(CC=CC3)C2c2ccccc2)=O)c1 Cc1ccc(SCC(=O)NCC2CC2CNC(c2ccc(C3CC3)o2)=O)cc1 C1(C(N(C)CC2(CNC(c3cnco3)=O)CC2)=O)CCCCS1(=O)=O C12(C(=O)NCCC(=O)NCC#C)CC(CN(C(c3cn(C)cn3)=O)C1)C2 C1(n2cc(C(CC)O)nn2)CCC(C(=O)NC(c2cccnc2)C)CC1 C1(CNC(C2N(CCC)CCC2)=O)CCCCN(C(=O)C(C)=C2CC2)C1 C1(C(=O)NC(C)(C)CCNC(c2ccnn2C2CCCCC2)=O)CCC12CCC2 N1(C(CCOc2ccc(OC)cc2)=O)CC2CC1CC2NC(=O)C(C)=C1CCC1 C(=O)(CCCCC#N)NCCOCCCN(C(=O)CCC1(C)CC1)C c1(C(N2CC(NC(c3ccc(OC)c(Br)c3)=O)C(F)C2)=O)cc2ccccc2o1 Cc1ccc(-c2cn(-c3ccccc3C(=O)N(C)C(C)C)nn2)c(C)n1 N1(C(c2cc[n+]([O-])cc2)=O)CC2(CCCN2C(c2ncn(-c3ccccc3)n2)=O)C1 N1(C(Cc2ccc(C)s2)=O)CC=C(CC(=O)NCC2(O)CCC(C)C2)CC1 c1(N2CCC(C)(C(=O)NC3CC3)C2)ccn2nccc2n1 N1(C(c2c(C)[nH]cc2)=O)CCC2(CC1)CC2NC(c1sccc1OC(F)F)=O c1(-c2n(CCC(N)=O)ccn2)cccc(S(=O)(=O)N2C(=O)CCC2=O)c1 c1(-c2nc(C(=O)NC(c3ccsc3)(C)C)sc2)c[nH]c2ncc(Br)cc12 C1(C(N2CCC(n3cc(-c4n(CC)ccn4)nn3)CC2)=O)Cc2nnc(C)n2C1 CC(CO)(C(=O)NC1CC2CCC1O2)NC(=O)CCCc1cnn[nH]1 S(=O)(=O)(c1ccc2ccccc2c1)N1c2nc(cs2)C1.C1(CC)CCCNCC1 C1(NC(CC2C=CC(NC(=O)CCCC3CCCO3)C2)=O)C2C=CC(C2)C1CO Cn1nc(-c2cccnc2)cc1C(=O)NC1CC1NC(c1ccon1)=O CC#CCC(C(=O)NCC(F)CNC(c1c(CC)noc1C)=O)c1ccccc1 C1(C(=O)NCc2nc(C(=O)OC)sc2)CCCCN1C(c1ccc(F)nc1)=O c1(C(N2CC(NC(CN(C)CC)=O)C(CO)C2)=O)ccc(C)cc1O N1(C(Cc2cn(CC)nc2)=O)CCN(C(C2C3CCCC23)=O)C(CC2CC2)C1 C1(C)(C(N(CCOC)C)=O)CN(C(=O)CNC(c2ccc(F)cc2)=O)C(C)(C)C1 Cc1ccc2c(c1)CN(CC(C1CCC1)NC(=O)OC(C)(C)C)CC2 C1(C(=O)NCC(CN(C(C2(OC)CCSC2)=O)C)(C)C)CC2(CO1)CC(F)(F)C2 c1(C(N2C(C)CC(CNC(=O)C3=CS(=O)CCC3)C2)=O)cc2ccccc2cn1 c1(C(=O)NC2CN(C(CC(C(=O)OC)C)=O)CC2O)cc2c(Cl)cccn2n1 C(c1c(Cl)cccc1Cl)=CC(=O)NCC(CNC(C(C)(Cl)Cl)=O)O C12(C(N3CC4CCN(C(c5ncn(C)c5)=O)CC43)=O)CCCC(=O)N1CCC2 c1(NC(C2C(NCc3cc(C)sc3C)CCC2)=O)c(F)ccc(Cl)c1F CC(C)(C(=O)NCc1cc(C(=O)NC2CCN(C(N)=O)C2)n[nH]1)C(F)F Cc1nc(NCc2nc(C3CC3)cs2)cc(=NCC2(C)C=CCCC2)[nH]1 N1(C(CCCOC(C)=O)=O)CC(=O)CC1C(=O)NCC12CCC(CC1)O2 c1(C(N2C(CCNC(C=C(COC)C)=O)CCC2)=O)sccc1C#N C1(NC(=O)CCF)CC2CC(C1)CN(C(=O)C(c1ccc(F)cc1Br)O)C2 C1(N(C(CC=CC=C)=O)C)CCCN(C(=O)CCc2nncs2)CC1 CC1=C(C(=O)NCC2(F)CC(CNC(=O)CCCN3CCCCC3)C2)CCO1 c1(C(N2CC(NC(c3cc(OC)c(C)cc3)=O)C(C)C2)=O)cccc([N+](=O)[O-])c1 C1(NC(COC2C(C)CCCC2)=O)CCSC12CN(C(=O)C(C)(C)C1CCC1)C2 c1(OC)c(C)ccc(NC(c2csc(C3CCCCC3)n2)=O)c1C C12CN(CC1(C)C)C2=O.c1(NC(C)=O)ccc(NC(c2cccn2C)=O)cn1 C1(c2n(CCC)nnn2)(NC2CCC(NC(C)=O)CC2)CCN(C(C)C)CC1 c1(C(C(=O)NC2C(NC(c3c(CCC)nns3)=O)CCC2)C)ccc(F)cc1F C#CC1(C(=O)NCCOCCC(=O)NC2CC(C)C2)CCCCC1 C1(C(=O)NC(c2cnn[nH]2)C)CC12CC(NC(c1ccncc1Cl)=O)C2 c1(NC(C(=O)NCc2c(C)cccc2)=O)ccnc2c1CCO2 C(CC(C)(C)C)(C(=O)N(CCC(C)O)C)NC(CC1CCC(C)CC1)=O C1(C(N(C(C(=O)OC)C)C)=O)CC(C)(C)CCN1C(c1cc(C(C)C)no1)=O C1(NC(c2c(C)ncs2)=O)CCCC12CCN(C(c1cc3n(n1)CCCO3)=O)C2 C1(C(=O)NC2C(NC(CC(C)CF)=O)CCC2)CC2CC(C1)CC(F)(F)C2 Cc1n[nH]cc1C(=O)NCC1(C(=O)NC(C)(C)CN2CCCC2)CC1 C(=O)(C1=CCCC1)N1CCC(N(C(=O)CN(CC(=O)NC(C)C)C)CC)C1 CC(c1ccc(F)cc1)=CC(=O)NC(Cc1ccccc1)CCC(=O)O CCC(C)(CCNC(=O)C(=CC1CCCCC1)F)NC(C1CC(C2CC2)C1)=O C(CC(C(=O)N(C)CP(C)(C)=O)NC(=O)Cc1cnccc1C)=CC N1(C(C(=O)NC(C)C)=O)C(C)CC2CN(C(c3ccc4ncncc4c3)=O)CC12 C1(NC(CC(CC)O)=O)CC2(CCCN(C(=O)C#CC3(CC)COC3)C2)C1 C1(CC(=O)NCC2C=CCN2C(c2ccnnc2O)=O)(OC)CCCCC1 c1(NC(C2CCCN(Cc3ccc(CC(=O)OC)cc3)C2)=O)c(O)cccc1O N1(C(C(CC#C)O)=O)CCCC(NC(c2cccn2Cc2ccncc2)=O)C1C C1(CC(=O)NCc2ccccc2)CC2(C1)CN(C(C1CCS(=O)(=O)C1)=O)C2 C1(CNC(C(CC)F)=O)(NC(c2ccccc2OC(F)F)=O)CCOCC1 O=C(C#Cc1ccc(Cl)cc1)NC1CCN(Cc2cc(F)c(F)cc2F)C1 CCCC(C)(O)C(=O)NC1(CN(C(=O)CCCOc2ccc(C)cc2)C)CC1.OCC Cc1ccc(C(=O)NCC2CCCCN2C(c2c(F)ccnc2Cl)=O)c(Cl)c1 c1(C(N2C(CC(=O)O)CC3(CCC3)C2)=O)c[nH]c2c(F)c(Cl)ccc2c1=O Cc1ncnc(C(N2CCC(C(C)(C)NC(c3c[nH]cc(F)c3=O)=O)C2)=O)c1C c1(NC(C)C(C2CCCCC2)NC(=O)CCC2CCCCCC2)ncc(I)cn1 c1(C(=O)NCC2(CNC(CC(C)C)=O)CCCC2)sc(Cl)cc1Cl CCC(CC)CCC(=O)NCC(C1CCN(C(=O)C(CN(C)C)N(C)C)CC1)C c1(-c2c(C)ccs2)ccc(CN2CCC(c3c(C(=O)NC)nccn3)C2)nc1C C(c1ncco1)=CC(N1CCC1CNC(=O)C(c1ccccn1)C1CCCC1)=O Cc1c(N)ccc(C(=O)NC2CS(=O)(=O)CC2NC(c2cocn2)=O)c1Cl C=CCC(C(=O)N1CC(N(C)C(C2(OC)CCOCC2)=O)C1)c1ccccc1 C1(C(N2C(C)(CNC(=O)Cc3csc(=N)[nH]3)CCC2)=O)CCCS(=O)(=O)C1 CCCCCCCCC(=O)N1CC2(C1)CN(C(C1CC(OC)C1)=O)C2 CC1CCC(NC(c2ccc[nH]2)=O)CN1C(c1cc(Cl)ncc1O)=O Cn1nc(Br)c2ncnc(N3CC=CC(NC(=O)CC4CC(O)C45CCC5)C3)c12 N1(C(C=C(CCC)CCC)=O)CC(N(C)C(c2[nH]c(=N)ccc2C)=O)C2(CC2)C1 c1(OC)cccc2cc(C(=O)NC(C)CC(C)NC(=O)C(C)(C)N3CCCC3)[nH]c12 C1(C(N2CCC(C(C)(C)NC(c3cn(C)nn3)=O)CC2)=O)CCC(N=[N+]=[N-])CC1 C(=O)(CC(C(=O)Nc1ccc(F)nc1)N1CCCCC1)OC C1(NC(CCN(C)CC)=O)C(CNC(=O)Cc2ccccc2Cl)CCC12CCC2 c1(CC)cc(C(=O)Nc2cccc(NC(=O)CN3CCCCC3C)c2)oc1CC N1(C(C2(C)N(C(c3c(CC)nn[nH]3)=O)CCC2)=O)CCC2(CCOCC2)C1 N1(C(C2N(C(C(C)C)=O)CCCC2)=O)CCN(C(=O)C#CC2CC2)CC(C)(F)C1 c1(C(=O)NC(C2CN(C(C3CCCCC(=O)C3)=O)CCO2)C)nc(Cl)ccc1Cl S(=O)(=O)(C1CN(C(C2(O)CC2)=O)C1)N1CCN(C(C2CCCC(C)C2)=O)CC1 c1(SC)ccc(C=CC(=O)NCC(C)N(C(=O)CCC2CCC(=O)N2)C)s1 C1(C)(C(=O)Nc2cncc(COC)c2)CC12CCN(Cc1ccc(C)s1)CC2 C12(C(=O)NC(C3(O)CCN(C(CC(C)CF)=O)C3)C)CC3CC(C1)CC(O)(C3)C2 Cc1cc(C)c(C(N2CCC(CNC(c3cnn(C)c3C3CC3)=O)C2)=O)cc1N C=CC(F)(F)C(=O)N(CC(=O)NCCOC1CCCC1)CCOC.C(C)(=O)O C1(F)(CNC(C2(Cl)C(C)(C)C2)=O)CCN(C(=O)CCCN2CCCC2)C1 C1(O)(CNC(c2cn(C3COCC3F)nn2)=O)CCN(C(=O)Cc2cnsc2)C1 c1(C(=O)NC2C(C#N)CN(C(C3(O)CC3)=O)C2)ccc2[nH]nc(Br)c2c1 c1(N(C(C(C(C)C)n2cncn2)=O)CC(C)C)ccc(Cl)c(Cl)c1 C1(CC)(NC(=O)CN(c2ccccc2)C)CCCN(C(=O)Cc2ccc(C)o2)C1 CON=Cc1ccc2cc(S(=O)(=O)NCCC3CCSCC3)ccc2c1 CCC(C)(O)C(=O)N1CC(C(NCP(C)(=O)OCC)=O)C(C)C1 N1(C(C(CC)(C)CNC(c2cc(C)c(C)s2)=O)=O)CCCC2C(=O)NCC12 c1(CC(=O)NC23CC2CN(C(C2(C(F)F)CC2)=O)C3)nsc2ccccc12 C(=O)(C#CC1CCOC1)C1(C(=O)OC)CCN(C(c2cc(C)cnc2O)=O)C1 CCC(C)C(C(=O)NC1CCC(O)CC1)N(C(=O)C1=CCCCC1)C c1(CCNC(C2CCC(F)(F)C2)=O)cccnc1O N1(C(C(CC)(C)C)=O)CCC2(NC(=O)Cc3cncnc3)CCCC12 C1(NC(CC=C(C)C)=O)CCC2CN(C(=O)COC3(C)CCC3)CC2C1 N1(C(C2CC2(F)Cl)=O)CCC2(CC1)CC2c1cn(Cc2ccc(O)c(O)c2)nn1 C(=O)(CCC(C)(C)[N+](=O)[O-])NC1CCCC(NC(CCCc2scc(C)n2)=O)C1 c1(C(N2CCN(C(c3ccc[nH]3)=O)CC2c2cn[nH]c2)=O)cc2c(s1)CCOC2 C1(C(=O)NC2(C)CC(NC(=O)Cn3ncc(O)nc3=O)C2)Cc2ccccc2S1 N1(C(c2cc(CC)[nH]n2)=O)CCC(NC(=O)C(C)CCC(C)(C)C)C2(CCC2)C1 C1(CNC(c2n(CC)cc(Cl)c2)=O)N(C(=O)C(F)=C2CCCC2)CCCC1(C)C N1(C(C(=O)Cc2ccc(F)cc2)=O)CC2(CC2)CC1CNC(=O)Cn1nccn1 C1(NC(C(C)SC)=O)COC2(CNC(=O)C(c3ccc(C)cc3)(F)F)CC1C2 c1(C(N(C(CNC(=O)Cc2cccs2)C2CC2)C)=O)cn(-c2cnn(C)c2)cn1 c1(C(N2C3C(C(=O)NCCC4C(C)CCCC4)C(C3)C2)=O)cc(F)c(F)cc1Cl N1(C(CCC=C=C)=O)CC2CCC(NC(=O)C=CCN(CC(F)(F)F)C)C2C1 c1(CC)cccc(NC(C2CC=CC(NC(=O)CNC(=O)CC)C2)=O)c1C N1(C(CC(=O)OC)=O)CCC(C)C1CNC(=O)CC1CCC(C)CO1 C1(NC(=O)Cc2cc(C3CC3)on2)CN(C(=O)C2=C(Cl)CCC2)CCC1O C1(CC(N2CCC(CC(C)NC(=O)C(C)CC)CC2)=O)(CSC)CCOCC1 S(=O)(=O)(c1ccc(CC#N)cc1)NC(c1ccccc1O)C C=CCCC(CC(C)C)C(=O)NC1CN(C(c2ccc(C)c(C)c2N)=O)C1 CCN=c1[nH]cnc2cc(C(=O)Nc3ccc(C(C)=O)cc3)ccc12 Cc1cccc(OCCC(N2CC3CC3(NC(c3cc(CO)oc3C)=O)C2)=O)c1 c1(C(=O)NC(C2(O)CCN(C(c3cc(Br)n[nH]3)=O)C2)C)noc2ccc(Cl)cc12 O=C1CCC2C(C(=O)NCc3ocnc3C(=O)NCC=CCl)C12 c1(C(CCCC2(NC(=O)C(=O)N(C)C)CC2)C)ccc(C(C)(C)C)cc1 C(=O)(C1CCCc2n[nH]cc21)NCCC(C)N(C(c1nccc(SC)n1)=O)C CC(CC(C)(C)C)C(=O)NC1CCC1C(N1CCC(O)(C(N)=O)CC1)=O C(=O)(C1=C(C)OCCS1)N(CCCC(=O)NC(CC)(C)CC)C CC1CCC(NC(c2cn3c(n2)SCC3)=O)CN1C(c1nnn(C(C)(C)C)n1)=O C(=O)(CCCCCOC)N1CCC(CN(C(C2C(C(=O)OC)CCC2)=O)C)CC1 C1(NC(c2cc(Cl)ns2)=O)CCCC(CNC(C2(Cc3ccsc3)CC2)=O)C1 c1(CNC(c2cc(C)cc(C)c2)=O)ccc2c(c1)CN(C(c1cncnc1)=O)C2 c1(N(C(=O)CN2Cc3ccccc3C2)CCO)nc2c(s1)CC1(CCOCC1)CC2 n1(C(CC)C)ncc(C(=O)NCC(C)N(C(=O)C(C)CC)C)c1C C1(C(=O)NCC(C)(C)CNC(=O)CC2(C)CC2(Cl)Cl)NC(=O)OC1(C)C C#Cc1ccc(C(=O)NC2C=CCN(C(=O)C(C)CC(N)=O)C2)c(C(F)(F)F)c1 O=C(CC1=CCCC1)NCC1C2CN(C(=O)CCOCC(F)(F)F)CC12 c1(-c2ccn(COc3c(Cl)scc3)n2)nc(C2CC2)nn1C1CC1 C1(NC(CSCCOC)=O)CC(NC(=O)C(c2cccc(Cl)c2)(C)C)C12CCC2 c1(C(N2CCOCC(NC(C3C(C)CC(C)O3)=O)C2)=O)cccc2c1ncn2C Cc1ccn2nc(C(N3CC(C)C(NC(C4CCSCC4)=O)C(C)C3)=O)nc2n1 c1(CC(N2C(C)CC(NC(c3cc(C)sn3)=O)C2)=O)cc2ccccc2c(O)n1 C12(C(=O)NCC3CCN(C(c4ccoc4)=O)C3)CC3CC1C2C3 CCC(C)(C)C(C(=O)N1CCCCC1CCCNC(=O)CCOC(C)C)OC CCCCC(CNC(=O)Cc1nc(O)n[nH]1)NC(c1ccc(-c2cccs2)s1)=O C1(F)(CNC(c2cnc(O)s2)=O)CCN(C(=O)C(c2ccc(Cl)cc2)O)CC1 c1(C(CC)NCc2c(F)cc(F)c(F)c2F)cccc(S(N)(=O)=O)c1 c1(C(C)=O)ccc(NC(c2cnc(NC(c3ccc(Br)cc3C)=O)s2)=O)cc1Cl Cc1cnc(C)c(NC(=O)C(C2CCN(C(=O)CNC3CCCC(O)C3)C2)C)c1 C1(CNC(C2CC=CCC2C(F)(F)F)=O)CC2(CCC2)CN1C(=O)CO N1(C(c2n(CC(C)C)ncc2)=O)CC2CCC(NC(=O)Cc3cn[nH]c3)CC2C1 C=CC(CC)CC(=O)NCCCCC1CCCN(C(=O)Cc2cn[nH]c2)C1 c1(C(=O)NCC2N(C(c3ncc(NC)nc3)=O)CC(OC)C2)c(C)[nH]c(C)c1C c1(OC)c[nH]c(C(=O)NCCN(C(C2CCOC(C)C2)=O)CC2CC2)cc1=O c1(C(=O)NC)ccc(C(=O)N(C)CC2(O)CN(C(=O)C=CCCC(C)C)C2)cn1 N1(C(C(=O)CC#C)C)CCNC1=O.c1(C(CNC)C)nn[nH]n1.C1C(=O)N1 C1(C(=O)Nc2ccc(N(C)C)cc2)(CC)CCN(c2ccc(C(=O)O)cn2)C1 C(c1ccc(I)o1)=CC(=O)OC.N1(CCO)CC1 C(=O)(CC(C)(C)CC(=O)OC)NC1CC(F)(CNC(c2c(COC)noc2)=O)C1 C1(CNC(c2c(CC)[nH]c(=N)s2)=O)C(C)CCCN1C(=O)C(O)C(C)C c1(CC)cc(C(=O)NC2CC23CCN(C(=O)CCCF)C3)cc(O)n1 Cc1cc(CC(N2CC(CCCCNC(C3(N4CCNC4=O)CC3)=O)C2)=O)cs1 N1(C(=O)CC(F)(F)F)CCC2CCN(C(C3(F)CC4(CCC4)C3)=O)CC2C1 N1(C(C=COCC)=O)CCC2(CCC(CNC(C3CN(C)C3)=O)O2)CC1 C(=O)(C1=CCSC1)NCCNC(C1CN(C(C(N2CCCCC2=O)C)=O)C1)=O C1(c2n(CC)c(N3CCC(CO)C34CC4)nn2)CCCCCCC1O c1(CNC(c2n(C(CC)C)nnn2)CC(C)C)cccc(Cl)c1Br c1(OC)c(NC(C2CCCN2C(=O)CC2CCCN2C(C)=O)=O)cnn1C C1(C(C)C(=O)NCC(C)(C)F)CCCN(C(C2(CF)CC(=O)C2)=O)C1 N1(C(C(C(C)C)(C)O)=O)Cc2ccccc2CC1CNC(=O)CC1CCN(C)C1 Cc1oc(C)c(C(N2CC(NC(=O)CCc3cnoc3)C(C)C2)=O)c1C c1(C(N2C(CN(C(CCOCCOCC)=O)C)COCC2)=O)cccc(C)c1F C1(NC(c2nnc(C)s2)=O)CC(O)CN(C(=O)Cn2cc(C3CC3)cn2)C1 C1(C#N)(C(N2CCC(OC)(CNC(C3CCC3(F)F)=O)C2)=O)CCCCCC1 C1(C(N2CCC(NC(Cn3nnc(=N)[nH]3)=O)(CO)C2)=O)CCc2nc[nH]c2C1 C1(NC(COC(CNC(C2(C(C)(F)F)CC2)=O)(C)C)=O)CC(F)(F)C1(C)C CS(=O)(=O)c1sccc1C(N1CCCC2OCCC12)C(=O)NC1CCOC1 N1(C(c2c(C)n(C)nn2)=O)CCN(C(=O)CC(C)NC(C2CCCC2)=O)CC1C c1(C(N=c2ccn(C)[nH]2)=O)csc2c1CCN(C(c1cc(F)nc(F)c1)=O)C2 C(=O)(CC(C(C)C)OCC)N1CCC(NC(C2(C=C)CCC2)=O)CC1 C1(CNC(COCCOCC)=O)CNCCN1C(C1CN(C2CCOC2)C1)=O c1(CC)cc(CC(N2CC(CC(F)C(=O)NCCCCc3cnc[nH]3)C2)=O)on1 CCCCC(CC)CC(=O)NC1CCC(N(c2nc(C)nc(Cl)c2C)C)CC1 c1(C(N(C)CCNC(C2(O)CCC2)=O)=O)ccc2c(c1)NC(C)CC(=O)N2 C(c1ccc(F)cc1)=CC(=O)NC1CCC(N(C)C(c2ccco2)=O)CC1 N1(c2ncnc(=N)[nH]2)CCCC1C1CCCCN1C(C1CCN1)=O.C1CCCC1 c1(C(N(C)C)=O)cccc(CNC(N2CCCC(n3cc(C4CC4)nn3)C2)=O)c1 C1(C)(CCC)CCN(C(=O)C(C)(C)CNC(C2CC=CCO2)=O)C1 c1(NCCN(C(C)=O)CC)ccnc(C(=O)OC)c1.C1(=O)C(C2CCOC2)N1 c1(C(=O)NC2(C(=O)O)C(C)C2)cccc(Cn2cc(-c3ccccn3)nn2)c1 CC1(C)CCCCC1CC(=O)NC12CCC(CC1NC(c1ccc(C#N)o1)=O)C2 CC1=C(C)CC(C(=O)NC2COCC2NC(c2c(Br)cnn2C)=O)CC1 C1(C(=O)NC(C)CO)CCN(C(c2cc(CO)on2)=O)CC1.CC(F)(F)C1(CO)CC1 C1(NC(C2CC(NC(C3C(C)CC3)=O)C2)=O)CCC(CN(C)C)CC1 CCCCC(C)C(=O)NC12CC1CN(C(c1conc1C1CCC1)=O)C2 c1(C(N2C(C(=O)Nc3cc(C)cc(O)c3)CC2C)=O)cc(C#N)ccc1C c1(C(N(C(C=CC(=O)N(CC(C)C)CCOC)C)CC)=O)ccccn1 N1(CC(n2nccn2)C)CCC(Cn2ccnc2)CC1 CC(C)S(=O)(=O)C(C)C(=O)N1CC(NC(c2nc(=O)n(C)[nH]2)=O)C(C(F)(F)F)C1 N1(C(=O)OC(C)(C)C)CCN(C(c2ccccc2OC(F)F)=O)CC1C(=O)O C1(CNC(c2ncccc2Cl)=O)C2CN(C(C3(CF)CC3)=O)CC12 N1(C(C2(C(=O)OC)CC2C)=O)CCC(C)(NC(=O)C(=Cc2cccnc2)C)C1 C(=O)(C(=O)N=S(C)(C)=O)NC(CCCNC(CN1C(C)CCC1C)=O)(C)C N1(C(CNC(C)=O)=O)CC2(C(=O)NCc3c(O)cccc3F)CCC1CC2 C(=O)(CCCC(=O)N(C)C)NC1CC(C)N(C(=O)COCc2ccnc(O)c2)C1 CS(=O)(=O)c1ccnc(N2CCOCC2CC(=O)Nc2cc(C#N)ccc2Br)n1 N12C3CCC1CC(C3)C(=O)OCC2.N1(C(C)=O)CCC(O)CC1 Cc1cnc2ccc(C(=O)NC3(CNC(C4(Cl)CC4(C)C)=O)CC3)cn12 Cc1nn(C)cc1CN(C(=O)CN1CC2CC2C1)C(=O)CN1CCC(CO)CC1 c1(C(C(=O)NCC)N(C2(C3CC3)CC2)C)cc2cccc(Cl)c2o1 N1(C(CCC)=O)CCCCC1C(=O)N(C)CC(c1scnc1C)N1CCOCC1 Cc1nc(C(C)C)nc(O)c1C(=O)NCC1C2CN(C(=O)CCNC(N)=O)CC12 C12(C(=O)NC3CC(N(CC)CC)C3)CC(CN1C(=O)C=Cc1nccs1)C2 N1(C(c2cn(CCC)nc2C)=O)CCCN(C(C2CCCCO2)=O)C(CO)C1 c1(C(=O)NCC2CN(C(CN(CC)CC)=O)C2)ccc(OC(F)F)cn1 Cc1cncc(C)c1C(=O)NCC(C)(C(C)C)NC(C1CC2CCC1CC2)=O C1(F)(CC)CCN(C(=O)C(n2cc(-c3nn(C)cc3C)nn2)C)C1 N1(C(C(C)=C2CCC2)=O)CCC(CCC(=O)N(C2(CCO)CC2)C)C1 c1(CC(C(=O)OC)n2cc(-c3ccn(C(C)C)n3)nn2)ccc(C)c(C)c1 c1(OCC(=O)NCC(CO)SC)ccccc1O.Cc1nc(CC(=O)O)cs1 CCCC(CCCNC(c1oncc1CC)=O)NC(=O)COCCSC.CC C=C1CCC(C(=O)NCCC2CCN(C(C3CC(OC(C)(C)C)C3)=O)C2)CC1 C1(NC(CSC(C)C)=O)COC2(CCN(C(C3(C#N)CC3(C)C)=O)CC2)C1 CCC(C)CCCCC(=O)NC1C(C)(C)C(NC(c2ocnc2C)=O)C1(C)C c1(C(=O)NCCCC(C)NC(C2(CC)CCCCO2)=O)nccc(C)c1F N1(C(c2c(C)ncnc2)=O)CC2(NC(c3cccn3C)=O)CCC1CC2 Cc1ccc2sc(C(=O)NC(C)CNC(c3ccc([N+](=O)[O-])cc3Cl)=O)cc2c1 N1(C(CN(C(=O)OC)C)=O)C(C(=O)N(CC(O)C2CCC2)C)CCC12CC2 C1(NC(c2c(SC)scc2)=O)CCCCC1NC(c1[nH]c(C)nc1C)=O O=C(CCCCCNC(C1(F)CC2(CCC2)C1)=O)NCCOc1ccc(F)cc1 Cc1csc2ncnc(N3CCC(C)C3CNC(=O)CCCc3ccsc3)c12 N1(C(C(C)OCC)=O)CCCC(N(C(=O)Cc2ccccc2Cl)C)C1 CC(C)CC(C(=O)NCCC(C)C(C)C)ONC(C1COC(=O)N1)=O C12(NC(C(C)(C)NC(CC3CCCC(C)C3)=O)=O)CCCN(CCC1)C2 CC(CCN1CCC(C)C1)C(=O)OC1CCCCC1 C12(CNC(CC3N(CC)CCC3)=O)CCC1CN(C(=O)Cc1c[nH]nc1O)C2 c1(C(=O)NCC2CCN2C(=O)Cn2cnnn2)cncc(C(F)(F)F)c1 C1(NC(C(Cn2ccnn2)NC(Cn2nnc(C)n2)=O)=O)CCN(C)CC1 c1(C(=O)NC(C(=O)NCC2N(C(C)=O)CCCC2)CCSC)cc2ccsc2s1 c1(CC)cc(N2CCC(CF)C2)nc(CCNC(=O)C(C)C(C)CC)n1 c1(COC)noc(COCC(C)CNC(c2cnn(CCN(C)C)c2)=O)n1 c1(SCCC(N2CCCC(N(C(C(CSC)O)=O)C)C2)=O)ncnc2[nH]cnc12 Cn1cccc(C(=O)NCC2(C(N3CCOC(CCF)C3)=O)CC2)c1=O C=C(Cl)CCC(=O)N1CCCC1(CC(C)C)C(=O)NC1CCN(CC)C1=O C(=O)(CCCCCC(C)O)NC1C(CNC(c2ccc(CC)cn2)=O)COC1 N1(C(C)C)CCC(C(=O)NC(C)(CNC(C2CC2F)=O)CO)CC1 CC(C)C(C)C(=O)N1CCC(CNC(C2CCCC(CF)C2)=O)CC1 CCC(C)(CC(=O)NCCN(CC(C)O)C(c1cccc(COC)c1)=O)C(=O)OC N1(C(CC2C(C)C2)=O)CCCC12CCN(C(c1cc3c(s1)CC(C)(C)C3)=O)C2 C(c1ccc([N+](=O)[O-])cc1)=CC(=O)NC1C(C(=O)OC)OCC1 C1C(C(C)(C)C)SCC(=O)N1.CCC(C(=O)NCc1ccncc1)c1ccccc1 c1(OC)cccc(NC(=O)CCN(CC2CC2)CC2CCCO2)c1 N1(C(C=C(C)C)=O)CC(C)CN(C(c2ccnc(O)c2Br)=O)C(C)C1 CC(CNC(=O)C(C)(C)S(=O)(=O)C1CC1)(CC1CCC1)N=c1cc(Cl)c(O)n[nH]1 O=C1CC2(CCN(C(=O)C(c3cccc(Oc4ccccn4)c3)(F)F)C2)CN1 c1(NCC2(COC)CC2)cc(Br)ccc1S(=O)(=O)NCc1cc(CN(C)C)on1 Cc1noc(C(F)(F)F)c1C(=O)NC1CN(C(=O)C#CC2CC2)CC1F c1(C(N2CCC(N(CCC)C(C3CC3CF)=O)C2)=O)ccc2cn(CC)nc2c1 CCC(O)C(F)(F)C(=O)NC(C1CN(C(c2cc(=O)n(C)cn2)=O)C1)C CCC(CCC(=O)NC(c1ccncc1F)C)NC(=O)C=Cc1ccncc1 CC#CCCC(=O)NC1(CCNC(=O)CCCCC2CCCCC2)CCC1 C(=O)(C(C)(C)C(=O)NC1CCC(C(N2CCC2(C)CC)=O)C1)OCC CCC(C)(CNC(=O)CCC1CCCN1C(=O)C(C)N1CCCC1)CO C1(C(N2CCC(N(c3ccc(C#N)nc3)C)C2)=O)CCc2cncn2C1 N1(C(C(CC(C)C)F)=O)CCC2OCCN(C(=O)CCC(=O)c3ccc[nH]3)C2C1 c1(-c2cn(Cc3ccc(N4C(=O)NCC4)cc3)nn2)ccc2nccnc2c1 C1(C(N2CCC(N(C(Cc3ccc(OC)cc3)=O)C)C2)=O)Cc2ccccc2C1 c1(C(=O)NCC(CCNC(C(C)(C)OC)=O)O)[nH]cc2c(=O)n(C)ccc12 C1(NC(C2CCN(C)CC2)=O)CC(F)(F)CC1NC(c1ccccn1)=O c1(N2CC(NC(CN3CCC(C)C3)=O)(CO)C2)ncc([N+](=O)[O-])cc1Br N1(C(c2ccc(OC)c(Cl)c2)C(=O)NCC)Cc2[nH]nc(Cc3ccccc3)c2C1 c1(C(=O)NCCCCCN(C(c2c(CC)ccs2)=O)C)cc(OC)cc(C)n1 C=CCC(CC(C)C)C(=O)N(C1CCN(C(c2nn(C(F)F)cc2Cl)=O)C1)C c1(N2CCC2)ccccc1[N+](=O)[O-].C1(C)(CN(C)C(C2CC2)=O)CCCCCC1 CC1CCCN(C(=O)CCn2ccnn2)C1CNC(=O)CCN1CCN(C)CC1 C1(C(F)(F)F)(C(=O)NC(C=Cc2c(C)nccc2)C2CCC2)CC2CCC1CC2 CCC(C)C(O)C(C)C(=O)N1CCC(OCCNC(=O)CCc2csnn2)C1 Cc1cc(C(=O)NCCC2(O)CN(C(c3cn(C)nc3Cl)=O)C2)cc(C)c1F C1(C(N2CC(CNC(C(C)(C)CO)=O)C3C2C3)=O)CC12C1CC3CC(C1)CC2C3 c1(-n2ccc(C(=O)NC3CC(N(C(C=CC(CC)C)=O)C)C3)n2)ccccc1C C1(OC)CN(C(=O)COCC2CC2)CC1NC(C1CCCCCS1)=O C1(N(C(c2c(COC)scc2)=O)C)CCCN(C(=O)Cc2cccnc2OC)C1 c1(C(=O)NCC(C)CNC(=O)C(C(C)(C)C)n2ccnn2)ccc([N+](=O)[O-])cc1 C1(F)(CNC(C(C)Cc2cccnc2)=O)CCCN(C(=O)CCC(N)=O)C1 N1(C(c2ccn(C(C)C)n2)=O)CC(C(=O)NC2CCCSC2)C(C)(C)C1 Cc1nc(Cl)ccc1C(N1CC(O)CC1C(=O)Nc1cnc(Cl)c(Cl)c1)=O CC1CCN(C(c2nonc2N)=O)CCN1C(=O)CC1CCCC1C Cc1ncn(C)c(=O)c1C(N1CC(NC(C2(C#N)CC3(CCC3)C2)=O)C(C)C1)=O C1(OC)CC2(C1)CC(C(=O)NCC(CO)NC(=O)CC1CCC(F)(F)CC1)C2 C=C(C)C(C)(C)C(=O)NC1CN(C(c2coc(C3CCCC3)n2)=O)CCC1CO N1(C(CC(CC)(C)C)=O)CCCN(C(C2(c3cccc(Cl)n3)CC2)=O)CC1C N1(c2nccc(=NCc3ccc(Cl)c(Br)c3)[nH]2)CCc2ncncc2C1 C(c1c(Cl)cccc1Cl)=CC(=O)N(CC(C)(C)NC(c1c(C)snc1)=O)C c1(OC)c(C(=O)NCCC2CCCN2C(=O)Cc2nonc2C)cc(Cl)cc1C Cc1nsc(N2CCC(O)(C(C)NC(=O)CS(N)(=O)=O)CC2)c1C#N CCCCC(O)C(=O)NCC1(NC(C2CCN(C)C2)=O)CCCCC1 CC1CC(CNC(=O)CC2CC=CC2)CN1C(=O)Cc1cccc(O)c1 N1(C(CC(CCC)C)=O)CC(NC(=O)Cn2ncc(Br)n2)CC(C)(C)C1 c1(C(=O)NC2CCN(C(CCSc3ccc(C)cc3)=O)C2)cc(N)c(F)cc1C C1(C(N(CC(C)NC(C=CCC)=O)C)=O)CC(=O)NC(=O)C1 C1(C(=O)N(N2CCOCC2)Cc2ccc[n+]([O-])c2)Cc2ccc(Cl)cc2S1 N1(C(C2(SC)CCC2)=O)CC2(CC(NC(c3ccccn3)=O)c3nccn32)C1 C1(C(N2CCOCC(CNC(C3(C)CCCCC3)=O)C2)=O)CC2C=CCC(C1)C2 c1(C(N2CC(C(C)(C)O)(CNC(CCCCCC)=O)C2)=O)cc2n(n1)CCCO2 c1(CNC(COCC#C)=O)cc(C(=O)NC2(C(N)=O)CC(CO)C2)n[nH]1 c1(CC)nn(C)c(Cl)c1C(=O)NCC(CNC(c1ncccc1Cl)=O)CO Nc1cc(Cl)nnc1C(=O)NC1CS(=O)(=O)CC1NC(=O)Cc1c[nH]nc1O C(CC(=O)NCC(O)CNC(c1cnn(CC(C)C)c1CC)=O)(C(C)C)OCC n1(CCN2CCN(C(C3(CCF)CCC3)=O)CC2)c(=O)oc2cccnc12 CCC(N=c1cc(OC)nc(Cl)[nH]1)C1CCN(C(c2ccccc2[N+](=O)[O-])=O)CC1 c1(C(N2CC(CCNC(C(C(C)C)O)=O)C2)=O)cc2ccnc(Cl)c2s1 C1(CCNC(c2cc(C)ncc2)=O)CN(C(c2scnc2C(F)F)=O)CC(C)O1 c1(C(=O)OC)cc(-c2cn(CC3CCCC(C)C3)nn2)cnc1OC CCCC(C(=O)NC(C)(CNC(c1occ(C)c1C)=O)C(C)C)C(C)C C(=O)(CC1=CSC2=NCCN12)NCC1N(C(CC(=O)N(C)C)=O)CCC1C1CC1 S(=O)(=O)(c1c(C)cccc1Cl)N1CC2(N(C(CC(CCC=C(C)C)C)=O)CC2)C1 N1(C(c2ccc(COCC)o2)C(=O)NC(CC)(C)C)CCn2ncc(C)c2C1 Cc1ccc(N2C3CCC2CC(NC(c2nccnc2N)=O)C3)c([N+](=O)[O-])c1 C1(CC=C)(C(=O)NCC(=O)N2CCCO2)CCN(C(=O)C(F)C(C)C)C1 c1(C(=O)NC2CCC(CNC(CCC#CC)=O)C2)cc(OC)c(S(N)(=O)=O)s1 C1(C(N2C(CN(C(C=NOC)=O)C)CCCC2)=O)OC2CCC1CC2 Cc1cc(C(=O)N(C(C)C(=O)N(C2CC(C)(C)C2)C)C2CC2)cc(F)c1 CC(C)(C)C(C(=O)NCC1CCC(F)(F)C1)NC(C1CC1C1CC1)=O c1(C(N2CCCC(N(C(C(C)NC(N)=O)=O)C)C2)=O)cc2ccccc2s1 CC1CC2(CCO1)CC2C(=O)NC1CCCCN(C(c2ncn(C)n2)=O)C1 C1(C(N(CC(C)NC(C2CC(NC(c3ccco3)=O)C2)=O)C)=O)CCCOC1C c1(C(N2C(CNC(CC3C(C)C3)=O)CC2)=O)cccc(-c2cnn(C)c2)n1 C1(O)(CNC(CC(C)C(F)(F)F)=O)CC2CCC(C1)N2C(=O)C(C)(C)O N1(C(c2ccc(CNC(C=C(C)C)=O)cc2)=O)CCN(C)C(=O)C1C C12(C(N3CC(C#C)(F)C3)=O)CCCC1CCN2C(C1CCC2(CCC2)C1)=O C1(NC(c2nnc3ccccn23)=O)CN(C(c2cc(=O)cc[nH]2)=O)CC2(CC2)C1 c1(C2(C(=O)NC3CCC(NC(C4(SC)CC4)=O)C3)CCC2)ccc2c(c1)OCO2 C1(CNC(CC2N(CC)CCC2)=O)CC2CCC1N(C(=O)CP(C)(C)=O)C2 N1(C(c2cc(C)c(C)o2)=O)CCC2(CCCN2c2nc(Cl)ncc2Br)CC1 CC1CCN(C(=O)CSCc2ccccc2Cl)C(CNC(c2cc[nH]n2)=O)C1 N1(C(c2ccns2)=O)CCC(C2CCN(C(c3cnc(C(F)F)s3)=O)C2)CC1 N1(C(C(C)N(C(CCCOCC)=O)CC)=O)CCC(F)(F)C(C)C1 c1(C(N(CCC(C(C)C)NC(=O)CC(C)CF)C)=O)ccc2c(c1)CN(C)CC2 Cc1sc2ncnc(N3CCCC(C)(CNC(=O)C=Cc4cnc[nH]4)C3)c2c1C N1(CC(=O)N(c2cccc(C)c2)CC)CCOC(C(=O)O)C1(C)C c1(C(=O)NCCN(CCCCCC)C(=O)CC)sccc1C#N.C1(=O)C(C)N1 Cc1ccc(C)c(C(=O)NC2CC(C)(CNC(=O)CC3CCCOC3)C2)c1 N1(C(C(C)OCCC(C)C)=O)CCOC2(C1)CN(C(C1CC1C(F)F)=O)C2 c1(C2C(NC(c3c(Br)n[nH]c3Br)c3n(CC=C)nnn3)C2)ccc(F)cc1 CCCC(C)(CCC)C(=O)NCC(CC(C)C)NC(c1cnn2c1OCC2)=O Cc1cc(C(N2CC=CC2C(=O)NCC2COC(=O)N2)=O)c(C)s1 C1(NC(C(C)OCC#C)=O)C2CC1CN(C(=O)C(N1CCC(C)C1)=O)C2 C1(NC(c2sc(CC)c(CC)c2)=O)CN(C(c2ccc(F)cc2O)=O)CC12CC2 C1(C(=O)NCC2CC(C(=O)NCC3CC(OC)C3)CO2)(CC)CCCCO1 Cc1cnc(C(=O)NCCN(C(c2n[nH]c(C)c2F)=O)C(C)C)c(Br)c1 C=CCCCCCN=c1ccn2ncc(S(=O)(=O)NC(C)CC(N)=O)c2[nH]1 C1(NC(c2nc(Cl)ccc2Cl)=O)(CO)CCCN(C(C2(Br)CC2)=O)C1 C(CO)(C(C)NC(c1cc(CNC(=O)CSCCC(C)C)[nH]n1)=O)SC c1(C(=O)NCc2c(C(=O)NC(CCSC)CO)con2)cnn(C)c1Cl CC1(C)CCOC1CC(=O)NC1CN(C(c2cccnc2SC(F)(F)F)=O)C1 C1(CNC(C2(CC)CCNC2=O)=O)CN(C(C2(C)CCC(=O)N2)=O)CCC1(F)F c1(C(=O)NCCC(=C)CNC(c2nn(CC)nc2C)=O)ccc2c(c1)CNC2=O C1(c2ccccc2)(CNC(C2CN(Cc3cc(I)n(C)n3)C2)C)CCCC(=O)N1 N1(C(CC(C=C)C)=O)CC(CC(=O)NCc2cc(OC)nn2C)CC1(C)C C1(NC(C#C)C(C)(C)OC)CCc2nc(C#N)sc2C1 c1(C(N2CCC(CCNC(C(c3nc(C)sc3)=O)=O)C2)=O)ccc(Cl)nc1C CCCCC(CNC(C1CN(C(=O)CCC2CC2C)CC1C)=O)CCC N1(CC=C)CCN(C(C2(C)C=CCN2C(=O)CC2CCCC3CC23)=O)CC1 c1(OC)ccc(C(=O)CN(C)C(c2cnn(C)c2)C)cc1Cl C1(NC(c2cccc(=O)o2)=O)CCC2(CC1)CC(NC(=O)C(O)CC1CC1)C2 c1(C(N(CC(C)NC(=O)C(C)OCCN(C)C)C)=O)cnc(C(C)(C)C)o1 c1(CC)cc(C)c(C(=O)NCCC(C)(C)CNC(=O)CC2(O)CCCCC2)o1 c1(C(=O)NCC(CC)(CC)NC(=O)C(O)C(C)OC)c(Cl)nc2ccccn12 c1(N(C(CN(C)C(C2CC(CC3CC3)C2)=O)=O)C)ccn(C)n1 N1(C(C(C)NC(CCC)=O)=O)CCC2(CC(NC(c3c(C)cccc3Cl)=O)C2)C1 N=c1c(C(=O)NCCC2CCN(C(=O)Cn3ncnn3)C2)c[nH]c2ccccc12 NC(=O)CC(O)C(=O)NC1CC2(C1)CC2C(=O)NCCOc1ncccn1 C1(C(N2CC(CNC(C3(CC#C)CCOCC3)=O)C2)=O)CC12CC(F)(F)C2 N1(C(c2c(Br)cn(CC)n2)C(=O)NC2CCCCC2)CCCSc2cc(C)ccc21 C1(O)(C(N(C)CCNC(C2CCC2C(C)(C)C)=O)=O)CCc2ccccc2C1 N1(C(c2cncc(CC)c2)=O)CC(C(=O)NCC2CC[Si](C)(C)C2)CCC1(C)C c1(C(=O)NCC2N(C(C(CCOC)C)=O)CC2)c(N)cccc1[N+](=O)[O-] Cc1ccc(C(=O)N(c2cc(Cl)ccn2)C)cc1Cl c1(CN(C(=O)C(C)(C)N(C)C)C)ccccc1CNC(=O)C(C1CCCCC1)O c1(C(N2CC(c3c(CNC(c4cn(CC)nc4)=O)nco3)C2)=O)csc(=NC)[nH]1 CCC(C(=O)NCC(C)CNC(c1ccc(C)s1)=O)N(C)C Cc1ccc(OCCC(=O)NCC(C(C)(C)C)NC(c2nn(C)cc2N)=O)cc1 CC(C(=O)N1CCC(CNC(=O)COCC2CCOC2)C1)S(N)(=O)=O N1(C(Cn2c(C)ncc2)=O)CC(NC(c2cc(C(C)C)cc(F)c2)=O)C(C#N)C1 C1(COC)(NC(C2CCC(=O)N2C)=O)CCN(C(C2CC(C)(C)C2)=O)CC1 C(CCCCCNC(c1ccc(Cl)cn1)=O)NC(c1c(COC)ncs1)=O C(c1ccc(F)cc1)=C(C)C(N1CC2CC1(CNC(=O)CC(C)C1CC1)C2)=O C1(C(=O)NC(CC)C(=O)NC(C23CC(CO2)C3)C)CCOC1(C)C N1(C(=O)NC(C)(C)CCCO)CCNC(=O)C(F)(F)C1 N1(C(c2c(CC)c[nH]c2)=O)CC(N(C(=O)CC2CC(C)(C)C2)C)C(F)C1 CC(C(=O)NCC1(NC(C2CC(N(C)C)C2)=O)CC1)N1CCCC1.N(C)C Cc1c(NC(c2ccc(Br)cn2)C)ncnc1N1CCC(C2CC2)C1 N1(C(CC(c2ccc(CC)cc2)C)=O)CCN(C(=O)CCCOC)C2COCC12 CC(CC(=O)N(C)CC1(O)CCN(C(=O)CN2CCOC2=O)CC1)P(C)(C)=O C1(O)(CC)CCCN(C(=O)CN2CCC(Cc3cnnn3C)CC2)C1 N1(CCCCCCC(N)=O)CCC2(CC1)NC(=O)N(CC(=O)O)C2=O C=C(C)CC(C(=O)NCC#CC#CCO)NC(=O)CC1CC1(C)C c1(C(N2CC3(CC(NC(C(C)n4cccn4)=O)C3)C2)=O)cc2cccnc2[nH]1 c1(NC(N2C(c3cn(C)nc3)CCC2)=O)ccc2c(c1)OCCO2 C(=O)(C(C)CCC(C)(C)C)NC(CNC(C1CCN(CC(C)C)C1)=O)C C1(NC(C(CC)N(C)C)=O)CC1C1CCCN(C(c2cc(C)n(CC)n2)=O)C1 C(=O)(C1=CS(=O)(=O)CCC1)N1CCCC(O)(CNC(c2[nH]cc(CC)c2)=O)CC1 O=C(CC1=Cc2ccccc2C1)NC1C=CCN(C(=O)Cc2cncnc2)C1 CCCC(CC)C(=O)NCC(C1CCN(C(=O)C(C)(C)c2ccsc2)CC1)(C)O c1(C(C)C)ncncc1C(=O)NC1COCC1NC(c1ccc(CO)cn1)=O CN1CCCC2C1CCN2C(=O)CC1CC2CCC1O2 N#Cc1ccc(C(N2CCC(C3CC3)(CNC(C3(CO)CCC3)=O)C2)=O)c(O)c1 CC(CCC(=O)N1CCC(C)(O)C1)NC(=O)CSC1CC1 C1(NC(c2c(SC)cc(F)cc2)=O)CN(C(=O)Cc2ccno2)C2(CCOC2)C1 c1(C(=O)NCCC2CCN(C(C)=O)C(C)C2)c(F)ccc2[nH]ccc12 CC1(C)OCCC1C(N1CCSCC1C(=O)NC1C=CC(CO)C1)=O c1(C(=O)NC2CC3(CC(NC(C(COC)C)=O)C3)C2)nc(Cl)c(Cl)c(N)c1Cl C1(CC(=O)NCc2cc(C(N)=O)no2)CCN(C(=O)C2=NOCC2)CC1 C1(CC(=O)NC(C2CC(NC(C3(CC=C)CCCC3)=O)C2)C)CC(CC)=NO1 c1(N)cc(F)cc(F)c1.C1(NC(=O)CCOCC2CC2)(CNC(=O)C2CC2)CCOC1 C12(C(=O)NCCCCCNC(C(CC=C)CC)=O)CC(CO)(C1)OC2(C)C c1(C(=O)NCC=C)ccc(C(=O)NCC(C)CN(C(=O)C(C)(C)OC)C)cc1 c1(CC(=O)NC(C(C2CCCCC2)NC(CC)=O)C)ccc([N+](=O)[O-])c(N)c1 c1(C(N(CCCN(C)Cc2nc(C(C)(C)C)n[nH]2)C)=O)cc(Cl)nnc1Cl CC1CCCC(NC(=O)CCCNC(=O)CCn2ccnc2)C1 c1(C(=O)NCC23CC2CN(C(C2CC2C(F)(F)F)=O)C3)ccc2oc(O)nc2c1 C1(NC(C(c2cncn2C)C)=O)CCC(NC(=O)C=CCN2CCCC2)C1 n1(CC)ccc(CNC(=O)CC2CCN(C(=O)C=Cc3ccoc3)C2)n1 C1(NC(C2(C)CC=CCO2)=O)CCN(C(c2scnc2Cl)=O)CC1O c1(C(C(=O)NC)N(C)CC2CC2(C)C)cccc2cncn12 N1(C(C2(CC)CC2)=O)CC2CCCC2(NC(c2onc(OC)c2Br)=O)C1 N1(C(c2c(C)c(=O)cc[nH]2)=O)CC2OCCN(C(=O)C(C)C)C2C1 C1(C(F)(F)F)(C(=O)NCC(C)CNC(=O)C(F)=C2CCCC2)CCOCC1 c1(NC)cncc(C(N2CCCC2C(=O)NCC2C3CCCOC23)=O)c1 C1(C(=O)NC(C)C(CO)NC(c2ccc(N(C)C)nn2)=O)CCC(F)CC1 CC(C)CC(=O)C(=O)NCC1CC(NC(=O)C(F)C(F)(F)F)C1 c1(CC)ncccc1-c1cn(CCCN(C(=O)CCC(C)=O)C2CC2)nn1 N1(C(c2ccnc(C(C)C)n2)=O)CC2CCC(CNC(c3csnc3Cl)=O)(C2)C1 C(=O)(C1=CNS(=O)(=O)N=C1C)NC1CC2CN(C(CCSCCC)=O)C1C2 CCCCC(CNC(c1cc(C)n(CCO)n1)=O)NC(C1CCCO1)=O CCC(C)(C)CC(=O)N1CC(NC(c2cc(NC)nc(Cl)c2)=O)C(C)C1 c1(CC(=O)NCCCC2(NC(C)=O)CC2)ccccc1C(N1CCOCC1)=O C(=O)(C1CCc2ccc(OC)cc21)NC(CCNC(c1n(CC)cnn1)=O)C c1(N2C(NC(c3nc(Cl)c(Cl)cc3Cl)=O)CC(OC)C2)ncc2[nH]ncc2n1 C(CCN=c1ncc(C2CC2)c[nH]1)NC(c1ccc(C)nc1)=O Cc1nn(C)cc1C(O)C(=O)NCCC(C)NC(c1nn[nH]c1C(F)(F)F)=O CCC(COC)C(=O)N1CCC(C)(NC(c2ccoc2Br)=O)C1 C(=O)(CCC(F)F)NC(C)CCCNC(C1(C)CC1C(F)(F)F)=O Cn1nc([N+](=O)[O-])cc1C(=O)NCC1(C)CCC(NC(=O)CSc2nncs2)C1 N1(C(CCCOCC)=O)CCOC2(C1)CN(C(c1cccc(Cl)c1F)=O)C2 N1(C(CCC(N)=O)=O)Cc2ccc(CNC(c3cn[nH]c3)=O)cc2C1 c1(C(N(C(CNC(CSCC#C)=O)C)C)=O)ccc(NS(=O)(=O)CCCC)cc1 Cc1cc(C(=O)NCCCN(C)C(c2cn(C)nc2C2CC2)=O)nnc1O N1(C(c2ncn(C)c2)C(=O)NC2CC2)CCSC2CCCCC12 c1(OCC(=O)NC2CCC(NC(c3cnn(C(F)F)c3Cl)=O)C2)ccc(F)cn1 c1(C(=O)NC2(CC=C)CCN(C(=O)C(C)NS(C)(=O)=O)C2)sc(C#N)cc1C N1(C(C(c2cccnc2)OC)=O)CC(NC(=O)C(O)CC(N)=O)C2(CC2)C1 C1(CC#C)(C(=O)N(C2CCC3CC23)C)CCN(C(C2CC2(C)C(F)F)=O)C1 N1(C(c2c(C)cccn2)=O)CC(C(=O)NC2CC(O)C2C(=O)O)C2(CC2)C1 N1(C(C2C(C)CCCC2)=O)CCCC2(CCN(C(C3CCC(C)(C)OC3)=O)C2)C1 C12(C(N(C)CCOCCc3cccc(Cl)c3)=O)CC3CC(C(=O)N1)C2C3 CC1Cc2ccccc2N(C(=O)C=Cc2ccc(C(C)(C)C)cc2)C1 N1(c2cc(C(N)=O)ncn2)CCC(NC(C2CSCCS2)=O)C2(CCC2)C1 CC1CN(C(=O)CCc2nccn2C)C1C(=O)NCC(C1CCCCC1)O C1(CNC(C2(C)ON=C(C)C2)=O)(CO)CC12CCN(C(c1cocn1)=O)CC2 N1(C(C2CC(NC(C(C)(C)OCC)=O)C(O)C2)=O)CC(C2CCCCC2)C1 N1(C(CC(COC)C)=O)CC=C(C(=O)NC2C=CC(CO)C2)CC1 N1(S(C(C)C)(=O)=O)CCOC2(CCCN(Cc3ncc(Cl)cc3F)C2)C1 CCC(CC(=O)NC(C)C(=O)NCC(C)(F)F)OC C1(C(N2C(C)CN(C(C3(O)CCOCC3)=O)CC2)=O)CC2CSCC(C1)C2 C1(C(=O)NCCC2N(C(COC)=O)CCCC2)CCc2nnc(C(F)F)n2C1 c1(CC(=O)NCCN(C(C2C(OC)CC2)=O)C)cnn(C(C)C)c1 c1(C(C)(C)SC)cn(C(C)C(=O)NC(CCN2CCCC2)=O)nn1 C1(NC(c2n(C=C)nnc2)=O)CN(C(=O)CCN2CCNC(=O)C2)C2(CCC2)C1 Cc1ncc(C(=O)NC(C)CCCNC(C2(C(C)(F)F)CC2)=O)[nH]1 N1(c2c(-c3c(C)cccc3)noc2C)CCS(=N)(=O)C(C)C1 N1(C(c2cc(C)[nH]n2)=O)CCC2(CC1)CN(c1ccnc(S(C)(=O)=O)n1)CCO2 N1(C(C2C(CC)OCC2)=O)CCCC(N(C)C(C2CCOC(C)(CC)C2)=O)CC1 N1(C(Cc2cnc(C)s2)=O)CCC2CCC12CNC(=O)C#CC(C)(C)C c1(C(N2CC3CCN(C(=O)CCC(F)F)C3C2)=O)cc(Cl)c(F)cc1F CCC(C)C(C(=O)N1CCCOC(CNC(c2cc(C)c(C)[nH]2)=O)C1)OC N1(C(c2c(CC)n(C)nn2)=O)CC(NC(=O)CN2CC=CC2)C(C2CC2)C1 c1(OC)cnc(Cl)cc1C(=O)NC(C1(CNC(=O)CCC(F)(F)F)CC1)C CC#CCCC(=O)NC1CCN(CCNC(C23CC2CNC3=O)=O)CC1 CC(O)C(F)(F)C(=O)NCC1CCCCN1C(=O)CCC(C)(C)O CCC(C(=O)N1CCCC1CNC(=O)C(C)=C1CCC1)SC N1(C(CC(C)(C)SC)=O)CC2CC(C1)N2C(C1CC1C(F)F)=O c1(C(N2CCC(C)C(NC(=O)Cc3cncnc3)C2)=O)cc(F)c(O)c(F)c1 c1(C(N(CC(O)CF)CC)=O)ccc(CNC(C2CC(=O)N(C)C2)=O)cn1 Cn1ccc2nc(N(C3CCCCNC3)C(c3cccc(Br)n3)=O)ncc12 C1(C(=O)NC(CC)COCC2CC2)COC2(C1)CN(C(=O)CC(C)=C(C)C)C2 n1(CC)[nH]cnc1=NC(=O)C(=O)N(C(C)CF)C N1(C(c2nc(C)n(C)n2)=O)CC2(CCN(C(C3CCCNC3=O)=O)CC2)CC1C C(=O)(C1=CS(=O)(=O)CCC1)N1C(C)CCC(NC(=O)C=Cc2ccc[nH]2)C1 C1(CC)CC(CC(=O)NCC(C)(C)CNC(=O)CC2(C)CCC2)CCO1 N1(C(c2cc(C)cc(O)n2)=O)C2CCC1CC(C(=O)NC1C3CCOCC13)C2 CCC(C)(CO)C(=O)N1CC2CC2(CNC(=O)COCc2nnc(C)s2)C1 N1(C(CC(C=C)CC)=O)CCCCCC(NC(c2occc2C)=O)C1 c1(CC)cccc(N(C)C)c1.C12CC(C1)NC(=O)C2N(C(C)C(=O)NC1CC1)C N1(C(CSc2ccc(C)cc2)=O)CC2=C(C1)CN(C(=O)C(c1cccn1C)=O)C2 c1(C(N2CCN(C(CC(=O)OC)=O)CC2)=O)ccc(F)c(SC)c1 C1(NC(C2(CCNC(C3CCC(=O)C3)=O)CCC2)=O)CCC2(CCC2)C1 CC1=C(C(=O)NCC2(CNC(=O)C(O)C3CC3)CCC2)Cn2nnnc2N1C c1(CC)noc(C)c1C(=O)NCC1CCCC1NC(=O)C(CC1CC1)OC C(=O)(C1CCCc2nc(C)[nH]c21)NCC(C)(C(C)C)NC(c1cncc(C)c1)=O c1(CN2CCC(C)(C(N3CCS(=O)CC3)=O)C2)cc([N+](=O)[O-])ccc1Br c1(SCC)ccc(C(N2CCCC2C2(c3ccc(COC)cc3)CC2)=O)cn1 CN1Cc2ccc(C(N3CCC(CNC(c4ncc[nH]4)=O)C3(C)C)=O)cc2C1 c1(C(=O)NC(CNC(CN=S(C)(C)=O)=O)C2CC2)scc2c1OCCO2 C1(C(=O)NC2CCCN(C(C3(C(=O)OCC)CC3)=O)CC2)C2CCC3C(C2)CC13 N1(C(c2ccc(Oc3nc(C)cc(SCC)n3)cc2)=O)Cc2cccc(Br)c2C1 Cc1ccn(C(C)C(=O)N(C(C)CN(C(=O)CN(C)C(N)=O)C)C)n1 c1(C2N(C(C3CC(F)(F)C3)C(=O)NCC)CCC2)ccc(C(C)(C)C)cc1 c1(NC(=O)NCC(F)Cl)ncc2nccnc2n1 Cc1cc(C(N2CCOC(C)(CNC(=O)COCCCF)C2)=O)c2n[nH]cc2c1 C1(NC(CCSC)=O)Cc2ccccc2C1NC(c1ccc([N+](=O)[O-])cc1F)=O CCCCCS(=O)(=O)CC(=O)NC1CN(C(C2CCCN2C=O)=O)CC2(CC2)C1 c1(CC)cc(OC)c(OC)cc1C(c1nnnn1C)NC(c1c(C)noc1C)C C1(C(=O)NC(C(O)CO)C2CC2)CC(O)CN1C(=O)CCc1cncnc1 N1(c2ccnc(NC(c3csnn3)C)n2)CCC(C)(C2CC2)C1 C1(NC(=O)Cn2cnnc2O)CCCC2CN(C(c3ccc(Cl)nc3O)=O)CC12 c1(C(N2CCC(CCCNC(C3C4CC5C(C4)C35)=O)CC2)=O)cc2scnc2[nH]1 c1(OC)cccc(C(=O)NC2(Cc3cccc4c3OCC4)CC2)c1[N+](=O)[O-] C1(NC(c2cnn(C)c2F)=O)CC(CNC(=O)COCC2CCC2)C12CCC2 c1(C(=O)NCCCN(C(=O)CC2(C)CC2F)C)cc2cc(Cl)sc2[nH]1 c1(C(=O)NCC(CNC(c2c(CCC)nco2)=O)O)cncc(OC(C)C)c1 N1(C(C=CC(C)C)=O)C2CCCC1CN(C(c1cccc(=S)n1O)=O)CC2 c1(N(C2CC2)CC)ccc(C(N2CCC(F)(CNC(=O)C(C)OC(C)=O)C2)=O)cn1 C(=O)(CC(=O)NCC(C)N(C)C(c1cnn(C2CC2)c1)=O)OC c12ccc(cc1)S(=O)(=O)N2.C1(N(C)CCN)CCN(CC2COC2)CC1.C1C(=O)N1 C(=O)(C1=CCCCN1C(=O)OC(C)(C)C)N1CC(OCC)C(O)CC1 c1(C(=O)NCc2ccc(-c3nn[nH]n3)[nH]2)ccc2occc2c1 C(C1=CCN(C(=O)C(c2ccccn2)O)CC1)NC(C=C(C)Cl)=O C(=O)(C(O)P(C)(C)=O)NC1C2CN(C(c3cc(OC(C)(C)C)ncc3)=O)CC21 c1(CC(=O)NCC2CC(F)(CNC(CN(C)CC)=O)C2)ccc(C)cc1 N1(C(COCCCN(C)C)=O)CC2CC2C1C(=O)NCC1(C)CC(C)=NO1 C1(NC(C2CCCN(C(C(CO)OC)=O)C2)=O)CC12CCOCC2 C1(C(CC)NC2CCN(CC(=O)O)CC2)CCCC(C)(C)C1 C#CC1CCCN(C(C2CCN2C(=O)CN(C)CCOC(C)=O)=O)C1 CC(CNC(=O)CC12CCCC1C2)C(F)C(=O)NC1CN2CCCC1C2 N1(C(COCP(C)(C)=O)=O)CCOCC(NC(=O)C(c2cccnc2)O)C1 C1(C(N2CCCC(C)C2C)=O)(CC)CCN(C(=O)CCC2CCCC2)CC1 Cc1cc(C(=O)NC2CC2NC(c2nocc2C(C)C)=O)sn1 C1(CCC)CC(C(N2CC3C(CNC(c4ccnc(OC)n4)=O)C3C2)=O)CCO1 c1(C(C(=O)NCCOCC)N(C(C)CCC(C)C)C)nn(C)nc1Br c1(CC(=O)NCCN2CCC(NC(C3(F)CCNC3)=O)CC2)c(Cl)cccc1Cl C1(CNC(C2CCCN(CC)C2)=O)CC2(C1)CN(C(=O)COc1ccon1)C2 C12(NC(c3nc(C)sc3C)=O)CCC(C(N3CC(C4CCCCO4)C3)=O)(CC1)C2 CCCC(CCC)C(=O)N1CCCC1CN(C(=O)COCc1nc(C)no1)C C1(C(=O)NCC(CCNC(c2cc(OC)ncc2)=O)O)Cc2cc(Cl)ccc2O1 c1(OC)cccc(Cn2nnnc2C2(NCCC=CBr)CCC3CC23)c1 c1(CC)ccc(F)c(C(=O)NCC2(C)CCN(C(c3nc(C4CC4)cs3)=O)C2)c1 Cn1ncc(C#N)c1C(N1CCC2(NC(=O)Cc3cnc[nH]3)CC2C1)=O N1(C(c2cncc(OCC)c2)=O)CCC2(CC(NC(=O)C(C)(C)S(C)(=O)=O)C2)C1 c1(C(=O)NCC2(NC(c3ccsc3Cl)=O)COC2)nc(Cl)ccc1F c1(NCCN(CC)CC)cc(=NC(C)c2ccc(O)nc2)[nH]c(C)n1 c1(C(N(c2c(-c3nn[nH]n3)ccc(OC)c2)C2CC2)=O)cn2cc(Cl)cnc2n1 N1(C(C2C(CNC(c3ccc(O)nc3)=O)CC2)=O)CCC2CCCC2CC1 N1(CC(N2CC(CC(F)C(=O)NCc3ccc(O)cc3)C2)=O)C(=O)CCCC1=O CC1(C)CC(=O)N(CC(=O)NCC2CCC2NC(C2(C3CCC3)CC2)=O)C1=O c1(C(=O)NC2C(C)(C(=O)OCc3ccccc3)CCC2)cc(Br)cnc1O c1(OCC(C)NC(CC(C)Sc2ccccc2)=O)ccc(Cl)cc1Br C12(CNC(C3(C)ON=C(C)C3)=O)CCC(CNC(=O)C#CC(C)(C)C)(CC1)CO2 CC1CC(NC(=O)CCc2cnn(C)c2)CN1C(c1coc(C(F)(F)F)c1)=O C1(CN(C)C(c2ccncc2F)=O)COCCN1C(=O)CCc1cncc(F)c1 C(CC(=O)NCC1(F)CCOCC1)(C(F)(F)F)NC(C(COC)C)=O C#Cc1ccccc1CC(=O)NC(C)(C)CCN(C(=O)CCCC#CC)C CC(C(=O)NCC1(NC(=O)C(F)=C2CCCC2)CCOC1)C(=O)N1CCOCC1 C1(C(=O)NC2(C)CN(C(c3cc(C(F)(F)F)cnc3O)=O)C2)CC2CC1C1CC21 CC(O)C(C)(C)CN=c1nc(N2CCCC(O)CC2)c2c([nH]1)CSC2 Cc1ccc(Cl)cc1C(N1CC(C)(NC(C2(c3cccnc3)CCCC2)=O)C1)=O C1(NC(c2csc(Cl)c2)=O)CCOCC1NC(C1CC(F)(F)C1)=O c1(CNC(C2C(C)CCCC2)=O)ccc(C#N)cc1F.C12CC(C)(C)CN1C2=O N1(C(CNS(C)(=O)=O)=O)CC2ON=C(CNC(c3ccc(CO)cc3)=O)C2C1 c1(CC(=O)NCC2(O)CN(C(CNC=O)=O)C2)ccc2nc[nH]c2c1 C(=O)(C1c2ccccc2C2CC1C2)NCC1C(CNC(C2(CCC=C)CC2)=O)C1 C(=O)(C1(C)CCCc2ccccc21)N(C1CC2CCCC(C1)N2C(=O)C1CC1)C c1(C(=O)NCCN(C(C)C)C(c2cccc(N)c2F)=O)ccc(F)cc1F C1(NC(CNS(N)(=O)=O)=O)COC2(C1)CN(C(c1cc(CO)on1)=O)C2 C1(NC(=O)NC2(c3cccc(Cl)c3)CCC2)CC2C(C1)C2(F)F c1(C(=O)NC2C(C)CCN(C(c3c(C(C)C)ncs3)=O)C2)n[nH]c2ccccc12 CC1CCN(C(C2CCSC2)=O)CCN1C(c1ccc(CO)c(F)c1)=O C1(NC(C=C(COC)C)=O)CC2C1CCN2C(c1nnn(-c2ccccc2)n1)=O Cc1cc(C(=O)NCC2CCN(C(=O)CCC3CC3(F)F)C(C)C2)cc(N)c1O N1(C(c2c(N)c(Br)ccc2)=O)CCC2CN(Cc3ccccc3)CC12 CC1C2CCCCC2CN1C(C1CC12CCN(C(c1cn(C)ccc1=O)=O)C2)=O C1(C(C)C)(C(=O)NCc2ncccc2F)CCN(C(=O)C(C)N=[N+]=[N-])C1 c1(C(=O)NCCCCNC(CCCc2nc(C)sc2)=O)nccc2c1NCCC2 C(CC1c2ccccc2CCN1C(=O)CSC)NC(C1N(CC)C(=O)CC1)=O C1(C(C)(C)NC(C2CC2(F)F)=O)CCN(C(=O)CCc2ccccc2)C1 c1(C(=O)NC2CN(C(C(=CC3CCCC3)C)=O)C2)ccc(Br)cc1O C1(CNC(CC(C)n2cccn2)=O)CCCC2CN(C(=O)CN(C)C(N)=O)CC12 c1(C(N2CCC(C(=O)NCC3CN(CC)C(=O)O3)(CF)C2)=O)cncc(F)c1C c1(NC(CC)CNC(C2CC23CCSCC3)=O)ncnc2onc(C)c12 CCC(C(=O)NC1CC(NC(c2c(Br)ccc(F)c2F)=O)C1)C(C)(F)F C(=O)(C(CC(C)(C)O)NC(=O)OC(C)(C)C)NC1CCCN(CC)C1 N1(C(c2ccncc2-n2cccn2)=O)CC2CS(=O)(=O)C2C1 c1(C(=O)OC)cc(=NCC2CCCCN(C(=O)CCc3ncccn3)C2)[nH]cn1 c1(CN2CC(=O)N(CCc3nnn(C)n3)C2=O)nc2cc(F)c(F)cc2[nH]1 Cc1ccccc1C(C)C(=O)N(C)CC1COCCN1C(C1CC1(F)F)=O Cc1nncc(CNC(=O)CC2C3CCCC3N2C(=O)CC2(C)CCOC2)c1C C1(C(N(C2CN(C(=O)C(F)=C3CCC3)C2)C)=O)CCC(=O)N2CCCC12 C1(C(=O)NC2CC(O)C2)CN(C(c2ccc(Br)cn2)=O)Cc2cccn2C1 C(=O)(CC(C)(C)NC(C1CC(CF)C1)=O)NCC(COC)(C)O N1(CCn2c(C)cc(C)n2)CCC2(CCCN(C(=O)CCc3ncccn3)C2)C1 Cc1nnn(C)c1C(=O)NCC1CN(C(=O)Cc2cnn(C)c2)CCO1 CC1(C)CCC(=CC(=O)NCC2CN(C(C3(Cl)CC34CCC4)=O)CCO2)CC1 c1(OCCC)ccccc1NCC(O)CN(C(=O)C(C)(C)CNC(=O)C1CC1)C c1(-n2c(-c3nc(OC)ccc3Cl)nc(CCCCC)n2)cc(Cl)ccc1OC c1(C(=O)NCC2(C)OCCN(C(Cc3cn(C)nc3)=O)C2)cnc2[nH]nnc2c1 CC1=C(C(=O)NCC2CCCN(C(=O)CCc3ccoc3)C2)CCCC1 c1(C(=O)NCCCC(C)NC(c2c(OC)n[nH]c2)=O)nn(C)nc1C C1(C(=O)OCC)(CO)CN(N2CC(CO)C(C)(COC)C2)C1 C1(C(=O)NCCC#C)CCC2(CN(C(c3cc(F)c(Cl)cc3C)=O)C2)O1 c1(C(=O)NC2C(CNC(Cc3cc(C)ns3)=O)C2)c(C)cc[nH]c1=N CC(C)(C)C#CC(=O)N1CC(CNC(c2ccc(NC3CC3)nc2)=O)C(O)C1 C(=O)(C1=CC2C=CC(C1)C2)N1CC(CC(C)NC(C(C(CC)C)NC=O)=O)C1 N1(C(C2CCOCC2)=O)CC2CCN(C(c3cc(C4CC4)ccc3F)=O)C2C1 N1(C(=O)OC(C)(C)C)CCCC12CCCN(c1ccc(=N)[nH]n1)C2 Cc1cc(C#N)ccc1NC(c1cnn(-c2ccccn2)c1C)=O N#Cc1cc(C(=O)NCC2CCN(C(c3cc(F)c[nH]3)=O)CC2)ccc1[N+](=O)[O-] c1(C(=O)NCC2CN(C(CC=CCC)=O)C(C)C2)cn(C)c2ncccc12 c1(C(=O)NC(CNC(Cc2ccc(OCC)cn2)=O)C)cc2ncccc2o1 CC1(c2cn(-c3ccccc3Cl)nn2)CCN(C(c2cnc(C(=O)O)[nH]2)=O)CC1 C1(C(C)C)C(C(=O)NCCC2CCC(C)(C)C2)CCN1C(c1ncccn1)=O Cc1nc(N2CC(CN(C(=O)C(=O)N(C)C)C)C2)c(C)c(C)n1 c1(C(=O)NNC2CC(CCNC(C(C)N3CCC3)=O)C2)c[nH]nc1C(F)(F)F c1(C(N2CC3N(C(C(=O)OCC)=O)C(CC3)C2)=O)c(C)nc2ccc(OC)nn12 c1(CC2(CC)CN(C(=O)NC(c3ccc(Cl)cc3)C(C)C)C2)ccccc1OC N1(C(c2oc(C)c(Br)c2)=O)C2CCC1CC(CNC(C1CC1(C)C)=O)C2 C1(CNC(C2C=CC(NC(C3CC(N(C)C)C3)=O)C2)=O)CCC(O)CC1 Cc1nc(Cl)[nH]c(=NCC2CN(C(=O)COCC3CCOC3)CCCO2)c1F C1(C(N2CCC(CNC(=O)CC3OCCO3)C2)=O)(OC)CC(CF)C1 c1(Oc2c(OC)cccc2)nccc(=NC(C)C2CCC(F)(F)CC2)[nH]1 c1(C(C)(C)C)cc(C(=O)NCCC2(NC(C3(C)CCCO3)=O)CC2)no1 N1(C(c2nc(OCC)sn2)=O)CCC(N(C(C2(C(C)(F)F)CCC2)=O)CC)CC1 C=CCC(CNC(c1ccc(OC)nc1)=O)C(=O)NCCCN1CC=CC1 C1(NC(c2cnnc(O)c2)=O)COC2(C1)CN(C(=O)Cc1cscn1)C2 C12(CNC(C(CC=C)(F)F)=O)CCCCC1CN(C(c1cc(OC)nn1C)=O)C2 C1(NC(c2c(CC)ocn2)=O)CN(C(C2(C)COC(=O)C2)=O)Cc2ccnn2C1 c1(C(N2CCCCC2)=O)ccnc(Br)c1.c1(N)ccc(-c2ccc(F)cc2)nn1 c1(CC(=O)NC2CC2CNC(c2nc(Cl)cs2)=O)coc(-c2cccs2)n1 C(=O)(C(F)C(C)(C)O)N1CC2C(CNC(c3c(C)oc(C4CC4)n3)=O)(C2)C1 c1(C(N2C(CNC(CCCNC(C)=O)=O)CCC2)=O)cccc2c1NCC(C)C2 Cc1nc(O)sc1C(=O)N(C1CN(C(=O)C(C)C(C)C)C1)C C(=O)(C1Cc2ccccc21)NCC(C(=O)NCC1(CC(=O)OC)CC1)O C1(C(N(CCOC)CC)=O)CCCCCN1C(c1cnncc1OC)=O C12CCN(C1(C)C)c1nnnn1C2.C1(C(C)C)CC(NC(=O)OC(C)(C)C)CO1 N1(C(C2(CC)CCCN2C(c2cncc(Cl)c2)=O)=O)CCCC2(CC2)C1 c1(C(=O)NC(CSC)(C)C(=O)N(C)CCOCCCO)ccc(C)c(O)c1 C1(CNC(C(C=C=C)C)=O)CN(C(c2ccn(C(F)F)n2)=O)CCC1(F)F C1(NC(=O)C=Cc2ncc[nH]2)CC2CCC(C1)N2C(c1ccc(F)c(Cl)c1)=O N1(C(C2CC(=C)C2)=O)CCC(N=c2cc(C)[nH]c(C(=O)OC)n2)C(C)C1 C(=O)(Nn1ccccc1=O)C1(NC(C2CC(C)OC2C)=O)CCC1 CC(O)CCC(=O)N1CC(O)CC1CNC(=O)Cc1cc[nH]n1 c1(C(C)C)cc(C(=O)NC23CCCN(C(=O)CC#N)C2C3)c2ccccc2n1 N1(C(CNC(CC)CC)=O)CCCC1CCC(=O)N(C(C)COC)C N=c1[nH]cnc2cc(C(=O)NC3CC(NC(C4C5CC(F)(F)CC45)=O)C3)ccc12 c1(C(=O)NC2CC3CN(C(C#CC(C)(C)O)=O)C2C3)ccc2c(c1)CCCS2 N1(C(CC(C)F)=O)C2CCC1CC(CNC(c1ccc(Cl)cc1C(F)F)=O)C2 C1(NC(=O)C(N2CCC3(CC3)C2)=O)COC2(CCCC2)C1 C(CCC(O)C(=O)NC1CCC(F)CC1)NC(c1c(C)noc1)=O C(=O)(C(CO)C(C)(C)C)N1CCC(NC(COCCCCCC)=O)C1 C(C(CNC(=O)Cc1cc(F)cc(F)c1)C(F)(F)F)NC(C1N(CC)CCC1)=O C1(CC)(NC(c2cnc(OC(C)C)cn2)=O)CCCN(C(c2occc2C)=O)C1 CC1(C)CN(C(c2cccc(Br)c2F)=O)CC1NC(c1cc[nH]c1)=O C(=O)(C(C)(C)C(=O)NC1(CNC(C2(OC)CCSC2)=O)CCCCC1)NC CC1(C)CN(C(C2CC3CCC2O3)=O)CC1CNC(c1cc(C(N)=O)ccn1)=O c1(NCCCC(C)C)ncccc1C(=O)N(C)NC(CCC1CC(OC)C1)=O C1(NC(C2(SC)CC2)=O)CCC(C(N2CCC(F)(C(N)=O)C2)=O)CC1 c1(C2(CNC(C)=O)CCC2)ncccc1F.C1(F)(CNC(=O)CC(C)F)CC(C)C1 c1(C(C)NS(=O)(=O)CC2(C)CCCOC2)ccc(Br)nc1F N1(C(=O)C(F)F)CCC2CCN(C(C3(C4CCCO4)CCC3)=O)C2C1 CC(C)(CC(F)C(=O)N1CCC(O)C1)NC(c1ccc(F)s1)=O N1(C(CC2C(C)CCO2)=O)CCC2CN(C(c3cc(Cl)ncc3Cl)=O)CC2CC1 N(C1CCOc2ccc(F)cc21)C(c1cc(CC)on1)c1nnnn1CCSC N1(C(C(C(C)OC)NC(=O)CC2CC2(C)C)=O)CC(=O)N2CCCC2C1 Cc1cc(C(=O)N(C2CCC3CC23)C)c(O)c(C)n1 C1(O)(CCNC(=O)Cc2nc[nH]n2)CCN(C(=O)CC2CC(=O)NC2=O)CC1 N1(C(c2ccn(CCCC)n2)=O)CC(C)N(C(=O)CCN2CCOCC2)CC1C c1(C(N2C(C)CCC(NC(Cc3nc(CC)sc3)=O)C2)=O)cc(Cl)c(OC)cc1C c1(CNC(C2(CC)COC2)=O)ccnc(C(=O)NOC2CCC(O)C2O)c1 N1(C(=O)OCC)CCN(C(c2cc3sc(C(F)(F)F)cc3s2)=O)CCC1C C1(CN2CC(C)(C(=O)Nc3nccc(OC)c3OC)C2)Cc2ccccc2C1 C#CCC(C)C(=O)NCC1CCC(CNC(=O)C(F)(F)C2(O)CCC2)CC1 c1(C(=O)NCC2N(C(CC(CCC)C)=O)CCC2CC)cc2ccccn2c1 c1(OC)ccc2c(c1)N(C(=O)CCC1OCCO1)CCN2C c1(C(=O)NC(C)C(C)(C)NC(=O)C(O)C(F)F)ccc2c(c1)CCCC(=O)N2 c1(OC)ccc2ccccc2c1CN1CCC1C(=O)NC1CSC1 C(C1Cc2ccccc21)NC(=NCCC#C)NCc1cnn(C)n1 C(=O)(C(C)(Cc1ccc(Cl)cc1)NC(=O)C(c1cccc(C)c1)=O)OC N1(CCNC(c2c(C)snc2)=O)CCC(NC(c2cncc(N)n2)=O)CC1 CCCCC(C)C(=O)NC(C1CCCN(C(=O)CNc2ccccc2)C1)C C(=O)(C1COc2ccc(Cl)cc21)NC1CCC(CNC(=O)CC2CCNC2=O)C1 Cc1[nH]nc2c(C(N3CCCC(NC(=O)C(C)N4CC(C)C4)C3C)=O)cccc12 C1(COCC)CC(N=c2[nH]c(N3CCC(C#N)C3)nc3c2CSC3)C1 C1(C(=O)NC(CC(C)C)C(=O)NC)(NC(C(C=C)CC)=O)CCC(C)(C)C1 N1(C(C23N(C(=O)OC(C)(C)C)C(CC2)CC3)=O)CC(C2CCCCC2)C1 c1(N2C3CC(=O)NCC2CC3)nc(=NCCc2ncccc2F)[nH]c2c1COC2 C=CCC(C)(CNC(=O)C(C1(C)CC1)NC(=O)CNC=O)CO N1(C(CCc2cc(C)on2)=O)CCC(N(CC(C)C)C(C2CC2C)=O)CC1 N1(CCC)CCCC(C(=O)NCC2CC(F)CN2C(c2cn(C3CC3)nn2)=O)C1 C(=O)(CC(C)CN(C)C)N(CCOC)CCNC(C1(C)CC1C(F)(F)F)=O N1(C(COCCOCC)=O)CC(N(C)C(C2CC3CCC2CC3)=O)C(C)(C)C1 C1(C(N2CC(CNC(CN(CCCCCC)C)=O)C2)=O)CC(C(C)=NO)C1(C)C C1(C)(CNC(c2c[nH]c(=NC)s2)=O)CN(C(C2(C)C=CCCC2)=O)CC1C Cc1nc(NC2C(C)CCC(C)(C)C2)c2cc(C)sc2n1 C1(NC(c2ccc(SC)s2)=O)(CO)CCN(C(c2nc(C)ccc2C)=O)CC1 c1(C(N2C(=O)NC(CC(C)C)C2=O)C)ccccc1[N+](=O)[O-] c1(C(=O)NCCCN(C(=O)Cc2ccc(C)cc2)CC)nn(C(C)(C)C)cc1Cl c1(C(=O)NC2CN(C(C3(CO)CC3(F)F)=O)CC2O)cc(F)c(F)cc1Cl C1(NC(c2ccccc2Cl)c2n(CCC)nnn2)CCCCC12CC2 N1(C(CNC(c2ccccc2CO)=O)=O)CCCC2(C1)CN(Cc1cc[nH]c1)C2 c1(C(=O)NC2CC2CN(C(C(=O)NCCCOC)=O)C)cc(Cl)c(OC)c(Cl)n1 c1(C(N2CCC(N(C(=O)CC=CC(C)(C)C)C)CC2)=O)cc(F)c(CO)c(F)c1 N1(C(c2sc(C)c(O)n2)=O)CC(NC(=O)C(O)C2CCCC2)C2CCCC12 N1(C(c2cccc(CC=C)c2)=O)CC2CCN(C(c3cc(C)c(Cl)s3)=O)C2C1 Cn1cc2c(n1)CCCC2C(=O)NCC1(C)CCN(C(c2ncc(F)cn2)=O)C1 C1C(F)(C(C)C)C(=O)OCC(C)C(=O)N1.C(C)(C)(CC(=O)OCC)NCC c1(C(N(CC(CO)(CO)NC(Cc2c(C)non2)=O)C)=O)cccc2ncsc12 N1(C(C2CCNC(=O)C2)=O)CCCCCCC1CNC(c1nc(C(C)C)oc1)=O N1(C(c2c(OC)scc2)=O)CCCC(C2(NC(C3COC4COCC34)=O)CC2)C1 C1(CC)CCCCCCN1C(=O)C(C)NC(C1CC(=O)C12CCC2)=O N1(C(CCC#CC)=O)CCCOC(CNC(=O)C(F)C2CCC2)C1 N1(C(CCCOCCC)=O)CC(C(F)(F)F)CC1CNC(=O)C(CC)SC C1(CC(=O)N(C2CCN(C(c3cnc(Cl)s3)=O)CC2)CCC)CCCS1(=O)=O C(=O)(C(CC)CC=C)NC(CC#C)C(=O)NC(C)CCCCC CCC(C(C)C)NC(=O)C#CCNC(c1cnc(C)o1)=O C1(N(CCOC)C(C2(C)CC2C(=O)O)=O)CCNCC1 C1(C(N)=O)CCCCN1C(=O)COC(C1CCN(c2cccc(F)c2)C1=O)=O C(=O)(C1=C(C)CCOC1)NCCCN(C(CCC(=C)C)=O)C CCCCCC(C)(C)C(=O)N(CC(=O)NC(c1cnn(C)c1)CO)C1CC1 CCC(CC(=O)NCC(CNC(=O)Cn1cc(Cl)c(C)n1)S(C)(=O)=O)C(C)(C)C c1(C(N2C(C(=O)N(CC(CC3CC3)CO)CCO)CC2)=O)ccnnc1O Cc1ccc(C(=O)N(CC(C)(C)CNC(C2CS(=O)(=O)C2)=O)C)cc1Cl C(CCCCNC(C1CN(CC(C)C)C1)=O)N(C(C(C)SC)=O)C c1(C(=O)NC(CCNC(c2nn(C)c(Cl)c2)=O)(C)C)ccc(O)c(Cl)n1 N1(C(C2(COC)COC2)=O)CCC(C)C(NC(c2ccncc2C(F)F)=O)C1 C1(CC(=O)NCC(F)(F)F)(OC)CN(C(C2(c3ccccn3)CC2)=O)C1 C12(C(C(F)(F)F)NC(=O)CCO)CC3CC(CC(C3)C1)C2.C1(C=O)CC1O c1(C2(C(=O)Nc3nccc(CN)c3)CCCC2)cccc(F)c1F Cc1cc(NC(=O)C2CC2)ncc1-c1nc(C2CCC3CC3CC2)no1 N1(C(CCSC)=O)CC2CC2C1C(=O)N(C)CCN(C)C(C)=O c1(C(=O)NC(CCCNC(c2c(C)cco2)=O)C)cnc(CC2CC2)nc1O c1(C(=O)NC(CCOC)CNC(=O)CC(C)C2CC2)c(C)cccc1O N1(C(=O)NC(c2ncc(C)[nH]2)C(C)(C)C)CCOc2ncccc2C1 c1(C(=O)OC)cc(I)c(Cl)cc1NC(C1CCN1C(c1sc(Br)nc1C)=O)=O Cc1ccc(C)c(OCC(N2CC(CC(=O)O)CC2C)=O)c1 C1(NC(c2cccnn2)=O)CN(C(c2snc(O)c2Cl)=O)CC2(CC2)C1 C1(CC)(CC)CCN(N2CCCCCN(C)C2C)CC1.c1(O)ccccc1 c1(OC)ccccc1C1CNCCN1Cc1noc(-c2ccccc2)n1 c1(CNC(c2ccncc2-c2ccc(C(F)(F)F)cc2F)=O)cccc(Cl)c1Cl c1(NC(=O)NC23CCC(C(=O)OC)(OC2)C3)cc(Cl)cc(F)c1F C1(OC)CCC2(C(=O)NC(C)C(C)C(=O)NCc3ccc(CO)o3)CC12 C(CCCCC(=O)NCc1c[nH]nc1C(=O)NC1COCCC1(F)F)OCC CC1OCCC1CC(=O)NCc1cc(C(=O)NCC(c2ccncc2)O)co1 c1(NCc2c(CC)nns2)ccc2ccccc2c1 C1(NC(CCCSC)=O)CCC2(CC1)CC(NC(c1cc(C)c(=O)n(C)c1)=O)C2 N1(C(c2ccccc2)CCOC)CC2CC1CN2C(C1CCOC(C)(C)C1)=O c1(-n2cc(C(COC)(C)O)nn2)cc(Cl)cc(Cl)c1.C1(C(C)=O)CCCO1 N1(C(CCCNC(N)=O)=O)C2CCC1CN(C(C1CSCC1c1ccccc1)=O)C2 C1(CNC(CCCN(C(C(C)CC2CC2)=O)C)=O)CCCOC1(C)C n1(CC(=O)NCCC2CN(C(=O)COC(F)F)C2)cnc(Br)c1 C1(NC(c2ccc(CC)o2)=O)CC12CCN(C(=O)CSCc1cccs1)CC2 C#CCCCCC(=O)N1CC(NC(=O)CCc2nnc(-c3ccsc3)o2)CC1C CCCC(C(=O)NC(C1(O)CN(C(=O)Cc2nc(C3CC3)cs2)C1)C)N(C)C C=C1CCN(C(=O)C(N2CCCCC2)C)C(C(=O)NCCc2c[nH]nc2C)C1 C1(NC(C(CC)Oc2ccccc2Cl)=O)CCN(C(=O)CO)CC1(F)F CC1(F)CCN(C(C2CC(CNC(C3CC34CCOCC4)=O)C2)=O)CC1 c1(NC(c2n(C(CC)(C)C)nnn2)C(C2CC2)OC)ccc2nccn2c1 n1(CC2CC(OCCC(=O)NCCOC)C2)cc(C(=O)Cn2cc(C)cn2)nn1 C1(CNC(CSCC#N)=O)CC2CN(C(=O)C(C3CCOCC3)F)CC12 O=C(C1=CCSC1)NCC1(C(=O)NCc2nn[nH]c2C2CC2)CCCO1 c1(C2(C(=O)NC3C(NC(=O)C=C(Cl)Cl)CC3)CC2)nccc2ccccc12 c1(C(N2CCC23CN(Cc2c(F)cc(Cl)cc2Br)C3)=O)cccc2c[nH]nc12 N1(C(C2C(C)(CC)C2)=O)CCCC(NC(=O)CNS(N)(=O)=O)C1CC CCCCC(O)C(=O)NC1C2CC1N(C(C1CCN(C3CCSC3)CC1)=O)C2 c1(C(=O)NC(C2CCN(C(CSC)=O)C2)(C)C)cc(C(=O)OC)oc1C CCCC(O)C(=O)N1CCC(CNC(c2ccc(-c3nnc(O)o3)cc2)=O)C1 CC1OC2(C(=O)NC3CN(C(=O)Cc4cnccn4)CC3C)CCC1CC2 C(CC(C)(C)CC(=O)NCc1cnc(OC)cn1)OC c1(C(=O)NCCN(C(C2C(C)(C(=O)OC)C2)=O)CC2CC2)ccc(OC)c(OC)c1 CCCCCCC(CC)C(=O)NCC1CCN1C(C12CCC(CC1)C(C)O2)=O C1(NC(CC(C)SC)=O)CCN(C(c2cc(N)cnc2Cl)=O)CC1F C1(OC)CC(CNC(=O)C=CC2CC2)N(C(c2cccc(C(=O)NC3CC3)c2)=O)C1 C1(OC)CCN(C(C2(F)CCN(C(c3cncc(C)n3)=O)C2)=O)C12CCC2 c1(CNC(C2CSCN2C(=O)CC2CCCC2)=O)ccncc1Cl C=CCCCC(C)(C)C(=O)N1CC2=C(C1)CN(C(C1SCCS1)=O)C2 CC1=C(C(=O)NCC2CC(C)CN(C(=O)CCC3CCCO3)C2)CCC1 C1(CC=C)(C(=O)NCC(=O)NOC)CCCN1C(=O)CCC1CCCCO1 c1(C(=O)OC)c(Cl)nc[nH]c1=NCC1(NC(c2cnnn2C(C)C)=O)CCCC1 c1(C(=O)NC(CC)CNC(=O)C=C(C)C(F)F)cc(OC)c(Cl)cc1Cl CCC(C)(COC)C(=O)NCC1CC(O)CN1C(=O)CCc1cocn1 c1(NC(C2(C(F)F)CCCO2)=O)cccc2c1OCCC2 C1(NC(=O)CCCc2cccs2)CN(C(c2cnns2)=O)CCC1CO c1(C(=O)NCCCC(C)NC(=O)C(C)NC(N)=O)cncc(F)c1 c1(OCC)nc(C(=O)NCCNC(=O)CC2CCC3CC23)co1 CC1CC(C(=O)NCC2CCN(C(c3cnn(CCF)c3)=O)CC2O)CC(=O)N1 C12N(CC1(C)C)C(=O)CC1CCN1C2.c1(C(=O)OC)csnc1OC N1(C(C(CC)(C)OC)=O)CCC(NC(c2ccnc(F)c2O)=O)C(C)(C)C1 c12cc(ccc1C#N)S(=O)(=O)N2.CC1CSCCN(NC2CCSC2(C)C)C1 c1(C(N(CC(CN(C)C)O)C)=O)cccc(OC2CC2)n1.C12(CCCO1)C(=O)N2 C(CC)(CC(C)CO)NC(CC1(C=C)CN(C(=O)Cn2cc(CO)nn2)C1)=O N1(C(CC=C=C)=O)CC2CCN(C(c3scnc3C(C)C)=O)CCC2C1 N1(C(CN(C(C)C)C(C2Cc3nccn3C2)=O)=O)CCC(F)C(O)C1 CC(C(=O)O)C(C)N1CC(Cn2ccc(C(F)(F)F)n2)S(=O)(=O)C(C)C1 c1(C(N2CC(C(=O)Nc3cc(C)c(F)cc3)CC2(C)C)=O)cc2cccnn2c1 N1(C(c2nc(C)sc2C)=O)CCn2nc(CNC(=O)C(C)c3ccsc3)cc2C1 C(=O)(C1=CC2(CCN(C(=O)C(C)C(C)COC)C2)C1)NCC1(C#C)CCCC1 CCC(C)CC(=O)C(=O)N1CCC1CC(N1CCCC(C)(C)C1)=O C#CC1CCN(C(C2COC(CNC(=O)C(O)C3CCCC3)C2)=O)C1 N1(C(C=CC(CC)C)=O)CC(C(F)(F)F)CC1CNC(=O)C(c1ccccc1)O C(=O)(CCC(C)(C)F)NC1CCC(C)(CNC(c2c(OCC)ccs2)=O)C1 C#Cc1cnn(CC(N2CCC(C(=O)NC(C)Cc3cccs3)(CF)C2)=O)c1 C(=O)(C(C)(C)C(=O)NCCC1CCN(C(=O)Cc2cnc[nH]2)C1)OC c1(C(=O)NCCCC(C)(C)NC(C2C(=C)CC2)=O)c(C)ccc(Br)c1N c1(OC)ccc(-c2cn(C3CCN(C(C4CC(O)C(F)C4)=O)C3)nn2)cc1Br c1(C(=O)NC(C2CCN(C(=O)Cc3sc(O)nc3O)C2)C)cncc(C2CC2)c1 c1(C(=O)NCCC2CCC(NC(=O)C3=COCCO3)C2)cccc2ccsc12 c1(C(N2CC(NC(=O)OCC)C2)=O)cc(CNC(c2csc(Cl)c2)=O)ccn1 c1(C(N2CC(NC(C3(OC)CC3)=O)C2)=O)ccnc(C)c1Cl C1(CCC)CCCN(C(=O)CCN(C(=O)CC2CCOC2)CC)CC1 c1(C(N2C(C(=O)NC(C#C)C)CC3CC32)=O)cc(Br)c(C)c(Br)c1 NS(=O)(=O)c1ccc(C(O)CNC(C2CC2c2cc(F)ccc2F)=O)cc1 N1(S(CCOCCOC)(=O)=O)CCC2(CC1)CC(=O)Nc1ccccc12 C(CCN(C)C(c1ccc(C)nc1O)=O)(C(C)(C)C)NC(CCC(=C)C)=O c1(C(N2CC(C)N(C(=O)Cc3ccc(O)cc3)CC2)=O)cccc2nsnc12 c1(CNC(C2(SCC)CC2)=O)n[nH]c2c1CN(C(=O)CCC(=O)NC)CC2 Cc1nc(C)c(F)c(=NCC2C(C)CCCN2C(c2scnc2C)=O)[nH]1 C1(CC)CCOCCN1C(C1CC2C(C1)C2(F)F)C(=O)NC C1(CNC(CCCCCC)=O)(NC(=O)CC(C)CN(C)C)CCC(F)(F)CC1 C(CO)(CCCCNC(=O)C=C1CC1)NC(CCOC(C)C)=O CN1CC=C(CC(=O)NC2CCN(C3CCN(C(C4(O)CC4)=O)CC3)C2)CC1 CCC(O)C(F)(F)C(=O)NC1CC2(C1)CC(C(=O)NC1CC(=O)NC(CC)C1)C2 C1(C(=O)N(CCCCNC(=O)CCC2CCCCO2)C)(COC)CC(=O)C1 Cc1cncc(C(=O)NCC2C(C)CCN2C(c2c(Cl)cnn2C(C)C)=O)n1 C#CC1(C(=O)N(CCCN(C)C)C)CCN(C(=O)COC(C)=O)C1 C12(CNC(=O)Cc3csc(Cl)c3)CCC(CC1)N2C(=O)Cc1cn[nH]c1 N1(C(CSCCC(C)C)=O)CCCC1CN(C(C1CC1(F)F)=O)C1CC1 C1(NC(c2cc(C)no2)=O)(CO)CCCN(C(c2ccnnc2O)=O)C1 N1(C(C(C)=CC)=O)CCCC2(NC(c3cccn4nccc34)=O)CC2C1 c1(NC(N(C2CC(CN)C2(C)C)c2n(C(C)C)ncc2)=O)c(Cl)nnc(Cl)c1O C(=O)(C1=NNC(=O)CC1)NCC1CCN(C(C2C3CC(C)(C3)OC2)=O)C1 Cc1ccc(C(N2CC(C(N)=O)(CNC(=O)CC3CC4(CC4)C3)C2)=O)cc1F C(=O)(CC(C)CCC(=O)N1CC=C(CNC(c2cccc(Cl)c2Cl)=O)CC1)OC C#CCCCCCCNC(=O)C(C)CNC(=O)CC1(O)CCOCC1 CC1CCN(C(=O)C=CC(=O)OC(C)(C)C)C1CNC(=O)CC1CCCO1 C1(C(=O)OC)CC(CNCc2cccn2CF)N(S(C)(=O)=O)C1 N1(C(CC#C)=O)CCCCC1CNC(c1cncc(Br)c1)=O c1(NC2C(SC)COC2)ncc(S(=O)(=O)NCc2cccnc2Br)cc1Cl N1(C(C(C)SC(F)(F)F)=O)CC2(CNC(C3(SC4CC4)CC3)=O)CCC1C2 c1(C(=O)NC2CCN(C(c3ccn(C(C)C)n3)=O)C2)n[nH]c2c1CCOC2 C=CCC(CNC(c1cnc(=N)[nH]c1)=O)C(=O)NC(C)(C)CCF c1(C(C)C(=O)NC2CC2NC(=O)CC2=NNC(=O)C2)ccc2ccccc2c1 N1(C(Cc2n(C)ccn2)=O)CC(O)CC1C(=O)NC1CN(C(N)=O)C1 C1(NC(C2(CC=C)CCCCC2)=O)CC(NC(C2(OC)CCCC2)=O)C12CCC2 C1(CNC(C=CCC)=O)CC(NC(c2ccn(CC)n2)=O)C(O)C1 c1(OC)c(C(=O)NCC(CO)NC(c2ccc(C(C)(C)C)[nH]2)=O)cc(Cl)cc1C N1(C(CC2(OC)CC2)=O)CCCC2(C1)CN(C(=O)C(C)N=[N+]=[N-])C2 C=CCC(C)(C(=O)NC1(CNC(c2cc(OC)nc(Cl)c2)=O)CCC1)N(C)C N1(C(CC2N(CC)CCCC2)=O)CCC2CC1CN2C(=O)CC(=O)OC C12(C(=O)NC(CCNC(c3cc(C(C)C)nn3C)=O)(C)C)CSCC1C2(F)F c1(C(=O)NC(CN(C(C(C=C)(F)F)=O)C)C)cncc2ccccc12 c1(CC(=O)Nc2ccc(NC(C3ON=C(C)C3)=O)cc2C)c(C)cc(O)cc1C Cn1cc(C(=O)NC2CCN(C(C3(C#N)CC3)=O)CC2)c(C(C)(C)C)n1 CCC(CCOC)C(=O)NC(C)(C)C(C)NC(=O)CN(C1CCC1)C C1(C(=O)NCCOCCC=C)CC1C1CN(C(C2CC3CC(=O)C2C3)=O)C1 Cc1cccc(NC(C2(NC(C3CC(=O)C3)=O)CCCC2)=O)c1 c1(C(=O)NC2CC(NC(c3cn(CC)nc3C)=O)C2)nn(C)c2c1CCC2 C1(NC(Cc2c(C)ncs2)=O)COCCN(C(=O)CCN2CCOC2=O)C1 N1(C(c2c(C)csc2)=O)CCN(C(c2[nH]c(O)nc2C)=O)C2(CC2)C1 CCC(CC)C(C)C(=O)N1CC2CC2(CNC(C2CC(n3ccnn3)C2)=O)C1 c1(C(N2CCC(OCC(=O)N(CCCCO)CCO)C2)=O)cc(O)nc(O)n1 C12(CNC(C(CC)F)=O)CCCC1N(C(c1ccc(Br)c(F)c1)=O)CC2 C(=O)(C(CC(F)F)NC(c1nccnc1N)=O)NC(C#C)CC(C)C C(=O)(C(CC(=O)OC)N(C)C)NCC1CC(NC(COCC(=C)C)=O)C1(C)C c1(OC)ccc(C(N2CC(CNC(C3CCN3C(C)(C)C)=O)C2)=O)cn1 CC(F)(F)C(C)(C)C(=O)NC1CC2CC(NC(=O)C(CO)NC(N)=O)C1C2 CC(C)CC(C)CN=c1[nH]c(N2CCOC(C(=O)N(C)C)C2)nc2cc[nH]c12 C(CCCCC(=O)NC(C(C)C)C1CCC1)N(C(CC(C)SC)=O)C C1(CNC(c2cnc(C(C)(C)C)[nH]2)=O)CCCN(C(=O)CC2CCNC2=O)C1 CCS(=O)CC(=O)NC1CCCC(NC(c2ccccc2C2CCCC2)=O)C1 N1(C(C2(F)CN(Cc3ccncc3Cl)C2)=O)CCc2nc[nH]c2C1 c1(C(N2C(C)(CNC(c3cc4scnc4[nH]3)=O)CCC2)=O)ccc2c[nH]nc2c1 N1(C(c2ccc(C(=O)OC)[nH]2)=O)CC2CCCN(C(=O)CN(C)C(C)=O)C2C1 c1(C(N2C(CCC)CN(C(C3(CO)CCCC3)=O)CC2)=O)ccc2occc2c1 c1(SC)nc(N2CC3CC3(C(N3CCN(C(C)C#N)CC3)=O)C2)c(Br)c(C)n1 c1(C(=O)NC2C3CN(C(CC4(NC(C)=O)CC4)=O)C2C3)cnc2n1CCC2 C1(CNC(C(CC)OCC)=O)(NC(=O)CCCSC(C)(C)C)CCCCC1C N1(C(c2c(C)c(Cl)ccc2)=O)CCC(NC(=O)CC2CCCCO2)C(CO)CC1 C1(C(N(C2CCN(C(CCc3c(C)nn(C)c3)=O)C2)C)=O)OCCN(C)C1=O c1(CNC(=O)Nc2c(C)nc(Br)cc2)cccn2ccnc12 C1(C(N2CCC3(CCCO3)C2)=O)CCCCCCN1C(C1CC2C=CC1O2)=O C(C(C)(C)C1=CCCC1)NC(CC1CC(C)N(C(=O)CC2=CCCC2)C1)=O C(C)(CO)(C(=O)N(C)CCNC(C1CCC(O)C1)=O)OC c1(C(C(=O)NCc2ccc(F)cc2)N(C(CC)C#N)C)nc(Br)ccc1OC CC1OCCC1(C)C(N1CC(OCCNC(=O)Cc2ccnc(O)c2)C1)=O c1(N2CCN(C(c3c(C(C)C)nns3)=O)CC(O)C2)ncnc2c1SCCC2 N#Cc1cn(CCC(=O)NCCCC2NC(=O)NC2=O)c(=O)nc1O N1(C(c2ccc(I)c(C)c2)C(=O)NCC(=C)C)C2CCC1CN(C)C(=O)C2 C(=O)(CCC(C)S(C)(=O)=O)NCC(C)(C)NC(CC(COC)C)=O Cc1cccc(C)c1-n1cc(C2CCN(C(=O)CC(O)C(C)C)C2)nn1 N#Cc1cc([N+](=O)[O-])cc(Cl)c1NC(C12CC1CN(S(=O)(=O)CCCCCl)C2)=O C12(NC(=O)CCSC(F)(F)F)CCCN(C(=O)Cc3cnoc3)CC1C2 CC1SCCC1N=c1cccc(S(=O)(=O)N2CCC3(CC2)CC(O)C3)[nH]1 CC1CC(O)CCN(C(C2CCCN(C(C3C4CC(=O)CC34)=O)C2)=O)C1 C1(C(N(CC(C)O)CCNC(CCSCC(C)C)=O)=O)CCCC(O)C1 N1(C(C(CC)N(CC)CC)=O)CCC(C2N(C(=O)C(C)CO)CC2(C)C)CC1 CC(c1cnn(C)c1)=CC(=O)NC(C)CNC(c1cn(C)c(C)n1)=O C1(C)(C(=O)NCC2(CCNC(c3c(C)n(C)cn3)=O)CC2)CCC(F)(F)CC1 Cc1cc(CCc2ccc(Br)cc2)ccc1S(=O)(=O)NNC(=O)CN1CCC1 C1(NC(CCCCC)=O)CCCCCN(C(=O)CCc2ccncn2)C1 C1(NC(CCSCCC)=O)CCN(C(c2ccccc2C)=O)C12CCC2 C(=O)(CC(O)CC(C)(C)C)N1CCN(C(CCCc2ccc(C)cc2)=O)CC1C c1(OCC=C)ccccc1C(c1nnnn1C)NC1CC2(CCC2)C1 c1(NCC2CCC(NC(Cc3cc(C)no3)=O)C2)nc2c(cc1C#N)CCOC2 c1(C(=O)NCC2CN(C(CCc3ccc(C)o3)=O)C2)ccc2ncccn12 N1(C(CC(C(=C)C)OCC)=O)Cc2occ(C(=O)NOCC=CCl)c2C1 CCC(C)C(O)C(=O)NCC1(c2ccccc2)CCN(C(C2CC2F)=O)CC1 N1(C(C2C(CC)C2)=O)CCC2(C=C(C(=O)NCc3ccccc3N(C)C)C2)C1 CCC(CCOC)C(=O)NCC1(O)CN(C(c2c(C)c[nH]c2CC(N)=O)=O)C1 CC1(C)CCC(NC(C2COCCC2NC(=O)Cc2cncs2)=O)C1 c1(OC)ccc2cc(NCCN(C(c3cc(C)n(C(C)C)n3)=O)C(C)C)ccc2n1 C1(C(N2CCC(C)(NC(C(C)c3cccs3)=O)C2)=O)CCc2ncnn2C1 C1(C(=O)NCc2n[nH]c(C)c2C)CN(C(=O)C(C2CCCCC2)O)CC(C)(C)C1 c1(NC(=S)N(C)C)cc(C#N)ccc1NC1CCCN(c2ccc(C)cc2)C1 N1(C(c2ccc(=N)[nH]c2Cl)=O)CCC2(CC1)CN(C(C1CCCCC1F)=O)C2 c1(OC)nccc(C(=O)N(CC(C)CNC(=O)CN(C)C(N)=O)C)c1Br c1(CC(=O)NC2CCC(N3CCN(C(C(C)(C)C)=O)CC3)C2)c(F)cccc1Cl C(=O)(C(C)(C)S(C)(=O)=O)NCC(CCOC)NC(C12CCC(CC1)O2)=O Cc1ccc(CNC(c2oc(CNC(=O)COCCCF)nc2C)=O)c(C)c1 c1(C(C)C)cc(C(N2CCC(F)(CNC(=O)C(C)(C)N3CCCC3)C2)=O)nn1C c1(CC)ccc(CN(CCCNC(=O)CCc2c(C)noc2C)C(C)C)cc1 c1(C2C(C(=O)NCC3(CN(C(=O)C(O)C(F)F)C)CC3)C2)ccccc1Cl C1(NC(CNS(N(C)C)(=O)=O)=O)CC2CC1N(C(=O)CC1CN3CCC1CC3)C2 c1(OC)c(C(N2C3CCC2CC(CNC(=O)C(C)C(F)F)C3)=O)nc(O)nc1O C1(C(=O)NC2CC=CCC2C(N2CC(CC(N)=O)C2)=O)(OC)CCC(C)C1 c1(C(N2CCCC(NC(C(C)(F)F)=O)C2)=O)ccc(F)cc1Cl C1(NC(C2C=CCCN2C(=O)C(O)CC2CCCC2)=O)CCCC2(CC1)CC2 CC1(C(=O)NCc2ncoc2C2CN(C(C3CC34CC4)=O)C2)C=CCC1 C=C(C)CC(C)C(=O)N1CCN(C(=O)Cc2ccccc2OC)C(C)C1 N1(C(C(C)OCCC(C)C)=O)CCCN(C(C2CC3CCC2O3)=O)CC1 N1(C(C(C)OC2CCCCC2)=O)CC2CCN(C(c3ccc(Cl)cn3)=O)C2C1 C(=O)(C(C#N)C(C)(C)C)N1C2CC(NC(c3cc(CC)no3)=O)C1CC2 c1(C(N2C(COC(=O)NC)CCCC2)=O)cccc(O)c1F C1(NC(Cc2cn(CC)nn2)=O)CCC(CC(=O)NC2CCCC2(C)CO)CC1 c1(COC)ccc(C(=O)NC2(CNC(C3CN(C)CC3C)=O)CCCC2)cc1 N1(C(C(C)S(C)(=O)=O)=O)Cc2ccccc2C(CNC(=O)C2=NOCC2)C1 n1(CC(=O)NCC2OCCN(C(C(CC)(C)OC)=O)C2)ccc(=O)n(C)c1=O Cc1nn(C(C)(C)C)cc1C(N1CCC(NC(=O)C=Cc2cc[nH]n2)C1C)=O C(=O)(CCC(=O)N1CC(O)(C(C)(C)CNC(C2(C)CCNC2=O)=O)C1)OCC C(=O)(C1=C2CCCN=C2NN1)N(C)CC1CCN(C(C2CCCC(C)C2)=O)CC1 C(C)(C(C(=O)Nc1cnn(CC)c1)C(C)C)NC(CCC)=O c1(NC(C2c3ccc(o3)N2C)=O)ccccc1OC.C1(CC)CCC1C C1(N(C(=O)C(CC)N(C)CC)CC#C)CCN(C(c2cnc(Cl)s2)=O)CC1 C12(NC(C)=O)CCN(C(c3ncc(Br)cn3)=O)CC1C2 CCCCC(CC(=O)NC1(CN(C)C)CCCC1)NC(C1CC(SC)C1)=O C(CC(F)F)(C(=O)NCC1(C)CCCC1)N(C)C(C1CC12CCCCC2)=O c1(-c2nc(C(C)O)nn2C2CCCOC2)ccc2ncn(C)c(=O)c2c1 C1(O)(CC(=O)NCCCN(CC(=O)N(CCCC)CC)C2CC2)CCCCC1 C1(CC(C)C)CCCCN1C(=O)CN(C(=O)CN1CCCC(O)C1)C C1(Cn2cc(C3(N(C)C)CCCC3)nn2)COCCN1C(c1ccncc1N)=O c1(CNC(C(CC)OC)=O)nc(C)c(C(=O)N(C)Cc2cnn[nH]2)o1 O=C(C1=CS(=O)CCC1)N1CCC2CN(C(=O)CCC3CCCCC3)C2C1 C(CC(=O)N=c1ccn(C)[nH]1)c1cnc(NC(C23CCCCC2C3)C)s1 C(C(CC(=O)NC1CC(C)(NC(c2ccc3nn[nH]c3c2)=O)C1)C(F)F)N(C)C C1(C(N2C(C(=O)NC3(COC)CCOCC3)CCC2)=O)CC2C(C1)C2(F)F C1(CC)CCCCC1C(=O)NCCOCCOCCNC(c1n[nH]c(C)n1)=O C1(NC(=O)C=CC2CC2)COCCC1NC(C1CC(O)C1)=O CC1C(NC(C2(C)CCCCC2)=O)CCN1C(C1CCC1CF)=O C1(C(=O)NC(c2cccnc2)C(=O)NCCOCC(F)F)CC2(CCC2O)C1 N#CC1CCN(C(=O)COC2CCN(C(=O)CC3CCC(=O)N3)C2)C1 N1(C(C2CCC(=O)NC2)=O)CC2CC(CNC(=O)Cc3ccc(O)cn3)C2C1 NC(=O)C(F)(F)CNC(=O)CNC(c1cn(CCO)nn1)=O C(=O)(C(F)CCC(=O)O)NC(C)(C)C.C(=O)(CC1(CC(=O)OC)CC1)OC c1(C(=O)NCCC2CCN(C(c3coc(CO)c3)=O)C2)cc2c(C3CC3)cccc2[nH]1 C1(CNC(C(CC)NC(N)=O)=O)CC2CCC(C1)N2C(=O)CC(C)(C)OC C12(C(COc3cc(-c4cn(-c5cccc(OC)c5)nn4)sn3)=O)CCCCC1C2 N1(C(CC2C(CC)C2)=O)CCCN(C(C2(CF)CC2)=O)CC1 c1(C(C)(C)C)cnc(CCC(=O)NCC2(NC(C3CSCCS3)=O)CCOC2)o1 c1(C(=O)NCC2CCN(C(=O)C(F)C3CCC3)C2)ccc(-c2ncc[nH]2)nc1 c1(C(=O)NCC2N(C(C3(CCOC)CCC3)=O)CC2)cn(C)c(=O)cc1C N1(C(c2c(OC)cccc2Br)=O)CCC=C(C(=O)Nc2cccnc2C(N)=O)C1 C1(CNC(c2c(OC)n(C)nc2)=O)(OC)CCN(C(=O)CCC2CC2)CC1 C#CCCCC(C)C(=O)NCCCCCCN(C(=O)C=CC(C)(C)C)C C1(N(C(C(CCC)C)=O)CC2CCC2)CCCN(C(c2ccc(F)cc2)C)C1=O Cc1cnc(Cl)c(S(=O)(=O)N2CCCC(C)(C(=O)Nc3cnncc3Cl)C2)c1 c1(CCC(=O)NC(CC)CNC(=O)C(CO)N(C)C)n[nH]c2c1CCCC2 CCCCCS(=O)(=O)CC(=O)N1CCCN(C(c2ccc(Cl)c(C)c2)=O)CCC1 CCC(C)(C)CCCC(=O)N(CC)CC1CCCCN1C(c1csc(CC)c1)=O Cn1ncc(C(N2CCOCC2CC(=O)NCC2=CCCCC2)=O)c1Cl c1(C(C(=O)NCCC)N(C2COC2)CC)c(C)cnn1Cc1ccccc1 c1(C(=O)NC2CC(C(=O)Nc3ccc(F)cc3CO)C2)c(Cl)cnc(Cl)c1Cl C(=O)(CCCc1cncs1)NC(CC)CN(C)C(c1ccc(C)o1)=O CC1(C)CN(Cc2ccccc2)CCC1NS(=O)(=O)CCOc1ccc(Br)cc1 CCC(C)(C(=O)N1CCC(O)(CCNC(c2cc3c(s2)CCC3)=O)C1)C(F)F C(=O)(CC(C)(C)C(F)F)N(CCOCCCNC(c1cnc(CC(C)C)[nH]1)=O)C CC(C)C(C)(CNC(=O)OC(C)(C)C)NC(c1ncc(Br)cn1)C S(=O)(=O)(c1cccnc1NC1CCCCC1C(F)(F)F)NCC(CN(C)C)(C)C c1(C(=O)NCCN(C(c2n(COC)ncc2)=O)C(C)C)nccnc1C(=O)OC C(=O)(C(C(C)(C)O)NC(c1cnn2c1CCC2)=O)NC(c1nccs1)C N1(C(CC=C)=O)CCN(C(c2cccnc2-c2ccc(C)cc2)=O)C(COC)C1 C=Cc1ccc(C(=O)NC(CCCC)C(=O)NC2(C(=O)NCC)CC2)cc1 S(=O)(=O)(c1ccc(=NCC(O)c2ccnn2C)[nH]c1)N(CCN(C)CCO)C c1(C(N2CC(O)CC(NC(CS(=O)(=O)NC)=O)C2)=O)ccnc2cc(F)cnc12 c1(OC)c(CCC(=O)NCC(O)CCOC)cccc1F c1(C(N2C3CCC2CC(NC(=O)C(F)(F)C(F)F)C3)=O)cnc2ncccn12 Cc1cn(C)nc1C(N1CC(C(O)C(N2CCC(N3CCC3)CC2)=O)C1)=O Cc1cc(NC(=O)CCc2cnn(C)c2)ccc1NC(=O)CC1CCC1C C1(C(C)C)CC(C(=O)N(CC(O)C(F)(F)F)C2CC2)CCO1 C1(C(N2C(CNC(C(C)(C)CC#N)=O)CC2)=O)CCc2nnc(Br)n2C1 CC(CC(=O)NC1CCCC1CNC(c1cccnc1OCC(F)F)=O)C(F)F C(=O)(CCCCCCN=[N+]=[N-])NCC1N(C(C(CCC)N(C)C)=O)CCCC1 N1(C(CNC(C(C)N(C(C)=O)CCO)=O)=O)CCN(C(=O)CSC(F)F)CC1 C1(C)(CNC(c2c(CC)oc(C)c2)=O)CN(C(=O)CC2C=CS(=O)(=O)C2)CCO1 c1(C(C(=O)NCCCNC(=O)CC2CC=CC2)(F)F)cccc(Cl)c1 N1(C(C2(CCNC(c3cccc(C)c3F)=O)CC2)=O)CCCCC(F)(F)C1 N1(C(CC(C)C2CC2)=O)CCCC(C(=O)NCC(C)OC2CCCC2)CC1 C(=O)(C1=CCC(C)CC1)N1CCN(C(C2CCN(C(C)=O)CC2)=O)C(CCO)C1 c1(C(N(CC(C)NC(C(C)O)=O)C)=O)cccc(OCF)c1 C1(CNC(C(CC)SC)=O)(NC(=O)C=Cc2cnn(C)c2)CCCCC1 C(=O)(N=c1[nH]n(-c2ccccc2)cc1C#N)c1cnn(CC(=O)OC)c1OC c1(C(=O)OC)c(Cl)nc[nH]c1=NCCC1CCCCN1C(=O)CC1CCOCC1 c1(OCc2cc(C(=O)N(C3CCN(OC)C3)C)n[nH]2)cnccc1OC Cc1cccc(N)c1C(N1C2CCC(C2)C1CNC(=O)C=CC(=O)NC1CC1)=O C1(NC(c2c(C)cns2)=O)CCOC(C(=O)NCCS(N)(=O)=O)C1 c1(CC)cc(NC(C2(CNC(=O)CN3CCCC3=O)CC23CCC3)=O)ccc1F C1(OC)CC(CNC(c2c[nH]nc2C(F)(F)F)=O)N(C(=O)C(F)CC2CC2)C1 c1(C2CCN(c3ccnc(NCC4(C(C(C)C)O)CC4)n3)C2)cc(F)cc(Cl)c1 C1(C(=O)NC2C(NC(c3ccc(N)cc3Cl)=O)CCC2)CS(=O)(=O)CC12CC2 C1(C)(C(=O)NC2C(NC(c3cc(COC)on3)=O)CCC2)CCNC(=O)C1 CCCC(CC)N=c1cc(C)[nH]c(=NCc2cc(C)cs2)[nH]1 C1(O)(CN(C(c2c(NC)cccc2)=O)C)CCCN(C(C2C=C(C)CS2)=O)C1 CC(C)C(CNC(c1csc(C(F)F)n1)=O)NC(C1(Cl)CC1)=O c1(OC(C)C)sccc1C(=O)N(C)CCOCCN(C)C(C1(O)CC1(C)C)=O C1(C(N2CCCC2Cn2cc(Cn3cccc3)nn2)=O)CC2CCCC2N1 Cc1ccc(C(C)C(=O)NCC2CC(NC(c3c(Br)noc3C)=O)C2)cc1 c1(NC(N2C(NC(=O)OC(C)(C)C)CCC2)=O)nnnn1C1CC1.c1(C)ccccn1 c1(C(=O)NCC(C2CC2)NC(C(CC=CC)C)=O)cc(C(C)(C)C)n(C)c1C c1(C(=O)NC2C(C)CN(C(c3cnn(CCF)c3)=O)C2)ccc(F)c(O)c1F CCC(C)CC(C)C(=O)N1CC(CO)(NC(=O)CN(c2ccc(Cl)cn2)C)C1 c1(-c2nc(-c3cc(C)nnc3)on2)cnn2cccc2c1 C1(OCCOC)CCN(C(=O)Oc2scc(C(C(=O)OC(C)(C)C)C)n2)C1 CC1CN(C(=O)C(F)(F)C(O)C2CC2)CCC1CNC(=O)COCCF C#CCCCC(C)C(=O)N(C(CC)CC(=O)NC(CC)C1CCC1)C c1(CC)ccc(CC(N2CCCCC2c2cccc(C)c2)=O)cc1 c1(C(=O)NCC2CCC2NC(C2CCC(=O)N2C2CC2)=O)cccc2occc12 CC1(C(=O)NCCNC(=O)CC2CCCCO2)COC(=O)N1 N1(C(c2cc(CC)nn2C)=O)CC2CC(NC(=O)CC3CCC(O)C3)C2C1 N1(C(C2CC(CC)C2)=O)CC(CO)C2(C1)CN(C(c1csc3ccccc13)=O)C2 C1(C(C)(C)NC(COCC(=O)OC)=O)CCN(C(=O)Cc2cc[nH]n2)C1 C1(O)(C(=O)NCc2cc(C(N(CC)OC)=O)on2)CC2CCC1C2 C=Cn1nccc1C(=O)NCC1CCCCN1C(c1cnn(CC(F)F)c1C)=O S(=O)(=O)(c1cccc(=NCCC2CC=CC2)[nH]1)N(CC(C)C)CC1(CC(C)C)CC1 C1(NC(c2c(CC)noc2)=O)CCCC(NC(c2cccc(Cl)c2OC)=O)CC1 C12(C(N3CCC(C(C)CNC(c4cccc(O)n4)=O)CC3)=O)CCCC1CCC2 c1(C(=O)NCC(CNC(CCS(C)(=O)=O)=O)F)cc(F)cc2ccccc12 C(=O)(C1=NOC2COCC12)N1C(C)CC(NC(C2CCNC2=O)=O)CC1 Cc1cc2n(n1)CCN(c1cc(C(F)(F)F)nc(-c3ccncc3)n1)C2 N(C1c2ccccc2CC1NC(c1ccc(CO)o1)=O)C(C1C(C)CCO1)=O N1(C(CCCC#CC)=O)CCC2(CCN(C(c3ccc(CN(C)C)cc3)=O)C2)C1 C1(CC(=O)NCC(C)(C2CC2)NC(CCSC)=O)C(=O)ON=C1C CCCCCCCCCCC(C)NC(=O)Nc1cc(Cl)cc(Br)c1F C1(OC)(CNC(c2cc(C)nn2-c2ccccc2)=O)CCN(C(=O)CC2CC2)C1 n1(CC(=O)OC)c(C)cc(C(=O)NC(CNC(=O)CC23CCC(CC2)C3)CO)c1C C(c1ccncc1)=C(C)C(N1CCOC(CN(C)C(C2CC2C(F)(F)F)=O)C1)=O C1(NC(C(C)CC2CC2)=O)(CO)CCN(C(c2coc(CO)c2)=O)CC1 c1(C(CC)C(=O)N2CC(NC(c3ccc(CN(C)C)o3)=O)C2)ccc(F)cc1 C1(NC(Cn2c(C)cc(C)n2)=O)CC12CCN(C(=O)C=CSCc1ccco1)C2 N1(C(c2cc(Cl)ccc2C(F)(F)F)=O)CCn2ncc(C3=CCCC3)c2C1 c1(C(N2CCCC(NC(c3cc(O)cc(O)n3)=O)CC2)=O)ccc2sccc2c1 N1(C(CN2CCN(C)CC2)=O)CCN(C(=O)CCS(C)=O)C2CCC12 N1(C(C(C)Cc2ccncc2)=O)CCN(C(=O)CSc2cn[nH]c2)CC(C)(F)C1 N1(C(c2cccc(Cl)c2)C(=O)NC2COC2)CC(O)C2(CCCC2)C1 c1(C(=O)NCC=CCNC(c2c(C)cccc2F)=O)[nH]nc2ncccc12 c1(NCC2N(C(=O)OC(C)(C)C)CC2)cc(CO)no1 c1(OCC)cc(=NC(=O)CC(=O)N2CCC3(CC(O)c4ccccc4O3)C2)[nH]o1 CC1CN(C(C2C(C)(C)C2(C)C)=O)CC(C)C1NC(c1cc(Cl)c(Cl)s1)=O C1(C(CC)C)CCCN1C(=O)C(C)N(C(=O)CCNC(=O)CO)C1CC1 N1(C(CC(CC)CN(C)C)=O)CC(C)N(C(=O)CC2(C)CCOCC2)CC1C c1(NC(CC(=O)N(C(C)CC(=O)NC2CC2)C)=O)cnn2c1CCCC2 C1(CC=C)(NC(=O)CC(C)N(C)C)CCN(C(=O)Cc2cc(C)ccc2F)CC1 C1(C(=O)NCC(C(C)(C)C)NC(c2c(SC)csc2)=O)CC(C2CC2)=NO1 N1(C(C(C(=O)OC)C)=O)CC(C2(NC(=O)CC3COCCN3C)CC2)C1 c1(C(C)NC(c2cc(CC)cc(CC(=O)OC)c2)=O)cc2n(n1)CCCC2 N1(C(CCCC=C)=O)CC2CN(Cc3ccc(O)c(C)c3)C2C1 c1(C(=O)Nc2c(C)nc(F)cc2)n[nH]c2c1CN(C(=O)Cc1scnc1C)C2 N1(C(C(CC(C)C)OC)=O)CC2CC(C1)C(CO)C2NC(=O)Cc1nc[nH]n1 CCCCCC(C)(CC)C(=O)NCCCCCCn1cc(C2CCCC2)nn1 N1(C(CC(CC)CC)=O)CC2(CCC2)CC1CNC(c1c(C)ccc(C)c1C)=O C=CC(C)(O)CC(=O)N1CCCC(c2n[nH]c(CNC(=O)CCSCC)n2)C1 C1(CC(=O)NC(C(=O)OCC)C)CC2(C1)CN(C(=O)CN(C)C(=O)C1CC1)C2 CCCCC(C)(CO)NC(=O)Cn1cnc(Br)n1 C(=O)(N=c1cnn(C2CC2)[nH]1)c1cccc(C(C)NC(=O)Nc2ccccc2)c1 C=C=CCCC(=O)NCCC(=C)CNC(c1occc1Br)=O c1(CN(C)C(c2ccc(O)cn2)=O)ccccc1CNC(c1cn(CCO)nn1)=O C1(NC(c2cnc(C(C)C)nc2)=O)CC(C)CN(C(c2cc(Cl)ccc2N)=O)C1 C=CCCCCC(=O)NC1(C(=O)NCCCC(=O)N(C)C)CC1(C)C C=C(C)CC(C(=O)NC(C)CCC(=O)NCCc1ncoc1C)OC Cc1ccc2c(c1)CC(C(=O)NCC1CCCN1)S2(=O)=O CC1=C(C)CC(C(=O)NC2CCC(Cn3cc(CCOCCO)nn3)CC2)CC1 CC1CC(C(N2CCN(C3CCN(C(=O)CC4CC4)CC3)CC2)=O)CC(C)O1 c1(COC)nc(C)c(NCC(=O)NC(c2ccccc2C)=O)s1 c1(C(N2CC(NC(C(C)OCCOCC)=O)C2)=O)cc2c(nc1O)CCOC2 N1(C(CNC(N)=O)=O)CC(C2CC2)(C(N2CC(O)(c3nn[nH]n3)C2)=O)C1 N1(C(C=C(C)C(F)F)=O)CCOC2CN(C(c3cc4[nH]ccc4s3)=O)CC12 c1(-c2cnc(NC(c3cccc(OC)c3O)=O)c(O)c2)cccc2c1OCC2 C(=O)(C(O)C(F)(F)F)NC(CC(N1C(CNC(C)=O)CCC1)=O)C1CC1 c1(C(N2CC(CC)C(NC(c3ccccn3)=O)CC2)=O)cncc2sccc12 N1(C(CCC(=O)NCCC)=O)CCCC(C(=O)NCCC(=O)OC)C1C N1(C(CC=C=C)=O)CCN(C(c2nnccc2C)=O)C(C)C1C C1(CCC(=O)OCC)NC(=O)N(CC2CCCS2(=O)=O)C1=O S(=O)(=O)(c1cc(C(=O)OC(C)(C)C)cs1)Nc1c(C)noc1-c1ccccc1 c1(CC(=O)N(CCC(C)NC(CSCC)=O)C)nc(Br)n(C)c1C C1(CC(=O)NCC2(NC(CCc3cc(C)[nH]n3)=O)CCCC2)CCCCC1(C)C c1(OC)cccc(-c2nc(C(C)CC(F)F)n(C3CCN(C)CC3)n2)n1 C1(C(N2CC(NC(C3(O)CCCCCC3)=O)CC(O)C2)=O)CN2CCC1CC2 C(N=c1[nH]c(N2CC3CC2C(F)(F)C3)nc2cccnc12)c1scc(C)c1 Cc1c(CCC(N2CC(NC(=O)C(C)C3CC3)C(O)C2)=O)cnn1C c1(NC(CC(CCC)NC(=O)OC(C)(C)C)=O)ccc2ccn(C)c2c1 CC1(C)CC(NC(=O)CC(CNC(=O)Cc2cncs2)C2CCC2)C12CC2 Cc1cc(CNC(C2(CC(C)C)CCN(C(=O)C(C)OC(C)C)C2)=O)cc(F)c1 c1(C(N2CC(NC(C(C)(CO)OC)=O)C(C(F)(F)F)C2)=O)cccn2nccc12 C(=O)(CCC(C)(C)C#N)N1CC(C(=O)NC(c2nn[nH]n2)CC)C2(C1)CC2 N1(C(C(CC)C2CCOCC2)=O)CCN(C(C2(C#N)CC2)=O)CC(C)C1 N1(Cc2c(C)nn(C)c2)CCC(C2CCCN(C(=O)C(=O)Nc3cccs3)C2)C1 C(=O)(C1=C(C2CC2)N(C)C(=O)N(C)C1c1cnc2c(F)c(F)ccc2c1)OC Cn1cnc2c1C(C(=O)NNC(=O)c1cccc3sccc13)CCC2 C1(C)(COC)CC(NC(=O)C=CSC)CN1C(c1oc(C)nc1C)=O c1(C(=O)NC2C(NC(CC=C=C)=O)CC2)ccc(C#N)c(Cl)c1 c1(NC(C2SCCN(C(C3CCN(C)C3)=O)C2)=O)cn2nc(Cl)ccc2n1 C1(c2nnnn2CC2CCOC2)(NC(CC(C)(C)C)C)CCC=CCC1 c1(-c2ccc(CC)o2)nc2ccc(C(=O)Nc3ccc(C#N)o3)cc2[nH]1 CCCC(CCC)CC(=O)NCC(CO)NC(=O)CCOc1ccc(OC)cc1 CCCCCCCC(=O)NC1CC(C(=O)N(CC(=O)OC)C)=CC1O c1(C(=O)NC2CCC(C(=O)NCC3CCN(CC)CC3)C2)cc(F)cc(Br)c1F C1(C(=O)NC(CC)COC)CC2CCCC2N1C(C1CC(=O)N(C)C1)=O C1(NC(c2cc(C)sc2C)=O)C2CCCN(Cc3snnc3C)C2C1(C)C c1(C(N(c2nc(SC)c(Br)cn2)C2CCNCC2)=O)cc(Cl)cc2nc[nH]c12 C12(CNC(C3C(C=C)C3)=O)CCC(NC(=O)CC3(NC(C)=O)CC3)(CC1)CO2 c1(NC(C)C(=O)NC(c2ccccc2)CNC(c2cnsc2)=O)ccccc1 c1(CNC(COCC(=O)O)=O)cn(C2CC2)cn1.c12cn-1nn2 c1(OC)ccc(C(N2CC(CNC(=O)Cc3cnc(C)s3)C2)=O)cc1C1CC1 N1(CC(=O)NC2(C3CN(C(=O)CC=C(Cl)Cl)C3)CC2)CCCCC(O)C1=O c1(C(N(CCOC)CCNC(=O)Cn2cccn2)=O)c(F)cc(C)cc1F C12(C(N3CC(COC)C3(C)C)=O)COC(C1)C(NC(c1c(C#N)ncn1C)=O)C2 c1(OC)oc(C)nc1C(=O)NC(C1CN(C(=O)C2=C(C)CC2)CCO1)C CC1(C)CCN(C(=O)Cn2cnnn2)C1C(=O)NCC(O)Cn1cccn1 C1(C(=O)NCCCCC2(NC(c3cnc(N(C)C)s3)=O)CC2)CC2(C1)CC(O)C2 C(=O)(C(CO)C(F)(F)F)N1CC2C(CC(=O)NC3(C)CC(F)(F)C3)(CC2)C1 C(=O)(C(O)COC)NCC1(CC(=O)N(CC(C)OC)C)CC1 c1(C(=O)NCC2C(NC(c3cccc(C(C)C)c3F)=O)C2)ccc2c(c1)NCC2 C(=O)(CC(C(=O)N(CC(O)CNC(=O)CN1C(=O)CCC1=O)C)NC(C)=O)OC c1(C(N(C(C)CCNC(c2cc(Cl)cnn2)=O)C)=O)ccnn(C)c1=O c1(C(=O)NC2C(CNC(Cc3cn(C)nc3)=O)CCC2)cc2n(n1)CCCC2=O C1(C(=O)NCC(C)Cn2ccnc2)CN(C(C2(C(N)=O)CCC2)=O)CCO1 CCS(=O)CC(=O)N1CCC(C)(CCNC(=O)Cc2ccnn2C2CCCC2)C1 N1(C(c2cn(CC)nc2)=O)CCC2CCN(C(=O)CC3=CCCC3)C2C1 C1(NC(C2C(C)CCO2)=O)CCCC(CNC(c2cccn2C2CCCC2)=O)C1 c1(-c2nc(O)cc(C)n2)nc(C2COc3ccccc32)nn1CC1CCCO1 Cc1nc(O)ccc1C(=O)NC1COCCN(C(C2CC2C)=O)C1 n1(CC(C)C)[nH]c(CC(=O)N(CCCCN(C)C(C2CCCO2)=O)C)cc1=O C1(NC(C2(CCCC)CC2)=O)CN(C(C2(c3ccccc3)CCCC2)=O)CCC1C C#CCCCCC(=O)N(CCNC(=O)C(c1ccc(F)cc1C)O)CCOCCO S(=O)(=O)(CC(=O)NCC(C1CCC1)NC(=O)C(=O)C(C)C)NCC N1(C(C2C(CC)CCC2)=O)CC2CC(C1)CN(C(c1cnc(S)nc1)=O)C2 C(=O)(C1CCS(=O)(=O)c2ccccc21)NC1CC(CNC(c2cc(C)no2)=O)C1 CCC(C)(CNC(c1n[nH]cc1Cl)=O)NC(C1CC(=O)C1C(C)(C)C)=O c1(N(C)C)cnc(C(N2CCCC(CNC(c3cocc3C(N)=O)=O)C2)=O)cn1 c1(OC)cc(Cl)c(Br)cc1NC(CCC(C)C)C(=O)OCCCF C1(C(C)(C(=O)NCCOCC)NC(C(F)=CC)=O)CCOCC=C1 N1(C(c2c(C)nncc2)=O)CC2(CCCC2NC(c2noc3ccccc23)=O)C1 Cc1c(CC(=O)NCC2(C)CC(F)(F)CN2C(=O)CNC=O)cccc1[N+](=O)[O-] N1(C(c2c(C)nn(C)c2)=O)CC2(C)CC1C2NC(=O)Cc1c[nH]nc1O N1(C(C2CCN(CC)C2)=O)CCC(NC(c2scnc2C2CC2)=O)C12CC2 C(=O)(C(C)S(N)(=O)=O)N1CC(C(N(C(c2ccncc2)C)C)=O)C(C)C1 c1(C(=O)OC)ncc[nH]c1=NCc1ccc(CNC(=O)C=C(C)Cl)c(F)c1 c1(C(C)C)ccc(C(=O)NC(C)CC(C)NC(c2ccc(C3CC3)cc2)=O)cc1 N#CC1(NC(c2cc[nH]c2)=O)CCN(Cc2ccc(O)cc2Br)C1 n1(CCC(N2CC(OC)(CNC(=O)CCC3CC3C)C2)=O)cnccc1=O C1(CN(C(c2cc(Cl)ccn2)=O)CC)CCCCN1C(=O)C1=COCC1 c1(C(=O)NCCCCNC(=O)Cc2cnc(C3CC3)[nH]2)cccc2nsnc12 c1(C(N2CCC(CNC(C3(C)CC(=C)C3)=O)C2)=O)cc2c([nH]1)CCC2 c1(CNc2c(CC(N3CCC(F)CC3)=O)cccc2)cccc2nccnc12 C1(C)(C(N2C3CCC(NC(CCOC)=O)(C3)C2)=O)CC(C(F)(F)F)=NO1 C(=O)(C(C(C)(C)C)N(C)C)N1C(C(N2C(C=C)CC2)=O)CSCC1 c1(C(=O)N(CCN(C2CC2(F)F)C2CC2)C2CC2)ccc(C(F)F)cc1C(F)(F)F CCC(CNC(C1CCN(C(C)=O)C1)=O)(CC)NC(c1cc(C(N)=O)[nH]n1)=O C1(CNC(CC2(CSC)CC2)=O)(CO)CCCN(C(=O)C(O)C(F)(F)F)C1 C1(N(C(Cc2scc(C)n2)=O)C)CCCN(C(C2CNC(=O)N2C)=O)CC1 N1(C(Cc2n(C)cnn2)C(N)=O)CCC(C(=O)OC(C)(C)C)c2ccccc21 N(C(=NCC1CC1c1ccccc1)N1CCc2c(F)ccc(F)c2C1)C(C)CC#N C(=O)(CC(F)(F)CS(C)(=O)=O)NC1C2(CCN(C(c3c(C)ccnc3)=O)CC2)C1 N1(C(C2N(C(C)=O)CC(O)C2)=O)C2CCC1CC(NC(c1ncccc1Cl)=O)C2 C1(CNC(C(C)SC(C)C)=O)CCC2(CN(C(C3CCC4(CCC4)CC3)=O)C2)O1 C1(C(N(C(C)CNC(c2coc(C(F)F)n2)=O)CC)=O)OCCC1C(C)C Cc1sc(C(=O)NCCOCCNC(=O)Cn2[nH]cnc2=N)c(C)c1C Cc1cc(C(=O)NCC(C)(F)CNC(=O)CC2=CCOCC2)c(C)c(C)c1 N1(C(c2cc(OC)n(C)n2)=O)C(CNC(=O)C(C)(C)CC(F)F)CC2COCC12 C1(C#CC(=O)N2CCC(C(C)NC(c3nc(C)ccc3C)=O)CC2)(CC)COC1 c1(CCC(=O)NC(C)CNC(=O)CC2(O)CCOC2)cccc(Cl)c1 C(CC(C)C)(C(=O)N1CCCC(N(CCF)C(c2ccc(Cl)s2)=O)C1)OC C12(C(N(C)CC3CCCN3C(c3cnoc3C3CC3)=O)=O)CC(C1)S(=O)(=O)C2 c1(C(N(C2CN(C(C(C)=C(CC)C)=O)CC2F)C)=O)cc(F)c(F)cc1OC c1(C(=O)NC(C)(CO)C(=O)N2CCC(n3ccnc3)C2)cccc2cc[nH]c12 C1(CCC)CN(C(c2cn(C)nc2OC)=O)CCN1C(=O)CC1CCC(=O)N1C c1(OCC)cccc(CC(=O)NCC(C)CNC(c2c[nH]nc2C(F)(F)F)=O)n1 c1(CC(C(=O)NCC(CNC(C2CC(CC)C2)=O)O)O)cccc(OC)c1 c1(C(N2CC(CCNC(c3n[nH]c(C)c3Cl)=O)OCC2)=O)cc(Cl)c(F)cc1F c1(C(N2CCC(C(=O)NC(COC)C(C)C)C2)=O)c(OC)cccc1C N1(C(C(=O)N(CCOC)C)C)C(=O)CCC1=O.C1(C(C)C)CCN(C(C)C(=O)N)C1 S(=O)(=O)(c1cccc(CCC(=O)OC)c1)Nc1n(CCOC)ccn1 C1(C(=O)NCC(F)(F)CC2CC2)CN(C(=O)Cn2nccn2)CC12CC2 N1(C(C2(C)CC=C(C)CC2)=O)C2CCC1CN(C(c1nnn(C(C)C)c1C)=O)C2 c1(C(N2CCCN(C(C(F)=CCC)=O)CC2)=O)cc2ccccc2c(OC)n1 CCS(=O)c1ccccc1OCCCNC(=O)N(C)C C1(NC(c2ccc(CCC)s2)=O)CC2CCC1C(NC(=O)C#CC(C)(C)C)C2 C1(CCC)CCN(C(=O)C(F)C2CC(NC(C3CC3Cl)=O)C2)CC1 N1(C(CC2C(CC)C2)=O)CC(NC(C2(C)CCCN(C)C2)=O)C(N=[N+]=[N-])C1 c1(NCC2C(C)C2C)[nH]c(=NCc2ccccc2C(C)(F)F)nc2ncn(C)c12 C1(CCC)CN(C(C2(NC(=O)CCCCNC(N)=O)CC(F)C2)=O)CC1CO C1(NC(c2c(CC)cccc2F)=O)CN(C(C2(O)CCSC2)=O)CC1S(C)(=O)=O c1(C(=O)NC23CC(NC(c4n(C)ncc4)=O)(C2)C3)nccc(F)c1Cl N1(C(C)C)CCN(C(=O)C(C(C)O)NC(C2CC=CC2)=O)CC1 c1(C(N2C(C(=O)NCC(CC)C(C)C)CC(OC)C2)=O)cc(C)nc(C)n1 N1(c2c(C)cncn2)CCN(C(c2c(F)cccc2Br)=O)CC1C CC1=C(c2ccncc2)CN(c2nc(N3CCC(C)(C)C3)c3c(n2)CSC3)CC1 c1(N2CC(OCCNC(c3c(C(C)C)noc3)=O)C2)ncccc1C#N C1(C(c2ccc3nc(N4CCCCC4)sc3c2)=O)CCc2nnnn2CC1 N1(C(C(CCC)(C)O)=O)C2CCCC1CC(NC(=O)CSc1nc[nH]n1)C2 C1(C)(CNC(c2n(C)cnc2)c2nnnn2C2COC2)CC=CCC1 Cc1cc(NC(=O)COC(=O)C(O)CC#C[Si](C)(C)C)n(-c2ccccc2)n1 c1(C(=O)NCC2(O)CC(CNC(c3c[nH]c(=O)cn3)=O)C2)ccc(Cl)cn1 c1(C(N2CCC(O)(C(C)NC(CNC(C)=O)=O)C2)=O)c(C)ncc2ccccc12 c1(N2CCC(NS(C)(=O)=O)C2)nc(N2CCN3CCCC3C2)nc2ccsc12 CC1=NN(C)C(=O)C1CC(=O)NC1(CNC(c2cn(C)cc2C(F)(F)F)=O)CC1 c1(C(=O)NCC2(C)CCC(NC(c3cc(CC)[nH]n3)=O)C2)cnn2cnnc2c1 C(c1ccncc1)=C(C)C(=O)NC1CC1NC(=O)C(C(C)C)N(C)C N1(C(c2cc(C)ncn2)=O)CCOCC(NC(=O)CC(O)C(C)C)C1 C1(C(=O)NC2(CNC(COC3(C)CCC3)=O)CCCC2)CC12CCOCC2 Cc1cc(Cl)c(Cl)cc1C(N1CCOC(CN(C(=O)C=CC(=O)N(C)C)C)C1)=O N1(C(C(=O)NC(C2COC2)C)C)CCN(C(=O)OC)CC1 C1(C(=O)NC(C(=O)Nc2cccc(Cl)c2)c2ccco2)CCCOCC1 c1(C(C)C(N2C(CNC(=O)C3=COCCO3)CC(O)C2)=O)c[nH]c2ccccc12 C=CCC(CC(C)C)C(=O)NC1(C(=O)NC2CC2O)CCC1 c1(CNC(C2CCC(C)C2)=O)ccc(CCNC(c2n[nH]c(C3CC3)n2)=O)cc1 C1(CNC(c2scnc2Cl)=O)COCCN1C(=O)CC1CCC(O)C1 c1(C(N2C(C)(CNC(Cc3ncc(C)o3)=O)CCC2)=O)ncnc2c1CCCC2 CN1CC2(CCN(C(c3cc(CNC(c4cn(C)c(=O)n4C)=O)no3)=O)CC2)C1 C1(NC(C2(C(=O)OC)C(=C)CC2)=O)CN(C(=O)C2=NOC(C)C2)CC12CCC2 N1(C(C(c2ccncc2)C)=O)CCC(C)C(CNC(c2cccc(Cl)c2)=O)C1 c1(OC)cnc(Cl)[nH]c1=NC1CCC2CN(C(=O)Cc3cc(C4CC4)on3)CC12 C1(C(=O)NC(CNC(C(c2nc(C)sc2)=O)=O)C(C)C)CC2CCC1O2 Cn1nc(C(=O)NCC2CN(C(c3ccc(C(N)=O)cc3)=O)CC2O)ccc1=O CC(CCC(=O)N1CCC(O)(CCNC(c2cnns2)=O)C1)N(C)C c1(C(N2C(CNC(C(CCSC)N(C)C)=O)CCC2)=O)ncnc(O)c1Cl C=CCCCC(C(=O)N1CCC(C)=C(C)C1)NC(=O)C(C)CC=CCC N1(C(C(=O)NCC)=O)CCn2c(CNC(C3CCN3C)=O)nnc2C1 N1(C(c2nn(C)cc2I)C(=O)NCCOC)CCCCCC1c1cccc(C)c1 N1(C(c2cnc(CC)o2)=O)CC2CC(NC(c3ccc([N+](=O)[O-])s3)=O)C1C2 CON1CCC(C(=O)NCC(O)CN(C)C(C2COCC2(C)C)=O)CC1 C(=O)(C1=CCCSC1)N1C(=O)C(O)CC1.C(C(O)CO)N(C(N)=O)C1CC1 C1(NC(c2cncc(NC)c2)=O)CC2CC(NC(c3cc(C)n(C)c3)=O)CC2C1 c1(C(=O)NC2C(NC(c3c(=N)cc[nH]c3)=O)CCC2)coc2cc(F)ccc12 CCCCCCC(C)NC(C1(F)CCCN(C(c2cnc3n2CCC3)=O)C1)=O C1(CN(C(=O)C(O)C2CC2)C)CCCCN1C(=O)C(c1ccccc1Br)(F)F O=C(CCCn1cc(CO)nn1)NCCNC(C1(c2ccccc2)CC1)C1CC1 C1(C2CCCCC2)(NC(=O)CCOCCCNC(C2COC(=O)N2)=O)CC1 c1(NC(C2C(NC(c3ccc(C)cc3F)=O)CCC2)=O)ncc2ccccc2n1 C(=O)(C1CCc2nccn21)NCCC(C)N(C)C(C1CN2CCN1C(C)C2)=O C=C(Cl)C(C)(C)C(=O)N1CCCC(N(C(=O)Cc2cccc(Cl)c2F)CCF)C1 CN=c1[nH]c(=NCc2cccc(C#N)n2)[nH]c(=NCC2=NOC3(CCC3)C2)[nH]1 CCC(CN=c1nc2c(ncn2CC)c(NCC(C)(CC)OC)[nH]1)OC c1(C(N2C(C(=O)NCCNS(C)(=O)=O)CCC2)=O)cc(C(F)(F)F)ccn1 Cc1ncccc1C(=O)NC(c1ccccc1)C(=O)NCCn1cccnc1=O c1(C(N2CCN(C(C(CC#C)C3CC3)=O)CC2C)=O)cc(F)cc(C)c1O CC1(NC(=O)CCCc2cccc(Cl)n2)CCCN(C(=O)Cn2cc(C#N)cn2)C1 Nc1ccc(C(=O)NCc2cn(Cc3cccc(OC4CCC4)c3)nn2)c(Cl)c1 O(NC(=O)C(C)(C)C(C)NC(=O)C(C)c1ccco1)CCOC C12(NC(c3c(C)n(C)nc3)=O)CCC(CNC(c3nccc(Cl)c3F)=O)(C1)OC2 N1(C(c2c(C)nn(C)c2N)=O)CCC2(CC1)CN(C(c1occc1Cl)=O)C2 N1(C(=O)CC2CNC(=O)O2)CC2CC(C1)N2C(C1(O)CCCC1)=O c1(C(=O)NCCC(C2CC2)NC(C(C)OCCOCC)=O)ccc(N)c(Cl)c1 CC1N(C(=O)C(N2CCC(S(=O)(=O)N(C)C)C2)=O)CCCC12CCC2 N1(S(CC)(=O)=O)CC2CCC1CN2Cc1cnc(Cl)cn1 C1(SC)CCCC1C(N1CC(C(N)=O)(CNC(=O)CC2(NC(C)=O)CC2)C1)=O C1(C(=O)OCC)CCN(CCC(=O)NC(=O)NCc2ccccc2Br)CC1C C=C1CCC(C(=O)N(C2CCCN(C(=O)C(F)OC)C2)CCF)CC1 C12(CC(=O)NCC(C)(CNC(C3CCOC3C)=O)OC)CCC(CC1)CC2 C1(NC(C2(COC)CC2)=O)CC2(CCCCN2C(C2SC3C=CC2CC3)=O)C1 N1(C(C(CO)NC(N)=O)=O)CC2(CC(NC(=O)CN3CCCC3=O)C2)C1 C1(C(=O)NCCN(C(C2C(OCC)C2)=O)C2CC2)CCC(O)CC1 c1(CC)cc(C(=O)NCC2(C(=O)N(C)Cc3cn(C)nn3)CC2)on1 c1(CCC(=O)NC2C(NC(CCC#CC)=O)CCCC2)c(Cl)cccc1[N+](=O)[O-] N1(C(C(C#C)(C)C)=O)CCC2(CC1)CN(C(=O)C(C)CCCCCC)C2 N1(C(C2(C3(C)CC3)CC2)=O)CCC(C=CC(=O)NCC(C)(F)C(C)(C)F)CC1 N1(C(=O)Nc2ccc(OC)cc2)CCC(C)C(NC(C2C=CS(=O)(=O)C2)=O)C1 C(C(=O)NC1CCN(C(C2CCCC(=O)C2)=O)C1C1CC1)(C(C)C)OCC C1(NC(c2ncn(C)n2)=O)CN(C(C2Cc3nccn3C2)=O)C2CCCC12 c1(C(CC(=O)NCCC2CC(NC(C=C(CC)CC)=O)C2)O)cccc(F)c1 N1(C=O)CC23CCC2(COC3)C1.C1(C(=O)NO)CCN(C(=O)C2CC3(CCC3O)C2)O1 C=CCC(C)C(=O)N(CCNC(c1ccc(C(C)C)cc1)=O)CC1CC1 C(N=c1c(Cl)c[nH]cc1[N+](=O)[O-])C1CN(C(COC)=O)C(C)C1 Cc1nc(C)c(CCC(=O)NC(C)C(C)NC(c2cc(N)cc(O)n2)=O)c(O)n1 N1(C(C(CCC)NC(c2ncn(C)n2)=O)=O)CCC(C)=C(F)C1 c1(C(=O)NCC2(CNC(c3cc(C(N)=O)on3)=O)CCOC2)ncncc1Cl N1(C(C2(C#C)COC2)=O)CCC(NC(C2CC3CCC2CC3)=O)C(C)(C)C1 c1(C(=O)NC2CCCC(CNc3ncc(I)cn3)C2)cc2ccccc2oc1=O c1(C(=O)NC(CCOC)C(=O)N(C)CC2CCCO2)cnn2ccccc12 N1(C(C(C=C)CC)=O)CCC(CCOC)(NC(c2ccc(=N)[nH]n2)=O)CC1 c1(OCC(=O)NCC(CCOC)NC(=O)CCF)ccc(F)cc1Br Cc1ccc(C(N2CC(C(C)NC(c3c(C)coc3C(C)C)=O)C2)=O)c(C)c1 CC1CCCCN(C(=O)C(C(C)(C)O)NC(=O)COC(C)(C)C)C1 C1(C(=O)OCC)CN(C(=O)O)CCC1O.c1(C(C)CNC)c(C)nn(CC)c1C C#CCCC(O)C(=O)NCCC1(O)CCN(C(C2(N(C)C)CCCC2)=O)C1 C(=O)(C(C)(C)CC(F)F)NCCC(CNC(CCCCCOCC)=O)O CCCC(CCCNC(c1ccc(OC)cc1Cl)=O)NC(C1(Cl)CC12CCC2)=O N1(C(C(C)OC)=O)CCC(C(C)(C)C)(CNC(=O)C(C(C)C)c2cccnc2)C1 C1(C(N(C)Cc2n(CC)ccn2)=O)CN(C)CCN1C(=O)C(C)COC c1(C(N2CCC(CN(C)C(c3scnc3C3CCCC3)=O)C2)=O)ccccc1Cl C1(COC)CCN(C(=NCc2scnc2C)NCC2CCOC2)C1 N1(C(CC(C)C2CC2)=O)CC2CCCCC2(NC(=O)Cn2ncnn2)C1 c1(-c2cn(CCC(=O)NC(C)CCN(C)C)nn2)ccc(C(F)(F)F)cn1 CC(C)(C)CC(C)(C)C(=O)NCC1CCC(NC(=O)COCc2nc[nH]n2)CC1 Cc1cc(C)n(Cc2nc(-c3cccc(F)c3)nn2C(C)C)c(=O)n1 CCCC(O)C(CO)NC(=O)CN(C(c1cc(C)nnc1C)=O)CC1CC1 N1(CC(C)(C)NC(=O)C=Cc2cccnc2)CCN(C(C2CCNC2=O)=O)CC1 C1(NC(C2(CC=C)CCOCC2)=O)CCN(C(C2(C#N)CC2)=O)CC1F S(=O)(=O)(c1cccc(NCC(C)Oc2ccc(F)c(Br)c2)c1)N(CCC(C)C)C c1(NC(=O)CC2CCN2)cc(-c2c(CO)cccc2F)cc2[nH]ccc12 C1(NC(c2ccc(Cl)nc2Cl)=O)CCN(C(C2(CC3CC3)CC2)=O)CC(O)C1 n1(CC)c(-c2nc(CCCO)nn2CCN2CCC(O)CC2)cnc1O CC1(C)CCCCCC1NC(C1(NC(c2cc[n+]([O-])cc2)=O)CC1(C)C)=O Cc1cnccc1C(N1CC(c2ccccc2)(NC(C2COC(=O)C2)=O)C1)=O C=CCC(CC)C(=O)NCCCOCCN(C(=O)C(C)C)C N1(C(CN2CC(C)C2)=O)CC2CC(NC(=O)C=CCN(C(C)=O)C3CC3)CC(C2)C1 C1(C(c2nnnn2C2CC2)(C)NCC2CCCC(C)(C)C2)Cc2ccccc2C1 CC1CCCN(C(=O)CCc2cn(C)cn2)C1CNC(=O)CN1CCC(C)(C)C1 c1(C(c2occc2Br)N(CCNC(=O)C(C)(C)C)CC)ccccc1F c1(CC(=O)NC(CNC(C(C)OC)=O)C2CCC2)ccsc1Cl O(NC(=O)CN(C(=O)CC)CCN(C)CC1CCCO1)CCC CN(CCCC(=O)N1CC(NC(c2cnn(C(C)(C)C)c2)=O)C2(CC2)C1)N=O CC1CN(C(=O)CS(C)(=O)=O)CCC1NC(=O)C(F)(F)C1CCOCC1 c1(C(C(C)NC(c2c[nH]c(C(C)(C)C)c2)=O)C)ccc(C(F)(F)F)cc1 c1(NC(C2CCN(c3cn(C)nc3)C2)=O)ccc(OC=C(F)F)cc1 C1(NC(C2C(CC)OCC2)=O)CCS(=O)(=O)C12CN(C(=O)C=C(Cl)Cl)C2 C(=O)(CCCC(F)F)NC(CNC(C1CN(C)C1)=O)C1CC1 CCCCCC(C)(C)C(=O)NCCCCN(C)C(C1CC(=O)N(C(C)(C)C)C1)=O CC1CN(C(C2CCC(F)CC2)=O)C(C)CN1C(=O)CCc1ccccc1C#N CCC(CC(=O)N1CCC(C)(C)C(C(=O)N(C)Cc2cnc[nH]2)C1)C(C)(C)C N1(C(=O)C2=CCOC2)CCN(C(c2ccc(-c3cccs3)o2)=O)C(C2CCC2)C1 C1(CC(=O)NCC(CNC(C2(C(C)C)CCCO2)=O)(C)C)CCCCCC1 N1(C(C2(O)C(C)(C)C2)=O)CCC2(CCOCC2)C(NC(=O)Cc2cn[nH]c2)C1 N1(S(c2c(C)cc(Cl)nc2)(=O)=O)CCC(N=c2ccnc(C(C)(C)CN(C)C)[nH]2)C1 n1(CC#C)c(C)cc(C(=O)N(C(C)C)CC2CCCCO2)c1C c1(C(N2C(CCN(C)C)CCC2)C(=O)NC2CCC2)ccc(F)cc1 Cc1cnc(C(=O)NC2CCCN(C(=O)CCc3nnc(C4CC4)o3)C2)c(F)c1 C1(NC(c2cnn(C)c2Cl)=O)CN(C(C2CCCC23CC3)=O)CC1(C)C C1(N(C(=O)C(c2ccc(O)cc2)=O)C)CC2CC(NC(=O)OC(C)(C)C)C1C2 C1(C(=O)NCCC(O)CNC(=O)CC2CCCC2O)(COC)CC(=O)C1 C1(C)(CC(=O)N(CCCOC)C)CCN1C(=O)C(C)NC(N)=O C1(N(C(=O)Cn2nnc(C)n2)CC)CCCN(C(C2CC3CCC2O3)=O)C1 C1(CNC(CC(=O)OC)=O)CCN(C(c2nn(C(C)(C)C)cc2Cl)=O)C1(C)C c1(NC(C2CC2NCc2ccc(F)s2)=O)ccc2sc(Cl)nc2c1 C(CC1=CCN(C(=O)C=C2CCOCC2)CC1)NC(=O)CC1CCC2CC12 C1(CC)CN(C(=O)C(CC2CCC2)NC(=O)C(=O)NC(C)C)CC1O N1(C(C2N(C(c3c(C)cccc3O)=O)CCC2)=O)CC(=O)NC2(CC2)C1 N1(C(c2cncc(O)c2Cl)=O)CCCC(C2CN(C(=O)C(O)C(F)F)C2)C1 CCCC(C)(C)C(=O)NC1CC(F)CN(C(=O)Cc2cccc(C(N)=O)c2)C1 CCC1=NOC(C(=O)NC2(C)CCCC2NC(c2csnn2)=O)C1 CCCC(C)(O)C(=O)N1CCC(CCNC(=O)CSc2cccc(C)c2)CC1 c1(COC)nc(Cl)cc(=NC2CC(NC(C3Cc4ccccc4CO3)=O)C2)[nH]1 C1(NC(c2onc(C)c2C)=O)CCCCC12CCN(C(=O)CC1CCOC1)CC2 c1(C(=O)NCCCN(C(C(C=CCCC)O)=O)C)cc2c(Cl)nccc2s1 N1(C(C(CC)N(C)C)=O)CCC(C2CC2)(NC(c2csc3ccccc23)=O)C1 N1(C(Cc2c(C)con2)=O)CC2CC(NC(C3CCOC4(CCC4)C3)=O)CC1C2 n1(CC)cc(C(=O)NC(C)(C)C=CC(=O)NCC(F)(F)CC2CC2)nn1 Cc1cccc(C)c1C(=O)NC1C=CC(C(=O)NCCCCc2ccccc2)C1 C#Cc1ccc(C)c(NC(C2CCCCCC2NC(c2cscn2)=O)=O)c1 c1(OCC(=O)NC(C)CCCNC(C2(C)COC2)=O)c(Cl)cccc1F Cc1cccc(CC(=O)NCc2cc(C(N3CCCC3CN(C)C)=O)co2)c1 C1(CCC2N(C(c3nc(C)[nH]n3)=O)CCC2)CCN(C(=O)CC2CC2C)CC1 c1(C(N(CCN(C(C(C2CC2)SC)=O)C)C)=O)cccc(CN2CCSCC2)c1 C1(CNC(C2N(N=O)CCC2)=O)CC2CCC1N2c1cc(C(F)(F)F)nc(Cl)n1 C(C(C)(COC)C(=O)N1CCCC(F)(C(=O)NCC(C)CC(F)(F)F)C1)OC N1(C(C(C(C)C)F)=O)CCC(O)(C(C)NC(=O)CCCCCn2cnnn2)CC1 CC1CCN(C(=O)N(C)Cc2ncnn2C)c2ccccc21 C1(C(=O)NC(C2CCN(C(C3(C)CC(F)C3)=O)C2)C)CCC1(C)C C1(NC(c2c(C(C)C)scn2)=O)C2CCN(C(=O)C=Cc3ccnn3C)CCC12 N1(C(C2(CC(C)C)COC2)=O)CC(CO)(NC(=O)C(C)n2ccnn2)C1 C12(NC(c3c(C)cc(SC)o3)=O)CCCC1N(C(c1ccc(Cl)cc1C)=O)CC2 C12(C(N(C3CCN(C(C45CCCN(CC4)C5)=O)C3)C)=O)CCC(CC1)CC2 CC1(C)CCCC(CC(N2CCC(CCNC(=O)Cn3cnnc3O)C2)=O)C1 c1(CC)cc2c(NCC3(CNC(c4coc(C(N)=O)c4)=O)CC3)ncnc2s1 n1(CCC)cc(C(=O)NCC2(CN(C(=O)CC(C)OC)C)CC2)c(C)n1 c1(CN2CC(C(C)NC(=O)C=Cc3ccccc3Cl)C2)c(Cl)cccc1B(O)O Nc1cc(F)c(C(N2CCC3CCC23CNC(c2cnsn2)=O)=O)cc1Cl N1(C(C(CC=CC)C)=O)CC(CC(=O)NCC(C)(O)CSC)CC1(C)C C=Cc1ccc(C(=O)NC2CCN(C(=O)C(C)C3CCC3)C(C)C2)cc1 C1(NC(c2cc(OCC)ns2)=O)CN(C(=O)C(COC)CC)C2CCCC12 CC(CC(=O)N1CC2CN(C(c3nc(Cl)ccc3N)=O)CCC12)C(F)(F)F CC1(O)CCN(CC(=O)NC2CCCCC2NC(=O)C(c2cccnc2)O)C1 C(CC(N=c1cc[nH]cc1C#N)C(C)C)N(C(Cc1ccc(C)nc1)=O)C C(CCC(C)C)(C(=O)NCc1ccnc(Cl)c1)NC(Cc1cc(C)n(C)n1)=O C1(CC(=O)NCC(CC)NC(c2ccc([N+](=O)[O-])s2)=O)CCCCC1(C)C c1(C(N2C(C)CN(C(=O)CC3CCCNC(=O)C3)CC2)=O)nc2cccnc2s1 O=C(N=c1nn[nH]s1)NC(Cc1cccs1)CO N1(C(C2CC2c2c(Cl)cccc2Cl)=O)CC2(CCOCC2)C1c1ccco1 c1(OCC)ccc(C(=O)Nc2cccc(C#N)n2)cc1OC.C12CC(C1)NC2=O C1(NCCC(=O)N(CCNC(c2c(CC)con2)=O)C2CC2)CCN(C)CC1 Cc1nn(CC(=O)NC(C2CCCN2C(=O)CC2CCSC2)C)c(=O)o1 c1(CNC(=O)NC2C(CC(C)C)CCCC2)ccc(F)cc1O C1(NC(=O)CC2CSC2)C(CNC(C2CC2c2ccco2)=O)CCC12CCC2 C1(C(=O)NCC2C(C(=O)NCC(C)NC(=O)OC)C2)CCCCC(=O)C1 C1(NC(CCCC(=O)NC2CC2)=O)CN(C(=O)C=CC2CCC2)CC12CCOCC2 C1(C(=O)NCC2(F)CC(CNC(c3nnsc3C)=O)C2)(OC)CCCOC1 c1(CC2C(C(C)NCC(COCC)O)C2)ccccc1 c1(SC)ccccc1O.c1(CC(N2CCC(c3ccccc3Cl)C2)=O)nc(C)cn1C c1(C(=O)NC2C(C)(CNC(c3csc(CO)n3)=O)CCC2)ccnc2[nH]cnc12 c1(C(=O)NC2CCN(C(CCc3ccc(C(=O)OC)[nH]3)=O)C2)ccc(Cl)c(C)c1 N1(C(C2(NC(CC(C)C3CCCO3)=O)CC(O)C2)=O)CCC(C2=NOCC2)C1 C=CCCN=C(NCc1cc(C)c(C)s1)NC(C)C1CC1 N1(C(c2cc(C)c(C)o2)=O)CC(C2CCN(C(C3CCOC3(C)C)=O)CC2)C1 C1(N(CC#C)C(C2CC2CC(C)C)=O)CCN(C(C2(CC#N)CCCC2)=O)CC1 c1(C(=O)NC(C)C(=O)NCCCNC(C2C(Cl)(Cl)C23CC3)=O)ccccc1Cl N1(C(CCOCC)=O)CC(NC(c2nscc2C)=O)C(n2ccnn2)C1 CCCC(C(=O)N1CCCCC1CNC(=O)C(C(C)CC)OC)S(N)(=O)=O CC1CN(C(=O)C=Cc2cnc[nH]2)CC1NC(=O)CCOc1cccc(F)c1 Cn1ccc(-c2noc(C3(C4CCNCC4)CCC3)n2)n1 Nc1cnc(C(=O)NCCCC2CCCCN2C(c2cnns2)=O)c(Cl)c1 c1(C(=O)NC(C)CCNC(=O)C(c2ccccc2F)O)cccc(P(C)(C)=O)c1 CC(=Cn1ccnn1)C(=O)NC1COCCC1NC(=O)CC1CCC(F)(F)CC1 C1(C(=O)OCC(C)CNC(=O)OC(C)(C)C)CCc2nn(C)cc2C1 N1(C(CC(CC)(C)NC(=O)CCOC(C)C)=O)CCC2CC2(OC)CC1 CC(C)C(CCN(C(=O)CCc1cc[nH]n1)C)NC(C1(O)CCCC1)=O C1(CNC(CCSC)=O)CN(c2nccc(C(C)(C)C)n2)CCCO1 C(=O)(C(O)C(F)(F)F)NC1CC(C)(CNC(c2ccc(F)c(Cl)c2)=O)C1 N1(C(C2C(CC)N(C(c3ccc(F)cc3)=O)CC2)=O)CC(OC)CC(C)C1 C1(C(=O)NCCCN(C(C2C(C(=O)OC)C=C2)=O)C)CCCCN1C Cc1ccc(C(C)(C)C(=O)NCC2CN(C(=O)C3=CCC3)C3CC23)cc1 c1(CC(=O)NC2CCC(NC(C34CCCC3C4)=O)CC2)c[nH]c2cnccc12 Cc1ccc(S(=O)(=O)NCC(N2CC3CCC(C2)C3O)=O)c(C)c1 c1(CCNC(C2CC2F)=O)ccc(CNC(C2CC(F)C2)=O)cc1 C(CCF)(C(=O)NCCCc1nccs1)NC(C1C(C)OCC1)=O c1(C(N(CC(CC)NC(c2cc(C(CC)CC)no2)=O)C)=O)nnc(O)cc1O C(=O)(C(=O)NC1CC1)N(CC(=O)N(CC(C)CO)C)CC#C.OCC c1(C(N2CC(O)(CC)C2)=O)ccc(CNC(=O)CSc2ccccc2)cc1 C1(C(N2CCC(COC)(CNC(=O)C(C)O)CC2)=O)CC(C(C)(C)C)=NO1 C1(C(=O)NCCc2nnc(C)s2)CC(C)CN(C(C2C=CC=CC=C2)=O)C1 C=CCN(OC)C(=O)C1CC(C)CN1C(C12C(=O)C3CC1C2C3)=O C1(C(N(CC(O)CO)CC)=O)CC12CCN1C(CCO2)C(C)(CCCOC)C1=O c1(OC)ccnc(OC)c1C(=O)NC1CCN(C(C2C(C)C2(F)F)=O)C1 C1(NC(c2cc(CC)on2)=O)COC2C(NC(c3csnc3OC)=O)COC12 N1(C(c2c(C)cnn2C)=O)Cc2nccn2CC(NC(=O)CCc2ccoc2)C1 c1(SCCC)cccc(C(=O)NC2CN(C(=O)C=NOC)CC2C(F)(F)F)c1 S(=O)(=O)(c1cscc1F)N(C)C.c12ccccc1SC(=O)C2 C1(C(N2CCC(CC=C)(C(N3CC(CO)C4(CC4)C3)=O)C2)=O)CC2(CCO1)CC2 C1(CC(=O)NC(C=C)(C)CC)CC2(CC2)CN1C(=O)CSC(C)(C)C c1(OCCC(=O)N(CCNC(C(CC)COC)=O)C(C)C)ccc(Cl)cc1Cl C(c1cnc2ccccc2c1)=CC(=O)OCC(c1cnn(C)n1)=O C1(NC(CSC(C)C)=O)CN(C(c2cnc(N)c(Cl)c2)=O)CC1S(C)(=O)=O C(=O)(CCC(F)F)NCC(CNC(=O)Cn1ccc(C(F)(F)F)n1)O [N-]=[N+]=NC1CC(C(=O)NC2CC3CCC2O3)N(C(c2ccc(C#N)cc2)=O)C1 Cc1ccc(-c2ccc(C(=O)NC3CC(F)(CNC(c4ccsn4)=O)C3)s2)s1 C1(C(=O)O)CN(C(=O)CC2CCCC(F)(F)CC2)CC12COC2 c1(C(N2CCC(CNC(c3cncs3)=O)C(F)(F)C2)=O)ccc2nc(O)[nH]c2c1 C(=O)(C1=Cc2ccccc2C1O)NC1C(C)(C(C)C)C1 C1(N(CC(=O)NC)C)CCN(C(=O)C(C)n2cccn2)C1(C)C c1(OC(C)C)c(C(c2nnnn2CC2CCOC2)NC(C)(C)CF)cccc1Cl C1(NC(CN(c2ncccn2)C)=O)CC2CC(C1)N(C(=O)Cc1ccc(Cl)s1)C2 C1(NC(c2nc(C)oc2C)=O)CCN(C(=O)CSc2nnnn2C)CC1C C#CCC(O)C(=O)N(C)CC1CCCC1NC(=O)CC1CCOC1=O N1(C(C(c2ccccc2Cl)C)=O)CC2CC2(CNC(c2ccsc2C#N)=O)C1 C1(CC)CN(C(=O)C(c2ccccc2F)O)CCC1NC(C1(Br)CC1)=O C1(NC(CC2(OC)CCCC2)=O)CC(CNC(C2CCC(=O)N2C(C)C)=O)C(O)C1 Cc1ccc(CC(=O)NCCN(C(=O)CC2CCCC(C#N)C2)C)c(Cl)n1 N1(C(C(CCOC)C)=O)CCN(C(c2cn(CCCF)nn2)=O)C(C)C1 Cc1cc(C(c2nnnn2C2COC2)Nc2cn(CCO)nc2C)sc1C C1(C(=O)NCC2(CN(C(=O)C=C3CCC(C)C3)C)CC2)(OC)CCC(C)(C)CC1 c1(OC)ccc(Cl)c(C(=O)NCCC2CCCCN2C(c2cccnc2C)=O)c1 N1(C(C(CC(C)C)O)=O)CCCCCC(NC(c2ccc3ncnn3c2)=O)C1 c1(NCCCCOC)cc(=NCC2CNC(=O)CO2)[nH]c(C(F)(F)F)n1 c1(C(N2CC(F)CC(NC(C(C=C=C)C)=O)C2)=O)ccc2cc(O)ccc2n1 CCCCCC(O)C(=O)N1CC2C(CNC(C3CCC(CCCC)CC3)=O)C2C1 C1(COC)(CNC(=O)Cc2cc(C)on2)CCN(C(c2ccc(SC)s2)=O)C1 N1(C(C(C)=CC=C)=O)CCC(C(C)C(=O)NCC2CN3CCC2C3)CC1 C=C=CC(C)C(=O)N(CCC(c1cccs1)NC(c1c(C(C)C)cnn1C)=O)C c1(C(=O)NC2CN(C(C(C)NC(C)=O)=O)CC(C)C2)c[nH]c2ccc(Br)cc12 C1(C(=O)NCC2(C(N)=O)CC2)CC12CCN(C(c1ncccc1F)=O)CC2 C1(CCC)CC(C(=O)N(C)CCNC(c2nc(C)n(C)n2)=O)CCO1 N1(C(C(CC2CCCC2)NC(C(CC=C)(F)F)=O)=O)CCC2(CC1)CN(C)C2 C1(CNC(CN(C(C)C)C)=O)CCC(CNC(C2CC3C=CC2C3)=O)CC1 C1(C(=O)OC)CC2(C1)CC(C(N1CCC1CNC(C1CNC(=O)N1C)=O)=O)C2 C(=O)(C(CC(C)C)CC(C)C)NCCN(CCOC)C(c1cc(F)ccc1C)=O c1(C(N2C3(CNC(C(COCC)N=[N+]=[N-])=O)CC(C2)C3)=O)nc(C)c(C)[nH]c1=O N1(C(C(C)OCCOC)=O)CCCC1C1(NC(=O)C(C)(C)C)CC1 c1(C(N(CCCNC(c2cc(C(CC)C)no2)=O)C2CC2)=O)cc(O)ccc1C S(=O)(=O)(c1cccc(Cl)c1)N1CC(CC(N2CCC(F)C2)=O)OCC1 C12(CNC(C3C=CCN(C(C4(Cl)CC4(F)F)=O)C3)=O)CC(CCO1)C2 C#CC1(C(=O)NCC2(N(C)C)CCC2)CCN(C(=O)CC(C)(O)C=C)C1 N1(C(N)=O)CC(C(=O)NCCNC(C2CC(O)C2)=O)C(O)C1.C1(S)CC1 c1(C(N(CC(CC)NC(C2CC2c2ccsc2)=O)C)=O)ccc(F)cc1[N+](=O)[O-] C1(NC(c2cc(CC)no2)=O)CCC2(CCN(C(C3(C(F)F)CC(=O)C3)=O)C2)C1 c1(C(C)C)conc1CC(N1CCC(CNC(c2cc(C3CC3)[nH]n2)=O)C1)=O N1(C(C(=O)Nc2ccc(C)cc2)=O)CC(C)N(C(c2cccc(Cl)n2)=O)CC1C C1(CC)CN(C(c2ccnc(OC)c2)=O)CCC1NC(=O)CC(=O)NCC1CC1 C(C(C)N=c1[nH]c(Cl)nc(C)c1F)NC(Cc1ccc(C)cc1Cl)=O c12n[nH]nc1C(=O)N2.C(=O)(C(C)(C)OC)N.C1(CN(CC)CC)CC(SCC)C1 N1(C(c2cc(CC)c(C)s2)=O)CCCC1C1CCCCN1C(=O)COC(C)(C)C C(CC(=O)NCCCCCC(C)C)(C(F)F)NC(c1ccc(C(C)=O)[nH]1)=O c1(CC)ccc(C(=O)NCC2CC(NC(=O)C(C)(O)CC(C)C)C2)cc1[N+](=O)[O-] S(=O)(=O)(c1ccc(Cl)cc1Cl)N1C2CN(C(c3cc(Br)cnc3F)=O)CC21 CCC(O)CC(=O)NC1CCN(C(c2nc(Cl)sc2C)=O)C1 C1(CC(N2C(CC)CC(C)C2)=O)CN(C(c2ccc([N+](=O)[O-])o2)=O)CC1(C)C N1(C(CC(C=C)CCC)=O)CCCCC2(C1)CN(C(=O)CC(F)(F)F)C2 C1(C(N(CCCN(C)C)C)=O)CN(C(=O)Cn2cc(CO)nn2)C(C)(C)C1 c1(COC)cc(C(N2CC(O)(C(C)NC(=O)CCCc3csc(C)n3)C2)=O)n[nH]1 Cc1cccc(C(=O)NC(C)Cc2cn(Cc3ccc(C(=O)O)o3)nn2)c1C c1(C(N2CC3CN(C(=O)OCc4ccccc4)CC3N2)=O)cc(Cl)c(F)cc1Cl N1(C(c2cc(SC)oc2)=O)CCC2(C=C(C(=O)NC(c3c(C)noc3C)C)C2)C1 c1(C(N(C(C)CNC(=O)C2=C(C)CCC2)CC)=O)c(F)ccc(F)c1O CCC(C)CCCCC(=O)NC(CCCOC)C(=O)N(C)CC1CCCCCC1 c1(C(=O)NCCC(C)NC(=O)CC2COC(=O)C2)ccnc2[nH]cnc12 c1(C(C)C(=O)N2CC(OCCNC(C3CC34CCC4)=O)C2)ccccc1Br C(=O)(C(CO)c1ccccc1)N(CC(C)(C)NC(=O)C(N)=O)C n1(CC(c2ccc(Cl)cc2)C)cc(C2CC2)ccc1=O C1(CC2(CNCn3cc(C(C)(C)C(=O)O)nn3)CC2)COc2ccccc2O1 c1(OC)cccc(NC(=O)C(c2nocc2C)N2CC(N(CC(C)C)C)C2)c1 Cc1ccc(OC(C)C(=O)NCCCN(C(c2cnnn2C)=O)C2CC2)cc1 CC1(C(N2CC3C(C(=O)NCc4cccc(Cl)n4)C3C2)=O)COC(=O)N1 c1(CCC)cc(C(=O)NC2CN(C(c3cnc(C(F)(F)F)s3)=O)CC2C)nn1C C(=O)(C1=CCCSC1)N1CCC(CCCCCNC(c2c(C)ocn2)=O)CC1 N1(C(CSCC=C)=O)CC2CCCC(C1)N2C(C1CC12CCOCC2)=O c1(-c2c(C(=O)NCC(CNC(CC3(C)CCCO3)=O)O)c[nH]n2)ccccc1Cl C12(CC(=O)NCCOCCCNC(=O)Cc3ccnnc3O)CCC(CC1)CC2 C1(NC(c2c(C(C)C)occ2)=O)CCC2(CCCN(C(=O)Cc3cncs3)C2)C1 c1(C(=O)NC(CNC(C=C(CCC)C)=O)(CC)CC)nc2n(c1Br)CCC2 c1(OCC(C)C)ccc(C(N2CC(O)(CCNC(C3(C)CSC3)=O)C2)=O)cc1 C1(NC(=O)CCSc2ccccn2)(CNC(=O)C(F)F)CCc2ccccc2C1 C1(CC(N2CCC(N(C(=O)CCN3CCCCC3)CC)C2)=O)CCS(=O)(=O)C1 C(C=CC(=O)NC1(CNC(=O)CNS(N)(=O)=O)CC1)(CC)=CC C1(C(=O)OCC)CCNCCC1NC(=O)NCCOc1cc(Cl)ccc1OC N1(C(CCC(=O)OC)=O)CCC2(CC1)CC(C)N(C(c1cnccc1OC)=O)C2 C(CC(F)(F)Cn1cc(CCO)nn1)CNCCCC=C C1(CNC(C(C)NC(CC)=O)=O)CC2CN(C(=O)C=C(C)C(F)F)CC12 CC1(C)CC(O)CCN1CC(=O)NCC1(c2c(Cl)cccc2Cl)CC1 Cc1n[nH]c2cnc(C(=O)NC3CN(C(C4CC5CCCCC45)=O)CC3C)cc12 n1(C(C)C)ccnc1C(N1CC(C)(CCC(=O)NCC2(CO)CC(C)C2)C1)=O S(=O)(=O)(c1ccc(Cl)cc1Cl)N1CCC2CN(C(C=CC)=O)CC21 C1(c2cn(CC3CC(CNC4CCCO4)C3)nn2)(N(C)C)CCOCC1 C(C)(C(O)C(=O)NC1CC(NC(c2cccc(N)n2)=O)C1)OC N1(C(CCN(C)CC)=O)CCC(CNC(=O)C=Cc2cn(C)nn2)C1(C)C c12ccccc1Sc1ccccc1NC2=O.C(C(C)C(=O)N(C)C)OC n1(CCC#C)c(N2CCC(Oc3ccccn3)C2)nnc1CC1CC1 C1(n2c(-c3ccc(C4CC4)o3)nc(-c3ccc(OC)nc3)n2)CCCC(F)(F)C1 c1(C(C(=O)NC(C(C)NC(=O)C=CBr)CO)(C)C)ccc2c(c1)OCCO2 C1(CNC(CC(CCC)O)=O)CCN(C(=O)Cn2ccnc2C)C12CCC2 c1(CNC(CC(=C=C)C)=O)c(C)nn2c1CN(C(c1csc(C(C)C)n1)=O)CC2 C(=O)(C1=C(Cl)CCCC1)NC1(C(N2CC(CC(C#C)C)C2)=O)CCCCC1 Cc1onc(CC(=O)NC2CC(C)N(C(C3CCCOC3)=O)C2)c1C#N c1(C(=O)NC2(CC)CCN(C(c3cc(C)n(C)c3)=O)CC2)cc(F)c(C)cc1F c1(NCc2cncc(OC)n2)nccc(=NCC2=CCCOC2)[nH]1 Cc1nc(-c2cccc(Cl)c2)[nH]c1C(=O)NC1CCCC1NC(=O)C1=COCC1 N1(C(c2nc(C)[nH]n2)=O)CCCC(C2CCCCN2C(=O)CC2CCN(C)C2)C1 c1(C(N2C(C(=O)NCCC(C)N(CCC)C)C(C)CC2)=O)cnc(O)c(C)c1 C(CCC(C)(C)C(=O)N1CC2CCC(CNC(=O)C3=C(Cl)CCC3)C2C1)OC C(=O)(C1=CC2CCC(C1)C2)N1CCC2(NC(C(N=S(C)(C)=O)=O)=O)C(C1)C2 Cc1ccn(CC(=O)NCC2(CNC(c3cncc(Cl)c3Cl)=O)CC2)c(=O)c1 Cc1cn2c(C(=O)NCC(C)(O)CNC(C3CC3C)=O)cnc2s1 N1(C(C2CCCN(C(CCc3cncc(C)c3)=O)C2)=O)CC2COCC2C1 N1(C(C(c2ccc(C)o2)C)=O)CC=CC(NC(c2ccc(Br)s2)=O)C1 c1(NC(=O)CCCCCl)ccc2[nH]ccc2n1 N1(C(COC(C)C)=O)CCCC2C1CCN2C(=O)Cc1csc2nccn12 C=C(C)C1OCCC1C(N1CCC(CCC(N2CCCC2C(O)CO)=O)C1)=O c1(C(N(C(CCNC(C(Cc2c(C)nc[nH]2)O)=O)C)C)=O)cc2ncccc2o1 Cc1cccc2cc(C(=O)NC3C4CCN(C(=O)CC(C)(C)O)C34)oc12 N1(C(c2cc(SC)oc2)=O)CCCC(C(C)(C)C(=O)NCC2(O)CC2)C1 c1(C(N(CC(CNC(Cn2ncc(C)c2)=O)O)C)=O)cc(F)c(Cl)cc1F Cc1ccc(Cl)c(OCC(N2CC3CC3(CNC(C3CCC(=O)N3C)=O)C2)=O)c1 C(=O)(CCC1=CCc2ccccc21)N1CCC(NC(c2coc(Cl)n2)=O)C(F)C1 c1(CC(=O)NCc2csc(CNC(c3cnn(CCF)c3)=O)n2)ccc(Cl)cn1 c1(C(=O)NC2CN(C(C)(C)C)C(=O)C2)cc(Cl)c(Cl)c(C(N)=O)c1Cl c1(CC(=O)NCC2CCN2C(C2C=CCC2)=O)ccc(-c2ccccc2)nc1 C1(CNC(C2(CC)CCOCC2)=O)CN(C(C2(CC)CCNC2=O)=O)CC12CC2 Cc1cc(Br)cc(C(N2CCOCC2C2CCC2)C(=O)NC2CC2)n1 Cc1cc(NC(=O)C2CC2)sc1C(=O)NC1CN(C(=O)Cn2cnnn2)CC1F N1(C(C(CC)OCC)=O)CC2(CCC(NC(=O)C(=Cc3c[nH]cn3)F)CC2)C1 c1(SC)ncc(C(=O)NC2CC2NC(=O)COc2ccc(C(N)=O)cc2)n1C c1(C(=O)NC2CCC(c3cncc(C(=O)O)c3)CC2)ccn2cnnc2c1 c1(CC(=O)NC2CCC(NC(CCCC)=O)C2)ncn2c1CCC2 C1(N(C(C(C2CCC2)OC)=O)C)CCCCN(C(c2ccc(C(N)=O)cn2)=O)C1 C1(CC(=O)NCc2c(C(N(c3cccc(O)c3)C)=O)n(C)nc2)CCCC2CC12 C(C(C)C)(C(C)C)NC(C1(NC(CN(C(=O)OCC)C)=O)CSC1)=O.OCC c1(NC(C2CCN2Cc2cc(F)c(F)cc2Br)=O)cc(Cl)c(O)cc1Cl CC1CC(NC(=O)Cc2cncc(F)c2)CN1C(=O)COC1CC=CC1 c1(C(N2C(CCOC)CN(C(c3cc(Cl)no3)=O)CC2)=O)cc(C)c(C)cc1C c1(C(=O)NCC2C(NC(C(C)NC(C)=O)=O)CC2)ccc(S(=O)(=O)NOC)cc1 C=CC(CC)CC(=O)N(CCCNC(=O)Cc1ccc(CC)c(F)c1)C c1(CNC(C2(C=C)CCC2)=O)cc(C(=O)NCC(C2CCCC2)O)ccn1 C12(C(=O)NC3CN(C(CNC(=O)CC(F)(F)F)=O)CC3O)CCCC(C1)OC2 CC#CCCCC(=O)NCC(C)(C)C(=O)N(CC(=O)NC)CC c1(C(N2CC(C3N(C(CC=C)=O)CCC3)(O)C2)=O)cc([N+](=O)[O-])nn1C C(=O)(CCCC(=O)N1CCC(=CCNC(=O)C(O)C2CC2)CC1)N(CC)CC N1(C(c2scc(C)c2)=O)CC(NC(c2cc3ccsc3s2)=O)CC12CCOCC2 C1(CNC(CC)=O)CN(C(c2cccnc2OC(C)C)=O)CC1C CC1=C(C)CC(C(=O)NCc2cc(C)c(C(=O)NCc3cccnc3C)o2)CC1 C12(CNC(CCOCCNC(c3c(CC)n(C)cc3)=O)=O)CCC(CC1)OC2 N1(C(CCC)=O)CC(NC(=O)CCC2CC2(Cl)Cl)CC2(CCC2)C1 N1(C(C2C(C)(C)COC2)=O)CC2CC1CN2C(=O)CCOCC(F)(F)C(F)F C12(NC(=O)CNCC3(O)CN(C(=O)CC4C=CCC4)C3)CC3CC(CC(C3)C1)C2 N1(C(c2nc(CCC)oc2)=O)CCC(C)(C)C(NC(c2ccc(OC)cc2)=O)C1 CCCCCC(=O)N(CCC(=O)NCCC(=O)N(C)C)C1CC1 c1(CNC(C2N(C(Cc3c(C)scc3)=O)CC2C)=O)ccc2c(c1)CC2 CC1(C)CC(CO)N(C(c2ccc(CNC(C3CC3[N+](=O)[O-])=O)nc2)=O)C1 C(=O)(CCC(C)O)NC(CNC(CCN(CC)CC)=O)C(C)C c1(C(N(CC)CC2CCOCC2)=O)ccc(-n2cc(CCC#N)nn2)c(C)c1 Cc1ncc(C(=O)NC(Cc2ccoc2)C(=O)NCC(C)CO)n1C C1(C(N2C3CC(C(N4CCCC5(CC5)C4)=O)C2CC3)=O)C2Sc3ccccc3C12 N1(C(C(CC)n2cccn2)=O)CCC2(CCCN2C(=O)CCNC(=O)CO)C1 N1(C(C2C(C)=CCC=C2)=O)CCCCC(N=c2nc[nH]cc2C#N)C1 c1(N(C)C)nc(Cl)c(C(=O)NCCCCCNC(C2(CO)CCOC2)=O)s1 C1(NC(c2n(CCCC)ncc2)=O)CC(O)CN(C(=O)CC2CCC=CCC2)C1 N1(C(C(CC)(F)F)=O)CCCC(F)(C(=O)NCCNC(=O)NCC)C1 N1(C(=O)Nc2cccc3ncsc23)CC2(CCCN2C(=O)CC2CCCC2)C1 c1(COC)cc(C(=O)N(CC(C)NC(c2snnc2C2CC2)=O)C)n[nH]1 C1(CNC(=NCC23C(C)(C2)C3)NCC(F)F)OC(=O)CC12CCC2 C1(NC(=O)C(F)C2CCOC2)CC1C1CCCN(C(c2c[nH]cc2C2CC2)=O)C1 N1(C(c2ccc(-c3ccccc3)o2)=O)CC(NC(C23CC(CO2)C3)=O)C(O)C1 C1(CC)(Nc2nccc(CO)n2)CCN(C(C2(CO)CC2)=O)CC1 CCC(C)(COC)C(=O)NN1CCCC1C(=O)NCCC1CC(C)C1 C1(NC(=O)CCN2CCCCC2)CCCC12CN(CC(=O)N(CCO)CCO)C2 N1(C(C(C=C)c2ccccc2)=O)CCC(C)C(NC(=O)CC(C)(C)CC)C1C Cc1cnc(C(C)(C)NC(C2CSCN2C(C2CCCN2C)=O)=O)[nH]1 N1(C(N2CC(C)C(C(=O)OC(C)(C)C)C2)=O)CC(C)C(F)(F)C1 C=CCC(CC(F)F)NC(C1C(CC)CCCN1C(=O)COC1CCOCC1)=O CC(C)CCC(C(=O)N(C1CC(OC)C1)C)NC(=O)CCC(C)(C)N(C)C N1(C(Cc2c(C)ccs2)=O)CCOC(CN(C)C(C2CCC(=O)N2C)=O)C1 N1(C(C(C=C)C)=O)CCN(C(C2CC3(CCC3)C2)=O)CC(C)(F)C1 C1(NC(C2(CCCC)CCCC2)=O)CCC(C)N(C(=O)Cn2ccnn2)C1 CC1CN(C(=O)C(C2(O)CCCC2)F)CC1NC(=O)Cn1cc(C#N)cn1 Cc1cccc(CNC(=O)C(C)(C2CC2)N(C)C(c2cncc(CO)c2)=O)c1F N1(C(C2(C(N)=O)CCC2)=O)CC23CCCC2(C1)CN(C(=O)CC1CC1)C3 C(=O)(C1CCc2ccccc21)N1C(C(=O)NCC(COC)(C)C)CSCC1 CC1(C)CC(C(=O)NC2CNC(=O)C23CC3)CCN1C(=O)C=CCO Cc1[nH]cc(C(=O)NC2CN(C(=O)C(C)C3(O)CCC3)CC2(C)C)c(=O)c1Cl C1(C(=O)NC(CN(C(c2occ(C)c2)=O)C)(C)C)CC12CC(O)C2 C#CC1(C(=O)Nc2ccc(OC)nc2)CCN(C(=O)C#CC2CC2)CC1 C(=O)(CCCCNC(C1CCCCN1C(c1ccc(F)s1)=O)=O)OCC N1(C(N2CCN(CCCOC)CC2)=O)CCC2(CC1)CC(C1CC1)=NO2 C1(OC)CN(C(=O)CCCCC2CC2)C(C)(CNC(=O)Cn2cc(CO)nn2)C1 C1(CNC(C2COC3COCC23)=O)CCC2(CN(C(=O)CC3CCOCC3)C2)O1 Cc1ncc(N)cc1C(=O)NCC=CCNC(=O)Cc1n[nH]cc1Br c1(C(=O)NC2CCN(C(C(C(CC)O)(F)F)=O)C2)sc2cccc(F)c2c1Cl C1(NC(c2cnc(S)[nH]2)=O)CC2CC(C1)N(C(c1ncsc1Br)=O)C2 Cc1nccc(CNC(=O)C=CCC(C)(C)NC(=O)Cc2cc[nH]n2)n1 C#Cc1ccc(C(N2CCCC(C)(N(C)C)C2)C(=O)NC2(C)CC2)cn1 c1(C(N2C(CNC(C(C=CC)O)=O)CCC2)=O)cnc2cnn(C)c2c1 C1(C(=O)Nc2scc(C)c2C(N)=O)CC12CCN(c1ncnc(C)c1Br)C2 N1(C(c2cccc(NC)c2)=O)CCCC(NC(=O)C=CS(C)=O)CC1 C(=O)(C=C1SCC(=O)N1C)N1CC(NC(C(CC=CCC)C)=O)C(OC)C1 C12(C(=O)NC3C(C=C)OCC3)COCC1CN(C(=O)Cc1cccc(F)c1)C2 c1(N2C(C)(CNC(C(C)NC(C)=O)=O)CCC2)ncc([N+](=O)[O-])cc1F CCCC(C)(C)C(=O)NCC1(O)CCN(C(C2CCSC2)=O)C1 C(=O)(C(=O)C(C)CC)NC(COCC)C(=O)N1CCC1C(C)O C1(OC)CC(CCNC(=O)CN2CCC2C)N(C(C2CCC=CCC2)=O)C1 n1(CC=C)nc(-c2ccc(OC)nc2)nc1-c1cccc(C2COC2)c1 c1(CC(=O)N(CC(C)N(C)C(C2CCC23CCC3)=O)C)c(F)cccc1F c1(NC(c2c(NC(c3c(C)scc3)=O)ccs2)=O)ncc(Br)nn1 C1(C(=O)NC2(C(=O)NCC(C)C)CSC2)CC2C(C1)C2(C)C C1(C(=O)NCC2CCCCC2)C2CN(C(c3ccc(CCO)cc3)=O)CC12 C(=O)(CCCCC(C)(C)C)N1CC(NC(C(CCCC)CC)=O)CC2(C1)CC2 C1(CCC=C)(C(=O)NCC(O)CO)CN(C(=O)Cc2ccc(Cl)s2)C1 C(C1CCCC1)=C(C)C(=O)NC(C)C(=O)NC(C)Cc1nn[nH]n1 c1(CN(C(CN2CCC(CCCC)C2)=O)C)ccccc1Cl C1(NC(c2cc(C)nn2C)=O)CCN(C(c2sc(=N)[nH]c2C)=O)C(C)C1 N1(C(CNC(=O)OC)=O)CC2CCC1CC2NC(C1CCC(F)(F)C1)=O N(C(=NCCN1CCOCC1)NCc1ccoc1C)CC1(OCC)CCSCC1 N1(C(Cc2c(C)nsc2)=O)CC2CC1CN2C(c1sc(=N)[nH]c1C1CC1)=O Cc1nncc(C(N2CCC(CCCNC(C3(Br)CC3)=O)CC2)=O)c1C C1(NC(c2c(C)c(Cl)ccc2)=O)CCN(C(=O)C2=CCCO2)CC1(C)C c1(C(N(CCCNC(=O)C(C)c2cc[nH]n2)C(C)C)=O)cc(N)nc(Cl)c1 C1(CCC(=O)NCC2N(CC(=O)N(C)CC)CC2)CCCN1C CCC(C(=O)NC(C1CCN(C(c2[nH]nnc2C2CC2)=O)C1)C)c1ccccc1 C1(CNC(c2c(C)nns2)=O)CN(C(=O)CCc2nncs2)CC1O C(=O)(C(N=[N+]=[N-])C(C)C)N1CCC(CC)CC1C(=O)N(CC(F)F)C c1(C(N2CC(NC(c3cnc(CC)[nH]3)=O)C(C)CC2)=O)ccc(Cl)cc1[N+](=O)[O-] C1(NC(C2(C)CN(C(C3CCC(CC)O3)=O)C2)=O)CN2CCC1(C)CC2 CC1(C)CCCC(NC(c2ncoc2CNC(C2CC3(CC3)CO2)=O)=O)C1 C1(NC(C(c2ccc(C)cc2)(F)F)=O)COCCN(C(c2cn(C)cc2C)=O)C1 C(CC(=O)Nc1ccc(OC(F)F)cc1)(C(F)(F)F)N1C(C)CCCC1 c1(N(C)Cc2ccc(OC)nc2)nc(N2CCC(F)CC2)nc2c1COCC2 c1(N2C(=O)CC(NC(CCC#C)(C)C)C2)ccc(Cl)c(Cl)c1 C1(C(N2CCN(CCNCC(F)(F)F)CC2)=O)CCOC12CCOCC2 c1(C(c2nnnn2C2(C)CC2)NCC2C(CCC)C2)cnn(-c2ncccn2)c1 C1(C(N(C2CCN(C(=O)CC3(O)CCCOC3)C2)C)=O)CCC(C(F)(F)F)CC1 Cc1c(C(N2CCOCC(CNC(C3(C)CCCN3C)=O)C2)=O)sc2cncn12 CC1CN(C(c2csc([N+](=O)[O-])c2)=O)CC1(C)CNC(=O)C(c1ccccc1)F C1(CC(=O)NCC(C)C2CCC2)CCCCN1C(C1OC2CCC1C2)=O c1(C(N(C(C)C)C(C23CC(CSc4ccccc4)(C2)C3)=O)=O)ccc(N)cc1Cl N1(C(C2C(=C)C2)=O)CC2CCC1CC2NC(=O)C(C)(C)CF CCCC(C(=O)NOCCCN(C)C)NC(c1cnc(O)n1CC)=O C1(C(N2CC(COC)(NC(c3cc[nH]c3C)=O)C2)=O)Cc2cc(F)ccc2O1 C(=O)(C(CC(C)C)C(N)=O)NC(C(C(=O)NC1(CCC)CCC1)C)C Cn1nc2c(c1C(=O)NCCCN(C(=O)CC1CC(C)(C)CO1)CCO)CCCC2 CC1(C#CC(=O)ON2C3C(=C4CCC(=O)N(C)C4=O)C(CC3O)C2)COC1 c1(C(N(C2CCCN(C(c3ccc(C=C)cc3)=O)C2)C)=O)cc(S(N)(=O)=O)cs1 CCCC(CC)CCC(=O)NC1CN(C(c2ccc(C#N)o2)=O)CC1O N1(C(C(CNC(CCCCC=C)=O)C(C)C)=O)CCC(C2CCC2)CC1 C1(CNC(C2CSCC(=O)N2)=O)CN(C(c2cocc2Br)=O)CCO1 C(=O)(CC1=CCN(C)CC1)NC(C)C(c1ccccc1)NC(C1(CCF)CC1)=O Cc1cc(F)c(C(=O)NC(C)CCNC(=O)CN(CC(C)(C)C)C)cc1Br C1(C(=O)NCC(C)N(CC)CC)CCN(C(c2ccoc2)=O)C1 C1(C(=O)NCc2cc(C)cc(C)c2)CC2(CCN(C(C3(C)CCC(=O)C3)=O)C2)C1 c1(C(=O)NC2C=CC(CNC(c3ccc(OC)s3)=O)C2)ccc2ccccc2n1 CC(=O)C(C)(C)CC(=O)NC(Cc1cc[nH]n1)C(=O)NCC1(C)CCN(C)C1 c1(OC)ccc(F)c(CC(=O)NC2CN(C(C3(C)CS(=O)(=O)C3)=O)CCC2O)c1 c1(C(=O)NC2C(OC)COC2)oc(CNC(C2(CO)CCC2)=O)nc1C C#CCC(C(=O)N(C1(C)CC1)C)NC(C1CCCN1C)=O C1(F)(C(=O)NCC(C)(C2CCC2)NC(=O)Cc2cnc[nH]2)CC1(F)F CC(O)CCCCCC(=O)OCC(N1CN(C)C(=O)C1C)=O C1(NC(C2(C)CSC2)=O)CN(C(C2(C)CCC2)=O)CCC1C(F)(F)F c1(C(N(C)CC2N(C(c3cc(C)on3)=O)CCC2)=O)c[nH]c(=N)nc1C N1(C(CNC(=O)NC)=O)CCN(C(c2cc(O)nc(C)n2)=O)C(C(F)F)C1 CC(C)CCCC(C)C(=O)N(C)CC1CCN(C(C2COC(=O)N2)=O)CC1 C1(NC(=O)CCC2CCC2)CCCC2CN(C(=O)CNS(N)(=O)=O)CC12 CCCC(C)C(=O)N1CCC(F)(C(=O)NCC(c2ccc(O)cc2)O)C1 c1(C(N2C(CC(=O)Nc3cc(C)ns3)CCC2)=O)ccc(C(F)(F)F)c(F)c1C C1(NC(C(CCN(C)C)O)=O)(CO)CCCN(C(=O)C(c2cccc(N)c2)O)C1 N1(C(CC(COC)C)=O)CCCC2(CCC2NC(=O)CCC2CC2(C)C)C1 C1(C(=O)NCc2cc(C(N(CC)CC)=O)no2)CCOC(C)C1 CC1CCN(C(C2CC(NCc3cc(Br)c(F)cc3F)C2)=O)CC1(F)F C1(OCC)CN(C(=O)C(C)N(C)C(C2CCCO2)=O)C1 c1(OC(C)C)ccc(CNC(=O)CC2CC(F)CN2)cc1F C1(NC(C(C)N2CCC2)=O)C(C)CCN(C(c2cscc2C(F)F)=O)C1C C(C1=CCCN(C(C2(F)CCCCCC2)=O)C1)NC(c1ncc[nH]1)=O C(CC(=O)NCc1cccc(CO)c1)(C(C)C)NC(CSCC#C)=O C1(C)(C(=O)NC(C23CCC(CC2)C3)CNC(CCNC(C)=O)=O)CCCS1(=O)=O C1(CC(=O)NCC(CC)(C)O)COCCN1C(C1CC(N=[N+]=[N-])C1)=O C1(NC(=O)CCOCC(F)(F)F)CS(=O)(=O)CC1N=c1ccnc(C2CCC2)[nH]1 N1(C(c2c(NC)snc2C)=O)CC(NC(=O)CCc2ccccc2)CC(O)C1 C1(CNC(CN(C(=O)OC)C)=O)CC(C(=O)N(C)CCN2CCOCC2)=NO1 c1(C(N2C(C(N(C(C(C)C)CO)C)=O)CCC2)=O)cccc2ccoc12 N1(C(C(C(C)C)O)=O)CC(CNC(c2nccc3ccsc23)=O)OC2(CCC2)C1 C(c1ccc(C#N)cc1)=CC(=O)NC1CCC(C)N(C(c2cccc(=O)o2)=O)C1 N1(C(C=C(C)CCc2ccccc2)=O)CC2OCC(NC(=O)C3=CCCS3)C2C1 CCC(O)C(C)(C)C(=O)N(C1(CC(N2CCC(c3cc[nH]n3)C2)=O)CC1)C c1(NC(C(c2cc(O)cc(Cl)c2)N2CCC(C(=O)NC)C2)=O)ccc(Cl)cc1F C1(C(=O)NCC(C)N(C(C(C2CC2)SC)=O)C)CC2(C1)OCCO2 c1(C(N2C(CNC(c3c(CC)non3)=O)C(C)CC2)=O)cncc(S(N)(=O)=O)c1 N1(C(C=Cc2cnc(C)s2)=O)CC(F)(F)CC1(C)CNC(=O)C1=CCCCC1C C1(NC(C=CCC)=O)CCC(N(C(=O)C(C(C)C)Oc2ccc(Cl)cc2)C)CC1 C12(C(N3C(CNC(c4ncsc4C4CC4)=O)CCCC3)=O)CCCN(CCC1)C2 c1(N(C)CCC2(O)CCN(C(=O)CN(C3CCC3)C)CC2)ccccc1[N+](=O)[O-] C12(CNC(=O)Nc3c(C)c(Cl)ncn3)CCC(CC1)C(C)(C)O2 N1(C(c2cnc(C(=O)OC)s2)=O)CCOC(C(C)NC(=O)CC2CCCC2)C1 Cc1[nH]nc2c1CC(C(N1CC3CC(NC(=O)Cc4csnn4)C3C1)=O)CC2 CCCC(C)(CCC)C(=O)NCC12CC(CN1C(=O)C(C)CCC(C)(C)C)C2 Cc1ccnc(NCC(C)(C2CC2)NC(=O)Cc2sc(C3CCC3)nc2C)n1 CC1CN(C(c2c(Cl)nsc2Cl)=O)CCCN1C(c1ccc(C(N)=O)cc1)=O C1(CC(N)=O)CCCCN1C(=O)CC1C=CC(NC(=O)C(c2cccnc2)O)C1 Cc1cc(C(=O)NC2COCC2NC(C2(C)CCC(C)C2(C)C)=O)cc(C)c1N CCC(CCCC(=O)NC(CC)(CC)CO)NC(=O)C(F)CC(C)(C)C c1(C(N(C2CN(C(C(CC=CC)CC)=O)CC2(C)C)C)=O)[nH]cc2c1CCCC2 c1(C(N2CC(C)(NC(C(CC)C(C)C)=O)C2)=O)cc2c(o1)CCCNC2=O C12(C(=O)NC(c3cncs3)C)CCC(CC1)N(C(C1CCOC1C)=O)C2 CCCCCCNC(=S)NC1CC(C(=O)O)C1 c1(CC(=O)N(CC(C)NC(=O)C(=Cc2c[nH]cn2)F)CCO)ccc(Cl)nc1 Cc1ccc(CN2CC3CC2C3C(=O)NCC(C)CN(C)C)c(F)c1 c1(OCC)cc(CNC2CCCN2C(c2ccc(F)c(F)c2)=O)cc(O)c1 C(CC(C)C(F)(F)F)NC(=O)NCC1CC(C)SCC1 C1(NC(c2ccc(C)cn2)=O)CCC2CN(C(c3cc(Cl)cnn3)=O)CC2C1 c1(C(N(CCN(C(Cn2c(C)ccn2)=O)C(C)C)C)=O)cnn2c1CCCN2 N1(C(C(COC)O)=O)CC2(CC(NC(c3cnc(OC)cc3C)=O)CO2)C1 c1(C(=O)NC(C2(O)CN(C(C3CC(F)CN3C)=O)C2)C)c[nH]c2ccc(F)cc12 C(=O)(C1=Cc2ccccc2OC1)N1CCN(C(=O)C=C2CCCCC2)C2C1CC2 Cc1ccn2ncc(C(=O)NC3CC(NC(c4cc(CO)[nH]n4)=O)C3)c2c1 C1(CNC(C2CC(C)C2)=O)CCN(C(C2CCN(S(C)(=O)=O)CC2)=O)C12CC2 C1(C(=O)NC23C(NC(C(C)=C4CC4)=O)CC(CC2)C3)CCn2nnnc2C1 C#CC(CC(C)(C)C)NC(c1[nH]ccc1CNC(C1(C)CC(C)(C)C1)=O)=O N1(C(=O)CC2(C(F)F)CC2)CCCC(N(C(=O)C(C2CCOCC2)O)CCO)C1 c1(C(C)=O)ccncc1NC(C1CCN1C(=O)Cc1cccc(F)c1)=O N1(C(CC2(CC)CCC2)=O)CCC2CCN(C(c3c(C)[nH][nH]c3=N)=O)CC12 c1(NCC2C(NC(C(CC)OC)=O)CCCC2)cc2nncn2c(C)n1 Cc1nc(C(=O)Nc2cn(C)c(C(=O)NCc3ccc(Br)cn3)n2)c(=O)[nH]c1C Cc1ccnc2c1CCN2C(c1cc(Cl)ccc1C(N1CCCC1)=O)=O CCCC(CCC)C(=O)N1CCC(NC(c2c(F)ccc(Cl)c2F)=O)CC(O)C1 C1(CNC(COCC(C)C)=O)C(O)C(O)CN1C(=O)CCNC(C1CCCO1)=O N1(C(CC2N(C)CCC2)=O)CC2CC2(CNC(c2cnc(Cl)s2)=O)C1 C=C(C)C1OCCC1C(=O)NC1C2CC1N(C(c1cnncc1C)=O)C2 C1(NC(=O)Cc2cnn(-c3ccccc3)c2)CCC2CC1CN2C(C1CC1F)=O C(=O)(CC(C(C)C)OC)N1C(CN(C(COCCC=C)=O)C2CC2)CCC1 C1(C(=O)NCC2CCN(C(=O)CSc3nc[nH]n3)C2)CC(c2ccncc2)=NO1 C1(CNC(c2c(C)n(C)nn2)=O)CN(C(=O)CC2CCCOC2)CCN1C N1(C(C=C(C)CCc2ccccc2)=O)CC(NC(=O)CC(C)C)CC(C)(C)C1 C1(C2CCCC2)(NC(C2C(NC(C3CCC=CCC3)=O)CCO2)=O)CC1 c1(NCC(C2CCCN(C(C(C)(F)F)=O)C2)(C)O)ncnc2c1ncn2C1CC1 C=CC1CCCN1C(=O)C(C)(CO)NC(C1COCC1C(N)=O)=O C(=O)(C(O)C(F)F)N1CC(C(C)NC(=O)CCCc2ccncc2)C1 c1(C(c2n(C(CC)C)nnn2)Nc2cnoc2)ccc(S(C)(=O)=O)s1 CC1CN(C(C2OCCC2NC(=O)CC2CC(F)C2)=O)CCC1(F)F C1(C(C)NC(=O)CCSc2cccs2)CCN(C(=O)CC(=O)N(C)C)CC1 N1(C(CN(CCOC)C)=O)CC(C)(CNC(=O)C(c2ccnn2C)O)CC1(C)C c1(C(N(CC(C)NC(=O)CC2(NC)CCOC2)CC)=O)sc(C2CCCC2)nc1C C(=O)(C1=NOC(CNC(c2ccc(C(N)=O)[nH]2)=O)C1)N(CCOCC)C N1(C(C(=O)NCC)=O)CC(C)C(NC(=O)C(c2c[nH]c3ccccc23)=O)C(C)C1 C1(CSC)CCCN(C(c2ccc(Br)cn2)C(=O)NCCCC2CC2)C1 C#Cc1cccc(C(=O)NCC(C)N(C(=O)C(C)OCCN(C)C)CC)c1C N1(C(C(C)OC2CCCC2)=O)CC(O)C(O)C1CNC(=O)C(C)(F)F N1(C(C2CC(=O)NC2)=O)CCCCC12CCCN(C(C1C=CCN1)=O)C2 N1(C(C2C(=O)NCC2)=O)CC2CCN(C(=O)Cn3nccn3)CCC2C1 C(=O)(CC(C)(C)CC(F)F)NCC(C)CNC(c1cnoc1C1CCOCC1)=O c1(CCNC(=O)Nc2cccc(COC)c2)ccc2[nH]ccc2c1 O=C(C1c2ccccc2CN1C(c1csc(Br)c1)=O)NCCCCCCCCO c1(CC)ncc(CNC(=O)Cc2cccc(NS(C)(=O)=O)c2)cc1C C(=O)(C1=CCC2CCC1N2C(c1nccnc1OC)=O)N1CCC(C)(CC)CC1 c1(OCC(=O)N(CCN(C(C)C)C(C2CC(N3CCCC3)C2)=O)C)cccnc1 CCCCCCCCCC(O)C(=O)N1CCCC(NC(c2cncs2)=O)C1C C1(CNC(c2cc(SC)ncc2)=O)C(C)CCCN1C(c1occc1C)=O C(=O)(C(C)CCC(C)(C)C)NCC(C)(CO)NC(Cc1ccc(SC)cc1)=O c1(OC)cncc(CCC(=O)NCC(O)CCNC(C2CC(O)(C(F)F)C2)=O)c1 N1(C(CC(=O)NC)=O)CCC2(CCCN(C(c3cc(C#N)ccc3Cl)=O)C2)C1 N1(C(C(=O)NC(c2cnc(Br)s2)C)=O)CCC(c2ccccc2)CC1C Cc1cc(-c2cccc(C(=O)Nc3nncn3C3CC3)c2)ccc1C=O c1(C(=O)NC(CC)CNC(=O)Cc2ccccc2SC)c(C)nn(C2CC2)c1Cl Nc1c(C(=O)NCCNC(c2[nH]nnc2-c2ccccc2)=O)cccc1F C1(C(C(=O)N(C)CC2CCO2)NC(C)=O)CCCCC1 c1(C(=O)NC2C=CCN(C(C3CCC(C)(C)C3)=O)C2)cscc1S(C)(=O)=O C1(NC(C=C(C)C2CC2)=O)C(CNC(c2cnn[nH]2)=O)CCC12CCC2 c1(C(=O)NCCNC(C)=O)cc(SC2(C(C)C)CC2)cc(N)c1 C(=O)(C(F)C1=CCCCC1)NCC1OCCCN(C(C2(C)CC2(Cl)Cl)=O)C1 C1(NC(C2CC(C)(C)O2)=O)CCN(C(=O)CCCCNC(N)=O)CC1O C1(CC(=O)NCC2N(CC)CCC2)CN(C(=O)CCCF)CCC1C N1(C(c2n(COC)ncc2)=O)CCN(C(C2CCC(C)(C)C2)=O)CCC1C c1(C(=O)NCC(C2CCC2)NC(C2(C)CC=CCC2)=O)cc2n(n1)CC1(CC1)C2 c1(NC(c2c(C)n(C)nc2C(=O)O)=O)nn(C)c2ccccc12 N1(C(C(C)OCC#C)=O)CCCC2(C1)CN(C(=O)C(F)(F)C(C)O)CCO2 C#CCC(C)(C(=O)Nc1cc(C)cnc1O)NC(=O)CC1CCC(C)(C)O1 N1(C(C(CC#C)(C)C)=O)CC2CCC1C1CN(c3cc(O)nc(SC)n3)CC21 c1(C(N2CC(CNC(c3c(C)csc3)=O)OCC2)=O)cc(Br)c(F)cc1F C1(C(=O)OCC)(C(=O)NCCC(C)NC(c2ccoc2Cl)=O)CC=CC1 c1(NC(c2c[nH]nc2C2CC2)=O)ccc(NC(=O)COCC(F)(F)F)cn1 C(CCCCC(=O)NCC1(C)CCCN1C(=O)Cc1ccc(F)cc1C)OC NS(=O)(=O)c1cc(C(=O)NCCCN(C(=O)C(F)(F)CO)C2CC2)co1 n1(C(C)C(=O)N(C2CCCS2)C)cc(C2(O)CSC2)nn1 N1(C(C2C(C)CCO2)=O)CCOC(C(=O)NC(C2CCOC2)CO)C1 N1(C(CC2CN(C)C(C(F)(F)F)CC2)=O)CCC23CCCCC2(C1)C3(F)F N1(C(C(=C)F)=O)CCC12CN(C(c1ccccc1OC)=O)C2 c1(OC)nscc1C(=O)NCc1cc(C(=O)NCCCCCC2CC2)no1 c1(C(=O)NCC(C(=O)Nc2ccc(OC)cc2)OC)ncnc(O)c1F C(CC(C(=O)NC(C)C(O)C(F)F)NC(=O)C(O)Cn1cncn1)OCC c1(C(=O)NCCN(C(c2ncccc2CO)=O)CC2CCOC2)snc(Cl)c1Cl c1(C(=O)NC2CCN(C(C(C)OCC#C)=O)C2(C)C)ccc2c(c1)B(O)OC2 c1(C(=O)NC2(C3N(C(C4C(CC)C4)=O)CCC3)CC2)c(OC)ccc(OC)c1N N1(C(=O)Nc2csc(Br)c2)CC(CO)CC12CCOCC2 CC1(C)CCN(CCNC(c2ccc(CNC(C3CC=CCC3)=O)o2)=O)C1 c1(C(C)=O)ncc(C(N2CCC(C3CCCN3C(=O)CC3CC(C)(C)C3)C2)=O)s1 C1(c2nc(C3C(C)(COC)C3)on2)(c2ccncc2)CCCCC1 c1(OC)ccc(C(=O)NC2CCN(C(c3cnc(F)c(C)c3)=O)CC2F)cc1Br CCCCCCCCC(=O)N1CCOCC1CN(C(=O)C(C)(CC)CO)C CC1(C)CCCC1CNC(c1[nH]ccc1-c1cccs1)=O C=CCCCC(C(=O)NC(CC)C(C)(C)C)NC(=O)COCCF c1(NC(=O)NNC(=O)c2ccsc2)cc(F)c(F)c(F)c1 C(=O)(CCCNC(c1cccnc1)=O)NC(C1CN(C(C23COC(C2)C3)=O)C1)C c1(C(N2C(COC)CN(C(=O)C=CBr)CC2)=O)ccnc2ccccc12 C#CC12CCC(C(=O)NC3CN(C(=O)CC4CCCC4)CC(C)(C)C3)(CC1)CC2 C(CNC(C1(C2CCCO2)CC1)=O)(CCOC)NC(CC1(OCC)CCC1)=O C1(NC(C2C(c3cn(C)nc3)C2)=O)CCCC2CN(C(=O)C(F)C3CCC3)CC12 CC(C)S(=O)(=O)c1ccccc1NC(=O)CC1(C)CCN1Cc1cccnc1Cl N1(C(c2ncn(CC)c2)=O)CCC2(NC(c3ccn4ccnc4n3)=O)CCCC12 c1(CC(=O)NC2CCN(C(C3CC(C)N(C)C3)=O)CC2)c[nH]c2ccncc12 c1(SCCC)cccc(C(N2CC(COC)(NC(=O)C(C)C(F)F)C2)=O)c1 N1(C(CCc2nc(C)c(C)o2)=O)CCCC2CN(C(=O)C(C)O)CC12 C12(NC(=O)CN3CC=CC3)CCOCC1CN(C(c1cccc(CO)c1)=O)C2 c1(OC)ccc(-c2cc(C(=O)NC3C4CN(CC(O)CO)CC34)n[nH]2)cc1 CC(C(=O)NCC1CN(C(C2(C)CC=CC2)=O)C1)S(N)(=O)=O c1(CC(=O)NCC(C)NC(c2cc(SC)oc2)=O)c(C)cc(C#N)cc1C c1(C(=O)NC2C(NC(c3cn(CCC=C)nn3)=O)COC2)cncn(C)c1=O N1(C(CCCOCCC)=O)CCCC(CO)(NC(c2oc(CC3CC3)nc2C)=O)C1 C1(COC)CN(C(c2c(C3CCC3)noc2C)=O)CCN1C(c1cscc1C)=O C(=O)(C1CCc2nccn21)NC1(CC=C)CCN(C(c2coc(C(F)F)c2)=O)C1 C1(C(N2CC(C)CC(NC(c3c(C)coc3C)=O)C2)=O)CCc2nncn2C1 C1(NC(C(C(C)C)OC)=O)CCN(C(c2sc(C(C)(C)C)nc2C)=O)CC1F Cn1cnc(CC(=O)NCC(C2CCOC2)NC(=O)COC2CCC2)c1 c1(C(N2CC(CCNC(C(C(CC)C)O)=O)C2)=O)ccc(F)c(S(N)(=O)=O)c1 c1(CC)ccccc1C(CNC(C1(Cl)CC1)=O)NC(=O)CCCOC CC(C)CCC(=O)NCC(=O)NC1C=CCN(C(=O)CSC2CCOC2=O)C1.O n1(CC)c(CNC(=O)CN(C(=O)CC2CCOCC2)C2CC2)nnc1O C(=O)(C(CC(C)C)OC)NCC12C(CN(C(c3c(CC)nc(C)[nH]3)=O)C1)C2 c1(OC)cc(F)c(F)cc1C(=O)NC1CC1NC(c1cc(CC2CC2)on1)=O c1(C(N2C3CC(NC(c4c(CC)nccn4)=O)C2CC3)=O)ccc(S(C)(=O)=O)s1 C1(c2cn(CCCCC3CC3)nn2)CCN(C)CC1.C(C(O)C(=O)N)=CCCC Cn1ncc(C(=O)NCC2CN(C(=O)CC3(O)CCC3)CCO2)c1Cl c1(N(CCC)CCNC(=O)C(C)OC)ccc(C(=O)OC)cc1[N+](=O)[O-] C1(CCNC(c2cc(C(F)(F)F)no2)=O)CCCN(C(=O)CC2CCOC2=O)C1 CC1CCCCC1(CNC(=O)Cc1cnccn1)NC(=O)CCCN=[N+]=[N-] c1(C(=O)NC2CCC(CNC(c3occ(C)c3C)=O)CC2)ccc2nccn2c1 c1(C(=O)NCC2(N(C(=O)CC3(C(F)F)CC3)C)CC2)cnco1 C1(C(=O)NCCC2CC(NC(c3ccc(=O)oc3)=O)C2)CC2CCC1O2 C(C)(CNC(c1cncnc1)=O)(C(C)C)NC(c1c(CC)scn1)=O C#CCC(C)(C)C(=O)N(CCNC(=O)C(CC=CC)NC(C)=O)CCOC C1(CC)CN(C(=O)C=CCOCCOC)CC1C(=O)Nc1ccccc1Cl CC1(C)CCC(C(=O)NC2C3CN(C(=O)C(C4CC4)C4CC4)CC23)O1 c1(C(=O)NC(C(C)NC(C2CCC2)=O)C)ccncc1C(F)(F)F CC(CN(C)C)C(=O)N1CC(C(O)C(=O)N(C)CCF)C1 c1(C(=O)NCC(CC)(C)NC(C2C=CCC2)=O)cc(C2CCCCC2)c(C)s1 C1(NC(COC2CC(NC(CN(C)C)=O)C2)=O)CC(C)(C)C12CC2 C(CC(=O)NCCC(C)OC)(C(F)F)NC(C1(CC)CC(C)(C)C1)=O C1(C(=O)NCC2(C)N(C(c3cc(C)sn3)=O)CCC2)CCc2ccnn2C1 c1(C(=O)NC2CC(C)(NC(C(N3C(=O)CCC3=O)CC)=O)C2)nccc(C)c1N c1(NC(C2CN(C(c3ccc(Br)c(F)c3)=O)CCN2)=O)ncc(Cl)cc1Br c1(C(=O)NCC2CCN(C(=O)Cc3ccc(Cl)cc3F)C2)ccc(Cl)c(Br)c1 c1(C(=O)NCC=CCNC(C2CCN(C)S2(=O)=O)=O)cc(F)c2ccccc2c1 N1(C(c2c(CC)nco2)=O)CC(NC(=O)CCCCCCSC)C2(CCC2)C1 C1(NC(COC)=O)CCN(C(c2cc(Br)sc2Cl)=O)C(C)C1 O=C(C1=CC2CCCC12)Nc1ccc(C(=O)OCc2cc(F)cc(F)c2)c(Cl)c1 C(=O)(CCCCCS(N)(=O)=O)NCC1(O)CN(C(c2ccc(OCC)nc2)=O)C1 C(=O)(CC(O)CC(C)(C)C)N1CC2N(C(c3n(CC)ncn3)=O)C(CC2)C1 C=C(C)CCN=C(NCC(c1ccco1)O)NC(c1ccc(Cl)c(F)c1)C N1(C(c2cnn(C(C)CC)c2)C(=O)NCC)Cc2ccccc2C1CCO CC(C(=O)NCC=CCNC(C1(C)CC1C(F)(F)F)=O)P(C)(C)=O N1(C(C2C(C)OC(C)C2C)=O)CCC(NC(=O)CCCCCO)C2(CCC2)C1 C1(CC)COCCN(C(CC2CCCC(NC(=O)CC(=O)OC(C)(C)C)C2)=O)C1 N1(C(C(CC)SC)=O)CCCC1(C(=O)N(C)CCOC)CC C12(CNC(=O)CC3=CCCC3)CCCCC1N(C(=O)COc1ccccc1)CC2 N1(C(C2CN(C(C)=O)C2)=O)CCC(O)C(NC(c2c[nH]nc2C2CC2)=O)C1 N1(C(c2n(CC)nc(C)c2)=O)CC(CNC(c2cnc(SC)s2)=O)CC1(C)C N1(C(=O)CC2CCC3(CCC3)O2)CCCCC2(C1)CN(C(C1CCCS1)=O)C2 C1(NC(C(CN(C)C)O)=O)CS(=O)(=O)C2CN(C(=O)C=CCO)CC12 Cc1cc(C(N2CCC(CN(C(=O)COCCCF)C)CC2)=O)c(C)nc1C c1(CNCC(C)C2CNC2)ccccc1CNS(C)(=O)=O CCC(C)C(C(=O)NC1CN(C(C)C)CC1C)N(C(=O)C=C(C)COC)C c1(C(N2CCC(N(C(C=CC(CC)C)=O)C)CC2)=O)ccc(Cl)c(F)c1 C(=O)(CCCCC(F)F)N1CC(NC(c2cnc[nH]2)=O)C2C1C2 c1(C(=O)NCC2(OC)CN(C(C3CCS(=O)(=O)C3)=O)C2)cc(O)cc(C#N)c1 C1(NC(C2CCC3(CC3)N2C(=O)CCC2CCCO2)=O)CC2(CCCC2)C1 C(=O)(CCCS(N)(=O)=O)NC1CCC(NC(C(C)Cc2ccncc2)=O)CC1 C1(NC(c2c(OC)csc2)=O)COC2(C1)CN(C(=O)C(C)(O)c1ccccc1)C2 C12(C(N(CC(C)CNC(c3cc(F)cnc3O)=O)C)=O)CCCC1CC(=O)CC2 c1(CC(N2C(CC)CN(C(=O)C(C)NS(C)(=O)=O)CC2)=O)nnc2n1CCCC2 c1(CC)ccsc1C(=O)NCCC1(O)CN(C(=O)CC(=O)OC)C1 C(Cc1ccccc1)(CC(=O)O)N(C)Cc1n(CC)ncn1 Cc1n[nH]c(C)c1C(C)C(=O)N(CC(C)NC(c1ncccc1C(F)F)=O)C C1(C(=O)NCC2CCC(NC(c3scnc3C3CC3)=O)C2)C(F)(F)C12CCC2 N1(C(C2(OC)CC2)=O)CC2CC1CC2NC(=O)Cc1cc(O)nnc1O C12CC(c3ccccc3)(C1)NC2=O.C1(CNC(C2CC(SC)C2)=O)CCCC1O C=C1CCC(C(N2CC3CC3(CNC(c3nc(C)oc3OC)=O)C2)=O)CC1 C1(C(=O)NC2CC2(F)F)COC2(CCN(C(c3ccncc3Br)=O)CC2)C1 c1(C(=O)NCCC(C)NC(C2(C(F)F)CCCC2)=O)c(F)c(F)cc(F)c1F C1(C(=O)NCC2CCN2C(=O)CN(C(=O)C(C)C)C)(SC)CCC1 C(=O)(C(=O)NOC)NC(c1ccccc1)C(=O)NC1(C=C)CCC1 c1(C(=O)NC(C2CCN(C(=O)CN3C(=O)CNC3=O)CC2)C)ccncc1Cl N1(C(C)=O)CCC(n2cncn2)C1.C1C(=O)N(C2CC2)CCO1 C1(C(=O)NCCN(C(=O)Cc2cccc(Br)c2)CC)COC2(CCC2)C1 CCCC(C(=O)NC(C)(CNC(C1(F)CCCCC1)=O)CO)c1ccc(Cl)cc1 c1(-c2n(CC(=C)C)nc(-c3ccc(OC)cn3)n2)cnn2c(OC)cccc12 c1(CC)cc(C(=O)NCC(C)(C(C)C)NC(=O)C(C)c2cccs2)cc(O)n1 CC1(C)CC(C)(C(N2Cc3ncsc3C2)=O)CN1C(c1csc(Cl)n1)=O Cc1cccc(-c2cn(C3CCN(C(C4CCCCS4)=O)C3)nn2)c1F C(C1C(=O)NC2CC(C2)CC(=O)N1)SCC.c1(NC(C)=O)cnn(C)c1 C(=O)(C(C)CC(N)=O)Nc1c(C2N(C(Cc3cc(C)no3)=O)CCCC2)n[nH]c1 O(NC(=O)CCC(C(C)C)NC(=O)C(CN(C)C)CC)CCOCC c1(CC)nc(C(c2nnnn2CC2CCOCC2)NC(C)CC2CC2)cs1 Cc1c(C(=O)NC2CC2NC(=O)C(F)(F)C2(O)CCCC2)cncc1Cl c1(C(=O)NC2C(CNC(c3ccc(OCC#C)cc3)=O)CC2)cc(C)cnc1C c1(C(N2C(CC(=O)Nc3c(OCC)cccc3)CC2)=O)ncc(F)cc1N Cc1nnc2n1CCC2(C)C(=O)NC(C)Cn1cc(CCO)nn1 c1(CCC(=O)NCCC2CCCN2C(c2cnc(C3CC3)o2)=O)cccnc1 O=C(C1=CCCCO1)NC1CN(C(c2ccc(-n3cncn3)c(F)c2)=O)C1 N1(C(CS(C)(=O)=O)=O)CCCC2(C1)CN(C(C1CC3CC1C3)=O)CCO2 C(=O)(C(C)CCC(C)(C)C)N(CCCNC(C(CC(C)C)O)=O)CCO n1(C(=O)NC(C)CCCCNC(=O)C(C)N(C)C)cc2ccccc2n1 N1(CC)CC(C(=O)N(CCCNC(C2CCCN(C(=O)OCC)C2)=O)C)NC1=O CC(CC(=O)NC(C)CN(C)C(c1ccnc(Cl)c1)=O)C(F)F CC(C)CCCC(=O)NC(CCN(C(=O)CC1CC1(C)C)C)C(C)C N1(C(=O)COC(F)F)CCN(C(c2ccc(CO)nc2)=O)C(C2CC2)C1 N1(C(C2CCCC(=O)O2)=O)CC(NC(=O)C=Cc2cncnc2O)CC2(CC2)C1 c1(C(=O)NCC(CC(C)C)NC(C2CNC(=O)N2C)=O)c(O)cccc1Cl C(C(=O)N=c1cc(C)o[nH]1)OCC(=O)NC1C(CNC(CC(C=C)(C)C)=O)CCC1 c1(C(N(C)CC2N(C(C(N3CCCC(O)C3)C)=O)CCC2)=O)nc(Cl)c(Cl)s1 c1(OC)cc(C(=O)NC2CCN(C(=O)C(C)(C)CF)CC2CO)c(Cl)cc1Cl c1(CC)sc(=N)[nH]c1C(=O)N(C1CCN(C(=O)CN2CCC(OC)C2)CC1)CC c1(C(=O)OCc2cc(=O)oc3cc(O)ccc23)cc(S(=O)(=O)N2CCCC2)ccc1Cl N1(C(CC(CC)C(F)F)=O)CC(NC(C2SCCCS2)=O)CC12CCOCC2 C1(C(c2n(CC(=C)C)nnn2)(C)NCC2(C)CC3(CC3)C2)(OC)CCCCCC1 C1(CNC(CS(=O)(=O)NC)=O)(COC)CCN(C(C2(C(=O)N(C)C)CC2)=O)CC1 c1(C(N2CCC(NC(c3c(C)nn(C)c3)=O)C2)=O)ccc(=O)n(C(C)C)c1 c1(C(N2C(C)C(O)CC2)=O)cc(O)nc2c1CN(C(C1CCN(C)C1C)=O)CC2 Cc1ncnc(C)c1C(=O)NCC1=CCN(CC(=O)NCC(C)C)CC1 N1(CCC)CCCC1C(N1CCC(C(=O)NCc2cccs2)C1)=O C1(NC(c2c(C)n(C)cc2)=O)CC2(C1)CC(C(=O)NC1CCN(C(C)(C)C)C1)C2 C1(C(=O)Nc2cccc(COC)c2)N(C(=O)CCc2cccs2)CCC1(C)C C(=O)(C(CC)C(C)(C)CC)N1CCN(C(c2cn(CCOC)nc2)=O)CC(O)C1 C1(CNC(C(C)NS(C)(=O)=O)=O)CN(C(c2ccc(F)cn2)=O)CC(C)(C)O1 CC1(C)CN(C(=O)CSC2CCCC2)C1C1CCCO1 CCCCCC(O)CC(=O)NCc1ocnc1C(N1CCCC1(C)COC)=O C1(CC)CN(C(C2CC(=O)N(C)C2)=O)CC1NC(c1cccc(OC2CC2)c1)=O CC1(NC(c2cccc(OC3CCC3)c2)=O)CCCN(C(=O)CC2CCOC2)C1 N1(C(C(C)O)=O)CCOCC(CNC(=O)CC2(C(F)F)CC2)C1 Cc1ccc(CCC(N2CCC(NC(c3cc(Cl)c[nH]3)=O)C(CO)C2)=O)cc1Cl CCCCCC(C)CC(=O)N(CCC(=O)Nc1cccc(C(C)F)c1)C CC1CCC(C)N1C(C)C(=O)N(C(C)CNC(=O)CCCc1cccs1)C C1(CN(C(=O)CC2CC(=O)NC2=O)C)CN(C(=O)CC2CCSCC2)CCO1 N1(C(c2cnn(C)c2Cl)=O)CCC2(CCN(C(C3CC(C(F)F)C3)=O)C2)C1 CC(F)(F)CCC(=O)N1CCC(N2CCN(C(=O)Cc3ccsn3)CC2)CC1 c1(C(N2CCC(NC(C(C)C3CC3)=O)C2)=O)ccc2c(c1)OCCO2 C1(O)(CN(C)C(C2CC(=O)CN2C(C2(C)CCCO2)=O)=O)CCCCC1 C(=O)(C1Cc2c(Cl)cccc21)N1CC(CNC(c2cncc(OC(C)C)c2)=O)C1 O=C1CCN(CC2(C3(SC(C)(C)C)CCCO3)CC2)C(=O)C(C2CC2(F)F)N1 C1(C(N(CCNC(=O)CCCn2ccnc2)C2CC2)=O)Cc2n[nH]cc2C(=O)N1 C(CN=c1cccn[nH]1)NC(N1CCC(n2ccnn2)C1)=O N1(C(CCS(C)=O)=O)C2CCCC1CN(C(C1CCC(=O)O1)=O)C2 c1(N2C(C)CN(C(c3ccnc(Cl)c3F)=O)CC(C)C2)ncnc2c1SCCC2 Cc1ocnc1C(=O)NC(C(=O)N(C)Cc1cn(C)cn1)C1CCOC1 N1(C(CCCC)=O)C2CCC1C(F)C(NC(C1(C(F)F)CCCC1)=O)C2 C1(C(N(CC(O)CNC(=O)CCc2ccoc2)C)=O)CC(C)(C)SC(C)(C)C1 c1(N(CCCC(=O)NC(CC2CCC(C)O2)=O)C2CC2)ncc(S(C)(=O)=O)cc1Cl C=CC(CCC)CC(=O)N1CC2(CC2)CC1CNC(c1cc(F)ccc1CC)=O n1(CC(C)NC(C2(C(F)F)CCCO2)=O)cc(CCC2CCCCO2)nn1 c1(CC(=O)OCC2CC=CCC2)ccc(NC(C2C(C)CCC2)=O)cc1 c1(C(=O)NCC2C(NC(C(CC)OC)=O)CC2)ccc2c(c1)nnn2C N1(C(C2(C#C)CCC2)=O)CC(NC(=O)CCc2cc(C)cc(C)c2)C2(CC2)C1 c1(OC(CC(=O)NC)C2CCC2)ccc(OC(F)(F)F)cc1.C1(=O)CCCCO1 C1(NC(COCCC(C)C)=O)C2CCC(C2)C1C(N1CCC(CO)CC1C)=O N1(C(C2CC(OCC)C2)=O)CCCC1c1cn(C2CC(O)C2)nn1 N1(C(CNS(CC)(=O)=O)=O)CC2CC1CN(C(C1CCC(C(N)=O)CC1)=O)C2 N1(C(=O)Nc2c(NC(c3cc(F)ccc3O)=O)nccc2)CCCC(F)(F)C1 C(=O)(C(CCC)OC)NCCCC1(NC(C(C=C)c2ccccc2)=O)CC1 Cn1nc(Br)cc1C(=O)NCC1CCCC1NC(=O)CCC1CCC1 N1(C(c2c(CNC(C(CSC)C)=O)cc[nH]2)=O)CC=CC12CCOCC2 c1(C(=O)NC(CNC(CC(CC)OC)=O)(C)C)cc(F)c2[nH]nnc2c1 C(CCC(=O)NC1(CN(C)C)CCOC1)=C(C)C.c12ccc(s1)C(=O)NC2 C(=O)(C#CC1CCCOC1)NCCC(C)(C)NC(=O)C1=CCCSC1 C1(C(=O)NC2CCN(c3ccccc3)C2)CC(=O)N(Cc2ccc(Cl)s2)C1 N1(C(C2(F)C(C)C2)=O)CCC(NC(=O)Cc2cccc(F)c2O)C(F)(F)CC1 C12(C(=O)NC(C34CCC(CO3)C4)C)COC(C1)C(NC(=O)C#CC1CCC1)C2 C1(NC(C(C)O)=O)CN(C(c2cc(Br)cn2C)=O)CC12CCOCC2 c1(C(N2CCC(F)(CNC(C3(C)C(C)C3)=O)C2)=O)ccc2c(c1)CC(C)(C)C2 c1(C(N2C(CNC(C(C)NC(C)(C)C)=O)CC2)=O)c2n(c(=O)n1C)CCCC2 Cc1ccc(C)c(C(N2CCC(N(C)C(c3cc(=O)n(C)cn3)=O)CC2)=O)c1N N1(C(c2cn(C)nc2O)=O)CC(NC(C2C=CCS2)=O)CC2(CCC2)C1 c1(CC)cc(C(=O)NCCCN(CCO)C(c2cnsc2)=O)ccc1C C1(NC(c2cc(Br)no2)=O)COC2CN(C(c3ccnnc3)=O)CC12 C(=O)(CCC(C)N(C)C)NC(C1N(C(C(=O)NCC)=O)CCC1)C c1(CC)noc(CC)c1CC(=O)NCC(C1CCCC1)NC(=O)C(C)(CO)OC C1(O)(CNC(C2C(C)(COC)C2)=O)CCN(C(c2cnc(C3CC3)s2)=O)CC1 c1(C(N2C(C)(CNC(c3cc(CO)on3)=O)CCC2)=O)cc([N+](=O)[O-])n[nH]1 Cc1nn(-c2ccccc2)c(C)c1CC(N1CCC1C(=O)N(C)CCO)=O C1(C(=O)NC2C=CC(C(N3CC(C(C)OC)C3)=O)C2)CC12CCOCC2 C(=O)(CCCCC(C)(C)C)NC12CC(C(=O)NC(C)C(C)(C)O)(C1)C2 N1(C(c2c(CSC)cccn2)=O)CC2CCN(C(C3CC(SC)C3)=O)CC2C1 c1(N2C(CCC(N3CC(C)NC(=O)C3)=O)CCC2)ncc2sccc2n1 C(=O)(C(C)(C)c1cncnc1)OCCOCC(=O)Cc1ccccn1 CC1COCCC1C(=O)N(C)CCN(C)C(c1cc(-n2cccc2)ccn1)=O N1(C(C(CC)(CNC(c2ccc(N)cn2)=O)CC)=O)Cc2ccc(C)nc2C1 N1(C(C(C)OCCCCCC)=O)CCCCC1CNC(=O)C(C)CC C(c1cncc(-c2cccc(C(N3CCCCC3)=O)c2)c1)=CC(C)(C)N(C)C C1(C(=O)O)CCC2CCC1N2c1nc(-c2ccc(C(F)(F)F)s2)ns1 c1(C(N(C)CC2CCN(C(=O)Cn3cnnc3)CC2)=O)cc([N+](=O)[O-])cnc1O CCC(F)C(=O)N1CCC(N(C(=O)CCC=CCC=C)CCO)C1 C1(C(=O)NCC(CC)NC(=O)COCC2(F)CC2)CCC(C(C)(C)C)CC1 c1(N(C2CCOCC2)C(=O)NC(C)C(C)n2cncn2)ccc2nccn2c1 Cc1oc(C(F)(F)F)nc1C(N1CCC(CO)(NC(c2cncc(N)n2)=O)C1)=O C(=O)(C(CC1CCCC1)CC)NC(c1c(C(=O)NCC(CCC)O)con1)C N1(C(C2(C)CC2)=O)CCC2(CCCN(C(c3cc4ccnc(Cl)c4s3)=O)C2)C1 c1(C(N2CC3(CC(NC(=O)CC4CS(=O)(=O)C4)C3)C2)=O)noc2cc(Cl)ccc12 c1(OC)c(C(=O)NCC2CCCN(CCC3CCS(=O)(=O)C3)C2)nc(O)nc1O N1(C(CC(C(C)C)NC(CC(CC)O)=O)=O)CCC12CCCSC2 c1(CCNC(=O)NC2CCCC2n2cccn2)cccc(F)c1 c1(SCNC(C)CCN=[N+]=[N-])ccc(S(N)(=O)=O)c(C)c1 CC1(C)CCCC(C(=O)NC2COCC2NC(c2cnc(=N)[nH]c2)=O)O1 c1(OC)ccc(F)c(C(N2CCCC2CCNC(c2cnc(S)[nH]2)=O)=O)c1 C(CC(=O)NOC1CCOC1)C1(CN(C)C(C2(CCN(C)C)CC2)=O)CC1 Cc1cc(F)c(C(=O)NC(C2CCOC2)CNC(=O)CC(C)(C)C)cc1F C1(OC)CC(NC(=O)C(c2ccc(NS(C)(=O)=O)cc2)N)C1(C)C C#CC1(NC(=O)C(CCOCCO)NC(=O)C(CO)NC(N)=O)CC(F)(F)C1 C1(O)(CN(C(=O)Cc2ccon2)C)CCCN(C(=O)C(=O)NCC(F)(F)F)C1 c1(C(=O)NC(CCN(C)C)C(N2CCC(F)(CF)CC2)=O)c[nH]c2ccccc12 CC(C)CC(O)C(=O)N1CCN(CCCNC(c2cc(Cl)no2)=O)CC1 n1(CC)c(C(N2CCNCC2C(=O)O)=O)cc2ccccc12 c1(C(=O)NCC(CNC(CC2CCC(C)C2)=O)(C)C)cc(S(C)(=O)=O)co1 C(=O)(C(O)CCCNC(=O)CC1(C#N)CC1)NC(C)(C)C(N)=O c1(OCC=O)ccc(N(CC)CC)cc1C.C(=O)(C(C)N(CC)CC)N N#Cc1ccncc1C(=O)NCC1OCCC1C(=O)N(CCCO)CCCO C(=O)(CS(=O)(=O)C(C)(C)C)N(C)CC1(O)CCN(C(C2(C(C)C)CC2)=O)C1 N1(C(C(C)Cn2ccnc2)=O)CCOC(C(=O)Nc2ccc(F)cc2O)CC1 C(=O)(CCN(OC)C(=O)C1(O)CCOC1)NCC(C#C)C(C)C N1(C(C(=O)NCCOC)=O)CCN(C(=O)CCc2cnco2)CC1C1CC1 C(=O)(C1=CCC(NC(c2cc[nH]c2)=O)C1)NCCC1C(C)CCO1 CC(C(=O)NNc1ccc(Br)c(F)c1F)OCC1CCCO1 c1(OC)nc(C(N2CCCC2(C)CNC(=O)C(C)C2CC2)=O)sc1C CCCCCC(=O)N1CC(NC(c2csc(-c3cccc(C)n3)n2)=O)C(C)C1 c1(C(=O)NCC2N(C(Cc3nc(C)[nH]n3)=O)CCCC2C)ncc2ccccn12 c1(SC)ccc(CCCC(=O)NC2C3CC2N(C(=O)CC2CCC(=O)O2)C3)cc1 C1(C(=O)NC(C)(C)CNC(=O)C=C2CCCCC2)(CC)CCC(F)(F)CC1 CC1(O)CCCN(C(=O)CONC(=O)C=C2CCOCC2)C1 c1(OC)cccc(C(CO)NC(=O)CC2CC(CNCc3ccncc3Cl)C2)c1 C(CC(C(C)(C)C)NC(c1cccc(C(F)F)n1)=O)N(C)C(c1cnn(C)n1)=O CC(C)CC(C(=O)N1CC2CC2(C(C)C)C1)ONC(=O)C1(CC(C)C)CC1 c1(C(=O)NCC2(C(F)F)CCN(C(c3c(SC)csc3)=O)C2)c(C)cnnc1O c1(CN(C(=O)C2=CC(C)(C)C2)CC)ccc(CO)c(F)c1.C12CCCCN1C2=O C1(C)(C(=O)NC(C2CCCN2C(=O)Cc2cn[nH]c2)C)CC1(C)C c1(C(=O)NCC(C)NC(=O)Cc2ccccc2Br)cc(C#N)c(F)cc1F Cc1c(NC(c2nc(-c3ccccc3)oc2C(C)C)=O)cnn1CCO C1(C(=O)NC2CCN(CC)C2)CCC(O)CN1C(c1ccc(=N)[nH]c1)=O C(=O)(CC(C)(C)C#N)NC1CCCC(N(C)C(c2ccc(C(F)F)s2)=O)C1 c1(SC)ncc(-c2cccc(CC(=O)NCc3cccc(C(F)(F)F)c3)n2)cn1 N1(Cc2scc(C(=O)NC3C(CC)CCO3)c2)CCOC(CC(N)=O)C1 c1(OC)cc(OC)cc(C(N2CCCCC2C(=O)NC(C)CN(C)C)=O)c1 N1(C(C2(CC#C)CC2)=O)CCC2CCN(C(c3cc(O)nc(O)c3)=O)CC2C1 CC(C)C(=O)CCCN1CCN(C2CCCCC2N(C)C)CC1 c1(Nc2cncc(CC(C(=O)O)NC(=O)OC(C)(C)C)c2)cc2n(n1)CCC2 C(=O)(C#CC1CCC1)N1CCC(C(C)NC(c2ccn(CC)n2)=O)C1 C(=O)(N=c1[nH]nc(SC)s1)NCC(CC)O c1(CCNC(N(C2CCCC(SCC)C2)c2ccccc2)=O)ccnc(C)c1Cl c1(C(=O)OC)cc2c(c(S(=O)(=O)Nc3cccc(N4CCCC4=O)c3)c1)CCC2 CCC(C)C(C(=O)NC(C)(CO)C1CC1)N(C(=O)C=C1CCC1)C c1(C(=O)NCC2CCN(C(C=Cc3ccc(CC)o3)=O)C2)ncc(Br)cc1C Cc1cncc(C(=O)N(C)CC2CN(C(=O)CSCc3csc(=N)[nH]3)CCO2)n1 C1(C(=O)NC(C2C3CC4C(C3)C24)=O)CC12CCN(C(C1(C)CC(F)(F)C1)=O)C2 C(=O)(CC1=CCCCC1)NC(CCCNC(=O)Cn1cnnn1)c1ccccc1 c1(C(=O)NC2C(NC(=O)C3=CCCOC3)CCCC2)ccc2c(c1)COCCN2 N1(C(CC2C(OCC)COCC2)=O)CC2CC(Nc3ccc(F)cc3)C1C2 C1(C)(C(C)C)CC1C(=O)N(CCNC(=O)Cc1cc[nH]c1)CCOCCO C1(CCC)CN(C(c2cc(C(=O)OC)cs2)=O)CCN1C(c1cccnc1Cl)=O N1(C(CCSC)=O)CCCC(O)(CCNC(c2cccc(F)c2C(F)F)=O)C1 c1(-c2cnc(SCC(=O)NCC3CC4CCC3C4)o2)ccccc1F C(=O)(CCC(C)(C)NC(c1cn(C)c(=O)n1C)=O)NCc1c(C)nn(C)c1 CCC(CC(F)(F)F)C(=O)N1CCC(CNC(c2cnc(C(=O)OC)cn2)=O)C1 C1(OCCC)Cc2cn3c(n2)SC(=N1)N3.c1ccccc1 Nc1cc([N+](=O)[O-])ccc1C(=O)NCC1CC1NC(c1ccccc1[N+](=O)[O-])=O N1(C(=O)CC2CC3CCC2C3)CC2CN(C(C3(Br)CC3)=O)CC(C1)O2 C#Cc1ccc(C(N2CCC(C=CC(N3CCC(CO)C(C)C3)=O)CC2)=O)cn1 C(=O)(C1CCCc2ncccc21)NC1CCN(C(Cc2c(C)nn(C)c2Cl)=O)C1 c1(C(N2CC(NC(C=CC(CC)=CC)=O)C3C2C3)=O)ccc2nncn2c1 Cc1cccc(C(=O)N(C)CCn2cc(CN3CC4CC4C3)nn2)c1Br CCCCC(CCCC)C(=O)N1CC(NC(=O)CCSc2nccn2C)C(C)C1 N1(C(c2cc(C)oc2)=O)CCC2CN(C(c3csc(=N)[nH]3)=O)CC12 S(=O)(=O)(c1ccc2c(c1)CN(C(=O)Cc1cc(C3CC3)on1)C2)N(C)C Cc1nc(NCc2ccc(N(C)C)c(C)c2)cc(=NCC2CCOCC2)[nH]1 C12(CNC(c3ccncc3)=O)CCCOC1CCN(C(c1cccc(Cl)c1)=O)C2 C(=O)(NNC(=O)NC1CC(Cc2ccccc2)C1)c1ccc(C)o1 N1(C(CCSCCC)=O)CC2CCC2(CCNC(c2nccnc2C(N)=O)=O)C1 C1(OCC)CCN(C(=O)CC2(OC)CN(C(=O)CC3(COC)CC3)C2)CC1C c1(C(N(CC(=O)NCc2c(C)nc(C)s2)C)=O)ccc(C)c(O)c1 n1(CCC)nc(C)cc1C(=O)NCC(C1CCCC1)NC(C)=O c1(C(N2C(CNC(=O)C(N)=O)CC(COC)C2)=O)cc(Cl)cc(Cl)n1 C1(C)(N(C(c2cscn2)C)C)CCN(Cc2ccccc2)CC1.C1(=O)CCCN1 c1(C(c2nnnn2CCCF)NC(CCCC)COC)ccc(N(C)C)cc1F c1(C(=O)NCCCNC(=O)C(F)Cc2ccccc2)cnc2[nH]nnc2c1 C1(C(=O)NC)CC(O)CN1C(=O)CC1CCCC1NC(=O)C=C1CCOCC1 C=CCCCCCC(=O)NC1CCN(C(=O)COC2(C)CCC2)CC1F c1(C(N2C(C)CC(c3ccccc3)C2)=O)cc2cccc(Br)c2cn1 c1(C(=O)NC2CCCC(C(=O)Nc3cnoc3)C2)cc(F)cc([N+](=O)[O-])c1 c1(C(=O)NCC(C)(C)NC(C(C(COC)C)C)=O)cc(C)c(F)cc1F N1(C(COC(C)=O)=O)CCC2(NC(=O)Cc3ccc(F)cc3Cl)CCCCCC12 CCC(CC(=O)N1CC2C(CNC(c3cncc4c[nH]nc34)=O)C2C1)C(C)C N1(C(C=C(C)C2CC2)=O)CCC(C)(C)C1CC(N1CCCC1)=O N1(C(CC(CC)C(C)C)=O)CCC2(CCCCC2NC(=O)CN(C)C)CC1 n1(CCOC)cc(NS(=O)(=O)CC2COCCO2)c(C)n1 C1(C(N2C(C(C)C)C(NC(C3CC(=C4CCC4)C3)=O)CC2)=O)CN(S(N)(=O)=O)C1 c1(C(=O)NC(CN(C)C)C(=O)NCCN2CC(CF)C2)cccnc1S N1(C(C)=O)C2CCC1CN(C(N1CCCCC1c1cnc(S(C)(=O)=O)s1)=O)C2 c1(COC)cc(F)c(S(=O)(=O)Nc2cccc(C(=O)N(C)C)c2)c(F)c1 Cc1cc2c(cc1NC(=O)CC(C)N(C)C(=O)NC(C)(C)C)CCO2 N1(C(c2c(C)ccnn2)=O)CCCC(CO)(NC(c2cccs2)=O)C1 Cc1noc2ncc(C(N3CC(NC(C4CCN(C)C4)=O)C(O)C3)=O)cc12 C1(NC(=O)Cc2c[nH]nc2O)CC(O)CN(C(c2ccc(C(F)F)c(F)c2)=O)C1 C1(C(=O)NC(c2n(CC)ncc2)C)CN(C(=O)CCP(C)(C)=O)CCC1O Cc1nnc(NC(C2(c3ccncc3)CC2)=O)n1C O=S(=O)(c1ccc(N2Cc3ccncc3C2)cc1Br)NC(CO)C1CC1 c1(NC(C)CCC(F)(F)F)ccc(S(=O)(=O)NCC2(C)CCCOC2)cc1C#N N#CC1(C(=O)NCC(O)CNC(C2CC23CCCCC3)=O)CCSCC1 c1(OC)ccc(C(=O)NCC2C3CN(C(C4(F)CC4)=O)CC23)c(OC)c1Cl C(=O)C(N)CCC(=O)OCC.N1(C(C)C)CCC(C2CC2)C1 C1(NC(C(C)(C)NC)=O)CCC2(CC1)CCN(C(=O)CCc1cc(F)ccn1)C2 N1(C(CN(c2ccc(Cl)nn2)C)=O)CC(C2(NC(=O)CN3CCCCC3)CC2)C1 CCC(COC)C(=O)N1CCC(CC(=O)NC(C)CC(C)CC)CC1 Cc1cc(C(=O)NCC=CCNC(C2CC2c2cccc(Cl)c2)=O)ncn1 CC(C)C(CCNC(C1(n2cccn2)CCC1)=O)NC(=O)Cn1ccccc1=O C1(CNC(CC2CC(OC)C2(C)C)=O)CC(C)CN(C(=O)CC2(OC)CCC2)C1 CC1CCCCC1(CNC(=O)C1=CCCOC1)NC(=O)C1=CCCOC1 Cc1cc(O)nnc1C(=O)NCCC1CN(C(C2(O)CCC2)=O)CC1C c1(C(=O)NC(C2CC(NC(C3(CF)CCOCC3)=O)C2)C)cccc(O)n1 C12(CNC(c3sc(C)c(-c4nc5cnccc5[nH]4)n3)=O)CCCCC1CCC2 N1(C(C2(NC(C3CC(CC)(CC)C3)=O)CCSC2)=O)CCC12CCC(O)CC2 C1(C2CC2)(CNC(C2C(OC)C2C)=O)CCN(C(=O)COCC2CCCOC2)C1 C1(C(=O)NC2CC(NC(CSc3n(C)ccn3)=O)C2)CCCCC1C#N N(C1CC2(CCN(C(=O)C(F)F)C2)Oc2ccccc21)C(C1(C#C)CCCC1)=O C(=O)(C(C)CC(N)=O)NC1CC(F)(CNC(c2c(C(C)C)scn2)=O)C1 C1(NC(C(C(C)(C)C)NC(C)=O)=O)CN(C(c2n[nH]c3c2CCC3)=O)CCC1(C)C C1(CNC(CCc2n(C)ccn2)=O)(NC(=O)CC#N)CCOCC1 c1(C(=O)NC(CNC(CC2CCC(C)C2)=O)(C)C2CC2)ncc2ccccn12 C1(C(N(CCC#N)Cc2ccccc2F)=O)C2C=CC(C2)C1C(=O)O N1(Cc2cccc(C)c2)CCCC(NC(=O)CNC(=O)CC(C)(C)C)CC1 C1(NC(c2nnn(CC)c2C)=O)CC(NC(c2occc2Br)=O)C12CCC2 N1(C(CC=CCNC(C2C(C)CCC2)=O)=O)CCCC2(C=CCO2)C1 c1(N)nnc(C(OC(F)(F)F)C)n1Cc1cccs1.C(C(C)C)CCC C1(CC(=O)NCC2N(C(CSc3n(C)ccn3)=O)C3C(C2)C3)CN2CCN1CC2 N1(CCNC(c2nnnn2C2CC2)C2(C)CSC2)CCc2ccccc2C1=O c1(-n2c(C(=O)NC3CC(CNC(CCOCC#C)=O)C3)cnc2)ccccc1Cl C(=O)(C1CCCc2nncn21)N1CCC(O)(CN(C)C(C2(C)CCOC2)=O)CC1 N1(C(C(CC=CC)CC)=O)CCC2CN(C(=O)C=Cc3scnc3C)CC12 c1(C(N2C(CNC(c3n(C(C)C)ncc3)=O)CCC2)=O)c(Br)cc(F)c(F)c1F CC(CC(=O)N1CCCC1CC(=O)N(C)CC1(C)CC1)C(C)(C)C c1(OCCC=C)ccc(C(N2CCC(C)(CCNC(=O)CCOCC)C2)=O)cc1 C(=O)(CCCCC#N)N(C)CC1CCC(CNC(c2cn[nH]c2)=O)O1 C(=O)(CC(F)(F)C(C)(F)F)NCC1CCC2(CN(C(CC(CC)CC)=O)C2)O1 C1(C2CC(NC(=O)NCc3ccc(C(=O)OC)cc3)C2)Cc2ccccc2O1 Cc1cc(C)c(C(N2CC(C(F)(F)F)C(CNC(C3CCCC3)=O)C2)=O)c(=O)o1 Cc1cc(C)c(NC(C2CC23CC(NC(=O)CC(C)n2cccc2)C3)=O)c(C)c1 N1(c2cc(C)nc(N3CCN(Cc4ccco4)CC3)n2)CCC2(CC(C#N)C2)C1 C1(CNC(C2(C#C)CCC2)=O)C2CCCC1N(C(c1nccc(Cl)c1Cl)=O)C2 C1(NC(CC=CC)=O)CC12CCN(C(c1nn(C)cc1N)=O)CC2 CC1Oc2c(F)cccc2C1NC(c1ccc(C#N)cc1Br)=O C1(C(=O)N(C)CCC2CCC2)(SC)CN(C(C2CCCC2O)=O)C1 C1(NC(C2CC23CC3)=O)CCN(C(C2SCCS2)=O)CC1O C1(OC(N(C(CN2CC(C)(OC)C2)=O)Cc2ccccc2)=O)CC2(CCCC2)C1 CCC1=C(C(=O)NCC23CC(NC(=O)CN4CCCC4CO)(CO2)C3)SCCO1 N1(C(C(CC)OC)=O)CC2C(CN(C(=O)CCC3CCCCC3)C)C2C1 C1(C(N2CC(O)(CNC(c3ccc(N)cn3)=O)C2)=O)Cc2nnsc2S1 c1cc2c(N3CCC4(CCCO4)CC3)[nH]c(=NCc3cn4ccnc4s3)nc2s1 c1(CN2CCC(C(C(=O)Nc3nc(C)sc3)C)CC2)cc(F)ccc1[N+](=O)[O-] N1(C(c2c(CC)csc2)=O)CCCC12CCN(C(c1cscc1OC)=O)C2 C1(CCC)CN(C(c2c(C)cnn2C)=O)CCN1C(C1CC1c1ccccc1)=O C1(C(=O)NC2CN(C(c3ncn(C)n3)=O)CC2O)CCCCNC1=O C#CCC(C)(C)C(=O)NCC(C)CN(C(=O)C(C)Oc1cccc(C(C)=O)c1)C C(=O)(CCCC(C)(C)NC(=O)C1=CCCCC1C)N1C(C(=O)NC)CC(O)C1 C1(NC(=O)Cn2cccnc2=O)CCN(C(=O)Cc2cnccn2)CCC1CO C(=O)(C(C)CC(C)(C)C)NCC1N(C(C2N(C(C)=O)CSC2)=O)CCCC1 c1(C(N2CC(C(C)NC(c3c(CC)n(C)cc3)=O)OCC2)=O)cccn(O)c1=O c1(N2C(CNC(C(=C)C)=O)C3CCC2C3)nc(C)cc(C#N)n1.C12(CC1)C(=O)NC2 N1(C(CC(c2cccc(F)c2)C)=O)CCC12CN(C(=O)Cc1ccon1)C2 C1(CNC(Cc2cc(C)ncc2)=O)C(C2CC2)CCN1C(=O)CC1CCC(C)C1 C1(CN(C(=O)CCCCN2CCCCC2)C)CCCN(C(=O)COCCCF)C1 c1(CC(=O)NCC2CC3CNC2C3)ccccc1OCc1ccccc1 Cc1[nH]nc(C(=O)NCCC2CCN(C(=O)Cc3cc(C4CC4)no3)C2)c1F C(=O)(C(C)(C)C(N)=O)N1C(C2(NC(C3CCN(C(C)C)C3)=O)CC2)CCC1 C(N=c1[nH]c2c(c(=NC3CCc4cccc(N(C)C)c43)[nH]1)COC2)c1c(C)nco1 C(CC(C)C(=O)N1CCC(NC(c2cc(C#N)no2)=O)C1)OC C1(NC(CCN(C(C2C(CCOC)C2)=O)C(C)C)=O)CC2CC2C1 c1(C(N2C(CNC(CC3(C)CCOCC3)=O)CCC2)=O)cnn2cccc(Cl)c12 C(CNC(c1n[nH]c(O)n1)=O)(C(=O)NCC(CC1CC1)CO)OC c1(CN=C(NC(COC)C)NCCn2ccnc2)ccc(F)c(O)c1 N1(C(C(CCC)OCC)=O)CC2(CCN2C(=O)CCC2CCC2)C1 N1(C(CN2CC(=O)N(CCCc3ccccc3)C2=O)=O)CCCC2(C1)OCCO2 N1(CC(=O)NCC(C)C)CC(NC(c2cnsn2)=O)CCC1C CC1CC(C(=O)NCCCCCCNC(=O)CC2CC(F)(F)C2)CCS1 CC1(C)CNC(=O)c2c(C(=O)NCCNC(C3Cc4cscc4C3)=O)coc2C1 N#Cc1cc(C(=O)NCC2CCN2C(c2nccc(Cl)c2F)=O)n2c1CCCC2 C=CC1(CC(N2CCOC3CC23)=O)CN(C(=O)CCC(C)N(C)C)C1 CCCCC(CC)CC(=O)N1CCC(C)(C)C(C(=O)NC2CC(O)(CO)C2)C1 CCCCCC=CCC(=O)NCCN(C(=O)C(C)OCC1CCCCO1)C(C)C O=C(CCC(F)F)NCCC1CCCN(C(c2cccc(OC(F)F)n2)=O)C1 c1(CN2CCCC(NC(C(C)(C)O)=O)CC2)cc(Br)c([N+](=O)[O-])s1 c1(C(N2CCC(C(N)=O)C(C)(C)C2)C(=O)NC)ccc2c(c1)CC(C)O2 Cc1cc(C#N)cc(C)c1C(N1CCCC1CNC(=O)C(O)c1ccco1)=O c1(C(=O)NCC(CC)NC(=O)C(C)S(C)(=O)=O)coc2c(F)c(Cl)ccc12 c1(C(=O)NC(CCCNC(Cc2ccc(C)cc2F)=O)C)cccc2c1NCC2 CCC(CCCC(=O)OCC1(O)CC2CCCC12)c1ccccc1 C(c1ccc(C)nc1)=CC(=O)NC(CCNC(c1c(CC)n(C)nn1)=O)C C#Cc1ccc(Cl)c(C(N2CCCC(CN(C(=O)C(C#N)CC)C)C2)=O)c1 n1(CCN(C(c2cnn(C(C)C)c2C2CC2)=O)C)c(=O)oc2ccccc12 N1(C(c2c(OCC)scc2)=O)CCC(C)(NC(=O)C(C)OCC)CC1.C(CC(C)C)O N1(C(C2(C(=O)OC)CC2)=O)CCC(C(C)(C)C)(CNC(C23CCN(CC2)C3)=O)C1 N1(C(=O)NC(c2ccc(F)cc2)CCC)CCCC1C1OCCO1 CC(C)CC(CNC(c1ncccc1N)=O)C(=O)NC(C)CCC=C(C)C C1(CNC(C=C(C)C(F)F)=O)CCC(CN(C(=O)C=C2CCCCC2)C)CC1 c1(OC)nc(Cl)ccc1C(N1CCCC1(C)Cc1ccc(C)c(F)c1)=O N1(C(c2ccc(C(CC)C)cc2)C(=O)NCCCC2CC2)CCOC2CCCC12 Cn1nc(C(=O)NC2CC(C(=O)NCCC(N)=O)C2(C)C)cc1O n1(CC(N2CC(NC(COC)=O)C(c3ccccc3)C2)=O)nnc2ccccc12 N1(C(c2cc(C)cc(Br)c2)C(=O)NC(C)C(=O)OC)CCC(C2CCOC2)CC1 Cc1cc(NC(C2CCCN2C=O)=O)cc(CNC(c2cc(CC3CC3)on2)=O)c1 C(=O)(CC(O)C(C)(C)C)NC(C)CN(C)C(c1ccccc1)=O C1(CC)C(C(=O)NCCOC2CCN(C(=O)Cc3cn(CC)nn3)C2)CCN1C CC1C(NC(c2cn(C(F)F)cn2)=O)CCCN1C(=O)CCC1CC1 CC1C(NC(=O)C(C)(C)C2CCCCO2)CCN1C(=O)CC(F)F CCC(CC)CC(=O)N1CC(CC(N2Cc3c[nH]nc3C2)=O)(OC)C1 N1(C(c2c(C)cc(C)nc2S)=O)CCOC2(CCN(C(=O)CSC(F)F)C2)C1 C1(C)(NC(COCC=C)=O)CC(NC(c2csc(C(C)(C)C)n2)=O)C1 N1(C(Cc2ccc(C)c(Cl)c2)=O)CCC2CN(C(=O)Cn3cnnc3O)CC2C1 C1(CCO)(NC(C(C)SCCCC)=O)CN(C(=O)C(CO)c2ccccc2)C1 C(=O)(C(O)C(C)(C)C)NC1(CC(=O)NCc2ccc(OC)cn2)CCC1 C1(C#N)(C(=O)NCCOCCN(C)C(c2cc(Cl)ccc2F)=O)CC12CCCC2 C1(CC(=O)Nc2cccc(C3CCOC3)c2)CCCS(=O)(=O)C1 Cc1ccnc(C)c1NC(C1CCC(NC(c2nccnc2Br)=O)CO1)=O CC(C)(C)CC(=O)NC(C1CC=CCC1)C(N1CCCC(CO)C1)=O C1(C(=O)NCC2C3CN(C(=O)C=CC=C(Cl)Cl)CC23)CCCCCS1(=O)=O Cc1ccc(C)c(N(C(=O)Cc2noc(COc3ccc(F)cn3)n2)C(C)C)c1 N(C(=NCCSC)NCCn1ncccc1=O)CC(c1ccc(Cl)cc1)OC C1(NC(C2(C)CC2)=O)CC2(CCN(C(C3CC(N4CCOCC4)C3)=O)C2)C1 CCC(C)C(C)C(=O)N1CC(c2ocnc2NC(=O)CC2(O)CCCCC2)C1 C(=O)(C1NCCc2cc(C#N)ccc21)Nc1c(C)n(-c2ccc(Cl)cc2)nc1 C1(CNC(=O)CC(C2CC2)C2CC2)CC2CCC1N2C(c1ccsc1Br)=O N1(C(C2(C)CC2)=O)CCCC(C2CC2NC(=O)CCCCCn2cnnn2)C1 C12(CNC(C3(CO)CCN(C(C(C)SCCCC)=O)C3)=O)CCCC1CCC2 C(=O)(CCCCCCBr)N1C(CC(N2CCN(CC(F)F)CC2)=O)COCC1 C1(CC)CN(C(c2c(CNC(=O)C=Cc3cnccn3)nnn2C)=O)CCO1 C1(C(=O)NC(C2CCOC2)(C)C)COCCC1NC(c1cccc(CO)c1)=O c1(C(N2CCC(O)(C(C)NC(CCSCC(C)C)=O)C2)=O)occ2c1CCOC2 c1(CC(N2CC(C(C)NC(c3c(C#C)c[nH]n3)=O)C2)=O)c[nH]c2cnccc12 N1(C(C2(C#C)CCCC2)=O)CCC2(CCC(CNC(C3CC3(Cl)Cl)=O)O2)CC1 N1(C(C(=O)NCCCSCC)C2=CCSC2)CCC2(O)CCOCC2C1 CCC(C)CCCC(=O)N1CCOC(CN(C(=O)CN2CCCS2(=O)=O)C)C1 C(CCCCC(=O)NC1CC1C(F)(F)F)NC(C1C(C)CC1)=O O=C1CC2CC(C1)CN(C(c1ccc(C(=O)Nc3cc(Cl)c(Cl)cn3)cc1)=O)C2 Cc1nc(Br)cnc1NC(C1CCCN(C(=O)CC#N)C1)=O Cc1c(NCCCc2ccsc2)ncnc1N1CCC(NC2CCC2)C1 C1(NC(C(C)CC2CC2)=O)CCC2(CCCN2C(=O)CC(C)(C)C(F)F)CC1 N1(C(c2c(C)ocn2)=O)CCC(C2CCN(C(c3ccnn3CC(F)F)=O)C2)C1 CCCCCCC(C)C(=O)NC1CC(C)(NC(c2cncc(Cl)c2)=O)C1 N1(C(C2C(C(C)O)C2)=O)CCCC(C2(NC(C3(O)CCCCC3)=O)CC2)C1 Cc1nccc(C(N2CCC2CNCC2(c3ccc(Cl)c(F)c3)CC2)=O)c1C C1(N(C(CN(S(CC)(=O)=O)C)=O)C)CN(C(=O)OC(C)(C)C)C2(CCC2)C1 CCCC(C#N)C(=O)NC1CCCCN(C(c2ccc(C(F)(F)F)nc2Br)=O)C1 N1(C(c2c(C)ocn2)=O)CCN(CCN(C)C(C2(C)CC=CCO2)=O)CC1 N1(C(=O)Nc2c(C)cccc2)C2CC1CN(Cc1ccnc(F)c1)C2 c1(C2CC(C(=O)NCCC3CCC(NC(c4sccc4F)=O)C3)C2)ccccc1 C1(NC(CCC=C)=O)CC2CC(NC(C3CCCC34CCC4)=O)C2C1 C1(C(N2C(CC(=O)NC)CN(C(=O)C=C(C)Cl)CC2)=O)CCCN2CCCCC12 c1(C(=O)NCCC2CCCN(C(=O)C(F)C3CC3)CC2)ccc2nn[nH]c2c1 N1(C(=O)CCOC2CC2)CCCC2(CCN(C(=O)CC3CC4CC4C3)CC2)C1 C(=O)(C1=C(C)N(C)c2nnnn2C1)N1CC(NC(=O)NC(C(=O)OCC)C)OCC1 Cc1nc(O)[nH]c1C(=O)NCC(C)(C)CN(C)C(c1ccc(Cl)o1)=O c1(C(=O)NCC2CCN(c3nnn(C)n3)C23CC3)ccc2c(c1)nnn2C Cc1cnc(N2CCOC(C(C)NC(c3cc(C4CCC4)on3)=O)C2)nc1O c1(CC(=O)NCC(C)NC(CC2C(C)=NOC2=O)=O)ccc(F)cc1F C(=O)(CCCC(OC)OC)N(CCC(C)C)CCC(N1CCC(CCC#C)C1)=O c1(CC)ccc(F)c(C(=O)N(C)CC2CCN(C(c3conc3CC)=O)CC2)c1 c1(C(=O)NC(C2CCOC2)CNC(C2(CC)CC2)=O)c[nH]nc1C1CCOCC1 N1(C(C2(COCC)CC2)=O)CCC(C(=O)Nc2ccccc2C(C)O)CC1 CC1CN(C(C2C(NC(c3ccc4[nH]ccc4n3)=O)C2(C)C)=O)CC(C)(C)C1 N1(S(C(C)(C)C)(=O)=O)CC2CC1CC2NS(=O)(=O)CC#N C#CCCC(O)C(=O)N1CC(C2(NC(C3CC(F)(F)C3)=O)CC2)C1 c1(CC(=O)NC(CCC)CNC(C2CCC2C)=O)cc(F)cc(F)c1 N1(C(C(C)Nc2ccn(C)n2)=O)CCN(C(c2cccnc2OC(F)F)=O)CC(O)C1 C#CC1COCCN1C(=O)CCC(CC)NC(=O)CCN(C)CCC N1(C(c2c(C)cc(F)cn2)=O)CCC(N(C(=O)CC2C=CS(=O)(=O)C2)C)C2(CC2)C1 C1(NC(C(Cn2ccnn2)NC(CCC(C)N(C)C)=O)=O)CCCN(C)C1=O C12(C(N3CCC(CC#C)CC3)=O)CCCC1CCN2C(c1sncc1CC)=O N1(C(c2c(C)nccc2)=O)CCC(C)(C)C1C(N1CC(c2cc(O)n[nH]2)C1)=O C1(C)(C(=O)NCC2(NC(CCC(C)(F)F)=O)CCOC2)Cc2ccccc2C1 c1(C(=O)NCCNC(=O)OC)ccccc1S(C)=O C1(C(N2CCC(O)(CNC(=O)CCc3cc(Cl)cs3)C2)=O)CC2C(C1)C2(F)F c1(OC)ccc(NC(=O)N(C2CC2)Cc2ccc(C)cc2)c(C(F)(F)F)c1 c1(C(C(=O)NCCOCC)N2CCC2C(=O)NC)ncccc1Br.C1CO1 C1(C(N2CC3CC(CNC(c4cccnc4)=O)C3C2)=O)CCc2ncsc2C1 N1(C(C2CCN(CC)CC2)=O)C2CCC1C(C(=O)NC1CC1(C)C)C2 C(C)(CC(=O)NC1CCN(CCOC)C1)NC(COCC(=C)C)=O c1(C(=O)NCC(CCOC)NC(=O)CC2CN3CCC2CC3)cn(C)ccc1=O C(CCO)(C(C)(C)C(=O)O)N1CC2C(C(N(C)CC3CCCC3)=O)C2C1 c1(CC(=O)NCC2CCN(C(COC(CC)C)=O)C2)ccc(F)cc1F Cc1ncncc1C(=O)NCC1COC(CNC(C2CCCN2C2CC2)=O)C1 c1(OC)c(F)ccc(F)c1C(=O)NCC1CC1NC(C1(P(C)(C)=O)CC1)=O CC(c1ccccc1F)=CC(N1CCCCC(NC(=O)C(C)CC(N)=O)C1)=O Cc1cc(C)n(C(C)C(=O)NC2CCCC2(C)NC(=O)Cc2cncs2)n1 CN=c1[nH]cc(C(=O)NC2CCC2NC(=O)CCc2ccccc2OC(F)F)s1 C1(C(=O)NCCN(C)C(C2CCCC2C(F)(F)F)=O)CCN(CCF)CC1 CCC(F)(F)CCN=c1nc2scnc2c(NCCOC2CCCCO2)[nH]1 OC1CN(Cc2cn(-c3c(F)cc(F)cc3F)nn2)CCc2ccccc21 C(=O)(CCS(C)(=O)=O)N1CCC(N(CC#C)C(c2ccc(O)nc2)=O)CC1 c1(OC)ncc(CC(=O)NC2(CNC(c3cccnc3OCCO)=O)CC2)cn1 c1(C(CNC(C2CC(OC)C2)=O)CNC(=O)CN2CC(CF)C2)ccccc1 n1(CC)ccc(CC(=O)NCCN(C(=O)C(C)OCC(C)C)C(C)C)n1 C1(CCNC(c2cccc(C)c2C)=O)CN(Cc2nc(=O)n(C)[nH]2)CCS1(=O)=O N1(C(Cc2cn(CC)nc2)=O)CCCCC(NC(c2nn[nH]c2Cl)=O)C1 C1(C(=O)NC(C2CCCC2)CNC(C2(CC(C)C)CC2)=O)CC=CC1 c1(C(=O)NC2C(C)CCN(C(=O)Cn3cccn3)C2)cc(F)c2c(c1)nnn2C C1(C(=O)NC)CN(C(C)=O)CCC1O.C12CCN(C1)C2=O C1(C(=O)NC2CN(C(c3ccc(C(N)=O)o3)=O)CC2CO)CCCCC1C1CC1 N1(C(c2ncc(C)o2)C(=O)Nc2ccc(OC)cc2C)Cc2c[nH]nc2C(C)C1 N1(C(C2=NN(C)C(=O)CC2)=O)CCC(C2CCCN(C(C34CC(C3)C4)=O)C2)C1 C1(C(N(C(CC(=O)N(CC#C)CC2CC2)(C)C)C)=O)CCC(C)=C(C)C1 CC1CN(C)CCC1N(C(c1cc(Cl)ccn1)C(=O)NCC1CCCO1)C C(C(F)C(=O)NC1(CO)CN(C(C2COCC2C(N)=O)=O)C1)N(CC)CC N1(C(c2cc(C)nn2C)C(=O)NCc2ccccc2)CCC2(O)CCOCC2C1 c1(CN2CCC(CNC(c3ccc(OC)cc3)=O)CC2)ccc(O)c(C)c1 n1(CC)cc(Cl)c(C(=O)NCC2CCCN2C(=O)C(C)(CO)OC)n1 n1(CCC(N2CC(C(C)NC(C(CC)NC(C)=O)=O)C2)=O)c(C)csc1=O N1(C(c2cc(Br)cs2)C(=O)NC(C(=O)OC)CC(C)C)CCC(C#N)CC12CC2 C1(CC(=O)NC(C(=O)NCC(F)(F)CO)c2ccco2)CC2(CC2)CO1 C(c1ccc2[nH]ccc2c1)=CC(=O)NC(C)C(C)NC(c1cocc1Br)=O Cc1ccc(C(=O)N(C(C)(C(=O)N(C)CC2CCCCO2)C2CC2)C)c(C)n1 Cn1cc(C=CC(=O)NCC2(C(=O)NCC(C)(O)C3(C)CC3)CC23CCC3)cn1 Cc1cc(F)ccc1CC(N1CCCC(CNC(C2CC(C(C)C)=NO2)=O)C1)=O C1(CNC(C(C(C)C)(C)C)=O)CN(C(c2ccnc(F)c2N)=O)CCC1(C)C Cc1cccc(OCOCC(=O)NCC(C)(C)CN(C(=O)CO)C)c1C C(=O)(C(C)S(C)(=O)=O)N(C1CCN(C(C2CCCC(OC)C2)=O)C1)CC O=S1(=O)CC2CN(Cc3ccc(Br)c(Cl)c3F)CC2(c2ccccc2)C1 CC1CN(C(=O)CC2(O)CCCC2)CC1CC(=O)NC1CC(=C2CC2)C1 N1(C(c2c(C)oc(Br)c2)=O)CCN(C(C2CC3CC3C2)=O)CC1C CCCCC(CC)CC(=O)NCC1(F)CC(CNC(=O)CC2CCCC23CC3)C1 c1(C(N2CC(COC)(CNC(=O)CN(C)CCO)C2)=O)cnn2c1CCC2 N1(C(C(CC)=CCCC)=O)CCCC(CCC)(NC(c2cccc(O)c2F)=O)C1 C(CCCCCC(=O)NCCCOC1CCC1)NC(C(C)N(CC)CC)=O c1(CC(=O)NC2C(OCC)CCCC2)ccc(F)cc1F c1(C(=O)NC(CCNC(C(C)OCC2CC2)=O)C)ncncc1N C1(NC(C2(CSC)CCOCC2)=O)CCN(C(C2CCOC2C)=O)CC(C)(C)C1 Cc1nc(O)ccc1C(=O)NCCC(C)N(C)C(c1cccc(CC2CC2)c1)=O N1(C(Cc2n[nH]c(=NC)s2)=O)CCC2C(C1)CN2C(=O)CCOC1CCOCC1 CCC(C)CC(C(=O)N(C)CCC1CC1)NC(=O)C(O)C1CCC1 C1(CCNC(=O)C=Cc2cocn2)CN(C(C2CC(n3ccnc3)C2)=O)CCO1 Cc1nccc(C(=O)NCC2CC(C)CN(C(C3CC34CC4)=O)C2)c1Cl c1(OCC(C)C)ccc(-c2cscc2C(=O)N(C2CC2)CC2CCN(C)CC2)cc1 Cc1cccc(C(N2CCCC2CNC(=O)CC2OCCCO2)=O)c1F c1(OC)ncc(C(N2CCC(O)C2C(=O)Nc2ccc(I)cc2F)=O)cc1F N1(C(c2cc(N)cc(F)n2)=O)CCCC2CN(C(=O)CC3COCCO3)CC12 N1(CC)CCN(C(c2cc(OCc3ccccc3)ccc2O)C(=O)NC)NC1=O C(CS(=O)(=O)c1ccc(C(=O)NCC2CCN(C(=O)CCC3CC3)C2)cc1)OC C1(C)(CC)COCCN1CCc1ccnc(C2CC2)n1 CN1CC(NC(c2cc(Cl)c([N+](=O)[O-])[nH]2)=O)CC12CCCC2 Cc1cc(O)n2ncnc2n1.C(=O)CCC(=O)N1CCN(S(C)(=O)=O)CC1 C#Cc1ccc(F)cc1C(=O)NC(CC)(CC)CCNC(C1(COC)CC1)=O N1(C(CCNC(=O)OCC)=O)CCN(C(=O)NOCC(O)CO)C(=O)C1 c1(C(N2CCN(C(CC(=C)Br)=O)C(C)C2C)=O)ccc2nc(O)sc2c1 c1(C(C2(CNc3nnnn3C3CC3)CCC2)NC(C)C)ccc(C(F)F)cc1 c1(C(=O)NCC(CNC(=O)COc2cccnc2Cl)O)ccnc2cc[nH]c12 c1(C(N(C(C)C(N2CCCC2CN(C)C)=O)CCC)=O)ccnc(OC)n1 CCC(C)C(O)C(=O)N(CCCOCc1ccccc1)C.C(=O)CN(C)CCO c1(N2CCCC(C(=O)Nc3cccc(C(C)C)c3)C2)ncc([N+](=O)[O-])cc1Cl c1(N2CCC(C)C(NC(c3ccco3)=O)C2C)ccc([N+](=O)[O-])cc1Br C1(C)(C(=O)NCC(N(C(c2cc[nH]c2C2CCC2)=O)C)C2CC2)CCC(=O)NC1 C1(C(=O)NC(C(=O)N(CCCC)C(C)CC)(C)C)COCCC1C c1(NC(C2CC(NC(c3ccc(Br)c(Cl)c3)=O)C2)=O)nc(Cl)ccc1O n1(CCCNC(=O)N=c2ccn(Cc3ccccc3)[nH]2)c(=O)oc2ccccc12 C12(CNC(=NCCCSC)NC(C3COC(C)(C)O3)C)CC3CC(CC(C3)C1)C2 C(=O)(C(C)CCCC(C)C)NCC1=CCN(C(C(c2ccccc2)OCC)=O)CC1 C(=O)(C(C)CC(C)C(C)=O)N1C(C(=O)NC2(C#C)CC(F)(F)C2)CC=CC1 c1(C(=O)NC2CC(C)N(C(=O)CCSC(F)(F)F)C2)ccc2oncc2c1 N(C1CCCc2cccnc21)(S(=O)(=O)Cc1ccc(-n2cccn2)cc1)CC c1(C(=O)NC2CCCC(NC(COC(C)C)=O)CC2)cnc2[nH]c(O)nc2c1 CC(C)C(O)C(=O)N1CC(C(N)=O)(CNC(=O)CCc2nnc(S)n2C)C1 c1(OC)ccccc1N(C(=O)CNCc1ccc(COC)o1)C N1(C(c2c[nH]c(=NC)s2)=O)CCC(C)C(N(c2ccccn2)CCCF)C1 N1(C(C(C)NC(C2CCOCC2)=O)=O)CC2CC(NC(=O)Cn3ncnn3)C1C2 c1(CC(=O)NC2CC(F)CN(C(=O)Cc3ccoc3)C2)c(Cl)cccc1Cl C=C1CC2CCC(C1)N2C(=O)C(c1cccs1)NC(=O)CC(CC)C(C)C N1(C(c2cc(Br)c(C)s2)C(=O)NCCCCCC)CCC(O)C(F)C1 CCCCCC(O)CNC(C1C2CC3C(C2NC(C2CN4CCN2CC4)=O)C13)=O N1(C(C(CC=C)CC)=O)CCCC2(C1)CN(C(C1COCCOC1)=O)C2 C1(NC(Cn2c(CC)ncc2)=O)CCN(C(=O)CCCCN2CCCCC2)CC1C c1(C(=O)NC2C(NC(=O)C(c3ccc(Cl)cc3F)O)C2)csc2ccccc12 c1(C(N2CC(NC(CCC(C)N(C)C)=O)C2)=O)ccc2c(c1)CCCS2 CC(C)(C(=O)N1C(CNC(c2cc(Br)c[nH]2)=O)CC2COCC12)S(=O)(=O)C1CC1 C(F)(F)(CN=c1ccc(COC)n[nH]1)c1c(C(=O)OC)ccc(OC(F)(F)F)c1 Cc1cc(C(=O)NCC2CCN2C(=O)CCSCC(C)C)nn1C(C)C c1(-c2c(OC)c(F)ncc2)cc2c(s1)CCN(Cc1ncc[nH]1)C2 c1(C(N2C(CN(C)C(C3CC34CCC4)=O)CC(F)C2)=O)ccnc2c1CCC2 C1(C(=O)NC2CCN(C(c3onc(C)n3)C)CC2O)CC2(C1)CC(C)(C)C2 N1(C(c2c(CC)con2)=O)CC(NC(=O)C(CCSC)NC(N)=O)CC12CCC2 N#Cc1ccc(NCCOC2CC2)cc1S(=O)(=O)NC1CC1 C#Cc1ccc(F)cc1C(=O)NCC1CN(C(C2C3CCC2(C)C3(C)C)=O)C1 c1(C(N(CC(C)C(=O)NC2(C(C)O)CC2)C)=O)cc([N+](=O)[O-])n[nH]1 N1(C(c2cc(C)c(C)[nH]2)=O)CC2CC3CC2C1C3NC(=O)C(C)SC(F)(F)F C(=O)(C1CCc2ccccc21)NC1CC(C)N(C(=O)C(C)Cc2ccccc2)C1 N1(C(C=C(C)C2CC2)=O)CC2(C1)CN(C(C1CC13CCCCC3)=O)C2 c1(OC)ccc2c(c1)OCCC2NC(c1ccc(Br)c2c1OCO2)=O N1(C(CN(C(C(C(CC)C)=O)=O)C2CC(C#N)C2)=O)CCC2(CCOC2)C1 c1(C(=O)NCC2(CCNC(C3CC(CF)C3)=O)CC2)cc(O)cc(Cl)c1 N1(C(C(n2cc(-c3csc(C4CC4)n3)nn2)C)=O)CCC2(CCO2)CC1 c1(C(N(CCC#C)C)=O)ccc2c(n1)CN(C(=O)CC1CCCCC1O)CC2 Cc1cnc2c(C(=O)NC3CN(C(C4CC4(Cl)Cl)=O)CC3O)cnn2c1 N1(C(c2c(CC)nccc2)=O)CC2CCN(C(=O)Cc3nc[nH]n3)C(C2)C1 C1(CNC(c2ccc(Br)cn2)=O)COCCN1C(=O)CC1C=CCC1 N1(C(CNC(C)=O)=O)CC(C)CC1c1cccc(F)c1 N1(C(CCC(C)O)=O)CCCC2(C1)C(NC(C1CCCS1)=O)CCN2C c1(CC(=O)NCCOC2CCN(C(C(CC)n3cncn3)=O)C2)c(C)noc1Cl C1(F)(CNC(CCC)=O)CCCN(C(C2(CC)CCOCC2)=O)CC1 C1(NC(C=C(CCC)C)=O)CC2CCC1CC2NC(C1(C)CCCC(F)(F)C1)=O c1(C(CCC)C)noc(CSc2cncn2C)n1 O=C(C1CCCn2cnnc21)NC1CN(C(c2nc(Cl)ccc2F)=O)C1 Cc1cnc(COCC(=O)NCCOC2CN(C(c3[nH]cnc3C)=O)C2)o1 N1(C(C)=O)CCCC2(NC(c3ccc(Br)s3)=O)CCCC12 C1(CNC(CC(CC)(C)C)=O)CC2(CCOCC2)CN1C(C1CC(C#N)C1)=O c1(C(N2CC(CC=C)(NC(c3cc([N+](=O)[O-])c[nH]3)=O)C2)=O)ccc(F)c(C#N)c1 C=Cc1ccc(NC(N2CCC(C(N3CCCC(C)C3)=O)CC2)=O)nc1F C1(CNC(c2ncc(C)nc2)=O)CN(C(C2(C)CCNC2=O)=O)CCCO1 C(=O)(CS(=O)(=O)C1CCCC1)NCC(CO)NC(=O)CCCC1CCC1 CC1=C(C)CN(C(c2sccc2CNC(c2ccn(C(F)F)n2)=O)=O)C1 c1(CC2N(C(=O)NCC(C(=O)OC)(F)F)CCC2)c[nH]c2ccccc12 C=C(Cl)CCC(=O)N1CC2C(CNC(c3c[nH]cc3-c3csc(C)n3)=O)C2C1 c1(C(N2CC3(CC(NC(C(C#C)(C)C)=O)C3)C2)=O)cc(Br)c2[nH]c(C)nc2c1 c1(CN=C(NCC(COC)F)NC(C)C2CC2)nnc2cccnn12 C(=O)(C1=CC2CCC(C1)C2)N1C(C(N(C)CCc2nccs2)=O)CCCC1 CCCCS(=O)(=O)NC(C)C(=O)NCCN(C)C(c1cc(C(C)(C)C)n(C)n1)=O N1(C(c2cn(CCC)nc2)=O)CCC(C(=O)NCc2cc(C(C)C)no2)C1CC N1(C(C=C(C)C2CC2)=O)CC(C(=O)NCC2(CO)CCCC2)CC(C)C1 C1(N(C(c2cc(COC)no2)=O)C)CN(C(=O)CS(N)(=O)=O)CCC1O N1(C(c2cccc3nonc23)=O)CC2C3CCC(C2C1)N(C(=O)C1=CCCC1)C3 C12(CNC(C(n3c(C)ncc3)C)=O)CCCC1N(C(c1cscn1)=O)CC2 CCCC(CNC(=O)CC1(C)CCOCC1)C(=O)N(CC)Cc1nc(CC)no1 C(CN=c1[nH]c(=NCCC(O)c2ccccc2)[nH]c2ccccc12)NC(C)=O Cn1ncc2c(NC3CS(=O)(=O)CC3NC(=O)C(F)(F)C(O)C3CC3)ncnc12 N1(C(C(CC)C)=O)CC(CO)C2(CCN(C(=O)Cc3c[nH]nc3O)CC2)C1 c1(C(N2CCC(NC(C(C=C)O)=O)C2)=O)ccc(-c2ccc(F)cc2)n1C C1(C(=O)NCC2N(C(CCOCCCOC)=O)CCC2C)CCCC(C)CC1 c1(NCC(C)N(C(C)=O)C)nc(=NC2CC(F)(CO)C2)nc(N2CCOCC2)[nH]1 c1(C(=O)NCCC(=O)NC(C)(C)C)cc(Br)cc2nn(C)cc12 N1(C(C2(S(C)(=O)=O)CCC2)=O)CCCN(C(=O)CCc2cccc(O)c2)CCC1 C(c1cc2ccccc2o1)=CC(=O)NC1CCCC(NC(C(C)(C)C(N)=O)=O)C1 c1(C(=O)NCC2CC(C)N(C(C3CCC3)=O)C2)nc2n(c1Cl)CCCC2 n1(C(CC)C)nnnc1C(c1ncc(I)s1)Nc1cnn(CCOC)c1 c1(Cc2c(C)nc3ccccc3c2)[nH]c(=NCc2cocn2)nc2c1ncn2C CCCCCC(C)(CC)C(=O)N1CC=CC(NC(=O)CSCCCC)C1 C(=O)(CC(P(C)(C)=O)c1ccccc1)NCC1N(C(CCC)=O)CCC1 Cc1ccc2c(CC(=O)NCC(CO)NC(C3CN(C(N)=O)C3)=O)coc2c1 C(=O)(C1=CCCOCC1)N(CC(CN(C(=O)CSc1nncn1C)C)O)C Cn1cc2c(CN3CCC(O)C(C(=O)Nc4cccc(Br)n4)C3)cccc2n1 Cc1cc(CC(=O)NCCOCCn2cc(-c3nc(C4CC4)cs3)nn2)sn1 O=C(CN=c1cc[nH]cc1)NC1CCCC(NC(=O)C(F)(F)C2CC2)CC1 Cc1c(C(=O)NC(C2CCCN2C(=O)C(C)SC2CC2)(C)C)cnn1CCO C=C(C)C(C)(O)C(=O)OC1CC(C(=O)NC2CCCCNC2=O)C1 c1(NC(c2cc(-c3ccccn3)c[nH]2)=O)cccc(C(F)(F)F)c1 Cc1cc(CNC(=O)CC2(O)CCC2)oc1C(=O)NCC1CCCC(C)C1 N1(c2n(C)nnn2)CCC2(CC1)CC(NC(c1cnc3c(cnn3C)c1)=O)C2 c1(C(=O)OC)nn2ncccc2c1NCc1cc(NC(C)=O)cc(C(N)=O)c1 c1(OC)cc(C(N2CC3CC2C3NC(=O)C(C)=C2CCCC2)=O)ccc1C#N C1(C(=O)NCCNC(=O)NC)CCCN(C(c2ns[nH]c2=O)=O)C1 c1(CC(=O)NCCCN(C(c2nnn(C)c2N)=O)CC)cc(F)ccc1OC CCCC(CCCO)C(=O)N1CCC(C)C1CNC(=O)CCCn1cccn1 C1(C(NOCC(C)C)=O)CC2(CC2)CN1C(c1ccc(=N)[nH]n1)=O N1(C(C(COC)Cl)=O)CCC12CCN(C(c1ccc(Cl)c(Br)c1)=O)CC2 C1(C(=O)NC(c2ncccn2)CC)CC(=O)CN1C(c1csc(C#N)c1)=O c1(N2CCC(CC(N3CCC(O)C3)=O)C2)[nH]cnc2nc(Br)cc1-2 C1(CNC(c2ncn(CC)n2)=O)CC(F)(F)CN1C(=O)CN(C)C(=O)OC c1(CC(=O)NCCC2(NC(=O)C(O)CN3CCCC3)CCCC2)cccc(O)c1 C1(=O)CCN(OC)C(=O)C=CC2CCCN12.c1(CC(=O)OC)ccsn1 N1(Cc2cccc(OCC)c2)CCC(NCc2c(C(=O)OCC)cco2)CC1 C(=O)(C(C)C1=CCCC1)N(C1CCCN(C(C2(CC)COC2)=O)CC1)C [N-]=[N+]=NC1(C(=O)NCCC2CC(NC(C3CCN3C3CCCC3)=O)C2)CC1 C(C)(C)(CC(=O)NCC1CN(C(C2CC2c2nc[nH]n2)=O)CCO1)N(C)C c1(C(N(CCCNC(=O)CC2CC2(Cl)Cl)C(C)C)=O)ccc2c(c1)C(C)CO2 C(=O)(C1=CCCC(C)(C)C1)NCC1COCCN(C(c2c(C)onc2)=O)C1 C(C(C)(C(=O)NCC1NC(=O)NC1=O)NC(c1cnn[nH]1)=O)SC C1(CC(=O)NC2(CO)CN(C(c3cc(C)[nH]c3)=O)C2)SC(=N)NC1=O C1(NC(CCNC)=O)(CO)CC(C(F)(F)F)(OC)C1 CC1CCC(C(F)(F)F)N1N1CCN(Cc2nncn2C)CC1 N1(C(C(CC)CC)=O)CC2CCCC(CNC(=O)C#CC3CCCCC3)C2C1 Cc1nc[nH]c1CC(O)C(=O)NC1COCC1CNC(=O)C=CC(F)(F)F C(=O)(CCCCCCCCCO)N1CCC(NC(C2C(CC(C)(C)C)C2)=O)C1 C1(NC(C2N(CC)CC2)=O)CC2(C1)CC2NC(=O)C(COC)COC C1(C(=O)NC(CC(=O)OC)C)CN(C(=O)CCCCC2CC2)CCN1C c1(C(=O)NC(CN(C)C(C23CC(C2)C3)=O)(C)C)cn(C)nc1Cl C1(C(=O)NC(C2(O)CCC2)C)CN(C(=O)C=CC(F)F)C1 CC(C)C(C(=O)Nc1cn(C)nc1C#N)C(C)NC(C1CCC2(CC2)C1)=O C1(OC)CN(C(c2ccco2)=O)CC1NC(C1CCC(C(F)F)CC1)=O C#Cc1cccc(C(=O)NC(CNC(=O)Cc2ccc(Cl)cc2)C2CCC2)c1C N(C1CCOc2c1ccc(Cl)c2Cl)S(=O)(=O)c1c(F)cc(Cl)cc1F C12(C(=O)NC3CC(NC(c4cnn(C5CC5)c4Cl)=O)C3)CCC(CC1)CC2 C1(CC)(CC)CCCN(C(=O)C(N2CCC(c3ncc(C(F)(F)F)[nH]3)C2)=O)CC1 Cc1nc(O)ccc1C(=O)N(CC(C)CNC(c1cccc(O)n1)=O)C C(CCC(C)(C)C(=O)NC(C1CCCOC1)CO)NC(C1N(C)CCCCC1)=O C(C(C)NC(c1ccc(OC2CC2(F)F)cc1)=O)(C(C)C)NC(C=CSC)=O c1(C(N2CC(CC)N(C(C3CCC3CF)=O)CC2)=O)cc2c(s1)CCOC2 Cc1c(C(C)NCC(C2(F)COC2)(C)C)cnn1-c1cccc(Cl)c1 Cn1[nH]c(=NC(=O)NC(Cc2ccsc2)C(=O)O)c2cnccc12 CC1CCCCC1(C)C(=O)NCC1CC(CNC(=O)Cc2c[nH]nc2O)C1 C1(NC(CC2(C=C)CN(C(C3CCC3(F)F)=O)C2)=O)CCN(C)CC1C#N N1(C(c2ccc(C3(C)CCO3)cc2)=O)CC2CC1CCC2NC(=O)CSC1CC1 c1(C(N2CC(C(N=c3ccn(C)[nH]3)=O)CC(F)(F)C2)=O)[nH]nc2c(Cl)cccc12 C=C(C(=O)N1CC2CC2(C(=O)NCCC(C)(C)O)C1)C(F)(F)F C1(n2cc(C(C)NC)nn2)CCCN(C(c2ccc(Cl)c(C(F)(F)F)c2)=O)CC1 CC(C)(N=c1[nH]cc(C#N)c2ccsc12)C(C)(C)c1ccccc1 CC1C(O)CCN1C(=O)CC1CCCCN1C(c1ccc(CO)cn1)=O C1(NC(C2(C)CN(C(C(C)NC(C)=O)=O)C2)=O)CN(C(C)C)CC1C c1(C(N(C2CCCC(NC(=O)C(C)(C)C(F)(F)F)C2)C)=O)cc2c([nH]1)CCCC2 Cc1ccc(C(=O)NC(C)(C)CC(=O)N(C)CCN(C)CCO)c(C)c1 C(=O)(C(CC1CC1)NC(=O)C=CC1CC1)N(CCN=[N+]=[N-])CC Cc1nn(C)cc1C(=O)NC(CNC(=O)CC1(N2CCCC2)CC1)C(C)C C(=O)(CCCC(C)C)N1CC(CCC)C(C(=O)NCCc2cc[nH]n2)C1 c1(C(N2CCN(C(C(C)OC)=O)CC2CCO)=O)cncc2nc(C)[nH]c12 Cc1cc(N)cc(C(N2CC(C(C)NC(=O)Cc3cccnc3Br)C2)=O)c1F C(C)(CC(=O)NC1C=CC(CNC(=O)C=CC2CC2)C1)OC N1(C(c2cc(CC)cc(C)n2)=O)CCC2CN(C(C34CC5CC3C4C5O)=O)CC12 C1(NC(CC(CCC)C2CC2)=O)CN(C(=O)CCC(=O)NCC)CC(C)(C)C1 c1(SC(C(=O)NCC=CCNC(CCNC(CC(C)C)=O)=O)C)cccc(Cl)c1 c1(C(N2CC(CNC(C3C(=C)CC3)=O)C2)=O)nccc2ccccc12 Cc1nn(C)c(C(=O)NC(C)CNC(=O)C(c2ccc(F)cn2)(F)F)c1[N+](=O)[O-] Cc1cc(C(C)C(=O)NC23CC(NC(=O)Cc4cc(C)on4)(C2)C3)cc(F)c1 C1(C(N(CC(=C)C)CC)=O)CC2CC1CC2NC(=O)CNC(=O)OC C1(C(=O)NCC#CCNC(c2c(CSC)cccn2)=O)CC(C)(C)CC(C)(C)C1 C1(C(N2CC(C)C(CO)CC2)=O)CC2CN(C(=O)C(C)OC(C)(C)C)CC2C1 N1(C(c2ccc(N(CC)CC)cc2)=O)CC2CCC2(NC(C2CC(O)C2)=O)C1 C1(CNC(C2OCCN(C)C2)=O)COCCN(C(c2cc(Br)co2)=O)C1 C1(C(N2CC(SCC)C2)=O)CCCC(NC(c2cc(CO)c(C)o2)=O)C1 C(c1cc[nH]n1)=CC(=O)NC(C(N1CCC(n2ccnc2)C1)=O)c1ccoc1 O=C(C1=C(Cl)CC1)NCC1CCN1C(=O)Cc1cc(Cl)sc1Cl C=CC1(CC(=O)NC2(C(=O)OC)CC2)CN(C(=O)CC2CCCN2C)C1 c1(C(=O)NC(CNC(CNS(N(C)C)(=O)=O)=O)C2CC2)cc2c(Cl)cncc2s1 C1(NC(c2c(SC)cnn2C)=O)CCCC(NC(c2cc(C(F)F)no2)=O)CC1 c1(C(N2CCC(Cc3ccccc3)CC2)=O)cc(Br)ccc1Cl CC(C(O)C(F)F)NC(=O)CC1CCCC1NC(c1cc[nH]n1)=O CC1CC(C(=O)NCCCC2CCCN2C(=O)CCc2cnn(C)c2)CC(C)O1 C(=O)(CC1=NN(C)C(=O)C1)NC(CCC(=O)NC(CC(C)(C)OC)C)C(C)C c1(COC(=O)C(C)C(C)O)cccc(-c2cn(C3CC4(C(=O)NC)CC34)nn2)c1 CCC(C)CC(C(=O)NCCC(C)(C)O)NC(c1cocc1C)=O C(CCN(C)C(c1ccnc(CO)c1)=O)(C(C)(C)C)NC(C(C)C#N)=O c1(C(N(C(C)C(N2CCC(SC)C2)=O)CCC)=O)cc(O)n(CC)n1 C12(CCNC(C3CN(S(CC)(=O)=O)C3)=O)CCC1CN(C(c1cc(C)co1)=O)C2 C1(C(=O)NC2(CCOC)CCN(C(=O)C=CC(C)C)C2)CCC2CC2CC1 C1(C)(C(=O)NCC23CC(NC(c4c(F)ccc(C)c4)=O)(C2)C3)CCS(=O)(=O)CC1 c1(C(=O)NCC2(O)CC(NC(C3CC34CC4)=O)C2)ncc(NC2CC2)cc1F C(=O)(CC(C)(C)C#N)NCCC(C)N(C(=O)C(C)N(CC(F)(F)F)C)C C#CCCCC(=O)NCc1ccccc1CNC(=O)C(C)C(=O)OCC CCCCC(C)(F)C(=O)NC(C)C(=O)N(C)CCc1cnc[nH]1 c1(-c2nc(CC(=O)OC)on2)c(C(F)(F)F)cccc1Cl.c1ccccc1 c1(C(=O)NC(C(C)NC(C2C(COC)C2)=O)(C)C)oc2ccc(Cl)cc2c1C N=c1[nH]c(Cl)c(Cl)cc1C(N1CCCC(CNC(=O)CC2CNC(=O)C2)C1)=O C1(OC)CN(C(=O)CCOC2CCCC2)C(C)(CNC(=O)CCF)C1 CON(CCC(=O)NC1CC(C)CCC1O)C(=O)C(F)C1CC2C=CC1C2 N1(C(C=CSC)=O)CC(C2CN(C(=O)CC3CCC34CCC4)C2)C1 c1(CC)cc(C(N2CCCC(NC(=O)Cc3cncn3C)CC2)=O)ccc1OC C1(C(=O)NC(c2ccc(F)cc2)CNC(c2cc[nH]c2)=O)CCCCCC1 c1(C(=O)NC2CC(NCc3cncc(C#N)c3)C2)ccnc2c1OCO2 N1(C(CCCSC(=N)N)=O)CCN(C(C2(C3CCCO3)CC2)=O)CC1 c1(C(N2C(C(C)(C)NC(C3C4COCC34)=O)CCC2)=O)cc(Cl)c(F)cc1O N1(C(C(C2CCC2)NC(C2CCC(C)CC2)=O)=O)CCc2sccc2C1 CC(CCCCNC(=O)C(C1(O)CCOCC1)(F)F)NC(=O)CC1CCCO1 Cc1cc([N+](=O)[O-])ccc1OC1CCN(C(c2cncc(Cl)c2Cl)=O)C1 C1(C(C)(C)CNC(=O)CCOC2CCC2)CCCN(C(c2ccc(F)nc2)=O)C1 N1(C(c2ccc(NC(C)=O)cc2F)=O)CCN(C(=O)C=CBr)C2(CC2)C1 C1(NC(c2cc(CC)ncn2)=O)CC2CC(NC(=O)Cc3ccsc3)C2C1 c1(C(N2CC(O)CC(NC(CC(C=C)(C)C)=O)C2)=O)cnn2ccncc12 N1(C(C(CCC)O)=O)CCCN(C(=O)Cc2cccc(Cl)c2OCC)CC1C c1(C(=O)NCC(C(C)C)NC(C2CC=C(C)CC2)=O)cc(Cl)cc(Cl)n1 c1(C(N2CCC(NC(C3CC(F)C3)=O)C2)=O)cncc(C2CC2)c1 N1(C(C=C(C)C(F)F)=O)CC2(C1)CN(C(c1coc(O)n1)=O)C2 N1(C(C(C2CCN(C(c3c(CC)cco3)=O)C2)F)=O)CCC(F)(CF)C1 C(=O)(CCCC(F)(F)F)N(C)CC1(NC(c2ncncc2F)=O)CC1 C1(C(=O)NC2CN(CC)CC2C)CN(C(c2nnn(C)c2N)=O)CCN1C CC(C)CCC(C(=O)N1CCC(C)(O)C1)NC(C1CC(N=[N+]=[N-])C1)=O C(=O)(C(F)(F)CCn1ccnn1)NC(C(C)C)(C)CNC(C1(C#N)CCC1)=O c1(CC(N2CCC3(C(NC(CCN(C)CC)=O)C3)C2)=O)c(C)nc(O)nc1O c1(C(N2CC(C)C(CNC(c3cc(F)cs3)=O)CC2)=O)cn2cccc(Cl)c2n1 N1(C(C(CNC(c2cc(C(C)=O)[nH]n2)=O)CC2CCCC2)=O)CC2CCC2(C)C1 c1(C(N2CCC(OCCCCCN(CC(=O)OCC)C)C2)=O)cc(CC)c(C)[nH]1 c1(OC)cccnc1CN1CCOCC1C(N1CCC(c2ccccc2)C1)=O c1(OC)ccc(NCCC(=O)NCCC2CCCN2C(=O)Cn2ncnn2)cc1 CC(C1=CCN(C)CC1)NC(C1CC2CN(C(=O)C=CCO)CC2C1)=O CCCCC(C(=O)N(C1CCCCCC1)CCNC(C1CC=CCO1)=O)C(C)C C(=O)(C1CCCn2ccnc21)N1CCC(OC)(CNC(=O)CNC=O)C1 N1(C(CC(C)F)=O)CCOC(C(=O)N(C2CCCCC2O)C)CC1 C1(c2cccc(C)c2)CN(C(c2ccc(-c3ccccc3)nn2)=O)C(C)CO1 S(=O)(=O)(c1ccc2[nH]c(=NCC(F)F)sc2c1)N(CCC(F)(F)F)C Cc1cccc(C2=CCN(C(=O)C(=O)N(C)C(C3CCCC3)C)CC2)c1 C1(CNC(c2c(CC)noc2C)=O)CCCCCN1C(C1CCCOC1)=O C(C(=O)NC(CC(C)C)C(=O)NCC1CCCCCC1)(C(C)(C)C)OC CC(C)CC(C)(C)C(=O)NCC(F)CNC(=O)Cc1ccc2nn[nH]c2c1 C1(F)(CNC(c2c(C)cco2)=O)CCN(C(=O)Cn2ncn(C)c2=O)CC1 N1(C(C(C2CN(C(=O)C(n3ccc(C)n3)C)C2)OC)=O)CCC2(C=CCO2)CC1 C1(O)(C(=O)NC(c2cccc(Br)c2)C)CCN(C(C2CCC(F)(F)C2)=O)C1 c1(NC(C2C(OC)CN(C(c3cncc(O)c3)=O)C2)=O)cc(F)ccc1C C1(N(C(=O)CCN2CCOCC2)C)CCN(C(=O)CCCCn2ccnn2)CC1 c1(CCC(=O)N(C)CC2CCCN(C(C3C(C=C)CC3)=O)C2)c(C)ncnc1O c1(C(=O)NCC(C)CNC(C2(O)CCC2)=O)cccc(C2CC(F)(F)C2)c1 CC1CCC(C(N2CCC(N(C(c3ccco3)=O)CC3CC3)CC2)=O)C(=O)N1 C1(C(N(CCC)CCC)=O)CN(C(c2cc(Br)ccc2C)=O)CCC1(F)F Cn1nc(C(=O)NCCCN(C(C2(CO)CCC2)=O)C2CC2)cc1Cl C12(C(N3C4C(NC(CN(C)C(N)=O)=O)C(CC4)C3)=O)CCC(C)(C(=O)O1)C2(C)C c1(C(N2C(C)C(NC(=O)CCCn3cncn3)CCC2)=O)ncnc2c1CCC2 C1(C(N2CC(C=C)(CC(=O)NCCC(O)C(F)F)C2)=O)CCCCCN1C C#CC1(C(N2CCCC(CC)CC2)=O)CCN(C(c2ccsc2)=O)C1 C(CCCC(=O)N1CC(CC(=O)NOC(C)C)CC1C)SC c1(C(=O)NCC(C)N(CC(N)=O)C)ccc(C(F)(F)F)o1 N1(C(c2c(C)n(C)nc2)=O)CCCC(C)C1CCNC(=O)C=C1CCN(C)C1 N1(C(C(c2ccc(F)cc2)C)=O)CCC(NC(C2CCN2C)=O)C12CC2 C1(NC(c2c(CC)cc(Cl)cc2)=O)CC12CCN(C(=O)C(C)CC(=O)OC)CC2 C12(C=O)CC1CCN2C(C1CC(C)(C)CO1)=O.N12CC(C1)N2C.S(C)(=O)(=O)N c1(C(N2CC(O)(CNC(C(C)NC(C)(C)C)=O)C2)=O)cc(F)ccc1OCCF CCC(C)(C)C(=O)C(=O)NC1CCCC(C(=O)NC(CO)C(=O)N(C)C)CC1 c1(CCC(=O)NCC2CC(O)CN2C(C2CC3CC2C3)=O)c(Cl)cccc1Cl c1(C(=O)NCC(C)(O)CNC(=O)CNS(C)(=O)=O)cc2nc[nH]c2cc1F N1(C(C(C=C)O)=O)C2COCC1CC(NC(=O)CC1CC(SC)C1)C2 N1(CC(N2CCN(C(c3c(C)nncc3)=O)CC2)=O)CC(=O)N(C)C1=O Cc1noc(C)c1CCNC(c1ccnc(Cl)n1)=O c1(OC(C)C)ccc(CN(c2ccccc2Cl)C)cc1C#N.c12nncn1C2 CC1(C)CCOC1C(=O)NCCC1(NC(C2CCCC2(F)F)=O)CCC1 c1(C(=O)NC2CCN(C(C(=O)NCC)=O)C2)ccc(F)c(Cl)c1N N1(Cc2cn(Cc3cc(C#N)on3)nn2)CC2OCCOC2C1 C(C(C)(C)CCl)(c1n(CCCCCC)nnn1)NCCC(=O)N(C)C C1(C(=O)NC2CCCC2)CC2CC2N1C(C1CC1c1ccc(Cl)cc1)=O CC1C(C)N(C(c2nn(C)cc2N)=O)CCN1C(C1CC2(CSC2)C1)=O CC(C)CCC(C(=O)NCCc1ncccn1)NC(c1cc(F)cc(F)c1)=O C12(NC(c3ccc(C)nn3)=O)CCOC(CNC(c3csc(C(C)C)n3)=O)(C1)C2 C(=O)(C(CO)C(F)(F)F)N1C(C)CC(CC(N2CC(=O)NC(C(C)C)C2)=O)C1 CC(C)C(CC(=O)NC(C)(CO)C1CCCC1)NC(C1(n2cccc2)CC1)=O N1(C(C(C)NC(=O)NC)=O)CC(C)(C)CC1CNC(c1ccc(CO)c(F)c1)=O Cc1ccc(C(N2CCCCC(N(C)C)C2)C(=O)NCc2cccs2)nc1Br c1(C(N(CC(CC)NC(=O)C(C)(C)C2CCCCC2)C)=O)scnc1C c1(C(=O)NCC2(NC(C3C(OCC)CC3)=O)CCCC2)ccnc(S)c1 N12CCC3(CCCC3C1=O)CC2.C1(C(=O)NCC2(OCC)CC2)CCCC(=O)O1 C12(NC(C3CCCC3)=O)CCN(C(c3ncoc3C3CCC3)=O)CCC1C2 S(=O)(=O)(c1ccc(C(C)(C)C)cc1)NCC1(CCO)CCC(C)CC1 c1(OC)ccc2c(c1)CCCC2NC(=O)Nc1nc(Br)c(C)cc1Cl c1(C(C)C)n[nH]cc1C(=O)NCc1n[nH]cc1C(N1CCC(CN(C)C)C1)=O N1(C(C2CCCCN(C(CC(=O)OC)=O)C2)=O)CCCC2CCCCC12 CC(C)C(C(=O)N(CCO)CCO)NC(=O)OC(C)(C)C.C12CCCN1C2 N1(C(C(COCC)N=[N+]=[N-])=O)CCC2(CC1)CC2C(N1CC(C(N)=O)(OC)C1)=O N1(C(c2c(C(C)C)ncnc2)=O)CC2CCC(CNC(=O)C(CO)N(C)C)(C2)C1 c1(OCC)ccc2cc(C(C(=O)NCCC#N)N(C3CCCOC3)C)oc2c1 C1(C(=O)NC2CC=C(C)CC2)CC2CCC(C1)C2 C1(NC(C2C(NC(C(C(C)OC)N(C)C)=O)CC2)=O)C2CCCC1CC2 N(C)(C(=NCC1=C(C)OCCS1)NC1CCC1)Cc1ccc(C(=O)NC)cc1 C(C(=O)NOC1CCOC1)(c1ccccc1)NC(C(C=C)OC)=O CC1CCCC(CC(=O)NC2CC3(C2)CC3C(=O)NCC2C3CN(C)CC23)O1 C1(NC(CCNC(COC)=O)=O)CC(C(=O)NC2CC3(CCOC3)C2)=CC1O N12CC3(CCC1CC3)C(=O)N1CCC(C=C)(C1)C2=O.c1(CO)ccccc1CO c1(C(=O)NC(CCOC)CNC(=O)C(O)CC(C)C)ccc2cc(Cl)ccc2c1 C1(NC(CC2CC(SC)C2)=O)CC(CC(=O)NC2(CN(C)C)CC2)C1(C)C N1(C(c2coc(Br)n2)C(=O)NC)CC(C(=O)OC)C2(CCCCC2)C1 C1(NC(C2C(C)OCCO2)=O)CS(=O)(=O)C2CN(C(=O)CCN3CCCC3)CC12 C1(N(CCC(=O)NCCN(C(C2CC2c2cccnc2)=O)CC)C)CCCCCC1 C1(CC)CN(c2ccnc(NCCOCCOC(=O)NC)n2)CC(C)S1(=O)=O CC1CC(C(=O)N(CC(O)CNC(c2cc3c([nH]2)CCOC3)=O)C)CC(C)(C)C1 c1(CC)ncc(C(=O)NC(CCNC(=O)C(c2ccc(Cl)s2)C)C(C)C)cn1 N1(C(c2c(C)nns2)=O)CCCCC1CNC(=O)Cc1ccn(C)n1 C#CCCC(O)C(=O)N1CC(NC(c2c(Cl)n[nH]c2C)=O)C(c2ccccc2)C1 N1(CCC(N2C(CN(C(C(C)SC)=O)CC3CC3)CCC2)=O)Cc2ccccc2C1 C1(C(=O)NC(C(C)C)CNC(c2cncc(Cl)c2)=O)CN(CP(C)(C)=O)C1 Cc1cnnc(O)c1C(=O)NCC1COC(CN=c2[nH]nc(C(F)F)o2)C1 C#Cc1cccc(C(N2CCC2CNC(=O)Nc2ccc(F)cc2C)=O)c1 C(CCO)(C(F)(F)F)NC(C1CC(C)(NC(=O)CSC(F)F)C1)=O N1(C(CCC)CC)CC(c2cn(Cc3cnn(C)c3Br)nn2)C(O)C1 C(=O)(C1=CNC2=NCCCN12)NC1(CO)CCCN(C(C(=O)N(C)C)=O)C1 c1(C(C(=O)NC(C)CC)N(CCOCC)C)ccc(CC)c(C)c1 C1(C(=O)NCCN(CCOC)C(C2SCCCS2)=O)CCC2(CC1)CC2 C1(OC)CC2CN(C(=O)CC3CCC(C)(C)C3)CCN2C1 CC(CO)CCN=c1cc[nH]cc1S(=O)(=O)NC1CC1F C(=O)(C1CCC(=O)c2ccccc21)N1CCN(C(CNC(CC)=O)=O)C(CF)C1 CN1CC(C(=O)NCCCOCCCO)N(C(C23CC(F)(C2)C3)=O)C1 N1(C(C(=O)N(CC)Cc2cccc(Br)n2)=O)CC2C(C1)C2(C)C c1(NC2C(=C)C2)ncc(Br)nc1NC(c1ccccc1)=O c1(CCNC(c2nnnn2C(C)C)C2(COC)CC2)cn(C(C)C)cn1 C12(NC(c3[nH]cc(CC)c3)=O)CC3CCC(C1C2)N3C(=O)CCOC1CCC1 C1(CC)CCN(C(C2CCCC(CF)C2)=O)C1C(=O)NC C#CC1CC1C(=O)N(CCNC(C1CCC1CF)=O)CC CCC(C)CC(C)C(=O)N1CCC(CNC(c2cccc(OC(C)C)c2)=O)C1 C(=O)(CC(C)(C)C=C)NCC1(CNC(C(C)OCC=C)=O)CCCCC1 CC1(C)COC(C(=O)NCC(C)(CO)NC(=O)CC2COCC2(C)C)CO1 C1(CNC(C2(COC)CC2(F)F)=O)CN(C)CCN1C(c1cc(O)ccc1F)=O N1(C(c2ccncc2)=O)CC2CCC(C1)N(C(c1cc(Br)c(F)c(F)c1F)=O)C2 C(CCC(=O)N(CC(C)NC(=O)CCCC1CCOCC1)C)=CC C1(C(=O)NC2CN(C(C3C(C)(C)C3CN=[N+]=[N-])=O)C2)CCC2(C1)N=N2 CC(F)(F)CC(=O)N1CCCCC1CC(N1CCC1N1CCOC1=O)=O N1(C(C2CC(C)OC2)=O)CC(C2CCCN(C(c3cnc(O)nc3O)=O)C2)C1 C=CCCCCCC(=O)N1CC(O)(C(C)NC(=O)C(CO)c2ccccc2)C1 C1(C(N2C(C(N3CC(C(C)NC(C(C)N(C)C)=O)C3)=O)CSC2)=O)CCOCC1 C=CCC(CC(C)C)C(=O)NCC1(NC(=O)CCc2ncccc2C)CCC1 c1(C(N2CC3CC3(C(=O)Nc3cncc(F)c3)C2)=O)c(C(F)(F)F)cccc1Cl Cc1c(C(N2CCC(O)(C(C)NC(=O)CN3CC(C)C3)C2)=O)sc2nccn12 c1(C(N2CCCC(NC(=O)C(=O)N)CC2)=O)c(Br)cc(Br)c(O)c1Br.CC(C)(C)O C12(C(N3C(CNC(C4N(C(C)=O)CCCC4)=O)CC3)=O)CCC(C)(C(=O)O1)C2(C)C c1(C(N2CCCC(C(N(CCCCC=C)C)=O)C2)=O)cccc(Br)c1O c1(CNC(C2CC(OC)CN2C(C2CCN(C)C2)=O)=O)c[nH]c2cnccc12 C12(COC)CN(C(=O)CCCn3cncn3)C(CNC(C3CCOC3)=O)(C1)C2 N1(C(=O)OC)CCC(C(N2CC(NC(C3(N4CCOC4=O)CC3)=O)C3CC23)=O)CC1 N(C1CCCc2c(F)cccc21)C(C=C(C)CS)=O C(=O)(CC(C(F)F)NC(=O)C(c1ccccc1)C)Nc1cnc(C)nc1 C1(NC(CCOC(C)C)=O)CCC(O)CN(C(=O)CN2CCN(C)CC2)C1 c1(C(=O)NCC(CC)NC(C2C3CCOCC23)=O)cn(C)nc1C1CCCC1 c1(C(=O)NCCC2C(C)C2)cc(CNC(=O)Cc2nccn2C)cs1 C1(C(N(CCCNC(=O)CC2CCCC2C)CCC)=O)CC(F)(F)C1(C)C C1(c2ccccc2)(NC(=O)NC(C)C(N)=O)CC(F)(F)C1 CCCCCC(C)(CC)C(=O)NCC1CCN(C(=O)C=CI)C1 C1(O)(CN(C)C)CCN(C(c2ccnc(CNC(C3(C)CCCS3)=O)c2)=O)C1 CC1(C)C2CN(C(c3sccc3NCc3ccc(N4CCCCC4)cc3)=O)CC12 c1(N(C)C)nc2cccc(C(=O)NCC3CCN3C(C3CS(=O)(=O)C3)=O)c2o1 c1(C(=O)NCCCC2N(C(C(C)OCCC=C)=O)CCC2)ccccc1[N+](=O)[O-] C(F)(C(=O)NCCC1CC(NC(=O)C(C)n2cnnn2)C1)OC C1(NC(CSCC(=O)OC)=O)CC2(CCN(C(c3ccns3)=O)C2)C1 C1(C(N(C)Cc2cn[nH]c2)=O)CC12CCN(C(c1cnc(S)nc1)=O)C2 c1(NC(C(C(C)C)OCC)=O)cccc(Cl)c1C.C12COCCC1NC2=O CCCCC(C)C(=O)NC(C)CC(C)NC(c1cn(CCO)nc1C)=O C12(C(=O)NC3(CO)CN(C(C=CC)=O)C3)CCCC1(C(N)=O)C2 N1(C(=O)NC2CCN(c3ccc(C)c(C)c3)C2=O)CC2(CCCC2)C1C(C)C S(=O)(=O)(c1cnn2ccc(=NCc3nccs3)[nH]c12)N1CC(COC)OCC1.C1CCOC1 C(=O)(CC1=NNC(=O)C1)N1CCOCC(CNC(=O)COCC2CCC2)C1 C1(C)(C(N2CC(CC(=O)NCC(C(C)C)O)OCC2)=O)C(C)(C)C1(C)C C(N=c1ccn(CC(=O)NCc2cccc(Br)c2)c(O)n1)c1ccc(C)cc1F C=Cn1nccc1C(=O)NC1(CN(C)C(C2ON=C(C)C2C)=O)CC1 C(CC(F)F)(C(=O)NCC1(C)CCCCO1)N(C(C1CN(C(C)=O)C1)=O)C CC1CC(=O)NC(C(N2CCCC2C2(C(=O)NCC(C)C#N)CC2)=O)C1 C1(NC(c2c(C(C)C)occ2)=O)CC(C)N(C(=O)CC2CC3(CCC3)C2)C1 c1(C(N2C(CN(C(C(C)SCC)=O)C)CCCC2)=O)ccc(F)c(F)c1 C1(C2CCN(C(C3(CC)CC3)=O)C2)CCCCN1C(=O)CCC(N)=O C1(C(=O)NCCNC(c2nccc(CC)c2)=O)CC2CCCC(C1)C2=O N1(C(c2ccn(CC)n2)=O)CCCCC(CNC(=O)Cc2conc2C)C1 CCCCCC(C)CC(=O)NCCOCC(N1CCCCCC1C(C)C)=O N1(C(c2c[nH]c(=NC)o2)=O)CCC(C)(C)C1C(=O)NC(c1ncc[nH]1)CO C1(CC(=O)NC2(C=C)CCC2)CCN(C(=O)C(F)=C(C)C)C1(C)C C1(NC(CC2C(C(=O)NCC3OCCC(C)C3)C2)=O)C2CCCC1CC2 C1(C(=O)NC2CC(C)(CNC(C3CC(O)C3)=O)C2)CCCC(C)(C)CC1 N1(C(CCCCCC=C)=O)CCC2CN(C(=O)CC3CCN(OC)CC3)CC2C1 C1(NC(c2cnc(Cl)s2)=O)CC12CCN(C(=O)CN1CC=CC1)CC2 S(=O)(=O)(c1ccc(Br)cc1)N1CCC(N2CCN(CCOC)CC2)C(F)C1 c1(OC)ccc(F)c2cc(C(=O)NCC(C)CNC(C3(F)CC3C)=O)[nH]c12 N1(C(C(CC#C)C)=O)CCCC2CN(C(C3CC(SC)C3)=O)CCC12 C1(CC)CN(C(c2ccc(C)s2)=O)CC1NC(c1nn(CC)nc1Br)=O N1(C(C2CN(CC)C(=O)C2)=O)CC(NC(=O)CC(C)C)CC12CCCC2 N1(C(c2ccc(CC)s2)=O)CC(CNC(c2ccc(C(C)=O)nn2)=O)CCC1C C1(CNC(C(CC=C)(C)C)=O)CN(C(c2ccc(CC)[nH]2)=O)CCC1(F)F CCC(CC(F)(F)F)C(=O)N(CC(C)NC(C1CC2(C1)CC(C)(C)C2)=O)CC N(C1CN(C(=O)CN=S(C)(C)=O)Cc2ccccc21)C(C(C(C)O)N(C)C)=O CC1(C)CC(C(=O)NC2COCC2C(=O)NCCOc2ccncc2)CCO1 C(=O)(C(C)CS(C)(=O)=O)NC(CC)CNC(=O)CC1CCCN1C(=O)OC C=CCC(C)(C)C(=O)NC1CCN(C(=O)C=Cc2ncc[nH]2)C(C)C1 c1(C(C)=O)ccc(C(=O)NCC2CN(C)CCN2C(=O)C(F)CC(C)C)cc1C C(C1c2ccsc2CCN1C(c1sccc1F)=O)NC(CSCC=C)=O N1(C(=O)NC2CCCCN2)CCc2nc[nH]c2C1c1ccc(F)cc1 C1(C(N2C3(CNC(CC4(C)CC4)=O)CCC2CC3)=O)CS(=O)(=O)CC12CC2 N1(C(C2N(C(C)=O)CCOC2)=O)CCC12CN(C(C1CCCCC(=O)N1)=O)C2 CC(C)CC(C(=O)NCCOCc1ccccc1)NC(=O)C(C)(C)Cl C(C(=O)N=S(C)(C)=O)NC(c1ccncc1C)c1n(CCSC)nnn1 C=CC1CCCN(N2CCN(c3nc(SC)ns3)CC2)C1 CC(C)(C)C(O)C(=O)NC1C2CC(NC(=O)C(C)(F)CC3CCCC3)CC12 C1(C(N2CC3C(CNC(=O)C(C4CCOCC4)O)(C3)C2)=O)(CF)CC2(CCC2)C1 c1(N(CC)CC)cccc(CCC(=O)NC23CC2CN(C(=O)CC(C)OC)C3)c1 CC1(C)COCCC1C(N1CCC(CNC(=O)Cc2csc(C(F)F)n2)CC1)=O CC(C)(C)C(C#N)C(=O)NCCN(C1CCCC1)C(c1cc(Cl)ncc1NC)=O N1(C(C=C(COC)C)=O)CCC(NC(=O)CSC2CCCCO2)C1C1CC1 C12(NC(C(CC=C)NC(C)=O)=O)CCC(CNC(c3ccsc3)=O)(C1)OC2 C1(CC(N2CC=CCC2)=O)CNC2(CCOCC2)CO1.NC(=O)CC(NO)=O C1(C)(CNC(CCC2(C)CC2)=O)CC(F)(F)CN1C(c1cccc(Cl)c1O)=O C1(C(C)C)CN(C(C2COCC2NC(C2CCC3CC2CO3)=O)=O)CCCO1 C1(CC)CCCN(C(c2ccc(CO)o2)=O)C1C(=O)NCC1(O)CCN(C)CC1 N1(c2nc(N3CCC(CCO)C3)cc(C)n2)CCC2(CCCCO2)C1 C(=O)(CC(CC)N(C(=O)C(C)O)C)NCC1(CCC)CCC1 N1(C(CCN(C(C)=O)C)=O)CCCCC1CNC(C1CC(CC2CC2)C1)=O C1(CNC(c2cc(OC)ns2)c2nnnn2C2CC(F)(F)C2)CC(C)(C)C12CC2 C1(NC(C(CC)CC)=O)C2CCN(C(=O)CC3CCCO3)CC12 c1(C(N2C(CNC(CC3C(C(=O)OC)CC3)=O)CC2)=O)cc(Cl)c(Cl)n1C C1(NC(C(C)(C)CC#N)=O)CCC2(CC1)CCN(C(c1conc1C1CC1)=O)C2 c1(CNC(C=C(C)C)=O)ccc2c(c1)CCC2NC(=O)C(F)(F)c1nccs1 CCCC(C(N)=O)N(C1CN(C(=O)CCn2cc(CCOC(C)=O)nn2)C1)C C(=O)(CC(C)C(=O)OC)NCCC1CCN(C(C(CC)CC)=O)C1 N1(C(c2c(C)nc(C)o2)=O)CCC(C2(NC(=O)CN3CCCS3(=O)=O)CC2)C1 c1(C(=O)NC2(CC=C)CCN(C(=O)C=CBr)CC2)[nH]c2c(C)cccc2c1C c1(OC)c(F)cc(C(=O)NCC(C2CC2)NC(C2CCC(C)(C)CO2)=O)cc1Cl c1(C2C(C(N(CCOC)C)=O)C2)noc(C)n1 Cc1csc(=NCC(=O)NC2(C3CN(C(=O)C(O)CCS(C)=O)C3)CC2)[nH]1 c1(C(=O)NC(C)CCC(=O)N2CCC(N(C)C)C2C)cc(O)cc(=O)o1 N1(C(C2CN(C)C(=O)N2)=O)CC2CCC1(CNC(=O)CCCS(N)(=O)=O)CC2 N1(C(C(C)CO)=O)C2CCCC1CC(NC(=O)Cc1ccccc1O)C2 CCC(C)C(O)CC(=O)NCC1(NC(=O)C2=C(C#N)CCC2)CCCCCC1 CC(C(C)C(=O)N1CCC(NC(=O)CSCC2CCCCO2)C(C)C1)S(C)(=O)=O N1(C(C2C(C(C)O)C2)=O)CC(CNC(C2CC2(C)C)=O)C1 c1(C(=O)NCC(C(=O)NCc2ccnn2C(C)C)OC)cccc(Cl)c1 N1(C(C(N2CCC(C)C2)=O)=O)CCCC(O)(CNC(C2CC(N(C)C)C2)=O)CC1 C1(COC)CCC(NC(=O)CC2CC(NC(=O)CSCC(C)C)C2)CC1 c1(C(=O)NC2C(CNC(CNC(C)=O)=O)CCC2)ccncc1Br N1(C(C(n2c(C)ncc2)C)=O)CC2(C(N3CC(C)C3(C)C)=O)CCC1CC2 c1(NC(C)C(C2CCCCC2)NC(C2CCOC2)=O)ncc(C#N)cc1Br N1(C(CC(CC)O)=O)CCC(NC(c2c(C)coc2C(C)(C)C)=O)C(CC)C1 C(=O)(C(CNC(=O)COC1CC(NC(=O)CCCn2cncn2)C1)OC)OC C1(F)(C(=O)NCC2C(C(NOCC3(C)CC3)=O)CCO2)CCOCC1 Cc1c(NC(=O)C(CCC2CC2)NC(c2csnc2Cl)=O)cnn1C N1(C(C(F)=CC)=O)CCC(CNC(c2n[nH]cc2-c2ccccc2)=O)C(C)C1 c1(C(N2CCN(C(C3CC=C(C)CC3)=O)CC2)=O)cccc(Br)c1N N1(C(C)C)CC(C(N2CCC(CNC(c3ccnn3C(C)(C)C)=O)C2)=O)CC1=O Cc1nn(C)cc1CCC(=O)NC1CN(C(c2nocc2Cl)=O)CC1C C1(CNC(C2(CCC)CC2)=O)CN(C(c2occc(=O)c2OC)=O)C(C)(C)C1 C1(C(=O)Nc2c(C)nsc2)(NC(c2cc[n+]([O-])cc2)=O)CCCC1C NC1COC2(CCN(S(=O)(=O)c3cccc(Cn4cnnc4)c3)CC2)C1 C(=O)(C1=CC2CCC(C1)C2)NCC1(CNC(C(CC#C)(C)C)=O)CC12CCC2 c1(C(=O)NCC(C)NC(=O)C(O)CF)cc(C(F)(F)F)ccc1[N+](=O)[O-] C=C(C)CC(C(=O)NC)NC(C)C(=O)NCc1ncoc1C(C)C C1(C(N)=O)CN(C(C2CCCC2NC(=O)C#CC2CC2)=O)CC12CC2 C12(CCOCC1)C(=O)OC2.C1(CCNC(=O)OC(C)(C)C)CCCC1(F)F c1(N2C(C(CC)O)CCC2)nc(=NCc2ccc(Br)s2)[nH]c(C)c1N C(=O)(C1=CCCCCC1)NC(CC#C)C(=O)NCC(C)(O)CN(C)C c1(C(N(C)Cc2cc(Cl)ccc2Cl)=O)cc2c(ncc3ccccc23)s1 C(N=c1[nH]c(=NCCCN2CCC(O)C2)c2ncccc2[nH]1)c1n(CC)ncn1 c1(CNC2C(C(=O)Nc3c(C)ncnc3)C2)c(F)cc(C#N)cc1F N1(C(C(C)C2CCCC2)=O)CC2CC(C1)N(C(c1noc3ncccc13)=O)C2 C1(CC(=O)N(CC(=O)NCCN(CC(F)(F)F)C)CCOC)CC1(C)C C1(c2n(C)ccn2)CN(C(=O)C(F)F)CCN1C(C12CC(F)(C1)C2)=O c1(-n2ncc(C(=O)NCC#CCNC(C(CC)(C)C)=O)c2C)ccc(F)cc1F N#Cc1ccc(CNC2(c3nnnn3CC(F)F)CCNCC23CC3)cc1F C1(N(C)C(c2nnn(-c3ccccc3)n2)=O)CCC(CNC(=O)CCC(N)=O)CC1 C12CC=CCC1NC2=O.C1(CC(C)C)(CNC(=O)NC(COC)C)CCC1 c1(C(N2C(CC(C)O)CCC2)=O)c(Cl)ccc(F)c1N c1(OCC)ccc(C(=O)NCCC2(NC(=O)C3CC3)CC2)cc1[N+](=O)[O-] C#CC1(NC(C2CC(F)CCN2C(c2c[nH]c(=N)c(C)c2)=O)=O)CC(F)(F)C1 N1(C(C(C)(C)C)=O)CC(C(=O)NC23CC(F)(C2)C3)C(F)(F)C1 O=S(=O)(c1cccc(=NCC2CCOC3(CCC3)C2)[nH]1)NCC1(O)CCC1 N1(C(C2N(C(CCCOC(C)=O)=O)CC2C)=O)CC2(CCN(C)CC2)C1 C1(C(=O)NC2C(SC)CCC2)CC(O)CCN1C(c1cc(F)cnc1O)=O C=C1CC(C(=O)NCC(C)C#N)(CNC(=O)COCC)C1 c1(C(N2CCC(NCCO)CC2)C(=O)NC)ccc(OC)nc1C C1(CC)CN(C(=O)COC2CCOC2)CCC1NC(c1ccnc(OC)c1)=O C1(NC(NCC(C(C)C)OC)=NCc2ccco2)CCn2c(C(F)(F)F)nnc2C1 c1(CNC(C(C(C)OC)NC(=O)CC2CNC(=O)O2)=O)nn(C)c(=O)n1C C1(N(C(C(=O)NCC)=O)C)CCN(C(c2cc(Br)ccc2F)=O)CC1C C(=O)(CC(C(F)(F)F)n1ccnc1)NC1CC(CNC(C(C)N2CCC2)=O)C1 N1(C(c2c(C)cccn2)=O)CCC(NC(C2CCC(=O)N2)=O)C(CO)CC1 c1(OCC)ccc(-c2ccc(-c3cnc(C)s3)cc2)cn1.C12CCN(CC1)NC2 c1(NC(c2cnn(-c3ccc(O)nn3)c2C(F)F)=O)nc2ccccc2o1 Cc1ccc(CNC(c2ccn(CC(F)(F)F)n2)=O)c2ccccc12 c1(OC(C)C(=O)NCC(CO)NC(c2cnc[nH]2)=O)ccc(F)cc1 C(=O)(C1CCC(=O)c2cccn21)N(C(CNC(C=C(CCC)CCC)=O)C)CC c1(CC)onc(C)c1C(=O)NC(C)C=CC(N1CC(N2CCOC2=O)C1)=O C(=O)(C1=CCC(F)(F)CC1)NCCCOCCNC(C1CCCC(=O)N1)=O C(C(C(=O)N(CCCOCCNC(C1CC1C)=O)C)C(F)(F)F)OC c1(C(=O)NCC2C(CNC(c3c(CC)nns3)=O)C2)cc2c(O)cc(Cl)cc2[nH]1 CC(N=c1nc2c(cnn2C)c(NCc2ccc(C(F)(F)F)o2)[nH]1)C1CC1 N1(CC)N=C(C(=O)N2CC=CC2CNC(c2cnc(C(C)(C)C)s2)=O)CCC1=O Cc1nccc(C(=O)NC23CC(NC(=O)CC4CCCN(C(C)C)C4)(C2)C3)c1Cl CC(C)CS(=O)(=O)CC(=O)N1CCOCC(CNC(=O)C(F)C2CCOC2)C1 C1(NC(C(CC)C)=O)CCN(C(=O)Cc2cccc(N)c2N)CC12CCC2 CC12CCN(C(c3ccc4ccoc4c3)=O)C1CN(C(=O)C1=CCCOCC1)C2 C1(OC)CC2(CCN(C(C3(C)CC(O)CN3C(c3coc(C)c3)=O)=O)C2)C1 C1(CC(=O)NC(CCOC)CNC(=O)C(C)N(C)C(C)=O)CCCCCC1 C(C(CNC(c1cnn(CCNC(c2cccc[n+]2[O-])=O)c1)=O)C(C)C)OC Cc1ccccc1CC(=O)N(C(C)(C)CC(=O)NCCN(C)CCF)C C1(CNC(C(C2CC2)OC)=O)CN(C(=O)CCc2nc[nH]n2)C2(CCC2)C1 c1(C(=O)NC2CC(CO)NC2=O)cccc2ccc(Br)nc12 Cc1c(C(N2CCCC(C)(CNC(C3CSCN3C)=O)C2)=O)cnc2ncnn12 C1(C(N2CCN(C)CC2)=O)CC2(CCCN2)C1.c12cccc(c1)CN2 Cc1ccc(F)c(CS(=O)C(C)C(=O)N(Cc2ccccn2)Cc2ccco2)c1 N1(C(c2c(C)nn[nH]2)=O)CCCC(NC(c2cn3c(n2)CCC3)=O)C1C CC(=O)C(C)(C)CC(=O)NC1CCC(NC(=O)C2=CCCSC2)C1 N1(C(CN(CCC#C)C)=O)CCC2OCCN(C(=O)C(C)CC)C2C1 N1(C(CSCC)=O)C2CCCC1CN(C(C1Cc3ccccc3C1)=O)CC2 c1(NC(c2ccc(N(C)C)cc2)CC)cccc(F)c1 N(C(=NCCCOS(C)(=O)=O)NC(C)CNC1CCC1)CC1CN(C(C)C)C1 C1(CNC(c2c(NC(C)=O)cc(C)cc2)=O)CC2CCC1N(C(=O)CC#N)C2 c1(CCC(=O)N(C(CC=CCC)=O)CC2CC2)c(C)noc1C C12(NC(CCc3cnc(C)o3)=O)CCCCCC1N(C(=O)CSCC(N)=O)CC2 C1(C(=O)NCC2(C)CCC(NC(CC(CCC)O)=O)CC2)CCc2nccn2C1 C1(NC(C2CC(C)(C)C2)=O)CC2CC(NC(c3ccc(Br)cc3Cl)=O)C1C2 C#CC1CCCN1C(=O)C(CC1CC1)NC(=O)C(C)(CO)OC c1(OC)ncccc1CC(=O)NC1CCN(C(=O)Cn2nccn2)C1 c1(C(N2CCC(C3(NC(C4C=CCC4)=O)CC3)C2)=O)ccc2cnccc2c1 Cc1[nH]nc2ccc(C(=O)N(C(C)CN(C)C(C3CCCCCC3)=O)C)cc12 C1(C(F)(F)C(=O)N2CCC(N(C)C(c3ccncc3Cl)=O)C2)(OC)CCCCC1 N1(Cc2cccc(-c3cccc(-c4nc(O)cc(C)n4)c3)c2)CCc2n[nH]cc2C1 C(=O)(C#CC1CCCO1)N1CC(OC)(CNC(c2ncccc2SC)=O)C1 C1(OC)(CNC(c2ccsn2)=O)CCN(C(c2ccnc(O)c2)=O)CC1 C1(CCOC)CCC(C(=O)Nc2ccc(-c3nn[nH]n3)nc2)CC1 C(=O)(C1=CCN(C(C2CC=C(C)CC2)=O)CC1)NCC1(SC)CCC1 CCCC(C(=O)NCC(C)(C)CC1CC1)NC(C1(OC(C)C)CCOC1)=O C12(NC(C(C)=CC)=O)CCC(CNC(=O)CC3(C#N)CCC3)(CC1)OC2 N1(C(c2c(F)ccc(OC)c2)=O)CCN(C(=O)CNC(N)=O)CC(C)C1 Cc1cc(Cl)cc(N)c1C(=O)NC1CCN(C(=O)C(C)CC(F)(F)F)C1 CC1CC(C(N)=O)CN(C(c2ccc(CNC(=O)C3=COCC3)o2)=O)C1 C=CCC(Cc1ccccc1)C(=O)NCSc1c(C)ccnc1OC C1(NC(CCc2ccc(C)nc2)=O)CC12CCN(C(C1CC1(C)C)=O)C2 c1(C2CN(C(c3cn(C(C)C)nn3)=O)C2)cccc(Cl)c1 C1(CNC(c2c(C)c[nH]n2)=O)CC(C(=O)NC(CO)C(F)(F)F)=NO1 N1(C(=O)CC2CCC=CCC2)CC(C2CCCN(C(C3CCS(=O)(=O)N3)=O)C2)C1 c1(C(=O)NC2C(CNC(c3cc(CC)on3)=O)CC2)ccc(=O)n(CCOC)c1 C1(CNC(c2c(CC)cco2)=O)(OC)CCN(C(c2cccc(CCO)c2)=O)C1 n1(CC)ncc(Cl)c1C(=O)NCC(C)N(C(=O)CC(C)C1CC1)C C(c1cccc(Cl)c1)=C(C(=O)NC1CCN(C(c2c(C)nc(OC)s2)=O)CC1)C c1(CC)cc[nH]c1C(=O)N(CCC(=O)NCCCCF)CCO N1(C(c2cc(C)nc(C)c2)=O)CCC2(CCCN2C(C2CCOC2(C)C)=O)C1 c1(C(=O)NC2CC(NC(C3C4CCN3CC4)=O)C2)ncc(F)cc1F C12(C(N3CCC(C(C)NC(C4CCN(C)C4)=O)CC3)=O)CCC(CC1)CO2 C1(CCNC(CSC)=O)COC(C)(C)CN1C(c1c(Br)cnn1C(C)C)=O C1(CC=C)(CO)CCN(C(c2nc(C)sc2C)=O)C1.C(=O)NCC=CCOC Cc1nc(=NCCN(C(=O)CCC2CCCCC2)CCC2CCCO2)[nH]cc1Br c1(C(=O)NCCN(C(=O)C(N2CCC(C)C2)=O)CC)ccn2nccc2n1 CN1CCCC(CCC(=O)N2CC(Cn3cc(CC4CCCNC4=O)nn3)C2)C1 O=S(=O)(c1cccnc1N1CCC2(C1)CC2(F)F)NCC(F)CO C(c1cccnc1)=CCNC(c1cn(CCNC(CSCCC#N)=O)nn1)=O c1(CN2CCC(C(C)C(=O)Nc3cncc(Br)c3)CC2)cccc2ccn(C)c12 C(C(CC(=O)O)CC(C)C)NC(C(=O)Nc1ccc(OCC)c(Cl)c1)C c1(CN(C(=O)Cn2nccn2)CCN(C(c2n(C)nnc2)=O)CC)cccc(Cl)c1 C(=O)(C1COc2cc(C)c(C)cc21)N(C1CCN(C(=O)CC(C)OC)CC1)CCC C1(NC(C(C)(C)C2CCN(C(=O)C(C3CCCCC3)=O)C2)=O)COCC(C)(C)C1 c1(C(=O)NCC(CNC(=O)CNC(c2ccco2)=O)OC)n[nH]c2c1CCCC2 c1(C(N2CCC(C(=O)N=c3cc[nH][nH]3)C2)=O)cc(F)c(Cl)cc1Cl C1(NC(C(C)OCC(F)(F)F)=O)CCC12CN(C(c1cn(C)[nH]c1=N)=O)C2 O=C(CC(C(F)F)c1ccc(F)cc1)N.C1COCCNC(=O)N1.C(CN(C)C)C1CC1 CCCCCC(O)CC(=O)NC12CC(C(=O)Nc3sc(C)cc3Cl)(C1)C2 C#CCCCC(C)C(=O)NCC(C)(C)CN(C)C(C1CCc2n[nH]cc2C1)=O N1(C(C(C)N(C(c2c(CC)cco2)=O)C2CC2)=O)CCCN(CC2CC2)CC1 c1(SCC#C)cccc(C(=O)NCC2CCCN2C(c2ccnc(C)c2)=O)c1 N1(C(CSCCCC)=O)CCC(CO)(CNC(c2nn(C)cc2C)=O)CC1 C1(NC(C2CC=CC2)=O)CC(C(F)(F)F)CN(C(c2cc(Br)ccc2I)=O)C1 N1(C(c2cnc(OC)s2)=O)CCCCC(N(C)C(C2(C)CCN(C)C2)=O)C1 CC(C)CCCC(=O)N1CCC(C(C)C(=O)NC(CN(C)C)CO)CC1 N1(CC2CCC(CCC(C)C)O2)CC2CCC1CN2C(c1cnn(C(F)F)c1)=O N1(C(C(C)C(C)O)=O)CCOCC(CNC(c2scnc2Cl)=O)C1 N1(C(=O)CCC2CCCCCC2)CCC2CN(C(C3(O)CCOCC3)=O)CC12 c1(CNC(C2CCC(C)C2)=O)nc(CNC(=O)CS(C)(=O)=O)cc(O)n1 CCC(C)(CNC(=O)CC1CN(C(C2CCC3(CC3)C2)=O)CCO1)CO C(CC(N)=O)(C(=O)NC1CCCC1CN(C)C)NC(c1nccc(OC)c1)=O c1(OC)cc2[nH]cnc2cc1C(N1CCCC(C)(OC)C1)=O C1(CCC(=O)NCCn2ncc(C)c2)CCCCN1C(=O)CC(C1CC1)C1CC1 c1(C(C)(C)C)ccc(C(N2CCC(NC(C3CC(C)(CN)C3)=O)CC2)=O)c(N)c1 N1(C(c2ccc(OC)cn2)=O)CCC(C(F)(F)F)C(NC(C23CC(C)(C2)C3)=O)C1 Cn1cc([N+](=O)[O-])cc1C(=O)NC1CC2C1CCN2C(C1CCC2(CC1)CC2)=O Cc1ccc(C(N2CC(C3CCN(C(C4CC5CC(=O)C4O5)=O)CC3)C2)=O)c(O)n1 c1(C(=O)NCC(C)CNC(C2CCOC2)=O)ccc(CN2CCCC2)[nH]1 Cc1cccc(C)c1CNC(=O)C(N1CCOC(C)(C(F)F)C1)CCOC(C)C N1(C(C(C(CC)O)C)=O)CCC=C(C(=O)NCC2CC(F)(F)C2)C1 CCCCC(O)C(=O)N1CC(CC(C)NC(=O)C(C)C(O)Cc2ccccc2)C1 C1(C(=O)Nc2cn(C)nc2)CCC(NC(=O)CCN2CCOC2=O)CC1 c1(CNC(C2C(NC(C3COCC(C)O3)=O)CC2)=O)cccc2ccnn12 c1(C(N2CC(C(C)NC(C3(C)CCCCO3)=O)C2)=O)ccc(O)c(Cl)n1 Cc1cc(CC(=O)NCC(C)N(C)C(C2CC3CC3C2)=O)cc(C)c1Br N1(C(CC(CCC)C)=O)CC2CCC(C1)N2c1ccccc1.C1CC2(CCC2)CO1 c1(OC(C)C)ccc(S(=O)(=O)NC(c2nc3cccc(Br)c3[nH]2)C)cn1 c1(N2CC(CC=C)(NC(c3cncc(C)c3)=O)C2)ncnc2c1ccn2C1CC1 N#Cc1cc(CNCC2(Nc3ccnc(C4CC4)n3)COC2)ccc1Br Cc1cc(CN2CCC(CNC(c3ccnn3CC3CCC3)=O)C2)no1 c12ccc(cc1)[nH]2.c1(N2CC(CNC(c3n(C)ccc3)=O)C2)ncc(Br)cn1 Cc1onc(C(=O)NC(C)C(C)NC(=O)CCc2ncc(F)cn2)c1[N+](=O)[O-] N1(C(CCC)=O)CC(NC(=O)CC(C)(C)CC)CC2(CC2)C1 c1(NC(N(CC(=O)NC2CC2)C)=O)csc(C#N)c1.C12CC1CNC2=O c1(C(=O)NC(CC)CNC(=O)CC(c2cccs2)NC(C)=O)cc(C)cc(F)c1 CC1=NNC(=O)C1CC(=O)NCC1(F)CCC(CNC(c2ccc(F)cn2)=O)C1 c1(NC(C)=O)ccc(F)c(C(=O)NCC(C)NC(C23CC(C2)C(C)(C)O3)=O)c1 C1(CC)C(C(=O)NC2CC(CO)C3CC23)CCCN1C(=O)C(C1CCOCC1)F c1(CSC)cc(C(=O)N(CCCNC(C2CC2(C)Br)=O)CCO)sc1C C(=O)(C1=C(Cl)CCC1)N(C1CN(C(C2(n3nccn3)CC2)=O)CC1F)C C(C(CC(C)(C)C)N(C=O)CC1CC1)OC CCC(C)C(C(=O)NCC1CN(C(=O)C2=NOCC2)C1)NC(N)=O C(C(=O)NCCCC1CCCN(C(=O)COCCCF)C1)(C(C)C)OCC C1(C(C)C)(C(=O)O)CCN(CC2CC(C)CO2)CC1 N#Cc1cccc(F)c1C(=O)Nc1csc(CN=c2[nH]cncc2F)n1 N12CCC(CC1)OC2=O.c1(CN(C(C)(C)C)CCO)cn(C(C)(C)C)nn1 c1(CNC2CCN(C(c3ccn(C)n3)=O)CC2F)cc(F)c(C#N)c(F)c1 c1(CC(N2CC(NC(C3C(CCC)C3)=O)C(C)C2)=O)cccc(Cl)c1F CCC(C)C(O)C(=O)NCC1(NC(=O)C#CC2(C(F)(F)F)CC2)CCCCC1C C(=O)(C1SCCc2ccccc21)NCCC1CC(NC(c2c(N)nccn2)=O)C1 CC(CC(=O)N1CCCC1(C)CNC(=O)COCc1ccncc1)C(F)(F)F Cc1nc(N2CC3CCC2CN3C(C2CCS2(=O)=O)=O)ccc1C#N c1(C(N2CCC(N(C(c3cccc(C)c3Cl)=O)C)C2)=O)ccc2c(c1)COCC2 c1(C(N2CCCN(C(C(C)C)=O)CC2C(C)C)=O)cc2cc(F)cc(F)c2o1 N1(C(CC=CC)=O)CC(CC(=O)N(CC)Cc2ccccc2)CC1C c1(C(N(CC(C)NC(c2ccccc2)=O)C)=O)cncc2cnccc12 N1(C(c2ncc(C)o2)C(=O)NC2CCC2)CCC(C2CCCC2(C)C)C1 C1(C(=O)NOCCCC2CC2)(OC)CCc2cc(Br)ccc2C1 N1(C(CCOC)=O)CCC2(CC1)CN(c1cccc(F)c1C#N)CCO2 N1(C(C(C=CC)O)=O)CCN(C(=O)CCCc2nc3ccccc3o2)CC(O)C1 C1(COC)(NC(c2cnc(O)o2)=O)CCCN(C(c2cccc(OC)n2)=O)C1 C1(F)(C(=O)NCCC2(O)CN(C(C3CCC(C(N)=O)C3)=O)C2)CC=CCC1 O=C1C(CN2CCCCCC2)CCCN1S(=O)(=O)Cc1cccc(Cl)c1O C12(NC(c3c(CC)noc3)=O)CCCC1CN(C(=O)C1=CC(C)(C)C1)C2 Cc1ccc(=NCCC(=O)N(C)CC2CCCCN2C(=O)C(O)C2CCC2)[nH]c1 N1(C(C2(SC)CCC2)=O)CCC(C)C(CC(=O)NCc2cc(C)on2)C1 O=C(C1=CCN(C(C2(C3(O)CCC3)CC2)=O)C1)NC1CCOCC1 C1(C(=O)NC(c2ccnc(F)c2)C)(NC(C2C(C)(C(C)C)C2)=O)CCOCC1 C(CCC(C)C)=CSCC(c1nccs1)C [N-]=[N+]=NC1CC(C(=O)NC2CC(CNC(c3ccnn3CCCO)=O)C2)C1 C(=O)(CCS(N)(=O)=O)NCC(N(C)C(C1CN(S(C)(=O)=O)C1)=O)C1CC1 CCC(C)(C)CCCC(=O)NC(C)C(C)C(=O)NC1CNC1 C1(NC(c2ccncc2O)=O)CC2(C1)CC(C(=O)NCc1ccc(F)cc1O)C2 N1(C(c2occ(C(=O)OC)c2)=O)CCCC(C(=O)NCC2(CO)CCCC2)C1 C(=O)(C#CC1CCOCC1)N1CCCN(C(C(CC)OC2CCCC2)=O)CC1 c1(NC)ccc([N+](=O)[O-])cc1C(N1CCC(C)C(NC(=O)CCCCOC)C1)=O c1(OC)ccc(-c2nc(C3CCC(C)C3)n(-c3ccnnc3)n2)nc1 C1(C(N2C(CN(C(C3CC=C(C)CC3)=O)C)CCC2)=O)CCCCCN1C C1(C(=O)NC2CCC(NC(=O)CC3CCC(=O)N3C)C2)(OC)CCCCCC1 N1(C(CC(CC)(F)F)=O)CC2(CCN(C(c3cc(Br)n[nH]3)=O)CC2)CC1C c1(OC)ncc(NC(C2(C)CCN2C(c2[nH]cnc2C)=O)=O)cc1F C1(NC(CCC(=O)NC)=O)C2CC3CC(C2)CC1(CNC(=O)Cc1cnsc1)C3 C1(C(=O)OC)(COC)CCCCN1C(c1cc(F)ccc1C)=O N1(C(C(CO)NC(N)=O)=O)CC2(C1)CN(C(=O)CC=Cc1ccccc1F)C2 C#Cc1ccc(C(=O)NCC(C2CC2)NC(c2sc(C3CC3)nc2C)=O)cc1F c1(NC(c2n(CCOC)nnn2)(C)C(C)OC)ccc(Cl)c(C(=O)OC)c1 S(=O)(=O)(c1c(C)nn(C)c1C)N1CC(CC)N(Cc2cc(C)nc(C)c2)CC1 C=CC(CCC)CC(=O)NC(CCSC)C(=O)NCC1CCCSC1 N1(CC(=O)NCC2CC(C(N)=O)C2)CCCCC1CNn1ccnn1 N1(C(c2cc(Br)ccc2F)=O)CCCC2C1CCN2Cc1ccc(F)c(F)c1F c1(NC(C2(CC)CCOC2)=O)ccc(NC(=O)C(C)C(C)(C)C)cc1C S(=O)(=O)(c1cccc2cccnc12)N1CCC(CC(N2CC(C)N(C)CC2)=O)C1 C(=O)(CC(C(F)(F)F)c1ccccc1)N(C1CCCN(C(C2OCCO2)=O)C1)C N1(C(C(CC)N(C)C)=O)CCC(C)(CNC(C2CC3(CCC3)C2)=O)C1 c1(C(=O)NC2C(NC(c3cnnc(O)c3)=O)COC2)n[nH]c2c1COCC2 c1(C(N2CC(O)(CNC(c3ccc(C(C)C)cc3)=O)C2)=O)[nH]nc([N+](=O)[O-])c1Cl N(C)(C1CN(C(=O)C=CSC)CCc2ccccc21)C(CCOCCCOC)=O N1(C(c2c(CC)c[nH]n2)=O)CCN(C(c2ccccc2CO)=O)CC(C)(C)C1 C1(NC(C2CCC(CNC(c3cc(C#N)[nH]c3)=O)O2)=O)CCc2nn[nH]c2C1 N1(C(C(C=C)CC)=O)C2CC1CN(C(=O)CCC(C)N(C)C)C2 C12(C(=O)NCC3N(C(C4COC5COCC45)=O)CC(O)C3)CCC(O)(CC1)CC2 C=C1CCN(C(=O)C(C)C(F)(F)F)C(C(N2CC(c3nncs3)C2)=O)C1 O=[N+]([O-])c1cnc2c(F)cccc2c1Oc1c(Cl)cc(C(=O)O)cc1Cl c1(C(N2C(Cn3cc(CC=C)nn3)C=CC2)=O)ccc(C(F)F)c(C(F)(F)F)c1 N#Cc1cc(F)c(C(=O)NC2CC(CNC(c3cn[nH]c3)=O)C(O)C2)c(F)c1 C(CC(=O)NC1CC(NC(=O)C(C)Oc2cccc(N)c2)C1)(C(F)(F)F)OC CCS(=O)(=O)NNC(=O)c1c(F)cncc1Br C(=O)(CCCCCS(N)(=O)=O)N(CCOC)CCNC(CC(=C=C)C)=O CC1CN(C(c2cscc2C2CC2)=O)CC(C)N(C(=O)CN2CCC(O)CC2)C1 C=CCC(C)(CC)C(=O)N1CC2CCC2(CCNC(c2ccn(C(F)F)n2)=O)C1 C12CCN(CCC(C(F)F)C3(CC)CCC(C)(CO3)NC1=O)CC2 c1(C(=O)NC(C(C(C)C)NC(=O)C2=CCCCO2)C)ccc2nsnc2c1 C1(CN(C)C(C2CCC2)=O)CCN(C(C2CCCN(c3cnccn3)C2)=O)CC1 C(C(O)C(=O)NC(C)(C)C(=O)N(C)Cc1ncn(C)n1)N(C)C C(C(C)(C)C(C)(C)C)NC(CC1(OC)CN(C(=O)CSCC(F)F)C1)=O O=S(=O)(c1ccc(O)nc1)N1Cc2cnc(C3CC3)nc2C1 C1(NC(CN(C)Cc2ccccc2)=O)CCCC1(C)CNC(C1CC2CC2C1)=O C(=O)(CCCCCC(C)C)N1CC(N(C(CCC(C)(C)OC)=O)C)C(C)CC1 CCCCC(CN(C(=O)CNC(c1ccc(F)cc1)=O)C)CC C=CCCC(C)(C)C(=O)N1CCCC(C)(NC(c2cnn(CC=C)c2)=O)C1 CN1CC=CCC1CC(=O)NC1CCCC1CNC(C1(C)CNC(=O)C1)=O c1(C(N=c2cc(C)o[nH]2)=O)ccc2c(-c3ccc([N+](=O)[O-])cc3)nn(C)c2c1 N1(C(c2cc(CNC(C3(C)CC3(F)F)=O)on2)=O)CC2CCC(C1)O2 CC1CC2CN(C(C3(NC(=O)CCC4CC(C)C4)CC(CO)C3)=O)CCN2C1 C1(C(=O)Nc2cn(CC)nn2)CC(O)CN1C(c1ccc(SC)cc1)=O c1(OC)nccc(C(=O)NCC2CC2CNC(=O)C=Cc2ccc(C(F)F)o2)n1 C1(C)(C(=O)NC(CCOC)C(C)C)CC(O)CN1C(c1ccc(F)c(O)c1)=O N12CCC3(CC1)CC(CO3)C(=O)Nc1cnc(Br)cc1C2=O.C(C)(C#N)OC N1(C(CC2N(C)CC=CC2)=O)CCCC(C)(C)C1CNC(=O)C(F)=C1CCCC1 CC1=C(C(=O)NC2CC(OCC(=O)NC3C4COCC34)C2)CCCO1 C1(CN(C(C2(C)CC2(C)C)=O)CC)CCCN(C(=O)CC2CN(C)C2)C1 C(=O)(CC(C)(O)COC)NCC(CC)NC(c1sccc1C(C)=O)=O C1(NC(COC(C)=O)=O)CCCC12CCN(C(c1occc1C(C)C)=O)C2 C1(CC(=O)NC2(CN(C(=O)CSC(F)(F)F)C)CC2)CCOC1=O CCCCC(CC)CC(=O)NC(CC)CCC(=O)NCc1nnc(O)o1 N1(C(c2c(CC)sc(=N)[nH]2)=O)CC2(C1)SCCC2NC(=O)CC1C=CCC1 N1(C(CCC(=O)OC(C)(C)C)=O)CCc2ccc(Br)cc2C1C(F)(F)F c1(CC)cccc(CC)c1CC(=O)NC(C)CCN(C(=O)Cc1ccn(C)n1)C c1(NC(CCC=C)(C)c2nnnn2C(c2ccccc2)C)ccc(C)c(F)c1 c1(C(=O)NC(CC=C)CNC(=O)C(C)NS(=O)(=O)CC)ncc(CC)cn1 N1(C(C(C)SCC)=O)CCC(NC(c2cccc(C(=O)NC)n2)=O)C2(CCC2)C1 C1(C(=O)NC(C#C)(C)CC)CC2CC2N1C(=O)CN1CC=CC1 N1(C(C2(CC)CCNC2=O)=O)CCC2CN(C(=O)C=CBr)CC2C1 c1(C(N2CC=CC23CCCC3)=O)coc2c(Cl)cc(Cl)cc12 N1(C(c2c(CC)nn(C)c2)=O)CCN(C)C(CNC(C2(O)CCSC2)=O)C1 C(C(C)(C)CNC(c1cnc[nH]1)=O)N(C(=O)C(F)(F)c1ccnn1C)C c1(C(=O)NC2(C)CCN(C(c3c(Br)cc(C)s3)=O)C2)cccn2nncc12 c1(CC(=O)NCC(C)CN(C)C(C2CCCCC2O)=O)ccc2c(c1)CCO2 Cc1ccc(OC(F)F)cc1C(=O)NCC(C(C)C)NC(=O)CNC=O N1(C(c2c(OC)cnc(Cl)c2)=O)CC=C(C(=O)NC2COCCC2OC)CC1 N1(C(C(CNC(COC2(C#C)COC2)=O)O)=O)C2CCCC1CC2 N1(C(C2C(CC)OCCC2)=O)CCCN(C(=O)C(C)(C)CN2CCOCC2)CC1 C1(N(C(C(C2CCOCC2)C)=O)C)CCN(C(c2coc(Br)c2)=O)CC1 C1(C)(C(=O)NCC(CCNC(C2(OC(C)C)CCC2)=O)O)CCN(C)C1=O c1(C(=O)NCC)ccc(C(=O)NC(C)C(c2ccc(Br)cc2)OC)cc1 N1(C(C(CO)N(C)C)=O)C2CCC1CC(N(C(=O)Cc1cncnc1)C)C2 Cc1[nH]nc(C(=O)N(CC(=O)NC2C(=O)OCC2CO)C)c1C CC1CCn2ncc(C(=O)OCC(c3c(Cl)nc4ccccn34)=O)c2C1 N1(C(Cc2cnc(C)o2)=O)CCCC(C2CC2NC(C2(C)CCC2)=O)C1 C1(C(=O)N(CCO)Cc2ccccc2)COCCN(C(=O)Cc2ccc(CO)o2)C1 c1(CC)cccc(C(=O)NCCn2cc(COC3CCOC3)nn2)c1F Cc1cnc(F)c(CNC(C2CC23CC(NC(C2CC2C#N)=O)C3)=O)c1 c1(CC(N2C(CN(C)C(c3cccc(C4CC4)n3)=O)CCC2)=O)ccc(N)cn1 c1(C(=O)NCCCCCCNC(C2C(C=C)(C(F)(F)F)C2)=O)c(C)nc(C)n1O CC1(C)CCC(CNC(=O)CS(=O)(=O)CCO)N(C(C2CCC(C(N)=O)O2)=O)C1 c1(C(=O)OC)ccc(Cl)c(C)c1OCCC1CC(C)C1 C1(C(=O)NCC(F)CO)COCCN(C(c2ccccc2O)=O)C1 C=CCC(CC=C)C(=O)N1CCC1CNC(=O)C=Cc1ccc(F)c(Cl)c1 c1(C(c2n(CC=C)nnn2)NCc2ccc(OC)cn2)cccc(C(N)=O)c1 C(=O)(C1=CCC(F)(F)CC1)N1C2C(CNC(c3c(C)nc(C)[nH]3)=O)CC(CC2)C1 c1(C(N2C3CCN(C(CS(N)(=O)=O)=O)C(C3)C2)=O)nncc2c1CCCC2 c1(OC)ccc(NC(C2CCN(C(=O)Cn3nc(C)cc3C)C2)=O)c(C)n1 C1(NC(C(=CC2CCCC2)C)=O)CN(C(C2(C#N)CCOCC2)=O)CCC1F CCC(C)(C)C(=O)C(=O)NOCC(=O)NC(c1ccccc1F)CO C(C(=O)NC1CCCCC1NC(c1nc(C)oc1OC)=O)(C(C)C)OCC n1(CC(=O)N(CC(C)(C)CNC(=O)Cn2cncn2)C)cc(S(C)(=O)=O)cn1 N1(C(C2CC(C#C)(O)C2)=O)CC(NC(=O)C(F)n2cccn2)CC2(CC2)C1 C(=O)(CC(C)COC)NC(CC)CNC(c1cnc(C(C)=O)s1)=O Cc1cc2c(cc(C(=O)NC3C(O)CC3O)n2CC(F)(F)F)s1 Cc1cc(C)c(C(=O)NCC(F)CNC(c2[nH]c(=N)ccc2C)=O)c(C)n1 C1(CC)CN(C(c2cn(CCNC(C3SCCS3)=O)cn2)=O)C(C)CO1 CC(C(=O)NCC1CC(F)CN1C(c1cc(Cl)cnc1O)=O)C(F)(F)F Cc1nc2ccc(C(C)NC(=O)C3=CCC(C)CC3)cc2o1 C1(C(=O)NCC2(C(N3CCCC3C(F)F)=O)CCC2)CCCC2CCCCC12 c1(C(=O)NC(CN(C(c2cn[nH]c2)=O)CC)C)ccc(OC2CC2)cc1 C1(N2CC(N3c4cc(on4)C3=O)C2)CC2CCCCC2NC1=O.CCOCC O=C(C1=CCCOCC1)NCCCNC(=O)CC1CCCC(O)C1 C(=O)(C(F)C(F)(F)F)N(C1CCN(C(=O)CNS(C)(=O)=O)CC1)C c1(OC)ccc(CN(C(=O)C(C)(N)CC2CCC2)Cc2cccnc2)cc1 c1(C(=O)NC2CN(C(C3(CC)CCCC3O)=O)C2)cc(F)cc2nn[nH]c12 c1(CN2C(CN=c3ccnc(N(C)C)[nH]3)CCC(C)C2)nn(C)c2ccccc12 C1(CC)CN(C(c2ncccc2Br)=O)CCC1NC(=O)CC1CCOCC1 c1(C(=O)NC2CC(C)N(C(c3cc(Cl)ccc3N)=O)C2)nc2ncccn2n1 C1(C)(CNC(C2(OC)CCCOC2)=O)CCN(C(=O)CNS(=O)(=O)N(C)C)CC1 Cc1cc(C(N2CCCC(c3nc(C)cs3)C2)C(=O)NC(C)C)cc(F)c1 CC1CN(CCCCNC(=O)C(=O)NCc2ccc(F)cc2F)CC(C)O1 C1(NC(C(CNC(c2ccccc2O)=O)O)=O)CC(O)C(O)C1 c1(OC)ncc(C)c(C(=O)NCC2CCN2C(=O)C(N2CCC(C)CC2)=O)c1Cl c1(CCCC)ocnc1C(=O)NC(C)(CNC(C1CC2CC2C1)=O)CO C=CC(C)(O)C(=O)NC1CC(NC(=O)C=CC=CCC)C1 C(CC(C)(C)CC(=O)N1CC2(C(N3CCC3(C)C(=O)NC)=O)CC1CCO2)OC CCCC(CNC(C12CN(C(=O)C(C)(C)C)CC1(C(F)(F)F)C2)=O)CCO C1(C(N2CCC(NC(=O)NC)C2)=O)C2CCC(C2)N1C(C1CC(C)C1)=O C(=O)(CCCCCCNC(c1cc(C)[nH]n1)=O)N1CCCC1.N(C)SC C1(C(=O)NCC2CCCC2NC(c2nonc2N)=O)(COC)CC1(F)F CC1CN(Cc2ccccc2)CC1C(N1CCC1NCCCc1ccco1)=O Cc1ccc(F)c(C(N2CSCC2C(=O)NCCCOCC(F)F)=O)c1 N1(C(C=CS(C)=O)=O)CC(NC(=O)CCCC2CCCCC2)CC1(C)C c1(NC(=O)OC2(OCC)C(C3CCCC3)(OCC)C2)ccc2c(c1)C(=O)CCC2 C(=O)(C(C)(F)CC1CCCC1)N(CCN(C(c1ccc(CC)[nH]1)=O)C(C)C)C N1(C(C2OCCC(C)C2)=O)CCCC(C2CN(C(C3(F)CCN(C)CC3)=O)C2)C1 N1(C(CCCN(C(C)C)C)=O)CCC(C)C(NC(c2cnc(N)c(Cl)c2)=O)C1 N1(C(c2occ(C)c2)=O)CC2(CCC2)CCC1CNC(=O)Cc1ccc(Cl)cn1 C#Cc1ccc(C(=O)NCC(C(C)(C)C)NC(=O)C=CS(C)=O)cn1 N1(C(c2ccc(OC)nc2)=O)CC2(CC2)CC1CNC(C1CNC(=O)C1)=O C(=O)(C(CC(F)F)NC(C1CCCC(CF)C1)=O)NCC1(COC)CC1 N1(C(C2CCN(C(c3cc(CC)oc3C)=O)CC2C)=O)CCCC2(CC1)CC2 N1(C(CC(c2ccc(C)cc2)(C)C)=O)CC2(CC(NC(C3(CCO)CC3)=O)C2)C1 c1(C(=O)NCC2CC(CNC(C=C(C)Cl)=O)OC2)ccc2ccncc2c1 C1(C(=O)OCC)CSCCN1C(c1nc(C)cs1)C(=O)NCCCOC N1(C(CC(=O)OC)=O)CCC2(CC1)CC2NC(C1CC=C(C)CC1)=O c1(C(=O)NC2CC(C(C)C)OC2)cc(Cl)c(Br)cn1 c1(CC)cccc(F)c1C(=O)NC1(C2CCCN2C(=O)CC(C)C(=O)OC)CC1 N1(C(CC2C(OCC)COCC2)=O)CC2CCC(C1)N2C(C1CC=CC1)=O C=CCCC(C(=O)N1CCCC(C)(O)C1)NC(c1c[nH]nc1C)=O Cn1cccc1C(=O)NCC(C1CCCC1)NC(c1ncoc1C(C)(C)C)=O c1(C(=O)NC(C2CCN(C(C(F)=C(C)C)=O)C2)C)ncccc1C c1(C(=O)NC(C)CCN(C)C(c2ccoc2CC(N)=O)=O)cc2cccn2cn1 c1(C(N(C2CCN(C(=O)CNC(=O)C3CC3)C2)CCC)=O)cn(C(C)C)cn1 Cc1ccc(C(N2CCCC(C)(NC(c3cc(Cl)c(Cl)[nH]3)=O)C2)=O)c(C)n1 c1(CN2CC(CC(N3CC(C)CC(COC)C3)=O)C2)cccc(Cl)c1[N+](=O)[O-] CC1CN(C(=O)C(n2ccc(Br)n2)C)CC1CNC(c1cnccn1)=O N#CC(C(=O)NCC1CCCN1C(c1cnc(Cl)s1)=O)C1CC1 n1(CCC)ncc(C(=O)NCC(C)(CO)NC(c2cccn2CC)=O)c1C1CC1 n1(CC(=O)N(CCNC(=O)CCc2ncc[nH]2)CC)cnnc1O.C1CS1 CCCC(CC)C(=O)NC(CNC(c1cc(C)n(CCO)n1)=O)CC(C)C C1(CCCNC(=O)Cn2cnnc2)CCCCN1C(=O)Cn1nnc(=O)[nH]1 CCCCCCC(CC)C(=O)N1CCCC1C1(NC(=O)C(CC)CCOC)CC1 c1(CC)nc(C(=O)N(C)CC2CCN(C(c3cnc(O)n3CC)=O)CC2)c(C)o1 c1(OC)ccc(C)cc1C(N1CCC(C)(C)C1CNC(=O)CC12CCCC1C2)=O C1(CN(C(C2C3CCC(=O)C23)=O)CC)CCCN(C(=O)CNS(=O)(=O)N(C)C)C1 c1(C(=O)NCCCN(C(C)C)C(C2CCOC(C(C)C)C2)=O)cccc[n+]1[O-] N1(C(C=Cc2ccc(CC)o2)=O)CCN(C(C2CCCC(CC)C2)=O)CC1CC C=CC1(C(=O)NCc2c(C)n[nH]c2C)CCN(C(C2CCCOC2)=O)C1 C(=O)(CC(O)CNC(=O)CCc1cc(C)no1)NC1(C(N(OC)C)=O)CC1 c1(CNC(NCCC(=C)Br)=NC)cc(C(C)(C)C)no1 C#CCCC(O)C(=O)N1CC(OC)CC1CCNC(=O)CC1COC(=O)C1 C1(C(N2CCC(O)(CN(C(Cc3nc(C)sc3C)=O)C)C2)=O)CCC2CCC1O2 C(=O)(C(CCF)NC(c1c[nH]nc1Cl)=O)NCC1C(C)(C)C1 C(CN=c1[nH]c(=NCC2CCCCC2O)c2cc(Cl)ccc2[nH]1)SCCOC N#CC1(C(=O)NCCCCCC(=O)N2CCN(C3CC3)CC2)CCCOC1 C1(O)(C(=O)NCCC2CCCO2)CC(F)(F)C1 c1(COC)cccc(C(N2CC(CNC(=O)CC3(C4CC4)CC3)CC2C)=O)c1 C#CCCCC(C(=O)NC(C)(C)C)N1CCCC(CCF)C1 N1(C(C2CCC(=C)CC2)=O)CC2CCN(C(=O)CC3CC3C3CC3)CC(C2)C1 N1(C(C(C=C)O)=O)CCCC(n2cc(-c3cc(OC)ccc3F)nn2)C1C c1(OCC(=O)N(CC(CNC(C(C)CC(F)F)=O)O)C)ccc2ccccc2c1 C(=O)(C(C)(C)COCC(F)F)NCC(C)N(C(=O)CCC1CCN(C)C1)C C12(NC(c3ccc(O)nc3Cl)=O)CCCC1N(C(=O)C(O)(C1CC1)C1CC1)CC2 C1(C(C)C)CCCN(C(c2sccc2Br)C(=O)NCc2csc(Br)c2)C1 C1(NC(c2n(CCOC)nnn2)c2cncs2)CS(=O)(=O)N(C)C1(C)C c1(C(N2C3CN(S(CCOCC)(=O)=O)CC32)=O)ccc(C#N)cc1C N1(C(C2(CC)CC2(F)F)=O)CCC2(CCCC2NC(=O)CC2CC=CC2)CC1 C1(C(CNC(C(C2CCC(=O)N2)C)=O)O)CCN(C(=O)Cc2ccccc2)CC1 C1(CNC(=O)C(O)C(F)F)CCCN(C(C2CCCCCCC2)=O)CC1 c1(SCC2C(C(=O)NCCNC(C3CCS3(=O)=O)=O)C2)nc2ccccc2s1 C#CCC(O)C(=O)NCC1CCN1C(c1ccc(C(F)(F)F)[nH]1)=O C1(Cl)(C(=O)NC2CC(C(=O)NC3(CCC)CCC3)C2)CC1(F)F c1(C(N(C2CCN(C(=O)CC3COCCO3)C2)CC)=O)ccc(C)c(F)n1 c1(C(C)NC(=O)Nc2ccc(C(N3CC4C(CO)C4C3)=O)nc2)ccccc1Br c1(C(C(=O)N(CCCNC(=O)C=CCO)C(C)C)O)cccc(Cl)c1 c1(C(=O)NCC2CCN2C(C2CC(F)(CO)C2)=O)cnc(C(F)(F)F)cn1 c1(NC(C(C)N(C(C2CCCC(OC)C2)=O)C)=O)cc(C)ccc1F c1(OC)ccc(CC(N2CC(OC)C(NC(C3(N=[N+]=[N-])CC3)=O)C2)=O)c(Cl)c1 C(=O)(CC(C)C(=O)NC(C(N1CC(C)(N(C)C)C1)=O)C1CCOC1)OC CC(C)(C)C(C)(C)C(=O)NCCN1CCN(C(=O)C#CC2CCCC2)CC1 C12(NC(C(C)(C)F)=O)CCCC1N(C(c1cnc3ccccc3n1)=O)CCC2 N1(C(=O)OC(C)(C)C)CC(F)CC1CC(=O)NC1CCCN(c2ccccc2)C1 c1(CN2C(C(=O)Nc3ccnn3CCCO)CCCC2)c(O)ccc(F)c1Br N1(C(Cn2c(N)ccn2)=O)CC2CC2(NC(c2cnc(S)nc2)=O)C1 Cc1cccc(CC(N2CCC(N(C)C(C3(C)CCN(C)C3)=O)C2)=O)c1C C1(C(N(CCCN(C(CC(=O)NCC)=O)C)C)=O)CCCC(C(=O)OC)C1 C=CCC(C)(C)C(=O)N1CCC(NC(=O)Cn2ncn(C)c2=O)C(C(N)=O)C1 c1(OC)c(C(=O)NCC2CCCN2C(=O)C(C)(C)CC2CC2)cc(Cl)cc1C C(=O)(C(F)(F)Cc1ccc(F)cc1)NC1CC(CCNC(COCCC=C)=O)C1 C(=O)(C(O)CC(C)(C)C)N1CC(C)C(CNC(C2CCCN2S(C)(=O)=O)=O)CC1 Cc1nc(C2(NC(C3(NC(=O)C(C)N4CCCC4)CCC3)=O)CC2)no1 CC#CCC(C(=O)NCC=CC)NC(C1CC=CCO1)=O C1(NC(CN(C2CCC2)C)=O)CC2CCC(C1)N2C(C1CCCC1(C)C)=O C1(C(=O)N(CC(=O)NC2CC(C(N)=O)C2)C)(COC)CCC1 C1(N(C(CCCN(C)C)=O)CCF)CCCN(C(=O)C(O)C(F)F)C1 c1(CC(=O)NCC2CC3CC(NC(C(CC#C)C)=O)C3C2)c(C)cc(OC)cc1C C=CC1CCCN(C(c2nnc(C)s2)C(=O)NCC(C)C)C1 C1(C(=O)NCCN(C2CCCCC2)C(=O)C(C2CCCCC2)O)CC2CCC2C1 c1(OC)cc(-c2nc(-c3cncnc3)nn2C(c2ccccc2)C)n(C)n1 O=C(C#CC1CCCOC1)NCC1CCCCN1C(=O)Cc1ccc(Cl)cc1 c1(C(=O)NC(C(C)NC(=O)C(C)(C)CN2CCOCC2)C)cnn2c1N(C)CC2 c1(C(N2CCC(N(C(CCCC(C)=O)=O)C)C2)=O)ccccc1S(C)(=O)=O O=C(C1=CCCCO1)NCC1(O)CCN(C(=O)CCC=Cc2ccccc2)C1 CCC(C)(C)C(=O)N1CC(CNC(c2cncnc2-c2ccccc2)=O)C(O)C1 CC(C)C(C(=O)N1C(CNC(c2cccn2C)=O)CC2CC12)c1ccc(F)cc1 c1(CC)ccc(O)c(NC(=O)CC(CC)NC(c2cc(C(N)=O)[nH]n2)=O)c1 C1(C2(C(=O)NCC(=O)N(C)C)CC2)CCCN1C(C1CN(C)C1)=O CCC(O)C(F)(F)C(=O)NCC1CN(C(=O)CC2CCC3CC23)C1 C1(C(=O)NC2CCC(NC(c3ocnc3C3CCC3)=O)CC2)CC2COCC2C1 CCCC(C)(C)C(=O)N1CCCC(NC(=O)C(O)CC2CC2)CC1 c1(CCC(=O)NCC2CC(F)(CNC(C=C(CC)CC)=O)C2)ccc(Cl)c(F)c1 C(CCCCCC(=O)N(C1CCCC1)CC)NC(c1c(CC)ncs1)=O C(=O)(C(O)(C(F)(F)F)c1ccccc1)NC1C(CNC(c2ccoc2)=O)CCC1 n1(CC(N2CC(N(C(=O)C3=CCOCC3)C)C(F)C2)=O)ncn2nccc2c1=O C(c1cccc(F)c1Cl)=CC(=O)NC1C(NC(C=CC(CC)=CC)=O)CCOC1 CC1(NC(C23CC(F)(C2)C3)=O)CCN(C(C2CC2C(C)(F)F)=O)CC1 n1(C(CC)C)nc(C(=O)NCC(CNC(=O)Cc2ccsc2)CO)cc1C C(C)(CNC(=O)CCCN1C(=O)CCC1=O)(C(C)C)NC(CNC(CCC)=O)=O C1(CSC)CC(NC(=O)C(=O)NC(C)Cn2cncn2)C12CCC2 c1(CC)ccccc1Cl.C12CCN(CC1)C(c1ccc(C(F)(F)F)cc1)C(=O)N2 c1(C(=O)NCC(C)(C)CNC(c2cncnc2)=O)cc(Cl)c([N+](=O)[O-])[nH]1 c1(CC(=O)NC2(CN(C)C(C3CN4CCN3CC4)=O)CC2)c(F)cccc1C#N n1(CCC)cc(Cl)c(C(=O)NC2CCN(C(=O)CC3OCCC3C)C2)n1 Cc1cc(=O)n(C)nc1C(=O)NCCNC(c1cccc(Br)c1F)=O c1(N(CC(C2CC2)OC)C)nc(NC2CCOC2)c2cnn(C)c2n1 C(=O)(CCC(C)(C)C)NCC(CCNC(c1cncc(NC)c1)=O)OC C1(NC(C(CC)OCC)=O)CC2CC(NC(c3cccnn3)=O)CC12 C=C1CCN(C(c2cnn(CCNC(c3ncoc3C)=O)c2)=O)C1 C(=O)(CCCCn1cc(NCc2ccc(OC)cc2)cn1)N(CCN(C)CC)CC Cc1ncc(C(N2CCOC(CNC(C3C4CNC(=O)C34)=O)C2)=O)c(=N)[nH]1 c1(CC)ncccc1C(N1CCC(NC(C2(N(C)C)CC2)=O)C1C)=O N1(C(c2c(C)cc(CC)o2)=O)CCCC(C)(C(=O)NCC2(C(C)(C)OC)CC2)C1 c1(C(=O)NC2C(C)(C)CN(C(=O)CCCC3CCC3)C2)nc2ccc(Cl)nn2n1 c1(CC)cc(NC(=O)CC(C)NC(=O)CCCCCn2cnnn2)cc(O)c1 c1(N2CCC3(C(C(N4CCC(C(=O)OC)C4)=O)C3)C2)nccc(S(C)(=O)=O)n1 C1(C)(CCNC(CC2CC(CC)OCC2)=O)CCN(C(C)=O)CC1 c1(C(N2CC(c3cn(CCCCC)nn3)C2)=O)ccc2n[nH]c(CCC)c2c1 c1(C(CNC(CC=CC=C)=O)N(C(=O)C(C)NC(=O)OCC)C)ccccc1 C1(CC(=O)NCCOCC(N)=O)CCCN(C(=O)C(c2ccccc2)O)C1 C1(C(N2CCC(C)C2CNC(c2cccc(CCO)c2)=O)=O)CC2(C1)OCCO2 c1(C(=O)NCC2C(NC(Cc3ccc(C)cc3Br)=O)C2)cc2ncccc2o1 C1(CNC(C(C)(C)OCC)=O)C(C)CCN1C(=O)CCC1OCCO1 C(=O)(C(CNC(C1OCCC1(C)C)=O)C(C)(C)C)N1CC(CC(C#C)C)C1 C1(CNC(c2ccc(C=C)cc2)=O)CN(C(=O)COCC(C)C)C2(CCC2)C1 CC1CC(NC(C2CC(O)C2)=O)CCN1C(c1cccc(C(F)F)c1Cl)=O c1(C(N2CCCC2C(c2ccccc2)O)=O)ncc(C2(O)COC2)s1 c1(C(=O)NC(C2CCN(C(C(CC)OCC)=O)C2)(C)C)nn(C)cc1COC C1(C(N2C(C)(CNC(c3ccc(C#N)o3)=O)CCC2)=O)Cc2cccnc2C1 C=CCCC(=O)NC(C1CC=CCC1)C(=O)NC(c1nc[nH]n1)C1CC1 C1(C(C(=O)NC2CC(F)(CNC(C3(C4CCCO4)CC3)=O)C2)F)CCCCCC1 N1(C(C(C(C)C)F)=O)CCC(C2CCCN(C(c3ccc(F)o3)=O)C2)CC1 c1(C(=O)OC)ccc(NC(=O)CCc2cc(C)ccc2C)cc1OC(C)C c1(CC(=O)NCC2C(NC(C(C)C3CCCO3)=O)CC2)sc(O)nc1O C1(CC=C)(NC(C2COCCC2(F)F)=O)CCCN(C(=O)CC(C)(C)CC)C1 N#Cc1ccccc1C(=O)NCC(CC(=O)N1CCCC1C(N)=O)C1CCC1 CCC(C)CCCCC(=O)NC1CCCC2CN(C(c3ccccc3O)=O)CC12 C1(O)(CNC(C(F)=C(C)C)=O)CC(NC(=O)C(O)c2cnc[nH]2)C1 c1(C(=O)NCC2C(NC(C(CC)SC)=O)C2)cc(C)c(C#N)c(C)c1 c1(C(C(N2CC(N(C(c3c(C)n[nH]c3)=O)C)C2)=O)C)cc(Br)ccc1F C1(C)(CSC)CN(C(=O)C(C)(C)C2CCN(C(=O)CCN(C)C(C)=O)C2)C1 C1(C(=O)Nc2c(C(N3CCC(CCOC)C3)=O)scc2)CCCC(=O)C1 c1(OCCC(=O)N(C(C)CNC(C2CC3CC2C3)=O)C)ccc(S(C)(=O)=O)cc1 C(=O)(C(C)C(C)CNc1ccc(SCC)cc1)N(CCCNC(CCC)=O)CCC N1(C(C2(OC)CCCC2)=O)CCC(NC(=O)Cn2nnnc2C)CC(C)(C)C1 C1(SCc2cn(CCC(=O)NCc3cnc(N(C)C)s3)nn2)CCCCC1CO c1(C(C)NCc2ccc(C(=O)OC)o2)cc2ccccc2[nH]1 n1(CC)cc2ccc(C(=O)NC(C)C(C(C)C)NC(c3c[nH]cc3C)=O)cc2n1 c1(Nc2cccc(SC)c2)ncnc(NCCCOc2ccccc2)c1C c1(CC)nc(C)c(C(=O)NCC2(F)CCC(CNC(c3n[nH]cc3CC)=O)C2)s1 C(CCCC(=O)NCC1C=CCN1C(=O)CC1CC1c1ccccc1)OCC c1(CC(=O)NC(C2CCN(C(=O)CSCC#N)CC2)(C)C)ccc2occc2c1 Cc1ccccc1SCC(=O)NCC1CC2CC2N1C(=O)Cc1sc(O)nc1O c1(COCC)nc(C)c(C(N2CCC(CNC(c3ncn(CC)n3)=O)CC2)=O)s1 CCCC(CCCNC(c1sccc1C(C)C)=O)NC(=O)C(C)C(F)F N1(C(CCCN(C)CC2CCCO2)=O)CCC(NC(C2CCC=CCC2)=O)CC1 c1(NC(C(CNC(=O)C=CC(C)(C)SC)OC)=O)cccc2c1OCO2 Cc1nnc2n1CCCC2C(=O)NC1CCN(C(=O)CCCC#N)CC1 N1(C(c2ccoc2Cl)=O)CCC2CCCN(C(=O)COCC(F)(F)F)C2C1 N1(C(=O)CC2CSC2)CC2C3CCC(C2C1)N(C(=O)CCN1CCCC1)C3 c1(CC)ccc(NC(=O)C(C)N(C(=O)C(C)(C)n2ccnn2)C2CC2)cc1O C=CC1(C(=O)NCC2CC3CCC2CC3)CCN(C(=O)CC2CNC(=O)O2)C1 N1(C(CCC=C)=O)CC(NC(=O)C(C)(O)C(C)c2ccccc2)CC2(CC2)C1 c1(CCCC(=O)N(C(CNC(CC(CC)C)=O)C2CC2)C)nc2ccccc2o1 C1(CCC=C)(C(=O)NCc2ncnn2C(C)C)CN(C(c2ccc(OC)o2)=O)C1 C#Cc1ccc(OC)c(C(N2CCC(CN(C(=O)Cn3cnc(=N)[nH]3)C)C2)=O)c1 C(C(C)C)(C(O)C(=O)NCCC1CCN(C(C2CC3(CCC3O)C2)=O)C1)OC C1(C(=O)NC2(O)CCC(C)(C)C2)Cc2c(O)cccc2N1C(=O)OC(C)(C)C Cc1nc2cncc(C(N3CC(CO)CC3CO)=O)c2[nH]1 C(=O)(CCC(C)(C)F)N1CC(C)C1C(N1CCCCC1C(=O)N(C)C)=O c1(C(C)(C)C(N2CCC(C)(NS(=O)(=O)CCCl)C2)=O)cccc(C#N)c1 N(C1CCCc2nn(C)cc21)c1cc(NC(C2CCCCCC2)CC)ncn1 C12(NC(C3CC34CCOCC4)=O)CCCC1(F)CN(C(=O)C(F)(F)C(F)F)C2 c1(NC(CC)C(=O)N(C)C)cncc(CNC(=O)OC(C)(C)C)c1 Cn1cnc(C(N2CC(C(N)=O)(CNC(C3(n4cnnn4)CC3)=O)C2)=O)cc1=O C1(C(F)F)(OC)CC(C(=O)N(CCCCN(C)C(C2(O)CCSC2)=O)C)C1 C1(NC(=O)Cc2sc(O)nc2O)CS(=O)(=O)CC1NC(c1ccnn1C(F)F)=O C1(C(N(c2nc(C)cs2)C(CC)C)=O)CC(=O)N(CC(F)(F)F)C1 C1(CNC(c2n[nH]c(C)c2C(F)(F)F)=O)CC(N=c2ccc(C#N)c[nH]2)C1 N1(C(CCCNC(C2=C(C)OCCC2)=O)=O)CC2CN(C)CC2(C)C1 C(=O)(C1CCc2ccccc21)NCC(CNC(=O)COC1CCCOC1)OCC Cc1cc(C(N2CC3(CNC(C4CCCC4)=O)CC2CCO3)=O)cc(C)c1Cl c1(C(N(CCC(=O)N(CC(C)C)C)C)=O)ccc2occc2c1 C(=O)(C1CCCc2nncn21)N1CCCC(NC(C=Cc2c(C)coc2C)=O)C1 c1(C(=O)NCC2N(C(COc3c(F)ccc(C)c3)=O)CC2)cnc2[nH]nnc2c1 C1(C(N2CC(C(N)=O)C2)=O)COCCN1C(=O)CCc1cncnc1 c1(C(N2C(C(C)C)CN(C(=O)CCC(=O)N(C)C)CC2)=O)cc(Br)cc(F)c1O C(=O)(CCCC(C)(C)C)NC(C)C(C)NC(c1nc(O)nc(O)c1F)=O c1(C(=O)NCCCC(C(=O)Nc2c(CC)cc(O)cc2)O)ccc2cc[nH]c2c1 C1(NC(c2n(CCCSCC)nnn2)c2cnn(C(F)F)c2)CCNC(=O)C1 c1(N2CCCC(OC)(CO)C2)nc(C)cc(=NCc2c(Cl)cccc2Cl)[nH]1 C1(NC(c2c(C)cc(F)cc2)=O)C2COCC1CN(C(c1n[nH]c(C)c1O)=O)C2 CC1(C)CCN(C(=O)C(N)=O)C(C(=O)NC2(C)CCC(=O)NC2=O)C1 c1(C(C)C)nc(NC(c2cn[nH]c2)C)cc(=NCc2cncc(C(N)=O)c2)[nH]1 c1(N2CCC(C)C(NC(=O)CCC(N)=O)C2)nccc(S(C)(=O)=O)n1 N1(C(C2CC(OCC)C2)=O)CCC(C(C)(C)NC(=O)C=CC2CCCN2C)CC1 N1(C(CNC(c2cccs2)=O)=O)CC(CNC(C2CC3CCC2O3)=O)C(O)C1 c1(CC(=O)NC2CC(F)(CNC(=O)CCC3CCCO3)C2)ccc(O)cc1 c1(CC)ccc(C(N2CCOCC2CN(C(=O)CC2CSCCS2)C)=O)cc1N CCC(F)(F)C(C)(C)C(=O)NCC1(C2CC2)CCN(C(c2nnn(C)n2)=O)C1 C1(CNC(c2cc(C)nc(Cl)n2)=O)CC2COCC2N1C(=O)C(C)CN(C)C C(Cc1ccccc1Br)(CC(=O)NN=c1ccn(C)[nH]1)NC(c1cnc(C)s1)=O C=C(C)C(C)(O)C(=O)NC1C2CN(C(c3cnc(CC)o3)=O)CC12 c1(C(=O)NCC(C)CN(C(=O)CC2CC2(C)C)C)csc2cc(Cl)cnc12 c1(CNC)ccc(NC(=O)C(Cn2cncn2)NC(=O)OC(C)(C)C)o1 N1(C(C2N(C(C(C)SC(C)C)=O)CCC=C2)=O)CCC(C)(C2CC2)C1 N1(C(C(OC)OC)=O)CCN(C(c2ccccc2C(N)=O)=O)CC2(CC2)C1 Cc1nn(C2CC2)c(C)c1CN=C(NC(C)C)NC1CCOC(c2ccccc2)C1 c1(C(=O)OCC)cc(NC(=O)CC2(C(F)(F)F)CCC(=O)NC2)ccc1OC CC(C)(CC(=O)NC1CCCN(C(=O)COc2ccccc2)CC1F)CC(F)F c1(N2CC(C)(NC(CCNC(=O)NC)=O)C2)c(C(N)=O)cccc1[N+](=O)[O-] c1(C(N(C)CC2CCN(C(C(C(C)(C)C)OC)=O)C2)=O)cnc2ccncc2c1 Cc1c(C(N2CC(NC(=O)C(C#N)=CC3CC3)C(C)C2)=O)ccn1C(C)C C(=O)(CC1=CCCCC1)N1CCCC(NC(C2CC(=O)N(c3ccccc3)C2)=O)C1 C12(C(N3CC(N(C(C4(COC)CCCCC4)=O)C)C3)=O)CC3CC(C(=O)N1)C2C3 C(=O)(CC1OCCc2ccccc21)N1CC(CCNC(c2c(CC)[nH]cc2)=O)C1 C#CCC(C)(C)C(=O)NCC(C)(CC)NC(c1cc(C(N)=O)no1)=O Cc1nc2ccc(C(N3CC(O)(CCNC(c4c(C)noc4N)=O)C3)=O)cc2[nH]1 c1(OC)cnc(C(N2CCC3C(NC(=O)CCC(=O)N(C)C)C23)=O)c(F)c1 Cc1ncc(Cl)cc1C(N1CC2CC(NC(=O)Cc3cc(O)nnc3O)C1C2)=O c1(C(N2CC(CC)N(C(=O)CC(C)F)CC2)=O)ccc(C#N)c(O)c1 C(C)(C)(C(=O)NCc1n[nH]cc1C(=O)NCCc1cocn1)OC(C)C C1(NC(C(C)OC)=O)CN(C(c2ccc(Cl)c(N)c2)=O)CCC1CO c1(C(N2CCC(O)(CC)C2)C(=O)NCCC)nn(CC(=O)OC)cc1C C(=O)(C(O)CN1CCCC1)NC1(C)CSC1.N12CC(C1)C2=O C(c1c(Cl)nc2sccn12)=CC(N1CC(NC(c2cc[nH]c2)=O)C(CO)CC1)=O N1(C(C2C(C)(C(F)F)C2)=O)CC2CC1C2C(=O)Nc1cnccc1C(N)=O Cc1cnc(F)cc1C(=O)NC1CCC(NC(=O)C(C(C)C)OCC(C)C)CC1 C(=O)(CCCCC(F)F)N1CC(NC(C=Cc2nnn(C)n2)=O)C(O)C1 C1(C(N2CCC(NC(C(C)Oc3cccnc3)=O)C2)=O)CN2CCN1CC2 C1(C(N2CCSCCC2C)=O)(CC)CCCN(C(c2ccc(C(C)=O)[nH]2)=O)C1 C1(C(N2C3CC(NC(c4cn(CC=C)nc4)=O)(C3)C2)=O)CCc2nn[nH]c2C1 C1(C(N(C)CC2(CNC(C3CCCC3)=O)CC2)=O)CC2CCCC(C1)C2 C1(C(=O)NC(CNC(c2cc(C(=O)OC)ncc2)=O)C2CC2)CC2CCC(C1)C2 c1(OC)ncc(C(=O)NC2COCC2CNC(=O)Cn2ncn(C)c2=O)c(C)n1 CCC(CC(F)F)C(=O)N1CC(NC(c2cc(C(N)=O)cc(C)c2)=O)CC1C C1(NC(c2c(CCC)nns2)=O)CN(C(c2oc(CN(C)C)nc2C)=O)CC1O c1(SC)ccc(C(=O)N(C)CC2(CNC(c3ccoc3C(F)(F)F)=O)CC2)cc1 c1(Cn2cc(C3C(OC)CN(C(C(C)=CC)=O)C3)nn2)cc2c(s1)CCC(C)C2 C1(C(NOC(CC)CC)=O)CCOCC1NC(c1ocnc1C)=O C1(C)(C(=O)Nc2cn(CC)nc2)CCN(C(=O)C(=Cc2ccco2)C)C1 c1(OC)ccc2cc(C(=O)NCC3CC3CNC(c3ccc(C)cn3)=O)sc2c1 C12(C(N3CCC(N(C(CCc4onc(CC)n4)=O)C)CC3)=O)CCCC(C1)OC2 C1(C(N(CCCNC(C(C2CC2)OCC)=O)C)=O)CCCC2(CCC2)O1 C1(C)(NC(C=CC(=O)CCNC(C2(CCOC)CC2)=O)(C)C)CNC1.C1(=C)CC1 C(CC(C)C(=O)N(CCNC(C1CC(=O)N(C2CCCC2)C1)=O)C(C)C)=CCC c1(SC)nc(Cl)cc(=NCC2CC(NC(C3CCCCC3O)=O)C2)[nH]1 N1(CC(=O)N(CC)CC2CCCN2C(=O)C(=Cc2ccco2)C)CCC(C)CC1 C1(C(=O)NCCCN(C(C(Br)=C(C)C)=O)C2CC2)CCN(C2CC2)C1=O C12(NC(C(C)N(C)CC3CC3)=O)CC1CN(C(c1sccc1-n1ccnn1)=O)C2 C12(NC(CCC(C)OC)=O)CCC(C1)N(C(C1(c3ccccc3)CCCC1)=O)C2 CC1CCN(C(=O)CN(C)CCN(C)C(C2(CO)CCC2)=O)C1 C(N=c1[nH]c2c(c(=NCC3CC34CCOCC4)[nH]1)CCC2)c1cc(C)on1 C(=O)(C(C)(C)COCC(F)F)NC(C)C(C)NC(c1ccncc1F)=O N1(C(C(C)Sc2ccc(C)cc2)=O)CCC(C2CN(C(c3cnccn3)=O)C2)C1 N1(C(CC(CC)C2CCC2)=O)CCN(C(c2ccc(C)nc2C)=O)C(CO)C1 c1(C(=O)NCC2N(C(C(C=C)(F)F)=O)CC2)ccc2c(C#N)c[nH]c2c1 C1(C(=O)NC2C3CN(C(C4(CC)COC4)=O)CC32)CCc2c(cnn2C)C1 N1(C(C2CCC(NC(c3nccc(C#C)c3)=O)C2)=O)CC2CCC(O)CC2C1 C1(COC)CCOC2(CCCC2)C1.N12CCN(CC(O)C1)C(=O)c1ccc2nc1 C1(C(=O)NCCC)CC2(C1)CC(NS(=O)(=O)CC1CCCN1C(=O)OC(C)(C)C)C2 C(=O)(C(O)C(F)(F)F)N1CC(NC(=O)CCCCc2ccc(Br)cc2)C1 N1(C(C2C(C)OCC2)=O)CC2CCN(C(=O)CCCn3ccnc3)C2C1 Cc1cc(C(=O)NC(C)CC(C)NC(=O)C=Cc2ccco2)cc(NC2CC2)n1 C1(CC(=O)NCC2CCCN(C(=O)COc3cnn(C)c3)C2)(OC)CCCCC1 C(=O)(C(CC(N)=O)NC(=O)CC1CC(=O)C1)NC1CCN(C(C)=O)CC1 c1(C(=O)NCC(C)C(F)C(=O)Nc2ccc(C3CC3)cc2)cncc2[nH]ccc12 c1(C(=O)NC(C)CCNC(c2ccc3c(c2)COC3)=O)ccc2c(c1)C(C)CO2 N1(C(COc2ccc(SC)cc2)=O)CC2CC1CC2NC(=O)CCn1cccn1 N1(C(c2cccc(C)c2Br)=O)CCCC(C2CN(C(=O)C(O)CC(C)C)C2)C1 CC1CCN(c2ccc(C(=O)NC3CC3NC(=O)CC3CC3)cc2)CC1 c1(CC(C)C)ccccc1C(N1CC(NC(C2CC2[N+](=O)[O-])=O)C(C(F)F)C1)=O C=C(C)c1cn(C2CCC(C(=O)NC(c3ccc(C(=O)OC)cc3)C)CC2)nn1 c1(CC(=O)OCC)nc(C)c(C(N2CCC2CNC(c2ccon2)=O)=O)s1 c1(C(=O)NC2C(C)CN(C(=O)CC3CCCCO3)C2)c[nH]c2ncccc12 C1(C)(NC(c2n(CCC)nnn2)c2occc2C)CCC(=O)N(C)C1 CCCC(O)(CCC)CC(=O)NC(C)C(C)NC(c1cnn(C)c1CC)=O C(=O)(C(C)C(O)C(C)CC)N(C(C)CNC(c1ccccc1)=O)CC c1(CN(C(c2c(C)c[nH]n2)C(=O)NC2CCOC2)C)cncc(F)c1 CCCCCC(O)CC(=O)NC1(C)CC(NC(c2coc(CO)c2)=O)C1 c1(CCC(N2C(Cc3cn(C(C)(C)C)nn3)CC2)=O)cccc2cccnc12 C(=O)(C1=C(C)N(C)c2ncnn2C1)N(C1CCN(C(c2c(CC)c[nH]c2)=O)C1)C N1(C(CCSC)=O)CCC(C2CCN(C(c3cncc([N+](=O)[O-])c3)=O)C2)C1 C(C(CCCC)NC(=O)Cn1cccn1)NC(C(F)=CCC)=O C(CCO)(C(=O)N1CCOC(CNC(=O)C=Cc2nccs2)C1)N(C)C C1(NC(C)C)CCN(C(=O)C(N2CCOCC2c2ccccc2F)=O)CC1 Cc1nc2ccccc2cc1CN(C(C1COCCN(CC2(CO)CC2)C1)=O)C N1(C(=O)CC2C=CCC2)CCCC(C2CN(C(=O)CC3(O)CCCCC3)C2)C1 C(=O)(C1CCCn2nccc21)NC(CNC(C1N(CC)C(=O)CC1)=O)CC(C)C N1(C(CSCC=C)=O)CCC2(C1)OCc1ccccc12 C1(NC(CCOC)=O)CN(C(C2(C)CS(=O)(=O)C2)=O)CCC1C CCCC(CNC(=O)Cn1nc(C)nc1C)C(=O)N1CCC=CC1C(=O)OC C1(C(N2C(CN(C(=O)C(F)(F)C3(O)CCCC3)C)CCC2)=O)CC12CCOC2 N1(C(C=CCOC)=O)CCC(C(N2CCC(C(C)C)(CO)C2)=O)C12CC2 C(C)(CC(C)NC(=O)CCOC1CCC1)NC(CN(CC)CC)=O c1(CC)nc(C)[nH]c1C(=O)NCC(C1CC1)N(C)C(c1cnc(C)nc1)=O c1(NC(C2C(NC(c3ncn(CC)c3)=O)CC=CC2)=O)ccc2nccn2c1 CC(C)C(F)(CNC(C1CCCCCC1)=O)C(=O)NC1CCOC2(CCC2)C1 C1(CNC(CN2C(C)CC2)=O)CCN(C(=O)COC(F)(F)C(F)(F)F)CC1(F)F C1(NC(=O)Cc2c(Cl)cccc2Cl)CCN(C(=O)CCc2cnoc2)C12CCC2 Cc1cc(N)n(CC(N2CC(CNC(c3sccc3C3CC3)=O)C(C)C2)=O)n1 C1(CCOC)CCN(C(c2cc(C(N)=O)no2)=O)C1.C1=CC(=O)NC1(C)C C12(CC=CCC1)C(=O)NC2.c1(CCNC(C2(C)CC(CO)C2)=O)ccc(O)nc1 N1(C(CC=CCC)=O)CCC(C)CC1CNC(=O)Cn1ccc(C)cc1=O C(c1ccccc1F)=CC(=O)NCC(CC)(C)NC(c1ccoc1C)=O c1(OCC(=O)OC)cccc(C(=O)NC2CN(C(C3SCCC3C)=O)C2)c1 N1(C(C(c2ccc(C)s2)C)=O)CCC2(CCC(NC(=O)Cc3cc[nH]n3)C2)CC1 C1(C(=O)Nc2cn(CC(C)(F)F)nc2)CCCCC(F)(F)C1 C(=O)(C(F)=CCF)NCC=CC(=O)NC(C1CCOC1)C#C C1(N(C)C(c2ccc(C(F)(F)F)s2)=O)CN(C(=O)C(F)F)CC1F CP(C)(=O)c1ccc(C(=O)NCC2CCCN2C(c2nsc3ccccc23)=O)cc1 N1(C(C2(C3CC3)CC2)=O)CCC2(CC1)CCN(CC(O)COc1ccccc1)C2 C#Cc1cnc(NC(=O)CN2CCN(C(=O)COCCOC)CC2)cn1 C12(C(N3CCCC(NC(Cc4cc(C)on4)=O)CC3)=O)CCCC1CC(=O)C2 C(c1ccc(C)cn1)=CC(=O)NC1C(NC(C(CCC)C)=O)C1 N1(Cc2n(C(C)C)ncc2)CC2(CN(C(=O)CCc3ccc(Cl)cc3)CCO2)C1 C1(C(N2C(C(=O)NCC(C)C#N)CSCC2)=O)CC2C(C1)C2(F)F c1(C(=O)NCCC(C)NC)cccc(NC(=O)CC2CC(N(C)C)C2)n1 C1(NC(c2c(CC)csc2)=O)CCCN(C(c2cnc(OC(C)C)cn2)=O)C1C C1(NC(C(C=C)O)=O)CN(C(=O)C(C)(C)CNC(C)=O)CCC1C N1(C(COCCCC)=O)CC2C(C(=O)NC(C)CS(N)(=O)=O)C2C1 c1(C(CC)C(=O)NCCCNC(=O)C=C2CCC(C)C2)c(C)noc1C c1(C(N2C3C(N(C(C(COC)C)=O)C)CC(C3)C2)=O)ccsc1S(C)(=O)=O c1(NC(c2cc(-c3nc[nH]n3)ccc2F)=O)c(F)cc(F)cc1Br C1(CC)CCN(C(C2CC2[N+](=O)[O-])=O)C1CNC(=O)CCn1ccnc1 c1(NC(C(C)NC(c2nccc(OC)c2)=O)=O)cn(C)c(=O)nc1O c1(NC(C(C)C)CCO)ccc(S(=O)(=O)N2C3CCC2CC3)c2ccncc12 C1(NC(c2cc(C)sc2)=O)C2CN(C(C3(c4ccc(O)nc4)CCC3)=O)CC12 c1(-c2n(C(C=C)C)nc(-c3ccnc(-n4cncn4)c3)n2)cccc2c[nH]nc12 c1(C(N2C(C(CNC(C(CC(C)C)C)=O)(C)C)CCC2)=O)cccc2c1NCC2 C(=O)(C=CS(C)(=O)=O)NC(C)CCNC(=O)CCC1NC(=O)NC1=O Cc1ccc2c(CC(N3CC(CNC(C4C=CCCC4)=O)C(C)C3)=O)c[nH]c2c1 C(c1ccccc1F)=CCC(N1C(C(C)NC(C2CCCS2(=O)=O)=O)CCC1)=O N1(C(C(CN(C)C)NC(c2cc(C(C)C)[nH]n2)=O)=O)CC(F)(F)C1C1CC1 N1(C(C(N2CCOCC2)C)=O)CCN(C(C2CCC=CCCC2)=O)CC12CCC2 N1(C(C2(C)CN(C(CC3C(C)(C)C(O)C3)=O)C2)=O)CCC12CC(C)(CO)C2 C1(C(=O)NCC2N(C(Cn3ncc(CC)c3)=O)CCC2)C2CCCCCCC12 C12(C(=O)NCCN(C(C3(C(=O)NC)CCC3)=O)C)CCCCC1CS(=O)(=O)C2 c1(NCC(=O)NCc2ncoc2CCNC(C2CCCCO2)=O)ccc(Cl)cn1 C(=O)(C(C)(O)C(F)(F)F)NCCSCC(=O)NCCn1c(C)cnn1 c1(C(=O)NC2C(NC(=O)CN3CCOC3=O)CC2)ccn2nnnc2c1 Cc1ncc(C(N2CCC(CCC(=O)NC(C)CC(C)C)C2)=O)c(=N)[nH]1 CC(C)C(C(=O)N(C1CCCCC1O)C)NC(=O)COc1cccnc1 CCC(C)C(C(=O)NC(CN=[N+]=[N-])C(=O)NCC1CC(C2CC2)=NO1)N(C)C CCCCC(CNC(c1ncc[nH]c1=O)=O)NC(=O)CC1(N2CCCC2)CC1 CC1C(C)N(C(c2nccc3nn[nH]c23)=O)CCN1C(=O)C(=O)C(C)(C)C c1(CN(C(=O)C(=O)N(C)CC2CC3CCC2C3)CC=C)ccc(F)cc1 c1(C(N(CC(C)CNC(C2CC23CC(F)(F)C3)=O)C)=O)cccc2[nH]ncc12 C1(C(=O)NC(CCN(C(c2cc(OCC)n[nH]2)=O)C)C)CCCC(C(=O)OC)C1 N1(C(=O)C=CC2CCOCC2)CC2(C1)CN(C(=O)Cc1cnoc1)CC2CO N1(C(C(C)NC(N)=O)=O)CCCC12CCN(C(=O)Cn1cnc([N+](=O)[O-])n1)C2 CC1Cc2cc(CC(N3CC(C)(NC(C4Cc5nncn5C4)=O)C3)=O)ccc2O1 Cc1nn2ncccc2c1C(=O)NC1CC1CNC(=O)CCOCC(F)(F)F Cc1ncc(CC(=O)NCC23CC(NC(=O)C(F)CC4CC4)(C2)C3)o1 c1(C(N2CC(O)CC2CNC(C2(CC(F)F)CCC2)=O)=O)cn2ncccc2n1 c1(C(=O)NCC(C)CN(C)C(c2nn(C)cc2[N+](=O)[O-])=O)nc2ccccc2[nH]1 C12(C(=O)NCc3cc(CC)[nH]n3)CC(CN1C(=O)C(C)NC(C)(C)C)C2 N1(C(c2c(C)nc(CO)nc2)=O)CCN(C(=O)CC2CNC(=O)C2)CC12CCC2 C(c1cccnc1)=CC(=O)NCCOCCC(=O)NCC1C(C)CCC1 N1(C(COc2c(C)cccc2)=O)C2CC1CN(C(=O)CCC(C)(C)F)C2 c1(C(N(C2CN(C(C(CC)N(C)C)=O)CC2O)C)=O)cc2cccc(C)c2nn1 c1(C(=O)NCC(CO)NC(C#CC(C)(C)C)=O)c[nH]ccc1=Nc1ccccc1 Cc1cc(Cl)c(C(N2CCC(O)(C(C)CNC(C3CS(=O)(=O)C3)=O)C2)=O)cn1 CC(C(=O)N1CC(NC(C2(C(F)(F)F)CCCC2)=O)C(F)C1)C(C)(C)O N1(C(c2c(OC)csc2)=O)CCN(C(=O)Cc2cc(Cl)n(C)n2)CC1CC(F)F C(C(F)(F)F)(C(C)(C)C(=O)OC)NC(C(CC(=C)C)N)=O C1(C(N2CCCC(CCF)C2)=O)CC(F)(F)CN1C(=O)CCC1CC1(F)F c1(Nc2c(C(N3CCOCC3)CN3CCCC3)ccc(Cl)c2)cc2ncnn2cn1 CCC(CC(=O)NC(C(=O)NOCCN(CC)CC)C1(C)CC1)C1CC1 CCCCCCC(F)C(=O)NC(C)CN(C)C(c1cn(C)[nH]c1=N)=O N1(C(C2CC(CNC(c3c(C(C)C)n[nH]c3)=O)C2)=O)CCOC2CC12 N1(C(C2CC(OC)C2)=O)CCC(C(C)(C)C)(CNC(=O)CN2CCC(C)(O)C2)C1 c1(NCc2cnn(CC)c2C)cc(=NCc2cc(Br)cc(C)n2)[nH]cn1 c1(C(N(CC(CC)NC(C(CCC#C)O)=O)C)=O)c(C)c(C)cc(C)c1C N1(C(c2c(C)cc(F)cc2)=O)CC(C)N(C(C2CCS2(=O)=O)=O)CC1C n1(CC(=O)NCCC2CCN(C(CC3C(=O)NC(=N)S3)=O)C2)ccc([N+](=O)[O-])n1 c1(OC)ccc(OC(C)CNC(=O)N(C23CC(F)(C2)C3)C)c(Br)c1 C12(C(N3CC(C)(C(N4C(C)(C)CC4)=O)C3)=O)CCCC1C2(F)F C1(C(N2CCC(N(C)C(c3ccc(=O)n(C)n3)=O)CC2)=O)CCCC1S(C)(=O)=O Cc1ccc(C(N2CC(NC(C3Cc4nncn4C3)=O)CC2(C)C)=O)c(O)c1 C1(S(C)(=O)=O)(C(=O)NCC2CN(C(C3=C(C)OCC3)=O)C(C)C2)CCOCC1 c1(NC(CC)CN(C(=O)C(C)CF)CC)ncc([N+](=O)[O-])cc1Br C1(C(=O)NC(CC#C)C)COC(CNC(c2c[nH]c(C(N)=O)c2)=O)C1 C12(C(=O)NCCC3CN(C(C(C4CC4)OC)=O)C3)C=CC(CC1)C2 c1(CC(=O)NC(C)(C)C=CC(=O)Nc2cnc(F)nc2)cccc(F)c1F CC(C)C(O)C(=O)NCC1CC(F)CN1C(=O)COCC1CCOC1 Nc1cc(Br)cnc1C(=O)NC1CCCN(C(C2CCOCC2)=O)CC1 CC1=NN(C)C(=O)C1CC(=O)NC1COCCN(C(C2CCOC(C)(C)C2)=O)C1 N1(C(=O)Nc2c(C)snc2)CCN(CC(=O)Nc2ccc(F)cc2)CC1 C(=O)(C(F)CC(C)(C)C)NCC(CCSC)OC.C1(OC)C(=O)N1 c1(C(N2CCC(NC(c3c(C)ncn3C)=O)C(O)C2)=O)cc(Cl)cc(Cl)c1O Cc1cc2nc[nH]c(=NCC3CC(CNC(c4ccoc4Cl)=O)CO3)c2[nH]1 Cc1ocnc1C(=O)NC(C1(O)CN(C(c2sccc2C(F)F)=O)C1)C CCC(F)(C(=O)OC)C(=O)N1CC2CC1CC2CNC(=O)CCC(C)C C=CC(C)(C)CC(=O)N1CC(CNC(C2C3CCCCCCC23)=O)(OCC)C1 N1(C(c2c(COC)cccn2)=O)CCCC(COC)(NC(=O)C#CC(C)(C)C)C1 Cc1ccc(-c2cc(C(=O)NC(C)CCN3CCCCC3)n[nH]2)c(C)c1 C1(C(N(CCCNC(C=C2CCC(C)CC2)=O)C)=O)CCC2C(CC1)C2(F)F N1(C(CC(CC=C)NC(=O)CCC=C(C)C)=O)CCCC(C)(C)C1C c1(CCC(=O)N(CCCNC(c2csc(O)n2)=O)C)cc(F)cc(F)c1 N1(C(COCCOC)=O)CC(NC(C2CCC(c3ccccc3)O2)=O)C(O)C1 c1(SC)cn(C)nc1C(=O)N(C1CCN(C(C2CCCCC2F)=O)CC1)C c1(NC(CC(=O)Nc2c(C(C)=O)cccc2)C)ncc2[nH]ncc2n1 C(C(C)(C(N)=O)NC(=O)CC1(CNC(c2cncc(O)c2)=O)CCCCC1)OC C(=O)(CC(C)CC(C)(C)C)N(C)CC1N(C(Cc2cn(CC)nc2)=O)CCCC1 C1(CC(=O)NC(C(=O)OC(C)C)C)CCCN(C(=O)CC2C=CCCC2)C1 C1(N(C(=O)CSCCC#N)CC)CCN(C(=O)CCSC2CCCC2)C1 Cc1ccc(OC2CCN(C(=O)C(c3ccc(F)cn3)(F)F)C2)cc1 C1(NC(CN(C(CC2(CSC)CC2)=O)CCOC)=O)CC2(CCCC2)C1 C1(C(=O)NC(CN(CC)CC)C)CCC(C)(C)N(C(c2cc(CO)nn2C)=O)C1 C1(c2cccs2)(C(=O)NC(CC)CNC(=O)C=C(C)C(F)F)CCCCO1 C(=O)(C1=NOC(c2ccccc2)C1)NCCCNC(C(c1cnccn1)C)=O CC1CN(C(C2(CCF)CCC2)=O)CCCN1C(c1cnn(C2CC2)c1)=O c1(CC)ncc(C(=O)N(C)CCN(C(=O)CCc2cnc(C)s2)C)c(O)n1 c1(C(=O)NCC(CO)NC(c2cccc(OC(C)C#N)c2)=O)n[nH]c2c1COC2 C1(CNC(C=CCN(C)CC)=O)CN(C)CCN1C(=O)CCNC(=O)NC c1(C(N(C(CC)CO)C)=O)ccncc1-n1cc(CC(C)(C)C)nn1 C12(NC(C#CC(C)C)=O)CCCC1N(C(=O)CSCc1csc(=N)[nH]1)CC2 N1(CC)OCC(N(C2CCOC(c3ccccc3)C2)C)C1=O CC1CC(CC(N2CCC2CC2CC2)=O)CN1C(=O)Cn1cccc1 c1(C(C)N(C)CC2CCCC2O)ccc(Br)s1 c1(C(N2CCC(C(C)NC(c3c(C)coc3)=O)C2)=O)cc(C(N)=O)ccn1 C#Cc1cnc(C(=O)NC23CCN(C(c4cn(C)cc4C)=O)CCC2C3)c(C)c1 N1(C(Cc2c(C)non2)=O)CC2(CC2)CC1CNC(=O)C(C)(F)F C1(Nc2ncc(C#C)cn2)CC2CC(C1)N(C(C1CCCCC1C(F)(F)F)=O)C2 C1(C(N2CC(C(C)NC(=O)CCCn3ccnc3)C2)=O)C(C)(C)C1(C)C N1(C(c2c(O)ccc(C)n2)=O)CCCC2(C1)C(NC(=O)CCC(C)C)CCN2C C(=O)(CC(C)C(F)(F)F)NCC(=C)CCNC(=O)Cc1cccc(C2CC2)c1 CC(CC(=O)NC1CCOC1C(N1CC(CC2CC2)C1)=O)N(C)C n1(CCC)ncc(CN(C(C(C)(C)C)c2nnnn2CCC2CC2)CC)c1C c1(CCC(=O)NCCN(C(c2c(NC)c(F)ccc2)=O)C)cccc([N+](=O)[O-])c1 c1(C(=O)NC)ccc(C=CC(N2CCC(N(C)C(C3COC(=O)N3)=O)C2)=O)cc1 n1(CC)cnc2c(NC(C)CC(N)=O)[nH]c(=NC(C)c3ccccc3)nc12 N1(C(C2CC(C)C(=O)CC2)=O)CC(O)(C2(CNC(c3cnn(C)c3Cl)=O)CC2)C1 C#Cc1cccc(CC(=O)NC(C)(CO)C(=O)NC(C)CC#CC)c1 c1(C(=O)NCCCCNC(c2cn(CC=C)nn2)=O)cc(Br)c([N+](=O)[O-])[nH]1 c1(C(C)C)ncc(C(=O)NCC(C)N(C(=O)C=CCO)C)n1C c1(NC(N2CCSCC2)=O)cc(O)cc(Cl)c1.C12CCN1C2=O c1(SCC)nc(NC2CCC3(C(=O)OC)CC23)cc(C)n1 C(=O)(CCCCCn1cc(CN2CCCCC2)nn1)N(C)CC1CCCO1 Cc1nc(C(N2CCCC2CNC(c2ncc3ccccn23)=O)=O)c(=O)[nH]c1C c1(C(N2CC(NC(COCc3n(C)ncn3)=O)C(CO)C2)=O)cccc(Cl)c1N CC(CCNC(=O)CCn1ncn(C)c1=O)CCNC(=O)C=C1CCC(C)C1 c1(-c2cn(C(C)C(=O)O)nn2)cccc(NC(CS(=O)(=O)NCCCC#N)=O)c1 C1(NC(c2cc(SC)oc2)=O)C(C)CCN(C(=O)Cc2ccc(Cl)cc2)C1C N1(C(c2cc(C)c(O)nc2)=O)CC2CN(C(c3cc(O)nc(O)n3)=O)CC2(C)C1 c1(C(=O)NCC(CC(=O)OC)NC(C(C(=O)OCC)OC)=O)ncc(Cl)cc1Cl N1(C(C2N(C(=O)OC(C)(C)C)CC2)=O)CCC2(CC2NC(C2CCCCC2)O)C1 C1(NC(Cn2cccc(C(=O)OC)c2=O)=O)CCCN(C(=O)CC2(O)CC2)CC1 c1(CCC)ccc(C(=O)NC(C2CCN(C(c3cc(C(C)=O)cs3)=O)C2)(C)C)[nH]1 CC1(C)CC(CO)(CNC(=O)CC(CC2CC2)NC(=O)C(=O)NC2CC2)C1 N1(C(C(C)N(C(c2c(C(C)C)noc2)=O)C)=O)CC2(CCCC2)C1 N1(C(C(=O)NCC)CCCCOC)CCCCC(C2CCOCC2)C1 C1(CC(=O)N(CCCC(=O)NCC2(OC)CC2)C)CC2(CCC2)C1 C=CCN(Cc1cccc(Br)c1)N1CCCC(C(=O)N(C)C)C1 CN1CCN(CC(=O)NC2(C)CC(NC(=O)CC34CCC(CC3)C4)C2)CC1 c1(CN2CCC(NC(=O)OC)CC2C)ccccc1S(=O)(=O)N(C)C c1(C(N2CCN(C(c3c(C)cc(C)o3)=O)CC2)=O)cccc2ncnc(O)c12 C(=O)(C(O)C(CCC)NC(=O)CNC(C1CC1C)=O)NC(CC#C)C(N)=O O=C1CC(C(=O)NC2CN(C(=O)C=Cc3cnccn3)CCC2CO)CC(=O)N1 CCCC(F)C(=O)N1CCCC1CCNC(=O)CC1CC(F)(F)C1 N1(C(CC2C(NC(Cc3c(C)noc3C)=O)C2)=O)CC2(C1)CC(C)(C)C2 C(C)(C)(CC(F)C(=O)N1CC(n2cnnc2)C1)NC(C(Br)=C(C)C)=O C(=O)(C1=C(C)CN(C(c2cn(C3CCOCC3)nn2)=O)C1)N(CC)CC CCCCCC(C)CC(=O)NC(c1ccnn1C)C(=O)NCc1cn[nH]c1 C1(NC(C2C(C)C2C)=O)CC(C)(CNC(C2CCCCO2)=O)C1 C1(NC(C(n2c(C)cc(C)n2)C)=O)CCN(C(=O)C#CC2CC2)CC1C C(=O)(C(C)(O)C(C)(C)C)N1CCC(CN(C(Cc2c(OC)ccnc2)=O)C)C1 c1(OC)ccc(CC(C)C(N2CCCC(CC(=O)O)C2)=O)cc1S(N)(=O)=O c1(N2CCCC(N(C)C(C3CC3F)=O)C2)ncnc2sc(-c3ccccc3)cc12 N1(CCCNC(C=C(C)C(C)C)=O)CCN(C(c2ncc(Br)cn2)=O)CC1 N1(C(CCC(=O)NCCC)=O)CCCC(C)(CNC(=O)CCc2cnoc2)C1 C1(NC(CC=CCCCCC)=O)CCC(C)N(C(c2cccc(C(N)=O)n2)=O)C1 c1(C(=O)NC(CCCNC(C(CC(C)C)OC)=O)(C)C)cc2cn[nH]c2cn1 CCCC(C(O)C(=O)N(C(C(N)=O)C1CC1)C)NC(=O)CN=[N+]=[N-] CCCCCC(C(=O)NC)NC(C1CN(Cc2c(OC)cccc2F)CCS1)=O N1(C(Cc2ccc(C)cc2C)=O)CC2(CCCC2)C1C(N1CCCC1CF)=O c1(-n2cc(CCOC)nn2)cccc(C(=O)NC2(C)CCSCC2)c1 c1(C(C)(F)F)cc(C(=O)NCC2(C)CCCN2C(c2cc(Cl)c(Cl)s2)=O)ccn1 n1(C(CC)C)nnnc1C(c1nnn(C)n1)NCc1cc(OC)no1 C=CCCCC(=O)NC(C)(C)CCNC(c1sc(=N)[nH]c1C)=O c1(COC)cc(NC(=O)N(CC(c2cccc(Br)c2)O)C)cc(Cl)c1 C(=O)(CC1OCc2ccccc21)N(CCCCN(C(=O)COC1CCOC1)C)C N1(C(C2(C=C)CCN(C(c3n[nH]c(C)c3C)=O)C2)=O)CCCCCCC1CC c1(C(=O)NC(C2CC(NC(=O)CCCN(C)C(C)C)C2)C)cn2c(n1)CCC2 C#CC1(C(=O)NCC2(N(C)C)CC2)CCN(C(=O)C2=CCCC2C)C1 C1(CC=C)(NC(C2CCC(C(N)=O)O2)=O)CCCN(C(c2cc(C#N)cs2)=O)C1 N1(CC=C)CCCCN(C(c2coc(CNC(C3CCCC(F)C3)=O)n2)=O)CC1 c1(C(N2C(CC(=O)NCCC3CC3)CCC2)=O)ccnn2ccnc12 n1(CC(C)CO)nc(CCN(C)C)nc1-c1cn(-c2ccccc2)nn1 C1(NC(c2cnc(CC)nc2C)=O)CCN(C(=O)C(C)(O)COC)C12CCCC2 Cc1oc(CO)cc1C(N1CCC(CNC(=O)C(C)Sc2ccccc2Cl)C1)=O C1(C)(CNC(=O)Nc2c(N(C(C)=O)C)cccc2)CCC(=O)NC1 c1(C(N(CCCCO)C)=O)cc(CNC(c2ccccn2)=O)[nH]n1 c1(OC)cc(C(=O)NC2CC(O)CN(C(=O)Cc3cnns3)C2)ccc1O C1(C)(CNC(CCN(C(C=C(C)C2CC2)=O)CC2CC2)=O)CCCCC1O C(C)(CCC#N)(c1n(CC=C)nnn1)NC(c1nc(COC)no1)C(C)C CN1CC(O)CCC1C(=O)NCCCOC1CCN(C(=O)C=CC(=O)N(C)C)CC1 c1(C(=O)NC(CC)CNC(c2ccn(C)c2C)=O)cnc(O)cc1C c1(CCC)ccc(NC(=O)CC2CN(C(C3CC(=O)C3)=O)CCO2)cc1 CN1C(=O)C(=O)N(CC(=O)NCC2(C)CCCN2C(c2ccno2)=O)C1=O C1(CCNC(CCOCCCNC(C(C2CCCCC2)C)=O)=O)CCCOC1 Cc1nnc(CCC(=O)NC2(C)CC(NC(C3CNC(=O)N3)=O)C2)n1C c1(C(CCCOC)NCCCCOC)ccc(OC)c(F)c1 N1(CC)CCC(C(=O)NCC(CNC(=O)COCC2CCCC2)CO)CC1 c1(CCC(=O)NC2(CCOCC)CN(C(C3CSCC(=O)N3)=O)C2)ccc(F)cc1 Cc1c(C(=O)N(C2CN(C(C3(C)CC3F)=O)C2)C)oc2ccccc12 Cc1nc(C(N2CCN(C(c3cc(CO)on3)=O)C(CF)C2)=O)c(C)n1C1CC1 N1(C(CC)=O)CCN(C(c2ccc(SC(F)(F)F)o2)=O)CC(C)(F)C1 N1(C(c2c(OC)nsc2)=O)CCCC2CN(C(=O)CCc3cscn3)CCC12 c1(C(=O)NC2C3CN(C(COCCSC)=O)C(C3)C2)nccc2occc12 C(=O)(C1=CCCCC1C)NCC(CC=C)NC(c1cc(CC)cc(Cl)c1)=O c1(CC)cc(CN2CCC(COCc3ccccc3F)CC2)n(C)n1 N1(C(Cc2cc(C)on2)=O)CCC2(CCN(C(=O)C(F)(F)C3CC3)CC2)C1 c1(N(c2n(C(CC)C)nnn2)C)ccc2cc[nH]c2c1.c1(SCC)ccc(NC)cc1C c1(C(N2C3C(C(=O)NC4CCC(C)CC4)C(C3)C2)=O)cccc2cccnc12 c1(NC(C(=O)N(C(C)CCN2CCCC2)C2CC2)=O)ncc(-c2ccncc2)s1 C(C(C(F)(F)F)N1CCN(C(c2cc(Br)n[nH]2)=O)CC1)NC(C(C)=CC1CC1)=O C1(C(NCP(C)(C)=O)=O)CCCC(NC(C2(C(C)(C)OC)CC2)=O)C1 C1(NC(C(CC)N(C)C)=O)CCSC12CN(C(c1cc(SC)oc1C)=O)C2 c1(C(=O)NCCC2CCN(C(Cc3n[nH]c(=N)s3)=O)C2)ccc2cnoc2c1 C1(CC)CCN(c2cc(N3CCN(CCCCO)CC3)nc(C)n2)CCO1 c1(C(=O)NCCNC(C(=O)NCC2CCC(O)C2)=O)ccc(F)c(F)c1 CC(Cc1ccncc1)C(=O)NCC(C)CNC(=O)COC1CC1 C1(NC(CCC#C)=O)CCN(C(c2cc(OC)c(Br)cc2F)=O)CC1(C)C S(=O)(=O)(C=Cc1ccccc1)N1C(C(=O)NS(=O)(=O)c2cccc(F)c2)CC1 CCCC(=O)N(CC(=O)NCCc1ncc[nH]1)CC(C)C O(NC(=O)C(CC)NC(c1ncoc1CC)=O)CCCC#C c1(NC(=O)NCc2cc(C)ns2)nc2cc(Cl)c(C)cc2s1 C1(N=[N+]=[N-])(C(N2CCC(CSC)C2)=O)CCN(C(=O)CC2CC(F)(F)C2)C1 C(CCO)(C(F)(F)F)NC(c1ccc(CNC(CC(C=C)C)=O)nc1)=O C(C(N=c1ccc2nnnn2[nH]1)C(C)C)NC(CC(n1c(C)cc(C)n1)C)=O C1(CC(=O)NCCc2ccn(CC)n2)(C(=O)O)CCCCC1 N1(CCNC(C2C(=C)CC2)=O)CCC(NC(=O)C(C)(C)OC(C)C)CC1 c1(C(=O)NC(C)C(C)(C)NC(=O)CC(C)n2cccn2)cnc(O)c2cncn12 c1(C(=O)NCC(=O)NCC(C)CNC(C2CCOC2)=O)cccc(Cl)c1 C1(C(=O)NC2(C)CCN(C(c3cc(C)nn3C)=O)CC2)CC12CCC(C)(C)CC2 c1(OC)cc(C(N2CCCC2C2(NC(=O)C(O)C3CC3)CC2)=O)cnc1Br c1(C(=O)NCCC(CNC(=O)C(F)=CC2CC2)O)ccc(C2CCOC2)cc1 Cc1ccc(C(=O)NC(C2CCCN2C(c2cc(C)on2)=O)C)c(O)n1 c1(C(N2CC(C(C)NC(C3CC34CCSCC4)=O)C2)=O)csc2c1CCCC2 c1(CN2CC(C(N3CC(O)C(F)C3)=O)C2)cc(F)c(Br)cc1Cl C(=O)(CCS(=O)(=O)C(F)(F)F)N1CC(NC(CC(CC)(C)C)=O)C(O)C1 C1(NC(c2cccc(Cl)c2Cl)=O)CN(C(c2cc[nH]c2)=O)CCC12CCOCC2 c1(CCN2CC(n3ncc(CNC(COCC)=O)c3)C2)ccc2oc(C)nc2c1 C1(O)(C(=O)NC(c2nocc2C(=O)N(C)CC2CCC2)C)CCOC1 c1(NC(CNC(C2(CC)CCCC2)=O)(C)Cn2cccn2)ncnc(C)c1OC N1(C(c2ccc(C)s2)=O)CC(C)OC2(CCN(C(C3CCCSC3)=O)C2)C1 Nc1c(C(=O)NCC2CCCC2NC(c2cccnn2)=O)ccc(Cl)c1Cl N12CC3(CC3)CC1CNC(=O)c1nsc2n1.C(=O)(CCC(F)F)OC n1(CC)cnc2c(NCC3(C)CC(C)(C)C3)[nH]c(=NCC(Br)=C(C)C)nc12 C12(C(=O)NC(CCNC(CCCCSC)=O)C)CC(CO)(C1)OC21CCC1 c1(CNC(C(C)=CCC)=O)cc(C(=O)N(CC(O)CC)C)cs1 CCCCC(CC)CCC(=O)NCCCNS(=O)(=O)c1cccnc1C(=O)OC c1(C(=O)NCC2C(NC(c3c(CC)onc3)=O)C2)c(C)cc(C)oc1=O CC1=C(C)CC(C(=O)NC(CCN(C(=O)CS(N)(=O)=O)C)c2cccs2)CC1 N1(C(COC)=O)CCN(C(=O)CCS(=O)(=O)N(C)C)CC(C)(F)C1.C1CO1 N1(C(CN2CCN(C(C(c3cccnc3)C)=O)CC2)=O)CCC2(CC1)CC2 c1(C(=O)O)ccc(Oc2ccc(Br)cc2)c(C(F)F)c1.CCC(N)CNC C(=O)(C=CS(C)=O)NC(C1CCN(C(CC2(COC)CC2)=O)C1)(C)C C1(C(=O)NC)CN(C(=O)C(C2(O)CCC2)NC(C2CCCOCC2)=O)CCO1 CC1=C(C(=O)NC(c2cccc(C(=O)O)c2)C(F)(F)F)Cn2ncnc2N1C c1(C(N(CCCNC(CCC(=C)C)=O)C)=O)nccc2ccccc12 N1(C(C2(C)CCCN2C(c2ccc(B(O)O)cc2)=O)=O)CCCC2(CCOC2)C1 c1(C(=O)NCC(C)N(C(c2ccc(F)c(O)c2)=O)CC)cc2c(nn1)CCCO2 CC1(C)CC(=O)NC1CNC(=O)C(C(C)(C)C)NC(=O)Cn1nccn1 C(=O)(C(C(C)C)NC(C)=O)N(CC=CCC(=O)N(C1CCCC1)CC=C)C(C)C N1(C(C(CCC)NC(N)=O)=O)C2CCC1C1CC1(NC(c1scnc1C)=O)C2 C1(N)CN(c2ncc(F)c(C)n2)CCC1(F)F.Cc1ccccc1CNC1CC1 N1(C(c2c(C#C)c[nH]n2)=O)CC(C(=O)NCC2CC(O)CCO2)C2(CC2)C1 N1(C(C(C)NS(C)(=O)=O)=O)CC2=C(C1)CN(C(=O)Cc1c[nH]ccc1=O)C2 N1(C(CC(C)C)=O)CC2CCN(C(c3cc[nH]c3)=O)CC2C1 c1(N2CC(CNC(=O)OC(C)(C)C)C3(C2)CC3)nc2ccccc2s1 C1(c2ccccc2F)(C2(C(NOCCC(C)O)=O)CC2)CC2(CC2)C1 C1(OC)CC(CNC(=O)CCC2CCOC2)N(C(c2n[nH]c(C)c2O)=O)C1 CC1C(NC(=O)CC2(C)CCC2)CCCN1C(c1csc(C(N)=O)n1)=O C1(C)(CCNC(c2c(OC)csc2)=O)CCN(C(C2(C)CC(C)C2)=O)C1 c1(OC)cc(C(N2CCCC(NC(=O)C(=O)O)C2)=O)cc([N+](=O)[O-])c1 C1(C)(C(=O)NC(C2CCN(C(N)=O)CC2)C)COC(=O)C1.C1CCN(C=O)C1 C1(CCOC2CN(C(C(C)NC(CC)=O)=O)C2)CC(C)CC(C)(C)C1 C(=O)(CCCCCO)N1CCC(N(CC#C)C(C2CC2(Cl)Cl)=O)CC1 C1(NC(c2n(COC)ncc2)=O)CCN(C(=O)Cc2cnccc2C)C12CCC2 Cc1cccc(COCC(=O)NCCC2CCN(C(C3CCCC(=O)O3)=O)C2)c1 Cc1ccnn1C(C)C(=O)N(C1CCN(C(=O)Cc2cnnn2C)C1)CCO N1(C(c2nnn(CC)c2C)=O)CC2CC1CN2C(=O)C(c1c(Cl)cccc1Cl)C CCC(C)(CCNC(c1cnc(C2CC2)o1)=O)NC(c1cc(Cl)ns1)=O C1(C(=O)NCC(=O)OCC)CCN(C(=O)C2(C)CCC(=O)NC2)O1 CCCC(C)(C)CC(=O)N1CCC(CC(=O)Nc2cc(C#N)ccc2C)C1(C)C C1(NC(CCOCCOC)=O)CCC2(CC1)CC2NC(=O)C(C)C(C)(C)C C(C)(C(=O)N(C)Cc1ccsc1)N(CCC)C(C1CC(OCC2CC2)C1)=O N#Cc1cccc(CCC(=O)NCCC2CN(C(C3CCSC3)=O)CCCO2)c1 c1(C(N2CCC(c3nccn3CC)CC2)C(=O)NCCCSC)cc(C)ccn1 c1(C(=O)NC2CCN(CCNC(C(CC)C(C)C)=O)CC2)ccc2nnnn2c1 n1(CC(=O)NCC(CN(C(=O)CC2(O)CCCCC2)C)O)ccc2ccccc12 CC1=NOC(=O)C1CC(N1CCN(CC2CN(C(c3occc3C)=O)C2)CC1)=O C1(CC)CN(C(C2CC2(F)F)=O)CCN1C(c1[nH]cnc1C)=O CCC(O)C(C)C(=O)N(C)CC1CCN(C(=O)CCC(=O)NC2CCCC2)C1 N1(C(C2(C)CC2)=O)CCCC(C2(NC(C3CN(CC(F)(F)F)C3)=O)CC2)C1 N1(C(C(CCC)O)=O)CC(NC(=O)CCSc2ccc(Cl)cc2)CC(F)C1 c1(OC)c(F)ccc(F)c1NC(C1(C)CCN(Cc2cc(Cl)cc(C#N)c2)C1)=O C(=O)(C1CCCc2ncnn21)N1C(C)CCC(NC(=O)C(C)(C)n2ccnn2)C1 c1(C(=O)NCC(=O)N(C(CC)CC)CC2(O)CCCCC2)cc(C)cc(C#N)c1 C(CCC(C)C(=O)NCC(C1CCN(C(=O)C=C2CCN(C)CC2)CC1)C)OC c1(C(N2C3CCC2C(CNC(=O)C(F)(F)C2CC2)C3)=O)ccc2c(c1)CCC2 N1(C(C2(CC)CCC2)=O)CCN(CC2CCN(C(C3CCC(C)C3)=O)CC2)CC1 C1(C(=O)NC(CC(=O)N(C2CCCCC2)C)C2CC2)CC2(CC2)CO1 C1(F)(CNC(c2n(C)nc(C(F)F)c2)=O)CCN(C(C2(C)CC(F)C2)=O)CC1 CC1(C(N2CCOC(CC(=O)NCC(O)C3(Cl)CC3)C2)=O)CC(C#N)C1 N1(C(C2CC(CCC)OCC2)=O)CC(C2(NC(=O)CC(=O)NC)CC2)C1 c1(C(N2CCC(C(O)CO)CC2)C(=O)NC(C(=O)OC)C)sc(Br)c(C)c1C N1(C(=O)OC(C)(C)C)CC(NC(=O)OCc2cc(Br)cnc2Br)CC12COC2 Cc1ccc(C(=O)NC2CCN(C(c3cc(N)ccc3O)=O)CC2C)c(O)n1 N1(N2CC(n3ncc(C(=O)OC)n3)C2)CCN(C)C2(CCOC2)C1 C1(CNC(C(COC)(C)C)=O)(CO)CCCN(C(=O)C(C(C)(C)C)SC)C1 N1(C(CSCCC(C)C)=O)CCCC(O)(CNC(C2CCCC(=O)N2C)=O)CC1 CC1(C)C=CC(NC(=O)NC2CC(OCC(F)(F)F)C2)CC1 C(=O)(CC(=O)N1CCCC1CN(C(=O)Cc1cccs1)C)NC Cc1[nH]nc2cc(C(=O)NC3CC3NC(c3c4c(nn3C)CCSC4)=O)ccc12 C1(NC(C(C2CCC2)OC)=O)CN(C(=O)C(C)(C)C#N)CC1c1ccccc1F C12CC13CCN(C3)C(=O)CCN2.Cc1cc(CNC(C2(F)CC2)=O)no1 CCC(O)CC(=O)NCCOCC(=O)NCC1CCC(=O)NC1 c1(C(N2CCC(C)(CCNC(CCCOCC=C)=O)C2)=O)cc(C)ccc1N c1(NCC(C)CNC(=O)CNC(=O)N(c2ccccc2)C)ccn2ccsc12 O=C1CCc2cc(CN3CCC4CC(C(N5CC=CC5CO)=O)C4C3)ccc21 c1(C(=O)NCCC(C)NC(C2CC3C=CC2C3)=O)ccc(-c2ncc[nH]2)cc1 C1(NC(CCN(C)C(C2CCC(O)CC2)=O)=O)CC(O)C(O)C1 C1(NC(c2c(C)ncnc2C)=O)CCC2CCN(C(=O)C(C)n3ccnc3)C12 C1CC(F)CCN1c1c(-c2cn(CC(CC=C)(C)C)nn2)cccc1.C(N)=O C1(NC(C(CSC)OC)=O)CN(C(=O)C=Cc2ccc(Br)cc2)C(C)(C)C1 c1(C(N2CC(NC(C3N(CC)CCCC3)=O)C(C)C2)=O)cc([N+](=O)[O-])ccc1C C1(NC(CSC(C)(C)C)=O)CN(C(c2cc(C(C)(C)C)ccn2)=O)CC1C(F)F c1(C(C(=O)NCC(COC)NC(=O)Cn2[nH]cnc2=N)C)cnn(C)c1 C(C1NCCc2sccc21)NC(C1(c2nccc(OC)c2)CCCCC1)=O C1(C(=O)NCC(CNC(c2ccc(C(N)=O)[nH]2)=O)CO)(COC)CCOCC1 N1(C(COC)C)CCN(C(=O)C=Cc2ccccn2)C(=O)C1 C1(CC)(NC(=O)CC2CCCC2)CCN(C(c2c(OC)cccc2Br)=O)CC1 C1(C(=O)NCCN(C(C2CC2c2nc(C(=O)N)no2)=O)CC)CC(C)(O)C1.OC C1(CNC(C(C(=O)OC)(C)F)=O)CC2CCC(C1)N2C(C1(CC2CC2)CC1)=O Cc1ccc(C)n1C(C)C(N1CC(O)(CCNC(C2CCCCN2C)=O)C1)=O N1(C(c2ccc(C(F)(F)F)o2)=O)CCC(Oc2cncc(Cl)n2)CC1 CCCC(C(=O)NC(C)(C)CCNC(=O)CC1CCC(F)(F)C1)OCC C1(NC(c2ccc3nccn3c2)=O)CS(=O)(=O)C2CN(C(c3ccsc3)=O)CC12 c1(CN2CC(NC(c3cc(-c4ccncc4)no3)=O)C2)cc(Cl)cc(Cl)c1Cl N1(C(C2N(c3cc(OC(C)C)ncn3)CC2)=O)CCN(C2CC2)C(=O)C1 c1(C(=O)NC2CN(C(C3(F)CC3)=O)CC2O)cccc(C(F)(F)F)c1Cl Nc1c(C(N2CC3(C(=O)O)CC2CCO3)=O)cc(F)cc1Br c1(C(=O)NCC2CC(NC(c3cc(C)sc3C)=O)C2)ccsc1S(C)(=O)=O N1(C(C2N(C(=O)COc3ccsc3)CCC2O)=O)CCOCC(C2CC2)C1 C1(C(=O)NC(CC)CCCO)C(C)OCCN1C(C1CCCC1O)=O C1(C(CNC2c3ncoc32)=O)CCC(C)(C)CC1.C1(COC)CCCC1 c1(NC(C2CC(F)CN2Cc2ccc(Cl)cc2)=O)cccc(OC(F)(F)F)c1Cl CC1CN(C(=O)C(c2ccccc2F)(C)O)CC1NC(=O)C=CC1CCC1 c1(C(=O)NCC(CC)NC(c2ccccc2OC)=O)cnc(C)nc1OC C12(C(N(C(C)CNC(C3(F)C(C)(C)C3(C)C)=O)C)=O)CCC(N(C)C)(CC1)CC2 c1(OCC)cncc(C(N2CCC(OCCNC(c3ccnnc3C)=O)C2)=O)c1 N1(C(c2cc(=N)[nH]cc2)=O)CCC2C(NC(C3CC3C(F)(F)F)=O)CC12 CC12CC3CC(CC(C(N4CCOC(CNC(=O)C5=NOCC5)C4)=O)(C3)C1)C2 c1(C(=O)NCC(CO)NC(c2ncc(C#N)cc2Cl)=O)cnc2[nH]c(O)nc2c1 Cc1csc(C(=O)N(C)CC2CCCC2NC(c2ccnn2CCF)=O)c1C C1(O)(C(N2CC(CNC(c3cccc(C)c3O)=O)C(C)C2)=O)CCCC(C)(C)C1 c1(NC(CC2CN(C(Cc3cc(C)cc(C)c3)=O)C2)=O)ncc([N+](=O)[O-])cc1Cl Cc1c(-c2nnc(C3CN(C(=O)OC(C)(C)C)C3)o2)ccn1C1CCCCO1 C1(NC(c2n(C(CC)C)nnn2)c2cc(C)on2)(CSC)CCS(=O)(=O)CC1 CCC(CC)C(C)C(=O)NC1CCN(C(c2cc(C)n(C)n2)=O)C1(C)C N1(C(C(C)=CC)=O)CCCOC(CNC(=O)CCC2CC2(Cl)Cl)C1 N1(C(C(c2c(C)noc2C)C)=O)CCCN(C(c2nc(Cl)ccc2N)=O)CCC1 C1(NC(c2c(C)cc(CC)o2)=O)CCN(C(c2sc(C(C)C)nc2C)=O)CC1O Cc1snnc1C(=O)NC(C1CC1C(=O)NC1(N2CCCC2)CCC1)C c1(C(N(C2C(C)CCN(C(CCC=CC)=O)C2)C)=O)cccc2c(C)ccnc12 Cc1ccc(F)c2[nH]c(C(=O)NC3CN(C(C4CCC(=O)N4C)=O)CC3C)cc12 C=CC1(C(=O)NCC2(C)CCC(=O)N2)CCN(C(=O)C(n2nccc2C)C)C1 CN1CCN(C(CC2(C)CC2)C(=O)Nc2ccccc2)CC1C1CC1 Nc1cccc(CC(=O)NCCCCC2CCCN2C(C2CCC(=O)N2)=O)c1N c1(CC)noc(CC)c1CC(N1CC(C(C)NC(C2(C)CC(F)C2)=O)C1)=O N1(C(CCCC(C)C)=O)C2CCC1CC(NC(c1conc1C1(C)COC1)=O)C2 C(=O)(C(CC(C)C)CC(C)C)NC1C(CNC(C(C=C)(C)C)=O)CCC1 C12(C(=O)NC3CC(N(C(c4c(C)nc(C5CC5)[nH]4)=O)C)C3)CCCN1CCC2 CC1COCC(CC(=O)NCc2cc(C(=O)N(C)CCN3CCCC3=O)on2)O1 C1(CN(c2nnc(-c3cccc(O)n3)n2CCC#N)C)CCc2c[nH]nc2C1 c1(-n2cc(C3CC(C(=O)NC(C(CC)C)=O)C3)nn2)cccc(Cl)c1 C12(C(=O)NC3(C(=O)NC4C=CC(C(=O)OC)C4)CC3)C=CC(CC1)C2 N1(C(C=CCCC)=O)CC(NC(C2(CO)CCOC2)=O)CC(C)C1 N1(C(CC2C(C)(C)C2)=O)CC(NC(=O)CSC(F)F)C2CCCCC12 c1(C(N(C(CNC(c2ccc(OC)cn2)=O)C)C)=O)ccc2ocnc2n1 c1(C(N(CCNc2cc(I)c(O)c(I)c2)CC)=O)ccc(OC)c(O)c1Cl C(=O)(C1=NOC(C)(C)C1)NC(C)C(=O)NC(C)Cc1ccnn1C N1(C(CC2CC(C(C)C)OCC2)=O)CCCC2(NC(=O)C(F)CC3CC3)CC2C1 C1(C(=O)NCC2(C(C(C)C)O)CC2)CCN(C(C2CC3CCC3C2)=O)CC1C.N c1(OC)cc(CC(=O)NC2CCCN(C(=O)C=C(Cl)Cl)CC2)cc(F)c1 c1(C(N2C(CN(C(=O)CC3COC(=O)C3)C)CCCC2)=O)cnc2ccnn2c1 c1(CC(C(N2C(OC)CSC2)=O)NC(=O)OC(C)(C)C)ccc(C)c(C#N)c1 N1(C(CCSCCNC(c2c(CC)nn[nH]2)=O)=O)CCC(C)C(CO)C1 N1(C(CCNC(COC)=O)=O)CC2(COC(CNC(=O)Cc3cnsc3)C2)C1 Cc1ccc(C(=O)NCC2CN(C(=O)Cn3cnc(Br)c3)C2)s1 C1(CC#C)(C(=O)OCC(C2CCCCO2)=O)CCCN(C(=O)OC(C)(C)C)C1 n1(CC(C)C)[nH]c(CC(=O)N(C2CN(C(=O)C(F)C3CCOC3)C2)C)cc1=O C1(NC(c2ncccc2O)=O)CN(C(c2cnn(C3CC3)c2)=O)CC12CC2 CC1(NC(=O)CC2C=CCC2)CCN(c2nncs2)CC1 CC1(C)C(C(=O)NCCc2ccc(-c3nn[nH]n3)cc2)CC12CCN2 C1(NC(C(CC)C(C)C)=O)CC2(CCN(C(=O)C#CC3CCCO3)CC2)C1 c1(C(CC)C(Br)NCC(=O)NCc2cn(CNC3CCC3)nn2)ccc(C#N)cc1 c1(C(N2C3C(CNC(C(CC)(C)O)=O)CC(CC3)C2)=O)ccc2cncn2c1C C=CC(C)(CC)C(=O)NC1CCN(C(C23CC(C)(C2)OC3C)=O)CC1C N1(C(c2[nH]cc(C)c2C)=O)CCN(C(C2(c3cccc(C#N)c3)CC2)=O)C2CC12 N1(CCC)CCCC1C(N1CC(CNC(C2COCC2C(N)=O)=O)(OC)C1)=O C(=O)(C1=CCCOCC1)NCCN(C(c1cncs1)=O)CC CC1COc2c(C(N3CC4(CSC4)C3)=O)cccc21 c1(C(N2CC3C(NC(c4ccc(CC)s4)=O)C(C3)C2)=O)cccc2nnn(C)c12 c1(C(=O)NC(C)CN2CCN(C(=O)C=C(Cl)Cl)CC2)cnc2[nH]cncc1-2 c1(OCC)ccc(C(N2CCC(F)(C(=O)NC(C)CCO)CC2)=O)cc1Br CCCCS(=O)(=O)Nc1cccnc1C(N1CCN(CCC)CC1)=O c1(-c2cccc(Cc3c(C)noc3C)c2)sc(=NCc2c(O)cccc2F)[nH]c1C C1(C(N(CCN(C(C2C(=C)CC2)=O)C)C)=O)COCCC1C c1(NC(C2(CNC(CCCCCCC)=O)CC2)=O)ccc2cccnc2c1 C(C(=O)NN1CCCC1C(N1CC(C#N)(SC)C1)=O)SCCCCC C(=O)(CCCCCCCCC1CC1)NCC1C(NC(C(C)(C)SC)=O)CCC1 c1(NC(c2nnn(C)c2C)(c2nnnn2C2CCCC2)CC)ccc(OC)cc1 N1(C(C2(C)CC(=C)C2)=O)CCC(NC(=O)CC2(C#N)CCC2)C(C)C1 C#CC1(C(=O)NC2CCC(CC(=O)NC(CC)CCO)CC2)CCCC1 c1(OCCC)cccc(C(=O)N(CCCN(C(=O)C(C)CSC(F)(F)F)C)C)c1 C1(C(=O)OCC)CN(N2CC(c3ccccc3)CC2C)CC2(CCC2)O1 O=C1CCCCC(C(N2CCCN(C(C3CCC(F)(F)C3)=O)CC2)=O)N1 C1(C)(CC)CN(C(c2cccc(OC3CC3)c2)C(=O)NC2COC2)CCO1 CC1(C)CC(CO)CCN1C(=O)CC(O)CNC(=O)CCc1cccnc1 CS(=O)C=CC(=O)N1CC(NC(C2(CO)CC(F)(F)C2)=O)C(CC2CC2)C1 c1(C(=O)OC)cccc(Cl)c1.C1(C(N(CCOC)CCN(C)CN)=O)CC2CCC1C2 C(=O)(CC1CCOc2ccccc21)N1CC(O)CC(NC(CN(C)C(N)=O)=O)C1 C(=O)(CC(O)CC)N(CCC(=O)N(C1CCN(C)C1)C)CC=C C1(CNC(C(C=C)(C)CC)=O)C2CCCC1N(c1nnc(CC(F)(F)F)s1)C2 c1(NCc2ccnc(C)n2)[nH]c(=NC2CCCN3CCCCC23)nc2sccc12 N1(C(c2c(C)con2)=O)CCC2(CC1)COC(CNC(c1cc(Br)n[nH]1)=O)C2 CCCC(C#N)C(=O)NCC(C)(CC)NC(=O)C=CCN1CCOCC1 N1(C(c2n(CC)nc(C)c2)=O)CC2CCC2(NC(c2ccoc2Cl)=O)C1 C(=O)(C(CCOCCO)NC(=O)C(C)C(=O)OC)NC(C(=O)OC)C1CC1 n1(C(CC)C)nnnc1C(CCC1CCCC1)NCCOCCO c1(CN2CCN(C(=O)Nc3cc(Cl)ccc3Cl)CC2)cc(F)cc(F)c1F c1(CC(=O)NC2CCN(C(CN(C(C)C)C)=O)CC2CO)ccc2nn[nH]c2c1 N1(C(c2cc(C(C)C)[nH]n2)=O)CCN(C(=O)C(O)Cc2cnc[nH]2)CC1C C(=O)(CC(C)(C)C)NC(C(C)C)Cn1cc(C2CCN(CC(C)(C)O)CC2)nn1 CC(C)C(CNC(=O)C(F)C1CCCC1)C(=O)NCC1CCOCC1 c1(OC(C(=O)N(CCNC(=O)CCCOC)CC)CCN)ccc(Cl)c(Cl)c1.OCN C1(C(C)NC(c2ccno2)=O)CCN(C(c2ccc(OCCO)cc2)=O)CC1 C1(=O)C(CCCC=C)NC(=O)CO1.C#CCC(C)(COC=O)CO.C1(O)CC1 c1(NC(c2nccc(OC)c2C)c2n(CCOCC)nnn2)c(F)cc(Cl)cc1Cl C1(CC)CN(C(c2ccc(CF)cc2)=O)CC1NC(c1cc(C#N)c[nH]1)=O N1(C(CC2CCCC(C)O2)=O)CC2(CC(NC(=O)C(=Cc3cccnc3)F)C2)C1 C1(C(=O)NC(COCC)C(C)C)CCCCN(C(=O)C(C)(C)O)C1 C=CCC(CC(=O)NC1CCOCCC1)NC(c1ocnc1C)=O c1(CC(=O)NC2C(CNC(C(COC)C)=O)CCC2)ccc2c(c1)CCN2C c1(-c2cccc(C#N)c2)n[nH]c2c1CN(C(c1ncc(Cl)cn1)=O)CC2 C(=O)(C1=CC2(CN(C(=O)C(C)C3CCOC3)C2)OC1)Nc1cncc(COC)c1 N12CC3C(C3C1)NC(=O)NC2=O.C(C(C)(C)N1CCCC1)N(C(C)C)CCN C1(OCC)COCC1N=c1[nH]c(=NC(C)Cc2ccc(Cl)cc2)[nH]c2c1CSC2 CCN=c1cc(-c2nc(Cc3ccc(C)cc3)n(-c3ccn(CC)n3)n2)cc[nH]1 CC(C)C(C(=O)NCC(CNC(C12CCCC1(C(N)=O)C2)=O)C(F)(F)F)C(C)C C1(CNC(C(CCC)C)=O)CCCC2(CN(C(=O)CC3CCOCC3OC)C2)O1 C=CCCC(C(=O)N1CCOCC1CN(C)C)NC(=O)C(F)CN(C)C C(=O)(NNC(=O)c1cc(C(C)C)on1)NCCOCCC CC1CC(N=c2c([N+](=O)[O-])c[nH]c3ccc(F)cc23)CCN1C(C1CCC1)=O c1(-n2cc(C(CCC)NC(c3ccccc3CO)=O)nn2)cc(F)ccc1C C1(C(N2CC(CC(=O)Nc3c(OC)nn(C)c3)(OC)C2)=O)CC2CC(=O)C1O2 Cc1cc(C(=O)NCC(=O)NCCN(C)C(c2cc(C#N)c[nH]2)=O)n(C)n1 N1(C(C(COCC)C)=O)CC2CCC2(NC(=O)COCC2CCOC2)C1 N1(C(Cc2c(OC)nccc2)=O)CCN(C(C2(c3nc[nH]n3)CC2)=O)CC1C N1(C(C(CC=CC)C)=O)CCC(NC(=O)C2=CCOC2)C1(C)C C1(NC(c2ccccc2-c2ccccc2)C)CC(C)N(c2nnc(C#N)s2)C1 CC(F)(C(=O)NCCC1CN(C(=O)CCCc2ccccn2)C1)C(F)(F)F c1(C(=O)NCC(CCCC)NC(c2cc3scnc3[nH]2)=O)n[nH]c2c1CC1CC21 C1(C(=O)NCC(CC)NC(=O)Cc2csc(CN(C)C)n2)CCS(=O)(=O)C(C)C1 C(=O)(C(CC=C)C(C)C)N(CC(=O)N(CC(C)(C)CO)C)CC#C N1(C(CCCNC(CC)=O)=O)CC(OC)CC(NC(c2cc(C)sc2C)=O)C1 Cc1csc(C(=O)NC2CCC2NC(C23COC(CO)(C2)C3)=O)c1Cl CC1CN(C(=O)Cc2ccc(O)nc2)CCN1C(c1coc(Cl)n1)=O CC1(C)OC(=O)C(CC(=O)NC2CC(NC(=O)CSc3nc[nH]n3)C2)O1 C12(OC)CCCCC(C(=O)NCCN(C(=O)C3=CCCS3)C)(C1)C2 c1(C(=O)NCC(N(C(C2N(C)CC2)=O)C)C2CC2)cc(Br)cs1 c1(C(C)(C)OC)nc(C)c(C(=O)NC(CNC(C2CCSCC2)=O)C2CC2)s1 c1(CN(C(=O)C(C)(F)F)C(C)C)cn(CC2CCCO2)nn1 N1(C(C(C2CCCC2)OC)=O)CC2CC2(NC(=O)COC)C1.C12CN(C1)C2=O N1(C(c2nc(C)oc2)=O)CCN2CCN(C(C3CC34CCCC4)=O)CC2C1 N1(CC)CCCC(C(=O)NC(C)(CO)C(=O)N(CC(C2CCCC2)O)C)C1 C(=O)(C1=COCCO1)N1CC(CCNC(=O)C2=COCC2)(OC)C1 c1(C(C)=O)cccc(-n2ncc(-c3noc(-c4csc(S)n4)n3)c2N)c1 N1(C(c2csc(Cl)n2)=O)CCOC(C2CN(C(=O)C=CC=C(Cl)Cl)C2)C1 C1(C(=O)NCC2=CCN(C(C3C(C)(CC)C3)=O)CC2)CC(c2cccnc2)=NO1 C=CCCCCC(=O)N1CCCC(NC(C2CCCC2F)=O)CC1 C1(NC(c2ccc(C3CC3)o2)=O)CN(C(C2CC3CCC2O3)=O)CC2(CC2)C1 C(=O)(CC(C)C(C)(C)NC(=O)CN1CCC(=O)CC1)NCc1cccc(OC)c1 C(C(COC)C(=O)N1CC(F)CC1Cn1cc(C2OCCO2)nn1)OC C(=O)(N=c1ccc(OC)c(OC)[nH]1)C1CCCN(c2ncc(CC)cn2)C1 Cc1cccc(C(=O)NCC2C3CN(C(c4ccc(F)cc4)=O)CC23)c1C#N C12(NC(C(C)NC=O)=O)CCC(C(=O)NC(c3ccsc3)(C)C)(CC1)C2 C1(O)(CNC(C2C3(CC3)C23CC3)=O)CCN(C(C2CCOC2=O)=O)CC1 C1(C#N)(NC(CN(C(c2cn(CCC)nc2)=O)CCOC)=O)CCOCC1 C(CC1CCC1)(C(=O)NOCCCCF)NC(=O)CC1CC=CC1.O=CO C(=O)(C(CNC(C1(OC)CC(C)C1)=O)C(C)C)Nc1cn(CC(=O)NCC)nn1 CC(CN=c1[nH]c(N2CC3OC3C2)nc2c1COC2)c1ncc[nH]1.C(F)(F)F C12(NC(c3ccc(F)cn3)=O)CCCCC1CN(C(C1CC3CCC1CC3)=O)C2 c1(C(=O)OCC)sc(C(=O)NCCC(O)CNC(C2CC2F)=O)c2c1CCCC2 C1(NC(c2scc(C)c2C)=O)CN(C(C23CCCC2(C(N)=O)C3)=O)CC1(C)C c1(C(=O)NCCCNC(C2(F)C(C)C2)=O)cccnc1OC(F)(F)F.C1(O)CCCC1 n1(C(C)C)ncc(C(=O)NCC2C3CN(C(=O)Cc4conc4C)CC23)c1N c1(OC)c(F)cc(F)c(N(C)CCN(C(=O)Cc2cncnc2)C)c1[N+](=O)[O-] C(N=c1cc(CCC2CCCC2)nc[nH]1)C1CS(=O)(=O)CC1O C1(NC(CCCOCCOC)=O)CN(C(c2csc(Cl)c2)=O)CC1n1ccnn1 C12(CNC(c3cc(C4CC4)[nH]n3)=O)CCC1CN(C(c1cc(Br)co1)=O)C2 c1(C(N(CC(C)NC(c2cc[nH]c2)=O)C)=O)ccnc(OCCN(C)C)c1 C1(CNC(C2(CCC)CCC2)=O)CCN(C(=O)CCC=CBr)CC1C CS(=O)(=O)C1(C(N2CCCOC(c3c(C(=O)NCCCl)cc(C#N)o3)C2)=O)CCC1 c1(C(N(CCN(C(C(C)(CO)OC)=O)C)C)=O)cc(C)c2sccc2c1 c1(C(N2CCC(C)(C#N)C2)=O)ccn2ncccc12.c12cccc(c1)CNC2=O N1(C(c2c(C#C)c[nH]n2)=O)CCC(C=C)(C(N2CCCC(CC(N)=O)C2)=O)CC1 C=CC(CC)CC(=O)NC1CCN(C(=O)CNC(c2c(F)cccc2Cl)=O)C1 C(=O)(CCCN=[N+]=[N-])NC1(C(N(CC(C)C(F)(F)F)C)=O)CSC1 N1(C(C2CCC(=O)N2)=O)CCC(C(N2CCC(Oc3ccc(F)cc3)C2)=O)C(O)C1 c1(C(=O)NCC(CNC(C(COC)(C)O)=O)C(F)(F)F)ccc(S(C)(=O)=O)cc1 CCCCC(CC)CCNC(c1sc2ccccc2c1Br)c1nnnn1C(C)C c1(-c2ccc(NC(c3ccc(Cl)c(Cl)c3)=O)c(O)c2)ccn2cnnc2c1 N1(C(=O)Nc2ncc(OC)s2)CC(C)SC(C)C1 N1(C(C2(C)CC=C(C)CC2)=O)CC2(CCC(CNC(=O)CNS(C)(=O)=O)O2)C1 c1(C(=O)NC2CC(F)(CNC(c3occ(C(N)=O)c3)=O)C2)cccc(F)c1 Cc1cccc(Cl)c1CC(N1CCC(O)(CNC(C2CCC(O)CC2)=O)C1)=O N1(C(c2nocc2CC)C(=O)NC(CC)C)CC(=O)N(C)C(C)C1 C#CC1(C(=O)NCC2CCCN2C(C2CC(N3CCCC3)C2)=O)CCC1 O=C(CCCCCl)NCC1CC1(F)F C=CCCCCCCC(=O)N1CCCC(C(=O)NCCC(C)CO)(CC)C1 c1(C(N2CC(F)(CNC(c3c(COC)ccs3)=O)C2)=O)cccc(Cl)c1Cl N1(C(c2cc(=N)[nH]cc2)=O)CC2CCN(C(=O)CCc3cnoc3)CCC2C1 C(C(CC(C)C)NC(c1csnc1Br)=O)NC(C1(NC(C)=O)CCC1)=O C(=O)(CCCC(=O)NCC(CO)NC(=O)C(CCC)c1ccccc1)OCC C1(CC=C)(NC(=O)Cn2cccn2)CCN(C(C2CC2(F)F)=O)CC1 CC(C)CCC(O)C(=O)N1CCN(C(c2ccc(Br)o2)=O)CC2(CC2)C1 c1(C(N2C(C)(COC)CC2)=O)c(C)nn(-c2ccc(C#N)cc2)c1C C(Cc1ccccc1)(CCNC(C1(Cl)CC1)=O)NC(c1cncnc1)=O Cc1nc(N2CCOCC(NC(=O)CS(=O)(=O)Cc3cccs3)C2)cc(Cl)n1 C1(COC)(CNC(C2(CC(C)C)CC2)=O)CCCN1c1nnc(-c2ccon2)s1 Cc1ccccc1-c1cn(C(C)CN(C(=O)CCN2CCCC2)C2CCC2)nn1 CC(CCC(C)(C)C)C(=O)NC1(C(=O)NC2CCn3cncc3C2)CC(F)C1 N1(C(CCN(C)CCO)=O)CCCC(C2CCN(C(=O)C(C)(C)CN(C)C)C2)C1 Cn1nc(Br)c2ccc(C(N3CC(F)CC3C(=O)NC(C3CC3)C3CC3)=O)cc12 N1(C(c2c(C)c(Cl)cnc2)=O)CC2CN(C(=O)CC(O)CCN(C)C)CC2(C)C1 Cn1ccc2ccc(C(N3CCCC3CC(=O)NCc3cncc(O)c3)=O)cc12 C1(C(=O)NCCN(C(C2CCN(C)C2=O)=O)CC)CCc2nc[nH]c2C1 CCC(CNC(C1(F)CCCN(C(=O)Cn2nccn2)C1)=O)C(C)(F)F C(=O)(CCCCCO)NCC(C)N(C(C(COC)C)=O)C c1(C(C)=O)ccc(C(=O)NCC2CC(NC(C3CCCC3C(N)=O)=O)C2)c(F)c1 C#CCC(C)C(=O)N1CCCC(CN(C)C(c2coc(C#N)c2)=O)C1 C1(NC(C(CC)C)=O)CCCN(C(=O)C=Cc2ccc(SC(F)F)cc2)CCC1 C(CCCC(C)(C)C(=O)NNC(=O)C1CCCCO1)NC(C(C)C(C)(C)C)=O c1(C(=O)NCC2OCCCN(C(c3ncc(C)cn3)=O)C2)cnc(O)n(C)c1=O C1(NC(C(CC)(C)C)=O)CC(F)(F)CC1NCC1CCN(C(C)=O)CC1 C1(NC(C2(CC)CN(C3(C#N)CC(C(=O)OC)C3)C2)=O)CC(O)C(O)C1 N1(C(CC(CCC)O)=O)CC2CC(C1)N(Cc1nn(C)c(=O)n1C)C2 N1(C(C=C(CC)C)=O)CCN(C(=O)CC(O)C2CCCC2)CC1CC(F)(F)F c1(CC)cc(C(N2CCCC(CC(N3CCC3C(=O)NC)=O)C2)=O)ncn1 O=S1(=O)CCc2cc(CNC(=NCCCC3CC3(F)F)NC3CCCC3)ccc21 c1(OC)cccc(O)c1C(N1CCN(C(c2cc(C)c(C)o2)=O)C(C(C)C)C1)=O Cc1cc(O)cc(Cl)c1C(=O)NC1CCCCC1CNC(=O)CCCN(C)C N1(C(CCOCC)=O)CC(NC(c2cnc(N(C)C)s2)=O)CC(C)C1 c1(CC(N2CCN(c3ncccc3F)CC2)=O)cc(F)ccc1C(F)(F)F C(=O)(C(F)CC(C)(C)C)NC1CC(CCNC(c2c(C)n(C)nn2)=O)C1 Cc1nnc2ccc(C(N3CC(NC(C4CC5(CCC5)C4)=O)C(C)C3)=O)cn12 CC1CNCC(CC(=O)NC(=O)CC(c2ccc(Cl)cc2)C2CC2)O1 c1(C(N2CCN(C(CC(=C=C)C)=O)CC(O)C2)=O)cnc2ccccc2c1C C1(N(N2C(C3(C=O)CC3)CCC2)C)C2CC3C(C2)C13.c12c[nH]c(c1)C2=O.CC C1(NC(c2nccc(OC)c2OC)=O)C(C)CN(C(c2cnc(Cl)s2)=O)CC1C C1(NC(C(c2ccc(C)cc2)O)C)CC(C)(C)OC(C)(C)C1 N1(C(CC2(C)CC2(F)F)=O)CC(NC(c2ccc(Cl)c(O)c2)=O)CC12CCC2 c1(-c2cnc(SCc3ccc(OC)cc3)o2)ccc(C)cc1C c1(NC(CCNC(C2C(C)C2)=O)=O)ccc(C(=O)NC2CCN(C(N)=O)C2)cn1 c1(COC)nc(=NC(=O)c2ccc(C(C)(C)S(C)(=O)=O)cc2)o[nH]1 C(=O)(C1=CCCN(C(C2CCN(C)C(=O)C2)=O)C1)Nc1c(C(C)C)cccc1 c1(OC)ccc(Cl)c(C(=O)NCC(C)CNC(c2nc(C)ccc2C)=O)c1F n1(C(C)C)ncc2c(NCC(F)CO)[nH]c(=NC3CCCCC3F)nc12 N1(C(CC(C)F)=O)CCc2c(c(CNC(C3CC3F)=O)nn2C)C1 C1(C(=O)NC(CNC(C2CC(CC)C2)=O)(C)CC)CCc2nnc(O)n2C1 c1(C(N2C(CNC(c3cnc(C)nc3)=O)CCCC2)=O)ccc2occc2c1O c1(C(=O)NC2CC(CNC(=O)C(C3CCCO3)C3CC3)C2)cccn2nncc12 C(=O)(CC1CC(C(C)C)c2ccccc21)NCC1C(NC(COC(C)=O)=O)C1 c1(C(=O)OC)ccc2nc(NC(c3ccc(Cl)cc3Cl)=O)[nH]c2c1 Nc1ccc2nc(N3CCCC(CO)(NC(=O)C=Cc4ccccn4)C3)sc2c1 c1(C(=O)NCC2(CNC(C(C)NC(N)=O)=O)CC(F)(F)C2)cc(S(N)(=O)=O)c[nH]1 N1(C(C(C2CCOC2)NC(C)=O)=O)CCC(NC(=O)C(C)N(C)C)C2(CCC2)C1 C(=O)(C(C)CC(F)F)NC(C(=O)NCc1ccc(C)cc1)C1CCC1 N(C1c2cc(F)ccc2CC1C)C(c1c(SCCOC)cccc1)=O c1(OC)ccc(C(=O)NC2CN(C(C3(C#N)CC(=O)C3)=O)CCC2C)c(C)c1 N1(C(C(CC)(C)O)=O)CCC(O)(CN(C)C(C2CN(C(C)=O)CCO2)=O)CC1 N1(C(c2c(NC)cnnc2)=O)C2CCC1C(NC(=O)COC1(C)CCCC1)C2 CC(=O)CCCC(=O)NCC1CN(C(c2cc(CN(C)C)on2)=O)CCC1C c1(C(=O)NCC2C(NC(C(C)(C)c3ccccn3)=O)CCC2)cnc2n1CCS2 N1(C(C2(CC)CCN(C(=O)CC3CCC(=O)C3)C2)=O)CCC2(CC1)CC2C#N C1(NC(C(CN(C(c2c(OC)csc2)=O)C)(C)C)=O)COCC1C1CC1 CC(C)(CC(=O)N1CC(C2(NC(c3ccc(O)nc3)=O)CC2)C1)C(F)F c1(C(N(CC(CNC(C2C(C(C)C)OCC2)=O)(C)C)C)=O)cnc2c[nH]nc2c1 c1(C(=O)NC2CN(C(=O)C=C3CCC3)C2)cc2sc(N3CCCC3)nc2s1 C12(C(=O)NCCCOCCNC(C(c3ccn(C)n3)C)=O)CCC(CC1O)C2 Cc1cc(C(N2CCC(C)C2CNC(c2cc[nH]c3nccc2-3)=O)=O)c(O)cc1F S(=O)(=O)(c1cnc(NCC2CC=C(C)CC2)c(Cl)c1)NC(CC)COC c1(CNC(C(CCOCCO)NC(CC(CC)C)=O)=O)cc(C)nc(C)c1 CN1CC(C(=O)NC2CC(NC(C3CC(=O)N(c4nccs4)C3)=O)C2)CC1=O C1(NC(c2c(SC)ccs2)=O)CN(C(=O)C(O)CC(F)F)Cc2ccnn2C1 N1CC(C)(C)OCC1CNC1CC(CNC(=O)CS(=O)(=O)NC)C1.CCCC1CC1 c1(NC(=O)Nc2cccc(CO)n2)ccc([N+](=O)[O-])cc1 CC(C(=O)NOC1CCN(C)CC1)NC(=O)C(=O)Nc1ccccn1 c1(Cc2c(C)ccs2)nc(Cn2cccn2)nn1C1CCSCC1 Cc1c(Br)c(C(=O)N(C)CC2(O)CCN(C(=O)C3=CC(C)(C)C3)C2)nn1C C(=O)(C1CCCc2ncc(C)n21)NC(C1CCCC1)CNC(CNC(C)=O)=O c1(C(=O)NC2(CCNC(c3ccsc3Br)=O)CCC2)c[nH]c(=O)cn1 c1(CCSC)cn(CC(=O)NC(COC(=N)O)Cc2ccccc2)nn1 c1(C(=O)NCC2C(NC(c3ncn(CC)c3)=O)C2)ccc(=O)n2c1CCCC2 N1(C(C(Cc2cn[nH]c2)NC(C(CCC)O)=O)=O)CCC(C)=C(F)C1 C1(NC(C(C)(C)N(CC(C)(C)C)C)=O)CC2(CCN(CNC(=O)OC(C)(C)C)C2)CO1 C1(C(N2CC(C#N)C(NC(C3(Br)CCC3)=O)C2)=O)Cc2ccccc2O1 Cc1ccc(F)c(C(N2CCSCC2C(=O)NC2CC(c3ncc[nH]3)C2)=O)n1 N1(C(C2OCC(C)(C)C2)=O)C2CCC1CC(CNC(c1c[nH]c(C(N)=O)c1)=O)C2 c1(OC)c(C(=O)N(C)CC2CCCN(C(C3(Cl)CC3(C)C)=O)C2)nc(O)nc1O C(=O)(C(C)(C)C1=CCSCC1)NCCCCNC(C(n1cnc(C#N)n1)C)=O c1(CNC(=O)CC2(NC(c3cnsn3)=O)CCC2)ncc(C(F)(F)F)s1 C1(C(N)=O)CN(C(=O)C(C2CCCCC2)F)CC1C(N1CC(O)CC1C(N)=O)=O C(=O)(C(C)C(=O)N1CCCC1CN(C)C(c1csc(-c2cnccn2)n1)=O)OC c1(CC(=O)NC(CNC(CCCCOC(C)C)=O)C(C)C)cccc([N+](=O)[O-])c1 N1(C(C(C)N(C(C)=O)C)=O)CC2(C1)CN(C(=O)CNC(c1ccc(C)cc1)=O)C2 Cc1cc(O)cc(C)c1C(=O)NCC1CCN(C(=O)Cc2nc[nH]n2)C1(C)C N1(C(C(C)S(C)(=O)=O)=O)CCC2C(CCCN2C(=O)CCCC(N)=O)C1 C1(CC(N2CCC(OCC)C2)=O)CCN(C(c2c[nH]ccc2=O)=O)CC1 C1(CNC(C2CC(F)C2)=O)CCCN(C(c2cccc(F)c2Cl)=O)CC1 N1(C(CC(C)(C)N(C(C(C(C)C)C2CC2)=O)C)=O)CC(O)CCC1C c1(CNC(C(=O)N(C2CCCOC2)CCCC)=O)noc2c1CCC2 C(=O)(C(C)(C)C1=CCS(=O)(=O)CC1)NC1C(C)CN(C(=O)CC2CCC2)C1 C1(C#N)(C(N(CCC)CC)=O)CCCN(C(c2ccc(OC)cc2)=O)C1 C(=O)(C1=Cc2ccccc2OC1)N1C2CCC(NC(C(N)=O)=O)(CC2)C1 C(CC(=O)NCc1cc(O)ccc1F)(C(F)F)NC(CC(C)F)=O C1(CC)CCCCC1NC(c1c(CNC(=O)C(=Cc2cn[nH]c2)C)cnn1C)=O C(=O)(C1=CCC(C)(C)CC1)NC1CCCN(C(Cc2scc(C)c2)=O)C1 n1(CCCF)nnnc1C(c1cscc1Br)NCCC(F)(F)F C1(NC(C2(C#C)CN(C(c3ccc(C(C)C)o3)=O)C2)=O)CCC12CCCC2 Cn1cc(Br)c(C(=O)NC2CCC(CCNC(=O)Cc3ccoc3)C2)n1 C1(N(C(C(N2CCCCCC2)C)=O)C)CCN(C(=O)Cn2nccn2)CC12CC2 N1(C(c2ccc(C(=O)OC)s2)=O)CCN(C)CC1CNC(=O)C(C)SC C1(C)(C(N2CCC(CCNC(c3cc(COC)no3)=O)CC2)=O)CCC(O)CC1 C1(C(=O)NC(c2nc(C)sc2)C)C2CCN(C(c3cc4n(n3)CCO4)=O)CC12 C1(C(N(CC(CC)C)C)=O)C(O)CCN1C(=O)COCC1CC1 C1(C(C(=O)NC2CC(CNC(c3ccc(SC(F)(F)F)o3)=O)C2)O)CCCCCC1 c1(C(=O)NC2(C)CC(NC(c3cnc(C4CC4)s3)=O)C2)cncc2cccnc12 C1(C(=O)NCC2CCOC2)(CC)CCN(C(=O)CCn2ccnn2)C1 C1(C(=O)N(c2ccncn2)CC2CCCNC2)CCC(F)CC1 Cc1nc(C)c(C(=O)NCc2occc2C(=O)NCC2(O)CCN(C)C2)o1 C(C)(CCCCN=c1[nH]nc(-c2ccccc2)s1)NC(C1C(OC)CCC1)=O N1(C(C2CC2C2CC2)=O)CC2CCN(C(C3(O)CCCC3)=O)CCC2C1 N1(C(C2CCCC2(F)F)=O)CCn2nccc21 CC1CN2CC(O1)C(=O)N1CCC(CC1)OC2=O.C(C#N)(C(N)=O)OC(C)C CC(C)(CNC(=O)CCN1CCC1)CN(C1CCCC1)C1CC1.C1(C(=O)N)COC1 C1(C(N2CCCC(CC)(NC(c3csc(=N)[nH]3)=O)C2)=O)CC2(C1)CC(C)(C)C2 O=C(CS(=O)(=O)c1ccc(C)cc1)NC1CCCC(CN=c2[nH]cncc2Cl)C1 N1(C(c2ccc(COC)o2)=O)CCCC(CN(C(=O)CCC(=O)OC)C)C1 C(CC1CC1)(C(=O)NC1CC(NC(=O)CCC2CCCN2C)C1)OC N1(C(C(c2cc(C)sc2)(C)C)=O)CC2CC1CN2C(=O)OC(C)(C)C CCCC(C)(C)CC(=O)N1CCCC1Cn1cc(CC2CCCCO2)nn1 C(=O)(C=C1SCC(=O)N1C)NCC1CCCN(C(C2CC(C(=O)OC)C2)=O)C1 N1(C(CC(CC(=O)OC)C)=O)CCC2(C=C(C(=O)NOCCC(F)F)C2)C1 C1(NC(C2N(C(C)=O)CC(O)C2)=O)CN(C(c2[nH]nnc2C)=O)CC1C1CC1 C1(CN(CC=C)C)CCN(N2CCCC2Cc2ccccc2)CC1 c1(C(=O)NCC2C(CNC(CCOCC#C)=O)C2)ncc(C(N)=O)cc1Cl c1(C(=O)OC)cnc2nc(NC(c3cccc(O)c3OC)=O)ccc2c1 c1(C(N(C)CC2CN(C(c3cnncc3O)=O)C2)=O)nc(O)[nH]c(=O)n1 C(=O)(C1CCNc2ccc(OC)cc21)N1CCC(n2c(CC)ncc2)CC1 C1(NC(CCCc2nc(C)sc2)=O)CN(C(=O)CC2CCCC(=O)N2)CC1C C=CCCCC(=O)N1CCCC(N(C(=O)Cc2csc(C(=O)OC)c2)C)C1 c1(C(=O)NCCCC2N(C(c3cnn(CC)n3)=O)CCCC2)cccc(C)c1C c1(C(N2CCC(CNC(Cc3cc(C)no3)=O)C(O)C2)=O)ccc2nccn2n1 c1(C(C(N2CCC(NC(=O)C=CCCC=C(C)C)C2)=O)=O)ccc(F)cc1 CC1OC2(C(=O)NCCCC(C)NC(=O)COCC(C)(C)C)CC1C2 C1(C(=O)Nc2ccc(N3CCNC3=O)cc2)CCc2nccn2CC1 N1(C(CNS(C)(=O)=O)=O)Cc2ccccc2OC2(C1)CN(C(=O)CNC(N)=O)C2 N1(C(CS(CC)(=O)=O)=O)CC(N=c2[nH]c(Cl)ncc2C2CC2)C1 c1(C(C)C(=O)NC2(CNC(=O)CCS(C)(=O)=O)CC2)cc2ccccc2s1 C(=O)(CC1=CCCCC1)NC1C(C)CCN(C(c2c(C)oc(C)c2Br)=O)C1 N1(C(c2c(OC)cc(C)cn2)=O)CC2CCC(NC(=O)C(C)(C)C(=O)NC)C2C1 C(=O)(C1=NN(CC)C(=O)CC1)NC1C2CN(C(C(C=C)C)=O)CC21 C1(CCC(C)C)(C(=O)OC)CCCN1C(=O)NC1(C#N)COC1 C12(C(=O)NCCC(C)NC(C3(CC#C)CC3)=O)C3CCC(CC13)C2(F)F c1(C(N2CC(SC)C(n3cc(CCC4CCC4)nn3)C2)=O)cc(C)c(F)cc1Br C(=O)(CCCCO)NC1CCC(N(C(c2ccn(CC(F)(F)F)n2)=O)CC)CC1 C1(NC(C(C)N(CCC)C(c2noc(CC)c2C)=O)=O)CCCCC1(F)F N1(CC(N2CCC3C(C2)CN3C(C2CCC=CCC2)=O)=O)CCCCCCC1=O C(C(C)(C)N(CC(C1(CC(=O)OC)CC1)=O)C)OCC N1(C(Cc2cc(C)no2)=O)CCC(F)(CNC(=O)CC2CCC3CC23)CC1 N1(C(C(CCSC)O)=O)C2CCC(C2)C1CNC(=O)CSc1cccc(Cl)c1 c1(NC(c2nnnn2C(C)C)CCOCC=C)ccsc1C c1(C(=O)NCc2c(CNC(=O)CC(F)F)cccc2)cccc(=S)n1O C1(CC(N)=O)CCC12CCN(CCNC(c1cccc3ccccc13)=O)CC2 C1(C)(C(=O)NCCOC2CN(C(COCCC)=O)C2)CC(C#N)C1 N1(C(c2n(C)cc(I)c2)=O)CCC(NC(=O)C=CC(C)(C)C)C1(C)C N1(CC#N)CCCN(C(c2c(O)cccc2O)=O)CC1 c1(NC(c2ccc(Cl)cc2)=O)ccc(Cl)cc1Cl.c12ncc(s1)NC(=O)N2 C1(CC(C)(C)C)CN(C(=O)COc2ccsn2)CC1NC(C12COCC(C1)C2)=O N1(C(CCC2CCCN(C(c3cnn(C)c(=O)c3)=O)C2)=O)Cc2ccncc2C1 C(=O)(C(C(C)C)C(C)C)Oc1c(OCc2cn(CCOC)nn2)cccc1Cl N1(C(C2CC(C)(NC(C3CC(C)(O)C3)=O)C2)=O)CC(CO)C(O)C1 c1(-c2n(C(CC)C)nc(-c3ccccn3)n2)cc2cnccc2[nH]1 C1(OC)CN(C(=O)C=CC2CCOC2)CCC1NC(c1cccc(OC)c1C)=O C(c1nc2ccccc2[nH]1)=CC(=O)NC1C(C(C)C)N(C(c2csnn2)=O)CC1 c1(CNC(C(C)=C2CCCC2)=O)ccc(C(=O)NCc2ccco2)cc1 c1(C(N2CC(CNC(c3csnn3)=O)C(O)C2)=O)cc(F)cc2cnccc12 C1(N(C(=O)NC(C)C(C)n2cccn2)C)CCC(C)(C)C1 N1(C(C(CC=C)CC)=O)CCCC(C)(C)C1CNC(c1ccc(F)o1)=O c1(C(=O)NCCOCCCNC(C=CCC)=O)ccccc1Sc1ccccc1 c1(NCCOCC)ncc(C)cc1S(=O)(=O)NCc1cc(F)ccc1C c1(C(=O)NCC(C)(C)NC(C(C(C)C)c2cnc(C)s2)=O)nccn2nccc12 C1(C(=O)NCc2ccc(C)o2)CC=CCN1C(=O)CCc1ccccc1 CCCC(C(=O)OC)C(=O)NCC1CC(F)CN1C(=O)CC1CCC(=O)NC1=O C#CCCC(C(=O)NC1CC(=O)N(C)C1=O)NC(=O)CC1CCCCCC1 C(C1CCOCC1)=CC(=O)N(C(C(=O)N(C1CCN(CC)C1)C)C)C1CC1 CCC(COC)C(=O)N1CC(NC(c2sc(Cl)cc2Cl)=O)CC1C CCC(C(=O)NCc1ccc(C(F)(F)C(F)(F)F)s1)C(C)O C(=O)(C1Cc2ccc(F)cc21)N1CC(CCNC(C2CCCC(O)C2)=O)C1 CC1CCC(NC(=O)CCCc2cncs2)CN1C(c1ccc(Cl)c(F)c1)=O C1(C(=O)NC(CC)CNC(C2CCC(C)(C)CO2)=O)CCC2(CCCC2)CC1 C(C(C(=O)N(C(C)CNC(c1cc(C2CCCCC2)[nH]n1)=O)C)OC)OC C(=O)(C(C)(C)CC(F)F)NC(C1CCC(C2CC(C)(c3ccccc3)C2)CC1)=O C1(C(C(=O)NCCC#N)N(CCOC)C(C)C2CC2)CCC(C)C1 N1(C(C(CC=C)(C)C)=O)Cc2occ(C(N3CC(=O)NC(CC)C3)=O)c2C1 c1(N(C)C=O)ccccc1Cl.c1(C2C(=O)N2)ccc(OCC#N)cc1.C1(NC)CC1 c1(C(N2C(C3CCCN(C(CC)=O)C3)CCC2)=O)sc(OC2CC2)nc1C N1(C(Cc2c(C)non2)=O)CCC2(CCCN(C(=O)CCC3CC3C)C2)CC1 C1(C(N2CCC(CCOC)(C(=O)OC)C2)C(=O)NC)CCCOCC1 c1(OC)c(C(=O)N(CCNC(=O)CN(C)CCO)C(C)C)cc(F)cc1F c1(NC(=O)NC2C(C)(C)CC2)nc2ccc(F)cc2s1 c1(OC)ccnc(O)c1C(=O)NC1CCC(N(C)C(c2nccn2C)=O)C1 C1(NC(c2c(OC)ccs2)=O)CCCCN(C(=O)C(c2ccc(F)cc2F)O)C1 c1(N2CCC(C)C(NC(c3n(C=C)ncc3)=O)C2C)nn2cc(C)nc2s1 c1(CN2C(c3c(C)ccc(OC)c3)CC2)cc([N+](=O)[O-])ccc1OCC(=O)O C1(NC(C2ON=C(CC)C2)=O)CCN(C(c2cnc(C3CC3)nc2O)=O)CC1C C1(C(=O)NC(C)Cc2nn[nH]n2)CC(O)CN1C(c1cnn(C2CC2)c1)=O N1(C(C(COC)O)=O)CCCC(O)(CN(C)C(c2cc(SC)n(C)n2)=O)C1 c1(C(=O)NCC2(O)CCCN(C(c3ccccn3)=O)C2)cc2cc(F)ccc2o1 C1(C2CCOCC2)(C(=O)NC2(C)CCN(C(=O)C(C)(C)CF)CC2)CC1(F)F CC1CCC(C(=O)NCC(CC)NC(C2CCCCN2S(C)(=O)=O)=O)CC1C c1(NC(C(=O)N(CCC)CCNC(c2csc(C)n2)=O)=O)ccc(C)c(C)c1 N1(C(C2C(C)C2)=O)CCCC2(CCCN2C(=O)C(c2ccc(Cl)cc2)O)C1 N1(C(C)C(N)=O)CCC(C)(NC(=O)CC2C=CCC2)C1 N1(C(CC2CN(C(C3C(C(=O)OC)C3)=O)C2)=O)CCc2c(O)noc2C1 C(=O)(C1=CC2(CCN(C(=O)C(COC)COC)C2)C1)N(CCCCO)CC N1(Cc2cccc(CCF)c2)CCC(C2(C3CCCN3)CC2)CC1 N1(C(C(C)OCC)=O)CCN(C(=O)CC2(OC)CCC2)C2CCCC12 CC(CNCc1cn(-c2ccccc2)nc1C(C)(C)C)S(N)(=O)=O c1(CC(=O)NCC(CNC(CN(c2ccccc2)C)=O)O)ccccc1CO c1(C(N2CC(CC=C)(NC(=O)Cc3cnns3)C2)=O)cc(N)cnc1C c1(CCC(=O)NC(CNC(C2CCC(COC)C2)=O)(C)C2CC2)cnn(C)c1C C1(C(=O)NC(C)CCN(C)C)(CNC(c2cc(COC)no2)=O)CC(C)(C)C1 c1(N2CCC(N(C)C(c3ccc([N+](=O)[O-])s3)=O)C2)nc(Cl)nc2nc(Cl)n(C)c12 C(=O)(CC(O)CCCC)NC(C(N1CC2(CC(=C)C2)C1)=O)CCC N1(C(c2cc(C)ncc2C)=O)CC(F)(F)CC1(C)CNC(=O)CCC1CC1(C)C C1(F)(CNC(C(Br)=C(C)C)=O)CC(NC(=O)CCc2ccccn2)C1 C1(N(C(c2cn(C(C)C)nn2)=O)C)CC1C1CC1C.c12cc(co1)CNC2=O c1(CC)ccc(F)c(C(=O)NC2CCCC(NC(C3CCC4CCC3O4)=O)C2)c1 N1(C(C(C(C)C)SC)=O)CCCN(C(c2ccc(C(C)=O)c(F)c2)=O)CCC1 c1(C(c2nnnn2C(C)(C)C)NC(c2csnn2)C)cccc2ccsc12 c1(C(=O)NC)c[nH][nH]c1=NC(=O)Nc1cc(C)c(-c2ccc(OC)nc2C)cn1 C1(C(c2nnnn2C2CCOC2)NCc2nc(C)c(C)o2)(OC)CCCCCC1 C1(C(=O)NOC2CC=CC2)C(C2CC2)CCN1C(=O)COC1CCCC1 C1(C(=O)NCC2OCCN(C(c3c(COC)cco3)=O)C2)CCCCC1(F)F C1(OC(C)=O)CCC(C(N2CCC2CNC(=O)COc2cccnc2)=O)C1 c1(C(N2CCCC(CCC#C)C2)C(=O)NCC(F)F)nc2ccccc2nc1C c1(C(N2C(C3(O)CN(C(CC(C)C4CC4)=O)C3)CCC2)=O)cc(Br)n(C)c1 C1(CNC(C2CC3CCC2C3)=O)CCCN(C(c2ccc(C(O)CF)cc2)=O)C1 c1(C(N2CC(NC(c3c(C)ccnc3)=O)C(CO)CC2)=O)cc(C)c(Cl)c(C)c1 c1(C(N2CC(CNC(C3C(CC)CCC3)=O)C2)=O)c(C)nc2sc(C)cn12 C1(NC(C2CC2F)=O)CCN(C(c2cccnc2C2CC2)=O)CC1F c1(CC)cc(N)ccc1C(=O)NC1CC(NC(=O)Cc2cn(C)nn2)C1 N1(C(CCCCCN(C(=O)CCN(C)CCO)C)=O)CCC2(CNC(=O)N2)C1 C1(CN(CCNC2CC2)CC)Cc2ccccc2O1 N1(C(C(Cn2cncn2)NC(c2cccc(C)c2)=O)=O)Cc2cccc(C)c2C1 Cc1nc2ccccc2nc1NC(=O)N(C(c1ccc(F)c(Cl)c1)CO)C C(CC(C)(C)C)(C(=O)NCCn1cc(C#N)cn1)NC(C(CCC)=CCC)=O C12(NC(C(CC)C#N)=O)CC3CC(C1)CC(NC(=O)CCC(C)S(C)(=O)=O)(C3)C2 C1(CC(C)NC(=O)CCOCCN(C)C)CN(C(C2(C)CSC2)=O)C1 Cc1[nH]c(C#N)cc1C(=O)NCC1C2CN(C(c3ccsc3Br)=O)CC12 N1(C(C2N(C(COC(C)(C)C)=O)CCCCC2)=O)CC(CO)C(C2CC2)C1 Cc1cc(=NC(=O)C2CC3(CC(NCc4cc(Br)c(O)cc4O)C3)C2)[nH][nH]1 Cc1cccc2c(C(=O)NCC(C3CCC3)NC(=O)C#CC(C)(C)C)cccc12 N1(C(C2CCC(CC)C2)=O)CCC(CN(C)C(C2(CO)CC2)=O)CC1 c1(C(=O)NCCCC2CCCN2C(=O)CSCc2cscn2)ncc[nH]c1=O N1(C(c2nc(CC)oc2)=O)CCN(C(=O)COC2CCC(C)CC2)C2CC12 CC(C(=O)NCCCN(CCO)C(c1cc(Br)ccn1)=O)C(C)(F)F Cc1cc(C)n2nc(C(N3CCC(CNC(=O)COC(F)F)C34CC4)=O)nc2n1 N1(C(C2C(COC)C2)=O)CCCN(C(=O)CC2CCS(=O)(=O)CC2)CC1 c1(N(C)Cc2c(C)cco2)nc2c(c(=NC(C)C3CC3)[nH]1)SCC2 C(=O)(C(CCS(C)=O)N(C)C)NC(CNC(c1c(C)nc(C)[nH]1)=O)C(C)C C(=O)(CC(C)CC(C)C)NCC(C1CCC1)NC(c1c(C)cno1)=O C1(N(C(=O)C=CCO)C)CC12CCC(NC(=O)CN1CCN(C3CC3)C1=O)CC2 c1(CC(N2CCC(N(C(=O)C(F)(F)c3nccn3C)C)C2)=O)ccc(O)c(F)c1 C1(OC)C(N=c2[nH]c(=N)[nH]c(=NCc3ccc(OCC(C)C)cc3)[nH]2)CC1(C)C CCCCC(CC(=O)NCCCCCF)NC(c1ncccc1F)=O c1(NCCN(CCC)C)ncccc1C(=O)CN1CCCC1=O c1(C(=O)Nc2scc(-c3cccc(CNC(C)=O)c3)n2)cc(I)ccc1Cl N1(C(C=CC)=O)CC(C(N2CCCC3(CCC3)C2)=O)CC(C)(C)C1 N1(C(C2C(C(=O)OC)C2)=O)CCN(C(=O)CCC2CCCCO2)CC1C C(=O)(CCCC(=O)OC(C#N)C1CC1)OC(C)(C)C c1(C(=O)NCC(C)CNC(c2ccncc2N=[N+]=[N-])=O)nc2n(c1Cl)CCCC2 c1(NC(C2CC(=C)CN2C(c2ccno2)=O)=O)cc2[nH]ncc2cc1OC C1(OC)CCC2(C(=O)NCC3CCCN3C(C3CCCCC3OC)=O)CC12 C1(C(N(CCNC(c2ccsc2Cl)=O)C2CC2)=O)COCCC1c1ccccc1 c1(C(N(C2CCC(NC(=O)Cc3ccccc3O)C2)C)=O)ccc(Cl)c(Cl)c1 c1(C(=O)NCCCC2(NC(C=C(C)C(C)C)=O)CC2)cn(CC2CCCO2)nn1 c1(C(=O)NC(C(=O)O)c2cccs2)ccc(Br)cc1C(F)F C1(NC(c2ccc(C(C)C)s2)=O)CN(C(c2cnc(C(N)=O)s2)=O)CCC1C C=CCC(C)(C)CC(=O)NC1CN(C(=O)C(N2CCCC(C)C2)=O)C2(CCC2)C1 C1(CC#C)(C(=O)N(CC(C)N(C)C(c2ccn(CCC)n2)=O)C)CCOC1 c1(CC2(NCC(=C)Br)CC2c2nnnn2C2CCCCCC2)ccccc1F c1(C(N2C(CC(N3CC(CC)OCC3)=O)CC2)=O)cc(C)cc(O)c1 C1(NC(=O)C(CO)c2ccccc2)CC2CCC(C1)N2C(=O)CN1CCCC1 C1(C(=O)Nc2ccc(OCC3CC3)cc2)C2Cc3ccccc3C12 C1(CC(=O)NCCCCN(C(=O)C=CC2CC2)C)COCC(C)(C)O1 N1(C(c2cc(C)on2)=O)CC(NC(=O)Cc2c(C)noc2Cl)CC12CCOCC2 c1(CC(=O)NCC#CCNC(c2ccc(C)cc2)=O)cccc(Br)c1Cl CCCC(C)(C)CC(=O)NC1(CC(=O)NCC(c2ccccn2)O)CCC1 N1(C(CC)=O)CCCC(C(=O)NC2C=CCN(C(C3CCCCN3C)=O)C2)C1 C1(CN(C(C2CCC2OC)=O)CC)CCCN(C(=O)C(c2cnn(C)c2)O)C1 c1(C(=O)NC2CCCC2NC(C2CCC2(F)F)=O)cnc2c(F)cccc2c1 C(C(C(=O)NCCCNC(N)=O)NC(c1cc(C)c[nH]1)=O)OCC C1(NC(CCc2onc(C(C)C)n2)=O)CN(C(c2ccns2)=O)C2CC12 CC1CN(C(C2(C)CC2(F)F)=O)CC1CC(=O)NCC12CCCC1C2 c1(C(=O)NC2(CF)CCN(C(CCc3n(C)cnc3)=O)C2)ncnc2c1CCC2 c1(C(=O)Nc2c(C)cc(NC(=O)CCS(N)(=O)=O)cc2)cn2c(n1)CCC(C)C2 Nc1cc(C(=O)NCC2CCC(NC(c3ccc(Cl)cc3Cl)=O)CC2)ncc1F C12(NC(C(F)=C(C)C)=O)CCCC1CN(C(c1cccc(Br)c1C)=O)C2 C(C1=NOC2CCCC12)OC(CC(c1ccccc1)NC(C)=O)=O C(=O)(CCCC(=O)N(C)C)NC(C)CCNC(=O)C(c1cccc(N)c1)O CN1CC(=O)NC(CC(=O)NC2COCCC2NC(=O)C(C)(C)O)C1=O C1(C(=O)NCCOCCC)(OCC)CCCN1C(=O)COC.CCSC c1(C(=O)NCC(C)(C2CC2)NC(C(CC(C)C)OC)=O)ccnc2[nH]cnc12 C1(C(N2CC(C(C)NC(=O)CCn3cncn3)C2)=O)Cc2nncn2C1 C1(C(N(CC(C)NC(=O)CCCC2CCOCC2)CC)=O)CC2CC1CO2 N1(C(=O)NC(CC)CNS(C)(=O)=O)CC2(CCCC2)c2cccc(F)c21 N1(C(C=C(CC)C)=O)CCC(C2(NC(c3ncn4c3CCCC4)=O)CC2)CC1 C1(C(=O)NCC2(C(=O)NC(c3cn(C)cn3)C)CC2)CC2(CSC2)C1 N1(C(C2CCC(=O)C2)=O)CCCCC1CCNC(c1cc(Cl)n[nH]1)=O N#Cc1cc(F)c(F)cc1NC.N12CCN(C(=O)C1)C(=O)CC1CCCN1C2=O Cc1nc(Cl)sc1C(N1CCN(c2noc(C)n2)CC1)C(=O)NCC1CCOC1 C(C(O)C(C)(C)C)N(C(CCCn1cc(-c2cn(CC)nc2)nn1)=O)CC1CC1 CC(C)CC(N)CC(=O)NC(C1CC2CC2C1)C C1(NC(C2CS(=O)(=O)CC23CC3)=O)CCCC12CN(C(c1ccc[n+]([O-])c1)=O)C2 c1(C(=O)NC2CCC(NC(CC(C)C3CCCC3)=O)C2)cn2cc[nH]c(=O)c2n1 N1(C(c2cnc(C(=O)OC)s2)=O)CCN(C(=O)CC(C)C)C2CC12 Cc1cc(F)c(C(=O)NC2CCN(C(C3CCCCN3C)=O)C2)c(F)c1 c1(CC(=O)NCCN(CCC)C(C2CN(C(C)=O)CCO2)=O)nnc(C)n1C C1(N(C(C)C(=O)NCc2ccco2)C)CCCCC1C C1(F)(C(=O)NC(CC)CN(C)C(C2CC(C)(CC)C2)=O)C(C)(C)C1(C)C C1(NC(Cc2c(C)non2)=O)CC(C(=O)Nc2ccc[n+]([O-])c2)C12CCC2 C1(C(=O)NC2CC(C(=O)NC(CC(=O)NC)C)C2)CC2(CCCO2)C1 C12CCCC3(CN(C3)N(C)C1)O2.c1(C(=O)N)cccc(C2(C)CC2)c1.C1(O)(C=O)CC1 c1(C(N2CC(C(N3CC(OCC)C3)=O)C2)=O)cc(NC(C2CCC(C)S2)=O)on1 C1(CC(=O)NC(CC=C)C2CC2)CCN(C(=O)CC2CC3(CCC3)C2)C1(C)C N1(C(C(CC)C)=O)CC2(C1)OC1(C)CC2(NC(=O)C=C2CC3CCC(C2)N3C)C1 c1(C(N(C2CCN(C(C34CCCCC3OCC4)=O)C2)C)=O)ccc(F)c(F)c1F c1(C(=O)NCCC(CC)(CC)NC(=O)C(O)CN(C)C)n[nH]c2c1CSCC2 C1(C2CCOCC2)(C(N(C)CC2CCCSC2)=O)CCNC1 CC1CCCC1CC(=O)NCCOCC(N1CC(C)(O)C1)=O c1(C(N2C(C)CC(NC(=O)CC(c3ccc(Cl)cc3)O)C2)=O)cccc(F)c1N C1(O)(CC(=O)N(C(C)CNC(=O)CC2OCCO2)CC)CCCCC1 N1(C(C2C(C(C)O)C2)=O)CCC2(NC(c3cc(Br)co3)=O)CCCC12 C12(NC(CCCSC)=O)CCC(F)(F)CC1CN(C(C1CCC1C(F)F)=O)C2 C1(C(=O)NCC(CN(C(=O)C(N)=O)C)(C)C)CCN(CCF)CC1 C(c1ccc(Br)cc1)=CC(N1CCN(C(c2cc(OCC)n[nH]2)=O)CC1)=O N1(C(C(CCC)(C)C)=O)CCOC2(CCCN(C(=O)CSCCOC)C2)C1 C1(C(N(CCC(C(C)C)NC(=O)CN2CCNC(=O)C2)C)=O)CN(C)CC(C)O1 Cc1cc(C(=O)NC2COCC2NC(c2conc2C(C)C)=O)ncc1C(F)F C12(CNC(C(CC)N(C)C)=O)CCC(CC1)CN2C(=O)CCNC(=O)CO CC1CCCC1(C(=O)N(CCCN(C)C)C)NC(C1CCCC1O)=O CCC(C)C(C)(c1nnnn1C1CC1)Nc1cnn(CCO)c1C c1(OC)cc(F)c(C(=O)NC(C)C(C)NCc2ccc3c(c2)OCC3)c(Cl)c1 Cc1cc(C(N2CC3CCN(C(=O)CS(C)(=O)=O)CC3C2)=O)ccc1[N+](=O)[O-] CC1(C)CCOC1C(=O)NCC1COCCN1C(=O)CCSc1ccccn1 C12(C(=O)NC3(CNC(=O)CCC4CCCCC4)CCCO3)CC3CC1C2C3O c1(N(C)Cc2c(CC(=O)OCC)cccc2)ccccc1S(=O)(=O)C1CCCC1 CC1CN(C(C2CCCN2C(c2ccc(O)c(F)c2)=O)=O)C(C)CO1 N1(C(C2(C)CC(=C)C2)=O)CCC2CCOCC2C1 c1cc(N2CC3CCC3C2)nc(N2CCC(C3CCCN3)C2)n1 C(=O)(C(O)CCCNC(=O)COc1ccccc1)NC(c1ncc[nH]1)C Cc1ccc(C)c(OCC(=O)NC2C3CC2N(C(=O)Cc2cc(C)nn2C)C3)c1 c1(C(=O)NC2CN(C(C(COC)COC)=O)CC(F)C2)cc(Cl)cc(C)c1OC C1(CCCC)CCCN1C(c1cc(CNC(=O)COC2CCCOC2)no1)=O C#Cc1ncccc1C(=O)NC(c1ccc(N2CCCS2(=O)=O)cc1)C C1(CCC(C)C)CCN(C(c2cnc(N(C)C)nc2)=O)CC1 c1(OC)cccc(C)c1C(=O)NC1CC1NC(=O)Cn1ccc(Br)n1 N1(c2nc(C#N)cc(C)n2)CC23CCCC2(CN(C(c2n[nH]cc2Cl)=O)C3)C1 c1(C(N2CC3CC(NC(CCC(=O)NC)=O)C3C2)=O)c[nH]c2cc(N)ccc12 C(=O)(C1=CC2C=CC(C1)C2)NC1CCC(CC(=O)NC(COC)C)C1 N1(C(N(c2ccc(NC(C)=O)cc2)C)=O)CCc2cc(Cl)ccc2C1C c1(C(C)C(=O)NCCCCCN(C)C(c2cc(C(N)=O)cs2)=O)ccc(Cl)cc1 C1(C(N(C2C(C)(C(C)C)C2)CC2CCCN2)=O)Cc2cc(Cl)ccc2C(=O)O1 Cn1nc2c(c1C(=O)NCCN1CCN(C(C3CCNC3=O)=O)CC1)CCCC2 C1(NC(C=Cc2c(C)ncs2)=O)CCCN(C(=O)CP(C)(C)=O)CC1 C12CN(CCO1)C(=O)C2.n1(CC(c2ccccc2)C)cc(C2(C)CCCO2)nn1 c1(CC)ccnc(C(N2CCC(C(=O)Nc3cccc(Cl)c3)C2C(C)C)=O)c1 N1(C(C=COCC)=O)CCC(NC(c2ccco2)=O)C(F)C1 c1(N2CC3OCC(NCc4cncc(C)n4)C3C2)ncnc(N)c1C#N N1(C(c2scc(OC)c2)=O)CCCC(C(C)NC(c2nnn(C(C)C)c2C)=O)C1 C12(OCC)CCC(C(N3CC(OCCNC(=O)C(O)C(C)C)C3)=O)(CC1)C2 N1(C(CCCN(C(=O)Cc2nccn2C)C)=O)CC2(CCCCCC2)C1 C1(NC(C2(CC)CCN(C(C3CCC4CC34)=O)CC2)=O)CCC2(CCC2)CC1 C1(C(=O)NCc2c(C(N3CC4C(CC)(C4)C3)=O)nco2)CC12CCCCC2 c1(C(N(CC(C)N(C(C2C(CCOC)C2)=O)C)C)=O)ccc(O)nn1 C12(CNC(CCSCC)=O)CC3CC(CC(NC(=O)C=CC4CCOC4)(C3)C1)C2 C1(F)(CNC(C(COC)NC(C)=O)=O)CCCN(C(=O)C2=CCCS2)C1 C1(CC=C)(C(=O)OC)CCCCN1CCC(=O)NC1CCCCCC1.C(C)=O C1(OC)(CNC(=O)C(C)SC)CN(C(c2occc2Cl)=O)C1 Cc1cccc(O)c1C(=O)NC1CCCC(NC(C2(CO)CC(F)(F)C2)=O)C1 C(C(C)(CO)OC)NC(CN(C(=O)CC(C)n1ccnc1)CCC)=O c1(-c2n(-c3cccc(Cl)c3)nc(C3CCCOC3C3CC3)n2)ccc2c(c1)COC2 c1(C(=O)NC2CC3CC(NC(C4CC4F)=O)C3C2)cc2ncccc2o1 C1(NC(=O)CC2CCOC2=O)C2CC1CN(C(=O)Cc1c(F)cccc1Br)C2 c1(C2C(C(=O)NC(C3CN(C(c4cc(O)no4)=O)C3)C)C2)cncn1C CCC(CN(C)C)CC(=O)NCCCCC(C)NC(c1cscc1OC)=O CC1CCN(C(=O)CC2CCCOC2)CCN1C(c1csnc1Br)=O C(C(C)(CC)C(N)=O)NC(C1N(C(COCC(=C)C)=O)CCC1)=O NC1(C(=O)NC(c2ccc(F)cc2)C2CC2)CC12CCC2 Cc1nccc(C(=O)N(CC(C)(C)C(=O)NCCC(O)C2CC2)C)c1N c1(C(N2C(CN(C(=O)C(=O)C(C)(C)C)CC)CCC2)=O)ccc(OC)c(Cl)c1 N1(C(CC2(OC)CN(C(C(C)OCCC=C)=O)C2)=O)CC(CO)C(C2CC2)C1 C1(C)(CCNC(C2C(OC)CC2)=O)CCCN1C(=O)C1CC1 n12c(nnc1CCn1ccnn1)N(C)CCC2.C1(C)CCCC1.CS c1(OC)noc(C)c1C(=O)NCCC1(O)CN(C(c2cncc(O)c2)=O)C1 N1(C(COc2c(C)cc(Cl)cc2)=O)CCC2CCCC12CNC(=O)C1=CCCS1 CC(=O)CCCC(=O)Nc1ccc(NC(C2CCCN2C(=O)OC)=O)c(C)c1 c1(NC(N2C(CC)CC2)=O)ccc(C)nc1 C(CCCC(=O)NCC1CCOC1C(=O)NC1CC(=CCN2CCC2)C1)OC CC1CCN(CC(=O)N(C(C)CN(C)C(c2ccn(CCF)n2)=O)C)CC1 c1(CC)ccncc1NC(=O)C(C1CN(C(C2CC(C)CC(=O)N2)=O)C1)OC N1(C(c2ccc(SC)cc2Cl)=O)CCC2CN(C(C3CCCC(C)O3)=O)CC12 C1(C(=O)NCc2scc(CNC(C(F)OC)=O)n2)CCC(=O)N1C(C)C C(CC(F)F)(C(=O)NCC1CCC(C)C1)N(C(COCCC)=O)C c1(C(=O)NCC(CN(CC(C)(C)C)CC)O)ccc(-c2nn[nH]n2)cc1 c1(C(=O)NC2CCC(CNC(C34CC3C4)=O)C2)cn2cc(Cl)cnc2n1 CCC(C)CCC(=O)N1CCC(Cn2cc(-c3cccc(C(N)=O)c3)nn2)C1 N1(C(CCOCCOCC)=O)CCC2(CCC2)C(NC(=O)C(C)NC(N)=O)C1 c1(OCC)cc(CNC(=O)C(N2CCC(C)(c3cccc(Cl)c3)C2)=O)cc(F)c1 c1(OC)cc(OC)c(C(=O)NC(CNC(=O)C(C)C(C)(C)C)C2CC2)cc1OC c1(C(C(=O)NC)N(CC(C)(C)C)CC)ccc(OC)c(SC)c1 C1(CC)CN(C(C2(C(=O)OCC3CC3)CC2)=O)CCC1NC(=O)Cn1nccn1 c1(CNC2CCCC(C(=O)NC3(C(C)C)CCOCC3)C2)ncc(Cl)nc1Cl C1(CC(=O)NCCC2(C(N(c3cn[nH]c3)CC)=O)CC2)CC(C)(C)CO1 N1(C(C2C(C)CC=CC2)=O)CCCC(O)(CNC(=O)COCC2CCC2)C1 c1(N(C(=O)CC2CC2)CCCN2CCOCC2)cc2nc(F)ccc2o1 N1(C(C2CC(OCC)C2)=O)CCN(C(=O)C2=NOCC2)C(CC2CC2)C1 C1(CC)CCN(C(=O)CS(C)(=O)=O)C1C(=O)NC(C)C(C)n1cccn1 CCC(C)C(O)C(=O)NC1CC(NC(=O)Cc2csc(-c3ccccn3)n2)C1 C1(C(N2C(CNC(C(CC#C)C)=O)CC(F)(F)C2)=O)CC2(C1)CC(C#N)C2 c1(C(=O)NC2CCCC(NC(CCCCC=C)=O)CC2)ccc(F)c(OC)c1F Cc1ccc(-c2ocnc2C(=O)NC(CNC(C2(C)CC2(F)F)=O)C2CC2)s1 C=C(CNC(=O)CC=CC)CCNC(=O)C(O)C1CC1 C1(C(N2C(C=CC(=O)N(C3CC(F)(F)C3)C)CCC2)=O)CC(=O)CC(=O)N1 c1(C(=O)NC2(CF)CCN(C(C(CC)N(C)C)=O)C2)cnn2ccc(C)nc12 c1(C2C(c3cc(-c4ccoc4)[nH]n3)C2)ccc(Br)cc1.C12CC1C(=O)NC2=O Cc1cc(-c2nc(-c3ccccc3F)nn2CCCOc2ccccc2)c(C)o1 N1(C(C(CC2CCCC2)NC(c2cc(C(C)C)no2)=O)=O)CCC2(CSC2)C1 CP(C)(=O)C1CCCCC1C(=O)NC1C2CC1N(C(C1CC1c1ccsc1)=O)C2 N1(C(CC(C)OC)=O)CC2(C1)CN(C(c1nnn3c1COCC3)=O)CC2CO N1(C(c2c(C)nco2)=O)CCC(C)C(CNC(=O)CSc2ccc(F)cc2)C1 c1(C(N2CCC(C=C)C2)C(=O)NCCCSC=CCNCC)cc(C)c(F)cc1Br c1(CC(=O)NCCN(C(C(COCC)C)=O)C(C)C)coc2cc(CC)ccc12 N1(C(COCC#C)=O)CCCC1C1CCCN1C(=O)CCCOC1CC1 S(=O)(=O)(c1c(Cl)nc2sccn12)N1CC(CNC(c2ccn(O)c(=O)c2)=O)C1 c1(C(=O)NC2C3CN(C(C4(COC)CCC4)=O)CC32)cncc(C(=O)OC)c1C S(=O)(=O)(c1ccccc1Br)N1CCC(N2CCN(C(C#CC)=O)CC2)CC1 C(CCCCCC(=O)NC12CCC(CC1NC(C1CCCNC1=O)=O)C2)SC S(=O)(=O)(c1cnc(N2CCC(N(C)C)C2)cc1C)NC(CCC=C)(C)C c1(C(C(=O)NC2C(CNC(C3(OC)CCC3)=O)COC2)(F)F)c(F)cccc1F CC1(C)Cc2ccc(C(N3CCC4(CCCN4C(=O)CS(C)(=O)=O)C3)=O)cc2O1 C1(C(N(C)CC2CCCCN2C(C2CC3(C2)CC3(F)F)=O)=O)COCCC1(F)F N1(C(C(c2n(C)c(Cl)cn2)(F)F)=O)CCC2(CCCC2NC(=O)CC#N)C1 C(=O)(C(C(C)(C)C)N1CCCCC1=O)NC(CNC(c1cc(CC)ncn1)=O)C C1(C(N(C)CCC2CCOC2)=O)CCCCN1C(=O)CCC(=O)N1CCCC1 c1(C(N2CC(CC(N3CC=CC(O)C3)=O)(OC)C2)=O)ccc(Cl)cc1O C1(OC)CN(C(c2sc(-c3ccn(C)n3)nc2C)=O)CC1NC(c1ccoc1)=O N1(C(c2ccc(C3CC3)nc2O)=O)CCC2(CCC2)C(O)C1 c1(C(=O)OC)ccc(CC(N2CCN(C(=O)COC(F)F)C3CC23)=O)cc1C C1(C(N2C(CNC(C34CC(F)(C3)C4)=O)CC(C)(C)C2)=O)CCc2nc[nH]c2C1 C1CCCCC(=O)N2CCCCC2c2cn1nn2.N12CCC(CC1)C2.CCOC c1(C(=O)OCC)cccc2nc(NC(C3(OC)COCC34CCC4)=O)[nH]c12 CCC(C)C(O)C(=O)NCCN1CCC(NC(=O)CCCn2cccn2)CC1 Cc1cc(C(=O)NCC2CC2CNC(=O)CCc2cc(F)ccc2Br)cnc1O c1(C(=O)NCC2(NC(C(C(C)C)OC)=O)CCCCC2C)cncc2ccsc12 c1(C(=O)NCC2C(CNC(C(F)=CC)=O)C2)c(C)ncn(C)c1=O CC1CCN(C)CCN1C(=O)CN1CCC(O)(C(Cl)(Cl)Cl)CC1 CCC(C)C(C(=O)NCC(C)(C)CNC(=O)CC1(O)CCC1)NC(N)=O Cc1cn2cc(C(=O)NCC34CC(CN3C(C3CSCCSC3)=O)C4)nc2s1 N1(C(c2c(C(C)C)nns2)=O)CC2CC(C1)C(CO)C2NC(c1nonc1N)=O N1(C(C2C=CC(NCc3cc(Cl)ccn3)C2)=O)Cc2cncnc2C1 c1(CC(=O)NC(CNC(c2c(CC)ocn2)=O)(C)C)cccc2cccnc12 c1(NC(C)=O)ccc(NC(c2cnnc(O)c2S)=O)c(Cl)c1 N1(C(C(F)=CCC)=O)CCC(NC(=O)COCc2ccccn2)C(CC)C1 c1(C(N2CC(CC)N(C(c3oncc3C)=O)CC2)=O)c(C)ccc(Br)c1F n1(CC)c(SC)nc2ccccc12.c12cn(nn1)CC(=O)NC(C)CCNC2=O CC(C(=O)NC1CCC1CNC(c1cc(C2CCCC2)nn1C)=O)P(C)(C)=O c1(C(N2CCN(C(c3ccnc(Cl)c3)=O)C3CC23)=O)cccc([N+](=O)[O-])c1Cl C=CCCCC(C(=O)NC(C)(C)CCCC)NC(=O)COCCCN=[N+]=[N-] C1(CCC(=O)NCC(N(C)C(C2(C)CC2(F)Cl)=O)C2CC2)CCCCN1C C(CN=c1ccnc(C(C)C)[nH]1)(CC(C)C)NC(C1Cn2c(C)nnc2CC1)=O C1(CCNC(CCNC(C)=O)=O)CN(C(=O)CS(=O)(=O)N(C)C)CCCO1 c1(NCC(C(C)C)C)cc(=NCC(F)CO)[nH]cn1 C1(CNC(C2(CSC)CC2)=O)C=CC(NC(=O)C(C)(C)C2CCCO2)C1 C(CCC(N)=O)(C(=O)N(CCCC)Cc1nccs1)n1cc(C(C=C)(C)O)nn1 C1(C(=O)NCC(C)(CO)c2ccccc2)CCCC2(CCNCC2)O1 C=CCC(CNC(c1ccc(C2CC2)o1)=O)C(=O)N1C(CO)CC1CO C12(NC(CSC)=O)CCC(CN(C(=O)CCc3n[nH]c4c3CCCC4)C1)C2 Cn1ccc2[nH]c(C(=O)NC3(C)CCN(C(=O)C(F)=C4CCC4)C3)cc12 C(=O)(C(C)CC(=O)OC)NCC1(O)CC(C(=O)NCC(C)N(CC)CC)C1 C1(NC(C2CCN(OC)CC2)=O)CS(=O)(=O)CC1N=c1[nH]ncs1 c1(OCC(=O)NCC(CNC(C(C(C)C)OC)=O)F)cccc(S(C)(=O)=O)c1 C(=O)(C1=CC2CCC(C1)C2)N1CC(O)(CCNC(c2cnc(OC)c(C)c2)=O)C1 CC1OCCCC1C(=O)NC12CC(C1)N(C(=O)Cn1ncnn1)C2 c1(C(N2CC(F)(C(=O)Nc3cn(C(C)(C)C)nc3)C2)=O)cccc(Br)c1 C1(CC=C)(NC(c2ccc(SCC)cc2)=O)CCN(C(C2(CC#N)COC2)=O)C1 c1(CC)cc(C(=O)NCC=CCNC(C2(C)CCCC2(F)F)=O)cc(O)n1 C=CCC(CC=C)C(=O)N1CCC(C(C)C(=O)NCc2ccc(Cl)o2)C1 C1(NC(c2ccc(C3CC3)cn2)=O)C2CC1N(C(C1(O)CC(CF)C1)=O)C2 C(=O)(CS(=O)(=O)CC(=O)NCC(CO)NC(=O)CC1C=CS(=O)(=O)C1)OC c1(C(=O)NCCC2C(C)CN(C(C3(CO)CCOCC3)=O)C2)cc(N)cc(O)c1 c1(C(N2CCC(N(C(=O)C=Cc3ncco3)CCC)C2)=O)cccn2cncc12 C1(N(C)C)CN(C(=O)C=CCC(C)(C)NC(=O)CCc2ccc[nH]2)CC1O N1(C(CC(=O)OCC)=O)CC2CC(C(=O)NC3C=CC(C)(C)CC3)C(C2)C1 C(=O)(C(C(C1CC1)OC)N(C(C)COCc1cccnc1)C)NCCOCC C=C=C(C)CC(=O)NCCCC(=O)NCc1cccc(OC)n1 C1(C(=O)NCCN(C(=O)COCCF)C(C)C)CCC1(C)C C=C(C)C(C)(O)C(=O)NCC(C(C)C)NC(c1cncc(N2CCCC2)n1)=O O(NC(=O)C(c1cccnc1)NC(c1ccn(CCF)n1)=O)CC(C)C N(C)(C1CN(C(=O)COC)CCc2ccccc21)C(CC(CC)SC)=O c1(C(=O)NC(CCNC(COCC#C)=O)C)cccc(C2OCCO2)c1 N1(C(C2(SC)CC(=O)C2)=O)CC(C(=O)NC2CC3(C2)CC(O)C3)CC(C)(C)C1 CCC(C#N)C(=O)NC(c1ccccc1)CNC(=O)C(C)(C)OCC(F)(F)F CCN(C(C)c1ccccc1Cl)N(C)C1CCN(c2ccccc2)C1=O CC1(C)C(c2cccc(C(F)(F)F)c2)CCN1CCc1ccccc1I Cc1cc(C2CCC2)ccc1C(=O)NCC(O)CNC(c1cncc(N)c1)=O c1(C(=O)NCC2(CO)CCN(C(C3CC=CCO3)=O)C2)ccn2c1CCCC2 S(=O)(=O)(C1CCC(=O)CC1)N1CCCC(N(c2nc(OC)nc(OC)n2)C)C1 C(=O)(C(C)CC)NC1CC(N(C(CSCCN(CC)CC)=O)C)C1 CS(=O)(=O)c1cc(C(N2CCC(O)C2c2ccc(Br)cc2)=O)cc(N)c1 CCC(C(=O)OC)C(=O)N1CC=CCC1C(N1CC(CO)C1(C)C)=O c12c(C)nn3c1CN(CC3)C(=O)C(=O)N2.C(=O)(C(F)(F)F)NCCOC C1(C(=O)NC2(CC=C)CN(C(C3(c4ccn(C)n4)CC3)=O)C2)C2CCC(=O)C12 c1(OC)ccc(CC(O)C(=O)N2CC(C)(O)C2)cc1.c1(C(=O)NC)cc(O)n(C)n1 C1(CC)(NC(=O)CO)CN(C(c2cncn2C)=O)C1 N(C1CCCc2c[nH]nc21)C(C(C(C)C)NC(=O)CC1(C)CCOCC1)=O CC1CCn2ncc(C(=O)NC3CC(c4ccon4)C3)c2C1 c1(OC)ccc(N)c(C(=O)NC(C)CCNC(=O)COC2CCOC2)c1 C(=O)(C(CO)N(CC(F)(F)F)C)N(C1CC(NC(=O)CN2CCCC2=O)C1)C C(=O)(C(CN=[N+]=[N-])NC(c1occc1C)=O)NCCc1n(CC)cnn1 c1(C(=O)NCC2(F)CCC(NC(C(C)(C)O)=O)C2)cn(CCO)c(=O)nc1O CCCCC(C)NC(C)(CCc1ccco1)c1nnnn1C1CCC1 N1CC(ONC(=O)CC(=CC2CCC2)C)C(C)(C)C1.C(=O)(C(C)(C)CC#N)N c1(CCC)cc(C(=O)NC(Cc2cc[nH]n2)C(=O)NC2CC=CCC2)n[nH]1 c1(C(=O)NC2CC(CCNC(C3CC=CCO3)=O)C2)ccc2nsnc2c1 c1(C(=O)NCCCC(=O)N2CC(OCC(=O)NC)C2)cc(C#N)ccc1N c1(C(C(=O)NC(CCCNC(c2cnc(SC)s2)=O)C)C)c(C)n[nH]c1C c1(CC(=O)NCC23N(C(C4CCC(C)C4)=O)CC(C2)C3)nn(C)c2ccccc12 C1(CNC(CC2CCN(CCC(C)(C)C)C2)=O)CCC2(CCC2)O1 c1(CC(=O)NCC2CN(C(c3csnn3)=O)CCCO2)csc2ccc(Cl)cc12 C1(CC)CCOCCN1C(CCC1CC=CCC1)C(=O)NCC(C)C N1(C(C(=Cc2ccncc2)C)=O)CCC2(C1)CN(C(C1CCCC(CF)C1)=O)C2 c1(C(=O)NC2CC(C(C)C)SCC2)cc(C#N)ccc1Cl c1(OC)ccc(CCC(=O)N(C2CC2)CC2CCCO2)cc1CO C1(CC)(NC(=O)C=CS(C)=O)CCN(C(=O)C(C)(C)CN2CCN(C)CC2)CC1 c1(C(=O)NC(CC)CN(C(=O)CCC2CC2(C)C)C)cccc2c1CCC2 C(=O)(C(F)(F)c1csc(=N)[nH]1)NCC(CN(C)C(C1(N(C)C)CCC1)=O)O O=C(CCCC1CCCC1)NCC1CC1CNC(=O)CNC(N1CCOCC1)=O c1(C(N2CCC(NC(c3cc(C)on3)=O)C(C)(C)C2)=O)cncc2nnn(C)c12 C1(CC)CCC(NC(C2COCCN2C(=O)C=C(C)c2ccco2)=O)CC1 N1(C(CC(C)c2cccnc2)=O)CC=C(CNC(c2cc(O)nc(O)n2)=O)CC1 Cc1[nH]nc2ccc(C(N3CC4(CC4)CC3CNC(=O)C(F)C3CCC3)=O)cc12 c1(C(=O)NCCCC(c2ccccc2)NC(CCC#C)=O)cc(Cl)c(Cl)s1 C1(C(N2CCC(NC(c3cc(C(=O)OC)oc3C)=O)C2)=O)CC2COCC(C1)C2 Cc1ccnc(N(CCCNC(c2cc(O)nn2C)=O)C(C)C)c1[N+](=O)[O-] c1(C(=O)NC(CCCNC(c2n(CC)ncc2)=O)C)nc(O)nc(O)c1N C1(O)(C(=O)NCCCC(C)C)CCCN(C(c2ccc(CC(=O)O)cc2)=O)C1.CN c1(NC(=O)NCCC#C)ccccc1-n1nc(C)cc1C CC1C2CC(C2NC(C2CCN(C)CC2)=O)N1C(=O)C1=CCCOC1 C1(C(C)C)(CO)CCN(C(=O)C(Cc2cn[nH]c2)NC(c2ncncc2Cl)=O)C1 C(CNC(=O)C(C)n1ccnc1)(CNC(=O)CC1(NC(C)=O)CC1)OC c1(CC)nc(C#N)cc(=NC(C)CNC(=O)Cc2ccco2)[nH]1 c1(C(N(CCC(=O)NCCO)CCCO)=O)ccc(=O)oc1 N1(C(CCCOCC)=O)CCCCC12CC(NC(=O)Cc1ccc(CC)cc1)C2 CC1CC2CCC(C1)N2C(=O)CC(C)NC(c1ccc2cc[nH]c2n1)=O C(=O)(C(C)(O)C(F)(F)F)NCc1nc(C)c(C(=O)NC2CCOC(C)C2)o1 C1(C(=O)NCC(CNC(c2ccc(C#C)o2)=O)C)CC2(C1)CC2(F)F CC(C)(C(=O)NC1CNC(=O)OC1)C1=CCN(C(c2cccc(=O)o2)=O)C1 C(=O)(C1=C2CCN=C2NC=C1)N1CCN(C(C(N2C(CC)CCC2)=O)=O)CC1 C1(CC(=O)N(C2(n3cccn3)CC2)CCNC(=O)C2CC2)CCCC1O C1(NC(Cc2cnc(C)s2)=O)C(CNC(=O)C(C)(C)CC#N)CCC12CCC2 C12(N(C)C(c3ccc(OC(F)(F)F)c(Cl)c3)=O)CC(N=[N+]=[N-])(C1)C2 C=CCC(C(=O)N1C(C(N2CC(C#N)C2)=O)CC2CC12)OC c1(C(=O)NCC2N(C(C(C)(C)O)=O)CCC2)ccccc1Sc1ccccc1 C(=O)(C(O)P(C)(C)=O)N(C1CC1)CC1CCN(C(C2N(C)CCC2)=O)CC1 c1(C(=O)NCCC2CC(NC(C3(Cl)CC34CCC4)=O)C2)ncccc1F C1(C(=O)Nc2c(C(=O)OC)csc2)CC(C)CN1Cc1cccc(CO)n1 N1(C(CC(C)n2cccc2)=O)CCC(O)C(N(C)C(C2CCCN2N=O)=O)C1 c1(C(=O)NC(CNC(CCSC)=O)(C)C)cc(C(F)(F)F)ccc1[N+](=O)[O-] C1(CNC(C=C(CC)C)=O)CN(C(c2ccnn2C)=O)CCC1C(F)(F)F C(c1nc2ccccc2[nH]1)=CC(=O)NC(C)CNC(c1cc(C#N)cn1C)=O C(=O)(CC(C)(CN(C)C)C(F)(F)F)N1CC(CNC(CCCC)=O)C(F)(F)CC1 c1(OCC)ccc(C(=O)NCC2CC2N)cc1OC.C(=O)(C(C)(C)F)C1CC1 C1(O)(CCNC(C(CCC)NC(C)=O)=O)CCCN(C(C2CC(=O)N2)=O)C1 C=CCC(C)(C)C(=O)N1CCCC(C(N2CCC(OCC3CC3)CC2)=O)C1 N1(C(CCC2CCN(C(c3nn(C)c(Cl)c3)=O)C2)=O)CC2OCCOC2C1 C(CC1CCCC1)(C(=O)NC1CC1)N(CCNC(=O)COC1CCCOC1)C1CC1 C(=O)(CC1=NNC(=O)C1)NC12C(CN(C(c3c(C)cc(N)cc3)=O)C1)C2 c1(NC(C(c2cn(C)nc2C(=O)O)C)=O)ccc(N2CCCC2)c(F)c1 c1(CN(C)C(=O)NCC(=O)NCC2CC2NC(c2ccc[nH]2)=O)ccco1 N1(C(C(c2ccccc2)C)=O)CC2CC(NC(c3cn4ccnc4s3)=O)C1C2 N1(C(CNC=O)=O)CC2CCC2(C(=O)NC2CC(O)C2)C1 C(=O)(C(C)C(C)C)NCCN(C(=O)COc1ccsc1)CC=C Cc1nc(C)c(C(N2CCC(NC(c3ccnc(N4CCCC4C)c3)=O)C2)=O)[nH]1 CN1CCN(C(c2cc(C3CC3)ns2)=O)C(CNC(C2(CO)CCCO2)=O)C1 C1(NC(Cn2c(C)nc(C)n2)=O)CC(NC(=O)CN(C)C)C12CCOCC2 Cc1[nH]nc2ncc(C(N3CCC(NC(c4csc(Cl)c4Cl)=O)CC3C)=O)cc12 C1(C(C)C)CN(C(=O)COCC(F)(F)F)CCC1NC(C1(CN(C)C)CCC1)=O Cn1cc(C(=O)NCC2(NC(=O)C=C3CCSCC3)CC2)c(-c2ccccn2)n1 c1(C(N2CCSCC2(C)C)C(=O)Nc2c(CC)cccc2)ccc2c(n1)CCC2 CCC(CC(C)C)C(=O)NC(Cc1ccco1)C(N1CC(=O)NC(=O)C1)=O N1(C(CC(CC)O)=O)CCC2(C1)CN(C(c1cc(C)ccc1N)=O)CCO2 N1(C(C2CC3C=CC2C3)=O)CCCC2(C1)CN(c1nccnc1F)CCO2 N1(C(c2nc(CC)sc2N)=O)CCC(C)N(C(=O)CC2CCSCC2)CC1 C1(CNC(c2n(CCC)nnn2)c2ccn(C(F)F)n2)CCC(=O)NC1 c1(C(N2CCN(C(c3c(CC)con3)=O)CC2C(C)C)=O)cc2nnn(C)c2s1 C1(F)(CNC(c2c(C)ccc(C(C)C)c2)=O)CCCN(C(=O)C=C2CC2)CC1 C1(C(N)=O)CCCN(CCC(=O)NCC2(O)CN(C(=O)C(C3CCOCC3)O)C2)C1 c1(CNC(C(CO)NC(C2C3CC(=O)CC32)=O)=O)ccc(F)c(F)c1 N1(C(C2(C)CCCN(C)C2)=O)CCC2(CC(C(=O)NC(CCO)C(C)(C)C)C2)C1 CC(C)C(C)CC(=O)NCC(C)(C)CC1CN(C(C2CCS(=O)(=O)CC2)=O)C1 N#Cc1ccc(N2CCC(C(=O)NCC3CC(NC(C4CCO4)=O)C3)C2=O)cc1 c1(CC(C)NN2CCCC(C3CCCCN3C)C2)ccc(OCC(F)F)cc1 c1(OC)c(C)nc(C2CC2)[nH]c1=NCC1(F)CCN(C(c2ccncn2)=O)CC1 c1(CC(=O)NCCN(C(=O)CC(C)CN(C)C)CC)ccc(F)cc1 C=CCCC(F)(F)C(=O)N1CC(CC(F)C(=O)NC(C2CC(C)(C)C2)CO)C1 C=CCC(C)(C)CC(=O)N1CCN(C(c2c[nH]nc2Br)=O)CC(CO)C1 N1(C(c2c(C)cco2)=O)CCCOC(CNC(c2ncccc2C(F)(F)F)=O)C1 C(=O)(CC1=CCCCC1)NC(C1CN(C(c2snnc2C2CC2)=O)CCO1)C c1(SC)ccccc1C(=O)N(CCCCCNC(=O)C=Cc1sccc1C)C c1(C(N2CC(F)(CNC(c3cn(C)nc3C(F)F)=O)C2)=O)ccc2ccnn2c1 C12(NC(c3[nH]cc(CC)c3)=O)CCCC1CN(C(=O)CSCCN(C)C)C2 C1(CN(C(=O)Cn2cnnc2O)C)CN(C(c2ccc(C3CC3)nn2)=O)CCO1 CC#CCCCC(=O)N1CCCOCCC1.C(CCCO)SC c1(OC)cc(N)c(Cl)cc1C(N1CC(NC(=O)C(C)(C)CF)CC1C)=O Cn1ccc(C(=O)NC2(CNC(c3cn[nH]c3)=O)CCOC2)cc1=O C1(CCC)CN(C(c2c(C)nn(C)c2F)=O)CCN1C(=O)COCC(C)C Cc1cccc2c(C(N3CC4(CC4)CC3CNC(C3CS(=O)(=O)C3)=O)=O)coc12 C(=O)(C(C)C(F)(F)F)NCC1(COC)CCCN1C(=O)CCC=CBr N1(C(C(CC2CCCC2)OC)=O)CCC2CN(C(c3ccns3)=O)CC12 c1(NCC(C)NC(=O)NC2(CC=C)CCC2)nccc(SC)n1 N1(C(c2cnc(COCC)s2)=O)CCN(C(C2CCO2)=O)CC2(CC2)C1 C1(NC(C(C)NC(=O)Cc2cccnc2F)=O)CC2(CCC2)C1O Cc1nc(NCCc2cnc(C)o2)cc(=NCc2nc(=N)[nH][nH]2)[nH]1 c1(CC)ncc(C(=O)N(C(C)CCNC(=O)CCOc2ccncc2)C)[nH]1 C1(C)(COC)CC(NC(c2[nH]cnc2C#N)=O)CN1C(=O)CCOCC(C)C N1(CCNC(C2(CC)CCC2)=O)C2CCC1CN(C(=O)C(C)(C)CC(C)C)C2 C(=O)(CC(C)(C)C(F)(F)F)N1CC(C)C(NC(C2CCCS(=O)(=O)C2)=O)CC1 N1(C(c2ccc(C(C)C)nc2)=O)CC2CCC1C(NC(=O)C(C)CC1CC1)C2 C(CCN=c1nc(O)c2ccccc2[nH]1)N1CCc2c(C(=O)O)ccc(F)c2C1 C#Cc1ccc(C(N2CC(NC(c3coc(CO)c3)=O)CC3(CC3)C2)=O)cc1F c1(C(=O)NC2CC(CCNC(C(C3CCC(=O)N3)C)=O)C2)c[nH]nc1F C1(C(=O)NCC(C)NC(C2(CC)CCC2)=O)CCC(=O)N1Cc1ccccc1F C1(C2CC2)(C(N2C(C#C)CC2)=O)CN(C(C2C3CCCOC23)=O)C1 c1(C(N(C(C)CNC(C2CC2(F)F)=O)CC)=O)cc2cccc(OC)c2[nH]1 N1(C(=O)C2=COCC2)CCC2(CCCCN(C(c3ncccc3C(F)F)=O)C2)C1 CC1CC(n2nc(-c3ccccn3)nc2C2(c3nccs3)CC2)CCO1 C=C1CC(C(=O)NC(c2ccccc2)COC)N(CS(=O)(=O)CC2CC2)C1 S(=O)(=O)(C1CCCCC1)N1CCC(NC(=O)CC(O)c2ccccc2)C(O)C1 c1(CC(=O)N(CC(C)NC(c2cc(C)oc2C)=O)C)ccc(O)c(C)c1 C12(C(N3CCC(COC)C3)=O)CC(CO)(CN1C(=O)C(C)c1cc[nH]n1)C2 c1(OCCOC)cncc(=NC(=O)CC2CC2C(N2CC3CCCC3C2)=O)[nH]1 CCC(CC)C(C(=O)NC1CCC(NC(c2cnoc2CC(C)C)=O)C1)OC c1(C(=O)NCC(C)(CO)NC(CCC2CC(C)C2)=O)cncc(N(C)C)c1 N1(Cc2nc(C(C)(C)C)on2)CCN(CC2CCC(F)(F)C2)CC1 N1(C(CC)=O)CCN(C(C2CCC23CCC3)=O)CC1c1cccc(Cl)c1 C1(C(N2CC3C(NC(c4c(CC)ncnc4)=O)C3C2)=O)CCC2CC(C)CN2C1 C=CCC(CC)C(=O)NC1C=CCCC1C(=O)N(C)CC1CC1 Cc1cccnc1C(C(C)C)NC(N1CCC(N2CCC2)CC1)=O c1(CC(=O)NCC2C(C(=O)NCc3ccc(C)s3)CCC2)ncccc1F c1(CCC(=O)NCC(c2ccccc2)NC(CNC(C)=O)=O)ccc(F)cc1Cl CC(N(C)N1CCC2NC(=O)OC2C1)C1CCOCC1 C1(C(N2CCC(C(C)NC(C3(CCOC)CCC3)=O)C2)=O)CC(O)CN1C(C)=O C1(NC(c2cc(SCC)ncc2)=O)CCC2CC1CN2C(C1COC(=O)C1)=O c1(C(=O)NCC23N(C(C4C(C)C4)=O)C(CC2)CC3)cc2c(nn1)CCCC2 N1(C(c2c(C)nccc2)=O)C2CCC1CN(CC(O)COCc1cccs1)CC2 c1(C(N2C(CC)CN(C(=O)C(F)(F)CO)CC2)=O)cc(C)nc2[nH]cnc12 Cc1ccc(F)c(N)c1C(N1CC2C(NC(=O)Cc3cnc(C4CC4)[nH]3)C2C1)=O N1(C(C)=O)CCC(NC(=O)C(C)(C)O)C1.C123CC(C1)(C2)NC3=O c1(C(=O)NC2(CNC(CC3CC(OCC)C3)=O)CCOCC2)ccc(C#N)cc1 N1(C(Cc2c(C#C)cccc2)=O)CCC2CCN(C(=O)CC(C)(C)OC)CC2C1 C1(CNC(Cc2nnc(C)o2)=O)CN(C(C2CCCC(=O)N2)=O)C2(CCC2)C1 c1(C(=O)NCC2(O)CC(NC(c3c(C#C)c[nH]n3)=O)C2)nc(OC)cc(OC)n1 CC(CC(N)=O)C(=O)N1CCCC(OCCNC(=O)CN2CSCCSC2)C1 CC(C)(C)C#CC(=O)NCC(CC1CC1)C(=O)N(CCO)C1CC1 Cc1nc(C(N2CCN(C(=O)Cc3csc(S)n3)C(CO)C2)=O)ccc1[N+](=O)[O-] C1(NC(C2(C)CC2)=O)CS(=O)(=O)C2CN(C(C3Cc4ccccc4CO3)=O)CC12 C1(NC(C2(CCCC)CCCC2)=O)CN(C(c2cn(C)cc2C)=O)CC12CC2 N1(C(c2cnnc(Cl)c2)=O)CCC2(CCCN(C(C3CCCC3)=O)C2)C1 N1(C(CN2CCN(C(CS(CC)=O)=O)CC2)=O)CCC2CCN(C)CC12 C1(C)(C(=O)NCC=CCSC)CN(C(C2C3CCC(F)C23)=O)C(C)(C)C1 C1(C(=O)Nc2ccccc2)C(C)(C)C1(C)C.CC1C(=O)NCC=CCNC(=O)N1 C12(C(N3C(C(=O)OC)C4CC4C3)=O)CC(CN(C(c3cc(F)ccc3F)=O)C1)C2 N1(C(c2cn(CC=C)nn2)=O)CCC(C)(C)C(NC(=O)CC(C)n2cccn2)C1 Nc1ccc(CCCNC(=O)NCCc2cc(Cl)ccn2)nc1 N1(C(C=C(C)Cl)=O)CC2CCCC(C1)N2C(c1nc(C)sc1Br)=O c1(CNC(=O)NC(c2cccs2)CC)cc2occc2s1 c1(C(=O)NCC(CC)(C)C(=O)NC(c2cccnc2C)C)coc2ccccc12 CC(C(=O)N1CC2CC3CC2C1C3)C(C)C(C)(C)C Cc1noc(C)c1CCC(=O)NC(C)(CNC(=O)C(O)Cc1cnc[nH]1)CO C(=O)(C(CCF)NC(c1ccc(O)nc1)=O)N1CCC(COC(C)=O)C1 N1(CC)C(=O)CCC1CC(N1CC2C(CNC(c3ccco3)=O)C2C1)=O N1(C(C(CCSC)OC)=O)CCC2C(C1)NC(=O)CN2C(c1ccc[n+]([O-])c1)=O S(=O)(=O)(c1cccc(=NCc2cc3c(s2)CCCC3)[nH]1)N(C)CC1(C)CCCO1 c1(C(CNC(=NC)NCCc2cc(C(F)(F)F)co2)O)cccc(C)n1 C1(n2cc(CCC(N)=O)nn2)CC2CCC1(NC(=O)CSCC(=O)O)C2 N1(C(CCc2cnc(C)s2)=O)CCC(NC(C2CCC(C(N)=O)C2)=O)C(O)C1 CC1CC(=O)NCCN1C(C(=O)NC1CC1)c1ccoc1 CC1CCC(N2CCCC2)CN1C(=O)NC(=O)NCC(c1ccc(O)cc1)O c1(N(c2nccc(N3CCC(O)CC3)n2)Cc2ccc(SC)cc2)ccc(C#N)cc1 c1(C(N2CC(NC(C3CC3F)=O)(CO)C2)=O)c(F)ccc(F)c1Br N1(C(c2n(C)ncc2)=O)CC(C(=O)NCc2ncc(C(=O)O)cn2)C(C2CC2)C1 c1(NCCc2ccc(SC)cc2)ccc(S(=O)(=O)N2CCOCC3CC23)cc1Cl c1(OCC(=O)NC2C(CNC(c3cnc(CC)[nH]3)=O)CC2)ccc(Cl)cc1F C#CC1(C(=O)N(C2CCCC2C)C)CCN(C(=O)C(C)C(C)C)C1 CC1CCN(C(=O)CC(C)C(C)(C)C)CCN1C(=O)Cc1cccs1 CC(C)C(C)(CNC(c1cccc(Br)c1)=O)NC(c1ccc(C2CC2)nc1)=O C1(C(=O)NCCN(C(=O)CCCN(C)C)CC)COC(C)C1 C1(CC)(NC(=O)CC2CCC(=O)N2)CCN(C(=O)C(O)Cc2cnc[nH]2)CC1 N1(C(C)=O)CCc2c(C(=O)Nc3cn[nH]c3)n[nH]c2C1 c1(C(N(C2CCN(C(=O)CC3CCOC3=O)C2)C)=O)ncc(Cl)n1C CN1C(=O)CSC1=CC(=O)N(C)CC1CCN(C(=O)COC2CCCOC2)CC1 CCC1=NOC(CC(=O)NCC(c2ccccc2)CNC(C2OCCO2)=O)C1 c1(OC)ccc(CCCCC(=O)NCCCCN(C)C(c2csnn2)=O)cc1 C12(NC(=O)CC3CCCOC3)CCCN(C(c3cc(F)c(F)cc3F)=O)CC1C2 c1(C(=O)NCC(c2cccc(C)c2)N(C(CCCC)=O)CC)scc(C)c1C C1(C(N(CC(C)NC(c2c(Br)cnn2C)=O)C)=O)CC12CCC(C)(C)CC2 C(=O)(C1CCCc2sccc21)N1C2(CN(C(=O)C(C3CC3)C3CC3)C2)CC1 Cc1ccn(C)c1C(N1C(C(=O)NCCCc2ncnn2C)CC1C)=O C1(OC)CC(NC(=O)C(=O)N(C)C)CN(C(=O)C=Cc2ccc(C)o2)C1 Cc1nc2cc(C(=O)NCC3CCCCN(C(C4CC4C#N)=O)C3)ccc2s1 c1(CC)ccc(OCCC(=O)NC(C)(C)CN(C)C(c2csc(C)n2)=O)cc1 c1(C(=O)NCC(CC=C)NC(C2(F)CCCOC2)=O)c[nH]c2c(C#N)cccc12 C1(C(N2CCN(CC=C)CC2)=O)CCC(O)CN1C(c1coc(C)n1)=O CC1(C)NC(=O)OC1CNC(=O)C(C1CCCC1)NC(C1COC(=O)N1)=O CN1CCN(C(=O)C(c2ccccc2F)O)CC1CNC(c1cccnc1Cl)=O N1(C(C2(NC(C3CC(=O)CS3)=O)C(C)(C)C2)=O)CC2(C1)CC2(F)F C1(C(N(CC(C)(C)CCC)C)=O)CCC2(CC2)C1.C(=O)(CCOCC(C)(C)C)OC CS(=O)(=O)CCC(=O)N1CC2C(CNC(=O)C(O)COCc3ccccc3)C2C1 c1(CC)ccc(C(=O)NC(CNC(c2cc(-c3ccncc3)[nH]n2)=O)CC)o1 C1(CNC(C(C2CC2)NC(C(C2CCOC2)OC)=O)=O)CCN(C)CC1 N1(C(Cc2c(C)ncnc2C)=O)CC2CN(C(c3ccnn3C)=O)CC(C1)O2 c1(OCC)noc(C)c1C(=O)NCC1CC(NC(c2csc(C3CC3)n2)=O)C1.OCC c1(OC)nccc(C(=O)N(CC(C)CNC(=O)CC2CCCCN2C)C)n1 c1(S)ccncc1OC.C(=O)(C(CN(C)C)NC(=O)C1CC1)NCCCOC c1(C(N2C(CN(C(CCCC(C)O)=O)C)CCCC2)=O)ccc(S(C)(=O)=O)o1 N1(C(CCNC(c2ccc(Br)o2)=O)=O)CC(NC(C2CC2F)=O)CC2(CC2)C1 C1(N(C)C)CCN(C(C2(C)CCN2C(c2cc(-c3ccncc3)[nH]n2)=O)=O)CC1 C(=O)(C(C)C(C)(F)F)N(C)CC1N(C(C(CC=C)NC(C)=O)=O)CCCC1 C#CC1(C(=O)NCc2n[nH]c(C)c2C)CN(C(C2CCN(C)C2C)=O)C1 C(C(C)CC(=O)NC(c1cccs1)(C)C)NC(c1cc(C)oc1)=O C1(O)(NC(C(C(C)N(C(=O)OC(C)(C)C)CC)C(C)C)=O)CCS(=O)(=O)CC1 C1(C(=O)NCCC2CCN(C)C2=O)CC(O)CCN1C(C1CC(N=[N+]=[N-])C1)=O c1(CC)sc(C(N2CCC(C)(c3cn(-c4ccccc4)nn3)C2)=O)cc1Br Cc1ccc(N2CCCCC2)c(NC23CCC(CC2C(=O)NS(C)(=O)=O)C3)c1 c1(C(N2C(C(=O)Nc3c(C)nc[nH]3)CC(F)C2)=O)ccc(O)cc1Br C(=O)(CCCCSC)NCC1(O)CC(CNC(COCCC)=O)C1 c1(OC)cccc(C(F)(F)C(=O)NCC(C)(C)CNC(C2(NC(N)=O)CC2)=O)c1 C=CC(C)(O)C(=O)NCC1(NC(c2ccnc(OC)c2)=O)CC1 C(=O)(C(C#N)(CC)c1ccccc1)NCC(C1CC1)NC(C1(CCC=C)CC1)=O C12(C(=O)NC(CCN(C(c3c(OC)n[nH]c3)=O)C)C(C)C)CCCC1C2(F)F C(C)(CCCCNC(=O)C(C(C)C)c1ccncc1)NC(c1c(C)con1)=O C1(CNC(C(COC)OC)=O)CC2CCC1N2C(=O)C=C(C)C C1(C(=O)NC(CC)(CNC(=O)COCC2CCCO2)CC)CCc2cncn2C1 c1(C(N(C(CNC(C2N(CCC)CCCC2)=O)C)C)=O)cnc2cnccc2c1 C1(CC)CN(C(=O)COc2ccccc2)CCN1C(=O)C(CCSC)NC(C)=O N1(C(C2OCCN(CC)C2)=O)CCOCC(C(=O)NCCCC(=O)NO)C1 c1(C(CCC(=O)NCC(C)N(C(C2CC(SC)C2)=O)C)=O)csc2ccccc12 N1(C(C(C2CC2)OCC)=O)CCCC(C(=O)Nc2ccc(CO)c(Cl)c2)C1CC Cc1cc(Cl)ncc1CC(=O)NCC1CCC(OC2CCCC2)CC1 CC(C)CC(=O)C(=O)NCCCN(C(c1cccc(F)c1)=O)Cc1ccccc1 C1(C(=O)NCC2(F)CCC2)COC2(C1)CN(C(C1CCC(F)(F)C1)=O)C2 N1(C(C2CCC(CC)O2)=O)CC=CC(NC(=O)Cc2nncs2)C1 c1(OC)cc(C=CC(=O)NC2CCCCN(C(=O)C(C)(C)C(C)C)C2)ccc1F C(=O)(CCS(C)(=O)=O)NCC#CC(=O)NCC(c1ccsc1)C CC1CN(C(C2CN(C)CCN2C(=O)CCc2ccn(C)c2)=O)Cc2nncn21 CC(C)CC(O)C(=O)NC1CCC(F)(CNC(C23CC(F)(C2)C3)=O)C1 N1(C(CCSCCCC)=O)CCN(C(=O)C2=CCOCC2)CC12CC2 Cc1ccc(C(N2CC3CC2CN3C(c2cnnc(O)c2)=O)=O)cc1N c1(CC(N)=O)ccccc1CC(=O)NC1CC(NC(=O)CSC(F)F)C(O)C1 C1(NC(c2n[nH]c(CC)c2Cl)=O)CCC2CCN(C(C3CCCC34CC4)=O)C12 N1(C(C=C(CC)CC)=O)CCCC1C(C)(C)NC(c1ccc(COC)s1)=O C(CS(=O)(=O)CC(=O)NC1CCN(C(c2cc(OC(F)F)n(C)n2)=O)CC1)OC Cc1nnc2n[nH]c(NC(c3cc(N)ccc3[N+](=O)[O-])=O)c2c1C c1(C(N(CCCN(C(COC(CC)C)=O)C)C)=O)c(F)ccc2ccncc12 C1(NC(=O)C=CC2CCC2)CCC12CCN(C(c1ccco1)=O)CC2 C1(CNC(C2C(C)C2C)=O)COCC1NC(=O)C(F)(F)C1(O)CCCC1 Cc1cc(C2CC2)ccc1C(=O)NC(C)CCCNC(C1CCCOC1)=O CC(C)C(C(=O)N(CC(F)(F)Cl)C)C(C)NC(=O)C(C)N=[N+]=[N-] C1(CNC(CC#N)=O)CN(C(c2cc(C(F)F)ccn2)=O)CC12CCOCC2 C1(CC(N2CC(OCCNC(C3(SC)CC(O)C3)=O)C2)=O)OC(C)(C)OC1=O C#CC1(O)CCCN(C(C2CC(C)N2C(=O)COc2ccn(C)n2)=O)C1 c1(C(N2CCN(C)C(c3ccc(F)cc3)C2)=O)ccc2c(c1)C(N)CC2 C1(C(N2CCN(C(C(C(C)C)(C)O)=O)CC2CCO)=O)CCOC2(CCC2)C1 c1(C(=O)NCc2cccc(CN(C(C(CC)F)=O)C)c2)ccc(CO)cc1OC C1(CNC(CCn2ncc(C)c2)=O)CN(C(=O)CCC2CCCO2)CCCO1 Cc1c(C(=O)NC2(CO)CCN(C(C3CS(=O)(=O)C3)=O)C2)cnn1CC(F)F CS(=O)(=O)c1ccc(OC(F)F)cc1F.C1(=O)CC(c2ccc(N)cc2)C(=O)O1 Cc1nc(C(=O)NC2CCN(CCNC(C3CCC3C)=O)CC2)c(C)s1 N1(C(CCNS(C)(=O)=O)=O)CC(CO)C2(C1)CN(C(=O)CC1CCCCCC1)C2 c1(OC)cc(N)c(F)cc1C(N1CCCC(NC(C2CCCC2(F)F)=O)C1)=O O=C(NNc1cc(F)c(F)cc1F)c1cnsn1 C(c1ccc(Cl)c(C(F)(F)F)c1)=CC(=O)NCC(CC)NC(C12CC(C)C1C2)=O C1(CCC(=O)NCCC(C)NC(C2(C3CCCO3)CCC2)=O)CCC(=O)C1 C=CCC(C)(CC=C)NC(=O)C(C(C)O)NC(=O)CCN1CCCC1=O C1(C(=O)NC2C3CN(C(C(C)NC(N)=O)=O)CC2C3)CC2CC(O)CC(C1)C2 c1(C(=O)NCC23CC(CO2)N(C(=O)C2=CCOC2)C3)c[nH]c2ccc(Br)cc12 c1(CC(=O)NCCCN(C(CCC(=O)NC)=O)CC)cc2ccccc2c(=O)o1 C1(NC(C(C)N(CC)CC)=O)CC2CC(C1)CN(C(=O)CCC1CCCCO1)C2 N1(C(C(C2CC2)OCC)=O)CC(NC(=O)CCn2cncn2)C(c2cnn(C)c2)C1 N1(C(C)C)CCOCC1C=NOc1ccc(F)c(F)c1 CC(C)CS(=O)(=O)CC(=O)NCCCN(CCO)C(C1CN2CCN1C(C)C2)=O c1(OC)cc(-n2nc(C3CCCC3)nc2CCCC2CC2C)cc(F)c1F C1(C(=O)NCC2C(CCC)C2)CCOCCN1C(=O)CCn1ccnn1 N1(C(C2(C)CCC2)=O)Cc2cccc(CNC(=O)CCc3cccnc3)c2C1 CCCCC(CO)NC(=O)CC(CC)NC(c1sccc1CO)=O CC1OCCOC1C(=O)NCC1(CO)CCN(C(C2C=CCC2)=O)C1 c1(CC(=O)NCC(C2CC(F)(F)C2)OC)c(Br)cncc1Br CCC(C)CCC(=O)NCCCN(C(=O)C(c1ccccc1Cl)O)CC C(=O)(CCCCN(C)C(C1CCCC1)=O)N(C(C=C)C1CC1)C C12(C(N3CCC(O)(CC)C3)=O)CC(CN(C(c3cn(C(C)C)nn3)=O)C1)C2 N1(C(c2ccn(CC)n2)=O)CCOCC1CC(=O)NCC(C)(O)C1CCCC1 C1(C(=O)NC2CCCC(NC(C3(CC#C)CCC3)=O)C2)CCC(C)(O)CC1 CC(CC(=O)OCC#CC(=O)NOCC=CCl)CC(C)(C)C.C(C)(C)C C1(CNC(C23CC(C)C2C3)=O)CN(C(c2c(O)cccc2Cl)=O)CC1(F)F C(=O)(CCCCCF)NCC1(C(C)NC(c2ccc(OC(C)C)nc2)=O)CC1 c1(CC)ccc(C(N2CCN(C(C3CC3(C)C)=O)CC2COC)=O)c(C)n1 N1(C(C(CSC)C)=O)Cc2nccn2CC(NC(C2(c3cc[nH]n3)CCC2)=O)C1 N1(C(C(SC)SC)=O)C2CCCC1CN(C(c1cc(C#N)c[nH]1)=O)C2 CN1CCN(C(=O)CCc2cnccn2)C(C(=O)NCC2(C3CC3)CCC2)C1 C(C(CC(C)C)NC(C1CCCN1CC)=O)NC(C=CCC)=O N1(C(CC(C)(C)C)=O)CC2(CNC(c3ccc(Cl)cc3)=O)CC1CO2 C(C(C)(C)C(=O)NCC(C(C)(C)C)NC(=O)C(C)CN1CCOCC1)NC(C)=O c1(CC(=O)NCCC(C)NC(c2c(SC)cnn2C)=O)ccc2sccc2c1 C1(C)(CNC(C(C)(C)OCCC)=O)CCN(C(C2CC2C2CC2)=O)C1 c1(C(=O)NC2CCCCC2NC(c2cccnc2O)=O)cc2c(nn1)OCCS2 c1(C(N(CCC)Cc2nc(-c3ncccc3C)no2)=O)cc2cc(O)ccc2[nH]1 N1(C(CN(C)C)=O)CCN(C(=O)Cn2ccnn2)CC2CCCCC12 C(=O)(CC1OCc2ccccc21)N(CC(C)NC(c1ccccc1O)=O)CC N1(C(c2cnc(C)s2)=O)CCC(NC(C2(F)CCS(=O)(=O)C2)=O)CC1C c1(C(=O)NC2(CNC(C(COC)(C)OC)=O)CC2)cccc2[nH]c(C)cc12 c1(C(=O)NCC(CNC(C)=O)F)cccn(CC(=O)OC(C)(C)C)c1=O c1(C(=O)NC(C)CN(C)C(c2ccn3c2CSCC3)=O)cc2nn[nH]c2cc1F N(C1CCCc2c1cnn2CCO)C(C1CCC(N)C1)C(=O)OC Cn1[nH]c(=NC(=O)C2CC(F)CN(Cc3cc(Cl)cnc3Cl)C2)cc1Cl CCCC(CNC(=O)CC1CCC(=O)N1)C(=O)N1CCCC1(CO)CO c1(NCc2cncc(OC)c2)cnc(F)cc1C(=O)Nc1c(C)cccc1Br C(=O)(C1CCc2ccccc21)N1CC(NC(CCc2c(C)noc2Cl)=O)(CO)C1 C1(CNC(CC(CC)SC)=O)C(OC)C(OC)CN1C(=O)CP(C)(C)=O c1(C(N2CC(NC(CCC(C)SC)=O)C(SC)C2)=O)cc2ccc(F)cc2o1 N1(C(C(C(C)C)O)=O)CC(C(N2CC(O)CC2(C)C)=O)CC(F)(F)C1 c1(C(N2CC(CN(C(C=CC(CC)C)=O)C)OCC2)=O)cn2cccc(F)c2n1 N1(C(c2c(CC)n(C)nc2)=O)CCN(C(=O)C=Cc2ccn(C)c2)C2CC12 c1(C(=O)NC2C(CNC(C3C(=C)CC3)=O)CCCC2)[nH]c2ccccc2c1C#N Cc1ccc(N)c(C(=O)NCC23CC(NC(=O)CCC4CCC4)(C2)C(C)O3)c1F c1(C(N2CCC(OC)(CNC(=O)C=C3CCOCC3)C2)=O)cnc2ncccn12 CN1CCN2CC1C(=O)Nc1c(ccs1)C2=O.C(=O)(C(=O)N(C)C)NC1CC1 C(C(C)(C(=O)N1CCCC1C(=O)NC1CC(C(C)O)C1)OC)OC C1(NC(C2=CCN(C)C2)=O)CCCCCN(C(c2ccc(O)nn2)=O)C1 C(C(=O)NC1CCN(CCNC(=O)CN2CCC(C)CC2)CC1)(C(C)(C)C)SC c1(NC(N2C(CCC(C)C)CCCC2)=O)ccc(F)c(S(N)(=O)=O)c1 N1(C(c2cnc(OC)s2)=O)CCOC(CNC(=O)CC2CC3CCC2C3)C1 CC(CC(C)(C)C)C(=O)NCCCN(C(=O)Cc1ncn2c1COCC2)C C1(S(N)(=O)=O)(C(=O)NC(CCN(C(c2cc(C)oc2C)=O)C)C(C)C)CCCC1 c1(CC(=O)N(CCN(CC)CC)CC)cc(OC)no1.C(C(C)C=O)SC c1(OC)cccc(CC(=O)NCC2(F)CC(NC(=O)C=C(C)C)C2)c1Cl C1(NC(=O)Cn2cnc(Br)n2)CCN(C(=O)CCn2cncn2)CC1O c1(C(N2C3C(NC(C#CC(C)(C)C)=O)CC(C3)C2)=O)cc2n(n1)CCNC2=O c1(CC(N2CC(C)C(NC(C3(C(F)(F)F)CC3)=O)C2)=O)cccc(C#N)c1 c1(C(N2CCC(n3cc(CNC(C4(O)CC4)=O)nn3)C2)=O)cc(Br)no1 N1(C(c2cc(OC)ns2)=O)CC(C2CCCCN(C(c3csnn3)=O)C2)C1 N1(c2ccnc(C(C)C)n2)CCC(NC(c2[nH]nc([N+](=O)[O-])c2Cl)=O)C(C)(C)C1 Cc1nc(C(=O)NC2CCCN(C(=O)C(C)(C)CN(C)C)CC2)c2ccccn12 N1(CCNC(C(c2cnn(C)c2)NC(c2c(C)non2)=O)=O)CCOCC1=O C=CCCC(c1nnnn1C(C)C(=O)OC)(C1CC1)NCc1ccccc1Cl Cc1nc(N2CCC(NC(=O)CC3CCCC(C)C3)C2)ncc1Br CC1(CNC(c2ccc(C3CC3)cc2)c2nnnn2CC2CC2)CC2CCC1O2 C1(NC(C2C(OCC)C2)=O)CCCCC1CNC(c1cc(C(C)(C)C)nn1C)=O c1(NCCC2N(C(c3cnccn3)=O)CCCC2)nc(Cl)nc2[nH]c(O)nc12 c1(C(N(C(C)C)CCNC(c2sccc2C(F)F)=O)=O)cccc2c1COCC2 CC(CC(=O)N1CCOC2(CCC2)C1)C(C)(C)NC(=O)CC1CNC(=O)O1 C1(NC(C2(CC=C)CC2)=O)CN(C(C2CCC2(C)C)=O)C2CCCCC12 Cc1cc(C)c2cc(-c3nc(C(C)C)nn3CCc3ccncc3)[nH]c2c1 N(C)(C1CN(C(c2cc(C)n(C)c2)=O)CCc2ccccc21)C(CC=CC=C)=O C1(C(=O)OC)CN(C(=O)NCCCC2CC2(C)C)c2ccccc2O1 c1(C(N2CCC(NC(c3cncc(Cl)c3)=O)(CO)C2)=O)cnc2ccccc2n1 C1(C(N(CC(C)NC(=O)C(=O)N=S(C)(C)=O)C)=O)CCCC1S(C)(=O)=O CC(Cc1cccs1)CN=c1nc(N2CCC(F)(CN(C)C)C2)c2c([nH]1)CCOC2 N1(C(C(C(C)O)C)=O)CC2CN(C(c3csc(Cl)c3)=O)CC(C1)O2 N1(C(C(C(=O)OC)OC)=O)CC2CN(C(C34CCC3CC4)=O)CC2C1 Cn1nnnc1C(C1CCN(S(C)(=O)=O)C1)NS(=O)(=O)CC1COC1 N1(C(C(CCSC)OC)=O)CCC(CCC(=O)O)C(C)C1 Cc1ccc(CNC(C23CC2CN(S(=O)(=O)CC#N)C3)=O)c(I)c1 CCCCC(CNC(c1coc(C(N)=O)c1)=O)NC(=O)Cc1cnc(C)s1 c1(C(=O)NCC(C)N(C(CCCN(C(C)=O)C)=O)C)cc(C)cc(O)c1 C1(CN(C)CCF)CNCCOC1 Cc1cncc(C(N2CCOC(CCNC(=O)Cc3ccc(C)s3)C2)=O)n1 c1(NC(C2(CC)CCC2)=O)cncc(-n2cccn2)n1 c1(N2CCN(C(C3(CC(C)=O)CCC3)=O)CC2)nccn2cnnc12 C(=O)(CCC1=NNC(=O)CC1)N1C(CNC(C2(CO)CCC2)=O)CCC(C)(C)C1 c1(C(N2C3C(NC(c4nc(C)oc4)=O)CC(C3)C2)=O)c(F)ccc(Br)c1F CC(C)(O)CC(=O)NC1COCC1NC(C1(c2ccnc(Cl)c2)CC1)=O N1(C(c2cc(C)sn2)=O)C2CCC1CC(C(N1CCC3(CCCO3)C1)=O)C2 C1(C(=O)NC2CC(C(C)N(C(=O)Cc3cnoc3)CCO)C2)CCCOCC1 N1(C(C2CC(n3cc(CN)nn3)C2)=O)CC(O)CC1CNC=O.CCO C#CCC(C)(C(=O)N1CCC(O)C(CO)C1)NC(C1C=CCC1)=O C=CC1(CC(=O)NCC(C)OC(F)F)CN(C(c2coc(C(F)F)c2)=O)C1 c1(-n2cc(CCCC(=O)NC(CC(CC)C)C(=O)O)nn2)c(F)c(F)cc(F)c1F c1(NC(C2N(C(C3N(C(C)=O)CCCC3)=O)CC2)=O)cc(Br)c(F)cc1Cl c1(C(N2CC(F)CC(C(=O)O)C2)=O)ccc2c(Cl)ccnc2c1.C1(CN)(C)CCC1 N1(C(Cc2nc(C)sc2C)=O)CC2CC(NC(C3CCCC34CCC4)=O)C2C1 c1(N2CC(NC(c3c(C)coc3C)=O)C(O)C2)ncc2c(Cl)cccc2n1 C=CCC(C(=O)N(CCC)CCNC(=O)C1=CCCS1)C(C)C c1(CCC(=O)NC(C(C)NC(=O)CCF)C)cnn(-c2ccccc2)c1 c1(CN2CC3(C(C(N4CC(=O)NC4)=O)C3)C2)cc(Cl)cnc1Cl n1(C(C(=O)NCC2(F)CC(NC(CCC)=O)C2)C)nc(C)c([N+](=O)[O-])c1C C1(C(=O)NCc2ccc(C(=O)OC)[nH]2)CC12CCN(C(c1ccc(Cl)cc1Br)=O)C2 C(c1cnc(C)nc1O)=CC(=O)NC1CC(CNC(c2oc(CC)c(C)c2)=O)C1 c1(C(N2CC(CNC(=O)C3=COCC3)C3(C2)CC3)=O)ccnc2ccccc12 c1(NC(=O)NCC(C)C(=O)O)nnc2ccc(COc3ccc(Cl)cc3)cn12 CCC(C)(COC)CN=c1[nH]c(=NCc2nc(C(N)=O)cs2)c2ccccc2[nH]1 N1(C(c2scc(C)c2)=O)CCN(C(c2ccc(C)o2)=O)CC1C#N c1(C(C)C(=O)NCCN(C)C(c2ccnn2CC2CC2)=O)cc(F)cc(F)c1 c1(C(=O)NC2CCOCC2NC(C2CSCCS2)=O)ccc2nn[nH]c2c1 CC1CN(C(C2(C(N)=O)CCC2)=O)CCC1NC(C1CN(S(=O)(=O)C(F)F)C1)=O Cn1c(-c2nc(CCCOC3CC3)nn2CCC(C)(C)C)cc2ccsc12 Cc1ncc(C(N2CC(Cn3cc(C4CCC5(CCC5)C4)nn3)C2)=O)c(O)n1 Cc1cc(NCC2CCCN(C(c3conc3C)=O)CC2)n2ncnc2n1 C1(C(=O)NC(CC)C(=O)Nc2ccc(Cl)cc2)CC2(C1)C(C(=O)O)C21CCC1 CCCC(O)C(=O)NCC(CC)NC(=O)CC1(C(F)F)CC1 N1(C(C(C)=C2CC2)=O)CC(CNC(c2ocnc2-c2ccccc2)=O)CCC1C c1(Cc2nc(=NCC3C(NC(C4CC(C)(F)C4)=O)CCC3)s[nH]2)ccc(Cl)cc1 N1(C(CCN2CC3C(C)(C)C3C2)=O)CCC2(CC1)CC(CO)C2 CC1(C)CCC(C(=O)NC2CC(C(F)F)(NC(c3ccc(O)cc3)=O)C2)CC1 N1(C(c2cc(COC)[nH]n2)=O)CC(O)CC1C(=O)NCCNC(=O)OC CC1(C)CCC(C(=O)NC2CCCC2CF)(NC(=O)COC2CCC2)C1 N1(C(c2c(C)scc2)=O)CCC(C)N(C(C23COC(CO)(C2)C3)=O)CC1 c1(C(=O)NCC(CC)NC(=O)C(N2CCCCCC2)C)cnc2n1CCCCC2 CC(C)C(C#N)C(=O)NC1CC(C)(C(N2CCCC(CN=[N+]=[N-])C2)=O)C1 Cc1cc(Br)c2oc(C(=O)NC(C)C(c3sccc3C)=O)cc2c1 c1(C(=O)NC2(C)CN(C(C(CC)SC)=O)C2)nc(Cc2ccccc2)sc1C C1(COC)CC(CNC(=O)C(c2ccc(Cl)cc2)=O)N(C(=O)Cc2cnn(C)c2)C1 c1(OC)ccc(C(N)=O)cc1C(=O)NC1CCCN(C(C2CC2OC)=O)C1 CC1CCN(C(=O)CN(C)C(N)=O)C(CNC(C2CCC3(CCC3)C2)=O)C1 Cc1nc(Cl)c(NC(C2CC(F)CN(C(=O)C3CC3)C2)=O)c(Cl)n1 N1(C(C2CCN(CC)C2)=O)CCC(C(N2CCC3(CCCO3)C2)=O)CC1(C)C c1(C(=O)NCCC2CC(NC(C(C)CC3CCCC3)=O)C2)cc2n(c1)CCOC2 c1(N2CC(C)C(NC(=O)Cc3ccc4c(c3)CCO4)C2)ncnc2cccnc12 c1(OC)nsc(OC)c1C(=O)NC(C)CCN(C(=O)Cn1cnnn1)C N1(C(CCOCC)=O)CCC2CCN(C(=O)C(c3ccccc3F)(C)C)CC2C1 C1(NC(C)=O)CCCC12CCN(C(=O)CS(=O)(=O)Cc1cnn(C)c1)CC2 C1(CC)CN(c2nnc(C(c3ccccn3)(F)F)n2CCC(=O)NC)CC(C)O1 c1(NC(C2CC3CC2(c2cccnc2)C3)=O)c(Cl)cc(I)cc1Cl C(=O)(C(=O)C(F)(F)F)N(C1C(N(C(C(C2CCC(=O)N2)C)=O)C)CCCC1)C C1(NC(c2cccc(OC)c2)=O)CCN(C(=O)Cc2ccc(O)cn2)C(C)C1 c1(CC(=O)NC2CC(CNC(C3C(COCC)C3)=O)C2)c(Cl)cnn1C CC1CN(C(=O)C(O)CCCNC(=O)Cc2ccc(F)cc2)CC(=O)N1C CC1CN(C(=O)CC(C(F)(F)F)c2ccccc2C(=O)O)CCC12CCOC2 C(=O)(CC1CCc2ccccc21)N1CC(C)(F)CN(C(=O)CC2CC2(Cl)Cl)CC1 C#Cc1cnn(CC(=O)NC(CNC(=O)COCC2CCOC2)(CC)CC)c1 C1(C(=O)N(CCC(C)NC(=O)CCC(C)CN(C)C)C)(OC)CCC(C)(C)CC1 N1(C(C(C)OCC)=O)CCC(C)(C)C(NC(c2cnc(CC)[nH]2)=O)C1 C1(C)(NC(c2cn(C)nc2)=O)CCCN(C(c2cnn3c2OCC3)=O)C1 c1(N2CCC(C(F)(F)F)CC2)nc(=NCC2CCC3CCC23)[nH]c2cccnc12 C1(N(C(c2c(-c3cncc(C)c3)nccc2)=O)C)CCCCN(CCO)C1 C(CC)(CCCC(=O)NCC[Si](C)(C)C)NC(C1(CC#C)CC1)=O CCCCCCC(=O)N1CCC(CNC(C2(C)CC2Br)=O)CC1 C12(C(=O)NC3CC4C(NC(CCC(=O)N(C)C)=O)C4C3)CCCN(CC1)C2 N1(C(c2nc(CCC)sc2)=O)CCn2c(CNC(C3C=CCC3)=O)nnc2C1 N1(C(CCOCCOC)=O)CCC(O)(C(C)NC(c2cc(C(C)=O)cn2C)=O)C1 c1(C(=O)NCC(C)(C2CCC2)NC(C23COC(CCO2)C3)=O)cc(F)cnc1O C1(C(=O)NCCC(CNC(CSc2cccc(C)c2)=O)O)CN2CCN1C(C)C2 N1(C(CC(C(C)C)NC(c2ccc(CC)s2)=O)=O)CCC2(CCC2)C(O)C1 c1(SCC(N2CC3C(NC(C=CC(=O)OCC)=O)(C3)C2)=O)ccc(C)cc1C Cn1cc2c(C(=O)NC3CCCC3NC(c3cnsc3)=O)cc(F)cc2n1 CC1CC(NC(c2ncoc2C(C)(C)C)=O)CN(C(=O)C=C2CCN(C)C2)C1 C(N=c1[nH]c(N2CCC(OCCOC)C2)nc(=N)[nH]1)c1n(C)nc(CC)c1Cl N1(C(C(C(C)O)N(C)C)=O)CC2(C1)SCCC2NC(c1cc2cnccc2o1)=O N1(C(C(CC)C#N)=O)CC(C2CCCN(C(=O)CNC(c3ccco3)=O)C2)C1 N1(C(C=CC)=O)CCC(CNC(=O)C(C)Cc2ccccc2F)(OC)C1 CCCCC(C(=O)N(C)CC1CCCN1C(c1ccc(O)c(Cl)n1)=O)NC(N)=O C1(C)(CC(=O)NCC2C(C)CCN(C(=O)CCC(F)F)C2)Oc2ccccc2O1 N1(C(CCCC2(NC(COCC#C)=O)CC2)=O)CC2CSCC2C1 c1(C(N2CCC(C(=O)Nc3ncc(C)cc3Cl)C(O)C2)=O)ccc(I)c(F)c1F c1(CNC(C2(OC)CC(C)C2)=O)ncccc1C(=O)NC(C1CCOCC1)(C)C Cc1sc(C)c2sc(C(=O)NC3CN(C(c4ccsc4)=O)CC4(CC4)C3)cc12 N1(c2ccnc(NC3C(CCCC)CCC3)n2)CCC2(CC1)CCN(C)C2 c1(C(N(C2CCN(C(CCC=C=C)=O)CC2)CC)=O)cc(C(=O)OC)cc(F)c1F C1(C(N(CC(C)N(C(=O)CCc2cn(C)cn2)C)C)=O)CCNC(=O)C1 C(=O)(C1=COCC1)N(CCCNC(=O)CC1(N2CCCC2)CC1)C1CC1 N1(C(C2C(OCC)C2)=O)CC2C(N(C(=O)CCc3ccsc3Cl)C)C2C1 N1(C(c2ccn(C(C)C)n2)=O)CCCC1C1CCCN1C(c1nc(=N)cc[nH]1)=O N1(C(C2CCN(C(C3(C)CNC(=O)N3)=O)C2)=O)CC2CC(O)CC1C2 c1(OC)cc(C(N2CC(O)(c3ncnn3C)C2)=O)sn1 C#CC(CC(C)(C)C)NC(=O)C(CCOCCO)NC(c1cccc(CO)c1)=O Cc1cc(C(=O)N(CCC(C)NC(C2CCC(=O)N2C2CC2)=O)C)oc1C N1(C(C(O)(F)F)C2CCCCC2)CCN(N2CCOC3COCCC23)CC1 Cc1nc(O)sc1C(=O)NCC1CCC1C(=O)NC1CCCCC1CCO C(=O)(C(=O)N=S(C)(C)=O)NCCN(C(c1ccc(CN(CC)CC)o1)=O)C1CC1 CCC(C)(CCC(C)C)C(=O)N1CCn2cc(C(N3CCC(F)C3)=O)nc2C1 C(=O)(C(O)C1=CCCCC1)NC(C)(CO)C(=O)NCC1(O)CCOC1 S(=O)(=O)(c1cccc(C#N)c1)N1CC(C(=O)Nc2c(C)c(Br)cnc2)NCC1 c1(C(N2C(CNC(CS(CC)(=O)=O)=O)CC(F)C2)=O)cc2cccnc2[nH]1 Cc1nn(C)c2nc(C(=O)NC3CCC(CNC(c4ccccn4)=O)C3)ccc12 S(=O)(=O)(c1cc(F)c(F)c(F)c1F)C(NNC(c1c[nH]c2ccccc12)=O)=O CC12CCC(C(=O)NCC3CC3NC(=O)Cc3csc(-c4ccoc4)n3)(C1)OC2 CC(C)(CCCNC(C1COCOC1)=O)C(=O)N1CC(CO)C(O)C1 N1(C(C(COC)C)=O)CCC(CC(N2CC(c3nncs3)C2)=O)CC1 C(C)(C(=O)NC1CC(OCC(=O)N(C)CCc2cccs2)C1)OCOC c1(OC)ccc(COCCO)cc1-c1cc(F)ccn1.N1CCC(O)(CC(=O)O)C1 C1(NC(C2CC23CCC3)=O)CCN(C(=O)CC2CCOCC2)C(C2CC2)C1 c1(SCc2n(C(C=C)C)nc(-c3cccc(N(C)C)n3)n2)noc2c1CCCC2 c1(NC(C(CCC)C)C)ncccc1S(=O)(=O)NC(CF)CF c1(-c2cc(C)c(O)cc2)ccc2ccnc(NCc3cn[nH]c3)c2c1 C1(N(C(=O)C=Cc2cn(C)nn2)C)CN(C(C2(n3cncn3)CC2)=O)CC1(C)C CC1C(NC(=O)CC2OCCOC2(C)C)CCCN1C(c1nn(C)cc1Cl)=O Cn1cncc(C(N2CCC(CO)C(NC(=O)CC3CS(=O)(=O)C3)C2)=O)c1=O C(C(C)(C)C(=O)NC(CO)C(C)NC(c1ccn(CC(C)C)n1)=O)NC(=O)OC N1(C(C(=O)NCC2CC2)=O)CCOC2CCN(C(C3CCCNS3(=O)=O)=O)CC12 c1(C(N2CCCC(CN(C(=O)Cc3c[nH]ccc3=O)C)C2)=O)cc(O)ncc1Br C(=O)(C1=CCCCC1)NC(CNC(c1c(C)cnn1C)=O)(C)C1CC1 C1(NC(C(C)C2CCCO2)=O)CN(C(=O)C(=C2CCCCC2)F)C2CCCCC12 N(C(=NCCCF)N1CCSC(CSC)C1)CC1C(C(=C)C)OCC1 c1(C(N2CCN(C)C(CNC(C3CC4(CCC4)C3)=O)C2)=O)[nH]cc2c1CCCC2 N1(C(C2C(C(C)O)C2)=O)CCC(NC(c2cncc(Cl)c2Cl)=O)C2(CCC2)C1 c1(C(C(=O)NC2CCCC2)N(C(CC=C)C)CC)cnc(C)[nH]1 CCCC(C)(O)C(=O)N1CCC(C2CCCN2C(=O)Cn2ccnc2C)CC1 c1(C(=O)NC2C=CC(CNC(=O)CCOC3CCC3)C2)ccc(O)c(F)c1 N1(C(C2(C#C)CC2)=O)CCC(c2nnc(CNC(=O)CC(C)(F)F)s2)CC1 N1(CC(CC)C)CCC2CCC(C1)N2C(=O)Cc1c(F)cccc1Cl c1(C(N(C2CCN(C(c3cccnn3)=O)C2)C)=O)ccc(C2CC2)nc1O c1(C(N2C(CN(C)C(C3(CC(F)(F)F)CC3)=O)CCC2)=O)ccc2c(c1)COCC2 C(C)(CO)(C(=O)N(C)Cc1ccncc1)NC(C1CC(CC)C1)=O c1(C(=O)NCCC2CCN(C(C=CCCC)=O)C2)ccc2ccc(Br)cc2n1 C1(n2cc(C34N(C(C(CCC)CCO)=O)CC(C3)C4)nn2)CCC(F)(F)CC1 CC(CC(=O)NC1CC(C)N(C(=O)COc2ccn(C)n2)C1)CC(F)(F)F CCCCCCC(C(=O)NCCN(C(c1c[nH]c(=N)s1)=O)CC)NC(C)=O c1(C(=O)N)cc(CSC)no1.C12CC(C1)CNC2.C(C)(C)(C)OC(=O)N Cc1cc(C(=O)NCC2CC2NC(=O)CCN(C(N)=O)CCO)c(C(F)(F)F)o1 C#CC1(C)CCCN(C(C2C3CN(C(C4(O)CCOCC4)=O)CC23)=O)C1 CCCC(C(=O)NC1CN(Cc2cc(C(F)(F)F)nn2C)CCC1C)C(C)C c1(C(N(CC(CCC=C)O)C)=O)cc(C#N)cc(C#N)c1 c1(SCC)cccc(NC23CC(C(N(C)Cc4cnccc4C(=O)O)=O)(C2)C3)c1F C(CCN=c1nc2scnc2c(NC2CCCC23CC3)[nH]1)N1CCC(C)CC1 Cc1cncc(CNC(C2CC(O)CN2C(=O)C=C2CCOCC2)=O)c1 N1(C(C23CC(C)C2C3)=O)CCCC2C1CCN2C(=O)CC1CCN(C)CC1 c1(CC2N(C(C(C)N(CCC)C3CC3)=O)CCC2)cccc2ccccc12 C12(CNC(C)=O)CN(C(c3ccc4c(c3)OCC4)=O)CC(F)(C1)C2 C1(C(=O)NCC(C)(C(C)C)NC(Cc2c(C)cccc2)=O)CC2C(C1)C2(F)F C1(NC(C2C(COC)C2)=O)CCOCC1NC(=O)CCN1CCC(C)CC1 C1(C(=O)NCCN(C(CCCOCC)=O)C2CCCC2)Cc2cccnc2C1 N1(C(CNC(=O)NC)=O)CCC(CCNC(c2cccn2C2CC2)=O)C1 c1(NC(C2(C)CCN(Cc3c(Cl)cccc3Cl)C2)=O)c(O)ncnc1O O=C1CC(C(N2CCCCC(NC(c3cnn4c3SCC4)=O)C2)=O)CC(=O)N1 CCC(CC)C(C)NC(=O)C(CC1CC1)NC(c1ccsc1OC)=O c1(C(N2CCC(C(C)NC(C(CC)NC(C)=O)=O)C2)=O)c(Cl)nn(C)c1Cl Cc1ccc(C(C(=O)NCc2cccs2)N(C2C3COCC23)C)nn1 c1(N2CCCC(C)(CC)CC2)cc(Br)ccc1S(=O)(=O)NC(CO)C1CCC1 c1(C(N2C(CNC(C(=O)NCC)=O)CC(OC)C2)=O)cn2ccc(F)cc2n1 C1(C(=O)OC)C(F)(F)C12CC(C(=O)NCC1CCC3C(C1)C3(F)F)C2 N1(C(=O)Cn2nnnc2C2CC2)CC2CCC(C1)N2C(C1CC(O)C(F)C1)=O C1(C(=O)NC2CC(C#C)C2)CCN(C(=O)OC(C)(C)C)C12CCSCC2 c1(CC(N2CCCC(NC(CC3C(C)=NOC3=O)=O)C2)=O)c(O)nc(=N)[nH]c1C N1(C(C2N(CCC)CCC2)=O)CCOC(C(N2CCC(F)CC2)=O)C1 c1(OC)cc(C(F)F)c(C(=O)NC2CCC(C)N(Cc3ccccc3)C2)cn1 C1(C(=O)NC2CCN(c3snc(CCOC)n3)CC2O)Cc2ccccc2CO1 CCC(CNC(=O)C=C(C1CC1)C1CC1)(CC)C(=O)NC(C)COC(C)C C1(CC(N2CCC(CN(C(=O)CC3C=CCC3)C)CC2)=O)CCCCC1(F)F c1(OC)cc(NC(=O)COC(c2cc(C)cc(O)n2)=O)c(Cl)cc1Cl C1(CC)CN(C(=O)CN(c2ccncc2)C)CCN1C(=O)C(C(C)C)OC C1(C(=O)NCC(CN(C(C(CC)F)=O)C)C)CCc2ccccc2O1 c1(NCc2occn2)nc2ccccc2nc1NCC1CN(C(=O)C2CC2)C1 C1(C(=O)NCCNC(=O)Nc2cccc(-c3ncn(C)n3)c2)(OC)CCOCC1 c1(C(N(C2CCC(NC(=O)C(C)(C)C)C2)C)=O)ccc(P(C)(C)=O)s1 C1(N(C(C2(C)CC(=C)C2)=O)C)CC(C)OC(C)C1.c1(C(=O)N)ccn(C(C)C)n1 Cc1ccc(Cl)c(OCC(=O)NC2CC(NC(=O)CC3CCC3C3CC3)C2)c1 c1(C(N(CCCCC(N2C(CCC)COCC2)=O)C)=O)cn2c(n1)CCC2 N1(C(C(C)CO)=O)CC23CCCCC2(C1)CN(C(=O)CC1CCCCC1)C3 c1(OC)cc(N)ccc1C(=O)NC1CCCC1NC(=O)C(C)CC1CCC1 c1(C(N2CCC(C)(CNC(C34CCCN3CCC4)=O)C2)=O)cc([N+](=O)[O-])ccn1 N#Cc1ccc(-c2cn(CC3CCN(C(c4ccc(Br)s4)=O)C3)nn2)cc1F c1(-n2ccc(C(=O)NCCCN(C)C(C34CCCCC3C4)=O)n2)ccccc1F N1(C(C=C(C)C)=O)CCC2C(C(=O)NC(C)C(O)C(F)F)C2C1 N1(C(c2cc(OC)ns2)C(=O)NC2CCCC2)CCOCC1P(C)(C)=O C1(C(C)C(=O)NC(C)C(F)F)CCN(C(=O)COc2cccc(F)c2)CC1 Cn1c(C(=O)NCC2(C(C)(C)C)CCN(C(c3csc(O)n3)=O)C2)cnc1Cl c1(C(=O)NC2CC(F)(CNC(c3cnsc3)=O)C2)cncc2[nH]ccc12 c1(C(=O)NC(CC(C)NC(c2cn(CC)nc2C2CC2)=O)C)cc2ccsc2[nH]1 C(CC(C(=O)NCc1cncs1)NC(=O)CCc1nc(O)n[nH]1)N(C)C N1(C(c2c(CNC(C3(CC)CCCCO3)=O)noc2)=O)CC2CCCC2(CO)C1 CC1C(=O)Nc2ccc(C(=O)NCC=CCNC(c3ccc4ccoc4c3)=O)cc21 C1(C(N2CC(NC(C(C)N3CCCC3)=O)C(F)C2)=O)CC(C)(C)CN1C c1(C(N2CCN(C(C3CCC(F)(F)C3)=O)CC2)=O)ccc(I)cc1[N+](=O)[O-] C(CC(C)C)(C(=O)NCCCCC1CC1)N(C(C(C(C)C)NC(C)=O)=O)C Cc1cnc2ccccc2c1C(=O)NCC1(O)CC(NC(=O)CNC=O)C1 C1(C(N(CCCOC(C)C)C)=O)CC(C)(C)CN1C(=O)CC1COCCO1 N1(C(C(Cc2ccc(C)cc2)C)=O)C2CCCC1CN(C(C1(F)CC1)=O)CC2 C1(C(=O)OC)C2CCCC1CN(C(=O)C(n1cc(-c3ccncc3)nn1)C)C2 C1(NC(c2c(C)occ2)=O)(CO)CCCN(C(C2CC2C(C)(F)F)=O)C1 c1(NC)ncccc1C(=O)NCC(C1CC1)N(C)C(c1sc(N(C)C)nc1Cl)=O c1(CN2CCC(Nc3nc(OC)c(F)cn3)CC2)cccc([N+](=O)[O-])c1 n1(CC(N2CCCC(C)(CNC(C(CCC)O)=O)C2)=O)c(C)nc2ccccc12 c1(CC)cnccc1C(=O)N(CC(C)(C)CNC(=O)C(C)C1CCOC1)C N1(C(CC(=O)OC)=O)CCN(C(C2CCN(S(C)(=O)=O)C2)=O)C(C2CCC2)C1 C1(F)(C(=O)NCCNC(=O)NC)CN(C(C2CN(C)C2)=O)C1 c1(C(=O)NCCC(C)N(C)C(C2Cc3nccnc3C2)=O)ccc2cncn2c1 Cc1nc(C)n(O)c1C(=O)OC(C)(C)C.C1(C)CC(=O)N1C.C1C(=O)N1 CC(C)C(C(=O)NCCc1cncs1)C(C)NC(c1ccsn1)=O c1(NC(C)=O)ncnc2c1nc(N(C(C)C(=O)O)C(c1ccccc1Cl)=O)n2C N1(C(CCCOCC=C)=O)CCC2(CCC2)C(NC(=O)CC2CCC(=O)C2)C1 C1(CNC(C(C)SC)=O)CCCC2CN(C(=O)C=CC3(C)COC3)CC12 C=C(Cl)CCC(=O)NCC(C1CC1)NC(=O)C(C)Oc1cccc(C(C)C)c1 c1(OC(C)C)cc[nH]c(=NCCCOC(C2CCC3(C2)CC3(F)F)=O)c1[N+](=O)[O-] C1(NC(C2CCC3CC3C2)=O)CCCN(c2ccc(-n3ccnc3)cc2)C1 C1(O)(C(N2CC=CC2Cn2cc(CCOCCO)nn2)=O)CCCCCC1 C(C(=O)NC(COC)CC(=O)N1CCCCC1)(C(C)C)OCC N1(C(C(COC)OC)=O)CCCCC1CC(=O)NCC(C1CC1)SC.C(C)=O C1(NC(COC)=O)CC2(CCN(C(c3ccnc(N(C)C)c3)=O)CC2)C1 C(=O)(C1=CC2(CCOC2)C1)N1CCCC(CCNC(CCCC#N)=O)C1 c1(OC)ccc(Br)c(CS(=O)CC(=O)N(c2ccc(Br)cc2)CC(C)C)c1 C(=O)(CC(C)(C)CNC(C1CC(C)(C)C1)=O)NC(c1ccnn1C)C C1(NC(CN2CCN(C)CC2)=O)CN(C(c2ccc(O)nc2)=O)CC1N=[N+]=[N-] CCC(CCC(=O)NCC(CC)(CC)OC)NC(=O)C(C)(O)COC C1(O)(C(=O)NCC2(C)CCCN(C(CC(=O)NCC)=O)C2)CCCC(C)(C)CC1 C1(C(=O)NCC2(F)CN(C(c3n(CC#C)ccc3)=O)C2)CCCCC1(F)F N1(CC(N2CC(F)(CNC(C3C(=O)NCC3)=O)C2)=O)CCCC(N(C)C)C1 C12(C(=O)NC3CC(NC(c4c(NC)nccc4)=O)CC3O)CCCN(CCC1)C2 Cc1cccc(CCC(=O)NCC2CCN(C(=O)C(N3C(=O)CCC3=O)C)C2)c1 C1(NC(CCC=C)=O)COC2(CCN(Cc3cccc4cccnc34)CC2)C1 c1(NC(C23C(CN(Cc4ccc(C(=O)OC)cn4)C2)C3)=O)ncc(Cl)cc1F C1(C(=O)NC2CC23CC(NC(=O)CSCC(N)=O)C3)(OC)CCC(C)C1 C(=O)(CCC1=CCCCC1)NC(CCC)CC(=O)NCC1CC(=O)N(C)C1 CC1=C(C(=O)N2CCC(CNC(C3(c4cncc(C#N)c4)CC3)=O)CC2)CCC1 CC(C)C(C)CC(=O)NCC(C)C(=O)N(CCCn1ccnc1)C n1(CC(=O)NC2CN(C(C=C(CCC)C)=O)C2)c(C(C)OC)nc2ccccc12 C(=O)(N1CCCc2nncn21)C1N(C(CC2OCC(C)(C)C2)=O)CCC(F)C1 c1(C(N2CC3(OCC(NC(CC4(C)CC4)=O)C3)C2)=O)cnc2c(c1)NC(=O)CS2 N1(C(Cc2cccc(C)c2F)=O)CCCCCC(NC(c2onc(C)c2C)=O)C1 C12(C(N3CCC(C)(NC(=O)CSC(C)(C)C)C3)=O)CCC(CO)(CC1)CC2 c1(SCC)ccccc1C(N1CCC(N(C)C(C2CCOC2C2CC2)=O)CC1)=O C1(NC(C(c2c(C)noc2C)C)=O)CC2CCC1N(C(c1n[nH]c(=N)[nH]1)=O)C2 N1(C(c2c(CC)ncs2)=O)CCOCC1CNC(=O)Cc1ccsc1Cl c1(C(=O)NCC(CC=C)NC(=O)CC=C(Cl)Cl)cc2cccc([N+](=O)[O-])c2[nH]1 N1(CC(=O)NCCCCC2CN(C(=O)Cn3cnnc3O)C2)CCCS1(=O)=O CN1CCCC12CCN(C(C1(CNC(c3cnc(=N)[nH]c3)=O)CCCO1)=O)C2 c1(C(=O)NC(CCOC)CNC(=O)CCn2cccn2)cc(Br)cnc1O C(=O)(CC(C(F)(F)F)OCC)NC12CC(NC(C=CC=CCCCCC)=O)(C1)C2 N1(C(C2C(OC(C)=O)C2)=O)CC2CC(NC(=O)CCCCC(N)=O)C(C2)C1 N1(C(C2CCC(C)(C)C2)=O)CCC2C(C1)CN2C(c1ccc(C2CC2)cc1)=O.C Cc1cc(Br)cc(C(N2CC(F)(F)CC2CNC(C2CC2CF)=O)=O)c1N c1(NC(c2cc(Br)cc(OCC)c2N)=O)nc2c(Br)cccc2s1 c1(CC)cc(NC(C2CC3CCC2N3C(C2C3C4CCC(C4)C23)=O)=O)cc(F)c1 C1(CNC(CN(CC)CC)=O)CN(C(=O)CC2CCOC2)Cc2nccn2C1 CCC(C)C(C(=O)N1CC=C(C(=O)N(CC2=CCSC2)C)C1)N(C)C S(=O)(=O)(c1ccc(=NCC2CC2(Cl)Cl)[nH]c1)NCc1ccc(N(C)C)c(F)c1 N1(C(C2CC(O)(CNC(c3cc(C)sn3)=O)C2)=O)CCC(C2CCC2)CC1 CCCC(C)(O)CC(=O)N1CCN(CC(=O)NC2CCCC2)CC1C C(=O)(CCP(C)(C)=O)NC(CNC(C(c1ccc(Cl)cc1)C)=O)CO C1(N(C(c2cnsn2)=O)Cc2ccccc2)CC12CCN(Cc1cnco1)CC2 c1(C(=O)NC(CC)CNC(c2nn(C)nc2Br)=O)ccc(C#N)nc1O C1(N(C(=O)CC2CCOCC2)C)CN(C(C2CCC(C(F)F)CC2)=O)CC1(C)C CC1CN2CCN1C(C(=O)NCC(C)CNc1ccc([N+](=O)[O-])cc1)C2 C1(C(=O)NC2C(NC(CCNC(N)=O)=O)CCCC2)Cc2cncn2C(=O)N1 C1(CCC)(NC(=O)C(C)CN(C)C(c2cnnn2C)=O)CCOC1 C(CCC(O)C(=O)NCc1nncs1)OC(C)C.C12(CC1)C(=O)NC2 C1(CNC(c2nc(C3CC3)cs2)=O)COCCN(C(c2cc(O)cc(Cl)c2)=O)C1 C#Cc1ccc(C(=O)NC(C)(C)CCCNC(c2coc(C(F)F)c2)=O)cc1F c1(C(=O)OC)cc(Cl)cc(Cl)c1NC(=O)C(N1CCCC1CSC)=O N1(c2nccc(OCC)n2)CCC(NC(=O)C(C)(C2CC2)OC)C(C)(C)C1 N1(C(CCC(=O)c2cccs2)=O)CCOC2(C1)CN(C(c1coc(Cl)n1)=O)C2 c1(C(=O)NCC(C)N(C(c2cc(C)sc2C)=O)C)cccc(S(C)(=O)=O)c1 N1(C(C(CC)NC(C)=O)=O)C2CCC1C(CNC(=O)C=C1CCSCC1)C2 C1(NC(CN(CCOC)C)=O)CCN(C(=O)C(c2cccc(OC)c2)C)C1(C)C c1(C(=O)NCC(C)CNC(C2CC2CF)=O)ccc(S(C)(=O)=O)c([N+](=O)[O-])c1 C(C(C(=O)NC1CCC(NC(=O)C(C)(C)O)C1)NC(C)=O)OC c1(C(N2C3C(NC(C(C)n4cncn4)=O)C(C3)C2)=O)ccc(O)nc1Cl CCC(C(=O)N1CCSCC1C(N1CCC(C(N)=O)CC1)=O)C(C)C C#CCCCC(=O)N(CCNC(c1ocnc1Br)=O)C1CC1 N1(C(COC(C)C)=O)CCC(C2CCN(C(C34CCCCC3C4)=O)C2)CC1 C(=O)(C(O)P(C)(C)=O)NCCC(C)N(C(CCC=CC)=O)C c1(C(N(C(C)C)C(C2CCN(Cc3cncc(F)c3)CC2)=O)=O)ccc(O)cn1 C1(NC(C=CC(C)C)=O)C2CC1N(C(C1(C(C)C)CC1)=O)C2 C1(NC(CCCCCC=C)=O)C2COCC1CC(NC(C1CCC(=O)C1)=O)C2 c1(C(N2CCC(CC3CCCO3)C2)C(=O)NCCC)nnc(-c2ccccc2)s1 c1(CN2C(C(=O)NCC3(C)OCCO3)CCCC2)cccc2nonc12 CCCCC(C)CCC(=O)N1CCC(N(C(c2cncc(F)c2)=O)CC)C1 C(=O)(C(CC(C)C)C(C)C)NC(CC(=O)NCC(CSC)(C)C)C(F)F C1(C(=O)NC2C=CCN(C(=O)C3=NOCC3)C2)Cc2nccn2C1 Cc1cc(C(=O)NC(C(=O)NCC2(n3cccn3)CC2)C2CCOC2)c(C)s1 C1(C(=O)NCC(C(=O)NC2CC(CC(C)(C)C)C2)C)COCCC1C C(=O)(CC1=CCCCC1)N1CCC(C=C)(C(=O)NCC(F)(F)COC)C1 c1(OC)ccc(CN2CCC(F)(C(=O)Nc3cncc(C(F)(F)F)c3)C2)cc1I C1(CNC(=O)C2CC2)CC2CCC(C1)N2c1ccnc(CO)n1 c1(NCC2(COC)CC2)cc(S(=O)(=O)N2CCC(CN3CCC3)C2)ccc1C#N O=C1CC(C(=O)NC2CCCCC2C(=O)NC2(c3ncc[nH]3)CC2)=NN1 c1(C(=O)NC2C(NC(C3(CC)CC3)=O)CCC2)ccc2c(c1)CCS2(=O)=O N1(C(c2c(OC)cc(OC)c(Cl)c2)=O)C2CCCC1CN(C(C1CC1C)=O)CC2 C=CC1(C(N2CC(OC)C(C)C2)=O)CCN(C(c2cnc(C3CC3)o2)=O)CC1 C(=O)(C1c2c[nH]nc2CN1C(=O)CCC1CC1C)NC1CN(CC)C(=O)C1 Cc1csc(CCC(=O)NCCOCCN(C(=O)CC2CCCC2O)C)n1 c1(-c2nc(-c3c(C)ccnc3)n(C3CCC(C)C3)n2)c2ccccc2nn1C Cc1nc(CCC(=O)NCCC2(CNC(c3nc(=O)n(C)[nH]3)=O)CC2)oc1C N1(CC(N2C(CNC(C(c3cccc(Cl)c3)OC)=O)CC2)=O)CCCCCC1 C1(C(=O)NCC2N(C(C=COCC)=O)CCCC2(C)C)CCn2c(C)cnc2C1 C1(C(=O)OCC)CCC12CCN(C(=O)Cn1cnnn1)CC2 Cc1cc(C(N2CCC(COC3CCOC3)CC2)C(=O)NCC(F)F)cc(Cl)n1 C1(C2CCOCC2)(C(=O)NCC(CCNC(=O)C=Cc2cc[nH]n2)O)CC1(F)F c1(Sc2ccc(C(=O)NCC(C)(C)CNC(=O)CC(F)F)o2)ccc([N+](=O)[O-])o1 C=CCC(C(=O)N1CC(C)(C)C1C1CC1)NC(C1CCC(N(C)C)C1)=O C(C1OCCc2ccccc21)N(S(=O)(=O)c1ccccc1)CCN(C)C(=O)OC CCCC(C)(C)CC(=O)N1CC(O)(CNC(=O)CC(C)CC(C)C)C1 C1(CNCCC(c2ccnn2C)C)CC2CC1(CO)C2 C(=O)(C1Cc2ccc(Cl)cc21)NCC(CNC(c1c(C)c(N)cc(O)c1)=O)(C)C c1(NCCCCOC(=N)O)cc(N)ccc1SC.C1(CC=O)(C(=O)OC)CC1 c1(-n2c(C(CC)C3CC3)nc(CCn3ccnc3)n2)cc(F)ccc1F C=CCC(CNC(C1OCCC1C(F)(F)F)=O)NC(c1cnc(C(C)C)s1)=O C(=O)(CS(=O)(=O)N1CCC(CC(=O)NCc2cc(CC)n[nH]2)C1)OCC C12(NC(CCCC3C(C)C3)=O)CCC(CC1n1cc(-c3ccncc3)nn1)C2 c1(C(=O)NCCCC(C)NC(c2ccc(CCCC)cc2)=O)c(F)cccc1Cl N1(C(c2cnc(CC)nc2)=O)CC2CCCC2(NC(c2cccn2C2CC2)=O)C1 N1(C(c2c(C)ncs2)=O)CC(NC(c2ccc(CN(C)C)cc2)=O)CC1CO Cn1cnc2c1CCCC2C(=O)NCC1(NC(=O)CC2COCCO2)CCC1 Cc1cc(S(N)(=O)=O)oc1C(N1CC2CC1CN2C(c1cnc(O)o1)=O)=O CC(C)(F)CC(=O)NCC1CC1CC(=O)NCCCCCC1CC1 N1(C(CNC(CC)=O)=O)CC(NC(=O)C(N2CCCCC2)C)CC1(C)COC c1(CC)nc(C(=O)NC2C=CC(CNC(c3cnncc3O)=O)C2)c(N)s1 N1(C(Cc2cc(C)[nH]n2)=O)CC2(CCN(C(c3cnn(C(C)C)c3F)=O)C2)C1 C1(C(=O)NCCOC2CN(C(COC(C)=O)=O)C2)CCc2nc(C)nn2C1.C C(CC(C)C)(C(C(=O)Nc1ccc2ccccc2c1)N1CCCCC1C#N)SC CC1(C)OCCN(C(C2C3CCCCC23)C(=O)NC2CCOCC2)C1(C)C CC(CN1CCOCC1)C(=O)N1CC(OCCNC(C2(CCC#N)COC2)=O)C1 c1(C(C)C)nn(-c2ccccc2)cc1NC(c1csc(-c2nn[nH]n2)c1)=O c1(C(=O)NCC2C(NC(c3ncc(OCC)nc3)=O)C2)cc2occ(Br)c2[nH]1 CCC(C)C(CC(=O)N1CC(CC)CC(C)C1)NC(=O)CNC(=O)C1CC1 c1(OC)cccc(F)c1C(N1CC(C(=O)NCc2cccc(C)n2)CC(F)C1)=O Cc1c(C(N2CCC(C)(CCNC(=O)CN3CC=CC3)C2)=O)noc1C1CC1 C1(CNC(C(c2nc(C)sc2)=O)=O)CCC(C)CN1C(=O)Cn1nccn1 C1(N(C(C(C)O)=O)C)CN(C(c2ccoc2CC(N)=O)=O)CCC1C Cc1ccc2c(C(N3CCC(NC(=O)C4=C(Cl)CC4)C(C)C3)=O)coc2c1 N1(C(CC(CC)O)=O)CC2CC(C(N3CC4(COC(C)C4)C3)C(C)SC)C(C2)C1 Cn1c(I)cc2c(NC(C3CSCCN3S(=O)(=O)CCCCCl)=O)ncnc12 c1(NC(C2C(O)CCN2C(c2ccc(O)cc2O)=O)=O)ncc(F)cc1Br C12(C(=O)NC3(CO)CCN(C(=O)Cc4ccc(Cl)c(F)c4)C3)CCCC1CCC2 N1(c2nnc(C(C)(C)C)o2)CC(NC(=O)C2=CCCCCC2)CC2(CC2)C1 CCCCC(CNC(=O)C(=O)NC(C1CCN(CC2CC2)CC1)C)CC c1(C(=O)NC(c2ccc(CC)cc2)CNC(=O)CCC(N)=O)csc2nccn12 C(=O)(C(O)CN1CCCC1)N(CC(C)C)CC(=O)NC1(C)CSC1 N1(C(CC2CC(SC)C2)=O)CC=C(CC(=O)N2CCCN3CCCC3C2)CC1 N1(C(C(C(C)C)c2ccc(Cl)cc2)=O)CC2CN(C(c3cc[nH]n3)=O)C2C1 Cc1cncnc1N1CCSCC1.C12CCN(CC1)C1CCC(CC1)N2.N(C)C C(=O)(C1=CCC2CCC1N2C(C12C(=O)C3CC1C2C3)=O)N1CC(OC)C2(C1)CC2 C1(C)(CNC(C(C)=C(CC)C)=O)CCC(NC(c2occc2C2CC2)=O)C1 CCC(C(=O)NCCc1cc(C(=O)NCC2(CO)CCOC2)no1)SC C1(NC(C2C(NC(CC3CC(CC)C3)=O)CCO2)=O)CCOCCC1C c1(C(=O)NC2(CNC(CN(CCOC)C)=O)CCOC2)cnn(SC)c1C c1(NC(C)=O)ccc(N(C)C)c(S(=O)(=O)N2CCCC(c3ncco3)C2)c1 N1(C(CC(C(=C)C)ONC(C23CCC(CC2=O)C3)=O)=O)CC2(CCC2)CC1CO C1(SCC(=O)NCC2C(NC(CCNC(=O)OCC)=O)C2)CCCCC1 c1(C(=O)NC2CC3CCC2N3C(=O)CC2CC2)cc(O)c2cc(F)cc(F)c2n1 N1(C(c2cc(COC)[nH]n2)=O)CC(CNC(=O)C(C)(C)CC#N)CCC1C N1(C(C(C2CCCOC2)OC)=O)CCC(N(C(=O)C2=CCOC2)CCO)CC1 CC(C(C)(C)O)NC(=O)C(=O)NCC1CCC1CN=[N+]=[N-] C#CC1CCCC(NC(=O)CCCCCN(C)C(C2(C#N)CC2(C)C)=O)C1 c1(-c2c(C(N3CC(CC)OCC3)=O)ccnc2)ccccc1C(F)(F)F Cc1ccc(S(=O)(=O)N(c2ccccc2)CC(O)COCCCC#N)cc1 C(=O)(N=c1c(Cl)c[nH]cc1Br)NC1(C)CCN(c2nc(C)nc3c2scc3)CC1 c1(CC)ccc(C(=O)NCC2(F)CC(NC(=O)C3=COCCO3)C2)c(C)c1 C#Cc1cc(C(N2CC3(C2)CN(C(C2(C)C(C)(C)C2(C)C)=O)C3)=O)cc(N)c1 c1(NC)cc(NC(c2cc(C(F)(F)F)n[nH]2)c2nnnn2C(C)(C)C)ccc1C Cc1cc(NC(=O)CN(C)C(C2COCCN2CC(F)F)=O)ccc1Cl CC(C)CC(C)CC(=O)NC1(C)CCCN(C(C2CCCOCC2)=O)C1 N1(C(C(C(C)(C)F)(C)F)=O)CCC2(CCCCC2NC(=O)CS(=O)(=O)C2CC2)C1 C1(CN(C)C(C2CC2F)=O)CN(C(C2CCCN2C=O)=O)CCO1 C(=O)(CC(C)CNC(c1nnnn1Cc1ccco1)c1cscn1)OC N1(C(=O)COC2CC2)CC2CC(C1)N(C(c1cc(Cl)c(F)c(Cl)c1)=O)C2 N1(C(c2c(SCC)cccc2)=O)CC(F)(F)CC1(C)CNC(C1C2COCC12)=O N1(C(CC=C)=O)CCC2CCN(C(c3cccc4nnn(C)c34)=O)CC12 c1(NC(C=CC(C)(C)NC(c2ncn(C3CC3)n2)=O)=O)ccc(F)cc1F c1(N(C)CC23CC(CO2)N(C(=O)OC(C)(C)C)C3)c(Cl)cccc1[N+](=O)[O-] CC(C)CC(C)CNC(N1CCC(c2ncccn2)CC1)=O C(c1csc2ccccc12)=CC(=O)NC1CCC(C)N(C(c2cc(Cl)no2)=O)C1 N1(C(C2CC(=C)C2)=O)CCC(NC(=O)C(C)(F)F)CC1c1ccccc1 C1(C2CN(C(=O)C(C)(C)c3ccno3)C2)(NC(C2CCC(OC)C2)=O)CC1 CCC(C)(C)CC(=O)N1CCC1(C)CC(=O)N(C(CO)C(C)C)C c1(CC(=O)NC2CCCC(NC(C3(O)CCOC3)=O)C2)nc2ncccn2n1 c1(CNC(C2C(C)=CCS2)=O)nnn(C)c1C(=O)NC1CCC2CCC12 C1(C(=O)NC(C)C)CCN1C(C)C.C1C(=O)N(CCOC)CCN1C.C(C)C C1(CC(N2CC(OC)(CNC(=O)C=CC(N3CCCC3)=O)C2)=O)CC(O)C1(C)C C1(C)(CNC(C(=O)NCCOC)=O)CN(C(C2(Cl)CC2(F)F)=O)CCO1 C1(NC(C(C)CF)=O)CCC(C)(C)CC1CNc1cc(O)nc(O)n1 N1(Cc2ncn(C)n2)CC(NC(=O)C=CC2CC2)C(O)C1 C1(CNC(C2CCCN2C2CC2)=O)CC2COCC2N1C(=O)COc1ccsn1 CCC(C#N)C(=O)N1CCC(N(C(c2cccc(CCN(C)C)c2)=O)CC)C1 C1(CNC(C(C)c2cccs2)=O)CN(C(=O)C2=NOC(C)(C)C2)CCC1(C)C C1(C(=O)NCCCN(C(=O)CCCc2cc[nH]c(=N)c2)C)C2CCCCCCC12 c1(N(CC(=O)NCC(C)(C2CC2)NC(=O)C(=O)C2CCCC2)C)ccc(Cl)cc1 C1(C)(NC(C(C)OCC#C)=O)CCCN(C(C2CCOC2)=O)C1 CCCC(C)(O)CC(=O)N1CC(CNC(=O)C(C)OC)CC1C.C1CO1 c1(C(N(CCNC(=O)Cc2cnn(CC)c2)CC)=O)cc(OC)ccn1 N1(C(c2c(C)ncs2)=O)CCCN(C(=O)Nc2ccccc2Cl)CC1 N1(C(CC(C)CNC(=O)Cc2cc[nH]n2)=O)CCC(C)C(O)C1 CCS(=O)(=O)CC(=O)N1CCC(C(=O)NC(C)CC(F)(F)F)C12CC2 C(c1cccs1)=CC(N1CCCC1C1CCN(C(C2(O)CCSC2)=O)C1)=O c1(CN(C(C2(NC(C(C=CC)O)=O)CC2(C)C)=O)C)cc(C)ccn1 c1ccccc1.C(=O)(C(=O)N1CC(CSc2ccsc2)C1)C(=O)NCCN c1(-c2n(CN(CCc3ccncc3)CC)ccn2)cccc(-c2n[nH]cc2C)c1 C1(NC(c2ccc(CN(CCC)C)o2)=O)CN(C(=O)C(C)S(N)(=O)=O)CC1(C)C C1(C(=O)NCC2CCN2C(=O)Cc2cc[nH]n2)(CC)CCOC1 c1(NC(C2CC(OCC3CCCCN3C(=O)CO)C2)=O)cc(C(F)F)cc(F)c1 Cc1c(C(=O)N(CCC(=O)NC(C2CCCC2)CO)CCO)cccc1O Cc1cc(COCC)oc1C(=O)NCCN(C(=O)CCN1CCC(O)CC1)C1CC1 n1(CCCC)nccc1C(=O)NCCC(C)N(C(=O)C=CC(C)CC)C CCCCCC(=O)N1CC(CC)(NC(=O)CCc2cnn(C)c2C)C1 c1(C(N2CCN(C(c3c(CC)csc3)=O)C(COC)C2)=O)ccc2cc[nH]c2c1 c1(CC(CCCCCC(=O)N(C(=O)CC(C)c2ccco2)C)C)cnccn1 C12(NC(N3C(CC)(CO)CCC3)=O)CCC(C1)N(Cc1ccccc1)C2 c1(C(N(C2CCCC2)C(=O)Cc2ccc(Cl)cc2Cl)=O)scc2c1CCCC2 N1(C(CC#N)=O)CCCC2CN(C(c3cscc3C(F)F)=O)CCC12 c1(C(N(C(C)C(=O)N2CC(CN(C)C3CC3)C2)CCC)=O)cnc[nH]1 c1(NC(Cc2cccc(OCc3ccc(C)cc3)c2)=O)cnc(Cl)c(C)c1 c1(OCC)ccc2cc(C(=O)N(C(C)CNC(C3CCCN3C=O)=O)C)[nH]c2c1 N1(C(C(COC)OC)=O)CCC(NC(C2(CC(C)=O)CC2)=O)C(C)(C)C1 N1(C(c2ccc(CNC(C(C)CC3CCC3)=O)s2)=O)CC2C(C)C2C1 c1(OC)cc(NC(N2CCN(CC(c3ccccc3)N(C)C)CC2)=O)ccc1C C1(NC(CC2OCC(C)(C)OC2)=O)CC2(CCN(C(=O)C(N)CN)CC2)C1 C1(NC(CNS(CCOC(C)C)(=O)=O)=O)CC(O)CN(C(=O)CN2CC=CC2)C1 C(=O)(C(O)C(C)C)N1CCC(C(=O)NC(CCC)C2CCC2)C1 C1(NC(CC(C2CC2)NC(=O)Cn2ccccc2=O)=O)CCCC(O)C1O c1(C(=O)NC(Cc2cccs2)CC(=O)N2CCCC(CO)C2)cc2ccoc2s1 CCS(=O)CC(=O)NCC(O)CNC(=O)CCc1nnc(S)n1C c1(NCCc2ccc(N)c(F)c2)cc(=NCCCc2n[nH]c(=N)o2)[nH]cn1 CC(CN1CCCCCC1)N=c1[nH]c2c(c(=NCC3CC(F)(F)CO3)[nH]1)CSC2 c1(C(N2CCOC(C)(CO)C2)C(=O)NCCCOC)cc(C(F)(F)F)cc(C)c1 N1(C(c2ccc(OC)c(OC)c2)=O)CCN(C(=O)C=CCO)C2CS(=O)(=O)CC12 c1(C(N2CC(NC(C(CC)NC(N)=O)=O)C(C)(C)C2)=O)c[nH]c(=N)c2[nH]ccc12 N1(C(CCN(C(=O)CC2COC(=O)C2)C)=O)CC2C(C1)C2(F)F CCC1=C(C(=O)NCC(C2CCC2)NC(C2(F)CCCN(C)C2)=O)CCCO1 N1(C(C)=O)CC2(NC(=O)Cc3cc(N(C)C)ccc3N)CCC1CC2 c1(-c2cn(CC(N3CCC(c4scc(C)n4)CC3)=O)nn2)ccc(F)cc1Br CCCC(C(=O)N(C)CC1COCCN1C(c1csc(=NC)[nH]1)=O)OCC c1(NC(C2CC23CCN(C(c2ccccc2Cl)=O)CC3)=O)cc(F)cc(F)c1Br c1(C(N2C(C)(CNC(C3C(=C)C3)=O)CCC2)=O)nc(C(F)(F)F)n2ccccc12 CC1(C)NC(=O)N(CCCC(N2CC3CC2(CNC(=O)C=CBr)C3)=O)C1=O C1(C2CCCCC2)(C(N2CCN(C(C3C(C(C)C)C3)=O)C(C3CC3)C2)=O)CC1 c1(CC(=O)NCC(CC)NC(=O)C(C)C2CCC2)ccn(C(C)C)n1 c1(C(N2CCC(CN(C)C(C3(C)CC=CCO3)=O)CC2)=O)nccc(C#N)c1F C1(O)(CCNC(Cc2cc(C)ns2)=O)CCCN(C(C2CS(=O)(=O)C2)=O)C1 N1(C(c2ccn(C)c2)=O)CCSCC1C(=O)NC1(c2ccccc2Cl)CC1 C1(C(=O)NC(C)(C)CC2(O)CCN(C(=O)CCF)CC2)C2CCC3C(C2)CC13 C=CCC(C(=O)N(C(C)CN(C)C(C1CCC(=C)CC1)=O)C)C(C)C c1(C(N(C2CN(C(C3(Br)CC3)=O)CC2O)C)=O)c(Cl)cccc1Cl N1(C(CC2C(=O)NC(=O)N2)=O)CCC2CC2(C(N2CCn3ncnc3C2)=O)CC1 c1(C(=O)NCC(c2ccccc2)N(C(COCC(=O)OCC)=O)C)csc(C)c1 C=CC1(C(N2CCOC(C3CC3)C2)=O)CCN(C(C2C(=C)C2C(=O)OC)=O)C1 c1(N2CC(NC(c3cnc4c[nH]nc4c3)=O)(CO)C2)nc2ncc(Cl)cc2s1 N1(C(c2ccc(C)c([N+](=O)[O-])c2)=O)CC(NC(C2(C)CC2)=O)CC12CCOCC2 c1(C(=O)NC2CC(C)(NC(c3coc(Br)c3)=O)C2)cc2nc[nH]c2cn1 C(=O)(C1CCc2ccccc21)NC(C)(C)CCC(=O)NC1CCN(C(C)(C)C)C1 CC(CCCC(=O)N1CCC(F)(F)C1)NC(=O)CN1CCC(F)CC1 C(c1ccccc1)=C(C(N1C(CNC(C(CC)NC(C)=O)=O)C=CC1)=O)C CC1(CNC(C2(C(F)(F)F)CC2)=O)CCCN(Cc2ccc(Cl)s2)C1 CC(C)S(=O)(=O)CC(=O)NCCN(C(=O)CN1CCSCC1)CC1CC1 N1(CCNC(=O)CCN(CCO)C(C2C3CCC(F)C23)=O)C(=O)CCC1=O C1(OC)CCC(F)(CNC(=O)C(n2cc(CN(C)C)nn2)C)C1 CC(CF)CC(=O)NC1(CNC(c2cccs2)=O)CCOC1 Cc1c(O)nc2ccccc2c1C(=O)NCC1CSCCN1C(=O)CC(C)(F)F c1(C(=O)NCC2CCCC(NC(CC3ON=C(CC)C3)=O)C2)ccn(C)c(=O)c1 C1(NC(Cc2n(C)ncc2)=O)CCN(C(=O)COc2ccc(Cl)cc2)CC1O N1(C(C=C(C)C)=O)CCCN(C(=O)Cc2ccccc2C(F)(F)F)CC1C(C)C N1(C(C2C(C#C)C2)=O)CCN(C(=O)CC2CCN(CC(F)(F)F)CC2)CC1CF c1(C(N(C)CC2(O)CN(C(C3(CCOC)CCCC3)=O)C2)=O)cc(O)ccc1F C(CC(O)C(F)(F)F)NC(C1(NC(Cn2ncc(CC)c2)=O)CC(F)C1)=O c1(OC)cc(C)c([N+](=O)[O-])cc1N1CCOC(c2ccc(C)s2)C1 Cc1ccc(F)c(CC(=O)NC(Cc2ccccc2)CN)c1 c1(C(=O)NC2(CNC(C(C)C3CC3)=O)CCOC2)ccc(S(N)(=O)=O)cc1F N1(C(C(C(C)C)F)=O)CCCC(C)(C)C1CNC(=O)Cc1ccns1 N1(C(c2c(CC)cno2)=O)CCC(C=CC(=O)N(C(C)CO)C)CC1 C1(C)(C(=O)NCCCC#C)CCN(C(c2ccc(F)c(F)c2)=O)CC1 Cc1c(Br)ccc(C(N2CCOC3(CC3)C2)=O)c1F.c12c[nH]nc1C(=O)N2 C1(NC(=O)CCF)CC(NC(=O)C=C2CCOCC2)C(O)C1 c1(CNC(C2(CO)CCC2)=O)cnn2c1CN(C(=O)COC1CCC1)CC2 O=C1NCC2(CC(N=c3[nH]c(N4CCOC(CF)C4)nc4ccc(Cl)cc34)C2)O1 N1(C(CN(c2ncc(Br)cn2)C)=O)CC2CCC(NC(=O)OC(C)(C)C)C2C1 N1(C(c2nccc(CC)c2)=O)CC2CC(NC(c3ccc(F)nc3)=O)CC2C1 N1(C(C2CC(SC)C2)=O)CC2(C1)CN(C(c1csnc1C)=O)CC2CO C(=O)(CC(C)(C)CNC(c1csc(CCOC)n1)=O)NC1CC(CC)C1 N1(C(c2c(CC)onc2C)=O)CCN(C(C2(CC)CCNC2=O)=O)C(COC)C1 C(CC1=CCN(C(c2ccc(C)c(Cl)c2Cl)=O)CC1)NC(C(CC)C)=O N1(C(CCCc2ccc(OC)cc2)=O)CC(NC(c2csc(O)n2)=O)CC1(C)C C1(c2n(CCCCCC)nnn2)(NCP(C)(C)=O)CCOC1C.c12cccc(c1)S2 N1(C(C(CCC)NC(=O)C=CC(=O)OCC)=O)CCCC2(C1)N=N2 N1(C(CCC(CC)OC)=O)CC2CCCC(C1)N2C(C1CC(CC)=NO1)=O C(=O)(C(C)(Cl)Cl)N(C)CCOCCCN(C)C(C1CC1(c1ccccc1)C)=O c1(C(=O)NC2CCC(CCNC(C3(CC)CCCC3)=O)C2)ncc(N)nc1C O=C1CC(=O)CC(C(N2CCC2CC(=O)NCCOCC(F)(F)F)=O)C1 C1(C(N2CCC(O)(CNC(CN3C(C)CC3)=O)CC2)=O)CC2CC1CC2(F)F O=C(N=c1c(Br)c[nH]cc1Br)C1(O)CCN(Cc2ccc([N+](=O)[O-])o2)C1 c1(N(C(C)CNC(c2ccnn2-c2ccccc2)=O)C)cc(Cl)nc(S(C)(=O)=O)n1 c1(CCC)cc(C(=O)NCC(O)CNC(=O)C(C)C(F)F)c(C)o1 c1(C(=O)NC(C2CCCC2)CNC(C(C)SCC)=O)cccn2c(C)cnc12 C12(C(=O)NC(c3ncc(C)[nH]3)CC)CCCC1CCN2C(=O)Cn1nc(C)nc1C C1(C(=O)NC(N(CCC)CCCCOCCC(=O)N)=O)CC(F)C(=O)N1.C1(=C)CC1 C(CCN(C(=O)CC=C(C)C)C)(C(C)C)NC(C1C(C(=O)OC)CC1)=O N1(C(C2(C)CC(C)OCC2)=O)CCCC2(C1)CN(C(=O)CSc1ccccc1)C2 CCCCC(C)(F)C(=O)NC(C1CN(C(=O)CC2CC(SC)C2)C1)C CC1(C)CCC(C(=O)NC2CCC2NC(=O)C(O)CCc2ccccc2)CC1 c1(C(N2CCC(C)(NC(c3nc(CC)oc3C)=O)C2)=O)cncc2ncccc12 c1(C(N2CC=C(CNC(C(C)NC(N)=O)=O)CC2)=O)cnn2c1C(=O)NCC2 Cc1nc(O)sc1C(=O)NC1COCC1CNC(c1c[nH]c(=N)o1)=O N1(C(CCCCCCC)=O)CCCC2C(NC(c3ocnc3CC)=O)C(C)(C)C12 c1(C(N2CCN(C(c3c(C)nnn3C)=O)C3(C2)CC3)=O)c(F)ccc2nc[nH]c12 O=C(NNc1ncc(F)cc1F)Sc1ccnc2[nH]nc(C(F)(F)F)c12 N1(c2cc(Nc3c(CC)ncnc3)nc(C(C)C)n2)CCn2ncc(C)c2C1 N1(C(C2N(C)CC(C)(C)C2)=O)CCC2OCCN(C(c3cc(=O)cc[nH]3)=O)C2C1 c1(-c2nc(CCCCC)nn2CCCO)cnc(N(C)C)c(Cl)c1 c1(C(=O)NC(C)CNC(=O)CC(C)(F)F)cc(S(N)(=O)=O)cc(Cl)c1F N1(C(c2c(C)coc2C(C)C)=O)C(C)CC2CN(C(=O)CNC(N)=O)CC12 C1(NC(C=CC(C)NC(C2(N(C)C)CC2)=O)=O)C2CCCC1CC2 C(=O)(C(C(C)O)NC(=O)Cc1ccsc1)NCc1c(C(C)C)con1 CN1CCc2nc(C(=O)NC34CCC3CN(C(=O)C(F)n3cccn3)C4)sc2C1 CCC(CC)CC(=O)N1CCC(N2CCC(NC(=O)C(O)C(C)CC)CC2)CC1 CC1CCOCCN1C(CC1CCCC1)C(=O)NCCN(C)C(=O)OC(C)(C)C C=C(Cl)CC(C(=O)N(C1CC2CC2C1)C)NC(c1ncc(C)cc1F)=O N1(C(c2cn(CC)nn2)=O)CCCCC(C(N2CC3CCC3(C)C2)=O)C1 Cc1ccc(C(=O)NCCCCCNC(c2cc3occc3s2)=O)c2c1CCC2 C(F)(c1ccccc1)=CC(=O)N(C1CN(C(=O)C(C#N)C2CC2)CC12CC2)C C#Cc1cncc(NC(=O)C(O)CCCNC(=O)C(C)SC)c1 CC1CCN(C(=O)Cc2csc(N3CCC(O)CC3)n2)CCN1C(=O)CCC#N c1(C(=O)NCC(C(C)(C)C)NC(=O)CCCn2ccnn2)cc(F)c(F)cc1F C12(C(=O)NC3C(CN(C)C)CCC3)CC(CCO1)N(C(C1CCC1(F)F)=O)C2 c1(CNC(COC2CCN(C(c3c(CC)cco3)=O)C2)=O)cccc(CO)c1 C1(C(N(CCC(=O)NCc2cc(CC)n[nH]2)C(C)C)=O)CCC(CC)CC1 c1(SC(CC)C(N2CC(O)CC2C(=O)OC)=O)cc(F)ccc1F C1(CCC)CN(C(C2C3CC(=O)CC23)=O)CC1CO.C1=CC(=O)NC(C)(C)C1 Cc1n[nH]c(C)c1CC(=O)NC1(CNC(=O)CCOCC(F)(F)F)CCOC1 C1(S(N)(=O)=O)(C(N2CC3C(NC(C4N(C)CC(O)C4)=O)(C3)C2)=O)CCCC1 c1(C(N2CC3CC(C2)N3C(c2c[nH]c3cnccc23)=O)=O)c[nH]c2ncccc12 CC1CC(CO)N1C(c1ccc(CNC(c2csc(=N)[nH]2)=O)o1)=O c1(N2CC(CC=C)(NC(=O)CCc3ccccc3F)C2)cc(C(N)=O)nc(Cl)n1 c1(C(=O)NC(C(C)C)(C)CNC(=O)C(C)S(C)(=O)=O)nn2cccnc2c1Cl N1(C(CC(C)NC(c2ccccc2)=O)=O)CCN(C(=O)C(F)(F)C2CC2)CC1C S(=O)(=O)(c1c[nH]c(C(N2CCCC(NC(C3(F)CCS(=O)(=O)C3)=O)C2)=O)c1)NC C#CC(CNC(=O)CC(C)NC(=O)C=CC(C)CC)C(C)C Cc1cc(Cl)ccc1C(=O)N(C1CCCN(C(=O)Cn2cnc(C#N)n2)C1)C c1(C(=O)N(C2CCO2)Cc2cccs2)ccccc1 c1(NC(N2CCCN3CCCC23)=O)cccc(P2(=O)CCCC2)c1 N1(CCC(F)(F)F)CCCC(N=c2ccnc(N3Cc4cccc(Cl)c4C3)[nH]2)C1 CC1CN(C(=O)C(O)(c2ccccc2)C2CC2)CCN1C(C1CCC(O)C1)=O c1(-n2cc(C(CC)C(N3CCCC(OC(C)C)C3)=O)nn2)cc(C)ccc1OC C1(NC(c2ncc(OCC)nc2)=O)C(C)CN(C(=O)Cc2scnc2C)CC1C Cc1cc2sc(C(=O)NC3CCN(C(=O)Cn4ccnn4)C3(C)C)cc2s1 C1(CC(N2CC(NC(=O)CCc3ccco3)CC2C)=O)(CC)CCOCC1 C1(C(=O)N)CCC(=O)N1CC.C(CC(=O)NCC(C)(C)OCCCCC)S S(=O)(=O)(c1ccc(N(C)Cc2ccoc2)cc1Cl)NC(CCOC)C(C)(C)C N1(C(C2(C)C=CCCC2)=O)CCC(C(=O)N2CCC(c3cc[nH]n3)C2)=C(F)C1 N1(C(C(=O)NCC)=O)CC(C)C(NC(c2ccc(-c3cccs3)cn2)=O)C(C)C1 C1(C(N(C(C(=O)OC)C)C2CC2)=O)CCC(c2ccc(C)cc2)CC1 c1(CNC(c2cc[nH]n2)=O)c[nH]nc1C(=O)N(CC(F)F)CC1CC1 N1(C(c2c(OC)n[nH]c2)=O)CC(NC(C2CCCN2C2CC2)=O)C2CCCC12 c1(SCC2(C)C(NC(=O)OC(C)(C)C)CC2)cnc(O)c(CO)c1 C1(NC(C2CCC(NC(CCC(C)OCC)=O)C2)=O)CCOC(C)(C)C1 N1(CC(=O)Nc2c(C(C)C)ncs2)CC(O)C(O)C12CCC2 N1(C(=O)OCCOC)CCN(N2CCCC(c3cnco3)C2)CC1 CC1CN(C(=O)CC2C=CCC2)CCC1NC(c1ccc(Cl)c(O)c1)=O N1(C(c2cnc(C)c(C#N)c2)=O)CC2(CCN(C(=O)Cn3cnnc3O)CC2)C1 c1(NC(CCN(C(CC)CC)C2(CC(=O)OCC)CCC2)=O)cnn(C)c1 C1(NC(C2(SC)CC2)=O)C=CCN(C(=O)Cc2ccccc2F)C1 c1(C(C)C)cncc(C(=O)NC(C)(CNC(c2ncccc2Cl)=O)C(C)C)c1 C1(F)(CNC(C2N(N=O)CCC2)=O)CC2CCC(C1)N2C(C1CC2(CC2)C1)=O c1(C(=O)NCC2CN(C(C(COC)C)=O)CC2O)cc(F)cc2cccnc12 C(=O)(C(O)(C(C)C)C(F)(F)F)NCC(CO)NC(CCCc1cc(C)no1)=O Cc1ccc(C(N2CCC(NC(c3oc(Br)cc3C)=O)C(F)C2)=O)cc1Br C1(CC(=O)NC2CN(C(C(C)(C)N(C)C)=O)CC2F)CC(c2ccccc2)=NO1 C=CCC(C(=O)NC1(CN(C)C(c2cnc(OC)s2)=O)CC1)C(C)C C1(NC(=O)Cc2ccc(C3CC3)cc2)COCCN(C(=O)C(O)C2CC2)C1 CC1(C)CCC(O)(CNC(C2COCCN(C(=O)C=CCN3CCCC3)C2)=O)C1 CC1CN(C(C2C3CCC2CC3)=O)CCC1NC(C1(n2cccn2)CC1)=O c1(C(=O)NC2CCCN(C(c3ccc(OC)c(N)n3)=O)C2)ccc(S(C)(=O)=O)o1 C(=O)(CC(O)C(C)(C)C)N(CC(C)NC(c1ccc(OCC)cc1)=O)C CC1CN(C(c2ccsn2)=O)CCN1C(=O)C(C1CCCCC1)F C1(C2CCCN(C(c3cc(Cl)sc3Cl)=O)C2)(NC(=O)CCc2ncc[nH]2)CC1 N1(C(C2=CCCN(C(C=C(C)c3ccco3)=O)C2)=O)CC(C)NC(=O)C12CC2 c1(C(=O)OC)ccc(OC)cc1C(=O)NC1CCCCN(C(=O)CC2(O)CC2)C1 c1(C(=O)NCC(=CC(=O)NCC2(SC)CC2)C)cc(F)cc(F)c1 C(=O)(CC(C)(C)CC(F)F)NC1C(F)CCN(C(CC2CCC(C)(C)CO2)=O)C1 CCCCC(F)C(=O)N(CC(C)NC(=O)C(C)c1ccco1)CC C(CCC(C)C(=O)N(C1CCCCN(C(=O)CCc2csc(=N)[nH]2)C1)C)OC CC1CC=CCC1C(=O)N(C1CCN(C(=O)Nc2cc(Cl)c[nH]2)CC1)CCO c1(C(N2CC(NC(c3cc(SC)oc3)=O)C(OC)C2)=O)cnc2n1CCC(C)C2 CC1(C)CC(=O)NCC1C(=O)Nc1cccn1Cc1cn(CC2C3CCCC23)nn1 C1(C(N(C2CCN(C(CCC=CCC=C)=O)C2)C)=O)CC2(CCC2OC)C1 C1(C(=O)NCC(C)CC(F)(F)F)(OC)CCCN(C(C)C(=O)N(C)C)C1 C(C(O)C(=O)NC(c1cnn(C)c1)C(=O)N(C1CCC1O)C)=CC C(=O)(C(C)C(F)(F)C(F)F)N1CCC(N(C(C2(C)CCNC(=O)C2)=O)CC)CC1 C1(CNCc2scc(COCC)c2)Cc2ccccc2N(C(=O)OC(C)(C)C)C1 c1(C(=O)NC2C(CNC(C(CC)C(C)C)=O)CC2)ccc2c(c1)NC(=O)CS2 c1(C(C)C)ncc(Cl)c(C(=O)NC2CC23CC(NC(c2ncncc2Cl)=O)C3)n1 C1(C(N(C(C(C)C)CO)C)=O)CN(C(C2COCCO2)=O)CC1(C)C c1(C(=O)NCC2CC(OC)CN2Cc2ccccc2)ncc(Cl)cc1F c1(C(=O)NC2C(NC(C(C(CC)C)O)=O)CCC2)cc(F)c(F)cc1OC Cc1[nH]c(C(N2CCCC(C)CC2)=O)c(C)c1C(=O)NCc1csc(C#N)c1 C#Cc1cnc(N2CC(=C(F)CNC(=O)CCc3ccccc3C(N)=O)C2)nc1 C1(O)(C(=O)NCC2CC(NC(C3(CCC)CC3)=O)C2)CCc2ccccc2C1 N1(C(C2C(C(=O)OC)C2)=O)CCC1C(=O)NCC1(CC)CC1 C1(C(=O)NCC(C2CCCCC2)NC(C(CC)F)=O)CCN(CCO)C(=O)C1 C1(CC(=O)NC2CC(NC(=O)CSc3ccccc3)C2)CCCCC(=O)N1 C(=O)(C(C)C(C)S(C)(=O)=O)N(CCCNC(C(C(CC)(C)C)=O)=O)C C(=O)(CN1C(=O)COc2ccccc21)NCC1(C)CN(C(C(C)O)=O)C(C)(C)C1 c1(OC)ccc(CC(N2CCC(=O)CC2C(=O)O)=O)c(Cl)n1 c1(C(=O)NC2CN(C(Cn3cc(C(C)=O)nn3)=O)CC2O)ccc2nccn2n1 N1(c2ccc(S(=O)(=O)N(C(C)C)C)cc2)CCc2c([nH]c3ccccc23)C1 N1(C(CC=C)=O)CCC(NC(c2cc(O)n(CC)n2)=O)CC1 c1(CC(=O)NCCC2CCCN(C(C3CC(C)(F)C3)=O)C2)noc2ccccc12 N1(C(c2c(C)nc(C)s2)=O)CC2OCC(NC(=O)CCOCC(F)F)C2C1 c1(C(N(C)CC2N(C(c3c(CC)onc3)=O)CCC2)=O)nsc2ccccc12 Cc1cc2cc(C(=O)NCC3CC(C)(C)CN3C(=O)CCC(F)F)oc2cc1C c1(C(=O)NC2C(NC(C(CCC)N(C)C)=O)C2)c(N)ccc(Br)c1F C1(C(C)(C)O)(CNC(c2ccnn2C2CC2)=O)CN(C(=O)CC2CC(F)(F)C2)C1 c1(NC)cnc(Cl)cc1C(=O)NC(C1CN(C(=O)C2=C(C)OCC2)CCO1)C c1(C(=O)NC2C(CNC(c3cn(CCC=C)nn3)=O)C2)onc(OC)c1Br O=C1CC2(CN(C(c3noc(-c4ccc(F)cc4F)n3)=O)C2)C(O)CN1 N1(C(COc2cccc(C)c2)=O)CCC(C)C(NC(=O)C=CCCC(C)C)C1C CC1CC(NC(=O)CCCn2cncn2)CN1C(=O)C=CCF C1(CCCNC(Cn2c(C)nnn2)=O)CN(C(c2cc(O)nn2C)=O)CCO1 c1(C(=O)NC(C2CCCCO2)C#C)cc2n(c1)CCCC2 Nc1ncc(C(N2CC(F)(F)CC2CNC(=O)Cc2cnc[nH]2)=O)cc1CO C1(C(N2C(C)(C)CC(NC(c3cnn4c3CCC4)=O)C2)=O)CNC(=O)CC1(C)C CC(C(=O)NCCC1(O)CCN(C(C2(c3ccno3)CC2)=O)C1)C(F)(F)F C1(OC)(CNC(c2ccc(C)c(Cl)c2)=O)CCN(C(=O)CCc2c[nH]c(=N)[nH]2)CC1 c1(NCc2cc(C)oc2Br)ccc(C)c(Br)c1 C12(C(=O)NC3CCN(C(C=CCC)=O)CC3(C)C)CC3CC(C(=O)N1)C2C3 C=CC(C)(O)CC(=O)N(C1CCN(C(=O)COCCCC)C1)CCC c1(C(=O)NC(CCCNC(CCN(CCC)C)=O)C)ncnc(C)c1OC C(N=c1[nH]c(Cl)ncc1F)C1N(C(C2(COC)C=CCC2)=O)CCCC1 CC(CSC1CC(OC(F)F)C1)C(=O)OC(C)(C)C CC1(C)CC(CNC(=O)Cc2c(Cl)cccc2Cl)N(C(=O)CC2(O)CCOC2)C1 c1(C(=O)NCC23CC2CN(C(C2CCCCO2)=O)C3)cc(O)nc(C2CC2)n1 C1(OC)CC2(C1)CC2N(C(=O)NCc1ccc(C)cn1)Cc1ccco1 N1(C(C2(C(C)C)N(C(CC(CC)CC)=O)CCC2)=O)CCCN2CCCC2C1 C1(NC(C2C(C=C)C2)=O)CCC(NC(=O)C(c2ccc(OC)cc2)O)CC1 C1(N(C(C2C3(CC3)C23CC3)=O)CC)CCCN(C(C2CC2C(C)(F)F)=O)CC1 Cc1cc(Br)cc2[nH]c(C(=O)NC3CC(CCNC(=O)C(C)(C)O)C3)cc12 C(c1cccnc1C)=CC(=O)NC1CCN(C(CN(C)CC)=O)C1C1CC1 CC1(C)CCC1C(=O)NC1COCC1NC(c1nscc1Br)=O N1(C(C=CC(=O)OC)=O)CCC2(CC1)CCN(C(c1cn(C)nc1OC)=O)C2 C=CCC(CO)NC(=O)CC1CCN(C(=O)C(C)CN(C)C)C1 c1(C(=O)NCC(CNC(CCc2nc(C)c(C)[nH]2)=O)O)ccc(Cl)cc1O CN=c1[nH]cc(C(N2CC(OC)C(NC(=O)C(n3ccc(C)n3)C)C2)=O)s1 C(=O)(C1=NOC(c2ccccc2)C1)N1C(CC(=O)NCc2cc[nH]n2)CCC1 CC(C)CC(C)CC(=O)N1CCC(CNC(c2cccnc2C2CC2)=O)C(C)C1 Cc1onc(C(F)(F)F)c1C(N1CCC(NC(c2nncs2)=O)C1)=O C1(C)(C(=O)NC2CC(F)(CNC(c3cn(CCC)nc3)=O)C2)CCCC1O C1(NC(c2csc(C)c2C2CC2)=O)COC2C(NC(=O)C(C)(C)N(C)C)COC12 c1(C(C)=O)nc(C(=O)N(C(C)CCNC(=O)Cn2ccc(C(F)(F)F)n2)C)cs1 CC1CCCCC1OCC(=O)NCC1CCN1C(c1cnc(C2CC2)[nH]1)=O c1(C(N2C3(C)CC(C2)OCC(=O)NC3)=O)ccn2cccc2c1.C(C(F)F)OC C1(C(=O)NCCCN(C(C)C)C(C2COC(=O)O2)=O)CC12CCOCC2 N1(C(CCSCC)=O)CCC(C(N2CCCC2n2ccnc2)=O)C1 C1(CNC(CCSC)=O)CC(C)N(C(=O)CNC(c2cccc(F)c2)=O)C1 C(CC(CO)NC(=O)CCN(C(=O)C(C)n1cccn1)C(C)C)SC c1(CC(=O)NC(C2CC(F)(CNC(=O)C=CC(F)F)C2)C)cnc2n1CCCC2C C1(CC(=O)N(C2CCCC2)CCNC(CCOCC#C)=O)CCCC(OC)C1 C1(C)(CNC(Cc2cc(CC)no2)=O)CCCN1C(c1ccc(CCO)cc1)=O c1(C(N2C(CNC(Cc3cc(OC)no3)=O)C(C)CC2)=O)cc2ccccc2o1 N1(C(C2CCN(C(c3c[nH]c(=NC)o3)=O)C23CC3)=O)CC(C)(C)OCC1C C1(CNC(C2(C)C=CCCC2)=O)CN(C(=O)CCC(CF)CF)CC12CCC2 c1(C(N2CC(C)C(NC(=O)C3=NNC(=O)C3)C2)=O)cc(Cl)nnc1Cl N1(C(C(C(CC)O)C)=O)CC2CCOC2(CNC(=O)CCc2cc(OC)no2)C1 CN1C(=O)CC(C(=O)NCC2CCCN(C(=O)Cc3nn(C)cc3Cl)C2)NC1=O C1(CC)(NC(C2CCCC2CNC(C2COCC(C)O2)=O)=O)CCCCCC1 c1(C(=O)NCCN(C(=O)C(C)(F)C(=O)OC)CCC)cc(C)cc(C)c1 N1(C(=O)C(Cl)(Cl)Cl)CCOCC(NC(c2cnc(-n3cccn3)cn2)=O)C1 C1(C(=O)NCc2occ(C(=O)NCC3(CO)CCN(C)C3)c2)CCC(O)CN1C C(=O)(C1=CCC(C)(C)CC1)NC(CC#C)C(=O)NCC=CC(C)(C)C CCC(C)(C)C(C(=O)N1CC2CCN(C(c3sc(C(C)C)nc3C)=O)C2C1)OC c1(C2(C(=O)NC3CC3)CC2)noc(-c2cn(C3CCOCC3)nn2)n1 n1(CC(=O)N(C)CC2CN(C(=O)COCC(F)F)C2)cnccc1=O CC(C)(N=[N+]=[N-])C(=O)NCC1(CNC(=O)C(F)n2ccnc2)CCC1 c1(C(=O)NCC(C)(C)NCC(c2ccsc2)C)cc[nH]c(=N)c1 C1(NC(c2sc(C)c(O)n2)=O)C(C)CCN(C(c2ccc(C)n2C)=O)C1C C1(C(N(C(C)=O)C)C)CCN(C(=O)CC2(CO)CCC2)CC1.C1CCC(=O)N1 C(CC(C)(C)C)(C(=O)N1CCOC(C#N)C1)NC(C(C=C=C)C)=O c1(OCC(=O)NCCC(CCOC)NC(C)=O)ccc(=O)n(CC(F)(F)F)n1.C(C)(=O)O c1(CNC(C(CNC(Cc2c(C)ccs2)=O)CC2CCCC2)=O)ccc(F)cc1O C1(C(N2CCC(O)C(CO)C2)=O)(COC)CCN(C(c2cnc(C)cn2)=O)CC1 c1(OC)cnc(C(=O)NCC23CC2CN(C(=O)C2=CCCCC2)C3)c(OC)n1 Cc1ccc2c(CN3CCC(NC(c4ccc(Cl)c(C)c4)=O)C(F)C3)c[nH]c2c1 C12(NC(c3coc4c3CCCC4)=O)CCC(CN(C(=O)C(F)n3cccn3)C1)C2 C1(C(=O)NC(C)Cc2ccco2)CC(NC(=O)COCC(F)F)C(O)C1 n1(CCC(C)(C)N)c(N2CCCC2)nnc1-c1ccc(C(N)=O)cc1.CSC C1(NC(C2CCC(F)(F)C2)=O)CN(C(c2nc(Cl)cs2)=O)CCC1O C1(CCNC(c2n(CC)ccn2)=O)CSCCN1C(c1cn(C2CCC2)nn1)=O CC(CC1=CCCCC1)NC(=O)CC1(CNC(=O)Cc2ccsc2)CC1 C#CCC(C(=O)N1CCC1C(=O)NCC(C)(C)C1CC1)C1CC1 c1(C(=O)NCCC(=C)CNC(c2oc(SC)cc2C)=O)c(C)ccc(C)c1C C1(CNC(C(C(C)O)(C)C)=O)CCN(C(=O)C(C2CC2)C2CC2)CCC1(F)F N1(C(COc2ccc(C#C)cc2)=O)CCC2C(C1)CN2C(c1ccoc1Cl)=O c1(C(=O)NC(CNC(CCCc2onc(C)n2)=O)CO)cc(Br)cnc1N N(C1CCOc2ccc(Br)cc21)C(C(N)Cc1cc(Cl)cc(Br)c1)=O Cc1nc(C2C(C(=O)NC34CC(NC(c5cn[nH]c5)=O)(C3)C4)C2(C)C)n[nH]1 N1(C(c2nn(CC)c(O)c2)=O)CC2(CC(NC(c3nc(O)c(C)s3)=O)CO2)C1 c1(CSCC(=O)N(C2CN(C(=O)Cc3nccn3C)CC2F)C)ccccc1Cl C1(NC(C(C)(C)NC(=O)NCCC)=O)C(C2CC2)CC(N=c2[nH]ccnc2F)C1 c1(C(=O)NC2CN(C(C(CSC)(C)C)=O)CC(O)C2)ccc2nc(O)sc2c1 C1(F)(CNC(c2ncc(Br)cc2F)=O)CCN(C(c2cc([N+](=O)[O-])cs2)=O)CC1 C1(NC(CC(C)(F)F)=O)COC2C(NC(=O)CC3(C)CC(F)(F)C3)COC12 Cc1cc(C(=O)NCC(=O)NCCOCCNC(=O)C(C)(C)C)ccc1C(F)(F)F Cc1[nH]nc(C(N2CCC(C(C)C(=O)N(CC(C)O)C3CC3)CC2)=O)c1O c1(C(N(CC(=O)N(C2CC2C)C)CCOC)=O)cn(C2CC2)cn1 C(=O)(CC1=NNC(=O)C1)NCC1N(C(Cc2c(C)nc(S)s2)=O)CCC1C c1(Cn2ncc(C(=O)NCCN(C(=O)CCCF)CCC)c2)ccccc1F c1(NC(CC2N(C(CCN(CC)CC)=O)CC2)=O)cccc(Cl)c1C Cc1nn(CC(N2CC3CC3(CNC(=O)C(C)CN(C)C)C2)=O)c(C)c1Br C1(CC)COCCN(C(C2CCN2C(C2(C)COC2)=O)=O)C1 C1(CCNC(c2c(C)nn[nH]2)=O)CN(C(=O)Cc2cncc(O)c2)CCS1(=O)=O c1(C(N2CCC(NC(C3C(COC)CC3)=O)C2)=O)cc(Cl)cc(Cl)c1OC c1(NC(C)=O)c(F)cncc1F.c12ccnc(c1)C(=O)N(C)C1CCN(C1)C2=O C1(C(=O)NC2CCC3CCN(C(CCCOC)=O)C32)CCc2nc(=N)[nH]cc2C1 c1(C(N2CCC(C)(CNC(c3cc(OCC)n[nH]3)=O)C2)=O)c(F)cccc1F C1(C(N(C(CC)COC)C)=O)CCOC1CNC(c1c[nH]nc1Cl)=O c1(C(N2C(C)CC(NC(=O)CCC#N)C2)=O)cnc2[nH]cnc2c1 c1(C(=O)NC(CN(C(=O)CC(=O)NC2CC2)CC)C)coc2cc(F)ccc12 C1(C2CCN(C(c3cnc(C(C)(C)CF)o3)=O)C2)(NC(C(CC)SC)=O)CC1 c1(CNC2(c3n(CCC)nnn3)CC3COCC23)cc(F)ccc1NC1CC1 c1(C(=O)NCC(CC=C)NC(=O)C(F)(F)COC)ccc(C)c(S(N)(=O)=O)c1 c1(SC)ccc2cc(C(=O)NC3CC3NC(C3OCC4CCCC34)=O)[nH]c2c1 c1(C(N2CC(N(C(C)(C)C)C(C3C(C)C3)=O)C2)=O)nc(N)cc2ccccc12 C12(C(=O)NCC3C(C(C)C)C3)C(NC(c3ccc[n+]([O-])c3)=O)C3CC1C2C3 c1(C(=O)NCC(CC(C)C)NC(=O)COCC2CC2)ccc([N+](=O)[O-])n1C C1(C)(C(=O)NCCCCCCN(C(c2n(C(C)C)ncc2)=O)C)CCOC(C)C1 c1(C(C)NC(C(CNC(C2N(C(C)=O)CCC2)=O)C)=O)ccnc(F)c1 c1(CC(=O)NCC2CC(NC(c3c(SC)ccs3)=O)CC2O)ccc2c(c1)CC2 N1(C(CCCCc2ccc(OC)cc2)=O)CCC(C2(NC(=O)CC3CC3)CC2)C1 C1(C(=O)NCCSC(C)C)(CC2CC2)CCCN1C(=O)CC(=O)N(C)C C1(CNC(c2csc(F)c2)=O)CC2(CC2)CN1C(c1cc(Cl)ccn1)=O C(C)(CC(=O)N(CCNC(C1(F)CCOC1)=O)C(C)C)SC C(N=c1[nH]c(=NCCOCCC(C)C)c2c(F)cccc2[nH]1)c1c(C)cc(Br)nc1 Cc1cc(C(N2C3CN(Cc4ccc(-c5ccccn5)cc4)CC23)=O)c(C)[nH]1 N1(C(c2cc(CC)c(C)s2)=O)CCC(NC(c2cc(C)c(F)cn2)=O)C(CO)C1 Cn1cc(C(N2CCC(CO)C(NC(=O)CCC3CC3)C2)=O)c(O)nc1=O c1(C(=O)NC23CCN(CC4CCCC(C)C4)C2CCC3)noc2c1CCCCC2 c1(OCC(=O)NC(C)CCCNC(=O)C(C)CC2CCCC2)ccc(CO)cc1 Cc1sc(=O)n(CC(N2CC(N(C)C(c3nc(=O)n(C)[nH]3)=O)C3(CC3)C2)=O)c1C c1(C(=O)NC(CCN(C(c2cccc(C(C)=O)c2)=O)C)C)ccc(N=[N+]=[N-])cc1 N1(C(c2ccc(OC)nn2)=O)Cc2ccccc2C(NC(C2(F)CCOC2)=O)C1 C1(CC(N2C(C(C)NC(C3CC(F)(CO)C3)=O)CCC2)=O)CCC(F)(F)CC1 N1(C(C(C)OC(C)=O)=O)CCC(O)(CNC(c2cc(C)ns2)=O)C1 C(=O)(C1=NOC(C)C1C)N1CCC(OCCNC(C(C(C)C)SC)=O)CC1 c1(CC(C)C)cc(C(=O)N(C)C(c2cn(CC3(F)CCOC3)nn2)C)n[nH]1 N1(C(C=CCOCCOC)=O)CC(NC(c2cc3sccc3[nH]2)=O)CCC1C c1(C(C)CC(=O)NCC(C)(C)CN(C)C(c2cscn2)=O)ccc(F)c(F)c1 CCCC(C)(C)C(=O)N1CCCC(CCNC(=O)CCCOCC)C1 c1(C(N2CCC(N(C)C(c3snc(O)c3Cl)=O)C2)=O)nnn2c1C(=O)NCC2 C(=O)(C1CCC(=O)c2cccn21)NCC1N(C(c2cn(C)nc2)=O)CCCC1 c1(C(C)NC(=O)N(CC(O)CO)CCN)ccc(OCC(F)(F)F)cc1F C1(C(N2CCC(C(F)F)(CNC(c3ccc(=N)[nH]c3)=O)C2)=O)CC2CCC(C1)O2 C1(F)(CNC(c2cn(CC=C)nn2)=O)CCCN(C(C2(C)CCCS2(=O)=O)=O)C1 N1(C(c2c(C)nn(-c3ccccc3)c2Cl)C(=O)NC)CCOCC(CN(C)C)C1 C1(NC(=O)CN2CCCC2=O)CN(C(C2CCSCC2)=O)C2CC12 N1(C(C(CC2CC2)OC)=O)CCOC(CC(=O)NCC(C)(O)C2CC2)C1 N1(C(C2C3CN(C(C(C)OC)=O)C2C3)=O)CCCN(C)CC1C N12Cc3ccc(cc3C1)C2=O.C1(C(C)C)(NC(=O)C(C)n2cccc2)CCC1 Cc1ccsc1C1CC1C(=O)NC(C)CNC(=O)C(C)SC1CN(C(C)(C)C)C1 c1(CC(=O)NCC2CCN2C(c2nc(Br)c[nH]2)=O)ccc(F)cn1 CCCCCC(C)CC(=O)N1CC2(CC(CC(=O)NCCC(C)SC)C2)C1 c1(CC(=O)N(C2CC2)Cc2cccc(C(F)(F)F)c2)cc2ccccc2c(=O)o1 C1(C)(C(=O)NCC(C)Cc2cn[nH]c2)CC(O)CN1C(c1ccn(C(F)F)n1)=O c1(C(=O)NC2C(N(CCC(=O)NCc3ccccc3)C)C2)cc2ccccc2o1 c1(OC)ccccc1C(C)NC(=O)CC1CCN(C(c2ccncn2)=O)C1 c1(C(N2C(C)(CC(=O)N(C3CC(C(N)=O)C3)C)CC2)=O)cnn2ccccc12 C1(NC(CCCC=C)=O)CC2(C1)CN(C(=O)C(C)S(N)(=O)=O)C2 c1(C(N2CC=C(CC(=O)N3CC4CCC3C4)CC2)=O)cnc2ccccc2c1 C1(CNC(c2cc(C)ns2)=O)CN(C(c2cc3ccsc3s2)=O)C2(CCC2)C1 N(C(=NCc1cc(CC(=O)OC)on1)N1CCC(C(C)(C)C)C1)C(CC)C CCCC(C)(O)C(=O)N1CC(NC(c2cc(OC)ns2)=O)C(SC)C1 c1(CN(C2CC2(Cl)Cl)S(C)(=O)=O)c(C(F)(F)F)oc2ccccc12 N(C(=NCC(Cl)C(F)(F)F)NCc1sc(N2CCCC2)nc1C)Cc1cc(C)on1 C1(C)(C(N2C(CN(C(=O)CC3(COC)CC3)CC)CCC2)=O)CCC(F)(F)C1 Cc1ccc2c(C(=O)NCC3CCCN3C(=O)C(C)CC(F)F)ccnc2c1Cl N1(C(C(C=C=C)C)=O)CCC(C=C)(C(=O)NCC=Cc2ccccc2)CC1 c1(CN(C)C(C2(NC(=O)CCn3cnc(=N)[nH]3)CC2(C)C)=O)cn(C)cn1 N1(C(Cc2cnc(C)[nH]2)=O)CCC(CNC(=O)C(C)C(F)(F)F)C12CC2 C1(C)(C(COC(C)(C)CNC(=O)OC(C)(C)C)=O)CCCO1.C1COC1 C=CC(C)(CCOC)C(=O)NC(CNC(c1cncc(C(C)C)c1)=O)C(C)(C)C N1(C(c2ccc(CC)[nH]2)=O)CC(NC(=O)C(C)CC(C)CC)CC12CCOCC2 O=C(C1=CN2CCS(=O)(=O)N=C2C=C1)NC1CCN(C(=O)C2=CCCOCC2)C1 C=CC1(c2cn(CC3CNC(=O)O3)nn2)COCCN1C(C1CC12CCC2)=O C1(N2C(=O)C(C)NC(=O)C(C)CC2)CCCCC1.C1(C(=O)N(C)C)CC12CC2 N1(Cc2c(C)cc(OCC#C)cc2C)CC(C)(C)C1C1CCCO1 N1(C(=O)OC)CCC(N=c2nc3scnc3c(N3CCC=C(c4ccco4)C3)[nH]2)C1 N1(C(c2cccc(SC)n2)=O)CC2CC(NC(c3ncc(Cl)s3)=O)CC1C2 c1(C(=O)NCC=CCNC(=O)Cc2cccnc2)cnc(Cl)c(Cl)c1 C1(CNC(c2csc(Br)n2)=O)CC2OCCC2N(C(=O)Cn2ccccc2=O)C1 c1(C(=O)NCC=CCNC(COCCCC#C)=O)cn2c(n1)COCC2 C=Cc1cnn(C)c1C(=O)NCC1CCCCC1NC(=O)CCCC(=O)N(C)C CCC(CC)CCCC(=O)N1CC2OCC(NC(=O)CCc3cncn3C)C2C1 c1(C(N2CCC(CC)(NC(=O)C(C)CC(F)F)CC2)=O)cc2c(s1)CCSC2 C#Cc1cc(C(N2CC(NC(c3ccnn3C=C)=O)CC2C)=O)cc(Br)c1 C(=O)(CCC(=O)NN(C)C)NC(CCCNC(CN(C1CC1)CC)=O)C C(=O)(CC(=O)N(C)C)NCC(C)(C)Cn1cc(C2CN(OC(CCC)=O)C2)nn1 Cc1ncc2n1CCN(C(=O)C(CNC(=O)CC1CC(=O)NC1=O)CC(C)C)C2 C(CCCCCN=c1[nH]c(Cl)ncc1C1CC1)NC(C1CCCC(C2CC2)O1)=O c1(CCC)ccc(C(=O)NC(C)(CNC(=O)C(C)N(CC)CC)C(C)C)cc1 N1(C(c2c(OC)cccn2)=O)CCN(C(=O)Cc2ccccc2Cl)C(CO)C1 N1(C(C=CC(C)=O)=O)CCOC(C(C)NC(C2(c3ccsc3)CC2)=O)C1 C1(CC)Oc2cc(Br)ccc2C1NCC(C)CC(F)F c1(OC)cccc2sc(C(N3CCN(C)C4CC34)=O)cc12 Cc1ccn2cnc(C(=O)N(C)CC3CN(C(=O)C(C)C(C)C4CCC4)C3)c2c1 c1(CC)ccccc1-n1nnnc1C(CCCSC)NCC.C1C(C(C)C)CO1 C1(NC(c2nccs2)=O)CC12CCN(Cc1ccc(O)c(O)c1O)CC2 C1(CC)(CNC(C2CCCC2NC(c2cc(Cl)n(C)n2)=O)=O)CCC(=O)N1 CCCC(CCCNC(=O)CCC(CC)OC)NC(=O)CCC1(C(=O)OC)CCC1 Cc1ccc(C(=O)NC(C2CC2C(=O)N(C)CC2CC2(F)F)C)cc1O C1(F)(CNC(c2cc(COC)[nH]n2)=O)CCC(CNC(=O)COCCCF)C1 N1(C(C=C2CCN(C)C2)=O)CCC2(CCC(CNC(=O)CC(C)(C)C)CC2)CC1 N1(C(C(C)=C2CCC2)=O)CCCC(CC(=O)NCCC2(C)N=N2)CC1 C1(NC(C2(SC)CC2)=O)CCCC(N(C)C(c2ccc(C(C)(C)C)[nH]2)=O)C1 O=C1CCC(C(N2CCC(O)C(NC(=O)C(O)C3CCCC3)C2)=O)CCO1 C(=O)(C#CC1CCOC1)N(CC(C(=O)NC1(CC=C)CC1)C)C N1(C(C(CC)N(C(=O)CC2(OC)CCC2)C)=O)CCOC(C)(CC)C1 Cc1ccc(F)cc1C(N1CC(CC(=O)NCC(O)C2CCC2)CC1C)=O c1(C(N2CC(OC)(CNC(c3cc4ccsc4s3)=O)C2)=O)cccn2ncnc12 Cc1nn2ccccc2c1C(=O)NCC1(F)CCC(NC(=O)C(C)N(C)C)C1 c1(C(=O)NCC(CNC(c2c(N)cc(C)cc2F)=O)C)ccc(F)c2ccsc12 c1(C(=O)NC(C=C)CO)ccc(CNC(=O)C=CC2(C)COC2)cn1 C(=O)(C(CN=[N+]=[N-])NC(c1ccn(C)c1C)=O)NCCn1c(C)nc(C)n1 C1(CCC)CCC(C(=O)NC2CC(NC(=O)C(N3CCC(C)C3)=O)C(O)C2)CC1 N1(C(C(C)SC)=O)CCC(F)(C(=O)NCC(O)C(C)C)CC1 CCCCCC(C)(C)C(=O)NCC1CCCN1c1nnc(C(C)(C)C)s1 N1(C(C=NOC)=O)CC2CN(C(c3cc4c(Cl)cccc4[nH]3)=O)CC2(C)C1 c1(C(N(CCC(=O)NCc2nncs2)C)=O)cccc[n+]1[O-] CC1CN(C(=O)COc2ccc(F)nc2)CCC1CNC(=O)CC1CCCC1 Cc1cc(Br)cc(C)c1C(c1nnnn1C(C)C)NCC=CBr C(=O)(C(C)(F)C(C)(C)F)N1C(C(N2CC(OCC)C2)=O)CC(=O)C1 c1(C(C(=O)NC(C)(C)C)N(CC(C)(C)OC)C)ccc(CC(C)C)cc1 c1(OC)cc(C(=O)NCC(C)CNC(=O)CC2CCOC2(C)C)sc1Cl CC#CCC(C(=O)N(CC(O)CO)C)NC(C1CCCS1)=O C(=O)(CCCC(=O)NCC1(C)CCN(C(c2ncncc2Cl)=O)C1)N(C)C C1(NC(C2(C)COC2)=O)CC2CCC1N(C(=O)C#CC1CCOC1)C2 c1(CC(=O)NCCN(C(C2(C#N)C(C#N)C2(C)C)=O)CC)cn2cc(C)sc2n1 c1(C(N2C(CC)CN(C(C3CCC(=O)N3)=O)CC2)=O)cc2cc(C)ccc2o1 c1(CC)cc(C(=O)NC2C3CN(C(C4CC(F)C4)=O)CC23)cc(N)c1 c1(C(=O)NCC2(F)CC(NC(C(COC)C)=O)C2)c(C(F)F)n[nH]c1C C(C(=O)N1CC(N(C(=O)COc2cc(C)on2)C)C(C)(C)C1)(C(C)(C)C)SC N1(C(C(CCC)c2ccccc2)=O)CC2(CCN2C(c2cnc(C)c(C)c2)=O)C1 c1(C(N(C(CNC(c2ccc(C(C)C)o2)=O)C2CC2)C)=O)cc(F)n(C)n1 c1(CC)cc(C(N2CCCC2CN(C(=O)C=C2CCSCC2)C)=O)no1 CCC1c2ccccc2CN1N1CC2(CC)CCCC2(CO)C1 CC1(CC(N2CC(OCCNC(C3CC3F)=O)C2)=O)CCCCCC1 c1(C(N2CC(CCNC(C(C)C3CC3)=O)C2)=O)ccc(=N)[nH]n1 C1(CCCNC(c2ncn(CC)n2)=O)CN(C(=O)CC2CN(C)CC2O)CCO1 C(=O)(C1=CC2C=CC1C2)NC1(C(NOCC=CC)=O)CCSC1 CCC(C(=O)OC)C(=O)N(CC(N1CCCC(COC)C1)=O)C1CC1 N1(C(C(=O)NC(C)C)=O)CCCC(CNc2cc(C(C)(C)C)on2)C1 C1(CC(N2CC3CC2CS3)C(=O)NC2COC2)CCCCCC1 N1(C(CN(C(C)C)C)=O)CC2C(C(=O)NC3CC(N(C)C(C)C)C3)C2C1 c1(C(=O)NC2(CC=C)CCCN(C(=O)C(F)C(C)C)C2)cc2c(C)sc(C)c2s1 C1(NC(C(C)SCc2ncccn2)=O)CC1C1CN(C(=O)C=CC(=O)N(C)C)C1 c1(C(=O)NC(c2ccc(C(F)(F)F)cc2)(C)C(N)=O)ccc(Cl)c(C(=O)O)c1Cl N1(C(c2c(CC)onc2C)=O)CC2CCC2(CC(=O)NC2CCC(O)C2O)C1 c1(N(c2ccccc2)C(C)=O)ccc(S(=O)(=O)NC2CC23CC3)cc1 Cc1nn2c(c1CNC(c1cnnn1C)=O)CN(C(=O)Cc1cncn1C)CC2 c1(C(N2CC(NC(C3(CC#C)CC3)=O)C(OC)C2)=O)c[nH]nc1[N+](=O)[O-] Cc1ccc(C2CN(C(C3CCCN(Cc4cnc(O)o4)C3)=O)C2)c(F)c1F CC1=NOC(CCNC(=O)CCOCCN(C)C(C2CCS2(=O)=O)=O)C1 N1(C(C2(COC)CCCO2)=O)C(C(=O)NOCC(O)COC)CCC12CC2 Cc1ccc2[nH]nc(C(N3C4CCC3CC(CCNC(=O)CNC=O)C4)=O)c2c1 Cc1noc2nc(C(=O)N(CCC(C(C)(C)C)NC(C3CC34CC4)=O)C)ccc12 c1(C(NNC(Cn2cc(OC)c(=O)cc2C)=O)=O)ccc2ccccc2c1 n1(C(C)C)cc(Br)cc1C(=O)NCC1CCN1C(C1C(C)CC1C)=O C1(CN(C)C(C2(Br)CC2)=O)CCCN(C(c2occc2F)=O)C1 CC(C)CC(CNC(=O)CC1CCC(=O)C1)C(=O)NC1CC(=C2CC2)C1 N1(C(C(C)C(=O)O)=O)CC(=O)NC(=O)C1 c1(OC)cc(C(N2CCC(=CC(=O)Nc3ncc(F)s3)CC2)=O)ccc1F C1(C(=O)NC2(CC=C)CCN(C(C3CCC(=O)N3)=O)C2)CCC2CCCCN12 CCCCC(C)(F)C(=O)N(CCC(C(C)(C)C)NC(c1c[nH]nc1Br)=O)C c1(N2CC(C)(C)OC3(C2)CC3)nc(NCC2CCCCO2)c2ccsc2n1 C1(C)(CC)C=C(C(=O)NCC2CC(NC(=O)COC3CCC3)CC2O)C1 C(=O)(CS(=O)(=O)C1CC1)NC1C(NC(CCN(c2ccccc2)C(C)=O)=O)C1 Cc1cc(C(N2CCCC2C(C)(C)NC(=O)CC2CCCCO2)=O)ns1 c1(Cn2cc(C3C4CN(C(C5(C)C=CCCC5)=O)CC43)nn2)cc(O)n2nccc2n1 c1(C(N2C(C(=O)Nc3c(Cl)ncc(C)c3)CSCC2)=O)cccc2cn(C)nc12 N1(C(C(C(CC)O)(F)F)=O)CCN2CCN(C(c3cncc(F)c3)=O)CC2C1 c1(CC(=O)NCC2C(C)CN(C(C3CC4CC4C3)=O)CC2)ccc2nn[nH]c2c1 CC(C)(O)C(C(=O)N1CCCC1)NC(=O)C(=O)NC1CCNCCC1(F)F c1(CC(C)C)nc(=NCC(C)CNC(C2(CN(C)C)CCCO2)=O)s[nH]1 N1(C(CSCC#C)=O)CCOC(CNC(c2c(Cl)n[nH]c2C2CC2)=O)C1 CCC(C)(CNC(=O)COc1ccn(C)n1)C(=O)N(CC(C)(C)CO)C c1(C(N(C2CCCC(NC(c3c(C)snn3)=O)C2)C)=O)cnc2c(c1)CCCO2 c1(NC(c2ccc(N3CC(C)OCC3)cc2)=O)cc(Cl)c(Cl)cc1O NS(=O)(=O)c1ccc(NCC(=O)NC2(CCNC(=O)CC3=CC=NC3)CC2)cc1 CCC(O)C(C)C(=O)N(C1CCN(C(=O)Cc2ccc(CO)c(C)c2)CC1)CC C1(CC(=O)N(CCNC(C2C(C)(CC)C2)=O)C2CC2)CCC(C(=O)NC)CC1 c1(NC(C2CC(N3CCCC3)C2)=O)ccc(Br)c(NC(C2CNC(=O)CO2)=O)c1 C12(C(=O)NCC(C)(CC(C)C)NC(C(C)=CC3CC3)=O)CCOC1CC(=O)NC2 c1(C(N2C(CNC(C(CC)C#N)=O)CC(OC)C2)=O)cnc(C(F)(F)F)c(F)c1 N1(C(c2c(C)c(C3CC3)on2)=O)CCCC2C(NC(c3csnn3)=O)C(C)(C)C12 c1(C(C(=O)NCCC2(NC(C(CC=C)C)=O)CC2)O)ccc(O)c([N+](=O)[O-])c1 N1(C(C(CCC)O)=O)CC2(COC(CNC(C3(CC)CC(C)(C)C3)=O)C2)C1 C(=O)(C1CCCn2ccnc21)N(C)CC1(NC(=O)CCS(C)=O)CC1 Cc1nc2c(N(CC(C)CNC(c3cc(C(F)F)ccc3Cl)=O)C)ncnc2s1 CC(C)CC(O)C(C)C(=O)N1CCSCC1C(N1CCC([N+](=O)[O-])CC1)=O N1(C(c2ccn(CC)c(=O)c2)=O)CC2CCCC(C1)N2C(=O)CN1CCCCC1 c1(CN(CCC)CCNC(=O)CC2CC2)ccccc1CNC(N1CC=CC1)=O CCC(O)C(C)C(=O)N1CCCCC(C(=O)NC2(C)CSC2)C1 c1(C(N(C(C(=O)N(CCOC)C)C2CC2)C)=O)csc(C)n1 c1(C(=O)NCc2cccc(NC(c3c(C)n(C)nc3)=O)c2)ncnc2c1CCC2 c1(CC(=O)NC2C(CNC(CCS(C)=O)=O)CC2)ccc(Cl)cc1F CC(C(=O)NCCOC1CN(C(C2CCN(c3ccccc3)C2)=O)C1)S(C)(=O)=O c1(CC#N)ccccc1C(=O)NC1CC(CNC(c2ccn(C3CCC3)n2)=O)C1 c1(C(=O)NC2C(C(N(C3C(=O)OCC3(C)C)C)=O)CCCC2)cccc(F)c1F N1(C(C2(F)CN(C(CC(CC)CN(C)C)=O)C2)=O)CC(C)(C)CCC1C c1(C(=O)OC)ccc(C(=O)NCC2CC2CNC(c2cc(C)n(C)n2)=O)cc1F c1(C(=O)NCC2(F)CC(NC(C3CCN(C)C3)=O)C2)cnc(O)c(Cl)c1 CC(C)CCC(=O)NC1CCC(C)(CNC(C2CC(OC3CC3)C2)=O)C1 C(=O)(C1CCc2cccnc21)NC(C(C)NC(c1cnn2c1CCC2)=O)(C)C c1(OC)cncc(C(N2CCC=CC2C(=O)NCC2(C)CCCOC2)=O)c1 Cc1cc(C(F)F)ncc1C(=O)NC1CCN(C(C2CCO2)=O)CC1O CCC(F)(F)CCN=c1[nH]c2c(c(=NCc3snnc3C)[nH]1)SCC2 C#CC1(O)CC(C(=O)OC2CCCN(CC(F)F)C2)C1 CC1Cc2ccccc2C(NC(=O)CCSc2cccc(F)c2)C1 C1(N(C(c2[nH]nc(OC)c2Cl)=O)C)CCN(C(=O)CSC(F)F)CC1C n1(CC=C)c(N2CCC(N(C)C(=O)OC(C)(C)C)C2)nnc1-c1coc(C)n1 Cc1cc(C)c(C(=O)N(C)CC2COCCN2C(C2CCN(CCF)CC2)=O)s1 c1(C(=O)NC2(c3cc(C)no3)CC2)ccc2c(-c3cc[nH]n3)nn(C)c2c1 Cc1oc(C(N2CC3CC2C3NC(=O)CC(C)CC(F)(F)F)=O)cc1S(N)(=O)=O N1(C(CC2CC(NC(CSCCC)=O)C2(C)C)=O)CCOC2CCC12 C=CCC(C)(CC)C(=O)NCCC1(CNC(=O)CC2(C)CCCO2)CC1 CCC(C)C(O)C(C)C(=O)NCC(C)(C)C#CC(=O)NC1COCC1F C(=O)(CC(CC(N)=O)CC(C)C)NC1C2(CN(C(CNS(NC)(=O)=O)=O)C2)CC1 N1(C(C(C)NC(CC)(C)C)=O)CCC(C)C(CNC(C2(CO)CCOCC2)=O)C1 N(C(=NCCc1ccsc1)NCC(F)F)Cc1cc(CC)on1 N1(C(C(CC#C)(C)NC(c2cnc(Cl)n2C)=O)=O)CCCC2(CCC2)C1 C1(CCNC(C2CCCC2NC(C2CC2C2CC2)=O)=O)CCCCO1 N1(C(c2cnc(CC)s2)=O)CC2C(CNC(=O)C(O)CSC)C2C1 C1(CC)CC(C(=O)NC2CC23CC(OC)C3)CCN1C(c1ccc(C(N)=O)[nH]1)=O c1(C2CC(=O)C2)nc(-c2ccc(C(F)F)cc2)nn1Cc1cccnc1 N1(C(C)=O)CCCC1C(=O)NC1CC1CNC(=O)CO.C(C)(C)O C(=O)(C1=CCC(C)(C)CC1)C(C(C)CNC(=O)C1CC1)=O.C12CCCCC1CN2 c1(C2N(C(=O)NC3(CC(=O)OC)CS(=O)(=O)C3)CCC2)ccc(O)c(OC)c1 C1(N(C(CN(CC)CC)=O)C)CN(C(c2ccc(OC)cc2Cl)=O)CCC1C C1(C(N2C(C(C)(C)NC(c3cn(C4CC4)cn3)=O)CCC2)=O)CC2C=CC1O2 N1(C(c2nc(C(C)C)sc2)=O)CCC(OCCNC(=O)C(C)C2CCCC2)CC1 CC1CC=C(C(=O)N2CCC(NC(c3cncc(C4CC4)c3)=O)C(C)C2)CC1 N1(C(c2n(C)cc(NC(=O)C(C)(F)F)c2)=O)CC(O)CC(O)C1 N1(C(C2(OC)CCOCC2)=O)CC2CN(C(=O)C=Cc3ccc(OC)o3)CCC12 N1(C(c2ccc(C)nn2)=O)CC2CN(C(C34CCC(C)(CC3)CO4)=O)CC2C1 c1(C(N(CCN(C(CC(CCC)C)=O)C)C)=O)ccc2c(c1)NCC2 N1(C(c2c(CCC)nco2)=O)CC2CCC1CN2C(C1(OC)CCC(C)C1)=O C1(NC(CC(=C)Br)=O)CC2CC1CN2C(c1c(OC)cccc1F)=O CCCCC(CCCC)NC(C1CN(C(=O)CC(C)F)CC1(C)C)=O N1(C(C(Cc2ccc(Cl)cc2Cl)NC(=O)OC(C)(C)C)=O)CCCC(F)(F)CC1 n1(C(C)(C)C)nnc2ccc(C(=O)OCC(C3CCOC3)O)cc12 N1(C(CN(C(=O)OCC)C)=O)CC2CC2C(CNC(c2ccccc2OC)=O)C1 N1(C(CCOCCOC)=O)CCCC(C(C)(O)CNC(=O)Cc2cnoc2)C1.C(C)(=O)O C1(C(=O)NC(c2noc(C)n2)CC)CCN(C(c2cc(C(C)=O)[nH]n2)=O)C1C CC1C(NC(=O)CCCC(F)(F)F)CC2CCC1N2C(c1cncc(Cl)n1)=O C(=O)(C(CC(C)C)ONC(c1cn(C)c(=O)cn1)=O)NCCc1c(C)nccn1 Cc1cn2ccc(C(=O)NC(C)C(C)NC(C3(C)CC(F)(F)C3)=O)cc2n1 c1(C(N2CCC(C)(CCNC(C3ON=C(CC)C3)=O)C2)=O)cccc2nncn12 C1(C(=O)NCC(C)(C)OCC(=O)NC2CCC(C)(C)C2)(NC(N)=O)CCCSC1 C1(NC(CC(CN(C)C)O)=O)CN(C(C2(F)CCCCC2)=O)CC2(CC2)C1 c1(NC)ccc(Cl)c(C(=O)NCC2(NC(c3ncnc(OC)c3F)=O)CC2)c1 C1(C(=O)NCC(=O)Nc2c(F)cccc2F)CCc2ccccc2C1 c1(C(=O)NCC(O)CNC(c2cc(F)c[nH]2)=O)ccc2c(c1)OCCCO2 Cc1cc(N(C)CCc2ccc(Br)cc2)nc(NC(C)C(c2ccccc2)O)n1 C1(NC(C(N)=O)=O)CCN(C(=O)C(O)CC2CCOCC2)C12CC2 c1(C(N2CCC3CN(C(C(C=CC)O)=O)CC3C2)=O)cc(Cl)cc2ccncc12 c1(CC(=O)NC2CCC2CNC(c2cccc(=O)o2)=O)cnc2ccccc2c1 c1(C(=O)NCC2CCCC(NC(c3nccc(OC)c3)=O)C2)cc(C)n(C)c1C c1(OC)cc(C)nc(N2CCC(C)C(NC(=O)C=Cc3cnc(C)s3)C2)n1 CC1CCCC(CC(N2CC(CNC(=O)CCCCNC(N)=O)CC2C)=O)C1 c1(OC)nn(C)cc1-c1ccc(CNC(c2c[nH]cc2C)=O)cn1 CC(CCC(C)(C)C)C(=O)NCC1CC12CCCC2 N1(C(c2ccc(N)c(Cl)n2)=O)CCC2CC2(NC(c2csc3nnsc23)=O)CC1 C1(NC(C(CC)(C)C)=O)CN(C(C2CCC=CCC2)=O)CCC1C C1(NC(CNC(CCC(C)C)=O)=O)CCN(C(C2(C)CCCO2)=O)CCC1(F)F Cn1ncc2cc(CNc3cc(-c4ccc(Cl)cc4)ns3)ccc12 N1(CC(=O)NCC(C)(CO)NC(C2CC(n3cccn3)C2)=O)CCC(=O)NC1=O N1(CCCCC)CCC2(CN(C(C3CCCOC3)=O)CC(C)O2)C1 c1(C(c2n(CC)nnn2)NCCC(C)COC)ccc(F)cc1 N1(C(CCCOC)=O)CCCC1(C)CCC(=O)NCC1(C(C)C)CC1 Cc1cc(=O)c(C(=O)NCC2=CCN(C(c3cc(C)n(C)n3)=O)CC2)cn1C C1(C(=O)NC(C(=O)NC2C(C)(C)C2)c2ccoc2)CC12CCCCC2 c1(C(=O)NCC(F)F)ncn2ccccc12.c12ccc(cc1)[nH]2 C1(NC(=O)CNC(=O)C2CC2)CC2CC(NC(c3cc([N+](=O)[O-])c[nH]3)=O)CC12 c1(N2Cc3c(c(O)nc(=N)[nH]3)C2)nccc(=NC(CF)c2cccc(F)c2)[nH]1 N1(C(CNC(C)=O)=O)CCCC(N(CCO)C(c2ncnn2C2CCOCC2)=O)C1 C(=O)(C(C)(C)C1=CCSCC1)NC(CN(C)C(C1CC2C=CC1C2)=O)(C)C Cc1ccc(C(=O)NCCC2CCC(NC(=O)C3=COCCC3)C2)c(C)c1 C1(OCCNC(=O)CCN2CCC(F)C2)CCN(C(=O)CC2COCCOC2)CC1 N1(C(C2N(C(c3cc(C(C)=O)[nH]n3)=O)CC(F)C2)=O)CCOCC(F)(F)C1 c1(-c2n(-c3cn(C)nc3)nc(-c3cc(F)cc(F)c3)n2)n[nH]c2c1COCC2 c1(C(=O)NCC2(OC)CN(C(=O)COc3ccccn3)C2)ccc2sccc2c1 c1(OC)ccc(Cl)c(CN2CC3CC(C2)N3C(c2cnc(OC)nc2)=O)c1F O=S(=O)(c1ccc(Br)cc1F)NC1CCC(Nc2ncnc3sccc23)C1 c1(-c2ccc(SC)nc2)cc(F)cc(F)c1C(=O)Nc1cc(C#N)ncn1 CC1(C)CCCCC(C(=O)NCCCC2CC2(F)F)C1 C1(NC(Cc2c(C)ocn2)=O)CC(C(=O)N2CCCC(F)(F)C2)=CC1O CC(C)CCCC(C)C(=O)NCCCCC(CO)NC(=O)COCCCN=[N+]=[N-] C1(NC(c2cn(CC=C)nn2)=O)CC2CN(C(c3cc(C(C)=O)on3)=O)CC12 N1(C(Cc2nc(CC)sc2)=O)CC2(NC(=O)C(CC)SC)CCCC2(F)C1 C1(COC)CN(C(=O)C(C)(C)C(=O)NC)CCN1C(C1CCN2CCOCC12)=O N1(C(COCCCCCC)=O)CCC(NC(=O)CSc2cncn2C)C(F)C1 c1(NC(C(c2cccc(Br)c2)(C)N)=O)ccc(S(F)(F)(F)(F)F)cc1 C=CCC(CNC(=O)C(C)=CCN(C)C)NC(C1CCCN1C1CC1)=O N1(C(C2N(c3ncnc(CC)c3F)C3C(C2)C3)=O)CCC2(CCNC2=O)CC1 c1(CC(=O)NC2C(C)N(C(=O)C(C)O)CCC2)cc(F)c(F)cc1F c1(C(=O)NCCCN(C(=O)Cc2cnc(C)s2)CC)c(F)ccc2[nH]ccc12 CCC(C)C(C)C(=O)NCc1ccc(C(=O)NCC(C)(C)C2CCC2)o1 N1(C(c2ccnc(C)c2N)=O)CC2CCC1CC2NC(=O)CC1COCC(C)O1 N1(C(C(C)NC=O)=O)CCCCC1CN1CCCC2(CC2)C1 c1(C(=O)NC2C3(CC(NC(c4cnnc(O)c4)=O)C3)C2)ncc(Br)cc1O c1(OC)cc(O)c(CNC2CN(C(=O)CC(=O)OC)CC23CC3)cc1OC C1(NC(CCC2CCCN(C(C(C)(C)CC3CC3)=O)C2)=O)CC(C)(C)OC1(C)C n1(CC)cccc1C(=O)NCCC(C)NC(c1ccncn1)=O N1(C(CC(c2c(C)cccc2)C)=O)CC(NC(=O)C=CC(=O)N(C)C)CC(F)(F)C1 N1(C(C(Cc2ccco2)N(C)C)=O)CC2CCCC2(NC(C2CC2(F)Cl)=O)C1 CC(C)(CC(=O)N1CCCCC(NC(=O)CSc2ccc(F)cc2)CC1)C(C)C C(CSC)(CN=c1nc(N2CCCC(CO)C2)c2c([nH]1)CCOC2)OCC C1(NC(Cc2c(C)cccc2)=O)CCCCC12CCCN(C(C1C=C1C)=O)C2 C=CCC(CNC(c1cnoc1-c1ccccc1)=O)NC(C1(C)CC1)=O Cc1nc2ccc(C(=O)NC3CCN(C(c4ccc(C(F)F)nc4)=O)C3)cc2o1 C1(CC)CCCC1N=c1[nH]c(N2Cc3ccccc3C2)nc2ncn(CC)c12 c1(SC)cc(C(N2CC(C(C)NC(c3csc(Cl)c3Cl)=O)C2)=O)c(C)o1 C12(C(=O)NC(C)CN(C(=O)Cc3nc(=N)[nH][nH]3)C)CC(CC(C)O1)C2 CC1CC(C(=O)N(C2CCN(C(=O)CSC(=N)N)CC2)CC2CC2)CCO1 N1(C(C(CCSC)O)=O)CCC(CC(F)F)(CO)CC1 N1(C(CCCCCOC)=O)CCC2(CC1)CC2C(=O)NCC1(C)CCCN(C)C1 C(=O)(C(F)(F)C(O)CC)NCC(CCCC)NC(=O)CCCOCCOC CC1(C)CN(C(=O)CCc2ccoc2)CC1CNC(=O)CSC1CC1 N1(C(CCCC#CC)=O)CCCC2CN(C(=O)C(C)(O)C3CCOCC3)CC12 c1(C(N2C(CNCc3cccc(OCC)n3)COCC2)=O)c(C)cc(O)cc1O N1(C(COCCCC#C)=O)CC(CNC(=O)CSCC=C)OC2CCCC12 CN1C2CCCC1CN(C(C1CC1C1CN(C(c3coc(C4CC4)n3)=O)C1)=O)C2 c1(C(N2CC3C(NC(c4cc(F)ncc4Br)=O)C3C2)=O)cn2ccc(Cl)cc2n1 C(=O)(CC(C(F)(F)F)SC)NCC1(CC)CCCCO1.C12(CCC1)C(=O)N2 c1(OC)cccc(COC(c2occc2NC(=O)CSC(C)=O)=O)c1 C1(C(N2CC(C)OCCC2)=O)CC2CCCC2N1C(=O)CCc1nncs1 c1(C(=O)NC(C)(C)CCCNC(=O)CCS(C)(=O)=O)cccc([N+](=O)[O-])c1Cl c1(CC(=O)NC2(CNC(C3(CCC)CCC3)=O)CC2)ccc(OC)c(Br)c1 c1(C(CN2CC(n3cc(CNC(C45CC(C4)C5)=O)nn3)C2)O)cc(F)cc(F)c1 c1(OCC(=O)NC2CC(O)C(F)C2)c(Cl)cc(Cl)cc1Cl C(CN=c1ccc(CO)c[nH]1)N(C(c1cc(OC)ncc1)=O)Cc1ccccc1Cl N1(C(CC2(OCC)CC2)=O)CCCC2(CCCN2C(C2(C3CCCO3)CC2)=O)C1 Cc1ccc(-c2cn(CC3CN(C(c4ccc(C)cc4C)=O)C3)nn2)c(C)c1 C1(CC)C(C(=O)NCC2CCC2C)CCCN1C(=O)CCC1CC1(F)F c1(C(N2CC(CNC(CC(C)OC)=O)C3(C2)CC3)=O)cc2ccccc2o1 Cc1nc(CCC(=O)NC(C2CN(C(C3(C)CC3(F)F)=O)C2)C)oc1C c1(CC)ncoc1C(=O)NCCCN(C(C1CCCO1)=O)CC1CCCC1 Nc1cc(F)cc(Cl)c1C(=O)NC1CCC2CCN(C(=O)CC3CCCCC3)C12 N1(c2nc(C)nc(C(C)C)c2)C(CNC(=O)CCn2cccn2)CC2COCC12 C(=O)(C(C)CC(C)(C)C)N(CCNC(c1c(C)n(C)cc1)=O)CCNS(C)(=O)=O C1(C(N2CC(C)(OCC(NOCC#C)=O)C2)=O)Cc2nccn2C1 C1(CCN(C(C(C)OC)=O)C)CCN(C(C2CC2C(F)F)=O)CC1 n1(CC)cc(NC(=O)C(C2CCCN(C(C3COCC3C(N)=O)=O)C2)(C)C)c(C)n1 C1(C)(CCNC(=O)NC2CC(C=C)C2)COCCO1 C(=O)(C(C)CC1CCCC1)N(N1CC2CC2C1)C.n1(C(C)C(=O)O)cc(C)nn1 C1(NC(C(CC)NC(C)=O)=O)CC(F)CN(C(=O)C(CC)(CC)c2ccccc2)C1 CC(C(=O)N1CCCC(CCC(=O)NC2(C3CC3)CC2)C1)C(C)(C)C CCC(C)CC(C)C(=O)N(C1CCN(C(C2CC23CCCC3)=O)CC1)CC1CC1 Cc1cn2c(n1)C(C(=O)NCC1CC(NC(=O)C(c3ccc(C)o3)C)C1)CCC2 Cc1cc2[nH]c(C(=O)NCC3(F)CCN(C(c4cc(Cl)ccc4O)=O)C3)cc2s1 C=CC(C)(C)CC(=O)N(C)CC1(O)CCN(C(=O)C(c2c(C)noc2C)CC)C1 c1(CONC(c2cccc(C3CC3)c2)=O)c(Cl)cccc1[N+](=O)[O-] c1(C(N2CCC(O)(CNC(C34CCC(C3)C4)=O)C2)=O)ccc(Cl)cc1Cl C#Cc1c[nH]nc1C(=O)NCC1CC(NC(=O)C(C)CC=C)C1 c1(C(N(CC(=O)NCCN(C)CC)CC(C)C)=O)cc[nH]c2nccc1-2 c1(C(N2CC(C(C)NC(c3cc(C(C)C)[nH]n3)=O)C2)=O)ccnc2c1CC(=O)N2 Cn1cc(C(N2CC(CNC(=O)C(=O)NCC3CC3)C(F)(F)C2)=O)c(O)nc1=O C1(CCNC(CCC)=O)(NC(c2ccc(C(N)=O)nc2)=O)CCOCC1 C1(NC(c2ccn(C3CCCC3)n2)=O)CC(CO)N(C(c2cccc(F)c2)=O)C1 N1(C(c2cnc(CC)[nH]2)=O)CC2(CCCC(CNC(=O)CCOCC(F)F)O2)C1 N1(C(C(n2cc(CCN3CCN(C)CC3)nn2)C)=O)CCC2CCC(C1)N2C c1(-c2cn(C(C)C(=O)NC(C)CCCCSC3CC3)nn2)c(F)cncc1F C1(C(N(CCCCNC(c2cc(C)cc(C)c2)=O)C)=O)CC2CC(O)CC(C1)C2 N1(C(c2c(C)ccc(F)c2)=O)CCC2CC2(C(N2CC(N3CCCCC3)C2)=O)CC1 N1(C(CCOC2CN(C(C(c3cncnc3)C)=O)C2)=O)CCCCCCC1C N1(CCNC(COCCCCC)=O)CCC(NC(=O)CC2CC(OCC)C2)CC1 CCCCCCn1nnnc1C(c1cccs1)NCC1(CC(C)C)CCC1 C(=O)(CCCCCNC(=O)C(C)C#N)N1CCC(OC)(CO)C1 C(=O)(C1(C)Cc2cccc(Cl)c21)NC(CN(C(C1CCN(C)C1)=O)C)(C)C CCC(C)C(O)CC(=O)NCCN(C)C(c1cnc2c[nH]nc2c1)=O C=Cc1cnn(C)c1C(=O)NC1CCCC1CNC(c1cnc(C)nc1CC)=O C1(C(=O)NCCCCCN(C(CC2C(C)OCC2)=O)C)CCCCNC1=O c1(C(=O)NC(CN(C(=O)Cc2cccc(O)c2F)CC)C)cnc(O)cc1C C12(NC(c3cccnn3)=O)CCCC1N(C(c1cncc(O)c1)=O)CC2 N1(C(CCC)=O)CCN(CC(C)NC(=O)C(C)(C)n2ccnn2)CC1 c1(NC(C2CC3CC3C2)=O)ccc(-n2cc(-c3ncccn3)nn2)cc1 C(C)(CCNC(=O)C(C)N(C)C)NC(COCCSC)=O C1(NC(C(CCC)CCC)=O)CN(C(=O)C(CN(C)C)CC)Cc2nccn2C1 N1(C(CC(CC)C2CC2)=O)CC2CN(C(C3(NC(C)=O)CCC3)=O)CC(C1)O2 C1(C(N2CC(C)C(CC(=O)N(CC(N3CC=CC3)=O)CO)C2)=O)CCC(C2CC2)C1 C(=O)(C(O)CCC(C)C)NC1CN(C(C2(OC)CCSC2)=O)CC1F N1(C(Cn2c(C)ccc2C)=O)CC2C=CC1C(C(=O)NCC1CC3(CC3)C1)C2 N1(C(c2sc(C)c(-c3ccccc3)n2)=O)CC(N)CCc2ccccc21 c1(C(N(CCNC(C)=O)CC2CC2(c2ccc(Br)cc2)F)=O)ccc(Cl)cc1Cl O=[N+]([O-])c1ccc2c(c1)C(NC1CCCCC13CCCCC3)CCN2 c1(CNC(=NC)NCCc2nccc(=O)n2C)cccc(P(C)(C)=O)c1 c1(CNC(=O)NC2CCN(Cc3ccccc3)C2)ccc2c(c1)OCCCO2 c1(NC(=O)C(N2CCN(c3cc(CCCCC)[nH]n3)CC2)=O)ccccc1F N1(C(CCNC(COC)=O)=O)CC(C(C)NC(=O)C(C)OC)C1 C1(C)(C(=O)NCC2C(NC(c3cn(CCC)nc3)=O)CC2)CC(OC)(OCC)C1 CCC(CCC(=O)NCC1CCC(C(=O)NC2(c3cc[nH]n3)CC2)C1)OC c1(OC)ncc(C(N2CCC(C)(NC(c3cn(C)ccc3=O)=O)C2)=O)cc1Cl N1(C(C(C2CCC2)OC)=O)CCCCC1C1CCCN(C(C2(C(N)=O)CC2)=O)C1 CCC(C)CC(=O)NCC1CCCCC1NCC(=O)Nc1nccc(CO)n1 CCC(CC(C)C)C(=O)N1CC2CC1CN(C(c1ccc(N(C)C)cc1F)=O)C2 C(CC(C(=O)NC1(C)CCCC1C)NC(c1ccc(N)cn1)=O)SC CC1(C)C(=O)NC2CCCN(CC(=O)NCCC3COc4ccccc4O3)C12 C1(COC)(CNC(C2CCSCC2)=O)CCN(C(C2COCCO2)=O)C1 C1(NC(C2(C)CCCC2)=O)CC=C(C(=O)N2CC(OC(=N)O)C2)C1 c1(COC)ccc(C(=O)NC2(CCCNC(=O)C(n3ccc(C)n3)C)CC2)s1 N1(C(CCOCCC)=O)CCN(C(=O)CNC(=O)OC)CC1C1CCCC1 C1(NC(C)=O)CCc2nncn2C1.c12ccc(cn1)C(=O)NC(C)C1(O)CN2C1 c1(C(N2CCC(C)C2CNC(=O)Cc2cccc(F)c2O)=O)cc(O)ncc1F N1(C(C(C)N(C)C)=O)CC(C(N2CC3CSCC(C3)C2)=O)C(C2CC2)C1 CC1(C)OC2(C(=O)NC3COC4CN(C(c5c[nH]ccc5=O)=O)CC34)CCC1C2 CCC(C)CCCCC(=O)N(C)CC1CCCN(C(c2cnc(COC)s2)=O)C1 c1(C(=O)NC(C)CC2CN(C(C3(C(N)=O)CC3)=O)C2)nccc2cccnc12 C(CC(C)C)(C(=O)N1CCN(C(c2ccc(F)cc2N)=O)CC1C(C)C)OC c1(C(=O)NCC(C)CN(C)C(C2CC2C(N)=O)=O)cncn1C C1(NC(=O)CCc2ncc[nH]2)CCCC12CN(C(C13CCCC1CCC3)=O)C2 C1(C(N(CCOCCCNC(CC=CCCCCC)=O)C)=O)CCNC(=O)C1 O=C(N=c1[nH][nH]c2ccc(F)cc12)c1cc(F)c(F)cc1Br N1(C(c2c(C)sc(-c3ccccc3)n2)=O)CC=C(C(=O)N2CCCC2CO)CC1 N1(C(c2c(C)nccc2Cl)=O)CCCN(C(=O)CCC2OCCO2)C(C)C1 Cc1ncnc(C)c1OCC(=O)NCC(C)(C)NC(c1ccsc1C#N)=O C1(CNC(c2n(C)ncc2)=O)CCCCN(C(=O)Cn2ncn(C)c2=O)C1 c1(C(N(C2CCN(C(c3ccc(O)nc3)=O)CC2)CCOC)=O)cc(=O)cc[nH]1 c1(C(N(C2CCCCN(C(=O)C(C#N)C3CC3)C2)C)=O)cnc2sccc2c1 C12(C(N(CCCN(C(=O)CN3CCC(N(C)C)CC3)C)C)=O)CCCC1CCC2 C1(C(=O)NCC(Cn2cc(-c3cncn3C)nn2)OC)CC(C)N(C)C1 C(=O)(CCC(C)(C)C)NC1C2CN(C(c3c(CC)nccc3)=O)CC21 N1(C(COCC)=O)CCN(C2CN(C(=O)CC(O)C3CCCC3)C2)CC1 c1(N(CCSC)C)nc2c(c(=NC3CCN(c4cccc(Cl)c4)C3)[nH]1)SCC2 N1(C(CC)=O)CCC2(CC1)CC2C(=O)Nc1cc(O)ccc1Cl N1(C(CCc2nc(C)c(C)o2)=O)CCC2(CC2NC(C2CC2C(N)=O)=O)C1 C1(c2noc(C3(C45CC6CC4C5C6O)CC3)n2)(CC)CCC(F)(F)CC1 CC(C)(O)C(F)(F)C(=O)N1CC2CC1(c1cn(-c3ccncc3F)nn1)C2 C1(NC(C(N2CCC(CO)CC2)C2C(C)C2)=O)CCC(F)(F)CC1 c1(C(=O)NC(COC)C(=O)N2CCCC2COC)cc(F)cc(F)c1 c1(C(=O)NCC(CCCC)NC(C2OCCN(C)C2=O)=O)ccc(C)cc1Cl Cc1ccc(C)c(C(=O)NC2CN(C(=O)C3=CCC3)CCC2CO)n1 Cc1ccccc1CC1CCCN1C(=O)NC(c1ncc[nH]1)CO c1(CCC(=O)N(C)CC2(O)CN(C(C(CC)N(CC)CC)=O)C2)ccc(C)cc1 C(=O)(C(C)(CC)CCC)NC1C(C(N(CC#C)CC)=O)CCC1 N1(C(CCC#CC)=O)CCC2CN(C(=O)C(C)(CC)C(=O)OCC)CC2C1 N1(C(c2n(CC)ccc2)=O)CCC(C(=O)NCC2(C3CC3)CCCO2)C1(C)C N1(C(C)=O)CCCCC1C(=O)N(CCNC(c1c(O)noc1C)=O)C1CC1 C1CCCC1NC(C1CCC1NC(N)=O)=O.N1(CCN(C)C)CCCC1 CC1(C)C(NC(=O)C=Cc2nccs2)CC1CC(=O)NCc1ccccc1F CC1(C)CC2(CC(C(=O)NCc3cccc(CNC(C4CC4(F)Cl)=O)c3)C2)C1 C#CCC(CC(=O)NCC12CCC(CC1)O2)NC(c1c[nH]nc1[N+](=O)[O-])=O C1(C(=O)NCC2CCN(C(C)=O)C2)(CNC(c2cc(C)n(C)n2)=O)CC2(CC2)C1 O=S(=O)(c1ccc(NC2CCCC3(C2)OCCO3)c(F)c1)NCC1CCCCS1 c1(C(c2n(C(CC)C)nnn2)NCc2cccnc2)cc(C)oc1C N1(C(c2cc(CO)ccc2Cl)=O)CC2CN(C(C3CCC3(F)F)=O)CC2C1 C1(NC(C2CC=CC2)=O)CCN(C(c2csc(-c3ccco3)n2)=O)CC1CO N1(C(CSCCNC(CC(COC)(C)O)=O)=O)CCC12CCCSC2 N1(C(CS(N)(=O)=O)=O)CCC(F)(CNC(=O)C(c2cccc(F)c2)O)CC1 C1(C(N(CCCC#C)C)=O)CCCCCCN1C(c1cc(CCC)on1)=O n1(CC(N2CC3CCC3(C(N3CCC(F)(F)C3)=O)C2)=O)nc2ccccn2c1=O C12CCCC1NC2=O.C(CC(OC)OC)NC(C1(C(=O)OCC)CC1)=O c1(C(N(CCN(C(c2ccc(Cl)s2)=O)CC)CC)=O)cnc(O)c(OC)c1 C1(n2cc(NC(CC(O)NC(C(C)Cc3ccnn3C)=O)=O)nn2)CCN(C)C1=O c1(NCCC2CCC(NC(C3(C#C)CC3)=O)C2)ncnc2[nH]c3ccccc3c12 Cc1cnc(C(=O)NC2CCCCC2CNC(=O)CC(F)(F)Cl)c(C)c1 Cc1nc(CC(=O)NC2(CN(C(=O)C(CO)N(C)C)C)CC2)c(C)s1 CC1CC(NC(=O)CCC(N)=O)CN1C(=O)CCCc1ccsc1 c1(NC(C2(C)CCN2C(C2(c3cccs3)CC2)=O)=O)cnn2ccccc12 CC(C)C(O)C(=O)NCC(C)CN(C(=O)CC1CC=CCN1C)C N1(C(c2cc(C)sc2C)=O)CCC2(CC2C(=O)Nc2ccc(O)cn2)C1 C1(NC(C=C(CCC)C)=O)CCS(=O)(=O)C12CN(C(c1c[nH]nc1F)=O)C2 c1(C(C)C)ccc(C(N2CC(CC(C)NC(=O)CC3OCCC3C)C2)=O)c(F)c1 CC1CCC=C1C(=O)N1CCCCC1CC(=O)NCCCS(N)(=O)=O C1(CNC(CC2N(CC)CCC2)=O)CC(OC)CN1C(=O)C=Cc1cscn1 CC(C(=O)NC1CN(C(=O)CN2C(=O)CCC2=O)CC1c1nccn1C)C(C)O C(=O)(C1CCc2cccc(=O)n21)NC(c1ccc(NCCC)cc1)=O N1(C(C(C=C)(C)C)=O)CCC2CN(C(c3n[nH]cc3C(C)C)=O)CC2C1 N1(C(=O)OC(C)(C)C)CC(CNC(C)CC2(O)CCC2)C(C)C1 c1(C(N2CCC(C(C)NC(=O)CNC(C3CCC3)=O)C2)=O)cccc(C(F)F)c1 c1(C(N(C2CCN(C(C3(F)CCCN(C)C3)=O)C2)C)=O)cc(F)cc(F)c1O C(C(C)(C)C(C)C)(c1nnnn1C1CCOC1)N.C(CC#N)SCC S(=O)(=O)(c1ccccc1-c1cc(Cl)cc(Cl)c1)N1CC(C(=O)NC)C2(C1)CC2 C1(NC(c2ccc(C3CC3)s2)=O)CC(F)(CNC(=O)C(F)(F)C2(O)CCCC2)C1 C=CC(C)(O)CC(=O)NCC1(C)CCN(C(c2cc(OC)ccc2F)=O)CC1 N1(C(C2(C(=O)OCC)CC=CC2)=O)CCOC(CN(C(=O)CCC(N)=O)C)C1 C(=O)(CCCC(=O)NC1CC(F)(CNC(c2csnc2OC)=O)C1)NCCC CC1(C)OC2CN(CCN3CC(=O)N(Cc4ccc(Cl)s4)C3=O)CC2O1 C(=O)(C(C)(C)CCF)NCC1CCC(CN(C(c2c(C)n(C)cn2)=O)C)CC1 C1(C(=O)NC(CNC(CC=C)=O)CC)CC(F)CN1C C1(NC(CCC(C)O)=O)CN(C(=O)CN2CCC2)CC1(C)C c1(C(N(CC(O)COC)CC)=O)c(CNC(=O)C(C)C(C)C)nnn1C c1(CC)onc(C)c1C(N1CCC(OCCCNC(=O)C=CC2CC2)CC1)=O Cc1cc(C(N2CCCC(CN(C(=O)CC3CCOC3)C)C2)=O)nc(C)n1 CC1(F)CN(C(=O)C=CC2CCOCC2)CCN(C(c2cccc(Br)c2)=O)C1 C1(C)(CC)C=C(C(=O)N(C2CN(C(c3cnn4cc[nH]c34)=O)C2)C)C1 CCC(CC(C)C)C(=O)N1CCC(OCC(=O)NCc2csc(C)c2C)C1 c1(OC)ccc2c(=NCC3(C)CCCS3)[nH]c(=NCC3CC4C=CC3O4)[nH]c2c1 c1(C(=O)NC(C)C)ccc(C(=O)NCCNC(=O)CCc2cccnc2F)cc1 c1(SC)cc(C(F)(F)F)ccc1CC(=O)NC1CC(C2CNC2)C1 c1(CC(=O)NC2C(OC)CN(C(C3CC34CC(O)C4)=O)C2)ccc([N+](=O)[O-])cc1 C1(C)(C(=O)NCC(COC)NC(=O)Cc2nnc(S)s2)CCC2(CC1)CC2 Cc1cc(CNC(=O)C=Cc2cn(C)nn2)oc1C(=O)N(C1CCC1)CCO C1(NC(CCC(C)=O)=O)COC2(CCN(Cc3cccc(O)c3)CC2)C1 c1(C(N2CC(C3N(C(C4(CC)CC4)=O)CCC3)(O)C2)=O)n[nH]c2c1CC(C)CC2 C1(NC(C2(NC(C)=O)CCCCC2)=O)CN(C(=O)C(C)C)CCC1C C1(C(=O)NC(CCCCNC(c2ncc(OC)cn2)=O)C)CNC(=O)CC1(C)C C(=O)(C(C)(O)CC(F)(F)F)N1CCCCC(CNC(CC(=C)C)=O)C1 C12(NC(CC3(C)CCN3C(=O)COCCF)=O)CCCN(CC1)C2 C12(NC(CCc3ccn(C)n3)=O)CCC1CN(C(C1CCOC(=O)N1)=O)C2 C1(c2cn(C)nc2)CN(C(C2C(F)(F)C23CC3)=O)CCN1C(c1cn(C)cn1)=O C12(CNC(CCC#C)=O)CCCC1CCN2C(=O)CC1CC2(CC2)C1 C1(CNC(CC2(OC)CCC2)=O)CN(C(=O)CCN2CCOCC2)CCC1(F)F C12(CNC(C3N(C(CCC)=O)CSC3)=O)CC(NC(=O)C=CC3CC3)(CCO1)C2 c1(CC(N2CCC(C)(NC(C3CCOC(=O)N3)=O)C2)=O)nc2ncccn2n1 C12(C(=O)NCc3cn(CC)nn3)C(NC(=O)CC3CCSCC3)C3CC1C2C3 c1(NC(C2(CNC(=O)CC3NC(=O)NC3=O)CC(=C)C2)=O)cc(C)nc(C)n1 C1(F)(CNC(=O)CCc2cccc(F)c2)CCCN(C(C2CCC(O)C2)=O)C1 C(=O)(CC(C(F)(F)F)NC(C1(C)CNC(=O)N1)=O)NCCC(C)N(C)C c1(C(N2CC3C(NC(C(c4ccc(F)cc4)C)=O)C3C2)=O)c(O)ccc(Cl)c1F CCCCCCCC(=O)N1CCC(C(N2CCC(NC(C)=O)C2)=O)(CO)C1 C#Cc1cncc(C(=O)NC2CCN(C(c3cc(C(F)(F)F)cnc3N)=O)C2)c1 N#CC1CCC(CC(=O)NCCNC(c2cncc(Br)c2)=O)C1 N1(C(Cc2onc(C)n2)=O)CC(CNCc2ccc(N(C)C)cc2)C(C)C1 CCCC(C(=O)N1CCCC1=O)C(C)C N1(C(=O)NC2CCCN(c3ccc(Cl)nn3)C2)CCC(O)C12CCC2 N1(C(C2(C=C)CCOCC2)=O)CC2CCC(CNC(=O)C(C)n3cccc3)(C2)C1 N1(C(CC(C)(C)O)=O)CCCC2CCN(C(c3ccc(C#N)s3)=O)CC12 C(=O)(CC(C(F)F)NC(c1coc(N(C)C)n1)=O)Nc1c(CC)nn(C)c1 c1(C(=O)NCCN(C(=O)CCCOC)CCOC)ccc(Br)c(C)n1 c12cn(C)nc1NC2=O.C(CCOC)(C(N)=O)NC(COCCOCC#C)=O c1(C(N2C(CNC(C(CC(=C)C)C)=O)C3CC3C2)=O)n[nH]c2ccc(OC)cc12 CC(C)(CNC(=O)CNC(c1cnn(C2CC2)c1)=O)CO c1(CNC(CC2CCN(C(C(C)C(c3ccccc3)O)=O)C2)=O)cccc(F)c1 CC1CCc2ccccc2N1S(=O)(=O)NC1CC12CCc1ccccc12 c1(C(C)CNC(=O)NC2CCC(NC(C3(C(C)C)COC3)=O)C2)ccc(F)cc1 N1(C(C2(C)CCCC2)=O)CCCC2(CCC(NC(=O)C=CC3CCCCC3)C2)C1 N1(C(c2cc(C)c(C)[nH]2)=O)CCCCCC1CNC(C12CC=CC(C1)OC2)=O C1(CC(=O)OC)CCC(S(=O)(=O)Nc2ccc(CO)cc2)C1 c1(C(=O)NCCCN(CCCNC(C2CC2Cl)=O)C)ccnc(OC(F)(F)F)c1 C1(C(N(CCNC(c2c(COC)cco2)=O)C)=O)CCCCC(=O)N1 N1(C(c2c(C)nc(O)[nH]2)=O)CC2(C1)CN(C(=O)CCc1cnc(O)[nH]1)C2 c1(CNC(C2CC23CCN(Cc2cc[nH]n2)CC3)=O)ccc2cncnc2c1 c1(CC2CCCN(C(c3c(C)n(CC(C)C)nc3)=O)C2)ccc(F)c(Cl)c1 C12(CC(N3CCCC(NC)C3)=O)CC3CC(CC(C3)C1)C2.CC1CC2(C=O)CC12 c1(-c2nc(OC)sn2)ccc2cc(NC(C3(CN(C)C)CC3)=O)ncc2c1 c1(C(=O)NCCCC(C)(C)NC(c2csc(C(F)(F)F)c2)=O)ccc(F)cc1O N1(C(=O)C(c2cccc(F)c2)F)CCN(C(=O)C2=CCSC2)C(C(F)F)C1 Cc1ncc(C(=O)NC2CN(C(=O)CCCc3cnccn3)CC2C)cn1 N1(C(CSC(=N)N)=O)CCN(C2CN(C(=O)CCC3CC3)C2)CC1 C=CCCCCCC(=O)NC1CCN(C(=O)CCc2nc(C)c(C)o2)CC1(C)C c1(C(=O)N(CCC(N2CCCCCCC2)=O)CC2CC2)c[nH]c2ccccc12 c1(C(=O)NCC2(NC(c3cc(C4CC4)on3)=O)CCOC2)[nH]nc2ncccc12 Cc1cc(C(=O)NCC2CCN2C(C2CC=CCC2)=O)c2cnccc2c1 CC(C)C(C(=O)NCCCC1(C)CC1)C(C)NC(=O)CC1CCC1 c1(C(=O)NC2(C)CCN(C(=O)Cn3cccn3)C2)cc(=N)[nH]c(Cl)n1 O=C1NC(=O)C(CC(N2CC(O)CC2OC(N2CCC2c2ccccc2)=O)=O)N1 Cc1noc(Cl)c1CC(=O)NC1(C)CC1.N(S(=O)(=O)N(C)C)C1C2CC(C2)CNC1 c1(NC(C2(C)N(Cc3ccc(CSCC)o3)CCC2)=O)nc2cc(F)ccn2n1 C1(NC(c2c(CCC)occ2)=O)CCN(C(=O)C(F)OC(F)(F)F)C12CCC2 C=CC(C)C(=O)NC1CCN(C(C2CCC2C#N)=O)C1 C1(C(N2CC(C(C)C)OCC2)=O)C2CCN(C(C3COCC3(C)C)=O)CC12 c1(CC(=O)NCC2(OC)CN(C(c3cnc(C)s3)=O)C2)ccc(Br)cc1I C1(NC(C2(C)C=CCN2C(=O)CN2CCCNC2=O)=O)CN2CCC1(F)CC2 C12(NC(CCNC(=O)OCC)=O)CCCC1CN(C(c1ccc(C)c(F)c1)=O)C2 CC1CC(=O)NCC1C(=O)N(CCCCN(C)C(C1(C2CC2)CCC1)=O)C N1(C(CCCC(C)NC(c2cc(=N)[nH][nH]2)=O)=O)CCC2(CCOC2=O)C1 N#CC1(NC(=O)CCN2C(=O)C=CC2=O)CCN(Cc2nccnc2Cl)C1 c1(CNC(c2c(C)oc(Cl)n2)=O)cnc2c(c1)CNC2=O N1(C(c2cccc(C#C)c2C)=O)CCC2(CCN(C(c3cnnnc3C)=O)C2)C1 N1(C(C(C)OC(C)(C)C)=O)CCC(N=[N+]=[N-])(C(=O)NCCCN=[N+]=[N-])C1 C1(F)(CNC(c2nc(C)[nH]n2)=O)CCCN(C(C2CCN(C3COC3)C2)=O)C1 N1(C(Cc2cccc(OC)c2)=O)CC2CC1CN(C(C13CC4CC1C3C4O)=O)C2 N1(C(c2cc(Br)cc(C)c2C)=O)CCC2CCN(C(=O)CC3CCCC3)CC12 C(C)(CC(C)(C)C)(c1n(CCC)nnn1)NCC1(P(C)(C)=O)CC1 CCC(CCC(=O)NCCNC(=O)CC1OCCC1C)NC(=O)CO c1(OC)c(C)cc(C)cc1C.C12CCC1CCNC2=O C(C)(CCC(=O)NCC1CCN(C(=O)CC2CCOCC2)C1)OC N1(C(C2(c3ccc(C)s3)CC2)=O)CC2CC1C2NC(C12CCCC1(C(N)=O)C2)=O C1(C2=CCOCC2)(CN(CCN(C)Cc2ccccc2)C)CCC1 C(=O)(CC1=CCN(C)CC1)NC1(C)CC(C(N2CCC(O)(CC(C)C)C2)=O)C1 c1(OCC)cc2[nH]nc(NC(=O)NN3CCNCC34CC4)c2cc1CC(C)(C)C C1(NC(C(CC)C(C)C)=O)CCN(CC=CC=CC)CC1(F)F C12(C(=O)NC3CC(CC#C)C3)CCC(NC(=O)C(CC3CC3)OC)(CC1)C2 C1(NC(c2nncc(CCC)c2)=O)CN(C(c2cc(C)on2)=O)C(C)(COC)C1 C1(CNC(c2cc(C(C)(C)C)oc2C)(c2nnnn2C)COC)COC2(CCC2)C1 C1(SC)C2CCN(C(N3CCOC(CNC(=O)OC(C)(C)C)C3)=O)CC12 Cc1oc([N+](=O)[O-])cc1C(N1CCN(C(C2(C)CC(C#N)C2)=O)CC1C1CC1)=O c1(C(C(=O)NC2CC2)N(C)CCOCC2CC2)ccc2c(c1)CCCC2 N1(C(C(C(C)C)C2CCC2)=O)CCC2CN(C(c3cncc4ccsc34)=O)CC12 c1(C(=O)NC2C(NC(=O)CCc3nc(O)n[nH]3)CCC2)cccc2c1CCO2 c1(CC)ccc(OC)cc1C(=O)NC1CCN(C(=O)C(O)C2CC2)C1C C(=O)(C(C)(O)C(F)(F)F)NC1C(NC(CCN(CCCCC)CC)=O)CCOC1 c1(N(C)CC2CCN(C(c3ccc(C)s3)=O)C2)nc(Cl)nc2ccccc12 CC(C(=O)NCC1(CN(C)C(C2(CN(C)C)CCCCO2)=O)CC1)S(N)(=O)=O c1(C(c2nnnn2C(C2(C)CC2)C2CC2)Nc2c(C)csc2)ccc(Cl)cc1F C1(C(=O)NCC(C)N(C(=O)C(C2CCOCC2)C)C)COC2(CO)CC1C2 N1(C(c2cncc(C)n2)=O)CCC(F)(C(=O)NCc2cn(C)nn2)CC1 N(C(=NCCN1CCCC1)N1CCC2(CC(C(F)F)=NO2)C1)CCF c1(CC(=O)N(C2(CN3CC(O)(C4CCCO4)C3)CCC2)C2CC2)ccc(O)c(F)c1 c1(C(C)NC2CCC(C)NC2=O)cc(Br)ccc1F c1(C(N(C)CCNC(C2CCC(C)(C)CO2)=O)=O)ccc(O)c2ccccc12 C1(O)(Cn2cc(CNC(C)=O)nn2)CCCN(C(c2ncc(C(C)C)s2)=O)CC1 CC1CN(C(c2ccc(N(C)C)cc2)C(=O)Nc2ccccc2Cl)CC1C(N)=O N1(C(c2cc(C(C)=O)no2)=O)CC2(CCCCN(C(=O)C(C)N(C)C(C)=O)C2)C1 C1(NC(CC(C)SC)=O)C(CNC(C2CN3CCN2C(C)C3)=O)CCC12CCC2 C(CCC(C)(C)NC(=O)CCc1cnc(C)o1)NC(C1(C=C)CCC1)=O C1(C)(CC=C(C)C)C=CCN1C(=O)CCCn1cc(-c2cccc(N)c2)nn1 C1(C(N)=O)CCCCC1C(=O)NC1CCCC(NC(C23CC(CO)(C2)C3)=O)C1 c1(NCc2nccc(OC)c2)cccc(F)c1C(=O)Nc1cc(Cl)cnc1Br N1(C(C2(CC)CCCN2C(c2csc(CO)n2)=O)=O)CCCC(F)CC1 C12(C(=O)NC3CN(C(=O)CC4CC5(CCC5)C4)CC(F)C3)CC1Cc1c[nH]nc12 CCC(C(=O)N(C1CCN(CC(=O)NC(c2ccccc2)C)C1)C(C)C)C(C)C n1(CCOC)nccc1C(=O)N(CC(C)CNC(=O)CN(c1ccncc1)C)C c1(C(N(CCCNC(=O)CSCC2CCCO2)C)=O)ccc(F)c(O)c1 C(=O)(C(Cn1cncn1)NC(=O)CCc1cc(C)[nH]n1)NC1(CCCC)CC1 c1(C(N2CC(COC)(CNC(c3c[nH]nc3C)=O)C2)=O)ccc2nc(C)cn2c1 C1(NC(C=CC(CC)=CC)=O)CN(C(=O)Cc2ccc(CC3CC3)cc2)CC1F CC1CC(=O)Nc2ccc(C(=O)NCC=CCNC(=O)C3=CCCCC3)cc2N1 S(=O)(=O)(c1ccc(C)cc1F)NCC(=O)NC1CN(C(C(CC=CCC)C)=O)C1 CCC(C)C(CC(=O)NCc1cn(-c2cccc(Cl)c2)nn1)NC1CC1 c1(C(=O)NCC(C)NC(=O)C2=COCCC2)cc2c(s1)C(C)(C)CCC2 C(=O)(C1CCc2c(Cl)cccc21)NCCNC(C=Cc1cnc(OCC)nc1)=O CCCC(C)(CCC)C(=O)NC1CCOCC1C(=O)NCCCCCN(C)C c1(CC(C(=O)NCCN(C(C(C)(C2CC2)NC(C)=O)=O)C)C)ccc(F)cc1F N=c1cc(C(N2CCC(CCCNC(c3cc(Cl)no3)=O)CC2)=O)cc[nH]1 N1(C(=O)CCCCO)CCC2(CCCN2C(C2CCCCS2(=O)=O)=O)C1 C(=O)(C1COc2ccc(Cl)cc21)N1CCC(N(C(C(=O)NCC=C)C)CCO)C1 c1(C(N2CCOC(CCF)C2)C(=O)NCC)c(C)nn(C)c1Cl C1(CC=C)(C(=O)NCC(C)(O)CNC(c2ccc(CC)[nH]2)=O)CCCC1 C1(NC(C2(C)CCCC2)=O)CC2CC(NC(=O)CCN3CCOCC3=O)C2C1 Cc1ccc(O)c(C(N2CCCC2C(C)NC(=O)COCc2nnc(C)s2)=O)n1 O=C(C#CC1CCCOC1)NCC12CCC(CC1)N2c1cnc(C(=O)OC)cn1 Cc1nnc(CCC(=O)NCC2CC2CNC(C2CC=CCC2C)=O)n1C C1(C(=O)OC)Cc2cc(Br)ccc2N1C(c1cccc(C(=O)N(C)C)c1)=O C(=O)(C(C)(C1CCC1)NC(C1CCNC1=O)=O)N(CC#C)CCF c1(C(=O)NC(CC(C)NC(C2CCCO2)=O)C)cccnc1O c1(C(N2C(C)CC(CC(=O)NCCc3ncon3)C2)=O)nnc(O)nc1O c1(C(=O)NC2C(NC(C3CCC(COC)C3)=O)COC2)ccc(Br)cc1 c1(NC(C2CC3CC3N2C(=O)C=Cc2cnccn2)=O)ccc(Cl)nc1Cl C1(C(=O)NCCCN(C(c2ccc(SC)s2)=O)C(C)C)CC2CCCCCC12 CCC(C)C(O)C(=O)NCCN(C(c1ccnc(OCCOC)c1)=O)CC C1(NC(C(CC)(C)O)=O)CCN(C(C23CCCN2CCC3)=O)CC(C)(C)C1 Cc1ccc(C(=O)NCC2(F)CC(NC(c3nncs3)=O)C2)cc1 N1(C(C(C)OCCN(C)C)=O)CCC(C(=O)NCC(F)(F)C(F)F)(OC)C1 C=CCC(C)C(=O)NCCC1CC(NC(c2cn(C)c(O)n2)=O)C1 N1(C(c2ccc(COC)cc2)=O)CCN(C)CC1CNC(=O)C=CC1CCCO1 C1(NC(CCOCC#C)=O)CC(NC(c2cnco2)=O)C(O)C1 c1(OCC)nc(Cl)ccc1S(=O)(=O)Nc1nnc(C2CCCCC2N=[N+]=[N-])s1 N1(C(CC(COC)C)=O)CCC(C(F)(F)F)n2nccc21 CC1(C)CCC1NC(=O)CCC1CCN(C(C2COCCO2)=O)C1 C1(NC(CC=C)=O)CCN(C(=O)CCC23CCC(CC2)C3)CC(O)C1 c1(N2CC(SC)C2)ccc(S(=O)(=O)NCc2nn(C)cc2C)cc1C#N c1(C(C)N(C(=O)C=CCNC(=O)CC2CCSC2)C)cccs1 C(CCC(C)C)(C(=O)NC1C2CCCC1CO2)NC(CCCCC#C)=O C(=O)(CC1=NN(C)C(=O)C1)NC1CN(C(CC2(OC)CCOCC2)=O)C(C)C1 C#CCC(CC(=O)NC1(CC)CCCCCC1)NC(c1ccc(O)c(F)c1)=O O(Nc1ncnc2c(Br)cc(F)cc12)Cc1ccc(OC=C)cc1 c1(NC(C2CN(C(=O)CC3CC4CCC3C4)CCN2)=O)ccc(Br)cc1 Cc1c(C(=O)NCCC2(NC(=O)CCCC(N)=O)CCC2)sc2cccc(F)c12 Cc1cc(-n2cc(C3(C)CN(C(=O)C(CO)N(C)C)C3)nn2)cc(C)c1Br C1(CNC(C2CC(CC)C2)=O)CC(C(=O)N(CC(C)C#N)C(C)C)=NO1 C(CC(=O)N1CC(CC2CC2)C1)(C(F)(F)F)NC(c1nc(N(C)C)oc1)=O C1(NC(=O)C2CC2)CC2CN(C(c3ccc(-n4cccn4)nc3)=O)CCN2C1=O C1(c2nc(C)on2)CCCN(C2CCN(CC3CC(=O)N(C)C3)CC2)C1 Cc1nc(CC(C)C)oc1C(=O)N(CC(C)(C)CNC(=O)CC(C)(O)C1CC1)C c1(C2N(c3cc(S(C)(=O)=O)ncn3)CCC2)ccc(S(C)(=O)=O)c(F)c1 C1(CCNC(=O)CCc2cnco2)CCC(NC(c2ccoc2Br)=O)C1 Cc1cnc(NCC2CN(C(c3csc(Cl)c3-c3ccccc3)=O)CC2C)nc1O C#Cc1cncc(C(=O)NC(C)C(C)NC(c2c(C)ccn2C)=O)c1 c1(C(C)NC(C23C(CN(S(C(C)C)(=O)=O)C2)C3)=O)cc2ccccc2cn1 C(C(=O)N=c1ccn(C2CCC2)[nH]1)N(C(=O)C(N1CCCC1=O)C)CCCC N1(C(C(C)(C)C)=O)CCC12CN(C(=O)CC1CCNCC1)C2.c12ccc(cc1)o2 C12COCCN1C(=O)CONC(=O)N(C)C2.Cc1cc(OC(C)(C)C)no1 C(C(CC)(CC)NC(=O)C(CC)n1ccc(C2CC2)n1)NC(C(CC)NC(C)=O)=O N1(C(C2CCN(C(C)C)CC2)=O)CC(NC(=O)CN(S(C)(=O)=O)C)C(C2CC2)C1 Cc1ccc2c(=NCc3cccnc3Cl)[nH]c(N3CCCCC(C)C3)nc2c1 CC(Cn1cccn1)C(=O)NCC1(C(=O)NCC2CC2Cl)CC1 Cc1c(Br)c(C(=O)NC(CNC(C2COCCO2)=O)C(C)C)nn1C c1(CC)ccc(C(=O)NC2CN(C(c3ccccc3NC)=O)CC23CC3)c(C)n1 c1(CC)onc(C(=O)NCC2(F)CC(NC(=O)Cc3cncc(O)c3)C2)c1C c1(C(=O)NC2CC2CNC(c2c(F)cc(F)cc2F)=O)cc2cc(F)ccc2s1 C1(NC(C2CC23CC3)=O)CCN(C(c2cnn3cc[nH]c(=O)c23)=O)CC12CCC2 C1(C(=O)NC(C(C)OC)C(=O)N2CCC2CC2CC2)CCC(C)(O)CC1 c1(C(N(CC(C)N(C(=O)CN(C)C(N)=O)C)C)=O)csc(=N)[nH]1 C(=O)(C1=NNC(=O)CC1)N1CCCC(N(C(=O)CC2CC2)CCN2CCCC2)C1 C1(O)(C(=O)OCC)CN(C(=O)NC(C2CCCCC2)C(=O)OC(C)(C)C)CC1O CC1CC(NC(=O)C(C2CCCCC2)=O)CCN1C(C1CSCC(=O)N1)=O c1(C(N(C)CC2CCCN2C(C2CCNC2=O)=O)=O)cc2c(O)ncnc2cn1 C1(C(N2CC(CNC(c3cnc(C(C)=O)s3)=O)C2)=O)CCc2nn[nH]c2C1 Cc1oc(C)c(C(=O)NCC2(NC(c3c[nH]c(C#N)c3)=O)CC2)c1Br c1(OCC(N2CCN(c3cccc(C)c3)CC2)=O)c(C)nc2ccccn12 C1(CNC(c2cc(C)[nH]n2)=O)CN(C(c2cccnc2SC(F)F)=O)C2CC12 c1(C(N2CC(NC(C3(N=[N+]=[N-])CC3)=O)C(C3CC3)C2)=O)ncn2c1CCCCC2 C12(NC(c3nc(COC)sc3)=O)CCCN(C(c3ccc(F)o3)=O)CC1C2 N1(CC2CC(OCC)C2)C(=O)CN(CCOc2cccc(C#N)c2)C1=O N1(C(C2C(CNC(CC)=O)C2(C)C)=O)CCC(F)(F)CC1 N1(CC(C(C)C)NC(=N)N)CCC2CN(C(C)=O)C2C1.CCCC(=O)O c1(OC)cc(OC)nc(N2CCCC2CNC(c2cc(F)cnc2Cl)=O)n1 CC(C)CC(F)C(=O)NCCOCCNC(=O)CC1CCCCC12CC2 C(=O)(CCC(C)(C)C#N)N(CC(=O)O)Cc1cn(Cc2c(C)nc(CC)o2)nn1 N1(C(C(CSC)O)=O)CCCC2(CCN(C(C3(CC(C)C)CC3)=O)C2)C1 N1(C(CCc2onc(C(C)C)n2)=O)CC2(CCN(C(C3CNC(=O)N3)=O)CC2)C1 c1(OC)c(C(=O)NCC2(O)CCN(C(C3(C(C)(F)F)CCC3)=O)C2)ncnc1C C(CC(=O)NC1CC(C(F)(F)F)C1)(C(F)(F)F)NC(c1nn(C)c(=O)cc1)=O CC(CCC(=O)N1CC=CC1Cn1cc(-c2nccn2C)nn1)N(C)C C1(NC(CC2(N(C)C(CC(N3CCOCC3)=O)=O)CC2)=O)CC(F)(CF)C1.C(=O)OC c1(C(N2CC3CN(C(c4nn(C)c(F)c4)=O)CC3C2)=O)cccc2cnccc12 C1(NC(COCCCOC)=O)C=CCCC1C(=O)NCCCCSC CC(C)CC(C(=O)N(c1nc(C2CCC(C)(C)CC2)cs1)C)c1cccc(Br)c1 N1(C(C(=C(C)C(F)F)CC)=O)CC(NC(C2(C3CCCO3)CCCC2)=O)CC(F)C1 N1(CC(C)C)CCC(NC(=O)C(=O)NCCN(C(C)C)C(C)C)C1 C1(NC(CN(C)C(N)=O)=O)CCN(C(=O)Cc2cc(Cl)sc2Cl)C1(C)C C1(NC(C(C)N(C(=O)COCC(C)C)CCC)=O)CCCN1 Cc1ncnc(O)c1C(c1ccccc1Cl)NC(=O)CCN1CCC(O)CC1 CC(C)(C)CC(C(=O)NCCNC(=O)OC)NC(C1CC=CCC1)=O C(=O)(C(CCC)S(N)(=O)=O)NCC(CC=C)NC(C1CC(n2cnnc2)C1)=O C(=O)(CC1OCCc2sccc21)NC(CNC(c1c(C)c(C(F)(F)F)n[nH]1)=O)C N1(C(CCOCC(C)C)=O)CCN(C(C2(CF)CCC2)=O)CC1 C1(C(=O)NC(C=C)CO)CN(C)CCN1C(c1cnncc1OC)=O CC1(C)C(=O)Nc2ccc(C(N3CC(NC(C4C=CCC4)=O)CC(F)C3)=O)cc21 C(c1ccco1)=CC(=O)NC(C(=O)N(CCCn1ccnc1)C)C1CCCO1 C(=O)(CC(C)(C)N(C)C)N(C1CCN(C(=O)C(C)OC(C)=O)C1)CC Cn1cccc1-c1cc(C(N2CC(CNC(C3CC3c3ccco3)=O)C2)=O)n[nH]1 N1(C(CCC#C)=O)CC23CCCC2(C1)CN(C(C1(CC)CCCO1)=O)C3 N1(C(C(COC)OC)=O)CCC(NC(=O)CNS(N)(=O)=O)C(O)C1 c1(OC)ccc(C(C)=CC(N2CCCN(C(c3ccoc3)=O)C(C)C2)=O)cc1 N1(C(C(C)CN(C)C)=O)CCC2(C1)CN(C(=O)COc1cn[nH]c1)CCO2 CC1(C)CN(C(C2SCCS2)=O)CC1C(=O)NCCC1=CCOCC1 O=C(N=c1[nH][nH]cc1Br)C1=NOC2(CCN(c3ncc(Br)c(C(F)(F)F)n3)C2)C1 N1(C(C2CC(CNC(C3N(C)CC(C)(C)C3)=O)OC2)=O)CCC2(CC1)CN(C)C2 C1(C)(C(=O)NCC2(C)CCN(C)C2)CN(C(=O)C2=NNC(=O)C2)C(C)(C)C1 CCC(CC)C(F)C(=O)NC1CC(C)(CNC(=O)COCc2nc[nH]n2)C1 CCCC(C)CC(=O)N1CCC(NC(c2cnn(-c3ccccn3)c2)=O)C1 C(=O)(C1=CN=C2N=CNN2C1)NCCC1N(C(C(C(COC)C)C)=O)CCC1 C1(C(=O)NC(CC)CCO)CC12CCN(C(=O)C=CC1CC1)C2 C1(NC(=O)Cn2ccnn2)CN(C(C2CCCOCC2)=O)CC1n1cccn1 CC1(C)CCCC(C(N2CCC(c3ccc(C#N)cc3)CC2)=O)O1 CC(C(=O)NC1CCN(C(=O)CCc2nncn2C)CC1O)S(C)(=O)=O C1(C(=O)NC2C(C(=O)NC3CC(C(C)O)C3)CC2)CC(C)(C)CO1 c1(C(=O)NC2CC(C)(CNC(C3CCC(=O)N3)=O)C2)cn2cccnc2n1 C(c1ccc(O)c(O)c1)=CC(N1CC(O)(CNC(CC2(C)CC(F)(F)C2)=O)C1)=O C1(C(=O)NC2CC(NC(c3nc(C(C)=O)sc3)=O)C2)Cc2c[nH]cc2S1(=O)=O c1(C(C)=O)cn(CC(N2CCCC2CNC(c2ocnc2C2CCC2)=O)=O)nn1 O=[N+]([O-])c1cccnc1N1CC(NC2CC2)C1 c1(-c2cc(Cc3n(C)ccn3)c(F)cc2)cc(O)c2ccoc2c1.n12ccnc1C2 N1CC2CC2C1C#N.Cc1cnncc1C(=O)NC1(c2ccc(Br)cc2)CC1 C1(C(=O)NCC2C=CCOC2)(CC)CCN(C(=O)C(O)Cn2cncn2)C1 CCCC(C)C(=O)Nc1ccc(-c2cn(CC3CCCC3)nn2)cc1 C1(CN(C(C(N2CCCCCC2)C)=O)C)CCN(C(=O)CC2CC=CCC2)CC1 c1(C(COCC(N2CC(CCCCNC(C=C(C)C)=O)C2)=O)C)cccc(F)c1 c1(CCC(c2n(CC)nnn2)(C)NC2(C(=O)NC)CC2)cccc(Br)c1 N1(C(C2(CC)CC(C)(C)C2)=O)CCC=C(CNC(c2n[nH]cc2C)=O)C1 C1(NC(c2c(CC)nc(C)[nH]2)=O)CCN(C(c2ncoc2Br)=O)C(C)C1 N1(C(C(C2CC2)OC)=O)CCCC(N(C)Cc2ncc(-c3ccc(C)cc3)o2)C1 c1(CCNC(=O)NCC(N(OCC)C)=O)ccc(C#N)cc1OC N1(C(CC(CNC(C(C)CC#N)=O)C2CCC2)=O)CCC2(COC(=O)N2)C1 c1(C(=O)NCCCN(C(C(C)C#N)=O)CCO)cc(Cl)ccc1CNS(C)(=O)=O C1(CC(=O)NC(CC#C)CC)C2CCCC2N1C(=O)CC1(C#N)CCOCC1 C(C(C)(C)CNC(=O)C(F)CC1CCCCC1)N(C(=O)C(F)n1cccn1)C C1(OC)CN(C(=O)CCc2ccsc2)CCC1CNC(=O)C(C)COC Cc1ccc2[nH]c3c(c2c1)CC(NC(N1CC(O)CC1(C)C)=O)CC3 Cc1ccc(C(=O)NCC2CC(NC(=O)CCOCC3CC3)C2)nc1O CC1(C)CCC=C1C(=O)N1CCN(C(c2ccc(C(F)F)nc2)=O)CC1C1CC1 N1(C(c2cc(C)nn2C)=O)CCC(NC(C2CC2C(N)=O)=O)C(F)C1 CC1OC2(C(=O)NC(c3cccc(Br)c3)CC3CC3)CCC1CC2 CCCCCC(O)C(=O)N1CC2(C(=O)NC3CCCC(F)(F)C3)CC1CO2 N1(C(CCc2n(C)cnn2)=O)CCCCC1CCNC(C1CC2CC1C2)=O C1(C2CCN(C(CCNS(CC)(=O)=O)=O)C2)CC(C)CCC1O n1(C(C)C)cc2c(n1)CC(C(=O)OCC1CCOCC1(C)C)CC2 CC1(C)CN(C(C23CCC(CC2)C3)=O)CC(C)(C)C1NC(=O)CCC1CCOC1 C(c1ccc2ncccc2c1)=CC(=O)NC(C)CCNC(=O)Cc1ccccn1 CC1(C)CCc2cnc(SCCON3CCN(c4cncc5nnnn45)CC3)nc21 N1(C(=O)NCCCC)CCC2(CCN(C(=O)Nc3ccc4ccccc4c3)C2)C1 c1(N2C3CC(NC(C4(CC)CCC(O)CC4)=O)C2CC3)ncnc2[nH]ccc12 N1(CC(=O)NCC(O)CCNC(c2cncc(Br)c2)=O)CC2CCC1C2 C1(C(=O)NC2CC(NC(c3cc(C(N)=O)[nH]n3)=O)C2)CCn2ncnc2C1 C1(CC)(CC)CCN(C(=O)C(C)N(C(=O)C(CC2CC2)OC)C)C1 C(=O)(C1=COCCO1)N1C(CNC(C2CC3(CCO2)CC3)=O)CCCC1 Cc1nc(N(C)C)sc1C(=O)NCC1CN(C(=O)C=Cc2ccn(C)c2)C1 N(C(=NCCC1CC(C)OC(C)C1)NC1CC(C)(F)C1)C(C=C)C C1(NC(c2ccc(CSC)o2)=O)CC(C)CN(C(=O)COCCN(C)C)C1 CC1CCCC(C(N2CCC(N(CC(=O)Nc3ccccc3)C)CC2)=O)C1 N1(C(C(CC#C)(C)C)=O)CC(NC(=O)CC=CCC)CC2(CC2)C1 CCC(C(=O)N(CC(C)NC(c1cc(C(C)(F)F)ccc1C)=O)C)C(C)(C)CC C1(NC(C(CCCC)(C)F)=O)CCC2(CC1)CC(NC(=O)CNC(=O)OCC)C2 Cc1ccc(C(=O)NC2(CO)CC(C)(C)C2)c(-n2cc(-c3ccnn3C)nn2)c1 CC(C)(C#N)CC(c1nnnn1Cc1cccs1)NC1CCCC1n1ccnn1 C(CC(C)(C)C)(C(=O)NCC1CCN1C(C1(C#N)CC2(CC2)C1)=O)OC c1(C(=O)NC2C(NC(c3cc(C)sc3)=O)CC2)c(C)noc1C(C)C CC1(CNC(=O)C(O)C(F)(F)F)CCCN(C(=O)CNC(N2CCCC2)=O)C1 Cc1ccc2nc(C)c(C(=O)N(CCNC(C34CCC3C4)=O)CC3CC3)cc2c1 C(=O)(C(C(C)C)N1CCCC1=O)N1C(C(C)NC(Cc2c(C)con2)=O)CCC1 c1(C(CC)CC)nc(C(O)C(c2ccccc2F)C)n(-c2ccc(SC)cc2)n1 C12(C(=O)NC(CC=CC)CO)CN(C(=O)OC(C)(C)C)CC(F)(C1)C2 c1(OC)ccc(C(=O)N(CC(C)CNC(=O)Cn2c(C)c(C)sc2=O)C)c(F)n1 c1(C(N(C)CC2(NC(C(C)=CC3CC3)=O)CC2)=O)ccc(OC(F)(F)F)c(C)c1 C1(C(=O)NC2(CO)CCCN(C(=O)C3=CCC3)C2)CN2CCCN1CC2 N1(C(CS(=O)(=O)NCC)=O)CCCC(CC)(NC(=O)Cc2ccccc2)C1 Cc1nccc(C(N2CCCC(CN(C(=O)CSc3n[nH]c(O)n3)C)C2)=O)n1 Cc1cc(C(=O)NC2CCC(CNC(C3(C)COCCO3)=O)C2)cc(N)c1Cl C1(C)(NC(C(C2CCCC2)OC)=O)CN(C(=O)C=C(C)C(C)C)C(C)(C)C1 C1(C(N2C(CNC(c3cc(OC)nc(C)c3)=O)CC2)=O)CCn2nncc2C1 N1(C(C(C)CCCc2ccccc2)=O)CC2(C1)CN(C(=O)C(F)C(C)(C)O)CCO2 c1(CC(N2CC(N3C(=O)CC(NC(C=CC=CC)=O)C3)C2)=O)ccc2[nH]ccc2c1 Cc1nc(CC(C)C)oc1C(=O)NC(C)(CNC(c1coc(C(F)F)n1)=O)C1CC1 C1(OC)CC(CNC(c2ccc(O)cn2)=O)N(C(c2ccc(F)o2)=O)C1 c1(SC)ccc(C(=O)NCCC2(NC(=O)CC(C)C3CCCO3)CCCC2)cc1 CC1CCc2n[nH]cc2C1C(=O)NCCN(C(c1sccc1C1CC1)=O)C1CC1 c1(C(N2C(C)(C(=O)Nc3nccc(OC)c3I)CC2)=O)cnn2cccnc12 C1(=O)CC(C(C)(C)C)Nc2cncc(c2)N1.C=CCC(CC)n1cc(COC)nn1 Cc1cncc(C(N2CCCC2C(C)(C)C(=O)NCc2ncc(C)s2)=O)c1 c1(C(=O)NCC2C(CNC(CCCC)=O)C2)c(F)ccc(C)c1Cl C1(NC(c2cc(C(C)(F)F)n[nH]2)=O)CN(C(=O)C(C)(C)C(F)F)CCC1CO Cc1nc(N2CCCC(Cc3cccc(F)c3)C2)sc1C(=O)NCCC(=O)NC C(CCCC(=O)NOC(CO)C(C)C)NC(CC(CCOC)(C)C)=O N1(C(C(CC)O)=O)CCC2CCC(C1)N2C(c1c(F)ccc(C#N)c1F)=O C=CCC(C)(CC)C(=O)NCC1COC(CNC(C23C4C5C2C2C3C4C52C)=O)C1 c1(C(=O)NC2CN(C(=O)CCc3ccncn3)C2)c(Cl)ccc(Cl)c1O c1(N2CCCN(C(c3c(OC)cccn3)=O)CC2)ncnc2ccc(O)cc12 C(=O)(C(F)C(C)CNC(=O)C(COC)COC)N(C1CC(=C)C1)C C1(C(=O)NC2CCC(CNC(=O)Cc3cncn3C)C2)(NC(C)=O)CCCCC1 C1(NC(C)C(C)n2cccn2)CC(=O)N(CCc2ccccc2O)C1 CC1CCCCC1(CNC(=O)CN(c1ccncc1)C)NC(=O)C#CC1CC1 Cc1c(C(=O)NC(C2CCOC2)CNC(=O)C(F)=CC2CC2)cnc2ncnn12 C(=O)(N(CC)OC)C1(CC=C)CN(C(C2CCCN2C2CC2)=O)C1 N1(C(c2sccc2C(F)F)=O)CCC2CN(C(=O)CCc3nncs3)CC2C1 c1(C(N2C(CC)(CC)CC2)=O)n[nH]c2c1CN(C(c1cnncc1NC)=O)C2 c1(C(=O)OC)c[nH]c(=NC2CCCC(NC(=O)CC3COCCO3)C2)cn1 CCS(=O)CC(=O)N1CC(C)(CCC(=O)NCC(C)(COC)OC)C1 n1(CC)nc(C)c(C(=O)NC2C=CCN(C(C3CC3C(=O)NC)=O)C2)c1Cl c1(C(N(CC(C)(C)NC(C(C)NC(=O)OC)=O)C)=O)sccc1SC S(=O)(=O)(c1cccc(CN)c1)Nc1c(=O)cc(C(=O)OC)n(C)c1 C12(C(N(CC(=O)OCC)C)=O)CC(C)(CN1C(=O)CSc1cn[nH]c1)C2 C1(NC(C(C)OCC=C)=O)CN(C(c2cn(CCOC)nn2)=O)CC1O C#CCCCCNC(=O)C#CCNC(c1cc(Cl)cs1)=O c1(NCC(=O)NC(CC(C)OCc2nccn2C(F)F)C)ccc(C#N)cc1F C12(C(=O)NCCCCC3CCN(C(C4CC5CC4CO5)=O)CC3)CC3CC1C2C3O N1(C(c2cc(OC)n(C)n2)=O)CCC2CCN(C(c3cncs3)=O)C2C1 N1(C(C2CCN(C3CCCC3)CC2)=O)CC(NC(C2(F)CC2)=O)CC12CCCOC2 C1(C(=O)NCC2C(C)OCC2)N(C(=O)CC2C(C)(C)C2(C)C)CCCC1(C)C C1(CNC(c2cccnc2S)=O)CCCC(NC(C2OCCO2)=O)C1 c1(N(C(C2=NOC(c3n(C)ncc3)C2)=O)CCC#N)nc2cc(C)cc(C)c2s1 C(=O)(C1=C2CCN=C2NC=C1)N1C2CC(CN(C(C34CCC(C)(OC3)C4)=O)C2)C1 CC1C(NC(=O)C(Cl)=CCl)CCCN1C(C1CC1c1ccccn1)=O C1(c2cn(C(C(=O)NCC3(OCC)CC3)C)nn2)CC(F)(F)C1(F)F c1(C2(C(=O)NC3CN(C(C=CC(CC)C)=O)CC3C)CC2)ccc(Cl)c(Cl)c1 C12C=CC(C1)CNC(=O)COC1CC1C(=O)N2.c1(COC)cccs1.C1CO1 c1(C(=O)NC2CC(NC(C3N(C)C(=O)CCC3)=O)C2)cc(Br)c(F)cc1F C(=O)(C1CCCc2cccnc21)N1CC(OC)(CNC(C2CC(=O)CO2)=O)C1 C(=O)(C1=NOC(CNC(c2cc(C3CC3)[nH]n2)=O)C1)N1CCCC(C(C)O)C1 CCC(O)CC(=O)NCCC(C(=O)NCC(C)C(=O)OC)OC N1(C(C2(CNC(=O)CC3C=CCCC3)CC(=C)C2)=O)CCC2(CCN(C)C2)C1 c1(C(N2CCCC(N(C(c3c(CC)cno3)=O)C)C2)=O)ccc(F)c(OC)c1F N1(C(C2(C)CC2(F)Cl)=O)CCC(C2CC2)C1CNC(=O)C1=COCC1 O=C(CCCC1CCCO1)NCC(O)C(=O)NCCc1ccncn1 C1(C(=O)NC(CO)CCO)C=CCN1C(c1cc(Cl)ns1)=O C(=O)(CCCC(F)(F)F)NCC(C)(CO)NC(c1ncc(C(N(C)C)=O)nc1)=O C1(C(=O)OC)CC(F)(F)CC1C(N1CCC(O)(CNC(=O)CN(C)C(C)C)C1)=O CC1CC2CN(C(=O)C(F)CC3CN(C(C4CCC5(CC5)C4)=O)C3)CC12 C(c1ccc(F)cc1)=C(C(=O)NC(CCNC(CC(CC)O)=O)C)C C(=O)(CC(C)C1CCCCC1)NCCC(C)N(C)C(C1(F)CCCC1)=O C1(CNC(C2CCC(C)CC2)=O)CCN(C(=O)C(C)Cn2cccn2)CC1O C1(NC(=O)CC2(C3CC3)CC2)CC(NC(c2csc(Cl)c2Cl)=O)C12CCC2 CCC(CC)(CCNC(C1CCN(C2CC2)S1(=O)=O)=O)NC(C1CC1F)=O CC1(C)Oc2ccc(NC(c3c(F)cc(Br)cc3Cl)=O)cc2O1 c1(C(N2CC3C(N(C(c4cc(CN(C)C)on4)=O)C)C3C2)=O)cccc(Cl)c1F C1(C(=O)NC(C2CCC2)C)COC2(C1)CN(C(=O)C(C)(C)F)C2 Cc1nc(CC(C)C)sc1C(=O)CNC(C1C2CN(C3CCSC3)CC12)=O CCCS(=O)(=O)CC(=O)NC1COCCN(C(=O)COCC(=O)OC)C1 C12(CNC(C(F)=CC)=O)CCCC1N(C(=O)COCP(C)(C)=O)CCC2 C(=O)(CC(C)(C)CCC)N1CC(CCC)N(C(c2cc(Br)ccc2O)=O)CC1 c1(C(=O)NC2CCC(CC)C2)sc(S(N)(=O)=O)c(OC)c1OC N1(C(CCNC(C(C)(C)C)=O)=O)CC(NC(=O)C2=C(Cl)CCCC2)CC(F)(F)C1 CC1=C(C(=O)N2CC(NC(c3cc(C4CC4)[nH]n3)=O)CC2(C)C)COCC1 c1(C(=O)NC(C2CCN(Cc3nccs3)CC2)C)cc(Br)c2ccccc2n1 c1(C(=O)NC2C(C)(CN(C(CCOC)=O)C)CCC2)ccc(Cl)c(N)c1 Cc1cnnc(O)c1C(N1CC(C(=O)NCC2CCC2C)CC(C)C1)=O c1(N(C(=O)CN2CC(C(N)=O)C2)CCCCNCC(=O)OC)cccnc1NC.CO c1(Nc2cc(NCCCOCCCO)nc(C)n2)cc(Br)c(F)cc1C CC1(C)CC(CNC(=O)C=Cc2ccco2)N(C(C2CC=CCC2)=O)C1 N1(C(c2c(Cl)csc2Cl)=O)CC2(C1)CN(C(C1(CO)CCC1)=O)CCO2 c1(OC)c(C(=O)NC2CC23CCN(C(=O)CO)CC3)cccc1[N+](=O)[O-] Cc1ccc(C(C)NC(N2CCC(Nc3ncccn3)C2)=O)s1 c1(C(=O)NC2C(NC(CCn3ccc(C)n3)=O)CC2)ccnc(N(C)C)c1 Cc1cocc1CN(Cc1ccccc1)CC1CCC1 Cc1cc(F)sc1C(=O)NC1CCCC1CNC(c1csc(Cl)c1Cl)=O C1(=CC(=O)NCC2C(CC(=O)NCCCCOCC)C2)CCCCC1 N1(C(C2(OC)CCSCC2)=O)CCCC2(CCCN2C(=O)C(C)CSC)C1 C1(CC(=O)NCc2nc3c(s2)CCC3)CC2(CCNC2)CO1 C(CC)(CC(F)F)Nc1ccc(NC(=O)NCCOCCCCCC)cc1 C(C(C)(C)CN(C(=O)CC1CCC2CC12)CNC(=O)COCCCF)OC N1(C(C(C)CC2CC2)=O)CCCC2C1CCN2C(C12COC(CF)(C1)C2)=O c1(CCC(N2C(CNC(C3C(CC)CCO3)=O)CCC2)=O)ccc([N+](=O)[O-])cc1 C(CCC(C(=O)N1CC2(CCC1CO)CC2)NC(=O)C(F)(F)C(F)F)OC C1(N(C(c2cnc(CC)s2)=O)C)CCCN(C(=O)CC(c2cccc(F)c2)C)C1 c1(CN2C(C(=O)Nc3cccc(O)c3)CC3CC32)c(Cl)cccc1[N+](=O)[O-] c1(CNC(C2CC(C)(NC(=O)C=Cc3nccs3)C2)=O)ccncc1F C1(CNC(C=CCN(C)CC)=O)C(CC)CCN1C(C1CC12CCCC2)=O c1(C(N(C)CC2CCCN2C(c2ccc(Cl)o2)=O)=O)cnn2c1CC(F)(F)C2 Cc1cc(CNC(=O)C=CCSCCC(C)C)oc1C(=O)NC1(O)CC(CO)C1 c1(C(=O)NC(C)(C)CCCNC(c2cn(CC3CC3)nn2)=O)ccc(Cl)cc1Cl Cc1ccc(CC(=O)NCCCCC(C)NC(c2cn(C(F)F)cn2)=O)c(C)c1 C(=O)(CC(C(F)F)n1cccn1)NC(CC)(CC)CCN C(C)(C)(CN=c1nc(SC2CC2)[nH]s1)C1CCN(C(C(C)CN(C)C)=O)CC1 CC1CN(C(C2(CC3CC3(F)F)CCC2)=O)Cc2cncnc21 c1(C(=O)NCCC(C)NC(C2(CCC)CCC2)=O)nnn2c1C(=O)NCC2 C(CC(C)(C)C)(C(=O)N1C(CC(N2CC(OC(C)C)C2)=O)C2CCCC12)OC c1(CC(=O)NC(COC)C(=O)NCc2cocn2)cncnc1O C1(C(N2C(C(C)O)CCC2)=O)CCCC(NC(C2CCN(C)C2)=O)CC1 c1(C(=O)NC(CCSC)C(=O)NC(C)C(=O)NO)cncc(F)c1C C1(c2cn(C)nc2)CN(C(C2(CF)CCC2)=O)CC1NC(C1CCOC1)=O N1(C(c2cc(C)[nH]n2)=O)CC2CC(C)N(C(=O)C(C3CCCO3)C3CC3)C2C1 C1(OCC)CCN(C(c2ccc(C)cn2)C(=O)NCc2ccccc2)CC1 CCN=C(NCc1cc2cc(C(=O)OC)sc2s1)N1CCCC(C(C)C)C1 c1(CN)nc2c([nH]1)CCN(C(=O)Nc1ccc(Oc3ccc(Cl)cc3)nc1)C2 c1(C(=O)NCC(CNC(c2coc(Br)n2)=O)OC)cc2ccccc2cn1 c1(SCC(=O)NCC(N(C(=O)C(F)n2ccnc2)C)C2CC2)cnn(C)c1 C(=O)(CCCCC(=O)NC1CN(C(=O)C=Cc2ccccc2)CC1N=[N+]=[N-])NC c1(C(=O)NC(CNC(Cc2c(C)n(C)nc2)=O)C(C)C)coc2c1COC2 C1(CC(=O)NC2(c3ncco3)CCC2)CCN(C(=O)CCc2cnn[nH]2)C1 Cc1nccnc1C(CNC(=O)NC(C)(C)Cn1ccnc1)N(C)C N1(C(c2c(C)nc(C3CC3)[nH]2)=O)CCCC(C)(C)C1CNC(C1CC1CF)=O N1(C(C2CC(CC)C2)=O)CCCN(C(c2nocc2C2CC2)=O)CC1C(C)C N1(C(C(CSC)O)=O)CC2(C(N3CCC3CN=[N+]=[N-])=O)CCC1CC2 c1(OC)ccc(F)cc1S(=O)(=O)NC1CCN(C(C2CCCN2C(C)=O)=O)CC1 c1(CNC(c2cncc(C#N)c2)=O)ccc2cncn2c1 C(C(=O)NCC(C)(C1CCC1)NC(c1occc1C)=O)(C(C)C)c1cnc(C)s1 CN1CCC(CC(=O)NCC2CC2NC(c2ccoc2Cl)=O)C1=O C(=O)(C(C)CC(N)=O)NCCC1(OC)CN(C(=O)CN2CCC2C)C1 Cn1nc(C(=O)NCc2csc(CNC(c3ncoc3C(F)F)=O)n2)cc1O c1(OC)ccccc1CCC(=O)N1CC(C(C)NC(=O)CSCC(N)=O)C1 C1(NC(CN(CCC)C)=O)CN(C(=O)Cn2nc(C)oc2=O)C2CCCCC12 CC1(Cc2cccc(F)c2)CCCN1C(=O)C(=O)Nc1ncccc1Cl CN1CCC(C)(C(N2CCC(NC(=O)CC3(C)CC(F)(F)C3)C(O)C2)=O)CC1 C1(NCC(=O)NC(CCOC)(C)C)CC2(C1)CC(O)(C(F)(F)F)C2 N1(S(CC(=O)OCC)(=O)=O)CC(CO)C2(CN(C(c3cc(F)c(Cl)nc3Cl)=O)C2)C1 c1(C(=O)NC(CCC)CNC(c2cc(CC)sn2)=O)cnc2cccc(C)n12 C1(O)(CNC(CCCN(C)C)=O)CCN(C(c2ccc(CCF)cc2)=O)C1 C1(C(=O)Nc2ccc(F)cc2)CCCN(N2CCC(n3cccn3)C2)C1 CN1CCN(C(C2CCC(=O)N(C)C2)=O)C(C(=O)NOC2CCCCC2)C1 N1(C(c2n(CCOC)ncc2)=O)CCCCC(CNC(=O)C(F)=C(C)C2CC2)C1 c1(CC(=O)NC2CC(CCNC(C(N3CCN(C)CC3)C)=O)C2)cc[nH]c(=N)c1 CN1C(=O)CCC12CCN(C(C1CCOCC13CCC3)=O)CC2 c1(CCC(=O)NC2C(NC(c3c(C)ncn3C)=O)CC2)ccc(F)c(F)c1F c1(CC)cc(C(N2CCCC2CN(C(c2csc(Cl)c2)=O)CCOC)=O)ccn1 Cc1cccc2c(C(N3CCOCC3CNC(=O)C(C)OCC(C)C)=O)coc12 C(=O)(CCS(N)(=O)=O)NCC(CC)(CC)NC(c1cn(CC)nc1C(F)(F)F)=O N1(C(CC2C(C)C2(F)F)=O)CCCN(C(=O)C=CC(=O)N(C)C)CC1 c1(NC(c2c(-c3c(F)cccc3F)cncc2F)=O)cccn2nccc12 N1(C(CCc2nc(C)c(C)[nH]2)=O)CCC2CN(C(=O)CNc3ccncc3)C2C1 C1(NC(c2n[nH]c(CC)c2C)=O)CCCC(C(=O)Nc2ccc[n+]([O-])c2)CC1 C(C)(C)(CCCCC(=O)N1CCCC(CN(C)C(c2cccc(O)n2)=O)C1)OC CC12CCC(C(N3CC4CCCC3(CNC(c3cccnc3)=O)C4)=O)(CC1)CO2 C(=O)(C(CNC(C1(C)CCCC1O)=O)CC1CCCC1)NCC1(C)CCC1 C(=O)(CC(C)C(=O)OC)NCCC(=C)CNC(C1(COC)CCC1)=O c1(CC(=O)NCC(C)(C)OCC(=O)N(C2CCCC2O)CC)cc(C)nn1C c1(C(=O)NC2CC(C(N3CCN(C(C)=O)CC3)=O)C2)cc([N+](=O)[O-])cnc1C C#CC1CC2CCC1N(C(C1(C(C)C)CCCN1C(=O)CCN=[N+]=[N-])=O)C2 Cc1coc(C(c2nnnn2CC2CC2)NCC2CCCCO2)c1 c1(N2CC(NC(c3ccc(COC)[nH]3)=O)C(C)CC2)ncc([N+](=O)[O-])cc1Br c1(OC)nc(C)ccc1C(=O)N(CC(C)O)CCNC(=O)CCc1cc[nH]n1 c12ccc(c([N+](=O)[O-])c1)NC1CN(CC1C)C(=O)C2.C1(C=O)CC1C(C)O.CO O=C(C1Cc2c(Cl)cccc21)N1CC(COC(=O)CC2CCCCC2)OCC1=O C1(CNC(C2C(OC)CCC2)=O)CC2(CO1)CN(C(c1cc(Cl)ccc1F)=O)C2 C(CCS(N)(=O)=O)c1cn(C2C(C3CC(NC(CSC)=O)C3)CCC2)nn1 N1(C(c2ccc(C)nn2)=O)CCC(CNC(c2nnc(O)cc2O)=O)C1(C)C N1(CC(=O)NCC2(NC(CNC(=O)NC)=O)CCCC2)CCS(=O)CC1 N1(C(C2C(=C)C2)=O)CCc2c(c(CNC(=O)CCc3cccnc3)nn2C)C1 c1(C(=O)NCC2CC(NC(Cc3nc(C)oc3)=O)C2(C)C)cc(C#N)ccc1Cl c1(C(C(=O)NCCC)N(CCCCOC)C)csc2c(Br)cccc12 N1(C(CNC(CCCCC)=O)=O)CC(NC(c2ncn(C(C)C)n2)=O)CCC1C Cc1oc(Br)cc1C(=O)NC1CCN(C(C23COC(CF)(C2)C3)=O)C1C1CC1 c1(C(N(C2(CC=C)CCNCC2)C)=O)ccc(Cl)c(Cl)c1 C1(CCNC(c2c(C#C)c[nH]n2)=O)CN(C(C23CC(C)(C2)C3)=O)CCS1(=O)=O N1(C(CC2(C#N)CCC2)=O)CC23CCCCC2(C1)CN(C(=O)CCN1CCC1)C3 CCC(C(=O)N1CC(CC(=O)NC(C)CN=[N+]=[N-])(OC)C1)n1cncn1 C(c1ccco1)=C(C)C(=O)N1CC(C(O)C(=O)N2CCC2NC(=O)C2CC2)C1 N1(C(c2c(C(C)C)cco2)=O)CCCCC(NC(=O)CCCC(F)F)C1 c1(C(=O)NC2CCN(C(C(C(=O)OCC)OC)=O)C2CC)cccn2nccc12 C(CC(=O)NCC1CC1NC(C1(C(N)=O)CC1)=O)(C(C)C)OCC c1(OC)ccc(F)cc1C(F)(F)C(=O)NC(CNC(=O)C(O)CSC)CC(C)C CCC(C(=O)NC(C)CNC(=O)NC)NC(=O)C=Cc1ccsc1 c1(CC)nnc2cc(NC3CC(NC(=O)CC4CC(C)(C)CO4)C3)ncn12 C1(C(=O)NC2(C)CC=CC2)CCN(C(=O)C(O)C(F)(F)F)C(C)(C)C1 C1(C(=O)NCCC2N(C(C(C)SC)=O)CCC2)CC2C=CC1O2 C(CC(=O)N1CC(C)(CO)CC1(C)C)(C(C)(C)C)NC(COCC(=O)NC)=O CN(CCCC(=O)NCCC1(CNC(c2cncc(Br)c2)=O)CC1)N=O c1(COC)nc(NCC2CC3OCCCC23)cc(=NC2CCOC2C)[nH]1 C1(N(C)C(c2cnc(C(C)(C)C)o2)=O)CN(C(C2CC23CCCC3)=O)CC1(C)C C(CN=c1[nH]cncc1I)C1CCC(NC(c2ccoc2Cl)=O)C1 C1(C=C)(C(N(C(C#C)C)C)=O)CCN(C(c2cc(Cl)c[nH]2)=O)C1 c1(NC(=O)NC2CCC(CC)C2)cnc2c(c1)c(=O)n(C)c(=O)n2C N1(C(C(C)n2cccn2)=O)CCN(C(=O)C2=COCC2)CC1c1ccccc1Cl Cc1cc(C(C2CCC2)NC(=O)C(=O)NC(C)C(C)CC)c(C)o1 C1(CC)COCCN1C(=O)C(CC1CCOCC1)NC(c1ccnc(CO)c1)=O CCCCCC(CC)C(=O)NC1(C2(C(=O)OC)CCCCC2)CCC1 C(=O)(C(F)C(C)CNC(C1(F)CC=CC1)=O)NC(CC#C)C(=O)OC N1(C(C(CC(C)C)F)=O)C2CCC1CN(C(C1CCS(=O)(=O)CC1)=O)C2 C(=O)(CC(C)(C)CCOC)N(C(CNC(C(C(C)C)NC(=O)OC)=O)C)C c1(OC)ccc(CC(C)C(=O)NC(CNC(=O)CNC(N)=O)C(C)C)cc1OC C1(C(=O)NCC#N)CC12CCN(Cc1ccc(O)cn1)CC2 c1(C(=O)NCC(C)NC(=O)C2Cc3c(Cl)cccc32)nnc(O)c2ccccc12 c1(NC(C(N2CC(C3OCCC(N)C3)C2)=O)=O)ccc(S(=O)(=O)NCCO)cc1 c1(C(N(C)CCN(C)C(C2CCC3(CC3)C2)=O)=O)csc(N=S(C)(=O)N(C)C)n1 C1(NC(COc2ccc(C)cc2Br)=O)CCCCN(C(=O)C#CC2CC2)CC1 CCCCC(C(=O)N(CCCCN(C)CCOC(C)CC)C)ON=C(C)C n1(C(C(=O)N(C2CC2)CC2(NC(C(C)SC(F)(F)F)=O)CC2)C)cc(Cl)cn1 C(=O)(C1=CCN(C(=O)CNC(=O)OC)CC1)NC(CCSCC)C N1(C(C(C=C)O)=O)CCC(C)(C)C(NC(=O)CC2(CC)CCC2)C1 c1(C(N2CCCC2)C)c(OC)cccc1O.C1C(C)(C)Cn2cc(nn2)CN1.C1(C)CC1 Cc1cc(F)cc(C)c1C(N1CCN(Cc2nccn2C(F)F)CC1)=O c1(C(=O)NCC(C2CC2)NC(c2c(CC)c(C)sc2)=O)cn(C)c(=O)n1C N1(C(C(CC)C)=O)CC(NC(c2cnn(CC(F)(F)F)c2)=O)CC12CCC2 c1(C(N(CC(CC)NC(C2CCCO2)=O)CC)=O)c(C)cc(C)nc1S C(=O)(CS(=O)c1cccc(OC)c1)N1CC(NC(C2CCC2)=O)CC(OC)C1 C(=O)(CS(=O)(=O)CC(F)(F)F)NCC1C(CNC(COCCC#C)=O)C1 N1(C(Cc2nnc(C)o2)=O)CCC(O)(CNC(=O)C(C)Cn2ccnc2)C1 CC(=O)CCN=C(NCc1nnc2n1CCCCC2)N1CCC(c2nncs2)C1 C#CC1CN(C(c2cnc(O)n2C)=O)CCN1C(c1ccc(C)c(C)c1)=O C12(CNC(Cc3cc(C)no3)=O)CC(NC(c3csc(C(C)C)n3)=O)(C1)C(C)O2 c1(C(=O)NC2C3CC(NC(C=Cc4cnc(C)s4)=O)CC32)cn2cnnc2cn1 C=C(C)C1OCCC1C(=O)NC1CC2(C1)CN(C(=O)COc1ccc(CC)cc1)C2 C(=O)(C(C)C(F)(F)F)NCC1CCCN1C(c1n(CC)cc(Cl)c1)=O N1(C(C(CCC)C(=O)OC)=O)CC(NC(C2CC(O)C2)=O)CC12CCOCC2 Cc1ccc(C(C)NC(=O)COC(C)(C)CNC(=O)CC2CC(C(N)=O)C2)s1 Cc1cc(C(=O)NC(C)CN(C)C(c2cccc(C3CC3)c2)=O)ccc1[N+](=O)[O-] C1(OC)CN(C(c2ccc(Cl)c(C)c2)=O)CCC1NC(c1cc(Br)nc(Br)c1)=O N1(C(CCNC(=O)NC)=O)CC2CCCC1CN(C(c1csc3nnsc13)=O)C2 c1(C(N2CCCC(NC(CC3(C)CCCCC3)=O)CC2)=O)cnc2n1CCCC2 c1(CC)cccc(C(N2CCC(NC(C3CCC(C(F)(F)F)CC3)=O)C2)=O)c1N C1(F)(CNC(C(C=C)O)=O)CCC(NC(c2cnccc2C(F)F)=O)C1 S(=O)(=O)(c1cc(Cl)c(Cl)s1)N1C2CN(C(CN3C(=O)CCCC3)=O)C(C2)C1 c1(C(=O)NCCCC(C)NC(c2scnc2Cl)=O)ccc(=O)n(O)c1 c1(N(C)CC2CC2(F)F)nc2c(F)cccc2c(=NC2CC2c2ccsc2)[nH]1 C(c1cccc(Cl)c1)=CC(N1CC(NC(=O)Nc2ccc(CC)cc2)C1)=O N1(C(c2cc(CN(C)C)on2)=O)CC(NC(=O)CC2CCC2(C)C)C2(CCC2)C1 C1(NC(c2c(C)nc(Cl)s2)=O)CN(C(c2c(F)cncc2F)=O)CC(F)(F)C1 C1(C(=O)NCCC(Cc2ccccc2)NC(=O)Cc2ccoc2)CCC(F)(F)C1 c1(OC)nc(C)c(C(N2CCCC2C(C)NC(c2c(C)cnn2C)=O)=O)s1 N1(C(Cc2c(OCC)cccc2)=O)CCCC2CN(C(=O)CS(=O)(=O)NC)CC12 c1(C(=O)NCC(N(C(=O)C(C2CCOCC2)O)C)C2CC2)nn(C)cc1Cl N1(C(c2ccc(OC)c(C(C)(C)C)c2)C(=O)NC)CC(C)C(N=[N+]=[N-])C1 C(CC(C)C(=O)NC12CC(C1)N(C(c1ccccc1SC(F)F)=O)C2)=CC N1(C(c2c(C)ncnc2O)=O)CCCC(O)(CNC(=O)C(F)(F)C(F)F)CC1 CCCC(CC(C)C)C(=O)N1CC(F)CC1CC(=O)N(CCCOC)C N1(C(C(CC)CC)=O)CCCC1C1CCCN1C(=O)COc1ccc(C)cc1 C1(C(=O)NC2(CNC(COC3(C#C)COC3)=O)CC2)CN(C)NC1=O c1(NC(=O)NCC2CCC(C)N2C)ccc2c(Br)nn(C)c2c1 N1(C(CCc2c(C)noc2)=O)CCC(O)C1CNC(=O)CC1CCC(C)CO1 C1(C2CCN(C(=O)Cc3ccc(Cl)nc3)C2)(NC(=O)CC2NC(=O)NC2=O)CC1 c1(C(=O)NC2(C)CCCN(C(c3cccc(Cl)n3)=O)C2)cc2ccc(F)cc2s1 Cc1csc(Cl)c1C(=O)NCc1cccc(NC(=O)COCCF)c1 N1(C(c2cc(CCC)[nH]n2)=O)C2CCC1C(NC(=O)C(C)CSC(F)(F)F)C2 C(=O)(C1=C(Cl)CCC1)N(C1CCN(C(=O)CSc2ccc(F)cc2)C1)CC CC(C)CCCC(=O)NC(CC1CC1)C(=O)NCC(C)(C)C(F)F C(=O)(C(C)(C)C(=O)NCCn1ccc(C(=O)NCCOc2cnn(C)c2)c1)NC C1(C(N(CCCCCCC)C)=O)CCCCC1(C)NC(c1nccc(C)c1N)=O N1(C(c2c(C)nsc2N)=O)CCC(C)C(NC(=O)CC2(C)CC2(Cl)Cl)C1 C1(NC(C=C(C)Cl)=O)CC(CO)N(C(=O)CCC=CBr)C1 N1(S(CC(=O)N(CCOC)C(C)C)(=O)=O)CCNC(=O)C1c1cccs1 C1(NC(c2cc(=O)cc[nH]2)=O)CC2C1CCN2C(c1cc(C(F)(F)F)no1)=O c1(N2CC3CC(NC(c4c(C(C)C)nn(C)c4)=O)C3C2)nc2cc(Br)cnc2s1 C1(C(N(CCNC(C2(C)CC(C(=O)OC)C2)=O)C)=O)COCCC1(F)F CC1CCN(C(=O)C(=O)N(CCCNC(C2CC2Cl)=O)C(C)C)CC1 N1(C(CC2C(C)C2)=O)CCN(C(=O)C(=O)Cc2cccc(F)c2)CC1CC1CC1 C1(C(N2CCC(CN(C(c3cc(C)sc3C)=O)C)C2)=O)CCCNS1(=O)=O CCC(O)CCc1cn(CC(=O)N(CC(N)=O)Cc2ccccc2)nn1 N1(C(c2n(C)ncn2)=O)CCC(NC(=O)CC(C)(C)C2CC2)C12CCC2 C(=O)(CC(O)C(C)CC)NC(CC(=C)Cl)C(=O)NCC1(C(N)=O)CCCC1 c1(OC)cc(OC)cc(C=CC(N2CCN(C(=O)CC3(C)CC3)CC2CF)=O)c1 C1(C(=O)NCCOC2CCN(C(C=CC)=O)C2)CCS(=O)(=O)N1 N1(C(c2ccnc(C(C)C)n2)=O)CC(NC(=O)C2=NOCC2)CC2(CC2)C1 N1(C(N2C(CC)COCC2)=O)CCCC2(C1)CN(C(c1ccc(O)cc1O)=O)C2 C1(CCC(=O)NCc2c(CC)nco2)CCCN(C(=O)C(O)C2CC2)C1 Cc1cccc(C(C)C(=O)NC2(CNC(=O)C=CC3CCCC3)CCC2)c1 c1(C(=O)NCC(C(C)(C)C)NC(c2cnc(CC)[nH]2)=O)cc(C)c(Cl)cc1F C(=O)(CC(C(F)(F)F)NC(C1CCC(=O)N1)=O)NCCc1c(C)nn(C)c1 CC1=C(CNC(=O)NCCn2ccc(C)cc2=O)S(=O)(=O)CCO1 N1(C(C(CC)CCOC)=O)CC2CCCC(C1)N2C(=O)CCC(C)O c1(C(=O)OC)cc(S(=O)(=O)NNC(=O)C(N)CC2CC=CCC2)ccc1Br C1(CC(N2CC(N(C)CC)C2)=O)CN(C(c2cc[nH]c2C)=O)CCC1C N1(C(C=COCC)=O)CCC(O)(C(C)NC(c2cc(-c3cnn(C)c3)on2)=O)C1 N1(C(C(n2ccc(C)n2)C)=O)CCN(C(C2CC=CCC2)=O)CC1CO C12(C)CCN(C(=NC)NC1)CC2.C1(C(=O)OCC)CCCC1C(C)C c1(C(N2CCCC(CCNC(CC(CC)C)=O)C2)=O)cn2cc[nH]c(=O)c2n1 C1(C(N2C(CCNC(=O)Cc3csc(S)n3)CCCC2)=O)CC2(C1)CC21CCC1 CCCCCCC(C)C(=O)NCCC1CCN(C(=O)C2=NNC(=O)CC2)CC1 c1(-n2cc(C(C)(C)NC(C(C)(C)Oc3ccccc3)=O)nn2)ccccc1Cl C1(C(N2C(CCC(=O)Nc3cncc(Br)n3)CCC2)=O)Cc2ccccc2O1 Cc1cc(C(=O)NC(CNC(C2(C(F)F)CCC2)=O)C2CCC2)c(O)c(C)c1 N1(C(c2c(C)ccc(C)n2)=O)CC2(C1)CN(C(C1COC(C)(C)CO1)=O)CCO2 c1(C(=O)OC(c2cc(Cl)sc2Cl)C)cc(O)nn1C C1(O)(C(C)NC(=O)CCc2cnn(C)c2)CN(C(c2[nH]nnc2C(F)F)=O)C1 C(CCCCC(=O)NC1CC(OC2CC2)C1)N(C)C(C1OCC2CCC1C2)=O N1(C(c2c(NC)nccc2)=O)CCCN(C(=O)CC2CCCNC(=O)C2)CCC1 C12(NC(=O)C(F)F)CCOCC1CN(C(c1cc(F)ccc1C(F)F)=O)C2 O=C1NC2(CO1)CC(C(=O)NCC1(NC(C3CC4(CCC4)CO3)=O)CCOC1)C2 C(=O)(C(F)(CNC(=O)CC1CC(C)=NO1)C(C)C)NCc1ccc(CC)cn1 CCC(C)(C(=O)N1CC(NC(c2ccc(Cl)c(C)c2O)=O)C2(CC2)C1)C(N)=O N1(C(c2n(C)cc(Cl)c2)=O)CCC2(C1)CN(C(=O)CC1CCCC(=O)N1)CCO2 CCCCCC(O)C(=O)N1CCCCC1CCCNC(c1cnc(NC)cn1)=O N(C1CC2(CN(C(c3ccn(C(F)F)n3)=O)C2)n2ccnc21)C(=O)C(O)C1CC1 N1(C(c2c(C)onc2-c2ccccc2)=O)C2CCC1CC(NC(=O)CC(C)O)C2 N1(C(c2n[nH]c(C)c2N)=O)CC2CC(NC(=O)C=C3CCC(C)C3)CC2C1 n1(C(C)C)ccc(C(N2CC(NC(=O)CN3CSCCSC3)C(C)C2)=O)cc1=O Cc1c(C(=O)NC(C2CCCN(c3ncnc(=N)[nH]3)C2)C)cnn1CC(C)(C)O N1(C(C2CC(C(=O)OC)C2)=O)CC2(C1)CN(C(C)=O)C2 C1(N(C(=O)CC23COC(C(=O)NCc4ccccn4)(C2)C3)CC)CCS(=O)(=O)C1 N1(C(CC(CC)C)=O)CC(C(=O)Nc2ccc(C)c(I)c2)CC(F)C1 C1(C(=O)NCCCC(c2ccccc2)NC(=O)OC(C)(C)C)CC2CCC2C1 C1(CNC(c2c(O)ncc(CC)c2)=O)CC2CCC(C1)N2C(=O)CS(C)(=O)=O C(=O)(C1=CCCCO1)NCCC(C)N(C)C(C1C2CC3C(C2)C13)=O c1(OC)ncc(F)cc1C(N1CCC(CC(=O)Nc2ncc(CO)cc2Br)C1)=O c1(C(=O)NCCCC2(NC(C3C(CC)OCC3)=O)CC2)cc2cc(Cl)ccc2o1 N1(C(C2C(C(=O)OC)CC2)=O)CCC2(CCN(C(c3csc4nnsc34)=O)C2)C1 c1(C(N2CC(NC(CCCCCOCC)=O)C(C)C2)=O)onc2cc(C)ccc12 c1(C(=O)NC2CCC2NC(c2ncoc2C2CC2)=O)cccc(CF)c1 C(=O)(C1=CC2C=CC(C1)C2)N1C(CCCNC(CCSC)=O)CCCC1 C1(C2CCCN(C(C3(C#N)CCCOC3)=O)C2)(NC(C(CC)C(C)C)=O)CC1 O=S(=O)(c1ccc(OC(F)(F)F)c(F)c1)NC(CC(F)(F)F)C(=O)O C(C(C)(C)CC(=O)NCC1(CNC(c2ccc(N)c(N)n2)=O)CC1)N(C)C C1(NC(CCCCC#C)=O)CCN(C(c2cncc(N)c2)=O)CCC1CO c1(C(=O)OCC)ccc(C(F)(F)F)c(NC(C)Cc2nc(C)no2)c1 C1(C)(C(=O)NC2(CC(=O)Nc3c(CC)csc3)CCCCC2)CCC(=O)NC1 C1(CC(CN(C)C)NC(=O)COC2CCCC2)CCN(C(=O)C(O)C2CC2)CC1 CCC(CC)C(C(=O)N1CCS(=O)(=O)C(CCNC(=O)CC(C)(C)OC)C1)OC C1(NC(C2(CC)CCCN2C(=O)CCn2cncn2)=O)CNC(=O)C1(C)C c1(OC)cc(C(=O)NC(C(N2CCCC2C(=O)N(C)C)=O)C2(O)CCC2)on1 C(=O)(CCC(=O)NN(C)C)N1CCCC(CCC)(NC(=O)C(C2CCC2)OC)C1 N1(C(CCCCC2(C)CC2)=O)CCCC(CNC(=O)CC2CCC(O)C2)CC1 O=C(C1SCc2cccnc21)N1CCC(CF)C1 N1(C(c2c(C)nn(CC)c2C)=O)CCC(C)N(C(c2cnc(C)cn2)=O)CC1 c1(C(C)NC(C(c2cccnc2)C)=O)cccnc1.C12(CCC1)COC(=O)N2 CCC(CC(C)C)C(=O)N1CCCC(Cc2cn(C(C)(C)C)nn2)C1 N1(C(C2N(C(c3cccc(C)c3Cl)=O)CC(C)C2)=O)Cc2cncnc2C1 C12(NC(CC(C)C)=O)CCC1CN(C(c1nccnc1N)=O)C2 C12CC(C1)CCC(=O)NCC(N(C)C)C1N(CC1)CC(=O)N2C.C1(CC)CCOC1 C(c1ccc(Cl)cc1F)=CC(N1CCN(C(C(C)NC(=O)NC)=O)C(C)C1)=O c1(C(N2CCCN(C(=O)CC3CC(F)C3)C(CO)C2)=O)cccc2scnc12 c1(CC(=O)NC(CNC(C2N(CC)CC2)=O)(C)CO)ccn2cncc2c1 Cc1nc(N2CCCC(C)(CNC(c3cc(C(C)C)on3)=O)C2)cc(C#N)n1 N1(C(c2n[nH]c(=N)s2)=O)CC2CCCC(NC(c3[nH]nc([N+](=O)[O-])c3Cl)=O)C2C1 c1(C(=O)NC2COCCN(C(=O)CC3(O)CCCCC3)C2)ccc2c(c1)COC2 c1(N2CCC(NC(CN(C)CC)=O)C(C)C2)ncnc2scc(C)c12 N1(C(C(C=C)O)=O)CCN(CC2(NC(=O)C(=Cc3ccco3)C)CC2)CC1 CC(C)C(O)C(C)C(=O)NC(C1(O)CCCCC1)C(=O)NCCCOCC1CC1 N1(C(CC(OCC)OC)=O)CCC(CN(C)C)C12COC2.C12CC(C1)CNC2=O c1(OC)c(C(=O)NC2(C)CN(C(=O)C(C)C(F)F)C2)ccc2c1CCC2 c1(CCNCC2N(CC(=O)Nc3ccc(Cl)cc3)CCCC2)cccc(Br)c1 c1(CCC)ccc(C(C(=O)N)N(CCOCCO)CCN(C)C)s1.NC c1(C(=O)NCC2C(Nc3ncc(C#N)nc3)CCCC2)ccn2nncc2c1 c1(CN2CCC(C(=O)OC(C)(C)C)C2)ccc(N2CCCC(C(N)=O)C2)cc1 N1(C(CC(C=C)CC)=O)CCOC2(C1)CN(C(c1cnc(N)cn1)=O)C2 Cc1ccc(NCCC(=O)NCC2C(C)CCCN2C(=O)CC2=CCCC2)c(Cl)n1 S(=O)(=O)(c1cccc(N2CCOC(C)(CCO)C2)n1)N1C(C)CCCC1 Cc1c[nH]cc(C(=O)NCC=CCNC(=O)C=Cc2ccncn2)c1=O C1(C)(C(N2C(COC)CCCC2)=O)CCCN(Cc2ccc(C(C)C)cc2Br)C1 c1(C(CNC(C2(OCC)CCSC2)=O)NC(CCCOC)=O)ccccc1F c1(C(N(C)CC2CCCN2C(=O)CC(C)(C)O)=O)c2c(nn1C)CCS(=O)(=O)C2 c1(C(=O)NC(CN(C(C(C)OC(C)(C)C)=O)C)C)cc(O)nn1C C1(NC(C(c2cn(C)nc2)O)=O)COCCC1C(N1CCC(F)C1)=O c1(C(C)C)cnc(O)c(C(=O)NCC2(C)CN(C(C)(C)C)CCO2)c1 C1(C(=O)NCC2(NC(C3C(=C)C3)=O)CCOCC2)CCc2nc(C)ncc2C1 C(C(F)C(=O)N(C)C)C(=O)NC1CC(N(C(C2C(C(C)C)C2)=O)C)C1 c1(-c2nnc(CC(=O)NON3CCOCC3)o2)ccc(Cl)cc1Cl C1(NC(C(c2ccc(C(F)(F)F)cc2)C)=O)CC(C)CN(C(=O)CCC(N)=O)C1 CC1(C)CCC(C(=O)OC2CC(C(=O)OC(C)(C)C)C2)OC1 CCC(O)C(CC)NC(=O)C(=O)Nc1ccccc1-c1nnnn1C(C)C N1(C(c2c(OC)n[nH]c2)=O)CC(C2CCCN(C(=O)C(O)CN3CCCC3)C2)C1 N1(C(c2c(C3(C)COC3)noc2)=O)CC(CNC(C2CC3CC3C2)=O)CC1(C)C N1(C(COC2(C#C)COC2)=O)CC23CCCCC2(C1)CN(C(=O)Cn1cccn1)C3 C12(C(=O)NCCc3cccc(C(F)(F)F)c3)CC3CC(CC(C3)O1)C2 c1(C(C(=O)NCCCC(C)(C)NC(=O)C=CSC)OC)ccc(Br)cc1 C(=O)(C1c2c[nH]nc2CCC1C)N(CCOCC)C.n1(CCO)cc(CC)nn1 Cc1cc(Cl)c(C(=O)N(C2CCC(NC(C3CCC34CCCO4)=O)CC2)C)cn1 C1(O)(CN2CCCC(CN(CC(=O)N(CC)CC3CCCO3)C)C2)CCCNC1 N1(C(C(C(=O)OCC)C2CC2)=O)CC(NC(C2(NC(N)=O)CC2)=O)C(C)(C)C1 N1(C(c2ccn(CC)c(=O)c2)=O)CC(C2CN(C(=O)C(C)Cc3ccco3)C2)C1 N1(C(COCC(=C)C)=O)CCN(C)C(C(=O)NC2(C)CCCC2(F)F)C1 C1(NC(=O)C(C2CCOCC2)O)CCN(C(=O)NC2CC2c2ccc(Cl)s2)CC1 C1(CCC)CN(C(c2cc(C(N)=O)cn2C)=O)CCN1C(=O)COCC1CC1 C1(CNC(=O)CC2CN3CCC2CC3)C(C2CC2)CCN1C(N1CCOC1=O)=O C(CCCCC(=O)N(c1ccc(O)c(C)c1)C(C)C(=O)O)NC(CC)=O c1(C(N2CCC(C(=O)OCC)C2)C(=O)NC)nc(F)ccc1Br c1(C(=O)NC2CC(NC(C(CC)C#N)=O)C2)c(F)cccc1[N+](=O)[O-] O=C(CS(=O)C(F)(F)F)NC1CCC(CNC(c2ccc(C3CC3)nc2O)=O)C1 C=C(Cl)C(C)(C)C(=O)N1CC2CC(C1)C2NC(c1[nH]c(C)c(C(=O)OC)c1C)=O C(=O)(CCC(=O)NN(C)C)NC1CC(NC(C(C(=O)OC)OC)=O)C1 c1(CC(C(=O)OC(C)(C)C)N(C)C)ccc2c(c1)CCN2.C12(OC)CN(C1)C2=O Cc1nc(N(C(=O)C(=O)N(C)C(C2(N(C)C)CCC2)C)C)sc1-c1ccc(CO)s1 CC(CC(C)(C)C)C(=O)N(C(C)(C)CC(=O)N1CC(O)C(F)C1)C O=C1OCCC2CN(S(=O)(=O)c3cccc(OC4CCCC4)c3)CC12 c1(C(=O)NCC(n2cc(Cn3ccc(C(=O)O)n3)nn2)C)ccnc2ncnn12 C1(OC)CN(C(=O)CCc2cncc(F)c2)C(C)(CNC(=O)Cn2cccn2)C1 c1(C(=O)NC2C(CNC(c3ccc(C(F)F)cc3)=O)C2)cc(O)cc(F)c1 Cc1ccc(C(N2CC(NC(=O)C=Cc3cccc(Br)c3)CC2C)=O)cc1C c1(C(N(C2CCN(C(=O)C(C)(C)O)C2)CC)=O)cc(F)c(OC)c(Cl)c1 N1(C(CNC(c2ncn(CC)n2)=O)=O)CCN(C(C2CC(=O)N(O)C2)=O)CC1 n1(C(CC)C)nc(C(N2CC(CCNC(=O)C(C)CO)C2)=O)cc1C c1(OCC(=O)Nc2ccnc(N3CCN(C)CC3)n2)ccc(Cl)c(Cl)c1 N1(C(C23CCC(C(N)=O)(C2)C3)=O)CCCCC(NC(C2CCCCO2)=O)C1 C1(NC(C(C)N(C)C(c2cc[nH]c(=N)n2)=O)=O)CCC(O)C(O)C1 C1(C(=O)NCC(=C)CCNC(=O)CC(C)n2cccn2)CC(=O)N(C(C)C)C1 C(=O)(CCCC(=O)OC)N(C)CCN(c1ccccc1)C(=O)COCCCF Cc1c(F)ccc(Br)c1C(N1CC(NC(c2cc(N(C)C)n[nH]2)=O)C(O)C1)=O N1(C(c2c(CC)ncs2)=O)CCC(C)C1CNC(=O)CSCc1cscn1 N1(C(CCC(=O)NC)=O)CCOC2(C1)CN(CC(=O)NCC1CCOC1)C2 c1(C(C(=O)NC)N(CCN(C)C)C2CC2)ccc(CC(C)C)s1 Cc1n[nH]c(=NC2CC3CN(C(c4oc5ccccc5c4Cl)=O)CC23)o1 c1(CC)ccccc1C(N1CCC(CCNC(=O)CCc2cncn2C)CC1)=O c1(C(=O)NC2CC(NC(C3(CC=C)CC3)=O)CC2O)ccc2cnoc2c1 N1(C(c2c(C)nc(COCC)s2)=O)CCCCC(CNC(=O)C2=COCCO2)C1 C(C(C)(CO)NC(c1cc(Br)c[nH]1)=O)NC(C(c1cnccn1)C)=O CCC(COC)C(=O)NCC1CC(NC(C2(C)CCCCO2)=O)C1 C1(C(N2CC(NC(C(CC)OC)=O)C(O)C2)=O)CC(=O)NC(=O)C1 C1(C(C)(C)NC(c2cnn[nH]2)=O)CCN(C(=O)C(F)C2CCC2)C1 CCCC(C)C(=O)NC1CCCC(CNC(c2ncccc2OC)=O)C1 C#CC1(C(=O)Nc2ccc(F)c(C)c2)CCN(C(=O)CN2CCC(C)C2)C1 N1(C(C(CC)N(C(=O)CC2CCCC3CC23)C)=O)CC2(CCC2)C1 c1(-c2nnc(CN(CCF)CC3CC(CC#N)C3)o2)ccccc1Cl C1(C(=O)NC2(CC)CCN(C(CCC=C)=O)CC2)Cc2ccccc2C1C c1(C(N2CCN(C(CCc3ccc(C)nc3)=O)CC2)=O)ccc(F)c2occc12 N1(C(C2(NC(C(CCC)O)=O)CCCCC2)=O)CCCC2(C=CCO2)C1 Cc1coc(C(=O)N(C(C)CNC(c2cn(C(C)C)nn2)=O)C)c1C CC1CN(C(=O)COC(F)(F)C(F)(F)F)CCC1CNC(c1cc(Cl)no1)=O C(=O)(C(F)C(=O)NC1CN(CC)CC1n1cc(CCN2CCOCC2)nn1)OC c1(-c2cccc(NCc3ccc(OC)nn3)n2)c(SC)cccc1F C1(C#N)(C(=O)NC2CC(C)N(C(=O)CN3CCC(O)CC3)C2)CCOCC1 C1(NC(=O)CNC(c2cc([N+](=O)[O-])n[nH]2)=O)CCCCCC1C(N1CCCC1)=O c1(C(=O)NC(C2CCOC2)CO)nc(Cl)sc1Cl C1(c2n(C(CC)(C)C)nnn2)(NCC(C)CC2CCCC2)COCC1CCSC c1(COC)cc(C(=O)N(C)CCN(C(=O)C(C2CCCCC2)O)C(C)C)on1 CCC(C(=O)NCCOC1CN(C(C2(CS(C)(=O)=O)CCC2)=O)C1)c1ccccc1 C1(CNC(C(C)(C)NC(=O)OC)=O)C2CN(C(C3(c4ccccc4)CC3)=O)CC12 c1(C(C)C(=O)NC2CCCC2NC(c2cc[nH]c2)=O)ccccc1F Cc1c(NCc2cn(C3CC3)nn2)ncnc1NC1CCSC(C)(C)C1 C12(C(=O)NCCCOC(=O)NC)CC(CO1)N(C(C1CC3CCCC3C1)=O)C2 C1(OCC(=O)NC(C)Cn2cc(-c3cnn(CCF)c3)nn2)C#CCCCCC1 C(CCCC(=O)N1CC(C)(NC(c2ccc(CC3CCCCC3)cc2)=O)C1)SC CC1NC(=O)OC12CN(C(=O)C(Cc1ccccc1Br)NC(=O)COC1CC1)C2 Nc1cnnc(NNC(=O)C2CCCCC2NC(c2ccc(Cl)cc2)=O)c1Cl c1(C(=O)NCCC(C)N(CCC)C)cc(CNC(C2CC2Cl)=O)on1 N1(C(Cc2c(C)cnn2C)=O)CC2(CC(NC(C3(N=[N+]=[N-])CC3)=O)CO2)C1 C1(OCCN(c2cnn(-c3cccc(F)c3)c2)C=O)CCCCCC1 C1(CNC(C(C#C)(C)C)=O)CN(C(=O)C(c2c(C)nn(C)c2C)C)C2(CCC2)C1 Cc1cccc(C(=O)NCC2COCCN2C(=O)Cc2cc(F)cc(F)c2)c1Cl C1(C(=O)Nc2cnc(C)c(Cl)c2)CC2(CCC2)CN1C(C1COCC(C)O1)=O c1(C(N2CC(N(C(CCCC(C)C)=O)C)C(C)(C)C2)=O)cccc2c1CCCC2 c1(NC(C2CC(F)CN2C(c2cncs2)=O)=O)cccc(-n2cncn2)c1 c1(NC(C2(C=C)CCC2)=O)ccc(NC(C2CC2C2CC2)=O)c(C)c1 CS(=O)(=O)C1CC(NC(=O)CN2CCN(Cc3cc(O)cc(O)c3)CC2)C1 N1(C(c2cc(C)c(C)s2)C(=O)NCC(F)F)CCOC2(CCCCC2)C1 C1(NC(CCSC)(C)c2nnnn2C2CCC2)COc2c(C)cccc2C1 C1(C(N)=O)CCN(CC2N(C(CC)=O)CCC2)CC1.c1(Cn2cccn2)ccco1 C1(C(=O)NCCCC2C=NNC2=O)(CC)CCCN(C(=O)Cn2cnnc2)C1 CC(CN=c1cccc(S(=O)(=O)NCc2ncc(Br)s2)[nH]1)C1CCCC1 c1(NCC(=O)NCC)nc(C)cc(=NCC(C)c2ccc(F)cc2)[nH]1 C(CC(C)(C)C)(c1n(CC=C)nnn1)(C1CC1)NC1C(C)CCC1C c1(C(C)(C)C)cccc2c1OCC2C(=O)N1CC(Cc2ccccc2)C1 C1(O)(CCNC(C(CCO)N(C)C)=O)CCCN(C(c2cscc2C#N)=O)C1 CC(=O)C(C)(C)CC(=O)N(C1CN(C(C2CC3CC3C2)=O)CC1C(F)F)C1CC1 C1(c2n(CCCSC)nnn2)(NC(c2cccc(Cl)c2Cl)C)CCCN(CC)C1 C=C=CCCC(=O)N1CCOC(CNCC2N(C(=O)OC(C)(C)C)CCC2)C1 c1(C2(NCc3cn(C)nc3)CC2)ccc(F)cn1 O=S(=O)(c1ccc(Br)cc1N1CCC2(CCC2)C(CO)C1)NCC(O)C1CCC1 C(CC1CC1)(C(=O)N(CCCN1CCCCC1)CC)NC(COC(CC)C)=O C1(C)(COC)CCCN1C(=O)C(N1CCC(C(=O)OC)(C(=O)OC)C1)=O C1(CNC(COCCC(C)C)=O)(NC(=O)CC2CCCSC2)CC(F)(F)C1 C(=O)(C1Cc2ccccc21)N(CCOC)CCNC(C1CC1C1CC1C)=O C1(CNC(C(CC)(C)C)=O)CCN(C(C2(C)CC2C(F)(F)F)=O)CC1C c1(OC)ccc(NC(c2coc(C(C)NC(C3(F)CCCC3)=O)n2)=O)cn1 Cc1[nH]nc2cc(C(=O)NCC3CCN3C(=O)C(C)(C)OCC(F)(F)F)ccc12 c1(CC)ncsc1C(=O)NC1CCCC1CNC(c1cc(C2(C)CC2)on1)=O N1(C(c2c(C)nc(C(C)C)s2)=O)CCC(CO)C(NC(c2nn(C)cc2Cl)=O)C1 C1(C(=O)NC(C2CCN(C(CC(C)OC)=O)CC2)C)CCC(C)=C(C)C1 C(=O)(C(C)(C)C(N)=O)N1C(C)CC1n1cc(CCC(O)CCc2ccccc2)nn1 c1(C(C(=O)NC2CN(C(CC(C=C)C)=O)C2)O)ccc([N+](=O)[O-])cc1 c1(CC(CNC(=O)NC2C3CCCCC23)CO)cc(F)c(F)c(F)c1 c1(OCC(C)C)ccccc1CN(c1cccc(N2CCC2=O)c1)C CCCCC(C)(F)C(=O)N1CCC(NC(C2CCC(C)(C)O2)=O)C(F)C1 C(CCCCN=[N+]=[N-])NC(CC1CC(NC(C2(CC=C)CCCC2)=O)C1)=O N1(Cc2c(C)n(C)nc2)CC2(CCCCC2)C1C(C)C C(=O)(C(C(F)(F)F)C(F)(F)F)N1CC(C2OCCN(C(CC(=O)OCC)=O)C2)C1 N1(C(CC(CC)(C)C)=O)C2CCC1CN(C(C13CCC1C3)=O)C2 n1(CCC(=O)NC2CC(N(C(C3C(CC)OCC3)=O)C)C2)c(C)cc(O)cc1=O N1(C(c2c(CNC(CC3C(=O)NCCC3)=O)ccs2)=O)CCOC2(CCC2)CC1 CN1CCN(C(c2ccc(=O)oc2)=O)C(CNC(c2cc(CO)n(C)n2)=O)C1 c1(C(N2CCC(NC(CCC(=O)NC)=O)(COC)C2)=O)ccsc1S(C)(=O)=O c1(C(N(CC(C)N(C)C(c2cnnn2C)=O)C)=O)cnccc1N(C)C c1(OC)nc2cc(N(C(=O)CC(C)c3ccccc3)C)ccc2o1 C(=O)(C1Cc2ccc(F)cc21)NC1CCN(C(C(C)NC(N)=O)=O)C12CCCC2 c1(C(=O)NC2C(NC(C3(OC)CCSC3)=O)CCC2)ccc(C2CC2)cc1Cl c1(CC(N2CCCC(C)(NC(c3cnc(C)[nH]3)=O)C2)=O)cccc(S(C)(=O)=O)c1 c1(CC(NOCC)=O)[nH]c(=NC2CCOCC(C)C2)nc2scnc12 CCCC(C(O)C(=O)Nc1ccc2nncn2c1)NC(C1OCCC1C)=O CP(C)(=O)C(O)C(=O)NCCN1CCC(NC(=O)CC2CC(F)(F)C2)CC1 c1(OC)ccc(Cl)cc1C(=O)NCCCNC(=O)Cc1cccnc1 c1(C(=O)NCC(CC)(CC)NC(C2CCCCCCC2)=O)cnc2[nH]cnc2c1 C1(C(=O)NCc2c(C(C)C)noc2)CN(C)CCN1C(C1C2CCC(F)(F)C12)=O c1(C(N2CCN(C3CN(C(C(C(=O)OCC)F)=O)C3)CC2)=O)cccn(C)c1=O Cc1cc(C(=O)NCCNC(C2CC2C)=O)c(C)n1C1CCCCC1 N1(CCC(=O)NC2CN(C(=O)C(O)C3CCC3)C2)C(=O)C2CCCCC2C1=O c1(C(N(CCN(C)C(c2ccncc2C(F)F)=O)C)=O)cccc(C(C)(F)F)n1 N1(C(N2CCC(NCC(C)(C)O)C2)=O)CC2CC1(C)C2.C(C(C)(C)C)O c1(C(=O)NCCC2(CNC(CSC)=O)CC2)cnc2c[nH]nc2c1 c1(C(N(CCCNC(c2n(CC)ccn2)=O)C)=O)cccc(P(C)(C)=O)c1 C1(CCC)(NC(=O)CC(C)(C)F)CCCN(C(c2ncccc2OC)=O)C1 N1(C(c2cc(OC)nc(Cl)c2)=O)CCC2(NC(=O)C=Cc3cnc[nH]3)CCCC12 N1(C(CCC2(C)CC2)=O)CC2CC2(NC(c2snnc2C2CCC2)=O)C1 c1(C(N2CCN(Cc3c(OC)ncc(Br)c3)C3C2C3)=O)ccc2sccc2c1O Cn1cc(C(=O)NCC2CC(C#N)(OCc3ccccc3)C2)n(C)c1=O C1(C(=O)NC2C(NC(c3ccnc4c3CCO4)=O)COC2)CCCC2(CCC2)C1 C(CC(=O)NC1CC2CC(NC(=O)CCSC3CCCC3)C1C2)(C(C)C)OCC C1(C)(CC)CC(NC(=O)CCC(C)C)CN1C(=O)CNS(=O)(=O)N(C)C N1(C(c2cccc(I)c2)=O)CC2CCC(C1)N2Cc1cccc(Br)c1F N1(C(c2c(C)csn2)=O)CCCCCC1C(=O)NCc1nncs1 C1(C(N2CC(N(C(C(CC)C#N)=O)C)C2)=O)CS(=O)(=O)CC12CC2 C1(CC(=O)N(CCCNC(c2ccccc2O)=O)CCO)CCCCC12CC2 Cc1ccc(Cl)c(N)c1C(N1CCC(NC(=O)C(C)N(C)C)C(O)C1)=O CC(O)C(C)(C)C(=O)NC(C1(O)CCCCC1)C(N1CC2CCC(C1)O2)=O N1(C(c2[nH]cc(C)c2)=O)CCOC(C)(CNC(=O)CC2(CN(C)C)CCCCC2)C1 N1(C(c2c(SCC)cc(Cl)cc2)=O)CCC(N(C)C(c2cnn[nH]2)=O)C2(CC2)C1 C(=O)(C1=COCC1)NC1(c2cn(Cc3ncc(Cl)cn3)nn2)C(C)C1 c1(C(N2CC3(CC(NS(CC=C)(=O)=O)C3)C2)=O)c(C)nc2ccccn12 Cc1nn(C)c(C)c1CC(N1CCSCC1CCNC(c1cncn1C)=O)=O c1(C(c2nnnn2C2COC2)NCC2(C)CCCC2(F)F)csc(S(N)(=O)=O)c1 S(=O)(=O)(c1cc(C(F)(F)F)cc(O)c1)Nc1c(C)ccc(SCCC)c1 C(CC1CCC1)(C(=O)N(CCCNC(c1cnc(C)s1)=O)CC1CCCC1)OC c1(CC(=O)NCC(C2CCN(C(=O)C(Cl)=CCl)CC2)C)ccc2sccc2c1 N1(C(CS(CC)=O)=O)CCCC(C)(NC(c2cnn(CC(C)C)c2C2CC2)=O)C1 Cc1cc(F)c(C(N2CCCC(C)(NC(=O)CSCc3ncc[nH]3)C2)=O)cc1F Cc1ncc(C(=O)NCC(C)NC(=O)C(c2ccc(F)cc2F)C)cc1N Cc1ccc(C(=O)NCC(c2cccc(Cl)c2)NC(C2CC2(C)C)=O)nc1 C(C(C)(C(=O)NC1CCCCC1)NC(C1CCCO1)=O)SC Cc1ccc(C(=O)NCC2CC2NC(c2c[nH]nc2-c2cccnc2)=O)c(N)c1 C(=O)(C1Cc2c(Cl)cccc21)N1C(CNC(CCCCNC(C)=O)=O)CCCC1 C(=O)(CC(C)(C)CC)N(C(CNC(C(CC)OC)=O)CC)C c1(CC)c(NC(C)=O)cccc1C(=O)OCC.C12(F)CC(C1)C(=O)NC1CC1C2 N1(CCC=CC)CCC2(CCCCN(C(=O)CCCOc3ccc(OC)cc3)C2)C1 c1(CC)nc2ccc(Cl)cn2c1C(=O)NCCN(C(=O)C1=CC(C)(CC)C1)C c1(C(N2CCC(NC(CC3C(C)=NN(C)C3=O)=O)C2)=O)ccc(C)cc1[N+](=O)[O-] C=CCC(CNC(=O)C(CC)=CC)C(=O)NCC(C)(O)C(C)CC c1(CNC(N)=O)ccc(C(N2CC3CC2C3NC(C2CC2Cl)=O)=O)cc1 CCC(=O)CCC(=O)NC(CC1CCC1)C(=O)NC1CN(C)CCC1O C1(OC)CN(C(c2[nH]c(O)nc2C)=O)CC1NC(C1(C2CC2)CC1)=O Cc1cc(C)c2onc(C(=O)NNC(=S)NCC(O)CC(F)(F)F)c2c1 C1(C(C(=O)N(CC(=O)NC)C)C)CCCN(C(=O)C=Cc2cocn2)C1 c1(C(=O)Nc2ccccc2)ccc(NCCNc2cscn2)cc1 c1(C(N2CC(NC(c3c(CC)c[nH]c3)=O)C2)=O)cc(O)c2ccccc2c1 Cc1nccn1CCNC(=O)C(C1(C)CC1)NC(C1CCC(C)O1)=O CCC(CC)CCCNC(=O)C(Cc1ccco1)NC(c1ccc(CO)o1)=O C12CCC(CC1)CNC2=O.C(C(O)CNC(=O)CC1CC1)OCC.C(=O)(N)NC c1(OC)ccccc1C(=O)NCC(CO)NC(=O)CC1CCC1C c1(CC)c(C(=O)NC2CC(O)(CNC(=O)C(C)(C)OC)C2)[nH]c(C)c1C(C)=O N1(C(CC(CC=C)NC(c2nccs2)=O)=O)C2CCC1CC(CO)C2 c1(COCC#C)cccc(NC(C2CC2NC(=O)CCc2cnn(C)c2)=O)c1 Cc1ccc(C=CC(=O)NCC2CC2CNC(=O)CCCC#N)s1 N1(C(COCC)=O)CCc2nc(C(=O)N(CCO)CCO)ccc2C1 N1(CC(=O)NCC(CN(C)C(c2cn(C3CC3)cn2)=O)(C)C)CCS(=O)(=O)CC1 C1(C(N2CCC(C)C(NC(C34CC(C3)C4)=O)C2)=O)C2CCC(C2)C1(C)C C#Cc1ccc(C(=O)NC2CN(C(C3CC(n4cnnc4)C3)=O)CC2OC)cc1 N1(C(CCCOC(C)C)=O)CCOCC(NC(=O)C(c2ccc(Cl)cc2)(C)C)C1 C=C(C)C1CN(C(=O)C(C2(O)CN(C(c3cn(C)nc3C)=O)C2)F)CCO1 C12CC(c3ccccc3)(C1)NC(=O)CCCOCCON2.C#CCN(C)C(C)=O C(c1ccccc1F)=CCOC(C(C)OCCC=C)=O C1(OC)CN(C(c2c(Br)noc2C2CC2)=O)CC1NC(c1ccoc1)=O CN1CC=C(C(=O)NC2CCC(CC(=O)NCC34CCC(CC3)O4)C2)C1 c1(-n2ncc(C(N(C3CC(NC(C4CNC(=O)C4)=O)C3)C)=O)n2)ccc(F)cc1 O=S(=O)(c1cc(Cl)cc(Cl)c1)N1CC2CN(Cc3cc(Br)ccc3Br)C2C1 c1(CC(=O)NCCCCC2CN(C(C)=O)C2)cnc(N(C)C)cn1 c1(C(=O)OC)ccc(F)c(Cl)c1.c1(OCCN2C(=O)C2)ccc(Cl)cc1 N1(C(C2C3CN(C(Cc4cc(C)on4)=O)CC32)=O)CCc2ccc(C#N)cc2C1 C(=O)(C(C)(CO)OC)NCC1C(C(N(CC(=C)Br)C2CC2)=O)CC1 CCS(=O)CC(=O)NCC12CC(CN1C(c1c(C)nsc1NC1CC1)=O)C2 c1(OC)cc(C)ccc1CN1CCC2(CC2C(=O)NC(C)Cc2ccccn2)C1 N1(C(c2nn(CC)c(C)c2)=O)CCC(CNC(=O)CCCCN(C)C)C12CC2 c1(C(=O)NC(CC)CNC(=O)CCc2csc(=N)[nH]2)cn2ccsc2n1 CN1CC(O)CC1C(=O)NCCCC(=O)NCC(O)C(F)(F)F C(c1ccccc1Cl)=CC(=O)NC1CC2CC1N(C(=O)COCc1nc[nH]n1)C2 C1(C)(NC(CN2C(C)CCC2C)=O)CCCN(c2ccncn2)C1 c1(C(N2CC(C)(NC(=O)COCc3nc[nH]n3)C2)=O)cncc(N)n1 c1(C(=O)NCC2C(NC(C)=O)COC2)c(-n2cnnn2)sc2c1CCC2 C(CC(C(=O)NC(CC1CC1)CC(=O)NCCCC1CCC1)OC)OC N#Cc1cc2cc(C(=O)NCC=CCNC(c3cnn[nH]3)=O)[nH]c2cn1 c1(OC)cccc(C2(C(=O)NCCCn3cc(C4(C(=O)O)CC4)nn3)CC2)c1 n1(C(C(=O)Nc2ccc(C)c(Br)c2)C)cnc2ccccc12 C1(CC(=O)N(C)CC2(N(C)C)CC2)N(C(c2cccs2)=O)CCC1(C)C N1(C(c2cc3occc3[nH]2)=O)CCCC2C1CCCN2C(c1ncon1)=O c1(CC)ccc(C(N2CCC(F)(CNC(C3CCCSC3C)=O)CC2)=O)c(F)c1 Cc1ccc(CC(=O)NC2(CCNC(=O)CNC(C3CCCC3)=O)CCC2)cn1 C1(NC(=O)COC(F)(F)F)C2CCC1CN(C(C1CC3CCC1NC3=O)=O)C2 C1(NC(CC(=O)OC)=O)C2CC3C1C3C2C(=O)Nc1cccc(F)c1C c1(SC)ccc(N)cc1C(N1CC2CC(NC(c3cc(C)c(C)[nH]3)=O)C2C1)=O C1(C)(C(N(C)CC2CCN(C)C2)=O)C=CCN1C(=O)Cc1cccnc1O C1(C(N(CCCF)C)=O)(NC(=O)C(=O)NCC2CC2)CCC(C)(C)C1 c1(C(=O)OC)ccc(C)nc1NC(C)(CNC(C1CCCN1C1CC1)=O)CC C1(C(N2C(CCNC(=O)COc3ccccc3)CCCC2)=O)CC2CC1C1CC21 N1(C(C(C=C)O)=O)CCOCC12COCCN(C(C1Cc3cccnc3C1)=O)C2 CC(C)CCCCC(=O)NC1CCCOC1c1ccccc1.C(=O)CC(C)C(F)F c1(C(=O)NC2(CNC(C3CC(C#C)(O)C3)=O)CCOCC2)nccc(Cl)c1C N1(C(c2ccc(CNC(C(C(C)C)N(C)C)=O)s2)=O)CCCC2(CCC2)C1 N1(C(C(COC)C(F)(F)F)=O)CC2(CCOCC2)CC1CNC(c1csnn1)=O c1(CC(=O)NC(CCN(C(C(=O)NCCOC)=O)C)C)ccc(C)cc1Br C=C(CC)CN=c1ccnc(NC2CCOCC2C)[nH]1 C1(CNC(c2n(CCCC)nnn2)C2CC2)CCS(=O)(=O)N1C.C(C)CCCCO N1(C(C2OCCN(C)C2)=O)CC2CC(F)(F)CCC2(N)C1 CCC(CSC)(c1nnnn1C1CCOC1)NCC=Cc1ccco1 c1(C(=O)NCC(C)N(C(C(n2ncc(C)c2)C)=O)C)noc2c1CC(C)(C)CC2 c1(C(=O)NC(COCC)CO)c(CNC(=O)C=CC2CC2)cnn1C N1(C(C2CC(SC)C2)=O)CC(CCNC(=O)CCc2nncn2C)OC(C)C1 c1(C(N2CCCC(NC(C=C3CCC(C)C3)=O)C2)=O)ccc2c(c1)COC2(C)C C1(C)(NC(c2cc(C)sc2)=O)CCN(C(c2cc(C)c(-c3ccccc3)s2)=O)C1 C12COCCN(C1)C2=O.C1(NC(=O)NOCC2CCSCC2)CC2(CCC2)CO1 N1(C(=O)C#CC2CC2)CCCC(C2CCN(C(c3ccc(C(F)(F)F)o3)=O)C2)C1 C1(NC(c2cccc(C3CC3)c2)=O)CCCCC1NC(C1(F)CCOC1)=O N1(C(=O)C2=CCC2)CCCC2(C1)CN(C(=O)C1SCCc3ccccc31)CCO2 CC1CCC(CC(=O)OCc2noc(COCc3ccccc3)n2)CC1 CC(C)(C)C(CC(=O)N1CC2CC1C2NC(C1CCC(CO)CC1)=O)C(F)F C1(C(=O)NC2(C)CN(C(=O)CC3(C)OCCO3)C2)CC2CCC1C2 C=CC1CN(C(=O)CC(CCC)NC(C2(C3CC3)CC(=O)C2)=O)CCO1 c1(C(=O)NC2CCCN(C(=O)Cc3ncc(Cl)s3)CC2)cc2ncccc2[nH]1 c1(CN2CCN(Cc3cc(C(=O)O)c(O)cc3)CC2)c[nH]c2cccc(O)c12 c1(N2CCCC(OCC)C2)nc2c(c(=NCC34CC(CCO3)C4)[nH]1)CC(C)CC2 c1(SCC(N2CCC(CC(=O)NC3(C(F)(F)F)COC3)C2)=O)ccc(F)cc1 C=CCC(CNC(C1(CC(=O)OC)CC1)=O)NC(=O)CC(C)n1cccn1 C1(CC(N2CC(C(C)NC(C3CC34CCCC4)=O)C2)=O)NC(=O)NC1=O C12CCC(C1)CCC(=O)N2.C(CCN=[N+]=[N-])NC(C1(CCOC)CC1)=O C(CCC(O)C(=O)NCc1ccc(CO)cc1)NC(C1(C)CCN(C)C1)=O C(=O)(CC(C)(C)C(F)F)N1C2C(NC(c3c(C)cncn3)=O)CC(C2)C1 C=CC1CN(C(=O)C(C)Cc2ccc(O)cc2)CC1NC(c1cnc(Cl)s1)=O c1(C(N2C(C(=O)Nc3ncc(Br)s3)CSCC2)=O)ccc2nc(CO)[nH]c2c1 C1(NC(c2c(CC)ocn2)=O)CN(C(=O)Cc2nc(C)sc2C)CC(C)(C)C1 N1(C(COC)=O)CCc2ccccc2C(NC(=O)C=Cc2cccc(Cl)c2)C1 c1(C(=O)NC2CC(C)(NC(=O)CCN3CCC3)C2)ccc2ccoc2c1 C12(C(=O)NC3(COC)CC3)CCN(C(C3CCC3C(F)F)=O)CCC1C2 c1(OCCC(N2CCC(C)(NC(CC3ON=C(C)C3)=O)C2)=O)cc(C)cc(C)c1 c1(-c2ccc(CO)cc2)csc(=Nc2cccc(O)c2)n1Cc1ccccc1Br CCC(CC1CCCC1)C(=O)N(CCCN(C)C(C1CC1c1cnn(C)c1)=O)C c1(C(=O)NCC(C)CN(C)C(C2C(C)C2(F)F)=O)cccc2nc(O)n(C)c12 C1(N(CC(=O)NC2CC(OC)C2)C)CC(C(=O)OCC2CC2)C12CCC2 C1(C)(OC)CCCN(C(C2CC(O)CN2C(=O)C=CC(F)(F)F)=O)CC1 Cc1cn2c(C(=O)NCC(C)NC(C3CCOC(C)(C)C3)=O)c(Cl)nc2s1 C1(C(N2CC(CNC(C3C(CC)CCO3)=O)C2)=O)CCCCC(F)(F)C1 C1(NC(=O)COc2ccsc2)CC2CC(NC(c3nc(Cl)cs3)=O)CC2C1 C1(N(C(C(CC)F)=O)CCO)CCN(C(=O)Cc2ccsc2C)CC1 C1(C(=O)NC(CNC(C2(CCOCC)CCCC2)=O)(C)C)CCCS(=O)(=O)N1 c1(C(N(CCC(C)NC(c2ccc([N+](=O)[O-])[nH]2)=O)C)=O)c[nH]nc1S(N)(=O)=O Cc1cc(NC(=O)C(CO)N(C)C)ccc1NC(c1oc(CO)nc1C)=O N1(C(C2(F)CCCN(C(C3CN(C)C(=O)CC3)=O)C2)=O)CCOCC(F)(F)C1 C(=O)(C(CC(C)SC)N1CCN(Cc2nc(CC)no2)CC1)NCCCC CCC(COC)C(=O)N(C)CC1C2CN(C(c3cccn3C3CCCC3)=O)CC12 NC1CCCN(C(=O)CCCn2ccnc2)C1C(F)(F)F C1(c2nc(CCN(C)C)n(-c3ccc(F)nc3)n2)CCC(F)(F)CC1 c1(OCC)c(-n2cc(-c3c(F)ccnc3F)nn2)cccc1F.C12CCCN1C2=O Cc1sncc1C(=O)NC1CCC1NC(=O)CCc1cnc(Br)s1 C1(NC(C(C)O)=O)C=CCN(C(=O)CNC(c2cccc(Cl)c2)=O)C1 N1(C(CC(C)OC)=O)CCN(C(=O)C(=Cc2cccn2C)F)CC1C1CCCC1 N1(C(COC2(C)CCC2)=O)CC(NC(C2CC2c2ccco2)=O)C(O)C1 Cc1cc(C(=O)NCC(N2CCN(C(=O)C3=COCCC3)CC2)=O)cc(N)c1Cl CC1(C)CCOC(C(=O)NCC2(C)CCCC2NC(C2CCS2(=O)=O)=O)C1 C1(NC(c2cc3occc3s2)=O)CCN(C(C2CC2(Cl)Cl)=O)CC1F N1(C(c2ncc(CC)cn2)=O)CCCC2CN(C(=O)CC(C)C(C)(C)C)CCC12 C=Cc1ccc(C(N2CC(OC)C(NC(=O)Cn3ncccc3=O)C2)=O)cc1 C1(C(=O)NCC(C2CC2)NC(c2cnn(CC(F)F)n2)=O)CCCCS1(=O)=O c1(N2CC(C)N(Cc3cccn3C)CC2)ncnc2c1CCC2 C1(C(=O)NCC23N(C)CC(C2)C3)CC(F)(F)CN1C(c1csnc1Cl)=O C=CCC(CNC(=O)C(N1CCCCC1)C)C(=O)NCCn1ccnc1C N1(C(C(C)N(C(C2C(=C)CC2)=O)CCC)=O)CCCN(C(=O)NC)CC1 C(=O)(C1CCCc2nncn21)N(CCC(C(C)C)NC(=O)C(Br)=C(C)C)C C12(CNC(=O)CSCC3CCCCO3)CC(CN1C(c1ccc(Cl)o1)=O)C2 S(=O)(=O)(c1cc(C(N2CC3CC2CCC3O)=O)n(C)c1)NC(C)C C(=O)(C1SCc2cccnc21)NC(C)CNC(c1cc(CO)ccc1Cl)=O C1(CC=C)(C(=O)NCCN(C(C)C)CC)CCCN1C(C1C=CCC1)=O C1(C(=O)OC(C)(C)C)CCCC2CN(C(N(C)CC3(C(F)(F)F)CCC3)=O)CCC12 C#Cc1ccc(C(=O)NC2CCCC(NC(C3CC34CC4)=O)C2)c(C)c1 c1(C(N2CCC3C(O)CC23)C(=O)NCCSC)ccc2c(c1Cl)OCO2 C1(CN(C)C(c2ccccc2)=O)CCCCN1C(c1ccncc1F)=O CCC(C(=O)NCCN(C(=O)CC(O)C1CC1)C1CC1)C(C)(C)CC C12(CC(=O)NCC(C)(C)Cn3cc(CO)nn3)COC(CF)(C1)C2 c1(C(=O)NC2C(NC(=O)C3=NOCC3)C2)ccc2c(=O)c3ccccc3sc2c1 C1(C(=O)NCC(CN(C(C(COC)C)=O)C)(C)C)Cc2c(F)cccc2O1 N1(CCN(C)C(C2COCCO2)=O)CCN(C(=O)CCc2cccc(Cl)n2)CC1 c1(C(N(CCOC)Cc2ccccc2C)=O)coc2c1CNC2 c1(OCC)cc(C=CC(=O)NC2CCCCC2NC(=O)CC2CC2)ccc1O C(C(C(C)C(C)C)NC(=O)CN1CC(=O)NC1=O)NC(c1c(SC)n(C)nc1)=O C1(CNC(C(CCC)(C)O)=O)CC2CCC(C1)N2C(C1CCCCC1O)=O Cc1cccc(CCNC(c2n[nH]cc2CNC(C2CC2(F)F)=O)=O)n1 c1(NC)ccc(NC(=O)C(=O)N(C)Cc2cnn(C)c2C)cc1F N1(C(COCC)=O)CCC(O)(CCNC(C2(n3cccn3)CCCC2)=O)CC1 CCS(=O)(=O)c1cc(F)ccc1NC(N1CCC(NC(c2ccccc2)=O)C1)=O N1(C(C(C(C)C)SC)=O)CC2CC(C)N(C(c3ccc4nnc(S)n4c3)=O)C2C1 C(=O)(CC1=CCN(C(=O)C(CCC)OCC)CC1)N1CC(C#C)OCC1 C(=O)(CS(=O)(=O)C(C)(C)C)NCC1N(C(C(C=C=C)C)=O)CC(F)(F)C1 N1(C(C(C)NC(=O)CCCCC2CC2)=O)CCCC12CCCOC2 C1(C(N(C(C)C(=O)N(CC(O)C2CCC2)C)C2CC2)=O)CCCCNC1=O N1(C(C(c2cccs2)N(CC=C)CC)=O)CCC(C(=O)NC2CC2)C1 C1(C(=O)NCC(CO)NC(c2cc(CO)[nH]n2)=O)CCN(CC2CC2)CC1 c1(OC(=O)N(C)Cc2c(C)cco2)cccc(F)c1 C(=O)(C(=O)CC(C)CC)NC(C(N1CCC(C(C#C)C)CC1)=O)CCF c1(C(N(C(C)CNC(=O)CC2CC3(CCC3)CO2)CC)=O)cnc(OC)c(F)c1 C1(c2ccc(C)nc2)NC(=O)N(C2CC2)C2=C1C(=O)NC21CCOC1 CC1(C)CN(C(C2C3COCC23)=O)CCC1NC(=O)C=Cc1cncnc1O Nc1c(C(=O)NCC2CCCN2C(=O)Cc2ccsn2)cc(F)cc1[N+](=O)[O-] Cc1ccc(Cl)c(C(=O)NC2CC(CCNC(c3cc(O)nn3C)=O)C2)c1 Nc1c(Cl)c(OCC(=O)NC2NC(=S)N(c3ccccc3)C2=O)nc(F)c1Cl N1(C(C2CCC(CC)O2)=O)CCC(C(=O)NCC2CN(C(C)C)C2)CC1(C)C C1(C)(NC(C(c2ccc(C)cc2)F)=O)CCCN(C(=O)C=C2CCCC2)C1 Cc1c(Cl)cnc(NC(=O)Nc2ncc(-c3ccccc3)cn2)c1Cl N1(C(C2(C)CCC2)=O)CCC(C2(NC(c3ccn4[nH]c(=N)nc4c3)=O)CC2)CC1 C1(NC(C2C(C(C)C)OCC2)=O)CC2CCC1N2C(=O)Cc1cccc(F)c1 CC1(F)CN(C(c2ccc(N)c(Cl)n2)=O)CCN(C(C2CCC3(CCC3)C2)=O)C1 CCC(CNC(c1cc(C2CC2)no1)=O)(CC)C(=O)N1CCC(C)(C)CC1 Cc1cc(N)c(C(=O)NCCc2ocnc2CNC(=O)CCC2CC2)cc1C C1(CC(=O)NCc2scc(CC)n2)CN(C(C2CC3(CC3)CN2C)=O)C(C)(C)C1 c1(C(=O)NCCN(C(c2cc(-c3ccco3)on2)=O)CC)cc2n(n1)CCC2 C1(C(=O)NC(C)Cc2ccncc2)CC=CCN1C(c1scnc1Cl)=O N1(c2c(S(=O)(=O)N3C(CC=C)CCCC3)cccn2)CCc2cc(Br)ccc2C1 c1(CNC(C(C)OCC2CC2)=O)cccc2c1CCN(C(c1sccc1F)=O)C2 C1(O)(C(C)NC(C(C)OCCCC)=O)CCN(C(=O)C(C)=C2CCC2)CC1 c1(C(C(=O)NC)OC)cn(N2CCCC2c2cc(C3CC3)on2)nc1C N1(CCC)C(=O)CCC1C(=O)NCCC1CCCN1C(c1cccnc1C)=O N1(C(CN(CC(=C)C)C2CC2)=O)CCCC1CC(N1CCC1C1CCCCC1)=O c1(SC)cc(C(=O)N(CCCCN(C)C(c2[nH]cnc2C#N)=O)C)oc1C C(=O)(C(C)CC(C)(C)C)NCCC1N(C(c2sc(C)c(O)n2)=O)CCCC1 c1(N2C(=O)CC(C(=O)NS(Cc3cccc(NC)c3)(=O)=O)C2)cnccc1C#N CC1CCN(CCn2cc(C(=O)N(C3CCOC3)CCO)nn2)c2ccccc2S1 C1(C)(OC)CC(NC(C2(N(C(=O)Cc3ccc[nH]3)C3CC3)CCC2)=O)C1(C)C c1(NC(CSCC(=O)NCC(C)NC(C2CCC(C)(C)O2)=O)=O)ccc(F)cc1 c1(OC)ccnc(F)c1C(=O)NCC1CC(NC(C2CC(C)OC2=O)=O)C1 C(CC(=O)NCC(=O)NC(C)CF)OC(C)=O c1(C(C)C)ccc(C(N2CC(NC(C3(C4CCCO4)CC3)=O)C(C)C2)=O)c(O)n1 C(CC(CNC(c1snnc1C(C)C)=O)NC(=O)CCc1cscn1)OC CC1CCC2(CO1)CN(C(C1(CO)CCCN(C(c3ncccc3N)=O)C1)=O)C2 N1(C(c2ccc(C)nc2C)C(=O)NCCOC)CCC2(CCN(C)C2=O)C1 c1(C(=O)OC)c(Cl)ccc(NC(c2cn(CCCCSC)nn2)=O)c1C Cc1ccc(C(C)(C)CC(=O)NCCC(C(=O)O)c2ccc(O)cc2)cc1 N1(C(C2(C)N(C(CN3C(C)CCC3)=O)CCC2)=O)CCc2sccc2C1 c1(C(=O)NCC2CCN(C(c3ccc(OC)s3)=O)C2)cc2c(Cl)cncc2s1 Cc1cc(C(=O)NC2CCSC23CN(C(=O)CC(C)C2CC2)C3)c(C)n1NC(N)=O c1(Nc2nccc(N3C4C(NC(C)=O)C(CCC4)C3)n2)cnc2ccnn2c1 C1(NC(C2(CC#C)CC2)=O)COCC1NC(c1cc(-c2ccc(C)s2)[nH]n1)=O c1(C(N(C2CCCN(C(C(CC)(C)C)=O)CC2)C)=O)ccccc1S(C)=O C1(NC(Cc2c(CC)cccc2)=O)CN(C(=O)CCCC(C)=O)CCC1C Cc1ncc(Br)cc1NC(=O)C(c1ccc(CN(C)C)o1)N(C1CCCCC1)C C(=O)(CC(C)CNC(=O)CC1CCC(=O)N1)NC(Cn1ncc(C)c1)C c1(CC)nc(C)[nH]c1C(=O)NC(C)(C)CNC(=O)CN1CCS(=O)CC1 Cc1cncc(C(=O)NCC2CC2CNC(c2cn(CC(F)(F)F)nc2C)=O)c1 c1(C(=O)NC23CC(NC(C4(SCC)CC4)=O)(C2)C3)nnn2c1CCCC2 c1(C(=O)NCC(C)(C)OCC(=O)NCC2(F)CC=CCC2)cccc2occc12 CC(C(O)C(F)F)NC(=O)COC1CN(C(C2(C)COC(=O)N2)=O)C1 C1(N(C(C(C)NC(=O)NC)=O)C)CCN(C(=O)COC)CC1 CCCC(CCCNC(c1cccc(CC)n1)=O)NC(c1cnc(C)c(N)c1)=O CC1(C(=O)NC2CCC2N2CCCC2)CCN(C(=O)C(CO)N(C)C)CC1 c1(CC)cccc(OCC(N2CC(COC)(NC(c3ccccc3C)=O)C2)=O)c1 C1(F)(CNC(C(C=C)c2ccccc2)=O)CCN(C(c2ccc(CCC)s2)=O)C1 Nc1c(Cl)cc(C(=O)NCC2CCN2C(=O)CSC2CCCCO2)cc1Cl C(=O)(CC1NC(=O)c2ccccc21)N1CC(CNC(c2cc(F)c[nH]2)=O)C1 C1(F)(CNC(C(C2CCC2)OC)=O)CCCN(C(C2CCC(C)O2)=O)C1 c1(C(C)C(=O)N2CC(NC(C3C=CCCC3)=O)C2)ccccc1F c1(N2C(=O)CC(C(=O)NCCNC(C3(C)CC=CCC3)=O)C2)ccc(F)c(F)c1 Cc1[nH]c(=NC2CCCN(C(=O)C(C)CC(N)=O)C2)ccc1C#N CCC(C)C(C(=O)N(CC(O)CF)C)N(C)C(c1cnn(C)n1)=O C(C(CC(C)C)C(=O)N1CCOC(C(C)C)C1)NC(c1cccc(C)c1N)=O c1(C(=O)NC2CN(C(c3cc(C)nnc3)=O)CC23CC3)c(F)cc(Cl)cc1F CC1OCCC1CC(=O)N(CC(C)(C)CNC(=O)CNc1nccs1)C c1(C2(CC(=O)NCC3CCC3NC(=O)CCC=CBr)CC2)ccc(F)cc1 N1(CCOCC(C)C)CC2(CC(NC(c3coc(C(C)C)n3)=O)CO2)C1 N1(C(c2c(CC)[nH]cc2)=O)CC(C(=O)NC2CC(C)CC(C)(C)C2)C(C2CC2)C1 CCCCC(CNC(=O)CCNC(c1cccs1)=O)NC(c1cc(Cl)cnn1)=O c1(C(=O)NC2CCN(C(CC(C)(F)F)=O)C2)cnc2ccc(Cl)cn2c1=O CC(CC(F)F)C(=O)NCC=CCNC(c1ccc(CNS(C)(=O)=O)o1)=O C1(C(=O)NC(CNC(COc2c(C)occc2=O)=O)(C)C)CCc2nccn2C1 c1(C(=O)NC(CN(C(c2cnc(O)n2CC)=O)CC)C)cn(C)nc1C Cn1nc2cccc(C(=O)NC34CC(NC(c5ccc(=N)[nH]n5)=O)(C3)C4)c2n1 C1(COC)(CNC(=O)C=CC(N)=O)CCCN1C(=O)CCc1cnn(C)n1 c1(OC)cc(=NC(=O)C2(CNC(c3cc(O)ncc3F)=O)CC23CCC3)[nH]n1C c1(C(=O)NCC#CCNC(=O)C=CC2CCOCC2)c(Cl)ccc2c1OCO2 c1(C(C)=O)ccccc1C(=O)NCCC(O)CNC(c1cc(Cl)ccn1)=O N1(C(COc2c(C)c(F)ccc2)=O)CCC(N=c2[nH]nco2)(c2ccccc2)C1 C(C(=O)N(C)CCN(C(C1(C(F)(F)F)CCCCO1)=O)C(C)C)(C(C)C)SCC CC1(CCNC(=O)C(C2CCC2)NC(c2cnncc2O)=O)CCOCC1 CC1(C)CCOC1C(=O)NC1CCCC1n1cc(CS(C)(=O)=O)nn1 Cc1nn2c(c1C(=O)N(CC(O)CN(C)C(c1cnnc(Cl)c1)=O)C)NCCC2 C(=O)(C(C)(C)CC1CC1)NC1CCC(CCC(=O)N(CC#C)CCF)C1 c1(CCNC(C(=O)NCCCC(=O)OCCOC)=O)ccc(C)c(Cl)c1 C1(C2CCC2)(C(=O)NCCC2OCCN(C(C3(C=C)CC3)=O)C2)CC1(F)F Cc1c[nH]nc1CNC(=O)C(F)C1CC(NC(C2CS(=O)C2)=O)C1 Cc1cc(CC(=O)NC2CC(C(=O)NCc3cc(Cl)ccc3F)C2)cc(C)c1 C(=O)(CC(C)(C)C(F)F)NCC1N(C(C(C(C)C)n2ccc(C)c2)=O)CC1 C1(CC)CCC(C)CN1C(C12CC1CN(C(c1cccc(C)c1)=O)C2)=O CCN=c1[nH]c(C(N2CCC(NC(=O)C=CC3CCOCC3)C2)=O)cs1 c1(CSCC(=O)NC2C(C)CCCC2)cc2cnccc2[nH]1 c1(OC(C)C(=O)NCC2CCN2C(=O)Cc2cn(C)nc2Cl)ccc(F)cc1 c1(C(N(C2CCC(NC(=O)CCN3CCCC3=O)C2)C)=O)cnc2[nH]ccc2n1 c1(C(N(CC(C)(C)NC(C=C2CCN(C)CC2)=O)C)=O)cc2sccc2n1C CC1CN(C(c2coc(C3CC3)n2)=O)CC1NC(c1cnc(C2CC2)s1)=O CC(C)CC(C)(CO)NC(C1C2CC3C(C2NC(c2c[nH]ccc2=O)=O)C13)=O c1(NC(c2ccccc2Cl)C)[nH]c(=NCC(C)CN2CCOCC2)nc2sccc12 N1(C(C2(S(C)(=O)=O)CC2)=O)CCS(=O)(=O)CC1.C123CC(C1)(C2)n1cc(nn1)C3 c1(OC)ncc(C(N2CC=CC(NC(c3ccc(C(C)(C)C)s3)=O)C2)=O)cc1C CC(CCC(=O)NCCC(O)CNC(c1cnoc1C1CC1)=O)c1ccccc1 c1(N(C)Cc2scc(C)c2)nc(=NC2CSC(C)C2)[nH]c2c1CCC2 C1(C2(NC(=O)C(Cc3cn[nH]c3)NC(=O)C(O)CC(C)C)CC2)(OC)CCC1 N1(C(c2c(SC)nccn2)=O)CCC(C)(C)C(CNC(c2ccccc2)=O)C1 C1(C(=O)OC)C=CCCN1C(C1CCC(CNC(=O)CC2CC(C)=NO2)C1)=O C1(C(=O)NCCN=[N+]=[N-])CCN(C(C2(C(=O)O)CCCN2)=O)CC1 C1(C(N(C)Cc2c(Br)cnn2C)=O)CCCN(C(=O)C(C)(C)C)CC1 CC(C)CS(=O)(=O)NC(c1cc(CF)on1)=O Cc1cncc(-c2cn(CC3CCCN(C(C4CCC4)=O)C3)nn2)c1 C1(C(N2CC(SCC)C2)=O)CCN(C(c2ccoc2CC)=O)C(C)C1 CC1C(NC(c2coc(C3CCCC3)n2)=O)CCN1C(c1ncccc1N)=O C1(=CC(=O)N(CC(CC)NC(=O)C(O)P(C)(C)=O)CC)CN2CCC1CC2 C(=O)(C#Cc1ccccc1)N1CC(NC(=O)Cc2cccnc2)C(F)C1 C1(CCC(=O)N(C(CC)CC)C)CCCCN1C(=O)C=Cc1cncn1C N1(C(c2ncc(Cl)cc2Br)C(=O)NCC2CCOC2)CCCC2(C=CCO2)C1 c1(N(C)C)ccc(F)c(C(N2CCCC(C)(C(=O)O)C2)=O)c1 C1(CC(C)(C)C)CN(C(=O)Cc2cc[nH]n2)CCN1C(c1c(CO)cnn1C)=O CC1(C)CCc2oc(C(=O)NCC3(CNC(=O)Cc4cnco4)CC3)cc2C1=O c1(C(=O)NC2CC(F)(CNC(C(CC)N(C)C)=O)C2)c[nH]c2nccc-2c1C c1(C(=O)NCC(CC)NC(=O)CC2CC2C2CC2)ccc(-n2cnnn2)cc1 C1(C(=O)NC(C)(C)CNC(C2(Cl)CC2(F)F)=O)C2CN(C(=O)OC(C)(C)C)CC12 S(=O)(=O)(c1csc(C(=O)NCC2CCN2C(c2ccc(F)cc2N)=O)c1)NC C(=O)(C1CCCc2ccccc21)NCCCCNC(=O)C(c1ccc(F)cc1)=O N1(OC(c2c(SCCCC)cnc3ccccc32)=O)CCC2(CC1)CCS2(=O)=O c1(OCC)ccc(CCCC(=O)NCCCNC(c2ocnc2C2CC2)=O)cc1 c1(CC2CN(CC3OCC4(CC(F)(F)C4)C3)C2)cnc2cc[nH]c2c1 N1(C(c2ccncc2O)=O)CC(C2CN(C(C3CC3C3CCC3)=O)C2)C1 N1(C(CC(C)F)=O)CCC(C)(NC(=O)COCC(C)(C)C)C1 N1(C(c2cc(Cl)ccn2)=O)CC2(C1)CN(C(C13CCC(F)(CC1)CC3)=O)CCO2 N1(C(CCc2ccc(C)nc2)=O)CC2CCC2(CC(=O)NCCCCN(C)C)C1 c1(C2C(C(=O)NCC3C(CNC(C4C=C(C)CS4)=O)C3(F)F)C2)cccc(Cl)c1 c1(C(N2CCC(CNC(=O)C(F)C(F)(F)F)C2)=O)nnn2c1CCCCC2 c1(C(=O)NC(CN(C(c2n(CC)ccn2)=O)C)C)ccc2c(c1)COCCN2 Cn1cnc(N2CCC(NC(=O)COc3cccnc3)C(F)C2)c(Br)c1=O CC(C)CCC(=O)N1CC(CN(C)C(c2ccnc(N(C)C)c2)=O)C1 CCC(C)(F)C(=O)N1CCC(F)(CNC(c2cnn(C(F)F)c2)=O)C1 c1(C(N2CC3C(NC(c4scnc4Cl)=O)C3C2)=O)nnn2c1CSCC2 C1(NC(Cc2nc(C)sc2)=O)C(C)CN(C(=O)CCCOCCN(C)C)CC1C c1(C(=O)NCCC2CC(NC(C(C)SCC)=O)C2)cnn(CC(F)(F)F)c1 CC1CCN(C(c2csc(Cl)c2)=O)CC1NC(C1(C(F)F)CCCC1)=O c1(C(=O)NCC(C(N2CC3(C(C(=O)OC)C3)C2)=O)N(C)C)cc(C#N)cn1C C1(CNC(c2cn(CCO)nc2)=O)COC(CNC(C2CSC2)=O)C1 CCCCC(CC)(c1nnnn1CC1CCOC1)NC(C)COCC c1(CNC(C2(C)CCCS2)=O)nnc2n1CCN(C(=O)C(c1ccccc1)=O)C2 N1(C(CC2(C=C)CN(C(c3cnns3)=O)C2)=O)CC(C)(C)C12CCC2 C(C(N=c1nc(-c2ccccc2)[nH]s1)C1CC1)NC(c1ccn2ccnc2c1)=O c1(CN(CCNC(C2CC23CCOC3)=O)CC)ccccc1C C1(C)(C(=O)NCCC2CC(NC(C3N(CC)CC3)=O)C2)CCN(C)C1 Cc1c(Br)noc1C(=O)NCC1CCCN1C(C1CC1c1ccccn1)=O CC12CCC3N4CCOCC1N(CCOCC)CC3(C(CN)C4)C(=O)NC2=O c1(-c2nc(C(C)SCC)nn2CC2CCCOC2)cnn2cc(F)cc(F)c12 C#CC1(C(N2CC(CCO)(CC)C2)=O)CN(C(=O)C(C)CC)C1 O=C1COc2cc(C(=O)NC3CC(F)CN(S(=O)(=O)C(Cl)(Cl)Cl)C3)ccc2N1 C(c1c(C)coc1C)=CC(=O)NCC(CCOC)NC(c1cc(COC)cs1)=O c1(CCC(=O)OCc2c(OCC#C)cccc2F)cnc2n1CCCC2 C(=O)(C#CC1(CC)CC1)N(C1CCCC(NC(c2cc(SCC)ncc2)=O)C1)C C1(C(=O)NCCCN2CCN(CC)CC2)CN(C(c2ccncc2)=O)CCN1C N1(C(C)=O)CCC(C(=O)NCC23CC(NC(=O)CC4CC4(C)C)(C2)C3)CC1 N1(CC)CCCC1CC(=O)N(C1CCN(C(c2scnc2COC)=O)C1)C N1(C(CCc2cccc(CC)c2)=O)CCCC2CN(C(CC)C(N)=O)CCC12 C12(CNC(CC=C)=O)CC(NC(C3CCC3C)=O)(CO1)C2 O=C(C1=NOC2(CCN(Cc3cc(O)ccc3Br)C2)C1)NCCCCCO c1(C(=O)NCCCCC2CN(C(C=CCC)=O)C2)cnc2c(c1)OCC(=O)N2 CC1(NC(=O)C(F)OC(F)(F)F)CCN(C(C2CC2c2cccc(OC)c2)=O)C1 c1(C(N2CC(NC(Cc3cc(C)[nH]n3)=O)C3C2C3)=O)cnc2cc[nH]c2c1 N1(C(C2CCC(=O)O2)=O)CC(C2CCCN(C(c3cccc4nccn34)=O)C2)C1 N1(C(C(=O)NCCOCC)=O)CC(OC)CC1(C)CNC(=O)CN1CCS(=O)CC1 C12(C(N3CC4CCC(NC(COCCOC)=O)(C3)C4)=O)C3CCC(CC13)C2(F)F Cc1cc(C(=O)N(C2CCN(C(C3NC(=O)CC3C)=O)CC2)CC2CC2)ccn1 C#Cc1cccc(C(=O)N(C2CCCN(C(=O)CC3COC4CC3C4)C2)C)c1Cl c1(C(N2CC(CC(C)NC(C3(CC#C)CCCO3)=O)C2)=O)cc(F)c(C)cc1O C1(C(=O)NCC(C(=O)N(C2(SC)CC2)C)N(C)C)(OC)CCCC1 C1(C(=O)NC2CN(C(C3(CC(C)C)COC3)=O)CC(C)C2)CCc2nccn2C1 Cc1c(C(=O)NC2CCC2NC(=O)C(C)CF)nnn1Cc1ccccc1 Cc1cc(CNC(C2CCC2CNC(=O)C=Cc2ccccc2)=O)ccc1F C(=O)(C(F)C(=O)NCC1(CC(=O)N(C)CC2CC2)CC1)OCC Cc1cc(OCCC(=O)NCC2COCC2NC(c2cc[nH]c2)=O)c(C)c(C)c1 c1(OC)cc(C(N2CCCN(Cc3ccccc3F)CC2)=O)cc(Br)c1O C1(CC(=O)Nc2cc(OC)cc(Cl)c2)CC(N=c2ccn3ncc(C#N)c3[nH]2)C1 C1(CCC)CN(C(=O)CC2CCC(C#N)C2)CC1NC(=O)CCN(CC)CC Cc1cc2cccc(C(N3CCOCC3CC3CCC3)=O)c2o1 c1(N(C)C)ncnc(NC2CC3CN(C(=O)C4=CC5CCCC45)CC23)c1[N+](=O)[O-] C(=O)(C1=CC2C=CC1C2)N1CCC(CC(N2CCC(CC#C)C2)=O)C1(C)C c1(C(N2CCC(C)(CNC(C34CCCN(CC3)C4)=O)C2)=O)nccc2ccsc12 C1(CNC(c2nc(C(C)OCC)sc2)=O)C(C)CCN1C(c1cccc(N)c1)=O C1(NC(CNS(C)(=O)=O)=O)CC(=O)N(C2CCCCCC2)C1 N1(C(CC2CN(C(c3c(C)n[nH]c3)=O)CC2C)=O)CCCCCC1C C1(NC(c2cc(CC)no2)=O)CN(C(=O)C(S(C)(=O)=O)C2CC2)CC2(CCC2)C1 C1(CCC)(NC(=O)CNC=O)CCCN(C(=O)Cc2cnc(Cl)cc2C)C1 C(Cc1ccccc1)(CCNC(=O)C=CC1CCC1)NC(COCC(=O)OC)=O C=C(CNC(N1CCN(C(=O)Cn2cncn2)CC1)=O)c1ccccc1 N1(C(C(COC)(C)C)=O)CCC(C)C(NC(=O)CN2CCCCC2=O)C1 C1(CNC(C(CC)O)=O)CC(F)(F)CN1C(c1cc(F)ccc1Cl)=O c1(CNC(C(C)c2cccs2)=O)nnc2n1CCN(C(=O)C(C#N)C1CC1)C2 c1(OC)ccc(C(=O)NCCC2(C)CCN(C(C3(C4CCC4)CC3)=O)C2)c(Cl)c1 c1(Cn2c(C(N3CCC4(C(C(=O)OC)C4)C3)=O)nnn2)ccc2c(c1)CCC2 c1(C(n2cc(Cn3nccc3C(=O)O)nn2)CC)ncnn1C.C1(=O)CON1 c1(NC(c2ccc(OCC(F)F)nc2)=O)ccccc1OC(F)(F)F CCC(C)CC(C(=O)N(C)CC1CN(C)C1)NC(C1CC(=O)N(CC)C1)=O c1(C2(C(=O)OCC)CCC2)c(Cl)cccc1Cl.C1(=O)CC(C)CO1 c1(CNC(NCC(C)S(C)(=O)=O)=NCC2CCN2C2CC2)ncnc2c1OCCO2 C1(NC(c2cnccc2C(F)(F)F)=O)C2CCC1N(C(C1(CO)CCCO1)=O)C2 c1(CC)ccc(S(=O)(=O)N2CCCC(C(N3CCOC(C)C3)=O)C2)s1 c1(C(=O)NC2CCC(CNC(=O)COCCF)CC2)ccc(F)c(O)c1F c1(C(N(CCN(C(C(C2CC2)OC)=O)C)C)=O)c(C)cc(Cl)cc1N c1(C(=O)NC2CN(C(C3ON=C(C(C)C)C3)=O)CC23CC3)cnn2c1OCCC2 c1(C(=O)NC(C(=O)NCC(C)CC2CC2)Cn2ccnn2)ccc(O)cn1 C1(CNC(C2C(OCC)CC2)=O)(CNC(C2(CF)CCC2)=O)CCCCC1 C1(C(=O)NCC2CC(NC(c3c(N)sc(C)c3C)=O)C2)CC(C(C)(C)C)=NO1 C1(CNC(Cn2c(C)nc(C)n2)=O)CC2(CCC2)CN1C(=O)C(C)C1CCCC1 N1(C(C2CCCS2(=O)=O)=O)CCN(C(c2ccc(O)nn2)=O)C2CCCC12 CN1CCCCC1C(=O)NCc1cn(CC(=O)NOCCCF)nn1 c1(Sc2cccc(C(N3C(C(=O)OCC)CC(O)C3)=O)c2)ccc(C#N)cc1F Cn1ncc2c(C(N3CC(NC(c4ccc[nH]4)=O)C(C)(C)C3)=O)cccc12 C1(NC(c2c(C)nc[nH]2)=O)CC2C(NC(C3CCC3C)=O)C2C1 CCN=c1ccc(C(=O)NC(C)CNC(=O)Cc2ccsc2Br)c[nH]1 C1(C(c2ccncc2Cl)N2CCC(n3cc(C(C)O)nn3)C2)CCCN1C=O CC1CC2CN(C(c3ccc(C(F)(F)F)s3)=O)CC2N1C(=O)CC1CC2CC2C1 c1(C(N2C(CNC(=O)CNC(=O)C3CC3)C=CC2)=O)csc2c1CCCC2 N1(C(C(c2cccc(C)c2)CN)=O)CCOC2(CCS(=O)(=O)C2)C1 N1(C(=O)NCCC2C(C)(C)C(=O)C2)CC(C(N2CCOCC2)=O)C(F)(F)C1 c1(C(=O)NC23CC(CNC(c4cc(OC)ns4)=O)(C2)C3)cc2sccc2[nH]1 CC(CF)CC(=O)N(CCNC(=O)C(F)=CCCF)CCc1ccccc1 CC1CCS(=O)(=O)CCN1C(c1ccn(C(F)F)n1)C(=O)NC1CCC1 C12(C(=O)NCC#CCNC(Cc3cccc(OC(C)C)c3)=O)CCC(C)(C1)OC2 c1(SC)ccc(C(N2CC(N(C(=O)C(O)CN3CCCC3)C)C2)=O)cc1 CCC(CC)CC(=O)NC1CCCCC1C(=O)NCCN1CCCC(O)C1 N1(C(C(COC)OC)=O)CCC(NC(=O)Cc2cccc(F)c2)C1CCO c1(C(N2C3(CNC(CN(C(C)C)C)=O)CCC2CC3)=O)cccc2c1CCO2 Cc1nc(CO)sc1C(=O)OCc1ncccc1C(C)(C)C C1(NC(C2CC=C(C)CC2)=O)C2CCCC1CC(NC(=O)CC(C)(C)C)C2 CC1(O)CCN(CC(N2CC(O)CC2CNC(=O)CC(F)(F)c2ccccc2)=O)C1 CC1CC(COC(=O)CCOc2cccc(C(C)(C)C)c2)CC(C)O1 c1(C(N2C(CNC(C(C)C)=O)CC(F)C2)=O)cccc(S(C)(=O)=O)c1F C1(CCCOC)CN(C(=O)CSCc2cccnc2)CCO1.C12CC1C(=O)NC2 N1(C(C=CC)=O)C(CNC(c2ncccc2OCC)=O)CC2CCCC12 CC1(C)CCCC(C(=O)NCC23CC2CN(C(=O)Cc2coc(C4CC4)n2)C3)C1 c1(N(C(=O)NC2CCOCC2F)Cc2nccc(C)n2)cc(F)ccc1C N1(C(CCc2cc(C)[nH]n2)=O)CC2(C=C(C(=O)N3CCOCC(C)C3)CO2)C1 N1(C(c2ccc(CC)cc2)=O)CCCC(CO)(NC(=O)C=C(C)C(F)F)C1 c1(C(N(CCN(C(c2cc(CC)c(C)cc2)=O)C)C)=O)nccn2cnnc12 c1(COC(=O)Cc2ccc(Cl)cc2Cc2c(F)cccc2F)c(F)cccc1F c1(OC)ccnc(C(=O)OCC(=O)NCC2CCC(C)O2)c1O CCCCC(C(=O)NC1CCN(CCCCCF)C1)NC(=O)OC(C)(C)C C(=O)(C1=CC2(CCOC2)C1)NC1CN(C(c2c(C)cnnc2)=O)C(C)(C)C1 C(c1ccccc1[N+](=O)[O-])=CC(=O)NC12C(CN(C(COCCC(C)C)=O)C1)C2 C(=O)(C(C#N)C(C)(C)C)NCC(C)(C)NC(c1ccc(Cc2nccs2)cc1)=O C1(C)(C(=O)NC(CC)CNC(=O)C(O)CCSC)CCCS1(=O)=O Cc1nnccc1C(=O)NC(CN(C)Cc1ccccc1)C(=O)NCCN=[N+]=[N-] C(=O)(C(C)C(O)C(C)C)NCCn1ccc(C(NOCCCOC)=O)c1 C(=O)(CCCC(C)C)NCc1nc(C(N(CC=C)CCC)=O)sc1 c1(C(C(=O)NCC2(O)CN(C(=O)Cc3csc(C4CC4)n3)C2)O)ccc(Cl)cc1 c1(OC)ccc2c(c1)CCC(C(=O)NC1CCCC1NC(C1(C(N)=O)CC1)=O)C2 Cc1nc(NCC(=O)Nc2ccc(F)cc2F)cc(=NCCOC2CCCC2)[nH]1 C1(NC(Cc2c(C#C)cccc2)=O)CN(C(=O)CCCC)CCC1(F)F c1(OC)c(Cl)ccc(Cl)c1C(N1CC(O)(CCNC(=O)C(C)O)C1)=O N1(CC(=O)NC2CCC(N(C)C(C3CCNC3=O)=O)CC2)CCCNS1(=O)=O Cc1ccc(NC(=O)CC(CC(C)C)NC(=O)CC(C)CN(C)C)c(C)c1O C1(NC(c2scc(C)c2)=O)CC12CC(NC(=O)CC1C=NN(C)C1=O)C2 C(=O)(C1=CC2CCCC12)NCC(C)(C)CNC(c1ccc(N)cc1O)=O c1(C(=O)NCC(C)=CC(=O)NCC(O)C2CCC2)ccc(O)nc1 c1(C(N2CCC(NC(C3CC34CC(F)(F)C4)=O)CC2)=O)cc2c(cn1)CCCC2 N1(C(c2ccc(CC)cc2)=O)CCCC2C1CCN2C(=O)CC1CC(=O)NC1=O N1(C(C2(CC)CN(C(=O)CC3CCCOC3)C2)=O)CC2CC2C2CC12 C#Cc1ccc(C(N2CC(C(C(=O)NCCC(C)CCO)OC)C2)=O)cc1C N1(C(C(C)SC)=O)CCCC2(CCCCC2NC(c2cn(C3CCC3)nn2)=O)C1 N1(CCC)CC(CNCC2CCCOC2)CC1=O C1(NC(c2c(OCCC)cccc2)=O)CCCC2CN(C(C3CC3OC)=O)CC12 N1(C(c2ccc(N(C(C)=O)CC)cc2)=O)CC2C(NCCCO)CS(=O)(=O)C2C1 C1(CNC(=O)C(C2CCCCCC2)O)C2CC1N(C(c1nc(Cl)cs1)=O)C2 c1(C(CCC)C)nc(-c2cc(C(C)C)nn2CCOC)n(CC(N)=O)n1 Cc1ccc(CN2CCCC(C(N3CC4CC(C3)O4)=O)CC2)c([N+](=O)[O-])c1 CC1CCn2cc(C(=O)NCc3nc(CNC(C4COC4)=O)cc(O)n3)nc2C1 Cc1nn(CCO)c(C)c1C(=O)N(C(C)CNC(=O)C(C)CO)C C1(NC(C(CSC)O)=O)CC2CC(NC(=O)C=C3CCCCC3)CC12 c1(C(=O)NCC2CCN(C(CCC=C=C)=O)C2(C)C)nc(C)c(C)[nH]c1=O N1(C(Cc2cnc(C)[nH]2)=O)CC2(C1)CN(C(=O)C(C#N)CC1CC1)CCO2 C1(NC(CC2C(=O)NC(=N)S2)=O)CCCCCN(C(C23CCC(F)C2CC3)=O)C1 C1(C2CCCCN2C(C2CC2F)=O)(CNC(=O)C(F)=CC2CC2)CCOCC1 c1(C(C)=O)cc(C(N2CCC(CO)(NC(C34CCC3C4)=O)CC2)=O)c(C)nc1C C1(CC(=O)NC(CCCC)C)N(C(=O)CSCCC(C)C)CCC1(C)C C12(NC(c3cccc(SC(F)(F)F)c3)=O)CC(C1)N(C(c1cncc(O)c1)=O)C2 c1(CC)cc(C(=O)NC2CCC(NC(=O)CN3CCCC3CO)C2)on1 C(C(C)S(C)(=O)=O)(c1ccc(C)cc1)N1CC2C(C(=O)NCCn3cccn3)C2C1 c1(C(N(CCN(C(C(C)OC2CCCC2)=O)C)C)=O)cccc(C2CCCC2)c1 c1(OC(c2ccnn2CCOc2cscn2)=O)cccnc1NC1CCCC1 Cc1ccnc(O)c1C(=O)N(CCCNC(=O)C(C(C)C)n1cnnc1)C C1(CCC(=O)NCCN(C(=O)C(CO)NC(N)=O)C(C)C)CC(F)(F)C1 C1(NC(C(C)OCC)=O)CN(C(c2cc(C)c(CC)nc2O)=O)CC1N=[N+]=[N-] c1(C(=O)NCC(C)NC(=O)Cc2cnco2)ccc(C2CCC2)cc1 C#CC(C)(C)C(=O)NCC1CCN1C(C1(n2ccnn2)CC1)=O N1(C(CC(=O)NC)=O)CCOCC2(C1)CN(C(=O)CN(C1CCCC1)C)CCO2 C(CC(CC)C(=O)NCC1(CNC(c2cnc(Cl)s2)=O)CC12CCC2)=CCCC C1(NC(C2C=C(C)CS2)=O)CC2CCC1CN2C(C1CCCN(C(C)C)C1)=O C123CCCC1N(CCC2)C(=O)CCOCC(=O)NC3.C(C(C)(C)C)OC(C)C C(N=c1nc2c(cnn2C)c(N2CCN3C(=O)NCCC3C2)[nH]1)C1CC(OC)C1 Cc1ccc(C(N2C3CCC2CN(C(C2CCN(C)C2C)=O)C3)=O)c(N)c1Cl C1(=O)C2CN(Cc3n[nH]cc32)C(=O)C(=O)C(CCC=C)N1.C(C)(C)(C)O.OCC c1(C(=O)O)cc2c(s1)CCC2=O.c1(C(N2CCCC2)=O)cc([N+](=O)[O-])n[nH]1 c1(C(=O)NC(C(C)NC(C2(CCOC)CCCC2)=O)C)cnc2ccc(F)cn12 C1(CC(=O)N(C(CCO)C2CC2)C)C2CCCC2N1C(C1CC=CCC1)=O CC(c1cnn(C)c1)=CC(N1CCN(C(C2CSCCS2)=O)C(C2CCC2)C1)=O c1(C(=O)NC(CNC(c2cnc(C)s2)=O)CC(C)C)ccc(Cl)c(F)c1 c1(C(=O)NCCCN(C(C2CC(C)=C(C)CC2)=O)C)ccc2n[nH]cc2n1 c1(NC(C)=O)cccc(F)c1C(N1CC(O)(CN(C)C(C2CCS2(=O)=O)=O)C1)=O C1(C(N2C(C(=O)NOC3CCOC3)CC(F)C2)=O)CC2(CCO1)CC2 N1(C(c2snc(O)c2Cl)=O)CCC2CCN(C(c3cc4ccccc4o3)=O)C2C1 N1(C(C2(F)CCC(C)CC2)=O)CCN2CCN(C(=O)CC3(CO)CC3)CC2C1 N1(C(c2c(C)ncnc2)=O)CCC(CNC(c2ccncc2)=O)C(C)C1 c1(OC)ccc(C(=O)NC2CCCC2NC(c2c(C)nn(C)c2Cl)=O)c(F)c1 c1(OC)ccnc(F)c1C(N1CCOC(CNC(=O)CCC(F)(F)F)C1)=O c1(C(N2CCc3cc(F)ccc32)=O)cc(Cl)c2cn[nH]c2c1 C1(C)(CNC(CC(CC)C2CC2)=O)CN(C(=O)CC2CC(C)(C)C2)CC1C Cc1ccc(Cl)c(C(O)CN2CCC(OCc3cccnc3)CC2)c1 N1(C(CCC(=O)NCCC)=O)C(CC(N2CC(CCO)C2)=O)C2CCCC12 C12(C(=O)NC(C3CCN(C(c4ccn(C(C)(C)C)c4)=O)C3)C)CC=CC(C1)OC2 CCC(O)C(C)(C)C(=O)NC1CN(C(=O)Cc2ccnc(F)c2F)CC1SC C(C1CN(C(C2C(C)C2C)=O)CC1C(N1CC(=O)NCC1C(C)C)=O)=CC N1(C(C(Cc2cn[nH]c2)NC(c2c(C)cns2)=O)=O)CC2(CNC(=O)N2)C1 N1(C(CC(C)F)=O)CC(C(N2CCC2CO)=O)CCC1C Cc1oc(S(N)(=O)=O)cc1C(=O)NC1CN(C(c2cc(F)cc(F)c2)=O)CC1C c1(NC(N(C)C)=O)cc(NC(=O)Nc2ccc(-c3ncn(C)n3)cc2)cc(Br)c1 CC1(CNC(=O)C(F)=C2CCC2)CCCN(C(=O)C(c2cccc(F)c2)O)C1 C1(CNC(c2cc(OC)n[nH]2)=O)CCCC2CN(C(=O)Cc3cncn3C)CC12 C1(O)(CN(C(=O)C(c2cccs2)NC(=O)CCc2ccoc2)CC)CCC1 c1(C(N2CCCC(CC(=O)Nc3ccc(C4CC4)nc3)C2)=O)cc([N+](=O)[O-])n[nH]1 CC(C)CS(=O)(=O)CCC(=O)N1CC2CC(NC(=O)C(C)N3CCC3)CC(C2)C1 c1(C(=O)NCC(C)N(C(C(C)NC(CC)(C)C)=O)C)cc2ccccc2c(O)n1 c1(C(=O)NCC(CN(C(=O)C=C2CC2)C)(C)C)cccc2c1OCCC2 C1(CCO)CCN(C(=O)C=CCCC(C)C)CC1.C=CC(C)C(=O)NC1CC1 N1(C(C2(C#C)CCC2)=O)CCCC(CN(C)C(C2(OC)CS(=O)(=O)C2)=O)C1 c1(C(=O)NCc2ncsn2)nnc(-c2ccc(Br)o2)o1 CCC(C(=O)NC1CN(C(=O)C(F)F)CC1(C)C)C(C)O c1(N2CCC(C(C)NC(CN(C(C)C)C)=O)C2)ncccc1C(F)(F)F C1(OC(C2CC3CC2(c2ccncc2)C3)=O)CCOC2(CCC2)C1 C1(CNC(C2(C#N)C(C)C2)=O)(CNC(=O)Cc2c(Cl)cnn2C)CCCCC1 C1(NC(c2cnc(C)s2)=O)CC2CCC(C1)N2C(=O)CCCc1cccc(F)c1 N1(C(c2nc(CC)oc2C)=O)CCCCC(NC(c2csc3nnsc23)=O)C1 c1(C(=O)NC2(C(N(CC(C(=O)OC)C)C)=O)CC(F)C2)cc(C)c(C)o1 N1(C(C2CC3(C(OC)CC3)C2)=O)CC2CCN(C(c3[nH]c(=N)sc3C)=O)CC2C1 N1(C(Cc2c(C)ocn2)=O)CCCC(F)(CNC(=O)CN2CCSCC2)C1 C1(OC(=N)O)CN(C(=O)CCOCCNC(C2(Br)CC2)=O)C1 N1(C(C2CCC(C)N(C(=O)CCc3ccsc3)C2)=O)CC2CN(C)CC2C1 C1(NC(C2N(CCC)CCC2)=O)CCN(C(=O)CN2CC(=O)N(C)C2=O)C12CC2 C1(C(N2CCC(CCN(C(CSC)=O)C)CC2)=O)CCc2nc(C)cn2C1 c1(C(C)=O)ncc(C(=O)NCCC(O)CNC(c2sccc2F)=O)s1 N1(C(CC(C)C)=O)CCC2CN(C(=O)C(F)Cc3ccc([N+](=O)[O-])cc3)CC2C1 C1(NC(N)=O)CCCC(CNC(c2coc(Cl)n2)=O)CC1 C#CCCCCC(=O)NCC12CC(CN1C(c1ccc(N)c(O)c1)=O)C2 C=CC1CCN(C(=O)CC2(C=C)CN(C(=O)CC3CCCC3C)C2)CC1 C(=O)(C1=C(c2cnco2)N(CC2CCCS2)C(=S)NC1c1ccc(=N)[nH]c1)OCC C(CCCC(=O)N1CCCC1C(C)NC(c1cnn(C)c1C(F)F)=O)SC c1(C(=O)NCCN2CCN(C(C=CCCC)=O)CC2)cc2c(s1)CCC2 c1(CC(=O)NC2C(CNC(Cc3nc(C)sc3)=O)C2)cccc(C(C)C)c1 n1(CC(N2C(CC(=O)NCc3ccsc3)COCC2)=O)ccc2c(F)cccc12 C1(C(N2CCC(C(C)NC(C3(O)CC3)=O)C2)=O)CC(C)(C)SC(C)(C)C1 C1(C(=O)NC(C)(C)CC2CCC2)C(C2CC2)CCN1C(C1CS(=O)(=O)C1)=O C(=O)(C1CCc2cccc(O)c21)N(C(C)(C)C)C(=O)COCc1cccnc1 C1(C(N2CC(n3cc(NC(c4cncnc4)=O)nn3)C2)=O)(C(F)F)CCCOC1 c1(CC(=O)NC2CN(C(CCCN(C(C)=O)C)=O)C(C)C2)ccc(C#N)cc1 c1(N2CC(CC(C)NC(C3CCCN(C(C)=O)C3)=O)C2)ncc(C)c(C)n1 C12(C(=O)OC)CC1CN(C(C1CN(C(c3cncc(OC)n3)=O)CCO1)=O)C2 CCCC(CC)C(=O)NC12COC(C1)C(NC(=O)COCc1nccn1C)C2 c1(C(=O)NC2C=CC(CNC(Cc3nc(CC)sc3)=O)C2)ccc(C#N)[nH]1 C(C(=O)N1CC(C(=O)NCCc2cc[nH]n2)C(C)C1)(C(C)C)SC c1(NC(C(CC#C)(C)NC(=O)C(C)OCC2CC2)=O)cc(C)cn(C)c1=O N1(C(C2(C)CCC(=O)N2)=O)CCN(C(c2ccc(N)c(Cl)c2O)=O)C2CCC12 CON1CC(C(=O)NCC(C)(C)OCCNC(=O)C(C)(C)C(=O)OC)CC1=O N1(C(c2cncnc2)=O)CCN(C(C2C3CCCOC23)=O)C2CCCC12 c1(C(=O)NCCCC(C)NC(C2N(CC)C(=O)CC2)=O)cc(=O)c(Br)c[nH]1 C12(C)CC(C1)C2.C1(CCC(=O)NCC(C2CCCN2C(N)=O)(C)C)CCCN1C N1(C(C(c2ccccn2)C)=O)CCC(C)(CNC(C2CN(S(C)(=O)=O)C2)=O)C1 C(CS(=O)c1ccccc1)NC(C(=O)NC(C1CC1c1cccnc1)C)=O C=C(C)CCC(=O)NCC1(CNC(c2csc(CCCCC)n2)=O)CCC1 C1(N(C(=O)CCC2CC2(C)C)C)C2CN(C(c3csnc3Br)=O)CC12 N1(C(c2nc(C)nn2C)=O)CCC2CCCC(C1)N2C(c1c(C)cncc1C)=O c1(CNC(C2CC(C)(NC(C3C(C(C)(C)C)C3)=O)C2)=O)ncc(Cl)cn1 C(=O)(CC(C)(O)CC(=O)O)N1CC(F)CC(NC(c2c(F)ccc(C)c2F)=O)C1 N1(C(C2CC(NC(c3c[nH]c(=NC)s3)=O)C23CCC3)=O)CCCCC2(CCC2)C1 C1(NC(C(C(C)C)NC(C)=O)=O)CC2CC1CC2C(=O)NC1CCOCC1 c1(C(=O)NC2CCCC(CNC(COCC=C)=O)C2)c(C)nn(C)c1Cl C1(C(=O)NC(C)CSCCO)(COC)CN(C(=O)Cc2ccccc2)C1 C1(N(C(c2cc(CCNC(CCOCC(C)C)=O)on2)=O)C)CCC(=O)N(C)C1 CC(O)C(C(=O)NCC1(F)CC(NC(c2cc[nH]c2)=O)C1)NC(=O)C(F)(F)F Cc1[nH]nc2ccc(C(N3CC4(NC(c5c[nH]ccc5=N)=O)CCC3C4)=O)cc12 C(=O)(CC(C)C(F)F)N1C(CC(=O)NC(c2onc(C)n2)(C)C)CCC1 c1(C2(CNC(CN(C(C)C(=O)N(C)C)C)=O)CCC2)ccc(F)cn1 C(=O)(C1CCc2nccn21)N1C2CN(CC1)C(=O)COC(=O)C2.C(=O)(NCC)NC c1(C(=O)NC2CC(NC(C3CC(C4CC4)C3)=O)C2)ccn(CC(F)F)c(=O)c1 C1(C(=O)NC2C(C(N)=O)CCC2)CCCN(C(=O)CC2CCOC2)CC1 c1(C(=O)NC2CCCC23CN(C(C2CC=CCC2)=O)C3)ccc2c(c1)CCOC2 C1(CC=C)(NC(c2ccoc2C)=O)CCN(C(C2(n3cccn3)CCC2)=O)C1 C(=O)(C(F)C(C)C(F)(F)F)N(CCCCN(c1nc(C)nc(C#N)c1)C)C c1(C(=O)NC2C=CC(CNC(C(C(C)C)C)=O)C2)cccc2c1CCN2 C1(C(=O)NCC(COC)(F)F)CCCN1NC(=O)C(O)CC1CCCC1 N1(C(c2ccc(CC)[nH]2)=O)CC(N=c2[nH]nc(C(F)F)s2)C2(CCC2)C1 c1(C(=O)NC2C(NC(C(c3cccc(OC)c3)O)=O)C2)cccc2ncsc12 Cc1ccc(C2(C(N3CCC(CF)(NC(C4C(C)C4(F)F)=O)C3)=O)CCC2)cc1 N1(C(CCN(C)CC)=O)CC(CNC(c2ccc(CNC(C)=O)cc2)=O)C2CC12 CCCC(CNC(c1c[nH]nc1C(F)F)=O)C(=O)NC(c1ccncc1)C Cc1nc(C(N2CCCC(CS(C)(=O)=O)C2)=O)ccc1OC(F)F N1(C(C(C)(CO)OC)=O)CC2CCC(C1)N2C(c1cccnc1NC(C)C)=O N1(C(c2ncc(OC)cn2)=O)CCCCC(NC(=O)C=C(F)c2ccccc2)C1 C1(NC(c2cnc(OC)s2)=O)CCCC1(C)CN(C(=O)CC1CCCCN1C)C C(=O)(C(C(C1CC1)C1CC1)N(C)CCc1nc(C)cs1)NCCC c1(OCC(=O)OC)ccccc1C(=O)NCC1CC(NC(=O)C(O)C2CCC2)C1 C1(C(=O)NCCC(C)N(C(c2ccc(SC)o2)=O)C)CC2OC(=O)OC2C1 N1(C(c2c(C(C)C)cccc2)=O)CC2CCC2(CNC(C2(CO)CC2(F)F)=O)C1 c12cc(F)ccc1O2.N1(C(c2c(OC)c[nH]n2)=O)CC(N(C)C)C(C)C1 N1(C(c2oc(CC)c(C)c2)=O)CCCC(C)(C)C1C(=O)NC(C)C(C)(C)O c1(C(N2CC(Cn3cc(CCN(C)CC)nn3)C2)=O)c(C)cnc2ccccc12 c1(OC)cc(CCN=C(NCC(C)C(C)(C)C)NC2CCC2)ccc1C c1(SC)cncc(C(=O)NCCCNC(C2(F)CC2c2ccccc2)=O)c1 Cc1ccc2ncnc(N3CCC(NC(c4nccn4C)=O)C(O)C3)c2c1 c1(C(=O)NC23CC(CNC(C(C(CC)C)C)=O)(C2)C3)ccc(Cl)c([N+](=O)[O-])c1 c1(C(=O)NCCC(C)NC(C2(NC(=O)OC)CCCCC2)=O)cc2c(s1)CCC2 CCC(CC(F)F)C(=O)NC1CCN(C(c2cc(-c3ccco3)on2)=O)CC1F Cc1cc2cccc(NC(c3csc(NS(=O)(=O)c4ccccn4)n3)=O)c2cn1 c1(C(=O)NCCN(C(CCC(C)SC)=O)CC(C)O)cnc(C)c(N)c1 CC(C)C(C(=O)NCC(O)CN(C)C(C1CCCCN1C)=O)n1cnnc1 C1(C(=O)NC(C2CN(C(=O)CS(=O)(=O)N3CCCCC3)C2)C)(CO)CCCCC1 CC12CN(C(C3(C4CC4)CC3)=O)C(C(N3CCC(C)(F)C3)=O)(C1)C2 C(=O)(CC(C)C(C)(C)C)N1CCCC(NC(c2c(C)n[nH]c2)=O)C1 c1(OC)c(C(N2CCC(NC(=O)CCC(C)(F)F)C(C)C2)=O)cccc1F c1(NC(C2CC=CCC2)C(=O)NC(C2CCCCC2)CC)coc(C)c1 Cc1oc2cc(C(N3CC(C)(NC(C4CCCCS4)=O)C3)=O)[nH]c2c1C Cc1nnc(C(=O)NC2CC(F)(CNC(c3cccn3-c3ccccc3)=O)C2)s1 C(=O)(C(=O)N=S(C)(C)=O)N1CCC(O)(C(C)NC(=O)CC2CC23CC3)CC1 Cc1cc(Cl)c(F)cc1C(=O)NC1CCCCC1C(=O)Nc1ccc(C#N)nc1 C1(NC(=O)CC2CC2)CCC2(CCC2)C1NCC(N1CCN(C(=O)NC)CC1)=O c1(C(=O)NC(CN(C(CSCCCC)=O)C)C)ccc([N+](=O)[O-])c(SC)c1 C1(NC(C=C(CC)CC)=O)COCCN(C(=O)C(F)=C(C)C)C1 c1(C(N2CC3C(NC(CN(CC(C)(C)C)C)=O)(C3)C2)=O)cn2cccnc2n1 C1(NC(c2cn(CC)nn2)=O)CC(C(=O)NC2CC(CN(C)C)C2)CC1O CN1CCC2CN(C(C3(NC(=O)CC4CCC(=O)NC4)CCCC3)=O)CCC12 c1(C(=O)NCC2N(C(C3=CC(C)(CC)C3)=O)CCC2)cc2c(C)nn(CC)c2s1 c1(CC(=O)N(CCNC(CCCc2onc(CC)n2)=O)CC)cccc(F)c1 C(=O)(C1=C(CCCCl)N(CC2CC2)C(=S)NC1c1cccc(Cl)c1)OCC C(=O)(CC(C)(CN(C)C)C(F)(F)F)NC1CC(NC(c2c(C)cccc2F)=O)C1 N1(C(CCOC)=O)CCC(O)(C(C)CNC(=O)C=C(Cl)Cl)C1 C(CC(O)C(=O)NCc1ccc(C(N2CCC2CC2CCCC2)=O)s1)N(C)C C1(C(=O)OCC)CN(C(=O)C(=O)NCc2nc(=O)n(C)[nH]2)c2ccnn2C1 n1(CC)nc(C(=O)NC2(C)CCN(C(C3(SC)CC(O)C3)=O)C2)cc1C O=C(C1=CS(=O)(=O)CCC1)NC1COC2C(NC(C3(O)CCC3)=O)COC12 Cc1nc(C(N2CC(N(C)C(c3cc(Cl)cn3C)=O)C(O)C2)=O)ccc1[N+](=O)[O-] c1(C(N(C2CCCN(C(CCCNC(C)=O)=O)C2)C)=O)cnc2ccnn2c1 C1(NC(c2n(C=C)nnc2)=O)CCC12CN(C(c1ccc(OC(C)C)nc1)=O)C2 C#Cc1cnc(C(=O)N(CC(=O)NC2C(C)C2(C)C)C)c(C)c1 c1(OC)ccc(CCCCC(=O)N2CCC(CC(C)NC(=O)C(C)O)CC2)cc1 c1(C(=O)NCCNC(CCCCCC(C)O)=O)cc(Cl)cc2c1NCCC2 S(=O)(=O)(c1cc(C=CC(=O)NCC(c2ccccc2)C)ccc1OCC)NCC c1(C(N2C(CNC(CCCOCC)=O)C(C)CC2)=O)cc2c(s1)CCC2 C1(C(=O)NCC2(F)CCC(NC(C3CNC(=O)N3)=O)C2)(CSC)CCOCC1 c1(C(=O)NC23CC(CNC(=O)C=C4CCCCC4)(C2)C3)ccc(F)c(Br)c1 C(=O)(CCC(F)F)NC(CN(C)C(C1CCCC1(C)C)=O)(C)C C(CNC(c1cc(C2CC2)[nH]n1)=O)(CC(=O)NCCc1csnn1)OC c1(C(=O)NC2C(NC(C3CC(C)OC(C)C3)=O)COC2)c(Cl)ccc(F)c1F Cc1cc(F)ccc1NC(=O)C(c1cc(Br)c(Br)o1)N(C)Cc1ccc(F)c(Br)c1 C1(C2CCCCC2)(NC(C2(C)C=CCN2C(c2ccc(O)cn2)=O)=O)CC1 c1(C(=O)NC(C(C)C)CNC(=O)Cc2cc(F)cc(Cl)c2)cccc2ncnn12 C(=O)(C(C)c1cc[nH]n1)NC(C1C(C(=O)NCCN(CCCC)C)C1)C n1(CC(=O)NC2C(NC(CCCC(C)C)=O)C2)ccc2cc(Br)ccc12 c1(C2(C(=O)NC3C(CNC(Cc4nnc(C)o4)=O)C3)CC2)cccc(F)c1F N1(c2c(F)cnc(OC)n2)CC2CN(OCC)CC2C1.c1(C)cc(Br)ccc1O c1(COC(C)(C)C)ccc(C(F)(F)F)c(Cl)c1.C12CC(C1)NC(=O)CN(C)C2=O N1(C(=O)OC(C)(C)C)CCCC(N=c2[nH]c3c(c(=NCC=CBr)[nH]2)CSC3)C1 CC(C)C(O)C(C)C(=O)N1CCN(C(c2cnc(O)n(C)c2=O)=O)CC1CO C1(C(N(C(C)CNC(=O)Cn2c(C)csc2=O)CC)=O)COC(C)(C)CO1 Cc1sc(C(N2CCN(C(c3cc[nH]c3)=O)C(C(F)F)C2)=O)cc1[N+](=O)[O-] C1(NC(=O)C=CBr)CCCN(CCCNC(=O)CNC(c2ccc(F)cc2)=O)C1 N1(C(c2n(CCC)ncc2)=O)CC2CC1CC2NC(c1cc[nH]c1)=O C1(CC)CN(C(c2cc(C#N)c[nH]2)=O)CCC1NC(=O)CC1CC(O)C1(C)C c1(CC(=O)NC2CN(C(=O)CN3CCCNC3=O)CC2C(F)F)cccc(Cl)c1 C1(C(=O)NCC2CCN(C(=O)Cn3cc(CO)nn3)C2)Cc2cscc2C1 CCCC(C)C(=O)NC1(COC)CN(C(c2cn(CC(F)(F)F)nn2)=O)C1 N1(Cc2cnc(OC)nc2)CCC(F)(C(N2CCN(C3COC3)CC2)=O)CC1 N1(CC(C)C)CCCCC1C(=O)NCC1CC(CNC(=O)COC2CCCC2)C1 C1(NC(COc2ccn(C)n2)=O)CC(NC(C2CC(=C3CCC3)C2)=O)C12CCC2 C(N1CC(C)CC(C#N)C1)c1onc(-c2c(Br)cc(OC)c(OC)c2)n1 C(=O)(CN=c1cc[nH]cc1)NC1CC(NC(CC(C)C)=O)C(O)C1 c1(OC)cc(Cl)c(Br)cc1C(=O)NCC(CO)NC(C1(Br)CC1)=O Cc1noc(C2CC2)c1C(=O)NC1CCC1NC(=O)CC(O)CN(C)C CC1CC(=O)CCN1CC(=O)Nc1ccnn1-c1cccnc1 C1(C)(CC)C=C(C(=O)N2CC(CN(C(=O)C(C)C3(O)CCC3)C)C2)C1 N1(C(CC2CC(=C)C2)=O)CC(CN(C2CC2C(C)(C)C)C(=O)C2CC2)C2(CC2)C1 c1(OC)cc(C(N2CC(NC(=O)C(C)(C)c3cncs3)C(O)C2)=O)cc(Cl)c1O C#CCCCCCC(=O)N(CC(C)(C)C(=O)NC1(CC=C)CCOC1)C C(C1(O)CCCc2ccccc21)NC(=O)C(=O)NC12COC(CF)(C1)C2 c1(CNC(C2(NC(C3CN(C(C)=O)C3)=O)CC(F)(F)C2)=O)nccc(C)c1F CC1(C(=O)NCCOCCCNC(C2CCOCC2)=O)CCC(=O)C1 Cn1nc(C(=O)NC2(C)CCN(C(c3cscc3C#N)=O)C2)cc1C1CCCO1 N1(C(CCC#C)=O)CC(NC(c2cc(O)cnc2Cl)=O)CC12CCC2 N(C(=NCc1ccnc(C(F)(F)F)c1)NC(CC)CC)C(C#C)C(C)C C1(C(=O)NCC2N(C(C(CC)C)=O)CCCC2(C)C)CC(c2cnn(C)c2)=NO1 c1(C(=O)NC2CN(C(c3ccnc(C)n3)=O)C(C)C2)cc2ccc(Cl)c(F)c2o1 Cc1nc(Cl)nc(N2CCCC2(C)CNC(c2ccc(O)nc2)=O)c1Cl C(=O)(CCCCCN=[N+]=[N-])NC(CC(C)C)CNC(c1cc2n(n1)CCO2)=O c1(CNC(CCSCCC)=O)cc(O)nc(CNC(=O)CCc2ccnn2C)n1 C(=O)(C1=Cc2cccc(OC)c2OC1)NCC12N(C(C(=O)NC)=O)CCC1CC2 C1(NC(C(COCC)C)=O)CC2CCC1C(NC(c1cc3c(ccn3C)[nH]1)=O)C2 Cc1ncnc(N2CCC(C(=O)NC(c3ccc(Cl)cc3)C3CC3)C(O)C2)c1Br C(=O)(C1CSc2ccccc21)NC(CNC(c1csc(C)c1C)=O)CO Cn1c(=N)[nH]c2cc(C(=O)NC3COC4(CCCN(C(=O)CNC=O)C4)C3)ccc12 c1(C(N2CCC3(CC(NC(c4cnn[nH]4)=O)C3)C2)=O)ccnc2ccccc12 N1(C(C(C(C)C)CO)=O)CCC2(CCCN(C(C3COC4COCC34)=O)C2)C1 C1(NC(c2nnc(C)s2)=O)CN(C(c2cnc3n2CCC3)=O)CC(C)(C)C1 C1(N(C(=O)CC23CCCC2C3)C)CCC(NC(=O)CCc2cccs2)CC1 c1(C(N2C(C)CC(NC(c3cn(C)nn3)=O)C2)=O)ccc2ccc(Br)cc2n1 N1(C(c2cccc(C)c2F)=O)CC(NC(C2CN3CCCC2C3)=O)C2(CCC2)C1 C1(CNC(c2ccc(C)cn2)=O)CCC(C)CN1C(=O)C(=O)NCC(F)(F)F C(=O)(C(C)(O)C(C)(C)C)N1CC(COC)N(C(c2ccc(F)c(SC)c2)=O)CC1 CCC(C)(C)C(O)C(=O)N1CCN(C(=O)C=C2CCC2)CC1C1CC1 CCCC(C)CC(=O)N1CCC(F)(CNC(c2ccc(COC)[nH]2)=O)C1 c1(C(=O)NC2CN(C(Cc3cc(C)nn3C)=O)CC2C)nccc(N)c1Cl N1(CC(=O)N(CC)CC)CCC(c2ccc(NC(C3(C)CC(C)=NO3)=O)s2)CC1 N1(C(C2(C)CC(C)(C)C2)=O)C2CCC1CC(NC(c1cc(Cl)cc(F)c1F)=O)C2 Cc1noc(C)c1S(=O)(=O)N1CCC(O)(C(N2CCC(C#N)C2)=O)C1 C(=O)(C#CC1(C)CCCO1)NC(C(=O)NCCC1CCC(C)C1)Cc1cn[nH]c1 CC1CCC(C)(C)CN1C(=O)NC(c1ccc(F)cc1Br)c1ccsc1 c1(C(N(CCNC(CC2CC(=C)C2)=O)C(C)C)=O)cc(F)c(Cl)c([N+](=O)[O-])c1 N1(C(C=CC(=O)OC)=O)CCN(N2CC(OC(=O)N(C)C)C3(CCC3)C2)CC1 N1(C(c2ncn(C)c(=O)c2)=O)CCCCCC(NC(C2CC3C=CC2O3)=O)C1 C1(C)(NC(=O)NCC(CC)(C)NC(=O)OC(C)(C)C)CN(C(C)=O)CCO1 C1(COCC#C)CCCN1C(=O)CCN(CC#C)C(C1C=CCCC1)=O N1(C(c2c(C)ccc(=N)[nH]2)=O)CCC2(CCCN2C(=O)C(C2CCCCC2)F)C1 c1(C(=O)NC2(CC=C)CCN(C(c3ccnnc3)=O)C2)cnc(Br)c(OC)c1 c1(CC)cc(C(N2CC(F)CC2CNC(C2(C)CCCCO2)=O)=O)ccc1F N=c1ncc(C(=O)NC2CCCCC2NC(c2cocc2Br)=O)c[nH]1 C(=O)(C(CNC(=O)OC(C)(C)C)CO)N(C(C)CN(C(=O)C=CCN(C)C)C)C c1(C(=O)NC2(C3N(C(CN(CCC#C)C)=O)CCC3)CC2)ccc(C(N)=O)nc1 C(=O)(CC(C)(C)C(C)=O)NC(C(=O)NCC(CC)(C)OC)C(C)OC N1(C(CCC(C(C)C)NC(C(n2ncc(C)c2)C)=O)=O)CCCC2CCCCC12 c1(CN2C(C(=O)NCc3ccccc3)CC2)cc2c3c(c1O)CCCN3CCC2 C1(NC(C2(CCC=C)CC2)=O)CCN(C(c2cnco2)=O)CC12CCC2 c1(NC(C(N2CC3CCC2C(O)C3)c2nc(C)c(Br)s2)=O)ccc2c(c1)CCC2 C1(C)(NC(C2CC(C=C(C)C)C2)=O)CCN(C(c2cccc(C(C)C)c2)=O)CC1 C1(C(=O)NCCCCCCN(C(C(C)NC(C)=O)=O)C)NC(=O)C2CCC12 C1(CNC(c2c(C)cncn2)=O)CC2(CCC2)CN1C(=O)CSC(C)C Cc1nccc(C(=O)NCCCC(C)(C)NC(=O)CN2CC3CCC2C3)c1N C1(NC(c2c(C)nccn2)=O)CC=C(C(=O)N(C)C(C)C2CC2)C1 N1(C(c2cc(OC)no2)=O)CC2CCN(C(c3ccn(C(C)C)n3)=O)C(C2)C1 C1(CNC(C)=O)CCCN(C(=O)C(C(C)(C)O)Oc2ccccc2)CC1 C(CCC=C(C)C)(C(=O)NC1CCC(F)(F)CC1)N(CCSC)CC N1(C(CS(CC)(=O)=O)=O)CCN(C(=O)Cc2ccc(C)cc2Cl)C(C)CC1C CC1(C)C2CC(C(N3CCCC3c3cn(CCF)nn3)=O)CC12 c1(C(=O)NCC23C(CN(C(CCc4c(C)ncs4)=O)C2)C3)cnc(N)c(Cl)c1 C(=O)(CCCCCN(C)C)N(CC(=O)NC1CCCS1)CC#C C(=O)(C1=NOC2COCC12)NC(CC(C)NC(c1ccc(C(=O)OC)o1)=O)C c1(COc2c(CNC(C(CC)C)c3ccco3)cccc2)cccc([N+](=O)[O-])c1 C1(CC)(NC(=O)CC2CC=CC2)CCCN(C(C2(SC)CC2)=O)C1 CC(C)(C)CC(O)C(=O)NC1CN(C(c2sccc2-n2cnnn2)=O)CC1O C1(NC(=O)C(F)=CC2CC2)CC(O)CN(C(=O)C(C2CCCCCCC2)O)C1 c1(OC)cncc(C(=O)NC(C)C(C)NC(=O)CCCn2cncn2)n1 Nc1c(C(N2CCCC(NC(C3(C(F)F)CCCO3)=O)CC2)=O)cc(F)cc1F Cc1noc(N)c1C(=O)NCCCCCN(C)C(C1CCC1n1ccnc1)=O c1(N(C)CC2CCCN2)cnc(C#N)cn1.c1(C=O)cnc(CC2CC2)s1 Cc1ccc2cc(C(N3CC4CC3CN4C(C3(O)CC(C)(C)C3)=O)=O)[nH]c2c1 C1(OC(CN(CC(C)=O)C(=O)COC(C)C)=O)CCOCC1 c1(C(=O)NC2CCN(C(C3(CC)COC3)=O)CC2F)nc2ccc(F)cn2n1 c1(CN2CCCC(Nc3ccc(C)cn3)C2)cncc(P(C)(C)=O)c1 C(=O)(C1OCCc2ccccc21)N1C(CNC(=O)Cc2ccc(F)c(Cl)c2)CC1 N1(C(C2CC(=C)C2)=O)CCCCC1C1(NC(=O)C(C)NC(=O)NC)CC1 C(=O)(C1=CC2(CN(C(=O)CN=c3cc[nH]cc3)C2)OC1)NCC(C)(C)C1CC1 Cc1ncn(C)c(=O)c1C(N1CC2CC2(NC(=O)CC2CC3(CC3)CO2)C1)=O n1(CC(=O)N(C2CCN(C(=O)CCCc3cc[nH]n3)C2)CC)cccc(C)c1=O CC(C)CC(CNC(C1(c2cc[nH]n2)CCC1)=O)NC(=O)Cc1cscn1 c1(NC(C2(O)CCN(C(c3cc[n+]([O-])cc3)=O)C2)=O)cc([N+](=O)[O-])cc(Cl)c1O N1(C(c2cc(CC)oc2C)=O)CC2CN(C(=O)CCCc3ccccc3)CC2C1 C(=O)(CCC(C)(C)NC(=O)C=CCF)NC1(COC)CCC1 C1(C(C)C)CN(C(=O)CCC(C)C#N)CCCN1C(=O)C=CC(F)(F)F n1(CC(N2CCC3C(NC(CC4(C)CC4(Cl)Cl)=O)C32)=O)cccc(N)c1=O N=c1[nH]c(N2CCn3c(cnc3Br)C2)nc2ccc(Br)cc12 C(=O)(CN=c1ccc(C#N)c[nH]1)NCC1C(CNC(c2c(C)cc(C)nc2)=O)C1 C1(NC(c2ccc(C#C)cn2)=O)C(CNC(=O)CC2(O)CCC2)CCC12CCC2 Cc1cc(=NCCc2ccco2)[nH]c(N(C)Cc2nc[nH]n2)n1 Cc1cc(F)ncc1C(=O)NC(C)CC(C)NC(C1(CF)CCC1)=O Cc1cc(Br)cc2cc(C(=O)NCC(C)CNC(=O)CC(C)(C)C#N)[nH]c12 CC1Oc2ccc(C(N3CCCC3CN3CCN(C4CC4)CC3)=O)cc2NC1=O c1(C(C(=O)NC2(CCNC(C(CC)NC(N)=O)=O)CC2)C)ccc(F)c(F)c1 N1(C(C2CCN(Cc3cc(Br)co3)C2)=O)CCCc2ccccc2C1 c1(NC(C2N(Cc3cc(C#N)c(Cl)cc3)CC(F)C2)=O)cccc2c(I)n[nH]c12 N1(C(=O)Nc2c(-c3n(CC)ncn3)cccc2)CCC2(CC1)CNC(=O)NC2 c1(CCCC(N2CCC(C(C)(C)NC(CCCC#N)=O)C2)=O)c(F)cccc1F N1(C(CCn2c(C)nc(C)n2)=O)CC(F)(F)CC1CNC(C1(Cl)CC1(F)F)=O c1(CCC(=O)NC(C2CCCN(C(COC)=O)C2)C)cc(OC)ccc1OC C1(CNC(C2(SC)CN(C(C3CC(=C4CCC4)C3)=O)C2)=O)CCCCN1C C1(CC(=O)N(CC(F)(F)F)CC)CN(CC2CCC(O)CC2)CCO1 c1(C(N(CCN(C(Cc2cc(OC)no2)=O)C)C)=O)cc2c(C)noc2cc1C C(=O)(C(CC(=O)OC(C)(C)C)N(C)CCNC(C)=O)NC(CCNCCNC)=O S(=O)(=O)(c1c[nH]ccc1=NC(CO)c1cccc(Cl)c1)NCCc1ccc(C)s1 c1(C(C#C)NC(=O)C(c2ccccc2)OC2CCCC2)ccccc1O c1(C(N(CC(C)NC(=O)CN2CCS(=O)CC2)CC)=O)cccc(Cl)c1Cl C1(NC(C(C(C)(C)C)O)=O)C2COCC1CC(NC(=O)C#CC1CCOCC1)C2 CN1CC(C)(C(=O)NCCCC2CN(C(C3(CO)CC3)=O)CCO2)CC1=O C1(N(C(=O)CCc2ccsc2)CC)CCN(C(c2cc(C(N)=O)c[nH]2)=O)CC1 Cc1cccc(OCC(C)NC(C)C)c1.c1(C(=O)NC)ccc(-c2nnc(S)o2)cc1 c1(C(N(CCNC(c2ccc(C)c(C)c2)=O)C)=O)ccc(N)c(C)c1C N1(C(Cc2scc(C)c2)=O)CCC(C2(NC(=O)CCn3cc(Cl)cn3)CC2)C1 C1(CNC(C(CSC)(C)C)=O)(NC(c2ccc(CO)o2)=O)CC2CCC1CC2 c1(C(N2CC(C)C(NC(=O)CC3CCCCCC3)CC2)=O)nccc2n[nH]cc12 C1(C(N(C2CCN(C(c3sc(O)nc3C)=O)CC2)CC#C)=O)CCC(N=[N+]=[N-])C1 C(=O)(C1=NOC(C)C1)NCCN1CCN(C(c2c(C)sc(O)n2)=O)CC1 N1(C(C(c2nc(C)sc2)=O)=O)CCCC(CCNC(c2cnoc2C2CC2)=O)C1 C1(O)(c2cn(CCOCC)nn2)CCN(C(C2(C)CCCC2(F)F)=O)CC1 N1(C(COC(C)C)=O)CCN(C(c2ccc(C(C)(C)C)o2)=O)C(C2CC2)C1 C1(C(NOCCC)=O)CC(C)CCN1C(C1CC=C(C)CC1)=O C1(C(=O)NCC2CC(NC(c3ncn(C(C)(C)C)n3)=O)C2)CCC2C(C1)C2(F)F C(=O)(C#CC1(CC)COC1)NC(CNC(COCCCOC)=O)CC C(=O)(CC(C)(C)NC(=O)C(CC1CCC1)OC)NC(COC)(C)C N1(C(Cc2scc(C)c2)=O)CCC2(CCN(c3nncs3)C2)C1 N1(C(c2nccc(SC)n2)=O)CC2CC(Nc3cc(O)nc(O)n3)CC1C2 c1(C(=O)NC2C(CNC(c3cn(CCCC)nn3)=O)C2)cc(F)ncc1OC N1(C(c2c(C)nc[nH]2)=O)CC(CNC(=O)CC2CN(C)C2)C(C)(C)C1 C(C(=O)N(C(CNC(=O)CCCCC1CC1)C1CC1)C)(C(C)C)SC Oc1ccnc(C2CCN(c3nccc(-c4cccnc4)n3)CC2)n1 C1(NC(CCCSC)=O)CCN(C(c2cnc(Cl)cc2Cl)=O)CCC1CO C1(C(=O)NCCCc2c(C)n[nH]c2)CN(C(=O)CCCC2CC2)CC12CC2 c1(CC)cccc(NC(=O)C(CNC(=O)Cc2cc(C)[nH]n2)OC)c1O C1(C(N2C(C3CCN(C(C4COC(C)(C)O4)=O)C3)CCC2)=O)Cc2cscc2C1 O=C(O)C(n1ccccc1=O)c1ccc(Br)cc1 N1(C(C(CC)(C)C)=O)CCN(C2CCNC2=O)C(C)C1 O=C1CC(C(N2CCCC2CNC(c2cccnc2C(F)F)=O)=O)CCN1 N1(C(CCOCC)=O)CC2CC(C)N(C(c3cncc4nc(C)[nH]c34)=O)C2C1 c1(NC(CNC(=O)CC2(O)CCCCCC2)=O)cccc2[nH]nc(O)c12 Cc1cnc(CC(=O)N(C2CCCCC2)CCNC(=O)C=C2CCC(C)C2)o1 c1(C(N2CCC(NC(CCc3c(C)ncs3)=O)(CF)C2)=O)c(C#N)cnn1C Oc1c(CC2CN(c3ncc(Br)cn3)CC23CC3)cccc1F c1(C(=O)NC2(CNC(c3occc3Cl)=O)CC2)ccnnc1O Cc1cc(C(N2CCC(NC(c3ccc(O)nn3)=O)C23CC3)=O)c(O)nn1 CN=c1[nH]c(C(N2CC(N(C(=O)CCCNC(C)=O)C)C(F)C2)=O)cs1 C1(C)(C(N(CC(CN(C(=O)Cc2cc[nH]n2)C)O)C)=O)CCC(F)(F)C1 c1(C(N(C)CC2(O)CCCN(C(C(COC)OC)=O)C2)=O)ccn2ccnc2c1 c1(CC(=O)NCCC(C)NC(C2CCO2)=O)c(F)cccc1F C1(C(N(CCN(C(=O)C(C)(C)c2cc[nH]n2)C(C)C)C)=O)CCCCO1 c1(C(=O)NCC(CNC(C(CCC)OCC)=O)(C)OC)c[nH]c(=N)c2[nH]ccc12 c1(CCNCC(=O)NNC(N2CC(=O)N3CCCC3C2)=O)ccc([N+](=O)[O-])c(O)c1.CS N1(C(C2CC=C(C)CC2)=O)CCN(C(=O)CC2C=CCC2)CC1C(C)C CC(C)(C)C(CO)C(=O)NC1C=CC(C(N2CC3OCC(CO)C3C2)=O)C1 CN1CCN(C)C(C(=O)NCC2CCC(NC(=O)Cc3ccsn3)C2)C1 C1(C(=O)NCCCCNC(C(CC)O)=O)CC12CC(NC)C2 c1(C(=O)NC2CC(C)(NC(c3ccnnc3)=O)C2)cc(=O)c2cc(F)ccc2o1 c1(CNC(C(C)N(C(C)=O)C)=O)cc(C(=O)NC(C)(CO)C2CC2)n(C)n1 c1(C(=O)NC2(C(N(C(C(=O)OC)C)C3CC3)=O)CC2)ccncn1 c1(OCC)ccc([N+](=O)[O-])c(C(=O)NCC23CCC(CN(C(C)=O)C2)C3)c1 c1(C(=O)OC(C2CC2NC(=O)OC(C)(C)C)C)cc(S(=O)(=O)N(C)C)c(C)o1 C(=O)(C1SCc2cccnc21)N1CCC(NC(=O)Cc2cnccn2)C(O)C1 N1(C(CC2CC(CC)C2)=O)CC2CCC1CC2NC(c1cnn[nH]1)=O C(=O)(C(C)(C)CCCCC)NCC1CC(NC(C2CC(=C)C2)=O)CC1O N1(C(C2(OCC)CCOCC2)=O)CC2CC(C1)N(c1cc(C)nc(SC)n1)C2 N1(C(C)=O)CC2(C1)CN(C(C1C=CC(CC(=O)NC3(CN(C)C)CCC3)C1)=O)C2 c1(C(=O)NC2(CO)CCN(C(C34CCCC3C4)=O)C2)ncnc(O)c1Br CC1CC(C(=O)N2CCC(NC(c3c(C(F)(F)F)cnn3C)=O)C2)=NO1 c1(C(=O)NCC(C2N(C(C=CC(CC)=CC)=O)CCC2)(C)C)ccc(C)c(O)n1 C(=O)(C1=C(C)CCCC1(C)C)NCC(C(C)(C)C)NC(CC(CC)(C)C)=O c1(C(=O)OC)cc(Br)ccc1NC(C1CN(C(c2ccc(SC)c(O)c2)=O)C1)=O n1(CC)nc(C)cc1C(=O)NC1CCCC(NC(C2CC(SC)C2)=O)C1 C1(C(=O)NC(C)CCNC(C2(C)CSC2)=O)CCc2cnn(C)c2C1 c1(CCC(=O)N(CC(CNC(C2C(CCOC)C2)=O)C)C)cccn1C N1(C(CCC(N2CCC(c3ncc[nH]3)C2)=O)=O)CCC2(C=CCO2)CC1 C(=O)(C(F)CCC(C)C)NCC(CCOC)NC(c1ccncc1N)=O c1(NC)ccc(F)cc1C(=O)NCCC1CCN(C(=O)C(C)CSC)C1 O(NC(=O)CCN1CCCC1)CC(=O)N(CCC)CCOC Cc1cc(C(=O)N(C)CC2(O)CCN(C(C3C4COCC34)=O)C2)n(CCO)n1 CCC(CNC(C1CNC(=O)CN1C(C1CCC(C)(C)C1)=O)=O)CC(C)C C1(CC)C(NC(C2CCCC2SC)=O)CCCN1C(=O)C(C)=C1CC1 CC12CCOC(C(N3CCC(NC(c4cccc(C(F)F)c4)=O)C3(C)C)=O)(C1)C2 N1(C(c2cc3ccc(Br)cc3o2)=O)CCC2CCN(c3ccccc3)CC2C1 c1(C(N2C(C(=O)Nc3c(C)cc(Cl)nc3)CCCC2)=O)onc2ccccc12 C(=O)(CCCC(C)(F)F)NC(CNC(COCC(=C)C)=O)C(C)C(C)C c1(-c2cn(-c3c(CC)nn(C)c3)nn2)cccc2cnccc12 C1(OC)CC2CN(C(C3C(C)(C)C3(F)F)=O)Cc3cccnc3N2C1 C(CCC)(C(=O)N1CCC(C)(NC(c2cc(OC)no2)=O)C1)=CCC C1(O)(CN(C(Cc2c(C)noc2Cl)=O)C)CCCN(C(C2C=CCC2)=O)C1 C(=O)(C(CC1CCCCC1)N(CCC#N)C1CC1)NC(C(=O)OCC)C c1(OC)ncc(C(=O)O)cc1NC1CCCNC12CC2 c1(N2C3CCC(NC(C(C(C)C)NC(C)=O)=O)C(C3)C2)ccc([N+](=O)[O-])c(O)n1 CC(C)C(F)C(=O)N(C)CC1(C)CCCC1NC(=O)CSc1ccc(O)cc1 C(c1ccnn1C)=CC(=O)NC(C1CCOC1)CNC(CCc1scc(C)n1)=O N1(C(c2c(C)c(F)cnc2)=O)CC(C)N(C(=O)C(C)C(C)C)C(C)C1 N1(C(c2c(C)nn[nH]2)=O)CCC2CCCC12CNC(c1cn(C)c(C)cc1=O)=O c1(C(=O)NC(CC)CNC(=O)C(C)CO)cc([N+](=O)[O-])ccc1SC1CCCC1 C[S+](C)CCC(O)C(=O)N1CCC(Cn2cc(-c3ccccc3C(=O)O)nn2)C1 N1(C(C2CC(CNC(CC(C)O)=O)OC2)=O)CC(CO)CC(C)(C)C1 C1(F)(CNC(c2c(CC)n(CC)nn2)=O)CCN(C(=O)C(F)=CC2CC2)CC1 N1(C(c2cn(CC)nn2)C)CC2CC3CC2C1C3.C1(CCC(=O)N)CCCOC1 N1(C(c2nc(OCC)oc2)=O)CCN(C(C2CC=CCO2)=O)CC1C1CC1 CC1CN(C(=O)CCN2CCN(C)CC2)CCC1NC(=O)C(C1CC1)C1CC1 C(C)(CO)(C(=O)NC1(c2cccs2)CC1)NC(C(C)c1cc[nH]n1)=O N1(C(=O)CCF)CC2CC(C1)N(C(=O)C(Cc1ccccc1)n1cnnn1)C2 N1(CCC(=O)NC(C(C)NC(c2cn(C)c(O)n2)=O)C)CCc2ccccc2C1 C1(NC(CC(CNC(CCCCSC)=O)O)=O)C(O)C2CCCC12 C(=O)(CCC(=O)NC1CC(NC(=O)CC(O)C2CCCC2)CC1O)OC(C)(C)C N1(C(C(CSC)O)=O)CCC2(CC1)CC2(CO)CNC(c1c(C)nsc1C)=O c1(CC(=O)NCCCC(C)NC(CC2ON=C(C)C2)=O)cccc(F)c1O c1(OC)c(C)csc1C(=O)NCC#CCNC(=O)Cc1cc[nH]c1 C1(NC(CC2C(C)CCC2)=O)CN(C(=O)CNC(=O)NC2CC2)CCC1(C)C c1(C(=O)NC)n[nH]c2c1CN(C(c1c(F)cc(Cl)cc1Cl)=O)C2 C1(CC(=O)NCC(C)CNC(C2CC(N(C)C)C2)=O)CCC2(CCC2)O1 c1(C(=O)NC2CCCN(C(CC3OCC(C)(C)OC3)=O)C2)ccnc2c1CCO2 c1(CN(C)Cc2cccc(C)c2)cc(Cl)c(Cl)n1C c1(NC(c2cnc3cccnn23)c2n(C)nnn2)cnn2c1OCC(C)(C)C2 Cn1cc(NC(=O)CC2CC(NC34CC(C3)C4)C2)c(OCCN(C)C)n1 C(CN=c1[nH]c2ccc(O)cc2s1)Oc1c(C(=O)Nc2cccc(=S)n2O)cccc1 N1(C(c2cn(CC)nc2)C(=O)NCC2CC2)CCC(C)C2(CCC2)C1 c1(C(CNC(C(C)SCCCC)=O)NC(=O)CCOC)ccccc1F C(=O)(C(C)(C)C1=CCN(C(C2CC2C(F)F)=O)C1)NCc1c(C)cn(C)n1 C1(NC(C2CC(C(C)C)C2)=O)C2CC(NC(=O)C(F)(F)CO)CC12 C1(NC(c2nc(CC)oc2)=O)CCN(C(c2cnc(C3CC3)s2)=O)C(C2CC2)C1 C1(NC(C2(CC#C)CC2)=O)CC(CNC(c2cnsc2)=O)C1 c1(C(=O)NCC2(O)CCN(C(c3cc(C)c(C#N)[nH]3)=O)C2)ncnc2ccsc12 C1(C)(CC)CN(C(C2CC(N(C)C(c3cncs3)=O)C2)=O)CCO1 C(=O)(CC1C(=O)N(C)c2ccccc21)N(CCNC(C1OCCOC1C)=O)CC C1(C(=O)NC2(C(=O)NCC3CC(N(C)C)C3)C(C)C2)CN(C)CCN1C Cc1cc2[nH]c(C(=O)NCC(C)(C)CN(C(=O)C(C)N3CC(C)C3)C)cc2o1 c1(C(=O)NCC2(C)CCC(NC(c3c(C)cccc3)=O)C2)cncc(C#N)c1 c1(CN(C(C2(OCC)CCS(=O)(=O)C2)=O)C)cnn2c1CN(c1nncs1)CC2 c1(CC)cccc(CC)c1CC(N1CCN(C(=O)C2=NNC(=O)C2)CC1)=O C1(OC)CN(C(c2cnc(CO)nc2C)=O)C(C)(CNC(c2ccc(C)s2)=O)C1 c1(C(c2n(CCCCCC)nnn2)NCc2cnoc2)c(C)nn(C(F)F)c1C N1(C(C(C)N(CCOCC)C2CC2)=O)CCC(C(C)(C)O)CC1.C1(C)C(=O)N1 c1(C(=O)NCC2(O)CN(C(CC(C)C)=O)C2)cc(Cl)nnc1Cl c1(N2CCC(C)(CC)C2)ccncc1S(=O)(=O)N1CCOC(C(C)(C)C)CC1 c1(N(C2(CNCc3cccc(C#N)n3)COC2)CCC)ccc(F)c(Cl)c1F c1(OCC(N2CCC(CCNC(COCCCC)=O)C2)=O)ccc(OC)cc1 N1(C(CSCC=C)=O)CC(C(=O)NC(CC)C(=O)NC(C)C)(CC)C1 c1(NC(=O)Nc2ccc(C)s2)ccc(CC(=O)NCCC2CCOC2C)cc1 N1(C(C2CC(C)N2C(c2cc(Cl)cn2C)=O)=O)CCOC2CCCC12 c1(C(=O)NC2CN(C(CC3(C=C)CCC3)=O)C(C)C2)[nH]cc2c1CCS2(=O)=O N1(C(c2ccc(COC)o2)=O)CCOC(CCNC(c2cc(SC)c(C)o2)=O)C1 Cc1cc(F)ccc1N(C)C(=O)N(C1CC1)CC1(c2ccc(Br)cc2)CCCC1 C1(OCC)COCCC1CC(=O)NCCN(c1coc(C2CCCC2)n1)CC C1(C(=O)NC2(CNC(=O)CSc3nncs3)CC2)CC12CCCCC2 CC1CCN(C(C2CC(O)CCN2C(c2cnnc(O)c2)=O)=O)C1(C)C C1(CNC(c2c(C)nc(CCC)s2)=O)CN(C(C2CCCCO2)=O)CCN1C c1(OC)ccc(N)c(C(=O)NCC2(NC(c3cscc3Cl)=O)CCC2)c1 c1(C(C)(F)F)cccc(C(=O)NC2CCCC(NC(=O)CC3OCCCO3)C2)n1 N1(C(CCCC(=O)NCCC)=O)CCC(C2(NC(c3nnc(C)s3)=O)CC2)C1 Cc1cc(=NC(CC2CC2)C2CC2)[nH]nc1N1CCc2c(O)ncnc2C1 C1(C)(C(=O)OC)CCCCC1C.C(CC(N)=O)N1C(=O)C=CC1C c1(OCC(=O)NCC(C)CNC(=O)CC2(C(F)F)CC2)ccc(Br)cc1 CC1(C)CN(C(=O)C(c2ccc(F)cc2F)=O)CCC1NC(=O)C1=NOCC1 N1(C(=O)CNc2ccccn2)CCOC(CCNC(C2CC(CF)C2)=O)C1 C1(NC(=O)C(C2CCCO2)C2CC2)CC2CN(C(=O)C=C3CCCCC3)CC12 c1(CC(C)CO)ccc(-c2nn[nH]n2)cc1.C1(N2CC2)CCCC(CC(F)(F)F)C1 c1(C(N(CCC(=O)NC2CCC2C)CC=C)=O)cn(C)c(C)n1 C(=O)(C#CC1CCCO1)NC1CCCCN(C(Cn2ncc(CC)c2)=O)C1 N1(C(C=CCC2(NC(=O)CC3C=CCC3)CC2)=O)CCC(F)(F)C(F)C1 CN1C(=O)CCC1C(=O)NCC(C1CCCN1c1nc(C(F)(F)F)ns1)(C)C C1(CC(=O)NCCN(C(c2cncc(CSCC)n2)=O)CC)CCOC(C)(C)C1 N1(C(CNC=O)=O)CC2(CC(CNC(c3ccc(F)c(C(=O)O)c3)=O)C2)C1 C1(C(=O)NC2CC(C(C)(C)O)C2)CC2(CCN1C(c1cncc(Cl)c1)=O)CC2 c1(C(=O)OCc2cccc(SCC)c2)ccc(Cl)c(Br)c1 c1(CNC(=O)C(=O)NCc2scc(NC(C3CCC(F)C3)=O)n2)ccc(F)cc1 c1(C(N(C2CN(C(=O)CNC(=O)C(F)(F)F)C2)C)=O)cn(-c2ccccc2)[nH]c1=N N1(C(c2ccc(OC)cc2O)=O)CCC2(CC1)CC2CNC(C1CC1C(C)C)=O C(=O)(CCCCC(C)(C)OC)N1CCCC(O)(CCNC(C(CC)C)=O)C1 c1(C(C)C)ccc(C(=O)NCC23CC2CN(C(=O)CC(C)n2cccn2)C3)cn1 CC(C)C(C(C)NC(c1cccc(N2CC=CC2)c1)=O)NC(=O)COC(F)F N1(C(C(C=C)(F)F)=O)CCN(C(c2nnn(CO)c2N)=O)C(COC)C1 c1(OC)cc(C(N2CCC(C)(NC(c3ccccc3F)=O)CC2)=O)cc(F)n1 O=C(C1=NOC(C(C)(C)C)C1)N1C(CNC(c2ncoc2C2CCCO2)=O)CC1 c1(C(=O)NC2CN(C(=O)CCN3CCCCC3=O)C2)cc(F)cc2nccnc12 c1(C(N2CCC(NC(C=C(C)C3CC3)=O)C2)=O)ccncc1-n1cccn1 c1(C(C)CC(N2CC3CC2C3NC(C2CCN(C)C2)=O)=O)ccc(F)cc1F C1(C(=O)NC2(C(=O)NCCc3cccnc3F)CCC2)Cc2nccn2C1 n1(C(C(=O)NCCN(CCOC)C(C2(CF)CCC2)=O)C)cc(C)cn1 C1(CNC(CCCCOC)=O)(NC(=O)C(C)c2cccs2)CC2CCC1CC2 CC1CC(C(=O)NC(C)CCCNC(=O)CCOCC(F)(F)F)Cc2nn[nH]c21 C(C1=CCCN(C)C1)NC(C1(CNC(C(CSC)OC)=O)CCC1)=O N1(C(c2ncc(C)cc2F)=O)CC(C(N2CCCC2C(C)(C)C)=O)CCC1(C)C CCCCC(CNC(c1csc(COC)n1)=O)NC(c1ccccc1Cl)=O N1(C(C2CC(C#C)(O)C2)=O)CC(NC(=O)C=Cc2cnn(C)c2)CCC1C CC1(C)CNCCN1C(=O)C(=O)Nc1ccccc1N1CCNC1=O N1(C(c2c(OC)c(C)sc2)=O)CC2CCN(C(=O)C(c3cnn(C)c3)O)CC2C1 N1(C(C=C(CC)C)=O)CC(CNC(=O)COc2ccc(Cl)cc2F)C2(CC2)C1 S(=O)(=O)(c1cc(C)cnc1NCC(C)(C)C(=O)NC)NCC(CC)(C)CO N1(C(C(CCC)CNC(=O)C(F)C(C)C)=O)CC(C)c2ccccc21 c1(C(=O)NC2CC(F)(CNC(C3C(CC)OCC3)=O)C2)cc(OC)ncc1F c1(C(N2C(CN(C(C3CC3(C)C)=O)CC)CCCC2)=O)cc2cc(Cl)ccc2o1 C1(c2n(Cc3c(SC)cccc3)ccn2)C(O)C(O)CN1N1CCC(OC)C1 CC(C)(C)C#CC(=O)NCC1(F)CCN(C(=O)CSc2ccccc2)C1 N1(C(C(C)OCCC#C)=O)CCCC(n2cc(CNC(=O)CCC3CC3)nn2)C1 n1(CC(=O)NC(C(C)NC(=O)CC2CCCCN2C)CO)ccc(=O)n(C)c1=O N(C1CSCc2ccccc21)C(CC(C)(C)C)c1ccc(Cl)cc1.C1CC(=O)N1 C1(NC(C(n2cc(Cl)cn2)C)=O)CCN(C(=O)C#CC2(C(F)(F)F)CC2)CC1C c1(C(N(C(C)C)CCN(C)C(c2ccc(N)cn2)=O)=O)c[nH]cc(Br)c1=O C12(C(=O)NC(CCNC(c3cc(COC)cn3C)=O)(C)C)CC(C)(C1)OC2C c1(NC2CCCCN(C(C(C=C)(C)O)=O)C2)ncc(S(C)(=O)=O)cc1Cl N1(C(C2C(C(=O)OC)C2)=O)CCN(C(C23CCC(CO)(CC2)C3)=O)CC1C1CC1 C1(C)(CNC(Cc2n(C)nnc2)=O)CN(C(c2ccc(Cl)s2)=O)C(C)(C)C1 C1(C(=O)NC(CN(C(c2cnsn2)=O)CC)C)CCCN(c2cnccn2)C1 C1(C(=O)OCC)Cc2cccc(NC(=O)N(CC(C)C)CCOC)c2C1 Brc1ccc2nc(CN3CCN4CCCCC4C3)cn2c1 C1(NC(C)=O)CN(C(=O)Cc2c(F)cccc2C#N)CC(C)(C)C1 c1(C(=O)NC(C)CN(C(=O)CCn2cnccc2=O)C)cc2c(s1)CCCC2 Cc1c(NC(=O)C(C)(C2CC2)N(C)C(C2CCOC2(C)C)=O)cccc1C#N c1(C(C(=O)NCC2CCCN2C(C2COC2)=O)O)ccc(Cl)cc1 c1(C(=O)NCC#CCNC(CC(=C)Br)=O)c(C)noc1C(F)F c1(OC(C2(OC)CCN(C(=O)OC(C)(C)C)CC2)=O)cnc2n1C(C)CCC2 C1(NC(=O)CC2CC=CC2)CN(C(C2CCOC2)=O)C2(CCOCC2)C1 CC1(C)CC(=O)NCC1C(N1CCN(C(=O)C=C2CCOCC2)CC1C(F)F)=O c1(C(C)(C)C)ccc(C(=O)NC2CCC2NC(c2ccccc2)=O)[nH]1 c1(C(N(C2CC(NC(C(C(C)O)NC(N)=O)=O)C2)C)=O)ccc2cnccc2c1 CC1CC=C(C(=O)N2CC(C(=O)NC3CC(CCC(N)=O)C3)C(F)C2)CC1 c1(SCC)ccc(CC(N2CCC(CNC(=O)CCn3cc(C)cn3)C2)=O)cc1 N1(c2ccnc(C)n2)CCN(C2CCCN(C(c3cnoc3C)=O)C2)C(=O)C1 N1(C(C(c2ccc(N(C)C)cc2)C)=O)CCCN(C(=O)C(N)=O)CCC1 N1(C(CC)=O)C(CNC(=O)C(F)(F)c2ccncc2)CC2CCCCC12 C(CC(N=c1[nH]c(Cl)nc2ccccc12)C(C)C)N(C(c1c(C)nc[nH]1)=O)C Cc1cc(CCNC(=O)C(CO)NC(C2CCNC2=O)=O)nn1C C1(CC)CCCC1(C)C(N1CC(C(C)NC(c2cnc(C(F)(F)F)nc2)=O)C1)=O C#CC1(C(=O)N(CC(C)C(=O)NCC2(CC)CCOC2)C)CCCC1 C1(NC(c2n(CCCC)ncc2)=O)CC(CNC(c2ccc(CC)o2)=O)C(O)C1 c1(C(=O)NCC=CCNC(Cc2nc(C)sc2C)=O)ccnc(O)c1Br C(=O)(N=c1nc(-c2cccc(CO)c2)[nH][nH]1)NC(c1cccc(C(=O)OC)c1)=O C1(NC(C=Cc2nc(C)sc2)=O)CCC12CCN(C(C1CC1(C)C)=O)CC2 C1(C(=O)NCC2(CNC(C3CCC(NC(C)=O)C3)=O)CC2)NC(=O)CC1C C1(C(N(CCN(C(C(C)=CC)=O)C)C)=O)CCN(C2CCS(=O)(=O)C2)CC1 c1(C(N2CCC(C)(NC(c3cc(Br)no3)=O)C2)=O)ccc(C2CC2)c(F)c1 N1(C(C(C)(C)OCC)=O)C2CCC1CN(C(c1oc(C)nc1CC)=O)C2 CC1(C)COCC(C(=O)NC2(C3CCCN3c3snc(Cl)c3C#N)CC2)O1 c1(-c2cccc(NC(=O)NC3CS(=O)(=O)NC3=O)c2)coc2ccc(Cl)cc12 C=CCCC(CC(C)C)C(=O)NC1(CNC(c2cscc2OC)=O)CC(F)(F)C1 c1(NC(C2(F)CN(C(C3CC(=O)N(C4CC4)C3)=O)C2)=O)ccnc(OC(F)F)c1 C1(C(=O)NCCN(C(c2c(C)noc2C(F)F)=O)C)CCCC2(CCOCC2)O1 Cc1ccc(Cl)c(OC(C)C(=O)NC(C)CNC(c2csc(S)n2)=O)c1 C=CC1CCN(C(=O)C(C2CCCOC2)NC(=O)NCC)CC1 N1(CC(=O)NCC2N(C(C(C)=CC3CC3)=O)CC=C2)CCCCC(O)C1=O Cc1c(C(N2CCC(NC(=O)CC3CCCC3)C3CC23)=O)cncc1Br C1(C(N2CCC(C3COC(=O)N3)CC2)C(=O)NC(C)C)CC2OC(C)(C)OC2C1 c1(C(=O)OC)cnn2c1CN(C(=O)NC1CN(c3ccc(O)cc3Cl)C1)CC2 c1(C(=O)NC2C(C(F)(F)F)CCN(C(C)=O)C2)[nH]nc2c1CCCC2(C)C c1(CC(=O)NCC(CC)(C)NC(=O)C(F)C(F)(F)F)ccc(C)cc1C CN1CCN(C(c2ccc(F)s2)=O)C(C(=O)NCCN2CCC(C)(C)CC2)C1 Cc1coc(C=CC(=O)NCC(O)CCNC(=O)CCCc2csc(=N)[nH]2)n1 C1(NC(C2C(C)(CC)C2)=O)(CF)CCN(C(c2ncccc2COC)=O)C1 c1(C2(C(=O)NCC3N(C(c4cn(CC=C)nn4)=O)CC3)CCC2)ccc(Cl)nc1 CCCCCC(C(=O)NCC1CCOCC1)N(CC)Cc1ccsc1 N1(C(C(C)CN(C)C)=O)CC(C(=O)NC2CC=CCC2)CC12CCC2 N1(C(C(CCC)CC)=O)CCC2(CC(C(=O)NCC(CO)N(C)C)C2)C1 Cc1cccc2cc(C(=O)NC34CC(NC(=O)C(=O)N(C)C)(C3)C4)oc12 C1(CNC(C(CC)Oc2ccccc2Cl)=O)(CO)CCCN(C(=O)CC(C)C)C1 S(=O)(=O)(c1ccccc1Br)Nc1c(C(=O)NC(C(=O)OC)C(C)O)csc1 Cc1nn(C)nc1C(=O)NC1(CF)CCN(C(c2sccc2Cl)=O)C1 C12(CNC(=O)C=CC=C(Cl)Cl)CN(C(=O)CC3CCCOC3)CC(F)(C1)C2 N1(C(c2cc(OC)ns2)=O)CCC(CF)(NC(=O)COC2CCN(C)CC2)C1 N1(C(C(C)O)=O)CC2CC(NC(=O)COc3ccc(F)cc3Br)CC(C2)C1 Cc1ccnc2nc(C(N3CCC(NC(=O)CN(S(C)(=O)=O)C)C3)=O)nn12 C(=O)(CC1=CCN(C)CC1)NCC(CO)NC(C1(C)N(C(=O)OC(C)(C)C)CC1)=O C1(C(N(CC(=O)NC(c2c(C)ncs2)C)CC(C)C)=O)CCCCC(=O)N1 c1(NC(c2n(C)nc(C)c2Cl)=O)cc(F)c(-n2ccnc2)cc1I S(=O)(=O)(c1cccc(=NCCC2OCCCC2(C)C)[nH]1)NCC1CCC(CC)CC1 c1(CCC(=O)NCC(CNC(C2(O)CCOC2)=O)OC)cscc1Br CCC(O)(CNC(=O)C(C)N(C(c1cnn(C)c1OC)=O)C1CC1)CC N1(C(c2ccc(COC)o2)=O)CC(NC(=O)CC2CCOCC2)C(C)C1 c1(C(N(CCCN(c2ncnc3c2COC3)C)C)=O)cc(F)cc2nccnc12 S(=O)(=O)(c1cnccc1N1CCC2(C1)OCCO2)NCCc1ncc(C)cc1C Cc1nc(SC2CCCC2)sc1CC(=O)NCCC(C)(C)NC(=O)C(CC)OC C1(NC(C2CC(C(C)=O)C2(C)C)=O)CN(C(=O)C=C2CCN(C)C2)CC1(C)C C(=O)(C(COC(C)C)NC(=O)CN(C(=O)CC(C)n1cccn1)C)OC C1(NC(COCCOCC#C)=O)CN(C(=O)CSCC(F)(F)F)CC(C(F)(F)F)O1 C(C(=O)N=c1ccn(CCO)[nH]1)(C1CC=CCC1)NC(CC1CCC(=O)CC1)=O N1(C(C2(CC)CCCO2)=O)CC2(CCCC(CNC(c3ccc(Cl)cc3)=O)O2)C1 CC(C)C(C(C)NC(=O)CO)NC(=O)CCNC(c1cc(-c2ccco2)[nH]n1)=O c1(C(N2C(C)CC(CC(N3C(C)CC(F)C3)=O)C2)=O)cccc(C#N)c1 N1(C(c2cc(CCC)[nH]n2)=O)CCN(C)C(C(=O)NC2CC=CCC2)C1 C1(NC(CC(=C)I)=O)CC12CC(NC(=O)C(O)C1CC1)C2 C1(NC(c2ccc(C)nc2)=O)CC2CN(C(c3cnc(Cl)s3)=O)CCN2C1=O c1(C(=O)NCC2CCC(NC(C(C(C)C)N(C)C)=O)C2)ccc(=O)n(O)c1 C1(NC(C2C(C(C)C)OCC2)=O)CC=CCC1C(N1CCCCC1CCO)=O C(C(C)C(C)C(=O)NCC1=CCN(C(c2cc(O)nc(OC)n2)=O)CC1)OC N1(ONS(c2c(C)sc(Br)n2)(=O)=O)CCC2(CC1)C(O)CC(C(=O)O)C2 C1(NC(C(C2CCCCCC2)C)=O)CCC(C)(NC(C23CC(C2)C3)=O)CC1 Cc1ccc(N2CC(C(=O)NCC3CCN(C)C3)CCC2=O)cc1C C(=O)(C(F)CCC(C)(C)C)NCCOCCCNC(c1cn(CCC)nc1)=O N1(C(C=C(C)Cl)=O)CC(C)(C)OCC1CNC(=O)COc1cc(F)ccc1F N1(C(C(C)CC(N)=O)=O)CC(NC(=O)C(C)N2CCCC2)CC12CCCCC2 CC1CN(C(C2(F)CCN(C)CC2)=O)CCC1CO O=C(CCCC(F)C(=O)O)N1CCCCC1c1nc(-c2cccs2)no1 c1(C(N)=O)cccc2c1CN(C(=O)CC1CCN(C(C3CCC(=O)O3)=O)CC1)C2 CCC(C)CC(C)C(=O)N1CCC(C)(C)C(c2cn(-c3cc(C)ccc3F)nn2)C1 C1(CNC(C(C)O)=O)CCC2(CN(C(c3ccc(F)cc3O)=O)C2)O1 C12(NC(C#CC3(C)CC3)=O)CCOCC1CN(C(c1ccns1)=O)C2 c1(C(=O)NCC(CNC(c2cnc(OCC)s2)=O)C)nc(O)nc(O)c1N N1(C(C(N)=O)=O)CC2(CCN(C(=O)Nc3ccc(Cl)c(NS(C)(=O)=O)c3)C2)C1 N1(C(CC2C(C)(C(F)(F)F)C2)=O)CCCC1(C)CNC(=O)CCC1CCCOC1 C1(NC(=O)Cn2nc(Cl)ccc2=O)CCOC2(C1)CC(C(=O)O)C2 c1(CC(=O)NC2(C)CC(NC(C(COC)OC)=O)C2)ccccc1CS(N)(=O)=O C1(CNC(C(C)NC(N)=O)=O)CN(C(C2CC2C2CC2C)=O)CCC12CCC2 C1(C2CCN(C(C3CCCCC3C)=O)CC2)(NC(c2cnc(C)c(N)c2)=O)CC1 c1(CC(=O)NC2(C)CC(NC(c3cn(C)c(=O)cc3)=O)C2)c[nH]c2ncccc12 C1(CC)CN(C(c2cn(C)c(C)n2)=O)CCC1NC(c1ccc(O)c(C)c1)=O c1(C(=O)NC(CNC(c2c(CC)n(C)nc2)=O)CO)ccn2c(C)ncc2c1 N1(C(c2ccc(CC(=O)OC)o2)C(=O)NCCOC)CCOC2(COC(C)(C)C2)C1 c1(C(N2CCCC(CNC(CCSC)=O)C2)=O)cc(Br)c(F)cc1N CC1(C)CN(C(=O)Cc2cncnc2)CC(C)(C)C1NC(=O)CCCCC(F)F CCC(COC)C(=O)NCC(CC(=O)NC(C)(CO)CO)C1CCC1 N1(CC(CCC)=O)CCOC2(CCSCC2)CC1 CCS(=O)(=O)NC(C)C(=O)N(CC(C)(C)NC(=O)C(C)c1ccco1)C C1(NC(c2n(CC)nc(C(C)C)c2)=O)CCCN(C(=O)C2=CCCO2)CC1 CC(C)(C)CCC(F)C(=O)N1CCCC1C1(NC(=O)CCCF)CC1 c1(CC)nn(C)c(CC)c1NC(=O)Nc1cccc(-n2ccnc2O)c1 C(C1CCOc2ccc(Br)cc21)NC(c1n[nH]c(C)c1F)=O c1(C(=O)NCC(C)(CO)NC(C2CC3CC3C2)=O)nc2n(c1Cl)CCCC2 C12(CNC(CC(C)C(F)F)=O)CN(C(C3CCOC3)=O)CC(F)(C1)C2 CC1(C)CCCN(C(C2CC=CCC2)=O)C1CNC(c1cc(C(F)(F)F)cs1)=O N1(C(C(C)CC2CC2)=O)CC2(CC(CNC(=O)Cn3cnnn3)C2)C1 C1(NC(CCCOCC)=O)CC(NC(c2cnn3c2CCC3)=O)C12CCC2 C1(N(C(C2C(=C)C2)=O)CC)CCN(C(=O)C=Cc2ncc[nH]2)CC1 N1(C(c2c(CC)cco2)=O)CCN(C(C2(CC(F)F)CCC2)=O)CC1COC CC1CC(F)(F)CN1C(C1CSCCN1C(=O)C=CC(F)F)=O Cc1cc(C(=O)NCC2CN(C(C3Cc4nccn4C3)=O)CC2O)c(C)cc1Cl c1(OC)cc(C(=O)OC2CN(C(C)=O)C2)cc([N+](=O)[O-])c1OCCF C1(C(N2CCN(C(CC3C(=O)NCCC3)=O)C(CO)C2)=O)CC2CC1CC2(F)F C1(CSC)(NC(=O)CCF)CCN(C(=O)CC(O)CNC(=O)OC(C)(C)C)CC1 c1(C(=O)NC(CCNC(CCC2C(C)C2)=O)c2cccs2)cc2cn[nH]c2cn1 CCC(C(=O)N1CCC(NC(c2sc(C3CCCC3)nc2C)=O)C1)C(C)(C)CC c1(C(=O)NC2CCCC2C(N2CCS(=O)CC2)=O)cc(O)nc(O)c1 C12(C(=O)NCC(COC)O)C(NC(=O)Cc3nonc3C)C3CC1C2C3 C(=O)(CCCCCNC(C1CC2COCC2C1)=O)N(CC(COC)(C)C)C N1(C(Cc2ccc(C#C)cc2)=O)CCN(C(=O)CSCC)C2COCC12 CC(C)(F)CCC(=O)NCC1(C(N2CCC3C(O)CC23)=O)CCCO1 CC(C)CCCCC(C(=O)O)NS(=O)(=O)c1ccc(Br)cc1NC(C1CCC1)C c1(C(=O)NCC2CN(C(CCc3onc(C)n3)=O)C2)cc(F)cnc1Cl C1(N2C(C(=O)NC(C3CC3(C)C)C)CCC2)CCN(Cc2ccsc2)CC1 C1(CC)CN(C(=O)C=Cc2cccc(CO)c2)CCC1NC(c1ccc(C)[nH]1)=O C12(C(N3CCCC(CCC#C)C3)=O)CCCC1CCN2C(C1CCCC(=O)C1)=O N1(C(C(CC)CO)=O)CC(NC(C2CCOC2CC)=O)CC12CCOCC2 C1(C)(C(N(C(C#C)C2CCC2)C)=O)C=CCN1C(C1OCCC1(C)C)=O C1(CNC(C=C=C(C)C)=O)CN(C)CCN1C(C1SC2C=CC1CC2)=O C1(NC(C2C(C(C)NC(C(C)=CC=C)=O)C2)=O)C(O)CC1O CCCCCC(=O)N1CCC(C(C)C(=O)Nc2cnn(C(C)(C)C)c2)C1 c1(C(=O)OC(c2ccc(Cl)cc2)CC)cnn2c1C(=O)N(C)CC2 C1(C(=O)NCC2(F)CC(NC(C3(C)CCCS3)=O)C2)CCC2(CCC2)CO1 C(CC(=O)NC(c1cccs1)C)N(C(=O)CN1CCCC1)CC#C C(CC(C)(C)CC(=O)NC(CCN(C)C)C(=O)N1CC(OCCF)C1)OC Cc1cnc2c(C(=O)NCC3CCC(NC(=O)CC(C)C(F)F)C3)cccn12 CC1CN(C(=O)CC2(C)CC2)CC1(C)C(=O)NCC12CC=CC(C1)OC2 C1(CC)(CC)CC(O)CN1C(=O)CC(O)CNC(=O)CCN(C)CCO Cc1cnncc1C(=O)NC1CC1NC(=O)CO C1(C(=O)NC(CNC(c2c(CC)nc(C)o2)=O)CO)CC2(CO1)CC(F)(F)C2 n1(CC(=O)NC2CN(C(C3(C)ON=C(C)C3)=O)CC(O)C2)c([N+](=O)[O-])cnc1C Cc1c(C(NC2CCCn3nccc32)=O)oc2ccc(I)cc12 c1(C(=O)NCCCCCOC)ccccc1-n1cc(-c2cccc(Br)c2)nn1 C1(C)(C(=O)NCC#CC(=O)NCCCCOC(C)C)CCCOC1 C(=O)(C(CCC1CC1)N(C)CC#N)NC1(C(=O)NCCSC)CCC1 N1(C(c2nc(OCC)sn2)=O)CCC(NC(=O)CC(C)(C)O)CC1C N1(C(C(C)=C2CCC2)=O)CCC(O)(CNC(c2cnc(-c3cnn(C)c3)s2)=O)C1 CC(F)(F)C(C)(C)CC(=O)NCC1(C)CC(F)(F)CN1C(=O)Cn1ccc(=N)[nH]1 N1(C(CC(COC)NC(=O)C(Cl)Cl)=O)CC2COCC2(C)C1 c1(C(=O)NC(C2CCN(C(COC(C)=O)=O)C2)C)cc([N+](=O)[O-])c2nsnc2c1 C(=O)(C(O)C1=CCCCC1)NC(CC=C)CNC(=O)CC c1(N(C)C(=O)OC(C)(C)C)ccc(C(=O)Nc2ccn(C3CCCC3)n2)cc1I C12(NC(CC(C)C3CC3)=O)CCC(CNC(=O)Cc3cc(C4CC4)on3)(C1)OC2 C(=O)(CC(C)CC(=O)NC(C)C(C)NC(=O)CC1CN(C(C)=O)C1)OC CCC(C)C(O)CC(=O)NCC1(O)CCCN(C(C2(COC)CC(F)(F)C2)=O)C1 S(=O)(=O)(c1ccc(NCC2(CC#N)CC2)c(C#N)c1)N1CC(C)CC(COC)C1 N1(C(C(C(CC)C)N(C)C(c2cnn(C)c2)=O)=O)CCCN(CC)C(=O)C1 Cc1cc(C(=O)NC2C3CN(C(=O)CCOC4CC4)CC23)c(C)cc1Cl C1(C2CN(C(C3CCCSC3)=O)C2)(Nc2cc(OCC)ncn2)CC1 N1(C(C2CC(CC)N(C(c3cc(C)cc(O)n3)=O)CC2)=O)CCC12CCCSC2 c1(CN2CC(C(=O)OC)OCC2C(c2c[nH]c(=NC)s2)=O)cnc2c(c1)CNC(=O)N2 C1(OC)CCCN(C(=NCCC(=O)Nc2ccncc2)NC2CCCC2)C1 CC(CC(N)=O)C(=O)N(C1CCCN(C(c2ccc(N)cc2)=O)C1)CC1CC1 c1(CC)ccc2[nH]c(C(=O)NCCN(C(C3CC(C)(C)O3)=O)CC)c(C)c2c1 C1(NC(c2cccc(C)n2)=O)CCN(C(C2CCC(C)C(C)C2)=O)CC1C CC(C(F)C(=O)NCCC(C)NC(=O)C1=CN=C2N=CNN2C1)C(F)(F)F c1(C(N(CC(N2CC(O)(C(C)NC(c3csnn3)=O)C2)=O)C)=O)ccc(Cl)cc1 c1(CCNC(CCN(C)C(C2CC2c2ccsc2)=O)=O)cc(O)ncn1 C=CCC(C(=O)N1CCC(NC(c2c(C)csc2Cl)=O)CC1C)C(C)C c1(CC(N2CCC(C(CNC(C(CC)O)=O)F)CC2)=O)ccc(O)c(C(N)=O)c1 N1(C(CCCn2cc(C(N3CCOC3=O)C)nn2)=O)CCC(C)(CC#N)C1 c1(CC)n[nH]cc1C(N1CC(C(C(=O)NCC(=O)NC)OC)C1)=O S(=O)(=O)(c1ccc(C(=O)O)c(F)c1)Nc1cccc(N(C)C)c1 c1(C(=O)NC2(C3N(C(C4C(C=C)CC4)=O)CCCC3)CC2)ccc(Cl)c(OC)c1 C(=O)(C(C(C)CC)N(C)C(C1CCCN1C(N)=O)=O)N(CCOCC=C)C c1(CN2CCC(CC(N3C(C(=O)OCC)CCCC3)=O)CC2)ccnc(Cl)c1Br N1(C(c2ccc(COC)c(N)c2)=O)CCC(C2CC2)C1CNC(c1nccs1)=O C1(CC(=O)N(CCN(C)CCO)C)CN(C(=O)Cc2ccc(F)cc2)CCO1 Cc1cc(C(=O)NCC(C2CC2)NC(=O)C(C)(F)c2ccon2)c(F)cc1N Cc1c(C(=O)NCCC(C)NC(=O)CC2C=CCC2)noc1C1CC1 c1(SC)cc(C(=O)NC(C)C(C)NC(c2ccc[nH]2)=O)ccc1N CCCC(CCC)C(=O)NCCC(C)NC(c1cc(Cl)nc(Cl)c1)=O c1(C(=O)NCC(c2cccc(OC)c2)C)cnn2c1SCC2 CCC(C(=O)NC(C)(C)CC(=O)NC(C)CCC1CCCC1)C(C)C C1(C(=O)NCCc2ncc(C)o2)N(C(=O)Cc2cnoc2)CCCC1(C)C CC1CN(C(=O)C(C)C(C)O)CC(C)N(C(=O)C=Cc2ccccn2)C1 C1(C(N2CCC(CCC#C)C2)=O)CC2C=CC1N(C(=O)CCCCOC)C2 C(C)(CC(C)NC(c1cn(-c2ccn(C)n2)cn1)=O)NC(C=C(C)C(C)C)=O C1(CC)(CNC2CCCN(C)CC2)CCCN(C(=O)OC(C)(C)C)C1 c1(C(N2CCCCC(NC(CCCC=C)=O)CC2)=O)oc2ccc(F)cc2c1C C(=O)(C1=NOC2COCC12)N1CCC(CN(c2ncnc(OC)c2OC)C)C1 c1(C(=O)NCC2C=CCN2C(=O)CCC2CC2(F)F)ccc2ccoc2c1 C1(C(=O)NCC#CCNC(c2cnc(C(=O)OC)s2)=O)Cc2nn[nH]c2C(C)C1 Cc1ccc2cc(C(=O)N(C3CCC(NC(=O)C(C(C)C)C(C)C)C3)C)[nH]c2c1 C1(C(N2CCC(C3N(C(=O)Cc4ccco4)CCC3)C2)=O)(CO)CCCCC1 C(=O)(C(=O)N=S(C)(C)=O)N1CCC(OC)(CNC(=O)C2=CC(C)(C)C2)C1 N1(C(CCCOCCC)=O)CC(CNC(c2oc(C3CC3)nc2C)=O)CC1C CC1CC2CCC(C(=O)NC3CCN(C(=O)C(C)(C)O)CC3F)CN2C1 C1(C(=O)NCC2(CN(C(c3nncc(OC)c3)=O)C)CC2)CN2CCN1CC2C c1(-c2nn(C(CC)CC)c(CSc3[nH]cnc3C)n2)ccc(N(C)C)cc1F C1(C(=O)Nc2cccc(OC)n2)CCC2(CCN(C(=O)C(C)Br)CC2)O1 Cc1cc(F)cc(C)c1C(N1CCC(CF)(NC(C2CCCCC2C)=O)C1)=O c1(OC)ccc(Cl)cc1CC(=O)NCC12CC(CN1C(C1(C)CNC(=O)C1)=O)C2 CN1CC(C)(C)CC1C(N1CCCC1C(C)(C)NC(c1cc2c[nH]nc2s1)=O)=O C1(C(N(CCCCCNC(C(Cc2c(C)nc[nH]2)O)=O)C)=O)CC12CCCC2 c1(CS(=O)(=O)N(c2csc(CO)n2)C(C2CNC2)C)ccccc1C(F)(F)F CCCCCCCNC(=O)C(CC1CCCC1)OC.C1(=O)COC(=O)CN1C c1(C(N(CC(CC)NC(=O)CNc2ncccn2)C)=O)n[nH]cc1C1CC1 C=CC1CN(C(=O)CSS(C)(=O)=O)CC1NC(c1ccccc1C1CCOC1)=O C1(NC(=NCc2c(C)cn(C)n2)NC2CCC2)CC(C2CCC2)C1 N1(C(C2(CNC(C(N3CCOCC3)C)=O)CCCC2)=O)CC2CCC(CO)(C2)C1 C1(C(N(CC(F)F)CCC)=O)CCN(C(=O)C2CC3(CCO2)CC3)O1 CC12CN(C(=O)OC(=O)C3CC3)CC(Nc3c(Cl)c(F)nc(F)c3Cl)(C1)C2 C1(C(=O)NCC=CCNC(=O)CC(c2ccccc2)c2ncc[nH]2)CC2CC1C2 CC1(C)CN(C(c2cccnc2)=O)C(CNC(c2nc(Cl)sc2Cl)=O)CO1 N1(C(c2cc(C)oc2)=O)CC2CCCC(N(C(=O)Cc3ccn(C)n3)C)C2C1 c1(CNC(C=C)Cc2ccc(F)cc2)cc2n(n1)CCCCO2 N1(C(=O)C2CC2)CCC2(CCCN2C(c2c(Cl)csc2Cl)=O)C1 c1(CC#N)c[nH]c2ccc(C(=O)NCCc3ccc(C(=O)C4CC4)cc3)cc12 C1(CNC(C(CCC)C)=O)(OC)CCN(C(c2cnc(O)cc2OC)=O)CC1 CCC(C(O)C(F)F)NC(=O)CSc1ccc(F)cc1F C1(C)(CNC(COC(C)(C)C)=O)CCN(C(=O)CCN2CCCCCC2)CC1 C1(CC(N2CC(C)(OCC)C2)=O)CN(C(C2CC2Cl)=O)CCO1 N1(CC(=O)N(CCc2ccc(OC)cc2)C)CCC2C(C1)NC(=O)N2CC(=O)O n1(CC(=O)NCC2(O)CN(C(C3C(C)CC=CC3)=O)C2)nc2c(n1)CCCC2 c1(CCC(=O)NCC2CC(NC(C(C)OCCOC)=O)C2)ccc(CC#N)cc1 C1(CC(=O)NCC(C)NC(=O)C=CBr)CC(C)OC1C C1(C2CCN(C(=O)C=Cc3cccs3)C2)(NC(C2CC3CCCCC23)=O)CC1 C1(CC)CCOCCN1C(=O)CC(C1CC1)NC(c1ccnn1C1CC1)=O c1(SCCC(=O)NC2CN(C(CCCCSC)=O)CC2O)ncnc2[nH]cnc12 N1(C(COCCC#C)=O)CCCC(N2CCN(C(=O)CCC3CC3(F)F)CC2)C1 C#Cc1cccc(C(=O)NCC2CC2NC(=O)C2=CC(C)(C)C2)c1Cl C=CC(CC)C(=O)NCC(C1CCC1)NC(c1cnn(C)c1)=O C(=O)(CCC(CF)CF)N1CCC(C(=O)NC(CCC)c2ccco2)C1C(C)C CCC(F)(F)CC(=O)N1CCCN(CCNC(=O)CCC2CCCCO2)CC1 C1(C(N(C2CN(C(=O)C=CC(=O)NCC3CC3)C2)C)=O)CCOCC1 C1(C(C(=O)OC)NC(c2conc2-c2ccccc2F)=O)CCCCC1C N1(C(c2[nH]cc(S(N)(=O)=O)c2)=O)CCC2CCC(C1)N2C(=O)CC1CCOCC1 c1(C(F)(F)F)cccc(-c2cncc(CNCC3CCC3(F)F)c2)c1 C(=O)(CC1OCCc2ccccc21)N1C(CNC(c2[nH]cc(C)c2)=O)CC2CC21 Cc1nc(CNC(C2CCCC2C(C)C)=O)oc1C(=O)NC1(CC(N)=O)CCC1 CC1CC(=O)NC(C(=O)N(CCCC(=O)NC2(C3CCCO3)CC2)C)C1 c1(C(N2CCCC(CN(C(CC=C)=O)C)C2)=O)c(C)cc(OC)cc1F C1(CNC(c2ccc(NC)cn2)=O)COC(C)(C)CN1C(c1cccnc1S)=O C1(C(=O)NCC2(OCC)CN(C(C(CC=CCC)C)=O)C2)CC2C(C1)C2(C)C c1(CC)cc(C)ccc1C(=O)NCC(CC)NC(c1cnc(Cl)c(N)c1)=O Cc1ncc(C=CC(=O)NC2CCCC2n2cc(C3CC3)nn2)s1 c1(C(=O)NCCC2CCN(C(c3ccc(C(C)C)o3)=O)C2)ccnc(C2CC2)c1 C1(CC(N2CC(F)(CC)C2)=O)CC(NC(=O)CN2CCNC2=O)C1(C)C C1(NC(c2cccnc2O)=O)CN(C(c2ncccc2Cl)=O)CC12CCC2 C1(C(=O)NC(C)Cn2cc(C)cn2)(CC)CCCN1C(=O)CCC(=O)NC C(=O)(C1=NOC(C)C1)N(CC(C)NC(c1sc(CC)c(Br)c1)=O)CC N1(C(C=C(COC)C)=O)CCOCC1CNC(c1cccc(-n2ccnc2)c1)=O c1(COCC)noc(C)c1C(=O)NC1(CNC(C2CC(C#N)(COC)C2)=O)CC1.OC c1(C(n2cc(C(C)(C)CN)nn2)C)ccc(F)c(F)c1.C(=O)(C)N(C)CCO C1(C(N2C(Cn3cc(CCC(C)=O)nn3)CCC2)=O)C2CC2C2CC12 N1(C(c2cc(COC)on2)=O)CCCC(CO)(NC(C2CCCCN2C)=O)C1 c1(C(=O)NC(C)CCCCNC(c2nocc2Cl)=O)cn2ccnc2s1 N1(C(CCCCCCSC)=O)CC2CCCC(C1)N(C(=O)Cc1cc[nH]c1)C2 c1(CCNC(C2(C)CC(NC(C(CC)n3ccnc3)=O)C2)=O)ccc(F)cc1 C=CCC(C(=O)NC1CCC(CCC(=O)NC(C)C(C)(C)C#N)C1)C(C)C C1(C(=O)NCC2CC(OC)CN2C(=O)C(=O)NC(C)C)Cc2ccccc2S1 C1(CNC(=O)C=CBr)COC(CNC(c2nc(C3CC3)cs2)=O)C1 N(C(=NCCC(F)(F)F)NC1CC1C)Cc1cccc(N(C)C)c1 C1(CCC(C)(C)NC(CC(C)n2cccc2)=O)CCCCN1C(=O)C=CCO N1(C(CCc2ncn(C)c2)=O)CCC(O)C1C(N1CC=CCC1)=O C=CCC(C)C(=O)NC(C)Cn1cc(Cc2scc(C(=O)NCC)n2)nn1 c1(C(=O)NC2CN(C(c3c(OCC)n[nH]c3)=O)CC2C)ccc(Br)c(C)c1F N1(C(CSCCC)=O)CC(CNC(c2c[nH]c(=N)cc2C)=O)C(C)(C)C1 CC1(C)CC(CC(=O)NC2CC(CCF)C2)N(C(C2CC2Cl)=O)C1 c1(C(N(C)Cc2ccc(CNC(=O)CC(C)(C)F)cc2)=O)cc2n(n1)CCO2 c1(C(N(OC)Cc2ccsc2)=O)cc(S(C)(=O)=O)ccc1OCSc1ccccc1 N1(C(CCSCCC)=O)CC(NC(c2cn(CCO)nn2)=O)C(CC)C1 N1(C(c2c(F)ccc(N)c2)=O)CC2(CCCC2NC(C2CCS2(=O)=O)=O)C1 Cc1ccnc(C(N2CCOC(CCCNC(=O)CN(C)C(N)=O)C2)=O)c1O CCC(CC(=O)NCCCOCCNC(c1cnn(C)c1Cl)=O)C1CCC1 Cc1n[nH]c(C)c1SCC(=O)NC(C)CC(C)NC(C1C2CC3C(C2)C13)=O C1(Cc2cccc(OCC)c2)CNCCC1C(N1CCC(C(N)=O)CC1)=O c1(C(N(C)CCn2ccnc2)=O)csc(CNC(=O)CC2(CSC)CC2)c1 N1(C(C)=O)CCN(S(=O)(=O)C2CC2)CC1C#N.c1(N)ccc(Cl)cc1C(F)(F)F C1(C(=O)NCC(C)Oc2ccccc2F)COCCC1c1ccccn1 CCC1=C(C(=O)N2CC=CC(NC(c3ccnc(F)c3F)=O)C2)CCCO1 C12CCC(C1)C(=O)N2.C(C)(C)(CNC(=O)CCC1CN(C(=O)OC(C)(C)C)C1)NC C1(NC(CNC(C)=O)=O)CC2CCC(C1F)N2C(C(CC(C)C)C(C)(C)C)=O CC1CN(C(c2c(CNC(=O)C=CCF)nnn2C)=O)CCC1O CC(C)(C)CC(C(=O)NCc1ccc(CO)o1)NC(C1CCSC1)=O CC1(C(=O)NCC2COCC2NC(=O)CNC(c2ccccc2)=O)CCOCC1 CCC(C)(O)CCNC(C1CCN(C(=O)C(C)N2CCCC2)C1C)=O N1(C(c2cn(C(C)C)nn2)=O)CC2(CC2)CC1CNC(C1(C2CCC2)CCC1)=O c1(C(=O)NC(C)C(CO)NC(c2ccc(F)c(N)c2)=O)cc2c(cn1)OCCO2 c1(CC(=O)NC(C2CCN(C(c3cc(F)c[nH]3)=O)C2)C)cc(Cl)ccc1O C1(OCC(=O)OCC)CCN(C(=O)C(=O)NC2(F)CCOCC2)CC1 c1(C(=O)NCC2(NC(c3cc(F)cc(N)c3F)=O)CC2)cc2c(=O)[nH]ccn2n1 CS(=O)(=O)C1CC(C(=O)NC2CN(C(c3cccnc3S)=O)CC2O)C1 c1(CC(N2CCC(N(C(=O)CNC=O)CC)C2)=O)cc(C)nn1C N1(C(CC=C=C)=O)CCC(C(=O)Nc2ccc3c[nH]nc3c2)CC1(C)C C1(N(C(C(C2CN(C(c3cncn3C)=O)C2)OC)=O)C)CCCCC1C C(C)(CC(C)NC(=O)CC1(C2CC2)CC1)NC(C=CC(C)C)=O C(c1cccnc1C)=CC(=O)NCC1C2CN(C(c3onc(CC)c3C)=O)CC21 C(c1cn(C)cn1)=CC(N1CCC(C(=O)NCCCn2c(C)ncc2)C1)=O c1(C(N2CCC(C(N(C(CC#C)C)C)=O)(CF)C2)=O)ccc(C#C)cc1C c1(NC(=O)NC2CC2C(N2CC3CCC(C2)O3)=O)cnc(C(F)(F)F)cc1Cl c1(C(=O)NCC(C)(C2CC2)NC(C(CC=C)N(C)C)=O)cc(S(N)(=O)=O)c[nH]1 N1(C(c2c(C)scc2)=O)C(C(N2CCOC(C(N)=O)C2)=O)CC2CC12 C1(NC(c2cc(SC)c(F)cc2)=O)CCC2CCN(C(=O)CC3(C)CCC3)C1C2 c1(C(NOCc2cn(CC)nn2)=O)cc(CNC(c2cc(C#N)c[nH]2)=O)ccn1 CC(C(=O)NCC(F)CO)(C1CCC1)NC(=O)Cc1ccsc1 c1(CCC)cc(C(N2CCC(CNC(=O)COCC(C)C)C2)=O)c(C)o1 N1(C(=O)COC2CCOC2)CCC2(CC1)CCN(C(=O)Cc1ccc(Cl)nc1)C2 c1(C(N2CCC3(C(C(=O)Nc4c(C)nsc4)C3)C2)=O)cc(Cl)cc([N+](=O)[O-])c1Cl C1(C(=O)NC2(CC=C)CCN(C(=O)CCC(C)(C)C)C2)CCn2nnnc2C1 c1(C(N(C(C)C(=O)NC(=O)Cc2ccco2)C2CC2)=O)ccnn1C N1(C(C(C)Sc2ccc(C#N)cc2)=O)CC2COCCC2(C(N)=O)C1 c1(OCC)cccc(OC)c1C(c1nnnn1C)NC1CC1(C)C C1(C(N(CC(O)C2CCC2)C)=O)CCCCCCN1C(=O)CCCNC(N)=O N1(NCCC(c2ccccc2)NC(=O)NC2CC(NS(C)(=O)=O)C2)CCCCC1 c1(C(N(C2C(C)CCN(C(C3C(=C)C3)=O)C2)C)=O)coc2ccc(C)cc12 N1(C(C(CCSC)OC)=O)CC2CN(C(c3n[nH]c(C)n3)=O)CCC12 N1(C(CC=CCNC(=O)C=Cc2cc[nH]n2)=O)CC2C3C=CC(O3)C2C1 N1(c2ncc(OCCOC)cn2)CC2(CCCC2NC(c2nccnc2N)=O)C1 c1(C(=O)NC)ccccc1-c1cc(C2(C(N3CCCC3CO)=O)CC2)no1 c1(C(N2C(C(=O)NCC3C(C(C)C)C3)CSC2)=O)ccc(Br)cc1 c1(O)ncccc1C(=O)NC1CC(NC(=O)C=CCCCOC)C1.c1ccsc1 C1(N(CCC)C(C2CC2C(=O)OC)=O)CCN(C(c2ccncc2F)=O)CC1 c1(C(C)C)ncc(C(N2CC(O)(CCNC(=O)CCC3CCC(=O)N3)C2)=O)o1 c1(OC)cccc(F)c1C(=O)NCC1CC(NC(=O)CCCc2nc(C)no2)C1 N1(C(c2nc(COC(C)=O)oc2)=O)CCSC(C)(C)C1.N12CCC(C1)C2 C(=O)(C(C)CC(N)=O)NC(CN(C(=O)CC(F)(F)Br)CC)C C1(NC(c2ccc[nH]2)=O)CC=C(C(=O)N2CCC2(CO)CO)C1 CC1CN(C(c2ccc(OC(F)F)cc2)=O)CC(C)N(C(C2(C3CC3)CC2)=O)C1 CC(C(=O)N(C1CCN(C(C2CCC(F)CC2)=O)CC1)CCO)C(F)F c1(NCC(C2CC(F)(F)C2)OC)ccc(S(=O)(=O)N2CCC(O)C(C)(C)C2)cn1 C#CCC(C)C(=O)N1CC2C(CN(C)C(c3ccncc3F)=O)C2C1 c1(C(=O)NC2CC(F)(CNC(c3csc(CO)n3)=O)C2)cccc(OC(F)F)n1 Cc1c(Cl)cc(C(=O)NC2CN(C(=O)C3=COCCC3)CC2C)cc1Br Cc1cc2cccc(C(=O)NCC34CC3CN(C(C3CNC(=O)C3)=O)C4)c2[nH]1 Nc1ncc(C(F)(F)F)cc1C(=O)NCCC(O)CNC(=O)C1=CCCCO1 C1(C(N(CCC(=O)N(C)Cc2c(C)cco2)C2CC2)=O)CCCC(=O)C1 NC(=O)CCCNC(=O)CC1CN(C(=O)N(CCCCl)CCO)C1 Cc1cc(CC(=O)N(CCNC(=O)COc2ccc(O)cc2)C2CC2)nn1C CC(CC(=O)NCCC1CN(C(C2(CO)CCOCC2)=O)CCO1)C(F)F c1(C(=O)NC(C2(O)CCN(C(C3CCC(C)CC3)=O)C2)C)cnc2ccsc2c1 N1(C(C(C)=CC)=O)CCC(NC(=O)Cn2nnnc2-c2ccccc2)C(CO)C1 C1(C)(CC)CC(NC(c2nnn(C)n2)=O)CN1C(c1ccc(N(C)C)cn1)=O c1(-n2c(C(CCCC)OC)nc(-c3cnn(CCO)c3)n2)ccc(F)c(C)c1 C(CCCCC(=O)N1CCCCC1CNC(c1cc(CN(C)C)on1)=O)OC c1(CNC(C2(C)COC2)=O)nocc1C(=O)NC1COC(C2CC2)C1 C(c1ccc(C(F)F)o1)=CC(N1C(CN(C(C(C)C2CC2)=O)C)CCC1)=O c1(CNC2C(C(=O)NC(C3CCOCC3)CC)C2)cccnc1Cl c1(C(N2CC3C(NC(COCCCC)=O)C3C2)=O)cc2ccc(C)cc2[nH]1 Cc1nc2n(n1)CC(C(=O)N(CCCNC(c1c(C)noc1C(C)C)=O)C)CC2 Cc1cc(C#N)sc1C(N1CC(F)(CNC(=O)C2=CCSC2)C1)=O N1(C(C(COCC)n2cc(-c3ccc(Cl)s3)nn2)=O)CC2(COC(C)C2)C1 c1(CC)c(C(N2CCC(CC(=O)NC(C)(C)CF)C2)=O)cnn1C c1(SCC)nccnc1C(=O)NCCC1CCCN(C(c2cnn(C)c2C)=O)C1 C(c1ccc(Cl)cc1)=CC(=O)NCC(C1CCC1)NC(C(C)OCCC(C)C)=O C(N=c1[nH]c(=N)[nH]c(=NCCCOC(=O)N(C)C)[nH]1)c1nn(C)c(C2(Cl)CC2)c1 C(=O)(CCCCC#N)NCC(CN(C(C(c1ccc(C(C)(C)C)cc1)C)=O)C)O Cc1ncc(CCC(=O)OCC23CC(F)C2C3)o1 C(=O)(C(F)(F)CCn1ccnn1)NC(C(C)C)CNC(C1CC1Br)=O N1(Cc2cncc(C)c2)CCC2(CC1)CC2NC(C1(c2cccc(O)c2)CC1)=O c1(C(C)=O)cc(C(=O)N(C2CCN(C(=O)CN3CCC(C)CC3)CC2)C)c(C)o1 C12(NC(c3c(CC)cno3)=O)CCCC1CN(C(c1sccc1OCC)=O)C2 Cc1cc(CNC(c2cc(CNC(c3snnc3C)=O)ccn2)=O)cc(C)n1 N1(C(=O)OCC)CCC2(CC1)CC2CNC(=O)C(C)(C)C(F)c1ccccc1 N1(C(c2c(C)ncn2O)=O)CCCC(C2(NC(C3(C(F)(F)F)CCC3)=O)CC2)C1 C1(C(=O)NCC(=C)CCNC(c2c[nH]c(=N)s2)=O)CCC(C)(C)C1 CC1CN(C(=O)C(C)(C)S(C)(=O)=O)CCC1N=c1[nH]c(C(C)(C)C)nc(=N)[nH]1 C(=O)(CC1OCc2ccccc21)NCC1(OC)CCN(C(C2(C#C)CC2)=O)CC1 C(=O)(CC1OCCc2ccsc21)N1C(COC)(CNC(=O)C2=CCC2)CCC1 N1(C(C2CCC(n3cc(C(C)C)nn3)C2)=O)CCOCC(C(C)(C)C)C1 N1(C(CCCSC)=O)CCN(C(C2CNc3ccnn3C2)=O)C2CS(=O)(=O)CC12 c1(CC(=O)N(C)CCOCCCNC(c2cc(CF)on2)=O)ccc(F)cc1F c1(SCC)ccc(C(N2CCC(O)(COC)C2)=O)cc1 C=C=C(C)CC(=O)N(C1CCN(C(=O)CN(C2CCS(=O)(=O)C2)C)CC1)C C(CNC(=O)C(=O)C(C)C)(N=c1[nH]c(Cl)c(C#N)s1)c1c(OC)cccc1 C(C)(C(O)C(=O)NCC(C)(C)CN(C(=O)CCNC(=O)CC(C)C)C)SC N1(C(C(C)OCCC=C)=O)CCC(C=C)(NC(c2cnc(C)c(OC)c2)=O)C1 O=C1CN(CCCN(C2CCCCC2)C(=O)C(=O)NC2CNCCO2)CCN1 c1(CC2CN(C(=O)NCC3(CO)CCC3)C2)cc(I)ccc1O C(=O)(C(F)(F)C(C)(C)O)NCC(COC)NC(c1ccc(C)c(C#N)c1)=O CC(C)CC(C)(C)C(=O)N1CCOC(C(C)NC(=O)CN(C)C(C)C)C1 C12(C(N(CCCN(C(=O)CC3CCC(=O)N3)C)C)=O)CCC(C1)C2 O=C(CCCCC1CC1)NCCC1(O)CN(C(=O)C(F)=C2CCCC2)C1 c1(C(=O)NCCNC(c2c(CCC)nco2)=O)ccc(=O)n(CCF)n1 C(=O)(C(C)(F)C(=O)N(CCC(=O)NCCCOCCO)C)OC N(C)(C(=NCC1CCCCC1)NCc1nc(-c2ccncc2)n[nH]1)CCCC C12(CNC(C3C(C=C(C)C)C3(C)C)=O)CC(CO1)N(C(=O)COCC1CC1)C2 c1(C(N2CC(C(N(CC(=C)C)CC(=C)C)=O)OCC2)=O)ccc(C)nc1C CC(C)(CC#N)C(=O)N1CCC(OCC(=O)NCC2(CO)CC3CC3C2)C1 Cc1[nH]nc2ccc(C(N3CC(NC(=O)CC(C)(C)O)CC(C)C3)=O)cc12 N1(C(CCc2cc(C)no2)=O)CCC(NC(=O)CCC#N)C(C(C)C)C1 N1(C(C)=O)CCOCC1Nc1cccc(Oc2cccc(I)c2)c1 C1(COCC)(CNC(C2(OC)CCCC2)=O)CCCN1C(c1ccsc1)=O C1(CNC(CCCC#C)=O)CN(C(C23CSCC2C3)=O)CC12CC2 c1(CC)nnc(C)cc1C(N1CCN(C(=O)C#CC(C)C)C(CO)C1)=O C(=O)(CC(O)CC1CC1)N(CC(C)NC(=O)COc1ccsn1)C c1(C(=O)N(CC(=O)NC2CC(CCOC)C2)C2CCC2)coc(N(C)C)n1 CCCC(CCCNC(=O)CCNC(C)=O)NC(c1ccc(F)c(N)c1)=O C=CC(F)(F)C(=O)N(C)CC1CCCN1C(=O)CN(C)CCOC C(c1ccccc1Cl)=CC(=O)NC1C(NC(=O)C=CC2CCOC2)CCCC1 C1(NC(c2c(F)cccc2F)=O)CC2(CCN(C(C3C4CCN3CC4)=O)CC2)C1 Cc1cc(Br)cnc1C(N1CC(CCNC(C2CC3(C2)CC(C)C3)=O)C1)=O c1(NC(C)=O)cc(N2CCC(CC(N3CCCC3NS(C)(=O)=O)=O)C2)nc(=N)[nH]1 c1(C(N(CC(C)(C)NC(C2CC(F)C2)=O)C)=O)nc2cncnc2nc1O CCCCC(CC)CCC(=O)NCC1CC(O)(CNC(=O)CCC(CC)OC)C1 c1(C(N2CC(NC(C(C)OCC=C)=O)CC23CCC3)=O)cncc(P(C)(C)=O)c1 c1(C(=O)NC2(CN(C(c3cc(CC)c(C)o3)=O)C)CC2)ccc(Br)nc1N c1(C(N2CCCC(N(C)Cc3nnc(S)n3C)C2)=O)cc(S(N)(=O)=O)co1 C(C(=O)N1CC(NC(C2CC3(CC3)C2)=O)C1)(C(C)C)NC(=O)OCC C1(NC(CS(=O)(=O)NC)=O)CCCC12CN(C(c1coc(CC3CC3)n1)=O)C2 CC1CN(C(C2CCN(C(c3ccnc(O)c3)=O)CC2)=O)CC(=O)N1 C(=O)(N1OC2C=CC1CC2)C1CC(C)N1C(c1cnc(O)c(F)c1)=O C1(CNC(Cc2ncc(C)o2)=O)CCN(C(C2CCCC2C)=O)CC1 CCCCCC(C(=O)NC(C1CCCN1C(=O)CC1CC1)(C)C)C(C)C c1(OC)cccc2c(CNC(C3COC(=O)C3)=O)coc12.C123CC(C1)(C2)C(=O)N3 C=CCC(C(=O)NCC1CNC(=O)O1)NC(=O)COC N1(C(c2c(NC)nccc2)=O)CCC(C)(C(=O)NC(C)COC(F)(F)F)CC1 CN1CC(=O)Nc2cc(C(=O)NC3CC3NC(=O)CCC(=O)NC3CC3)cnc21 Cc1ccc(C(=O)NC(CNC(c2ccc(C(O)CF)cc2)=O)CC(C)C)cc1 C1(CCNC(c2ccn(CC(C)C)c2)=O)CN(C(C2CS(=O)(=O)C2)=O)CC(C)O1 C12(C(c3nnnn3C3CCOCC3)NCC(C)OCCO)CCC(CC1)OC2 N1(Cc2cn(-c3cccc(CC(=O)OC)c3)nn2)CCCCC2(CCOCC2)C1 C1(NC(C2CCC(=C)CC2)=O)CN(C(=O)C(C)C2CCC2)Cc2nccn2C1 c1(C(C(=O)NCC(=C)C)N(C)CC2CCCCO2)sc(Cl)cc1Br N1(C(COCCCCC)=O)CCC(C)(CNC(c2c(CO)noc2C)=O)CC1 N1(C(CC(=C)Br)=O)CC2C(CNC(C3(C)CS(=O)(=O)C3)=O)C2C1 C1(COC)(NC(=O)C=C2CCCCC2)CCN(C(C2(C3CCCO3)CC2)=O)CC1 N1(C(C(CCN(C)C)N(C)C)=O)CC2CCN(C(c3ccsc3Cl)=O)CC2C1 c1(CC)ccc(C(N2CC(CNC(=O)CCCN=[N+]=[N-])CC(C)C2)=O)cc1F CC(Cn1ccnc1)C(=O)NCCN(C1CCCC1)C(=O)CC1CCCO1 C1(CNC(COCCOC)=O)CC2COCC2N1C(C1CC12CC2)=O N1(C(CC(C)(C)F)=O)CCC2C(CCCN2C(=O)Cc2ccc(CO)cc2)C1 CCC(CCOC)C(=O)NCC1(F)CC(NC(=O)Cc2ccsc2)C1 c1(N2CCC(=CC(=O)NC3CC(=O)N(C4CC4)C3)CC2)cccc([N+](=O)[O-])c1 C(C(C(=O)NOC1CC1)C(C)(C)C)NC(C(CC)SC)=O C1(CNC(C(CO)N(C)C)=O)CC2CCC1N(C(=O)C=Cc1cccc(O)c1)C2 c1(N2CCOCC(NC(C(CCSC)O)=O)C2)ccn2c(Br)cnc2n1 C(=O)(C(C)(C)C1=CCN(C(=O)C2=C(Cl)CCCC2)C1)NC1(C#C)CCCOC1 C1(C(C)(F)F)CCN(c2ccnc(NCC3COCCN3CC3CCC3)n2)CC1 Cc1cc(C(N2CC(CNC(=O)Cn3c(C)ccc3C)C(C)C2)=O)c(Cl)cc1F CC(N=c1[nH]c(=NC(C)c2ccc(C(C)(C)C)cc2)c2[nH]ccc2[nH]1)C1CC1 C(CN=c1[nH]c(C)nc(Cl)c1CC)(C1CCCC1)NC(c1ccn(CC)n1)=O c1(N2CCC(CC=C(C)C)C2)nccc(-c2ccccc2)n1 Cc1cc(C)c(C(N2CC(C3(NC(=O)CC(C4CC4)C4CC4)CC3)C2)=O)c(C)c1 c1(C(=O)NC2(C)CC(NC(C(CCC)OCC)=O)C2)c(F)cncc1Cl C=CCC(C)(CC)C(=O)NC1CC2(C(=O)NC3CCCCC3C#N)COC1C2 CC1(C)CC(NC(=O)CN2CCCCC2)CN1C(=O)C(S(C)(=O)=O)C1CC1 Cc1c(Br)ccnc1C(N1CCN(C)CC1CNC(=O)COCC(F)F)=O C1(C(=O)NCCC(CNC(=O)Cc2sccc2C)OC)CC12CCCC2 N1(C(C2(OC)CCSCC2)=O)CCC(C2(NC(c3csnc3C)=O)CC2)C1 N1(C(C(CC(F)F)NC(C=CC2(C)COC2)=O)=O)CC(O)C2(CCCC2)C1 C1(C)(C(N2CCC(N(CCC)C(c3ccoc3Cl)=O)CC2)=O)CCC(C)(C)CC1 c1(CN2CC(C(=O)NC34CC(CO)(C3)C4)C2)cc(OC(F)(F)F)cc(Cl)c1.O Cc1nc(C(=O)NC2CN(Cc3ncccc3O)CC2F)ccc1F c1(C(=O)NCCC(C)N(C)C(C2(CCF)CCC2)=O)ccc(-c2cnn(C)c2)o1 CC(C)C(CCN(C)C(=O)Nc1cc(C2CCOCC2)no1)N(C)C c1(C(c2cscc2Cl)=O)ncc(Cl)c(=NC2CCCC23CNC3)[nH]1.CO C1(C(N2CCCN(C(C(C=C)(C)CC)=O)CC2)=O)COc2ccc(O)cc2O1 N1(C(Cc2ccc(C)cc2)=O)CCN(C(c2ccnnc2)=O)C2COCC12 Cc1cc(Cl)c(C(=O)NC2CC(F)(CNC(=O)C(O)Cn3cncn3)C2)cc1N N1(C(C2C(NC(C(C)n3ccnc3)=O)C2(C)C)=O)CCC(C2(C)CC2)C1 C#CC1(C(N2CCN(C(C3CC(OC(F)F)C3)=O)CC2)=O)CCOCC1 c1(NCC23CC(NC(CNC(=O)OC)=O)(C2)C(C)O3)cnc2nccn2c1 N1(C(C2(NC(C3=C(C)CC3)=O)CCOCC2)=O)CC(C)CC(C)C1 C1(C(=O)NC)CCC(NC(C2CC(N)CN2C)=O)CC1 Cn1c(O)nc2cc(C(N3CCC(CNC(=O)COCCCF)CC3)=O)cnc12 N1(C(CC(CC)CC)=O)CCN(C(=O)CNC(=O)CN(C)C)CC(O)C1 N1(C(CC(CCSC)O)=O)CC2CC3CC2C1C3NC(c1cocn1)=O N1(C(C(C(CC)O)C)=O)CC2CCC1CN2C(c1sc(F)cc1Cl)=O CC1CC(CNC(c2ccc(C(F)(F)F)nc2)=O)CN1C(c1ccc(O)cn1)=O N1(C(CC2(C)CCN2C(=O)C=Cc2cocn2)=O)CC2C(C1)C2(F)F C1(C(N(CCC#C)C(C)C)=O)CN(CC2(COC)CC2)CC1C C1(N(C(CSCCN(C)C)=O)C)CCCN(C(=O)Cn2cc([N+](=O)[O-])cn2)CC1 C1(NC(C2CCCS2(=O)=O)=O)CCS(=O)(=O)C12CN(C(c1cc(C3CC3)on1)=O)C2 C(=O)(CC(C)(C)C#N)N(C(C)C(=O)NC1(C)CC(F)(F)C1)C CN=c1[nH]c(C(=O)NC2CC(CNC(c3cn(C(C)(C)C)nc3C)=O)C2)cs1 c1(N2CC(CC=C)(NC(=O)C(C)SC(F)(F)F)C2)cc2nncn2cn1 C(=O)(C(O)CC(F)F)N(C)C1CC1.c1(C2c3cn(nn3)CC2)cccc(Cl)c1 C1(COC)(NC(C2COCC(C)(C)O2)=O)CCCN(C(c2ccco2)=O)C1 c1(CCC(=O)NC2C(NC(Cc3nc(CC)sc3)=O)CC2)cnn(C)c1C N1(C(C2N(C(c3c(OC)cccc3Br)=O)CC(C)C2)=O)CCCC2(CCOC2)C1 C1(C(N2CCC(C(C)C)C2)=O)CCCCN(C(=O)Cn2cncn2)C1 c1(OCC)ccc(C)cc1NC(=O)C(N1CC(C(F)(F)F)OC(CO)C1)=O N1(C(C(CCSC)O)=O)CC2(CCCC2)C1C(=O)NCc1ccc(C)nc1 C(=O)(CS(=O)c1ccc(Cl)cc1)NC1CCN(C(CCSCC)=O)C12CC2 Cc1cccc(OCCC(=O)NC(C2CCOC2)CNC(=O)CCC=CBr)c1C c1(C(=O)NC2COCCN(C(C3C(C)C3)=O)C2)nn(C)c2ccccc12 C1(CNC(CC(CC)C)=O)CC12CCN(C(c1coc(C(F)F)n1)=O)CC2 N1(C(=O)Nc2cncc(-n3cccn3)n2)CCC(O)(C2(C(=O)O)CCC2)CC1 C1(NC(COC(C)=O)=O)CCCC1(C)NC(=O)CCOCC(F)F c1(OC)ccc(-c2nc(CP(C)(C)=O)n(CC3COC(C)(C)C3)n2)nc1 C1(C(N(C2CC2C2CC2)C)=O)N(C(c2cccc(F)c2)=O)CCC1(C)C Cc1ccc2nc(N3CCCC(C(=O)O)C3C)[nH]c2c1 C1(NC(CCC(N)=O)=O)CC2CC1N(C(=O)CCOc1cccnc1)C2 C1(N(C(C(C)=C(C)C)=O)C)CCCN(C(=O)C(O)C(F)F)CC1 C1(C(=O)NC(C)CCNC(=O)C=Cc2cncn2C)CCc2nccn2C1 CP(C)(=O)CCCNC(C1CC(F)CN1C(C1CN(C(N)=O)C1)=O)=O N1(C(c2cn(CC=C)nc2)=O)CC(NC(C2(F)CC=CCC2)=O)C(C(F)F)C1 Cn1cncc1C(O)C(=O)NC1CCN(C(=O)CCc2nc(O)n[nH]2)C1 c1(OC)ccc(C(=O)NCC2CC(C)N(C(=O)C=CCN(C)C3CC3)C2)cc1Br N#Cc1ccnc(NCC(C2CCCCC2)NC(C2CC(C3CC3)=NO2)=O)n1 C12(NC(C(C=C)O)=O)CCCCC1CN(C(c1nccc(OC)c1F)=O)C2 N1(C(C=CCOC(C)(C)C)=O)CC(NC(c2scnc2-c2cccs2)=O)C(O)C1 C1(C(N(CCCCC=C)C)=O)CCCCC1NC(=O)Cc1sccc1C c1(OC)cccc(CCC(=O)NCC(O)CCNC(c2sncc2C)=O)n1 c1(C(=O)NCCC2CC(OC)CN2C(=O)C(O)C2CC2)ccn(C)c(=O)c1 N1(C(C(Cn2cccn2)NC(c2c(C)c[nH]n2)=O)=O)CCN(C)C(C)C1 C1(CNC(CCCCOC)=O)CC2CCCCC2N1C(c1ccc(OC)nc1)=O C12(C(=O)NC3CCC(CNC(c4c(C)cncc4)=O)C3)CCCC1CC(=O)C2 c1(CC)ncc(C(=O)NC(C)CC2CN(C(C3CCN(C)C(=O)C3)=O)C2)c(O)n1 c1(N2CCC(C)C(CO)C2)nc(=NCCC2OCCC2(C)C)[nH]c2ccsc12 C1(CNC(C2CC(OC(C)C(=O)Nc3cc(Cl)cn3C)C2)=O)CC(C)(C)CCO1